c1ccc(-n2cc(CSc3ccc4c(c3)OCCCO4)cn2)cc1 ZINC000217500009 EI On-Demand Unstable TERT 0 41 COc1ccc(CCNc2ccc(C(=O)O)cc2S(=O)(=O)NC[C@@H]2CCCO2)cc1OC ZINC000217500040 JF In-Stock Unstable PTGDR 17 40 COc1ccc(CCNc2ccc(C(=O)O)cc2S(=O)(=O)NC[C@@H]2CCCO2)cc1OC ZINC000217500040 JF In-Stock Unstable SCMU_MYCTU 0 44 N=C(N)c1ccc(NCCON)cc1 ZINC000217500097 AC For-Sale Unstable ACR 69 43 N=C(N)c1ccc(NCCON)cc1 ZINC000217500097 AC For-Sale Unstable ST14 29 44 N=C(N)c1ccc(NCCON)cc1 ZINC000217500097 AC For-Sale Unstable KLK_PIG 42 33 CN1CC[C@@H](Nc2nc3ccccc3s2)C1=O ZINC000217500111 BD On-Demand Unstable BCL2L1 51 35 COc1ccc(CCNc2ccc(C(=O)O)cc2S(=O)(=O)NC[C@H]2CCCO2)cc1OC ZINC000217500126 JF In-Stock Unstable PTGDR 17 40 COc1ccc(CCNc2ccc(C(=O)O)cc2S(=O)(=O)NC[C@H]2CCCO2)cc1OC ZINC000217500126 JF In-Stock Unstable SCMU_MYCTU 0 44 O=C(COc1ccccc1F)Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1 ZINC000217500128 FH On-Demand Unstable CETP 22 44 CN(C)[C@@H]1CCN(c2ccc(CBr)cn2)C1 ZINC000217500177 CE For-Sale Unstable TLR7 17 45 C[C@@](O)(CNC(=O)c1ccccc1Cl)c1cc2ccccc2s1 ZINC000217500184 EI In-Stock Unstable ECR 44 37 C[C@@](O)(CNC(=O)c1ccccc1Cl)c1cc2ccccc2s1 ZINC000217500184 EI In-Stock Unstable E3UJZ5_SPOLI 40 36 CN1CC[C@H](Nc2nc3ccccc3s2)C1=O ZINC000217500197 BD On-Demand Unstable BCL2L1 51 35 CN(C)[C@H]1CCN(c2ccc(CBr)cn2)C1 ZINC000217500263 CE For-Sale Unstable TLR7 17 45 C[C@](O)(CNC(=O)c1ccccc1Cl)c1cc2ccccc2s1 ZINC000217500281 EI In-Stock Unstable ECR 44 37 C[C@](O)(CNC(=O)c1ccccc1Cl)c1cc2ccccc2s1 ZINC000217500281 EI In-Stock Unstable E3UJZ5_SPOLI 40 36 Cc1cc(NC(=O)NCCc2cccc(Br)c2)ccc1Br ZINC000217500335 HJ For-Sale Unstable RAF1 24 42 Cc1cc(NC(=O)NCCc2cccc(Br)c2)ccc1Br ZINC000217500335 HJ For-Sale Unstable Q8MMZ8_EIMTE 0 42 Cc1cc(NC(=O)NCCc2cccc(Br)c2)ccc1Br ZINC000217500335 HJ For-Sale Unstable NCE103 23 45 CCCc1ccc(S(=O)(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)cc1 ZINC000217500391 HH For-Sale Unstable ALOX15 39 40 O=C(O)c1ccc(NC[C@@H]2CCCO2)c(S(=O)(=O)NC[C@@H]2CCCO2)c1 ZINC000217500419 GD In-Stock Unstable TNK2 44 37 N[C@@H]1CCCN([C@@H](c2ccccc2)c2ccc(O)cc2)C1 ZINC000217500466 CF For-Sale Unstable OPRD1 0 42 N[C@@H]1CCCN([C@@H](c2ccccc2)c2ccc(O)cc2)C1 ZINC000217500466 CF For-Sale Unstable OPRK1 0 42 N[C@@H]1CCCN([C@@H](c2ccccc2)c2ccc(O)cc2)C1 ZINC000217500466 CF For-Sale Unstable OPRL1 19 42 O=C(c1cccc(N2CCOCC2)c1)N1CCOc2ccc(CO)cc2C1 ZINC000217500497 FE In-Stock Unstable EPHB4 42 33 O=C(c1cccc(N2CCOCC2)c1)N1CCOc2ccc(CO)cc2C1 ZINC000217500497 FE In-Stock Unstable AKR1C3 31 43 O=C(O)c1ccc(NC[C@H]2CCCO2)c(S(=O)(=O)NC[C@@H]2CCCO2)c1 ZINC000217500504 GD In-Stock Unstable TNK2 44 37 O=C(O)c1ccc(NC[C@@H]2CCCO2)c(S(=O)(=O)NC[C@H]2CCCO2)c1 ZINC000217500587 GD In-Stock Unstable TNK2 44 37 O=C(O)c1ccc(NC[C@H]2CCCO2)c(S(=O)(=O)NC[C@H]2CCCO2)c1 ZINC000217500662 GD In-Stock Unstable TNK2 44 37 O=C(Cc1ccc(F)cc1F)N1C[C@@H]2CCC[C@H](C2)C1 ZINC000217500683 CG In-Stock Unstable HTR2A 19 40 CN1C(=O)N(C)C(=O)C(Cc2ccc(CC3(CN4C[C@@H]5C[C@H](C4)Cn4c5cccc4=O)C(=O)N(C)C(=O)N(C)C3=O)cc2)(CN2C[C@@H]3C[C@H](C2)Cn2c3cccc2=O)C1=O ZINC000217500729 KD In-Stock Unstable CHRNA4 36 59 CN1CCC(CNC(=O)c2ccc(/C=C\C(=O)O)s2)CC1 ZINC000217500740 DD For-Sale Unstable HTR4 43 34 CN1CCC(CNC(=O)c2ccc(/C=C\C(=O)O)s2)CC1 ZINC000217500740 DD For-Sale Unstable HTR1F 46 32 CN1CCC(CNC(=O)c2ccc(/C=C\C(=O)O)s2)CC1 ZINC000217500740 DD For-Sale Unstable CACNA1I 65 39 CC[C@@H](C)c1ccccc1NC(=O)NCCc1cccc(Br)c1 ZINC000217500803 GK For-Sale Unstable ACAT 0 51 CC[C@@H](c1cccc(Cl)c1)N1CCC[C@@H](N)C1 ZINC000217500860 CG For-Sale Unstable OPRL1 0 50 CC[C@H](C)c1ccccc1NC(=O)NCCc1cccc(Br)c1 ZINC000217500889 GK For-Sale Unstable ACAT 0 51 CCOc1ccc(C(=O)N2CCC[C@@H]2c2ccccn2)o1 ZINC000217500891 CG In-Stock Unstable ADAM17 0 44 CCOc1ccc(C(=O)N2CCC[C@@H]2c2ccccn2)o1 ZINC000217500891 CG In-Stock Unstable COLA 92 38 CCOc1ccc(C(=O)N2CCC[C@@H]2c2ccccn2)o1 ZINC000217500891 CG In-Stock Unstable CPT1A 83 38 CCOc1ccc(C(=O)N2CCC[C@@H]2c2ccccn2)o1 ZINC000217500891 CG In-Stock Unstable PREP 48 35 CC[C@H](CSC)N1C[C@@H](C)NC[C@@H]1c1ccccc1 ZINC000217500931 CG For-Sale Unstable CACNA1C 15 42 CC[C@H](CSC)N1C[C@@H](C)NC[C@@H]1c1ccccc1 ZINC000217500931 CG For-Sale Unstable CACNA1B 27 42 Cc1cc(I)ccc1NC(=O)c1cc(Br)ccc1I ZINC000217500936 KK For-Sale Unstable Q25615_ONCVO 57 42 CC[C@H](c1cccc(Cl)c1)N1CCC[C@@H](N)C1 ZINC000217500957 CG For-Sale Unstable OPRL1 0 50 CCOc1ccc(C(=O)N2CCC[C@H]2c2ccccn2)o1 ZINC000217500967 CG In-Stock Unstable ADAM17 0 44 CCOc1ccc(C(=O)N2CCC[C@H]2c2ccccn2)o1 ZINC000217500967 CG In-Stock Unstable COLA 92 38 CCOc1ccc(C(=O)N2CCC[C@H]2c2ccccn2)o1 ZINC000217500967 CG In-Stock Unstable CPT1A 83 38 CCOc1ccc(C(=O)N2CCC[C@H]2c2ccccn2)o1 ZINC000217500967 CG In-Stock Unstable PREP 48 35 COc1ccc([C@@H](C)N2CCC[C@@H](N)C2)cc1 ZINC000217501047 BE For-Sale Unstable CHRM2 16 48 c1ccc(-c2cnc(N3CCN(c4ncccn4)CC3)cn2)cc1 ZINC000217501084 DE On-Demand Unstable SORD 38 47 O=C(NCCc1cccc(Br)c1)NC1CCN(Cc2ccccc2)CC1 ZINC000217501103 HH For-Sale Unstable CHRM2 23 42 O=C(NCCc1cccc(Br)c1)NC1CCN(Cc2ccccc2)CC1 ZINC000217501103 HH For-Sale Unstable CHRM1 15 46 O=C(NCCc1cccc(Br)c1)NC1CCN(Cc2ccccc2)CC1 ZINC000217501103 HH For-Sale Unstable DRD2 26 58 O=C(NCCc1cccc(Br)c1)NC1CCN(Cc2ccccc2)CC1 ZINC000217501103 HH For-Sale Unstable DRD4 57 61 O=C(NCCc1cccc(Br)c1)NC1CCN(Cc2ccccc2)CC1 ZINC000217501103 HH For-Sale Unstable ACHE 49 54 O=C(NCCc1cccc(Br)c1)NC1CCN(Cc2ccccc2)CC1 ZINC000217501103 HH For-Sale Unstable HRH2 29 49 O=C(NCCc1cccc(Br)c1)NC1CCN(Cc2ccccc2)CC1 ZINC000217501103 HH For-Sale Unstable DRD3 22 58 O=C(NCCc1cccc(Br)c1)NC1CCN(Cc2ccccc2)CC1 ZINC000217501103 HH For-Sale Unstable KCNH2 15 45 O=C(NCCc1cccc(Br)c1)NC1CCN(Cc2ccccc2)CC1 ZINC000217501103 HH For-Sale Unstable CHRM3 28 46 O=C(NCCc1cccc(Br)c1)NC1CCN(Cc2ccccc2)CC1 ZINC000217501103 HH For-Sale Unstable VACHT_TETCF 0 42 O=C(NCCc1cccc(Br)c1)NC1CCN(Cc2ccccc2)CC1 ZINC000217501103 HH For-Sale Unstable SIGMAR1 63 72 O=C(NCCc1cccc(Br)c1)NC1CCN(Cc2ccccc2)CC1 ZINC000217501103 HH For-Sale Unstable SSTR5 57 39 O=C(NCCc1cccc(Br)c1)NC1CCN(Cc2ccccc2)CC1 ZINC000217501103 HH For-Sale Unstable BCHE 0 48 O=C(NCCc1cccc(Br)c1)NC1CCN(Cc2ccccc2)CC1 ZINC000217501103 HH For-Sale Unstable CCR3 60 46 O=C(NCCc1cccc(Br)c1)NC1CCN(Cc2ccccc2)CC1 ZINC000217501103 HH For-Sale Unstable UTS2R 19 41 O=C(NCCc1cccc(Br)c1)NC1CCN(Cc2ccccc2)CC1 ZINC000217501103 HH For-Sale Unstable SLC6A5 24 45 O=C(NCCc1cccc(Br)c1)NC1CCN(Cc2ccccc2)CC1 ZINC000217501103 HH For-Sale Unstable EPHX2 23 55 O=C(NCCc1cccc(Br)c1)NC1CCN(Cc2ccccc2)CC1 ZINC000217501103 HH For-Sale Unstable CXCR3 44 41 O=C(NCCc1cccc(Br)c1)NC1CCN(Cc2ccccc2)CC1 ZINC000217501103 HH For-Sale Unstable MCHR1 54 51 O=C(NCCc1cccc(Br)c1)NC1CCN(Cc2ccccc2)CC1 ZINC000217501103 HH For-Sale Unstable CACNA1G 30 42 O=C(NCCc1cccc(Br)c1)NC1CCN(Cc2ccccc2)CC1 ZINC000217501103 HH For-Sale Unstable CCR8 15 44 O=C(NCCc1cccc(Br)c1)NC1CCN(Cc2ccccc2)CC1 ZINC000217501103 HH For-Sale Unstable NPFFR1 54 37 O=C(NCCc1cccc(Br)c1)NC1CCN(Cc2ccccc2)CC1 ZINC000217501103 HH For-Sale Unstable ADIPOR1 0 44 O=C(NCCc1cccc(Br)c1)NC1CCN(Cc2ccccc2)CC1 ZINC000217501103 HH For-Sale Unstable ADIPOR2 0 44 COc1ccc([C@H](C)N2CCC[C@@H](N)C2)cc1 ZINC000217501125 BE For-Sale Unstable CHRM2 16 48 C[C@@](O)(CNC(=O)c1ccc(Cl)s1)c1cc2ccccc2s1 ZINC000217501147 FI In-Stock Unstable F10 23 48 C=C1CC[C@H](O)C/C1=C/C=C1\CCC[C@@]2(C)[C@@H]1CC[C@@H]2[C@H](C)[C@H](O)CCC(C)(C)O ZINC000217501168 HK For-Sale Unstable VDR 141 65 C=C1CC[C@H](O)C/C1=C/C=C1\CCC[C@@]2(C)[C@@H]1CC[C@@H]2[C@H](C)[C@H](O)CCC(C)(C)O ZINC000217501168 HK For-Sale Unstable CYP24A1 44 55 C=C1CC[C@H](O)C/C1=C/C=C1\CCC[C@@]2(C)[C@@H]1CC[C@@H]2[C@H](C)[C@H](O)CCC(C)(C)O ZINC000217501168 HK For-Sale Unstable CYP27B1 25 44 N[C@@H]1CCCN([C@@H]2CCc3ccccc32)C1 ZINC000217501202 BE For-Sale Unstable SLC6A1 0 47 COc1ccc(NC(=O)[C@@H](c2ccccc2)S(=O)(=O)c2ccccc2)cc1Cl ZINC000217501205 HJ On-Demand Unstable DHODH 15 41 COc1ccc(NC(=O)[C@@H](c2ccccc2)S(=O)(=O)c2ccccc2)cc1Cl ZINC000217501205 HJ On-Demand Unstable MMP13 19 41 COc1ccc(NC(=O)[C@@H](c2ccccc2)S(=O)(=O)c2ccccc2)cc1Cl ZINC000217501205 HJ On-Demand Unstable COLA 56 38 COc1ccc(NC(=O)[C@@H](c2ccccc2)S(=O)(=O)c2ccccc2)cc1Cl ZINC000217501205 HJ On-Demand Unstable CPT1A 55 38 COc1ccc(NC(=O)[C@@H](c2ccccc2)S(=O)(=O)c2ccccc2)cc1Cl ZINC000217501205 HJ On-Demand Unstable CPT2 43 34 COc1ccc(NC(=O)[C@@H](c2ccccc2)S(=O)(=O)c2ccccc2)cc1Cl ZINC000217501205 HJ On-Demand Unstable GRM4 36 52 COc1ccc(S(=O)(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)c(C)c1 ZINC000217501231 IG For-Sale Unstable TGFBR1 32 40 C[C@](O)(CNC(=O)c1ccc(Cl)s1)c1cc2ccccc2s1 ZINC000217501233 FI In-Stock Unstable F10 23 48 O=[N+]([O-])c1ccccc1OC[C@@H]1CN(Cc2ccccc2)CCO1 ZINC000217501248 EF In-Stock Unstable DRD4 20 68 O=[N+]([O-])c1ccccc1OC[C@@H]1CN(Cc2ccccc2)CCO1 ZINC000217501248 EF In-Stock Unstable SIGMAR1 18 43 CCOC(=O)C1CCN(C(=O)c2cc(I)ccc2O)CC1 ZINC000217501258 HE On-Demand Unstable PTR1 49 38 CCOC(=O)C1CCN(C(=O)c2cc(I)ccc2O)CC1 ZINC000217501258 HE On-Demand Unstable L3MBTL3 50 38 COc1ccc(NC(=O)[C@H](c2ccccc2)S(=O)(=O)c2ccccc2)cc1Cl ZINC000217501282 HJ On-Demand Unstable DHODH 15 41 COc1ccc(NC(=O)[C@H](c2ccccc2)S(=O)(=O)c2ccccc2)cc1Cl ZINC000217501282 HJ On-Demand Unstable MMP13 19 41 COc1ccc(NC(=O)[C@H](c2ccccc2)S(=O)(=O)c2ccccc2)cc1Cl ZINC000217501282 HJ On-Demand Unstable COLA 56 38 COc1ccc(NC(=O)[C@H](c2ccccc2)S(=O)(=O)c2ccccc2)cc1Cl ZINC000217501282 HJ On-Demand Unstable CPT1A 55 38 COc1ccc(NC(=O)[C@H](c2ccccc2)S(=O)(=O)c2ccccc2)cc1Cl ZINC000217501282 HJ On-Demand Unstable CPT2 43 34 COc1ccc(NC(=O)[C@H](c2ccccc2)S(=O)(=O)c2ccccc2)cc1Cl ZINC000217501282 HJ On-Demand Unstable GRM4 36 52 O=C(NCCc1cccc(Br)c1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217501323 IG For-Sale Unstable HRH2 24 45 O=C(NCCc1cccc(Br)c1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217501323 IG For-Sale Unstable BMP1 45 40 O=C(NCCc1cccc(Br)c1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217501323 IG For-Sale Unstable SIGMAR1 15 54 O=C(NCCc1cccc(Br)c1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217501323 IG For-Sale Unstable NOS2 84 36 O=C(NCCc1cccc(Br)c1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217501323 IG For-Sale Unstable SSTR3 48 30 O=C(NCCc1cccc(Br)c1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217501323 IG For-Sale Unstable FAAH 19 40 O=C(NCCc1cccc(Br)c1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217501323 IG For-Sale Unstable MCHR1 27 47 O=[N+]([O-])c1ccccc1OC[C@H]1CN(Cc2ccccc2)CCO1 ZINC000217501340 EF In-Stock Unstable DRD4 20 68 O=[N+]([O-])c1ccccc1OC[C@H]1CN(Cc2ccccc2)CCO1 ZINC000217501340 EF In-Stock Unstable SIGMAR1 18 43 C[C@@H](c1ccccc1)N1CCC[C@@H](N)C1 ZINC000217501348 BE On-Demand Unstable DPP4 18 40 CCOC(=O)CN1CCO[C@@H](COc2cccc([N+](=O)[O-])c2)C1 ZINC000217501428 DD In-Stock Unstable CACNA1C 55 36 CCOC(=O)CN1CCO[C@@H](COc2cccc([N+](=O)[O-])c2)C1 ZINC000217501428 DD In-Stock Unstable CACNA1D 81 36 C[C@H](c1ccccc1)N1CCC[C@@H](N)C1 ZINC000217501429 BE On-Demand Unstable DPP4 18 40 CCOC(=O)N1CCN(C(=O)NCCc2cccc(Br)c2)CC1 ZINC000217501448 GE On-Demand Unstable P2RY12 52 43 CCOC(=O)N1CCN(C(=O)NCCc2cccc(Br)c2)CC1 ZINC000217501448 GE On-Demand Unstable HPN 30 41 CCOC(=O)CN1CCO[C@H](COc2cccc([N+](=O)[O-])c2)C1 ZINC000217501518 DD In-Stock Unstable CACNA1C 55 36 CCOC(=O)CN1CCO[C@H](COc2cccc([N+](=O)[O-])c2)C1 ZINC000217501518 DD In-Stock Unstable CACNA1D 81 36 O=C(NCCCN1CCOCC1)c1cc(Br)ccc1I ZINC000217501520 JF On-Demand Unstable EGFR 15 43 O=C(NCCCN1CCOCC1)c1cc(Br)ccc1I ZINC000217501520 JF On-Demand Unstable DRD2 23 42 O=C(NCCCN1CCOCC1)c1cc(Br)ccc1I ZINC000217501520 JF On-Demand Unstable HTR2A 25 41 O=C(NCCCN1CCOCC1)c1cc(Br)ccc1I ZINC000217501520 JF On-Demand Unstable HTR2C 29 41 O=C(NCCCN1CCOCC1)c1cc(Br)ccc1I ZINC000217501520 JF On-Demand Unstable DRD3 49 44 O=C(NCCCN1CCOCC1)c1cc(Br)ccc1I ZINC000217501520 JF On-Demand Unstable EPHX2 21 43 O=S(=O)(c1cccc(-c2nnc(SCc3cnn(-c4ccccc4)c3)o2)c1)N1CCCCC1 ZINC000217501605 JI On-Demand Unstable GSK3B 15 41 O=S(=O)(c1cccc(-c2nnc(SCc3cnn(-c4ccccc4)c3)o2)c1)N1CCCCC1 ZINC000217501605 JI On-Demand Unstable GSK3A 48 41 COC(=O)CN1CCO[C@@H](COc2cccc([N+](=O)[O-])c2)C1 ZINC000217501625 DC In-Stock Unstable CACNA1C 44 35 COC(=O)CN1CCO[C@@H](COc2cccc([N+](=O)[O-])c2)C1 ZINC000217501625 DC In-Stock Unstable CACNA1D 73 35 CC[C@H](CSC)N1C[C@@H](Cc2ccccc2)NC[C@@H]1C ZINC000217501705 CG For-Sale Unstable CACNA1B 23 41 COC(=O)CN1CCO[C@H](COc2cccc([N+](=O)[O-])c2)C1 ZINC000217501709 DC In-Stock Unstable CACNA1C 44 35 COC(=O)CN1CCO[C@H](COc2cccc([N+](=O)[O-])c2)C1 ZINC000217501709 DC In-Stock Unstable CACNA1D 73 35 NC(=O)CN1CCO[C@@H](COc2cccc([N+](=O)[O-])c2)C1 ZINC000217501818 CC In-Stock Unstable CACNA1D 49 32 NC(=O)CN1CCO[C@@H](COc2cccc([N+](=O)[O-])c2)C1 ZINC000217501818 CC In-Stock Unstable ACR 18 42 CC1(C)CC[C@@H](N2CCC[C@@H](CN)C2)c2ccccc21 ZINC000217501851 CG For-Sale Unstable SLC6A1 0 40 CC1(C)CC[C@@H](N2CCC[C@@H](CN)C2)c2ccccc21 ZINC000217501851 CG For-Sale Unstable OPRL1 17 56 NC(=O)CN1CCO[C@H](COc2cccc([N+](=O)[O-])c2)C1 ZINC000217501893 CC In-Stock Unstable CACNA1D 49 32 NC(=O)CN1CCO[C@H](COc2cccc([N+](=O)[O-])c2)C1 ZINC000217501893 CC In-Stock Unstable ACR 18 42 O=C(NCCc1cccc(Br)c1)Nc1cc(F)ccc1F ZINC000217501904 FI For-Sale Unstable RAF1 25 41 CC1(C)CC[C@H](N2CCC[C@@H](CN)C2)c2ccccc21 ZINC000217501941 CG For-Sale Unstable SLC6A1 0 40 CC1(C)CC[C@H](N2CCC[C@@H](CN)C2)c2ccccc21 ZINC000217501941 CG For-Sale Unstable OPRL1 17 56 CN1CCO[C@@H](COc2cccc([N+](=O)[O-])c2)C1 ZINC000217501985 CD In-Stock Unstable CHRNA10 51 39 COc1cccc([C@@H](C)N2CCC[C@@H](N)C2)c1 ZINC000217502029 BE On-Demand Unstable CHRNA10 23 43 CC[C@H](c1cccc([N+](=O)[O-])c1)N1CCC[C@@H](CN)C1 ZINC000217502047 CF For-Sale Unstable CACNA1D 43 33 CN1CCO[C@H](COc2cccc([N+](=O)[O-])c2)C1 ZINC000217502069 CD In-Stock Unstable CHRNA10 51 39 CN(C)[C@@H]1CCN(c2cc(Cl)ccc2CBr)C1 ZINC000217502092 DG For-Sale Unstable NOS3 18 42 CC[C@@H](c1cccc([N+](=O)[O-])c1)N1CCC[C@@H](CN)C1 ZINC000217502120 CF For-Sale Unstable CACNA1D 43 33 COc1cccc([C@H](C)N2CCC[C@@H](N)C2)c1 ZINC000217502131 BE On-Demand Unstable CHRNA10 23 43 CN(C)[C@H]1CCN(c2cc(Cl)ccc2CBr)C1 ZINC000217502183 DG For-Sale Unstable NOS3 18 42 O=C(NCC1CCCCC1)c1cc(Br)ccc1O ZINC000217502226 DG For-Sale Unstable CACNA1I 59 35 O=C(NCC1CCCCC1)c1cc(Br)ccc1O ZINC000217502226 DG For-Sale Unstable PYK 85 38 CN(C)[C@@H]1CCN(c2ccc(Cl)cc2CBr)C1 ZINC000217502297 DG For-Sale Unstable NOS2 21 45 CN(C)[C@@H]1CCN(c2ccc(Cl)cc2CBr)C1 ZINC000217502297 DG For-Sale Unstable NOS3 22 45 O=C(NCCc1cccc(Br)c1)N1CCN(c2ccccn2)CC1 ZINC000217502311 GF On-Demand Unstable DRD4 25 43 O=C(NCCc1cccc(Br)c1)N1CCN(c2ccccn2)CC1 ZINC000217502311 GF On-Demand Unstable GPBAR1 0 43 O=C(NCCc1cccc(Br)c1)N1CCN(c2ccccn2)CC1 ZINC000217502311 GF On-Demand Unstable SLC6A7 0 43 O=C(NCC1CCCCC1)c1cc(I)ccc1O ZINC000217502340 FG For-Sale Unstable CACNA1I 58 32 Cc1ccccc1-c1cccc(C(=O)N(C)CC[C@@H]2CCCCO2)c1 ZINC000217502351 EJ In-Stock Unstable OXTR 28 47 Cc1ccccc1-c1cccc(C(=O)N(C)CC[C@@H]2CCCCO2)c1 ZINC000217502351 EJ In-Stock Unstable AVPR1A 0 47 CN(C)[C@H]1CCN(c2ccc(Cl)cc2CBr)C1 ZINC000217502381 DG For-Sale Unstable NOS2 21 45 CN(C)[C@H]1CCN(c2ccc(Cl)cc2CBr)C1 ZINC000217502381 DG For-Sale Unstable NOS3 22 45 O=S(=O)(NCCn1nc(-c2ccccn2)c2c1CCCC2)c1ccc2ccccc2c1 ZINC000217502410 IH For-Sale Unstable HTR7 20 48 O=S(=O)(NCCn1nc(-c2ccccn2)c2c1CCCC2)c1ccc2ccccc2c1 ZINC000217502410 IH For-Sale Unstable TRY2_BOVIN 61 36 Cc1ccccc1-c1cccc(C(=O)N(C)CC[C@H]2CCCCO2)c1 ZINC000217502428 EJ In-Stock Unstable OXTR 28 47 Cc1ccccc1-c1cccc(C(=O)N(C)CC[C@H]2CCCCO2)c1 ZINC000217502428 EJ In-Stock Unstable AVPR1A 0 47 CC1(C)CC(NC(=O)c2cc(Br)ccc2I)CC(C)(C)N1 ZINC000217502445 JI On-Demand Unstable EZH2 59 43 O=S(=O)(NCCn1nc(-c2ccccn2)c2c1CCCC2)c1cccc2ccccc12 ZINC000217502530 IH For-Sale Unstable NPY2R 37 41 O=S(=O)(NCCn1nc(-c2ccccn2)c2c1CCCC2)c1cccc2ccccc12 ZINC000217502530 IH For-Sale Unstable NPY5R 16 41 O=S(=O)(NCCn1nc(-c2ccccn2)c2c1CCCC2)c1ccc(F)c(Cl)c1 ZINC000217502625 IH For-Sale Unstable HTR7 15 45 FC(F)Oc1ccc(-c2nnc(SCc3cnn(-c4ccccc4)c3)o2)cc1 ZINC000217502630 HJ On-Demand Unstable GSK3B 17 45 FC(F)Oc1ccc(-c2nnc(SCc3cnn(-c4ccccc4)c3)o2)cc1 ZINC000217502630 HJ On-Demand Unstable GSK3A 49 45 FC(F)Oc1ccc(-c2nnc(SCc3cnn(-c4ccccc4)c3)o2)cc1 ZINC000217502630 HJ On-Demand Unstable TERT 25 41 CC[C@@H](c1ccc(Cl)cc1)N1CCC[C@@H](N)C1 ZINC000217502719 CG On-Demand Unstable SLC6A1 41 38 O=[N+]([O-])c1cccc(OC[C@@H]2CN(Cc3ccccc3)CCO2)c1 ZINC000217502745 EF In-Stock Unstable MGLL 0 41 O=[N+]([O-])c1cccc(OC[C@@H]2CN(Cc3ccccc3)CCO2)c1 ZINC000217502745 EF In-Stock Unstable ABHD6 0 41 CC[C@H](c1ccc(Cl)cc1)N1CCC[C@@H](N)C1 ZINC000217502793 CG On-Demand Unstable SLC6A1 41 38 COc1cc([C@H]2N3CCc4ccccc4[C@H]3CN2S(=O)(=O)c2ccccc2)ccc1OS(=O)(=O)c1ccccc1 ZINC000217502820 KJ In-Stock Unstable FKBP1A 23 42 O=[N+]([O-])c1cccc(OC[C@H]2CN(Cc3ccccc3)CCO2)c1 ZINC000217502835 EF In-Stock Unstable MGLL 0 41 O=[N+]([O-])c1cccc(OC[C@H]2CN(Cc3ccccc3)CCO2)c1 ZINC000217502835 EF In-Stock Unstable ABHD6 0 41 COC(=O)c1cccc(NC(=O)NCCc2cccc(Br)c2)c1 ZINC000217502854 GH For-Sale Unstable PPIA 24 48 COC(=O)c1cccc(NC(=O)NCCc2cccc(Br)c2)c1 ZINC000217502854 GH For-Sale Unstable CCKAR 0 41 COC(=O)c1cccc(NC(=O)NCCc2cccc(Br)c2)c1 ZINC000217502854 GH For-Sale Unstable CCR3 30 41 COC(=O)c1cccc(NC(=O)NCCc2cccc(Br)c2)c1 ZINC000217502854 GH For-Sale Unstable RAF1 19 41 COC(=O)c1cccc(NC(=O)NCCc2cccc(Br)c2)c1 ZINC000217502854 GH For-Sale Unstable ROCK2 22 40 COC(=O)c1cccc(NC(=O)NCCc2cccc(Br)c2)c1 ZINC000217502854 GH For-Sale Unstable EPHX2 16 46 COC(=O)c1cccc(NC(=O)NCCc2cccc(Br)c2)c1 ZINC000217502854 GH For-Sale Unstable Q8MMZ8_EIMTE 22 41 COC(=O)c1cccc(NC(=O)NCCc2cccc(Br)c2)c1 ZINC000217502854 GH For-Sale Unstable KCNK3 60 34 CCCNc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217502861 EG In-Stock Unstable AKR1C3 50 39 CCCNc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217502861 EG In-Stock Unstable LIMK2 43 40 COc1cc([C@@H]2N3CCc4ccccc4[C@H]3CN2S(=O)(=O)c2ccccc2)ccc1OS(=O)(=O)c1ccccc1 ZINC000217502897 KJ In-Stock Unstable FKBP1A 23 42 CCOC(=O)CN1CCO[C@@H](COc2ccc([N+](=O)[O-])cc2)C1 ZINC000217502924 DD In-Stock Unstable SLC27A4 50 34 CCOC(=O)c1ccc(CNC(=O)NCCc2cccc(Br)c2)cc1 ZINC000217502942 HH For-Sale Unstable PDS 61 43 CN(Cl)CCCN1c2ccccc2CCc2ccccc21 ZINC000217502972 DI For-Sale Unstable HRH1 17 76 CN(Cl)CCCN1c2ccccc2CCc2ccccc21 ZINC000217502972 DI For-Sale Unstable SLC22A2 18 76 CC(C)Nc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217502989 EG In-Stock Unstable AKR1C3 50 42 CC(C)Nc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217502989 EG In-Stock Unstable LIMK2 46 41 CCOC(=O)CN1CCO[C@H](COc2ccc([N+](=O)[O-])cc2)C1 ZINC000217503019 DD In-Stock Unstable SLC27A4 50 34 COC(=O)c1ccc(CNC(=O)NCCc2cccc(Br)c2)cc1 ZINC000217503044 GG For-Sale Unstable PDS 50 39 CCCCNc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217503095 EG In-Stock Unstable AKR1C3 44 38 CCCCNc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217503095 EG In-Stock Unstable LIMK2 42 39 CCCCCCNC(=O)c1cc(Br)ccc1O ZINC000217503110 DG For-Sale Unstable ASAH1 96 40 CCCCCCNC(=O)c1cc(Br)ccc1O ZINC000217503110 DG For-Sale Unstable PYK 100 47 CCCCCCNC(=O)c1cc(Br)ccc1O ZINC000217503110 DG For-Sale Unstable PSBA 0 40 O=S(=O)(NCCn1nc(-c2ccccn2)c2c1CCCC2)c1ccc2c(c1)OCCO2 ZINC000217503160 IF For-Sale Unstable PKM 22 40 CCCCC(=O)NCCCC[C@H](N)C(=O)O ZINC000217503161 BC In-Stock Unstable CNR1 0 46 CCCCC(=O)NCCCC[C@H](N)C(=O)O ZINC000217503161 BC In-Stock Unstable GRIA3 15 41 CCCCC(=O)NCCCC[C@H](N)C(=O)O ZINC000217503161 BC In-Stock Unstable NOS1 0 62 CCCCC(=O)NCCCC[C@H](N)C(=O)O ZINC000217503161 BC In-Stock Unstable NOS2 0 59 CCCCC(=O)NCCCC[C@H](N)C(=O)O ZINC000217503161 BC In-Stock Unstable GRM8 25 41 CCCCC(=O)NCCCC[C@H](N)C(=O)O ZINC000217503161 BC In-Stock Unstable GRIK3 42 41 CCCCC(=O)NCCCC[C@H](N)C(=O)O ZINC000217503161 BC In-Stock Unstable S1PR2 15 40 CCCCC(=O)NCCCC[C@H](N)C(=O)O ZINC000217503161 BC In-Stock Unstable NOS3 19 53 CCCCC(=O)NCCCC[C@H](N)C(=O)O ZINC000217503161 BC In-Stock Unstable EPHX2 28 50 CCCCC(=O)NCCCC[C@H](N)C(=O)O ZINC000217503161 BC In-Stock Unstable GRIK2 19 41 CCCCC(=O)NCCCC[C@H](N)C(=O)O ZINC000217503161 BC In-Stock Unstable GRIK1 43 47 CCCCC(=O)NCCCC[C@H](N)C(=O)O ZINC000217503161 BC In-Stock Unstable BHMT 56 36 CCCCC(=O)NCCCC[C@H](N)C(=O)O ZINC000217503161 BC In-Stock Unstable NOD1 129 73 CCCCC(=O)NCCCC[C@H](N)C(=O)O ZINC000217503161 BC In-Stock Unstable CQSS 42 36 CC(C)CNc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217503203 EG In-Stock Unstable PTGER4 0 42 CC(C)CNc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217503203 EG In-Stock Unstable MTNN 80 38 CC(C)CNc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217503203 EG In-Stock Unstable AKR1C3 43 38 CC(C)CNc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217503203 EG In-Stock Unstable LIMK2 42 39 O=C(NCCc1cccc(Br)c1)NCCc1cccc(Br)c1 ZINC000217503254 II For-Sale Unstable AMP1_PLAFQ 29 40 CC[C@@H](C)Nc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217503285 EG In-Stock Unstable AKR1C3 41 38 CC[C@@H](C)Nc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217503285 EG In-Stock Unstable LIMK2 42 39 CCCN1CC[C@@H](NC(=O)CN(C)Cc2cccnc2)C1 ZINC000217503348 CD In-Stock Unstable C3AR1 45 38 O=C(NCCc1ccc(Br)cc1)NCCc1cccc(Br)c1 ZINC000217503363 II For-Sale Unstable LIG1 0 41 O=C(NCCc1ccc(Br)cc1)NCCc1cccc(Br)c1 ZINC000217503363 II For-Sale Unstable CAN2 0 40 CC[C@H](C)Nc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217503373 EG In-Stock Unstable AKR1C3 41 38 CC[C@H](C)Nc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217503373 EG In-Stock Unstable LIMK2 42 39 CCCN1CC[C@H](NC(=O)CN(C)Cc2cccnc2)C1 ZINC000217503420 CD In-Stock Unstable C3AR1 45 38 Cc1ccc(NC(=O)NCCc2cccc(Br)c2)cn1 ZINC000217503462 EH For-Sale Unstable RAF1 34 41 Cc1ccc(NC(=O)NCCc2cccc(Br)c2)cn1 ZINC000217503462 EH For-Sale Unstable Q8MMZ8_EIMTE 22 41 Cc1ccc(NC(=O)NCCc2cccc(Br)c2)cn1 ZINC000217503462 EH For-Sale Unstable NAMPT 32 43 CC(C)(C)Nc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217503479 EG In-Stock Unstable LPL 32 40 CC(C)(C)Nc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217503479 EG In-Stock Unstable AKR1C3 57 41 CC(C)(C)Nc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217503479 EG In-Stock Unstable LIMK2 42 40 Cc1ccc(NC(=O)NCCc2cccc(Br)c2)nc1 ZINC000217503573 EH For-Sale Unstable GYRB 0 40 Cc1ccc(NC(=O)NCCc2cccc(Br)c2)nc1 ZINC000217503573 EH For-Sale Unstable LUCI_LUCLA 22 40 CCN1CCO[C@@H](COc2ccc([N+](=O)[O-])cc2)C1 ZINC000217503692 CD In-Stock Unstable KCNJ1 18 40 O=C(O)c1ccc(NC2CC2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217503707 EF In-Stock Unstable SFRP1 85 34 O=C(O)c1ccc(NC2CC2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217503707 EF In-Stock Unstable LIMK2 36 40 O=C(O)c1ccc(NC2CC2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217503707 EF In-Stock Unstable WNT3 58 32 CC[C@@H](c1ccccc1)N1CCC[C@@H](N)C1 ZINC000217503721 BF On-Demand Unstable OPRK1 0 46 O=C(Nc1ccc(I)cc1)c1cc(Br)ccc1I ZINC000217503752 KJ For-Sale Anodyne Q25615_ONCVO 92 60 O=C(Nc1ccc(I)cc1)c1cc(Br)ccc1I ZINC000217503752 KJ For-Sale Anodyne PSBA 0 41 CCN1CCO[C@H](COc2ccc([N+](=O)[O-])cc2)C1 ZINC000217503761 CD In-Stock Unstable KCNJ1 18 40 NC[C@@H]1CCCN([C@@H]2CCCCc3ccccc32)C1 ZINC000217503798 CG For-Sale Unstable SLC6A1 0 45 NC[C@@H]1CCCN([C@@H]2CCCCc3ccccc32)C1 ZINC000217503798 CG For-Sale Unstable HTR3B 0 41 O=C(NCCc1cccc(Br)c1)Nc1ccc(Br)cn1 ZINC000217503807 GH For-Sale Unstable POL 0 58 CC[C@H](c1ccccc1)N1CCC[C@@H](N)C1 ZINC000217503810 BF On-Demand Unstable OPRK1 0 46 O=C(O)c1ccc(NC2CCCC2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217503814 FH In-Stock Unstable CCR8 41 41 O=C(O)c1ccc(NC2CCCC2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217503814 FH In-Stock Unstable AKR1C3 27 40 O=C(O)c1ccc(NC2CCCC2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217503814 FH In-Stock Unstable SFRP1 82 33 O=C(O)c1ccc(NC2CCCC2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217503814 FH In-Stock Unstable LIMK2 46 39 O=C(O)c1ccc(NC2CCCC2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217503814 FH In-Stock Unstable WNT3 65 32 COc1ccc(SCc2cnn(-c3ccccc3)c2)cc1 ZINC000217503888 CI On-Demand Unstable GRM4 18 42 COc1ccc(SCc2cnn(-c3ccccc3)c2)cc1 ZINC000217503888 CI On-Demand Unstable NPBWR1 40 36 O=C(NCCc1cccc(Br)c1)Nc1ccc(Cl)cn1 ZINC000217503908 FH For-Sale Unstable POL 0 64 COc1ccc(CCS(=O)(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)cc1 ZINC000217503921 IF For-Sale Unstable TGFBR1 27 43 O=C(O)c1ccc(NC2CCCCC2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217503935 FH In-Stock Unstable EPHX2 21 40 O=C(O)c1ccc(NC2CCCCC2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217503935 FH In-Stock Unstable NS5B 0 40 O=C(O)c1ccc(NC2CCCCC2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217503935 FH In-Stock Unstable CCR8 38 42 O=C(O)c1ccc(NC2CCCCC2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217503935 FH In-Stock Unstable SFRP1 82 33 O=C(O)c1ccc(NC2CCCCC2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217503935 FH In-Stock Unstable LIMK2 42 39 O=C(O)c1ccc(NC2CCCCC2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217503935 FH In-Stock Unstable WNT3 62 33 CC[C@@H](C)[C@H](NC(=O)[C@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217503990 KG In-Stock Unstable BMP1 57 35 CC[C@@H](C)[C@H](NC(=O)[C@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217503990 KG In-Stock Unstable POL 0 42 Cc1ccccc1-c1nnc(SCc2cccc3cccnc23)n1Cc1ccco1 ZINC000217503997 HK On-Demand Unstable HCRTR2 15 44 O=C(NCCc1cccc(Br)c1)Nc1cc(Cl)ccn1 ZINC000217504008 FH For-Sale Unstable PPIA 21 40 O=C(O)c1ccc(NCCC2=CCCCC2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217504036 HI In-Stock Unstable LIMK2 41 39 CNCC(=O)c1ccc(S(C)(=O)=O)cc1F ZINC000217504037 BC For-Sale Unstable PTGS2 23 40 CNCC(=O)c1ccc(S(C)(=O)=O)cc1F ZINC000217504037 BC For-Sale Unstable LOX1.1 47 39 CNCC(=O)c1ccc(S(C)(=O)=O)cc1F ZINC000217504037 BC For-Sale Unstable O49150_SOLTU 49 39 COc1ccc(-n2ccnc2SCc2ccc3ccccc3n2)cc1 ZINC000217504112 EJ On-Demand Unstable CYSLTR1 40 41 COc1ccc(-n2ccnc2SCc2ccc3ccccc3n2)cc1 ZINC000217504112 EJ On-Demand Unstable PDE10A 32 45 O=C(NCCc1cccc(Br)c1)Nc1cc(Br)ccn1 ZINC000217504115 GH For-Sale Unstable TYK2 15 40 O=C(O)c1ccc(NCCO)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217504137 ED In-Stock Unstable AKR1C3 41 40 O=C(O)c1ccc(NCCO)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217504137 ED In-Stock Unstable LIMK2 44 42 O=C(NCCCc1ccccc1)NCCc1cccc(Br)c1 ZINC000217504221 FH For-Sale Unstable SDH1 0 48 O=C(NCCCc1ccccc1)NCCc1cccc(Br)c1 ZINC000217504221 FH For-Sale Unstable SCN5A 0 40 O=C(NCCCc1ccccc1)NCCc1cccc(Br)c1 ZINC000217504221 FH For-Sale Unstable HDA106 0 43 O=C(O)c1ccc(NCCCO)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217504241 FD In-Stock Unstable LIMK2 38 40 CS(=O)(=O)c1ccc(C(=O)CCN)c(F)c1 ZINC000217504244 BC For-Sale Unstable PTGS2 32 40 CS(=O)(=O)c1ccc(C(=O)CCN)c(F)c1 ZINC000217504244 BC For-Sale Unstable LOX1.1 49 40 CS(=O)(=O)c1ccc(C(=O)CCN)c(F)c1 ZINC000217504244 BC For-Sale Unstable O49150_SOLTU 52 40 O=[N+]([O-])c1ccc(OC[C@@H]2CN(Cc3ccccc3)CCO2)cc1 ZINC000217504275 EF In-Stock Unstable LTA4H 22 44 O=[N+]([O-])c1ccc(OC[C@@H]2CN(Cc3ccccc3)CCO2)cc1 ZINC000217504275 EF In-Stock Unstable SIGMAR1 26 64 O=[N+]([O-])c1ccc(OC[C@@H]2CN(Cc3ccccc3)CCO2)cc1 ZINC000217504275 EF In-Stock Unstable MGLL 0 50 O=[N+]([O-])c1ccc(OC[C@@H]2CN(Cc3ccccc3)CCO2)cc1 ZINC000217504275 EF In-Stock Unstable ABHD6 0 50 O=C(O)[C@@]12C[C@@H]3C[C@H](C1)C[C@@](n1ncc(Nc4cccc(C(F)(F)F)c4)c(Cl)c1=O)(C3)C2 ZINC000217504295 JK In-Stock Unstable TRPM4 0 41 OC[C@@H]1O[C@H](n2cccc2)[C@H](O)[C@@H]1O ZINC000217504298 AB For-Sale Unstable ADORA1 45 40 OC[C@@H]1O[C@H](n2cccc2)[C@H](O)[C@@H]1O ZINC000217504298 AB For-Sale Unstable SLC29A1 73 36 OC[C@@H]1O[C@H](n2cccc2)[C@H](O)[C@@H]1O ZINC000217504298 AB For-Sale Unstable ADORA2A 19 40 OC[C@@H]1O[C@H](n2cccc2)[C@H](O)[C@@H]1O ZINC000217504298 AB For-Sale Unstable ADK 29 40 OC[C@@H]1O[C@H](n2cccc2)[C@H](O)[C@@H]1O ZINC000217504298 AB For-Sale Unstable CDA 73 44 OC[C@@H]1O[C@H](n2cccc2)[C@H](O)[C@@H]1O ZINC000217504298 AB For-Sale Unstable ADORA3 17 40 OC[C@@H]1O[C@H](n2cccc2)[C@H](O)[C@@H]1O ZINC000217504298 AB For-Sale Unstable FIMH 77 42 C[C@@](O)(CNC(=O)c1cc(=O)c2ccccc2o1)c1cc2ccccc2s1 ZINC000217504322 GH In-Stock Unstable BCHE 33 43 COc1cccc(CN(C)C(=O)c2ccc(O)cc2O)c1 ZINC000217504324 CE On-Demand Unstable ROCK1 32 49 COc1cccc(CN(C)C(=O)c2ccc(O)cc2O)c1 ZINC000217504324 CE On-Demand Unstable MTNR1A 31 42 COc1cccc(CN(C)C(=O)c2ccc(O)cc2O)c1 ZINC000217504324 CE On-Demand Unstable MTNR1B 27 41 COc1cccc(CN(C)C(=O)c2ccc(O)cc2O)c1 ZINC000217504324 CE On-Demand Unstable ROCK2 40 44 COc1cccc(CN(C)C(=O)c2ccc(O)cc2O)c1 ZINC000217504324 CE On-Demand Unstable HSP90AB1 56 59 COc1cccc(CN(C)C(=O)c2ccc(O)cc2O)c1 ZINC000217504324 CE On-Demand Unstable HSD17B2 50 58 COc1cccc(CN(C)C(=O)c2ccc(O)cc2O)c1 ZINC000217504324 CE On-Demand Unstable CDC42BPA 0 44 N#Cc1cc(C(=O)Nc2ccccc2)c(N)nc1SCc1cnn(-c2ccccc2)c1 ZINC000217504336 II On-Demand Unstable ATR 46 36 O=C(NCCCCc1ccccc1)NCCc1cccc(Br)c1 ZINC000217504343 GI For-Sale Unstable SIGMAR1 16 44 O=C(NCCCCc1ccccc1)NCCc1cccc(Br)c1 ZINC000217504343 GI For-Sale Unstable SCN2A 17 43 O=C(NCCCCc1ccccc1)NCCc1cccc(Br)c1 ZINC000217504343 GI For-Sale Unstable MTNR1A 32 47 O=C(NCCCCc1ccccc1)NCCc1cccc(Br)c1 ZINC000217504343 GI For-Sale Unstable MTNR1B 31 47 O=C(NCCCCc1ccccc1)NCCc1cccc(Br)c1 ZINC000217504343 GI For-Sale Unstable FAAH 39 48 O=C(NCCCCc1ccccc1)NCCc1cccc(Br)c1 ZINC000217504343 GI For-Sale Unstable SCN5A 0 43 O=C(NCCCCc1ccccc1)NCCc1cccc(Br)c1 ZINC000217504343 GI For-Sale Unstable SLC6A5 23 47 O=C(NCCCCc1ccccc1)NCCc1cccc(Br)c1 ZINC000217504343 GI For-Sale Unstable CES1 45 36 O=C(NCCCCc1ccccc1)NCCc1cccc(Br)c1 ZINC000217504343 GI For-Sale Unstable AMP1_PLAFQ 33 48 O=C(NCCCCc1ccccc1)NCCc1cccc(Br)c1 ZINC000217504343 GI For-Sale Unstable HDA106 0 43 O=C(NCCCCc1ccccc1)NCCc1cccc(Br)c1 ZINC000217504343 GI For-Sale Unstable CRTM 55 43 O=[N+]([O-])c1ccc(OC[C@H]2CN(Cc3ccccc3)CCO2)cc1 ZINC000217504350 EF In-Stock Unstable LTA4H 22 44 O=[N+]([O-])c1ccc(OC[C@H]2CN(Cc3ccccc3)CCO2)cc1 ZINC000217504350 EF In-Stock Unstable SIGMAR1 26 64 O=[N+]([O-])c1ccc(OC[C@H]2CN(Cc3ccccc3)CCO2)cc1 ZINC000217504350 EF In-Stock Unstable MGLL 0 50 O=[N+]([O-])c1ccc(OC[C@H]2CN(Cc3ccccc3)CCO2)cc1 ZINC000217504350 EF In-Stock Unstable ABHD6 0 50 COCCNc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217504354 FE In-Stock Unstable CPT1A 43 30 COCCNc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217504354 FE In-Stock Unstable AKR1C3 48 37 COCCNc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217504354 FE In-Stock Unstable LIMK2 42 42 CS(=O)(=O)c1ccc(C(=O)CCN)cc1F ZINC000217504360 BC For-Sale Unstable LOX1.1 32 40 CS(=O)(=O)c1ccc(C(=O)CCN)cc1F ZINC000217504360 BC For-Sale Unstable O49150_SOLTU 31 40 NC(=O)C[C@H](NC(=O)[C@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217504367 KC In-Stock Unstable SSTR4 44 31 NC(=O)C[C@H](NC(=O)[C@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217504367 KC In-Stock Unstable CCKAR 48 35 O=C(O)[C@]12C[C@@H]3C[C@H](C1)C[C@](n1ncc(Nc4cccc(C(F)(F)F)c4)c(Cl)c1=O)(C3)C2 ZINC000217504373 JK In-Stock Unstable TRPM4 0 41 COc1ccc(S(=O)(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)c(OC)c1 ZINC000217504378 IF For-Sale Unstable TGFBR1 33 40 C[C@](O)(CNC(=O)c1cc(=O)c2ccccc2o1)c1cc2ccccc2s1 ZINC000217504420 GH In-Stock Unstable BCHE 33 43 OC[C@@H]1O[C@H](n2cccc2)[C@@H](O)[C@@H]1O ZINC000217504452 AB For-Sale Unstable ADORA1 45 40 OC[C@@H]1O[C@H](n2cccc2)[C@@H](O)[C@@H]1O ZINC000217504452 AB For-Sale Unstable SLC29A1 73 36 OC[C@@H]1O[C@H](n2cccc2)[C@@H](O)[C@@H]1O ZINC000217504452 AB For-Sale Unstable ADORA2A 19 40 OC[C@@H]1O[C@H](n2cccc2)[C@@H](O)[C@@H]1O ZINC000217504452 AB For-Sale Unstable ADK 29 40 OC[C@@H]1O[C@H](n2cccc2)[C@@H](O)[C@@H]1O ZINC000217504452 AB For-Sale Unstable CDA 73 44 OC[C@@H]1O[C@H](n2cccc2)[C@@H](O)[C@@H]1O ZINC000217504452 AB For-Sale Unstable ADORA3 17 40 OC[C@@H]1O[C@H](n2cccc2)[C@@H](O)[C@@H]1O ZINC000217504452 AB For-Sale Unstable FIMH 77 42 COCCCNc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217504465 FF In-Stock Unstable AKR1C3 42 36 COCCCNc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217504465 FF In-Stock Unstable LIMK2 38 41 C[C@H](N)C(=O)c1ccc(S(C)(=O)=O)cc1F ZINC000217504480 BC For-Sale Unstable PTGS2 28 44 CCOc1ccc(S(=O)(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)cc1F ZINC000217504502 IG For-Sale Unstable BUB1 48 34 COc1cccc(CN(C)C(=O)c2cc(I)ccc2O)c1 ZINC000217504505 GG On-Demand Unstable ROCK1 31 48 COc1cccc(CN(C)C(=O)c2cc(I)ccc2O)c1 ZINC000217504505 GG On-Demand Unstable MTNR1A 32 41 COc1cccc(CN(C)C(=O)c2cc(I)ccc2O)c1 ZINC000217504505 GG On-Demand Unstable MTNR1B 33 41 COc1cccc(CN(C)C(=O)c2cc(I)ccc2O)c1 ZINC000217504505 GG On-Demand Unstable ROCK2 39 48 COc1cccc(CN(C)C(=O)c2cc(I)ccc2O)c1 ZINC000217504505 GG On-Demand Unstable HSP90AB1 50 55 COc1cccc(CN(C)C(=O)c2cc(I)ccc2O)c1 ZINC000217504505 GG On-Demand Unstable HSD17B2 46 56 COc1cccc(CN(C)C(=O)c2cc(I)ccc2O)c1 ZINC000217504505 GG On-Demand Unstable CDC42BPA 0 42 CC(=O)c1ccc(OCC2CC2)cc1F ZINC000217504534 BF On-Demand Unstable SHC 24 44 CC(=O)c1ccc(OCC2CC2)cc1F ZINC000217504534 BF On-Demand Unstable CHRNA10 40 41 COc1ccc(CC(=O)NC[C@@](C)(O)c2cc3ccccc3s2)cc1OC ZINC000217504546 GG In-Stock Unstable TRPV1 23 44 COc1ccc(CC(=O)NC[C@@](C)(O)c2cc3ccccc3s2)cc1OC ZINC000217504546 GG In-Stock Unstable MT-ND1 25 40 COc1ccc(CC(=O)NC[C@@](C)(O)c2cc3ccccc3s2)cc1OC ZINC000217504546 GG In-Stock Unstable NCE103 19 44 COc1ccc(CC(=O)NC[C@@](C)(O)c2cc3ccccc3s2)cc1OC ZINC000217504546 GG In-Stock Unstable CAN2 0 44 C[C@@H](N)C(=O)c1ccc(S(C)(=O)=O)cc1F ZINC000217504566 BC For-Sale Unstable PTGS2 28 44 O=C(O)c1ccc(NCc2ccccc2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217504572 GH In-Stock Unstable AKR1C3 41 40 O=C(O)c1ccc(NCc2ccccc2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217504572 GH In-Stock Unstable REP 0 40 O=C(O)c1ccc(NCc2ccccc2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217504572 GH In-Stock Unstable LIMK2 55 43 CC(C)(C)c1ccc(-c2nnc(SCc3cnn(-c4ccccc4)c3)o2)cc1 ZINC000217504580 GK On-Demand Unstable TYMS 0 43 CC(C)(C)c1ccc(-c2nnc(SCc3cnn(-c4ccccc4)c3)o2)cc1 ZINC000217504580 GK On-Demand Unstable GSK3B 18 48 CC(C)(C)c1ccc(-c2nnc(SCc3cnn(-c4ccccc4)c3)o2)cc1 ZINC000217504580 GK On-Demand Unstable GSK3A 51 48 CC(C)(C)c1ccc(-c2nnc(SCc3cnn(-c4ccccc4)c3)o2)cc1 ZINC000217504580 GK On-Demand Unstable TERT 26 43 COc1ccc(Nc2cc(C)nc(Nc3ccc(N)cc3)n2)cc1 ZINC000217504585 DH In-Stock Unstable GALR2 67 45 COc1ccc(Nc2cc(C)nc(Nc3ccc(N)cc3)n2)cc1 ZINC000217504585 DH In-Stock Unstable AGPAT2 40 38 COc1ccc(CC(=O)NC[C@](C)(O)c2cc3ccccc3s2)cc1OC ZINC000217504625 GG In-Stock Unstable TRPV1 23 44 COc1ccc(CC(=O)NC[C@](C)(O)c2cc3ccccc3s2)cc1OC ZINC000217504625 GG In-Stock Unstable MT-ND1 25 40 COc1ccc(CC(=O)NC[C@](C)(O)c2cc3ccccc3s2)cc1OC ZINC000217504625 GG In-Stock Unstable NCE103 19 44 COc1ccc(CC(=O)NC[C@](C)(O)c2cc3ccccc3s2)cc1OC ZINC000217504625 GG In-Stock Unstable CAN2 0 44 CS(=O)(=O)N1CCN(C(=O)NCCc2cccc(Br)c2)CC1 ZINC000217504648 GD On-Demand Unstable TRY2_BOVIN 37 40 CS(=O)(=O)N1CCN(C(=O)NCCc2cccc(Br)c2)CC1 ZINC000217504648 GD On-Demand Unstable HPN 32 42 C[C@@H](Nc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1)c1ccccc1 ZINC000217504680 GI In-Stock Unstable LDHB 0 41 C[C@@H](Nc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1)c1ccccc1 ZINC000217504680 GI In-Stock Unstable LIMK2 27 45 Cc1cc(N2CCCC2)nc(Nc2ccc(N)cc2)n1 ZINC000217504695 CF In-Stock Unstable GALR2 59 47 Cc1cc(N2CCCC2)nc(Nc2ccc(N)cc2)n1 ZINC000217504695 CF In-Stock Unstable TERT 21 40 COc1cccc(NCc2nnc(SCc3cnn(-c4ccccc4)c3)n2C2CCCCC2)c1 ZINC000217504704 JK On-Demand Unstable VCP 42 39 COc1ccc(Cl)cc1S(=O)(=O)NCCn1nc(-c2ccccn2)c2c1CCCC2 ZINC000217504715 IG For-Sale Unstable CPT1A 49 35 COc1ccc(Cl)cc1S(=O)(=O)NCCn1nc(-c2ccccn2)c2c1CCCC2 ZINC000217504715 IG For-Sale Unstable CPT1B 43 35 O=C(NCCc1cccc(Br)c1)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217504744 JF For-Sale Unstable TRY2_BOVIN 23 40 O=C(NCCc1cccc(Br)c1)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217504744 JF For-Sale Unstable TGM2 72 43 O=C(NCCc1cccc(Br)c1)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217504744 JF For-Sale Unstable F13A1 83 43 O=C(NCCc1cccc(Br)c1)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217504744 JF For-Sale Unstable AKR1C3 51 39 O=C(NCCc1cccc(Br)c1)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217504744 JF For-Sale Unstable NAMPT 40 37 O=C(NCCc1cccc(Br)c1)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217504744 JF For-Sale Unstable HPN 33 43 C[C@H](Nc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1)c1ccccc1 ZINC000217504755 GI In-Stock Unstable LDHB 0 41 C[C@H](Nc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1)c1ccccc1 ZINC000217504755 GI In-Stock Unstable LIMK2 27 45 Cc1cc(N2CCOCC2)nc(Nc2ccc(N)cc2)n1 ZINC000217504800 CD In-Stock Unstable GALR2 43 38 Cc1cc(N2CCOCC2)nc(Nc2ccc(N)cc2)n1 ZINC000217504800 CD In-Stock Unstable EPHB4 79 38 Cc1cc(N2CCOCC2)nc(Nc2ccc(N)cc2)n1 ZINC000217504800 CD In-Stock Unstable STAT6 56 34 Cc1cc(N2CCOCC2)nc(Nc2ccc(N)cc2)n1 ZINC000217504800 CD In-Stock Unstable SMG1 49 42 O=S(=O)(NCCn1nc(-c2ccccn2)c2c1CCCC2)c1ccc(C(F)(F)F)cc1 ZINC000217504828 JH For-Sale Unstable OXTR 29 43 Cc1ccc(S(=O)(=O)N2CCN(C(=O)NCCc3cccc(Br)c3)CC2)cc1 ZINC000217504832 JG For-Sale Unstable TRY2_BOVIN 26 42 Cc1ccc(S(=O)(=O)N2CCN(C(=O)NCCc3cccc(Br)c3)CC2)cc1 ZINC000217504832 JG For-Sale Unstable MMP3 16 46 Cc1ccc(S(=O)(=O)N2CCN(C(=O)NCCc3cccc(Br)c3)CC2)cc1 ZINC000217504832 JG For-Sale Unstable TGM2 67 41 Cc1ccc(S(=O)(=O)N2CCN(C(=O)NCCc3cccc(Br)c3)CC2)cc1 ZINC000217504832 JG For-Sale Unstable MMP7 16 46 Cc1ccc(S(=O)(=O)N2CCN(C(=O)NCCc3cccc(Br)c3)CC2)cc1 ZINC000217504832 JG For-Sale Unstable F13A1 79 39 Cc1ccc(S(=O)(=O)N2CCN(C(=O)NCCc3cccc(Br)c3)CC2)cc1 ZINC000217504832 JG For-Sale Unstable NAMPT 39 40 Cc1ccc(S(=O)(=O)N2CCN(C(=O)NCCc3cccc(Br)c3)CC2)cc1 ZINC000217504832 JG For-Sale Unstable HPN 34 49 O=C(O)c1ccc(NCCc2ccccc2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217504873 GH In-Stock Unstable AKR1C3 38 50 O=C(O)c1ccc(NCCc2ccccc2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217504873 GH In-Stock Unstable LIMK2 58 44 COC(=O)[C@@H](NC(=O)c1cc(Br)ccc1O)C(C)C ZINC000217504887 EE On-Demand Unstable PYK 94 39 Cc1ccc(Nc2cc(C)nc(N3CCNCC3)n2)cc1 ZINC000217504902 CE In-Stock Unstable GALR2 25 43 Cc1ccc(Nc2cc(C)nc(N3CCNCC3)n2)cc1 ZINC000217504902 CE In-Stock Unstable KARS 54 35 C[C@@](O)(CNC(=O)c1ccccc1Br)c1cc2ccccc2s1 ZINC000217504908 GI In-Stock Unstable ECR 19 40 COC(=O)[C@H](NC(=O)c1cc(Br)ccc1O)C(C)C ZINC000217504946 EE For-Sale Unstable PYK 94 39 O=C(N[C@@]12C[C@@H]3C[C@@H](C[C@@](Cl)(C3)C1)C2)N1CCOCC1 ZINC000217504961 CE In-Stock Unstable EPHX2 16 43 COc1ccc(CCNc2ccc(C(=O)O)cc2S(=O)(=O)Nc2ccccc2)cc1 ZINC000217504962 IH In-Stock Unstable ADRB2 39 41 COc1ccc(CCNc2ccc(C(=O)O)cc2S(=O)(=O)Nc2ccccc2)cc1 ZINC000217504962 IH In-Stock Unstable ADRB1 32 41 COc1ccc(CCNc2ccc(C(=O)O)cc2S(=O)(=O)Nc2ccccc2)cc1 ZINC000217504962 IH In-Stock Unstable CYSLTR1 17 41 COc1ccc(CCNc2ccc(C(=O)O)cc2S(=O)(=O)Nc2ccccc2)cc1 ZINC000217504962 IH In-Stock Unstable ADRB3 54 41 COc1ccc(CCNc2ccc(C(=O)O)cc2S(=O)(=O)Nc2ccccc2)cc1 ZINC000217504962 IH In-Stock Unstable BMP1 33 42 COc1ccc(CCNc2ccc(C(=O)O)cc2S(=O)(=O)Nc2ccccc2)cc1 ZINC000217504962 IH In-Stock Unstable PRTN3 44 31 COc1ccc(CCNc2ccc(C(=O)O)cc2S(=O)(=O)Nc2ccccc2)cc1 ZINC000217504962 IH In-Stock Unstable PTPRB 54 39 COc1ccc(CCNc2ccc(C(=O)O)cc2S(=O)(=O)Nc2ccccc2)cc1 ZINC000217504962 IH In-Stock Unstable PTGDR 38 42 COc1ccc(CCNc2ccc(C(=O)O)cc2S(=O)(=O)Nc2ccccc2)cc1 ZINC000217504962 IH In-Stock Unstable AKR1C3 46 44 COc1ccc(CCNc2ccc(C(=O)O)cc2S(=O)(=O)Nc2ccccc2)cc1 ZINC000217504962 IH In-Stock Unstable AKR1C2 48 38 COc1ccc(CCNc2ccc(C(=O)O)cc2S(=O)(=O)Nc2ccccc2)cc1 ZINC000217504962 IH In-Stock Unstable LIMK2 43 43 C[C@](O)(CNC(=O)c1ccccc1Br)c1cc2ccccc2s1 ZINC000217504988 GI In-Stock Unstable ECR 19 40 COc1ccc(Nc2cc(C)nc(N3CCNCC3)n2)cc1 ZINC000217505014 CD In-Stock Unstable GALR2 63 57 CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217505030 KG In-Stock Unstable PGC 49 31 CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217505030 KG In-Stock Unstable FCER2 57 33 CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217505030 KG In-Stock Unstable SSTR4 44 33 CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217505030 KG In-Stock Unstable CCKAR 17 40 CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217505030 KG In-Stock Unstable TIMP3 45 35 CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217505030 KG In-Stock Unstable CAPNS1 61 35 CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217505030 KG In-Stock Unstable HLA-DRB1 52 33 CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217505030 KG In-Stock Unstable REN 68 40 CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217505030 KG In-Stock Unstable CAPN1 74 39 CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217505030 KG In-Stock Unstable CAPN2 107 39 CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217505030 KG In-Stock Unstable FPR1 78 39 CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217505030 KG In-Stock Unstable NPR 79 35 CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217505030 KG In-Stock Unstable KISS1R 55 32 COc1ccc(CCNc2ccc(C(=O)O)cc2S(=O)(=O)Nc2ccccc2)cc1OC ZINC000217505069 JH In-Stock Unstable COLA 44 43 COc1ccc(CCNc2ccc(C(=O)O)cc2S(=O)(=O)Nc2ccccc2)cc1OC ZINC000217505069 JH In-Stock Unstable CPT1A 46 32 COc1ccc(CCNc2ccc(C(=O)O)cc2S(=O)(=O)Nc2ccccc2)cc1OC ZINC000217505069 JH In-Stock Unstable PTPRB 42 36 COc1ccc(CCNc2ccc(C(=O)O)cc2S(=O)(=O)Nc2ccccc2)cc1OC ZINC000217505069 JH In-Stock Unstable PTGDR 36 40 COc1ccc(CCNc2ccc(C(=O)O)cc2S(=O)(=O)Nc2ccccc2)cc1OC ZINC000217505069 JH In-Stock Unstable PTGDR2 21 40 COc1ccc(CCNc2ccc(C(=O)O)cc2S(=O)(=O)Nc2ccccc2)cc1OC ZINC000217505069 JH In-Stock Unstable AKR1C3 30 41 COc1ccc(CCNc2ccc(C(=O)O)cc2S(=O)(=O)Nc2ccccc2)cc1OC ZINC000217505069 JH In-Stock Unstable SCMU_MYCTU 0 50 Cc1cc(N2CCN(C)CC2)nc(N2CCNCC2)n1 ZINC000217505126 CB In-Stock Unstable HRH4 56 56 Cc1cc(N2CCN(C)CC2)nc(N2CCNCC2)n1 ZINC000217505126 CB In-Stock Unstable SORD 23 41 C[C@@H]1CN(C[C@@H](O)COc2cccc(CN)c2)CCCO1 ZINC000217505167 CC For-Sale Unstable ACOX1 71 32 C[C@@H]1CN(C[C@@H](O)COc2cccc(CN)c2)CCCO1 ZINC000217505167 CC For-Sale Unstable ABCB1 57 46 CCOC(=O)NCCNC(=O)NCCc1cccc(Br)c1 ZINC000217505170 FE For-Sale Unstable PDS 40 39 NCCNc1ccc(Nc2ccccn2)nn1 ZINC000217505239 BC In-Stock Unstable KARS 19 42 C[C@H]1CN(C[C@@H](O)COc2cccc(CN)c2)CCCO1 ZINC000217505243 CC For-Sale Unstable ACOX1 71 32 C[C@H]1CN(C[C@@H](O)COc2cccc(CN)c2)CCCO1 ZINC000217505243 CC For-Sale Unstable ABCB1 57 46 O=C(O)c1ccc(NC[C@@H]2CCCO2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217505276 GF In-Stock Unstable TNK2 56 39 CC(C)(C)OC(=O)N(CCN)C(=O)NCCc1cccc(Br)c1 ZINC000217505283 GF For-Sale Unstable PAPA1_CARPA 16 42 C[C@@H]1CN(C[C@@H](O)COc2ccc(CN)cc2)CCCO1 ZINC000217505340 CC For-Sale Unstable ACOX1 42 30 C[C@@H]1CN(C[C@@H](O)COc2ccc(CN)cc2)CCCO1 ZINC000217505340 CC For-Sale Unstable ABCB1 41 42 O=C(O)c1ccc(NC[C@H]2CCCO2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217505358 GF In-Stock Unstable TNK2 56 39 CC(C)(C)OC(=O)N1CCN(C(=O)NCCc2cccc(Br)c2)CC1 ZINC000217505401 HG For-Sale Unstable GPR119 37 43 C[C@H]1CN(C[C@@H](O)COc2ccc(CN)cc2)CCCO1 ZINC000217505421 CC For-Sale Unstable ACOX1 42 30 C[C@H]1CN(C[C@@H](O)COc2ccc(CN)cc2)CCCO1 ZINC000217505421 CC For-Sale Unstable ABCB1 41 42 c1cc(Nc2ccc(N3CCNCC3)nn2)ccn1 ZINC000217505441 CD In-Stock Unstable PRKD1 44 43 c1cc(Nc2ccc(N3CCNCC3)nn2)ccn1 ZINC000217505441 CD In-Stock Unstable PKD2 0 43 c1cc(Nc2ccc(N3CCNCC3)nn2)ccn1 ZINC000217505441 CD In-Stock Unstable KARS 55 35 C[C@@H](CCc1ccccc1)N1CCC[C@@H](CN)C1 ZINC000217505475 BF For-Sale Unstable ACE 35 41 C[C@@H](CCc1ccccc1)N1CCC[C@@H](CN)C1 ZINC000217505475 BF For-Sale Unstable SLC18A2 45 39 C[C@@H](CCc1ccccc1)N1CCC[C@@H](CN)C1 ZINC000217505475 BF For-Sale Unstable SIGMAR1 19 42 O=C(O)c1ccc(N2CCCC2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217505478 EF In-Stock Unstable KCNQ2 70 37 O=C(O)c1ccc(N2CCCC2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217505478 EF In-Stock Unstable TAAR1 28 43 O=C(O)c1ccc(N2CCCC2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217505478 EF In-Stock Unstable AKR1C3 36 42 O=C(O)c1ccc(N2CCCC2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217505478 EF In-Stock Unstable SFRP1 71 34 O=C(O)c1ccc(N2CCCC2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217505478 EF In-Stock Unstable LIMK2 45 41 O=C(O)c1ccc(N2CCCC2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217505478 EF In-Stock Unstable WNT3 59 32 CC(C)(C)OC(=O)N1CCC(NC(=O)NCCc2cccc(Br)c2)CC1 ZINC000217505514 IH For-Sale Unstable SIGMAR1 16 47 CC(C)(C)OC(=O)N1CCC(NC(=O)NCCc2cccc(Br)c2)CC1 ZINC000217505514 IH For-Sale Unstable EPHX2 38 45 CC(C)(C)OC(=O)N1CCC(NC(=O)NCCc2cccc(Br)c2)CC1 ZINC000217505514 IH For-Sale Unstable GPR119 42 46 N[C@@H]1CCCN([C@@H](c2ccccc2)c2ccc(F)cc2)C1 ZINC000217505515 CG For-Sale Unstable OPRL1 22 45 N[C@@H]1CCCN([C@@H](c2ccccc2)c2ccc(F)cc2)C1 ZINC000217505515 CG For-Sale Unstable SLC6A3 32 40 C/C(=N/O)c1ccc2[nH]ncc2c1 ZINC000217505552 AD For-Sale Unstable MAOB 16 45 C/C(=N/O)c1ccc2[nH]ncc2c1 ZINC000217505552 AD For-Sale Unstable JAK2 20 45 C/C(=N/O)c1ccc2[nH]ncc2c1 ZINC000217505552 AD For-Sale Unstable ROCK2 39 45 C[C@H](CCc1ccccc1)N1CCC[C@@H](CN)C1 ZINC000217505557 BF For-Sale Unstable ACE 35 41 C[C@H](CCc1ccccc1)N1CCC[C@@H](CN)C1 ZINC000217505557 BF For-Sale Unstable SLC18A2 45 39 C[C@H](CCc1ccccc1)N1CCC[C@@H](CN)C1 ZINC000217505557 BF For-Sale Unstable SIGMAR1 19 42 O=C(O)c1ccc(N2CCCCC2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217505580 FG In-Stock Unstable KCNQ2 66 36 O=C(O)c1ccc(N2CCCCC2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217505580 FG In-Stock Unstable TAAR1 28 42 O=C(O)c1ccc(N2CCCCC2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217505580 FG In-Stock Unstable AKR1C3 32 42 O=C(O)c1ccc(N2CCCCC2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217505580 FG In-Stock Unstable SFRP1 65 33 O=C(O)c1ccc(N2CCCCC2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217505580 FG In-Stock Unstable LIMK2 41 40 O=C(O)c1ccc(N2CCCCC2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217505580 FG In-Stock Unstable WNT3 50 32 O=C(O)c1ccc(N2CCCCC2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217505580 FG In-Stock Unstable BRPF1 0 41 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable ADRB1 35 42 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable DRD4 43 33 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable HRH2 24 45 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable CYSLTR1 17 40 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable PPIA 28 41 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable ADRB3 33 42 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable LDHA 37 40 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable BMP1 30 41 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable NQO2 43 46 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable CA1 24 47 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable TRPV1 24 54 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable PTGER3 15 44 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable MMP13 18 44 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable CCKAR 34 50 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable CCR3 59 47 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable RAF1 64 46 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable MTNR1A 112 45 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable MTNR1B 97 47 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable ROCK2 31 57 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable CCKBR 35 50 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable EPHX2 33 42 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable FLT4 19 41 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable CA12 17 47 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable PTGDR 31 52 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable CA9 19 47 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable MCHR1 28 44 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable Q8MMZ8_EIMTE 53 46 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable TAAR1 41 37 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable AKR1C3 61 57 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable NCE103 30 47 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable AKR1C2 52 37 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable IMDH_CRYPV 27 42 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable KDM4E 21 42 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable KCNK3 96 44 COc1ccc(CCNC(=O)Nc2cccc(C(=O)O)c2)cc1 ZINC000217505624 DF For-Sale Unstable KCNK9 62 34 O=C(O)c1ccc(N2CCOCC2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217505690 FE In-Stock Unstable MTOR 24 43 O=C(O)c1ccc(N2CCOCC2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217505690 FE In-Stock Unstable PIK3CG 0 43 O=C(O)c1ccc(N2CCOCC2)c(S(=O)(=O)Nc2ccccc2)c1 ZINC000217505690 FE In-Stock Unstable PIK3C2B 0 47 COc1ccc(CCNC(=O)N(C(C)=O)c2ccc(N)cc2)cc1 ZINC000217505724 EF For-Sale Unstable MTNR1A 53 38 COc1ccc(CCNC(=O)N(C(C)=O)c2ccc(N)cc2)cc1 ZINC000217505724 EF For-Sale Unstable MTNR1B 44 38 CCOc1ccccc1[C@H](O)[C@@]1(N(C)C)CCC[C@@H](C)C1 ZINC000217505748 CH For-Sale Unstable HCN1 41 31 CCOc1ccccc1[C@H](O)[C@@]1(N(C)C)CCC[C@@H](C)C1 ZINC000217505748 CH For-Sale Unstable HCN4 41 31 C[C@@H](c1cccc(F)c1)N1CCC[C@@H](N)C1 ZINC000217505786 BE On-Demand Unstable CHRNA10 44 41 COc1ccc(CCNC(=O)Nc2ccc(NC(C)=O)cc2)cc1 ZINC000217505811 EG On-Demand Unstable CA2 24 54 COc1ccc(CCNC(=O)Nc2ccc(NC(C)=O)cc2)cc1 ZINC000217505811 EG On-Demand Unstable ADRB1 26 45 COc1ccc(CCNC(=O)Nc2ccc(NC(C)=O)cc2)cc1 ZINC000217505811 EG On-Demand Unstable TSHR 49 34 COc1ccc(CCNC(=O)Nc2ccc(NC(C)=O)cc2)cc1 ZINC000217505811 EG On-Demand Unstable ADRB3 38 41 COc1ccc(CCNC(=O)Nc2ccc(NC(C)=O)cc2)cc1 ZINC000217505811 EG On-Demand Unstable BMP1 28 46 COc1ccc(CCNC(=O)Nc2ccc(NC(C)=O)cc2)cc1 ZINC000217505811 EG On-Demand Unstable NQO2 58 39 COc1ccc(CCNC(=O)Nc2ccc(NC(C)=O)cc2)cc1 ZINC000217505811 EG On-Demand Unstable CA1 49 54 COc1ccc(CCNC(=O)Nc2ccc(NC(C)=O)cc2)cc1 ZINC000217505811 EG On-Demand Unstable RAF1 54 43 COc1ccc(CCNC(=O)Nc2ccc(NC(C)=O)cc2)cc1 ZINC000217505811 EG On-Demand Unstable MTNR1A 95 47 COc1ccc(CCNC(=O)Nc2ccc(NC(C)=O)cc2)cc1 ZINC000217505811 EG On-Demand Unstable MTNR1B 75 43 COc1ccc(CCNC(=O)Nc2ccc(NC(C)=O)cc2)cc1 ZINC000217505811 EG On-Demand Unstable ACR 30 41 COc1ccc(CCNC(=O)Nc2ccc(NC(C)=O)cc2)cc1 ZINC000217505811 EG On-Demand Unstable CA12 33 54 COc1ccc(CCNC(=O)Nc2ccc(NC(C)=O)cc2)cc1 ZINC000217505811 EG On-Demand Unstable PTGDR 23 46 COc1ccc(CCNC(=O)Nc2ccc(NC(C)=O)cc2)cc1 ZINC000217505811 EG On-Demand Unstable CA9 33 54 COc1ccc(CCNC(=O)Nc2ccc(NC(C)=O)cc2)cc1 ZINC000217505811 EG On-Demand Unstable Q8MMZ8_EIMTE 44 43 COc1ccc(CCNC(=O)Nc2ccc(NC(C)=O)cc2)cc1 ZINC000217505811 EG On-Demand Unstable IDO1 30 50 COc1ccc(CCNC(=O)Nc2ccc(NC(C)=O)cc2)cc1 ZINC000217505811 EG On-Demand Unstable NCE103 40 54 COc1ccc(CCNC(=O)Nc2ccc(NC(C)=O)cc2)cc1 ZINC000217505811 EG On-Demand Unstable PROKR1 43 31 C[C@H](c1cccc(F)c1)N1CCC[C@@H](N)C1 ZINC000217505859 BE On-Demand Unstable CHRNA10 44 41 C[C@@](O)(CNC(=O)C1c2ccccc2Oc2ccccc21)c1cc2ccccc2s1 ZINC000217505873 HK For-Sale Unstable GRM8 42 34 CN(Cc1ccccc1Br)C(=O)c1cc(I)ccc1O ZINC000217505907 II For-Sale Unstable HSP90AB1 17 52 CCOc1ccccc1[C@H](O)[C@]1(N(C)C)CCC[C@@H](C)C1 ZINC000217505916 CH For-Sale Unstable HCN1 41 31 CCOc1ccccc1[C@H](O)[C@]1(N(C)C)CCC[C@@H](C)C1 ZINC000217505916 CH For-Sale Unstable HCN4 41 31 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable CA2 57 56 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable ADRB2 34 45 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable ADRB1 38 45 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable ADRB3 42 45 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable BMP1 90 52 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable CA1 68 56 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable CA7 29 47 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable MMP13 64 42 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable RAF1 42 41 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable CA4 25 55 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable CA5A 23 47 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable CA14 37 47 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable MTNR1A 64 41 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable MTNR1B 52 38 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable MMP2 42 47 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable MMP3 62 43 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable MMP8 42 47 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable MMP14 15 47 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable PTPRB 58 43 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable MMP9 62 47 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable EPHX2 18 40 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable MMP12 33 42 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable TGM2 15 43 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable CA12 70 56 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable PTGDR 15 42 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable MMP7 49 43 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable CA9 74 56 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable MMP1 68 47 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable Q8MMZ8_EIMTE 34 41 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable IDO1 30 48 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable NCE103 54 55 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable MTCA1 43 45 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable P96878_MYCTU 62 45 COc1ccc(CCNC(=O)Nc2ccc(S(=O)(=O)O)cc2)cc1 ZINC000217505922 FE For-Sale Unstable NAMPT 42 44 C[C@](O)(CNC(=O)C1c2ccccc2Oc2ccccc21)c1cc2ccccc2s1 ZINC000217505953 HK For-Sale Unstable GRM8 42 34 CCCCCNc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217506013 FH In-Stock Unstable ADRB2 0 45 CCCCCNc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217506013 FH In-Stock Unstable ADRB1 0 45 CCCCCNc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217506013 FH In-Stock Unstable PLA2G4B 41 34 CCCCCNc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217506013 FH In-Stock Unstable AKR1C3 43 37 CCCCCNc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217506013 FH In-Stock Unstable LIMK2 41 38 COc1ccc(CCNC(=O)Nc2cccc(S(=O)(=O)O)c2)cc1 ZINC000217506028 FE For-Sale Unstable CA2 33 51 COc1ccc(CCNC(=O)Nc2cccc(S(=O)(=O)O)c2)cc1 ZINC000217506028 FE For-Sale Unstable HRH2 17 43 COc1ccc(CCNC(=O)Nc2cccc(S(=O)(=O)O)c2)cc1 ZINC000217506028 FE For-Sale Unstable BMP1 70 46 COc1ccc(CCNC(=O)Nc2cccc(S(=O)(=O)O)c2)cc1 ZINC000217506028 FE For-Sale Unstable NQO2 48 42 COc1ccc(CCNC(=O)Nc2cccc(S(=O)(=O)O)c2)cc1 ZINC000217506028 FE For-Sale Unstable CA1 37 49 COc1ccc(CCNC(=O)Nc2cccc(S(=O)(=O)O)c2)cc1 ZINC000217506028 FE For-Sale Unstable TRPV1 0 53 COc1ccc(CCNC(=O)Nc2cccc(S(=O)(=O)O)c2)cc1 ZINC000217506028 FE For-Sale Unstable MMP13 42 39 COc1ccc(CCNC(=O)Nc2cccc(S(=O)(=O)O)c2)cc1 ZINC000217506028 FE For-Sale Unstable CCR3 44 46 COc1ccc(CCNC(=O)Nc2cccc(S(=O)(=O)O)c2)cc1 ZINC000217506028 FE For-Sale Unstable RAF1 43 51 COc1ccc(CCNC(=O)Nc2cccc(S(=O)(=O)O)c2)cc1 ZINC000217506028 FE For-Sale Unstable CA4 24 51 COc1ccc(CCNC(=O)Nc2cccc(S(=O)(=O)O)c2)cc1 ZINC000217506028 FE For-Sale Unstable MTNR1A 102 46 COc1ccc(CCNC(=O)Nc2cccc(S(=O)(=O)O)c2)cc1 ZINC000217506028 FE For-Sale Unstable MTNR1B 85 44 COc1ccc(CCNC(=O)Nc2cccc(S(=O)(=O)O)c2)cc1 ZINC000217506028 FE For-Sale Unstable MMP2 23 42 COc1ccc(CCNC(=O)Nc2cccc(S(=O)(=O)O)c2)cc1 ZINC000217506028 FE For-Sale Unstable MMP3 34 41 COc1ccc(CCNC(=O)Nc2cccc(S(=O)(=O)O)c2)cc1 ZINC000217506028 FE For-Sale Unstable MMP8 27 42 COc1ccc(CCNC(=O)Nc2cccc(S(=O)(=O)O)c2)cc1 ZINC000217506028 FE For-Sale Unstable PTPRB 40 37 COc1ccc(CCNC(=O)Nc2cccc(S(=O)(=O)O)c2)cc1 ZINC000217506028 FE For-Sale Unstable MMP9 44 42 COc1ccc(CCNC(=O)Nc2cccc(S(=O)(=O)O)c2)cc1 ZINC000217506028 FE For-Sale Unstable CA12 36 49 COc1ccc(CCNC(=O)Nc2cccc(S(=O)(=O)O)c2)cc1 ZINC000217506028 FE For-Sale Unstable PTGDR 26 51 COc1ccc(CCNC(=O)Nc2cccc(S(=O)(=O)O)c2)cc1 ZINC000217506028 FE For-Sale Unstable MMP7 26 41 COc1ccc(CCNC(=O)Nc2cccc(S(=O)(=O)O)c2)cc1 ZINC000217506028 FE For-Sale Unstable CA9 38 49 COc1ccc(CCNC(=O)Nc2cccc(S(=O)(=O)O)c2)cc1 ZINC000217506028 FE For-Sale Unstable MMP1 46 42 COc1ccc(CCNC(=O)Nc2cccc(S(=O)(=O)O)c2)cc1 ZINC000217506028 FE For-Sale Unstable Q8MMZ8_EIMTE 32 51 COc1ccc(CCNC(=O)Nc2cccc(S(=O)(=O)O)c2)cc1 ZINC000217506028 FE For-Sale Unstable AKR1C3 22 43 COc1ccc(CCNC(=O)Nc2cccc(S(=O)(=O)O)c2)cc1 ZINC000217506028 FE For-Sale Unstable NCE103 38 48 Cc1onc(-c2ccccc2Cl)c1C(=O)NC[C@](C)(O)c1cc2ccccc2s1 ZINC000217506062 IK In-Stock Unstable GPBAR1 40 48 Cc1onc(-c2ccccc2Cl)c1C(=O)NC[C@](C)(O)c1cc2ccccc2s1 ZINC000217506062 IK In-Stock Unstable BLAACC-4 0 42 Cc1onc(-c2ccccc2Cl)c1C(=O)NC[C@](C)(O)c1cc2ccccc2s1 ZINC000217506062 IK In-Stock Unstable SUGE 0 42 Cc1onc(-c2ccccc2Cl)c1C(=O)NC[C@](C)(O)c1cc2ccccc2s1 ZINC000217506062 IK In-Stock Unstable BLA_LAT-2 0 42 N[C@H](Cc1c[nH]c2ccccc12)C(=O)N[C@H](CCC(=O)O)C(=O)N[C@@H](Cc1cnc[nH]1)C(=O)N[C@@H](CC(=O)O)C(=O)Nc1ccc2c(C(F)(F)F)cc(=O)oc2c1 ZINC000217506081 KD In-Stock Unstable OPRM1 15 41 N[C@H](Cc1c[nH]c2ccccc12)C(=O)N[C@H](CCC(=O)O)C(=O)N[C@@H](Cc1cnc[nH]1)C(=O)N[C@@H](CC(=O)O)C(=O)Nc1ccc2c(C(F)(F)F)cc(=O)oc2c1 ZINC000217506081 KD In-Stock Unstable EDNRB 19 40 N[C@H](Cc1c[nH]c2ccccc12)C(=O)N[C@H](CCC(=O)O)C(=O)N[C@@H](Cc1cnc[nH]1)C(=O)N[C@@H](CC(=O)O)C(=O)Nc1ccc2c(C(F)(F)F)cc(=O)oc2c1 ZINC000217506081 KD In-Stock Unstable EDNRA 26 40 N[C@H](Cc1c[nH]c2ccccc12)C(=O)N[C@H](CCC(=O)O)C(=O)N[C@@H](Cc1cnc[nH]1)C(=O)N[C@@H](CC(=O)O)C(=O)Nc1ccc2c(C(F)(F)F)cc(=O)oc2c1 ZINC000217506081 KD In-Stock Unstable MC4R 48 49 N[C@H](Cc1c[nH]c2ccccc12)C(=O)N[C@H](CCC(=O)O)C(=O)N[C@@H](Cc1cnc[nH]1)C(=O)N[C@@H](CC(=O)O)C(=O)Nc1ccc2c(C(F)(F)F)cc(=O)oc2c1 ZINC000217506081 KD In-Stock Unstable CCKAR 87 43 N[C@H](Cc1c[nH]c2ccccc12)C(=O)N[C@H](CCC(=O)O)C(=O)N[C@@H](Cc1cnc[nH]1)C(=O)N[C@@H](CC(=O)O)C(=O)Nc1ccc2c(C(F)(F)F)cc(=O)oc2c1 ZINC000217506081 KD In-Stock Unstable MC3R 69 49 N[C@H](Cc1c[nH]c2ccccc12)C(=O)N[C@H](CCC(=O)O)C(=O)N[C@@H](Cc1cnc[nH]1)C(=O)N[C@@H](CC(=O)O)C(=O)Nc1ccc2c(C(F)(F)F)cc(=O)oc2c1 ZINC000217506081 KD In-Stock Unstable MC5R 72 49 N[C@H](Cc1c[nH]c2ccccc12)C(=O)N[C@H](CCC(=O)O)C(=O)N[C@@H](Cc1cnc[nH]1)C(=O)N[C@@H](CC(=O)O)C(=O)Nc1ccc2c(C(F)(F)F)cc(=O)oc2c1 ZINC000217506081 KD In-Stock Unstable GRPR 67 34 N[C@H](Cc1c[nH]c2ccccc12)C(=O)N[C@H](CCC(=O)O)C(=O)N[C@@H](Cc1cnc[nH]1)C(=O)N[C@@H](CC(=O)O)C(=O)Nc1ccc2c(C(F)(F)F)cc(=O)oc2c1 ZINC000217506081 KD In-Stock Unstable MMP11 80 35 N[C@H](Cc1c[nH]c2ccccc12)C(=O)N[C@H](CCC(=O)O)C(=O)N[C@@H](Cc1cnc[nH]1)C(=O)N[C@@H](CC(=O)O)C(=O)Nc1ccc2c(C(F)(F)F)cc(=O)oc2c1 ZINC000217506081 KD In-Stock Unstable CCKBR 57 46 N[C@H](Cc1c[nH]c2ccccc12)C(=O)N[C@H](CCC(=O)O)C(=O)N[C@@H](Cc1cnc[nH]1)C(=O)N[C@@H](CC(=O)O)C(=O)Nc1ccc2c(C(F)(F)F)cc(=O)oc2c1 ZINC000217506081 KD In-Stock Unstable GHSR 36 47 N[C@H](Cc1c[nH]c2ccccc12)C(=O)N[C@H](CCC(=O)O)C(=O)N[C@@H](Cc1cnc[nH]1)C(=O)N[C@@H](CC(=O)O)C(=O)Nc1ccc2c(C(F)(F)F)cc(=O)oc2c1 ZINC000217506081 KD In-Stock Unstable MC1R 104 49 N[C@H](Cc1c[nH]c2ccccc12)C(=O)N[C@H](CCC(=O)O)C(=O)N[C@@H](Cc1cnc[nH]1)C(=O)N[C@@H](CC(=O)O)C(=O)Nc1ccc2c(C(F)(F)F)cc(=O)oc2c1 ZINC000217506081 KD In-Stock Unstable KISS1R 75 36 N[C@H](Cc1c[nH]c2ccccc12)C(=O)N[C@H](CCC(=O)O)C(=O)N[C@@H](Cc1cnc[nH]1)C(=O)N[C@@H](CC(=O)O)C(=O)Nc1ccc2c(C(F)(F)F)cc(=O)oc2c1 ZINC000217506081 KD In-Stock Unstable TMPRSS6 16 44 CCOC(=O)c1ccc(N2CCC3(CCCC3)CC2)nc1 ZINC000217506099 CG On-Demand Unstable HDAC1 24 46 COc1ccc(CCNC(=O)Nc2ccc(C(C)C)cc2)cc1 ZINC000217506109 DI On-Demand Unstable CA2 21 50 COc1ccc(CCNC(=O)Nc2ccc(C(C)C)cc2)cc1 ZINC000217506109 DI On-Demand Unstable ADRB2 27 41 COc1ccc(CCNC(=O)Nc2ccc(C(C)C)cc2)cc1 ZINC000217506109 DI On-Demand Unstable ADRB1 44 44 COc1ccc(CCNC(=O)Nc2ccc(C(C)C)cc2)cc1 ZINC000217506109 DI On-Demand Unstable ADRB3 56 41 COc1ccc(CCNC(=O)Nc2ccc(C(C)C)cc2)cc1 ZINC000217506109 DI On-Demand Unstable BMP1 32 43 COc1ccc(CCNC(=O)Nc2ccc(C(C)C)cc2)cc1 ZINC000217506109 DI On-Demand Unstable NQO2 30 41 COc1ccc(CCNC(=O)Nc2ccc(C(C)C)cc2)cc1 ZINC000217506109 DI On-Demand Unstable CA1 46 50 COc1ccc(CCNC(=O)Nc2ccc(C(C)C)cc2)cc1 ZINC000217506109 DI On-Demand Unstable CTSL 18 47 COc1ccc(CCNC(=O)Nc2ccc(C(C)C)cc2)cc1 ZINC000217506109 DI On-Demand Unstable SCN2A 18 42 COc1ccc(CCNC(=O)Nc2ccc(C(C)C)cc2)cc1 ZINC000217506109 DI On-Demand Unstable RAF1 43 40 COc1ccc(CCNC(=O)Nc2ccc(C(C)C)cc2)cc1 ZINC000217506109 DI On-Demand Unstable MTNR1A 70 41 COc1ccc(CCNC(=O)Nc2ccc(C(C)C)cc2)cc1 ZINC000217506109 DI On-Demand Unstable MTNR1B 61 43 COc1ccc(CCNC(=O)Nc2ccc(C(C)C)cc2)cc1 ZINC000217506109 DI On-Demand Unstable NPY5R 24 43 COc1ccc(CCNC(=O)Nc2ccc(C(C)C)cc2)cc1 ZINC000217506109 DI On-Demand Unstable EPHX2 15 50 COc1ccc(CCNC(=O)Nc2ccc(C(C)C)cc2)cc1 ZINC000217506109 DI On-Demand Unstable F7 26 47 COc1ccc(CCNC(=O)Nc2ccc(C(C)C)cc2)cc1 ZINC000217506109 DI On-Demand Unstable ACR 24 43 COc1ccc(CCNC(=O)Nc2ccc(C(C)C)cc2)cc1 ZINC000217506109 DI On-Demand Unstable CA12 30 50 COc1ccc(CCNC(=O)Nc2ccc(C(C)C)cc2)cc1 ZINC000217506109 DI On-Demand Unstable PTGDR 15 43 COc1ccc(CCNC(=O)Nc2ccc(C(C)C)cc2)cc1 ZINC000217506109 DI On-Demand Unstable CA9 32 50 COc1ccc(CCNC(=O)Nc2ccc(C(C)C)cc2)cc1 ZINC000217506109 DI On-Demand Unstable MMP1 19 40 COc1ccc(CCNC(=O)Nc2ccc(C(C)C)cc2)cc1 ZINC000217506109 DI On-Demand Unstable Q8MMZ8_EIMTE 37 40 COc1ccc(CCNC(=O)Nc2ccc(C(C)C)cc2)cc1 ZINC000217506109 DI On-Demand Unstable NCE103 38 50 COc1ccc(CCNC(=O)Nc2ccc(C(C)C)cc2)cc1 ZINC000217506109 DI On-Demand Unstable P96878_MYCTU 23 43 COc1ccc(CCNC(=O)Nc2ccc(C(C)C)cc2)cc1 ZINC000217506109 DI On-Demand Unstable ACAT 0 46 CC(C)CCNc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217506118 FH In-Stock Unstable LIMK2 41 38 Cc1onc(-c2ccccc2Cl)c1C(=O)NC[C@@](C)(O)c1cc2ccccc2s1 ZINC000217506145 IK In-Stock Unstable GPBAR1 40 48 Cc1onc(-c2ccccc2Cl)c1C(=O)NC[C@@](C)(O)c1cc2ccccc2s1 ZINC000217506145 IK In-Stock Unstable BLAACC-4 0 42 Cc1onc(-c2ccccc2Cl)c1C(=O)NC[C@@](C)(O)c1cc2ccccc2s1 ZINC000217506145 IK In-Stock Unstable SUGE 0 42 Cc1onc(-c2ccccc2Cl)c1C(=O)NC[C@@](C)(O)c1cc2ccccc2s1 ZINC000217506145 IK In-Stock Unstable BLA_LAT-2 0 42 CCN(CC)[C@@H]1CCN(c2ccc(Cl)cc2CBr)C1 ZINC000217506158 EI For-Sale Unstable NOS2 20 40 CCN(CC)[C@@H]1CCN(c2ccc(Cl)cc2CBr)C1 ZINC000217506158 EI For-Sale Unstable NOS3 19 41 COc1ccc(CCNC(=O)Nc2ccc(C(=O)O)cc2)cc1 ZINC000217506226 DF For-Sale Unstable CA2 22 54 COc1ccc(CCNC(=O)Nc2ccc(C(=O)O)cc2)cc1 ZINC000217506226 DF For-Sale Unstable ADRB2 16 42 COc1ccc(CCNC(=O)Nc2ccc(C(=O)O)cc2)cc1 ZINC000217506226 DF For-Sale Unstable ADRB1 38 43 COc1ccc(CCNC(=O)Nc2ccc(C(=O)O)cc2)cc1 ZINC000217506226 DF For-Sale Unstable HRH2 19 45 COc1ccc(CCNC(=O)Nc2ccc(C(=O)O)cc2)cc1 ZINC000217506226 DF For-Sale Unstable PPIA 17 40 COc1ccc(CCNC(=O)Nc2ccc(C(=O)O)cc2)cc1 ZINC000217506226 DF For-Sale Unstable ADRB3 37 42 COc1ccc(CCNC(=O)Nc2ccc(C(=O)O)cc2)cc1 ZINC000217506226 DF For-Sale Unstable LTA4H 46 43 COc1ccc(CCNC(=O)Nc2ccc(C(=O)O)cc2)cc1 ZINC000217506226 DF For-Sale Unstable BMP1 24 43 COc1ccc(CCNC(=O)Nc2ccc(C(=O)O)cc2)cc1 ZINC000217506226 DF For-Sale Unstable CA1 44 54 COc1ccc(CCNC(=O)Nc2ccc(C(=O)O)cc2)cc1 ZINC000217506226 DF For-Sale Unstable CTSL 19 40 COc1ccc(CCNC(=O)Nc2ccc(C(=O)O)cc2)cc1 ZINC000217506226 DF For-Sale Unstable P2RX1 17 40 COc1ccc(CCNC(=O)Nc2ccc(C(=O)O)cc2)cc1 ZINC000217506226 DF For-Sale Unstable CCR3 21 40 COc1ccc(CCNC(=O)Nc2ccc(C(=O)O)cc2)cc1 ZINC000217506226 DF For-Sale Unstable SCN2A 26 42 COc1ccc(CCNC(=O)Nc2ccc(C(=O)O)cc2)cc1 ZINC000217506226 DF For-Sale Unstable HDAC8 15 43 COc1ccc(CCNC(=O)Nc2ccc(C(=O)O)cc2)cc1 ZINC000217506226 DF For-Sale Unstable RAF1 61 43 COc1ccc(CCNC(=O)Nc2ccc(C(=O)O)cc2)cc1 ZINC000217506226 DF For-Sale Unstable MTNR1A 74 40 COc1ccc(CCNC(=O)Nc2ccc(C(=O)O)cc2)cc1 ZINC000217506226 DF For-Sale Unstable MTNR1B 66 38 COc1ccc(CCNC(=O)Nc2ccc(C(=O)O)cc2)cc1 ZINC000217506226 DF For-Sale Unstable ROCK2 17 58 COc1ccc(CCNC(=O)Nc2ccc(C(=O)O)cc2)cc1 ZINC000217506226 DF For-Sale Unstable NPY5R 16 41 COc1ccc(CCNC(=O)Nc2ccc(C(=O)O)cc2)cc1 ZINC000217506226 DF For-Sale Unstable EPHX2 35 42 COc1ccc(CCNC(=O)Nc2ccc(C(=O)O)cc2)cc1 ZINC000217506226 DF For-Sale Unstable F7 23 43 COc1ccc(CCNC(=O)Nc2ccc(C(=O)O)cc2)cc1 ZINC000217506226 DF For-Sale Unstable ACR 52 44 COc1ccc(CCNC(=O)Nc2ccc(C(=O)O)cc2)cc1 ZINC000217506226 DF For-Sale Unstable CA12 30 54 COc1ccc(CCNC(=O)Nc2ccc(C(=O)O)cc2)cc1 ZINC000217506226 DF For-Sale Unstable PDGFRA 43 38 COc1ccc(CCNC(=O)Nc2ccc(C(=O)O)cc2)cc1 ZINC000217506226 DF For-Sale Unstable PTGDR 25 44 COc1ccc(CCNC(=O)Nc2ccc(C(=O)O)cc2)cc1 ZINC000217506226 DF For-Sale Unstable CA9 35 54 COc1ccc(CCNC(=O)Nc2ccc(C(=O)O)cc2)cc1 ZINC000217506226 DF For-Sale Unstable MCHR1 18 43 COc1ccc(CCNC(=O)Nc2ccc(C(=O)O)cc2)cc1 ZINC000217506226 DF For-Sale Unstable Q8MMZ8_EIMTE 57 43 COc1ccc(CCNC(=O)Nc2ccc(C(=O)O)cc2)cc1 ZINC000217506226 DF For-Sale Unstable AKR1C3 33 44 COc1ccc(CCNC(=O)Nc2ccc(C(=O)O)cc2)cc1 ZINC000217506226 DF For-Sale Unstable NCE103 37 54 COc1ccc(CCNC(=O)Nc2ccc(C(=O)O)cc2)cc1 ZINC000217506226 DF For-Sale Unstable AKR1C2 46 44 COc1ccc(CCNC(=O)Nc2ccc(C(=O)O)cc2)cc1 ZINC000217506226 DF For-Sale Unstable NOD1 16 42 COc1ccc(CCNC(=O)Nc2ccc(C(=O)O)cc2)cc1 ZINC000217506226 DF For-Sale Unstable NOD2 33 42 CCN(CC)[C@H]1CCN(c2ccc(Cl)cc2CBr)C1 ZINC000217506246 EI For-Sale Unstable NOS2 20 40 CCN(CC)[C@H]1CCN(c2ccc(Cl)cc2CBr)C1 ZINC000217506246 EI For-Sale Unstable NOS3 19 41 CSCC[C@H](NC(=O)[C@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217506263 KF In-Stock Unstable TACR1 0 40 CSCC[C@H](NC(=O)[C@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217506263 KF In-Stock Unstable SSTR4 44 31 CSCC[C@H](NC(=O)[C@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217506263 KF In-Stock Unstable FPR1 40 40 COc1ccc(CCNC(=O)Nc2cccc(Cl)c2Cl)cc1 ZINC000217506335 EI On-Demand Unstable ADRB3 15 40 COc1ccc(CCNC(=O)Nc2cccc(Cl)c2Cl)cc1 ZINC000217506335 EI On-Demand Unstable BMP1 30 46 COc1ccc(CCNC(=O)Nc2cccc(Cl)c2Cl)cc1 ZINC000217506335 EI On-Demand Unstable NQO2 39 42 COc1ccc(CCNC(=O)Nc2cccc(Cl)c2Cl)cc1 ZINC000217506335 EI On-Demand Unstable CA1 15 44 COc1ccc(CCNC(=O)Nc2cccc(Cl)c2Cl)cc1 ZINC000217506335 EI On-Demand Unstable TRPV1 32 61 COc1ccc(CCNC(=O)Nc2cccc(Cl)c2Cl)cc1 ZINC000217506335 EI On-Demand Unstable PTGER3 26 42 COc1ccc(CCNC(=O)Nc2cccc(Cl)c2Cl)cc1 ZINC000217506335 EI On-Demand Unstable RAF1 42 43 COc1ccc(CCNC(=O)Nc2cccc(Cl)c2Cl)cc1 ZINC000217506335 EI On-Demand Unstable MTNR1A 107 45 COc1ccc(CCNC(=O)Nc2cccc(Cl)c2Cl)cc1 ZINC000217506335 EI On-Demand Unstable MTNR1B 86 44 COc1ccc(CCNC(=O)Nc2cccc(Cl)c2Cl)cc1 ZINC000217506335 EI On-Demand Unstable PTGDR 23 42 COc1ccc(CCNC(=O)Nc2cccc(Cl)c2Cl)cc1 ZINC000217506335 EI On-Demand Unstable CA9 19 44 COc1ccc(CCNC(=O)Nc2cccc(Cl)c2Cl)cc1 ZINC000217506335 EI On-Demand Unstable Q8MMZ8_EIMTE 32 43 COc1ccc(CCNC(=O)Nc2cccc(Cl)c2Cl)cc1 ZINC000217506335 EI On-Demand Unstable NCE103 24 45 COc1ccc(CCNC(=O)Nc2cccc(Cl)c2Cl)cc1 ZINC000217506335 EI On-Demand Unstable PROKR1 43 31 COc1ccc(CCNC(=O)Nc2cccc(Cl)c2Cl)cc1 ZINC000217506335 EI On-Demand Unstable CAN2 0 45 Fc1ccc(N2CC[C@@H](N3CCCC3)C2)c(CBr)c1 ZINC000217506377 EG For-Sale Unstable L3MBTL3 67 40 CC1CCN(C(=O)c2nc(C(C)C)no2)CC1 ZINC000217506392 BE On-Demand Unstable LIPE 16 40 CC1CCN(C(=O)c2nc(C(C)C)no2)CC1 ZINC000217506392 BE On-Demand Unstable TRPC6 43 37 C[C@@](O)(CNC(=O)c1cc(C2CC2)on1)c1cc2ccccc2s1 ZINC000217506451 EG In-Stock Unstable S1PR3 0 41 COc1ccc(CCNC(=O)Nc2ccccc2C#N)cc1 ZINC000217506455 CF For-Sale Unstable ADRB1 46 48 COc1ccc(CCNC(=O)Nc2ccccc2C#N)cc1 ZINC000217506455 CF For-Sale Unstable BMP1 26 43 COc1ccc(CCNC(=O)Nc2ccccc2C#N)cc1 ZINC000217506455 CF For-Sale Unstable NQO2 26 41 COc1ccc(CCNC(=O)Nc2ccccc2C#N)cc1 ZINC000217506455 CF For-Sale Unstable CA1 15 46 COc1ccc(CCNC(=O)Nc2ccccc2C#N)cc1 ZINC000217506455 CF For-Sale Unstable TRPV1 0 57 COc1ccc(CCNC(=O)Nc2ccccc2C#N)cc1 ZINC000217506455 CF For-Sale Unstable CTSK 23 42 COc1ccc(CCNC(=O)Nc2ccccc2C#N)cc1 ZINC000217506455 CF For-Sale Unstable CTSL 23 44 COc1ccc(CCNC(=O)Nc2ccccc2C#N)cc1 ZINC000217506455 CF For-Sale Unstable MTNR1A 74 42 COc1ccc(CCNC(=O)Nc2ccccc2C#N)cc1 ZINC000217506455 CF For-Sale Unstable MTNR1B 61 39 COc1ccc(CCNC(=O)Nc2ccccc2C#N)cc1 ZINC000217506455 CF For-Sale Unstable CTSS 15 44 COc1ccc(CCNC(=O)Nc2ccccc2C#N)cc1 ZINC000217506455 CF For-Sale Unstable CA9 24 43 COc1ccc(CCNC(=O)Nc2ccccc2C#N)cc1 ZINC000217506455 CF For-Sale Unstable VIPR1 18 41 COc1ccc(CCNC(=O)Nc2ccccc2C#N)cc1 ZINC000217506455 CF For-Sale Unstable ABCG2 18 41 Fc1ccc(N2CC[C@H](N3CCCC3)C2)c(CBr)c1 ZINC000217506463 EG For-Sale Unstable L3MBTL3 67 40 CCNC(=O)NCCn1nc(-c2ccccn2)c2c1CCCC2 ZINC000217506477 DE For-Sale Unstable TGFBR1 36 40 C[C@](O)(CNC(=O)c1cc(C2CC2)on1)c1cc2ccccc2s1 ZINC000217506531 EG In-Stock Unstable S1PR3 0 41 CC[C@@H](C)c1ccccc1NC(=O)c1cccnc1F ZINC000217506537 CH For-Sale Unstable G2YM83_BOTF4 74 39 COc1ccccc1CN(C)C(=O)c1cc(Br)ccc1I ZINC000217506545 JI On-Demand Unstable HSP90AB1 20 41 CCOC(=O)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217506562 EG For-Sale Unstable BMP1 28 43 CCOC(=O)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217506562 EG For-Sale Unstable NQO2 25 41 CCOC(=O)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217506562 EG For-Sale Unstable CA1 27 46 CCOC(=O)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217506562 EG For-Sale Unstable TRPV1 0 55 CCOC(=O)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217506562 EG For-Sale Unstable RAF1 32 40 CCOC(=O)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217506562 EG For-Sale Unstable MTNR1A 74 42 CCOC(=O)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217506562 EG For-Sale Unstable MTNR1B 60 37 CCOC(=O)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217506562 EG For-Sale Unstable MMP3 16 42 CCOC(=O)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217506562 EG For-Sale Unstable SLC6A5 23 48 CCOC(=O)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217506562 EG For-Sale Unstable MMP9 16 42 CCOC(=O)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217506562 EG For-Sale Unstable CAPN2 16 45 CCOC(=O)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217506562 EG For-Sale Unstable CA12 18 54 CCOC(=O)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217506562 EG For-Sale Unstable PTGDR 0 45 CCOC(=O)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217506562 EG For-Sale Unstable CA9 21 54 CCOC(=O)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217506562 EG For-Sale Unstable MMP1 18 42 CCOC(=O)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217506562 EG For-Sale Unstable Q8MMZ8_EIMTE 24 40 CCOC(=O)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217506562 EG For-Sale Unstable NCE103 23 46 CCOC(=O)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217506562 EG For-Sale Unstable ABCG2 27 46 C[C@@H](CCc1ccc2c(c1)OCO2)N1CCC[C@@H](CN)C1 ZINC000217506565 CE For-Sale Unstable SSTR3 109 38 CC(C)C[C@H](NC(=O)CCC(=O)O[C@@H]1O[C@@H]2O[C@@]3(C)CC[C@H]4[C@H](C)CC[C@@H]([C@H]1C)[C@]42OO3)C(=O)N[C@@H](CO)C(=O)O ZINC000217506577 KD In-Stock Unstable Q9N6S8_PLAFA 46 38 Cn1ccnc1CN1CCN(C(=O)c2nc3ccccc3[nH]c2=O)CC1 ZINC000217506579 FC In-Stock Unstable EGLN1 0 40 CCCNc1ccc(C(=O)O)cc1S(=O)(=O)NCCCOCC ZINC000217506583 ED In-Stock Unstable PLA2G4B 41 33 CC[C@H](C)c1ccccc1NC(=O)c1cccnc1F ZINC000217506608 CH For-Sale Unstable G2YM83_BOTF4 74 39 C[C@@](O)(CNC(=O)c1ccc(OC(F)(F)F)cc1)c1cc2ccccc2s1 ZINC000217506638 GI In-Stock Unstable GCGR 40 36 C[C@@](O)(CNC(=O)c1ccc(OC(F)(F)F)cc1)c1cc2ccccc2s1 ZINC000217506638 GI In-Stock Unstable TRPV1 0 49 C[C@@](O)(CNC(=O)c1ccc(OC(F)(F)F)cc1)c1cc2ccccc2s1 ZINC000217506638 GI In-Stock Unstable SHH 46 36 COc1ccc(CCNC(=O)Nc2ccc(O)cc2)cc1 ZINC000217506644 CF For-Sale Unstable CA2 23 53 COc1ccc(CCNC(=O)Nc2ccc(O)cc2)cc1 ZINC000217506644 CF For-Sale Unstable ADRB2 27 49 COc1ccc(CCNC(=O)Nc2ccc(O)cc2)cc1 ZINC000217506644 CF For-Sale Unstable ADRB1 48 55 COc1ccc(CCNC(=O)Nc2ccc(O)cc2)cc1 ZINC000217506644 CF For-Sale Unstable ADRB3 45 49 COc1ccc(CCNC(=O)Nc2ccc(O)cc2)cc1 ZINC000217506644 CF For-Sale Unstable BMP1 24 52 COc1ccc(CCNC(=O)Nc2ccc(O)cc2)cc1 ZINC000217506644 CF For-Sale Unstable CA1 43 53 COc1ccc(CCNC(=O)Nc2ccc(O)cc2)cc1 ZINC000217506644 CF For-Sale Unstable TRPV1 0 52 COc1ccc(CCNC(=O)Nc2ccc(O)cc2)cc1 ZINC000217506644 CF For-Sale Unstable RAF1 28 42 COc1ccc(CCNC(=O)Nc2ccc(O)cc2)cc1 ZINC000217506644 CF For-Sale Unstable MTNR1A 84 42 COc1ccc(CCNC(=O)Nc2ccc(O)cc2)cc1 ZINC000217506644 CF For-Sale Unstable MTNR1B 75 39 COc1ccc(CCNC(=O)Nc2ccc(O)cc2)cc1 ZINC000217506644 CF For-Sale Unstable ROCK2 16 61 COc1ccc(CCNC(=O)Nc2ccc(O)cc2)cc1 ZINC000217506644 CF For-Sale Unstable SLC6A5 21 50 COc1ccc(CCNC(=O)Nc2ccc(O)cc2)cc1 ZINC000217506644 CF For-Sale Unstable EPHX2 19 44 COc1ccc(CCNC(=O)Nc2ccc(O)cc2)cc1 ZINC000217506644 CF For-Sale Unstable ACR 23 40 COc1ccc(CCNC(=O)Nc2ccc(O)cc2)cc1 ZINC000217506644 CF For-Sale Unstable CA12 31 53 COc1ccc(CCNC(=O)Nc2ccc(O)cc2)cc1 ZINC000217506644 CF For-Sale Unstable PTGDR 23 45 COc1ccc(CCNC(=O)Nc2ccc(O)cc2)cc1 ZINC000217506644 CF For-Sale Unstable CA9 35 53 COc1ccc(CCNC(=O)Nc2ccc(O)cc2)cc1 ZINC000217506644 CF For-Sale Unstable Q8MMZ8_EIMTE 37 42 COc1ccc(CCNC(=O)Nc2ccc(O)cc2)cc1 ZINC000217506644 CF For-Sale Unstable NCE103 25 53 C[C@H](CCc1ccc2c(c1)OCO2)N1CCC[C@@H](CN)C1 ZINC000217506653 CE For-Sale Unstable SSTR3 109 38 CC1(C)CC[C@@H](N2CCC[C@@H](N)C2)c2ccccc21 ZINC000217506689 CG For-Sale Unstable SLC6A1 0 43 CC1(C)CC[C@@H](N2CCC[C@@H](N)C2)c2ccccc21 ZINC000217506689 CG For-Sale Unstable OPRL1 18 53 Clc1ccc(-c2ccsc2)cc1Cl ZINC000217506711 BJ For-Sale Anodyne KMO 0 43 C[C@](O)(CNC(=O)c1ccc(OC(F)(F)F)cc1)c1cc2ccccc2s1 ZINC000217506722 GI In-Stock Unstable GCGR 40 36 C[C@](O)(CNC(=O)c1ccc(OC(F)(F)F)cc1)c1cc2ccccc2s1 ZINC000217506722 GI In-Stock Unstable TRPV1 0 49 C[C@](O)(CNC(=O)c1ccc(OC(F)(F)F)cc1)c1cc2ccccc2s1 ZINC000217506722 GI In-Stock Unstable SHH 46 36 CCCCc1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217506749 EI For-Sale Unstable CA2 20 51 CCCCc1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217506749 EI For-Sale Unstable ADRB1 30 43 CCCCc1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217506749 EI For-Sale Unstable AGTR1 15 42 CCCCc1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217506749 EI For-Sale Unstable INHA 44 44 CCCCc1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217506749 EI For-Sale Unstable ADRB3 25 40 CCCCc1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217506749 EI For-Sale Unstable BMP1 24 51 CCCCc1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217506749 EI For-Sale Unstable CA1 36 51 CCCCc1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217506749 EI For-Sale Unstable SCN2A 29 50 CCCCc1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217506749 EI For-Sale Unstable S1PR4 31 40 CCCCc1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217506749 EI For-Sale Unstable RAF1 42 41 CCCCc1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217506749 EI For-Sale Unstable S1PR3 29 42 CCCCc1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217506749 EI For-Sale Unstable MTNR1A 90 44 CCCCc1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217506749 EI For-Sale Unstable MTNR1B 76 43 CCCCc1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217506749 EI For-Sale Unstable MMP3 15 41 CCCCc1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217506749 EI For-Sale Unstable CFTR 43 34 CCCCc1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217506749 EI For-Sale Unstable S1PR2 43 39 CCCCc1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217506749 EI For-Sale Unstable S1PR1 19 42 CCCCc1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217506749 EI For-Sale Unstable EPHX2 19 45 CCCCc1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217506749 EI For-Sale Unstable SPHK1 23 42 CCCCc1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217506749 EI For-Sale Unstable S1PR5 28 40 CCCCc1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217506749 EI For-Sale Unstable CA12 28 51 CCCCc1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217506749 EI For-Sale Unstable PTGDR 22 46 CCCCc1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217506749 EI For-Sale Unstable CA9 30 46 CCCCc1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217506749 EI For-Sale Unstable Q8MMZ8_EIMTE 36 41 CCCCc1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217506749 EI For-Sale Unstable NCE103 39 51 CCCCc1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217506749 EI For-Sale Unstable P96878_MYCTU 23 52 CCCCc1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217506749 EI For-Sale Unstable ACAT 0 49 CCCCc1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217506749 EI For-Sale Unstable PSBA 0 42 CCCCNc1ccc(C(=O)O)cc1S(=O)(=O)NCCCOCC ZINC000217506755 FE In-Stock Unstable PLA2G4B 47 34 Nc1[nH]nc(C(=O)NCCc2ccncc2)c1Cl ZINC000217506769 CD In-Stock Unstable CA5B 17 45 Nc1[nH]nc(C(=O)NCCc2ccncc2)c1Cl ZINC000217506769 CD In-Stock Unstable CA5A 15 45 Clc1cccc(N2CC[C@@H](N3CCCC3)C2)c1CBr ZINC000217506770 EH For-Sale Unstable L3MBTL3 67 40 CC1(C)CC[C@H](N2CCC[C@@H](N)C2)c2ccccc21 ZINC000217506778 CG For-Sale Unstable SLC6A1 0 43 CC1(C)CC[C@H](N2CCC[C@@H](N)C2)c2ccccc21 ZINC000217506778 CG For-Sale Unstable OPRL1 18 53 Cc1ccsc1/C=C\C(=O)Nc1ccccc1[C@@H](C)O ZINC000217506806 CH For-Sale Unstable UL26 36 44 Cc1ccsc1/C=C\C(=O)Nc1ccccc1[C@@H](C)O ZINC000217506806 CH For-Sale Unstable SCAF_EBVB9 29 44 Clc1cccc(N2CC[C@H](N3CCCC3)C2)c1CBr ZINC000217506859 EH For-Sale Unstable L3MBTL3 67 40 COc1ccc(CCNC(=O)NCCc2ccc(O)cc2)cc1 ZINC000217506863 DE On-Demand Unstable ADRB2 28 48 COc1ccc(CCNC(=O)NCCc2ccc(O)cc2)cc1 ZINC000217506863 DE On-Demand Unstable ADRB1 36 48 COc1ccc(CCNC(=O)NCCc2ccc(O)cc2)cc1 ZINC000217506863 DE On-Demand Unstable ADRB3 31 53 COc1ccc(CCNC(=O)NCCc2ccc(O)cc2)cc1 ZINC000217506863 DE On-Demand Unstable CA1 15 50 COc1ccc(CCNC(=O)NCCc2ccc(O)cc2)cc1 ZINC000217506863 DE On-Demand Unstable TRPV1 0 51 COc1ccc(CCNC(=O)NCCc2ccc(O)cc2)cc1 ZINC000217506863 DE On-Demand Unstable MMP13 18 43 COc1ccc(CCNC(=O)NCCc2ccc(O)cc2)cc1 ZINC000217506863 DE On-Demand Unstable MTNR1A 80 48 COc1ccc(CCNC(=O)NCCc2ccc(O)cc2)cc1 ZINC000217506863 DE On-Demand Unstable MTNR1B 63 41 COc1ccc(CCNC(=O)NCCc2ccc(O)cc2)cc1 ZINC000217506863 DE On-Demand Unstable MMP8 15 44 COc1ccc(CCNC(=O)NCCc2ccc(O)cc2)cc1 ZINC000217506863 DE On-Demand Unstable SLC6A5 18 52 COc1ccc(CCNC(=O)NCCc2ccc(O)cc2)cc1 ZINC000217506863 DE On-Demand Unstable MMP12 15 43 COc1ccc(CCNC(=O)NCCc2ccc(O)cc2)cc1 ZINC000217506863 DE On-Demand Unstable CA12 15 53 COc1ccc(CCNC(=O)NCCc2ccc(O)cc2)cc1 ZINC000217506863 DE On-Demand Unstable PTGDR 24 41 COc1ccc(CCNC(=O)NCCc2ccc(O)cc2)cc1 ZINC000217506863 DE On-Demand Unstable CA9 25 53 COc1ccc(CCNC(=O)NCCc2ccc(O)cc2)cc1 ZINC000217506863 DE On-Demand Unstable MMP1 24 44 COc1ccc(CCNC(=O)NCCc2ccc(O)cc2)cc1 ZINC000217506863 DE On-Demand Unstable TAAR1 16 40 COc1ccc(CCNC(=O)NCCc2ccc(O)cc2)cc1 ZINC000217506863 DE On-Demand Unstable NCE103 27 42 COc1ccc(CCNC(=O)NCCc2ccc(O)cc2)cc1 ZINC000217506863 DE On-Demand Unstable PROKR1 55 40 COc1ccc(CCNC(=O)NCCc2ccc(O)cc2)cc1 ZINC000217506863 DE On-Demand Unstable AKR1B10 50 37 O=C1CC2(CCN(C(=O)/C=C\c3ccccc3)CC2)CN1 ZINC000217506869 CD On-Demand Unstable CCR2 43 39 O=C1CC2(CCN(C(=O)/C=C\c3ccccc3)CC2)CN1 ZINC000217506869 CD On-Demand Unstable GPR183 0 45 Cc1ccsc1/C=C\C(=O)Nc1ccccc1[C@H](C)O ZINC000217506882 CH For-Sale Unstable UL26 36 44 Cc1ccsc1/C=C\C(=O)Nc1ccccc1[C@H](C)O ZINC000217506882 CH For-Sale Unstable SCAF_EBVB9 29 44 CC[C@H](C)[C@H](NN)[C@@H](c1ccccc1)[C@@H](C)CC ZINC000217506912 BH For-Sale Unstable AOC3 17 47 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable CA2 18 48 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable ALOX5 19 47 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable ACHE 0 49 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable ADRB3 31 40 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable LTA4H 47 37 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable ANPEP 29 42 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable BMP1 109 45 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable NQO2 26 43 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable CA1 20 48 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable TSPO 17 41 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable SIGMAR1 22 47 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable MMP13 69 44 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable CTSK 23 40 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable SCN2A 18 43 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable ADAM17 38 41 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable HDAC8 15 44 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable CA5B 15 40 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable MMP16 0 42 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable MTNR1A 98 43 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable MTNR1B 86 39 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable MMP2 55 48 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable MMP3 67 49 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable MMP8 47 48 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable MMP14 20 40 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable SLC2A1 0 41 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable FAAH 26 40 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable NPY5R 25 45 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable CAPN1 17 45 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable MMP9 73 49 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable CASP1 17 41 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable CAPN2 22 41 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable MMP12 39 48 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable PTGDR 23 44 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable MMP7 31 45 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable CA9 21 47 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable MMP1 75 49 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable POL 0 45 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable AMP1_PLAFQ 38 42 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable SLC10A1 24 40 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable HT1 0 44 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable PROKR1 43 31 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable PTGES 24 47 COc1ccc(CCNC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217506939 EH On-Demand Unstable LMGT2 0 44 Cc1cc(CBr)cnc1N1CC[C@@H](N2CCCC2)C1 ZINC000217506953 DF For-Sale Unstable L3MBTL3 41 36 COc1cccc([C@@H]2CCN(C(=O)Cn3nc(C)cc3N)C2)c1OC ZINC000217506997 ED In-Stock Unstable FDFT1 41 36 Cc1cc(CBr)cnc1N1CC[C@H](N2CCCC2)C1 ZINC000217507027 DF For-Sale Unstable L3MBTL3 41 36 N[C@@H]1CCCN([C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217507031 CD For-Sale Unstable DRD2 23 49 N[C@@H]1CCCN([C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217507031 CD For-Sale Unstable DRD4 40 40 N[C@@H]1CCCN([C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217507031 CD For-Sale Unstable ACHE 39 45 N[C@@H]1CCCN([C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217507031 CD For-Sale Unstable DRD3 29 46 N[C@@H]1CCCN([C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217507031 CD For-Sale Unstable VACHT_TETCF 0 46 N[C@@H]1CCCN([C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217507031 CD For-Sale Unstable SIGMAR1 64 45 N[C@@H]1CCCN([C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217507031 CD For-Sale Unstable DPP4 20 40 N[C@@H]1CCCN([C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217507031 CD For-Sale Unstable SLC18A3 28 43 COc1ccc(CCNC(=O)N2CCC(C(=O)O)CC2)cc1 ZINC000217507069 DD On-Demand Unstable DRD4 40 31 Cc1noc(C)c1CC(=O)NC[C@](C)(O)c1cc2ccccc2s1 ZINC000217507073 EG In-Stock Unstable P2RX7 26 52 COc1cccc([C@H]2CCN(C(=O)Cn3nc(C)cc3N)C2)c1OC ZINC000217507087 ED In-Stock Unstable FDFT1 41 36 Cc1noc(C)c1CC(=O)NC[C@@](C)(O)c1cc2ccccc2s1 ZINC000217507149 EG In-Stock Unstable P2RX7 26 52 O=C(NCCn1nc(-c2ccccn2)c2c1CCCC2)Nc1ccccc1 ZINC000217507160 FH For-Sale Unstable TGFBR1 24 42 C[C@H](c1ccc(F)cc1)N1CCC[C@@H](CN)C1 ZINC000217507166 BF On-Demand Unstable CCR3 41 38 COc1ccc(CCNC(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000217507181 II For-Sale Unstable OPRM1 24 47 COc1ccc(CCNC(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000217507181 II For-Sale Unstable DRD3 16 47 COc1ccc(CCNC(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000217507181 II For-Sale Unstable OPRD1 36 47 COc1ccc(CCNC(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000217507181 II For-Sale Unstable OPRK1 32 48 COc1ccc(CCNC(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000217507181 II For-Sale Unstable OPRL1 26 41 COc1ccc(CCNC(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000217507181 II For-Sale Unstable BMP1 51 36 COc1ccc(CCNC(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000217507181 II For-Sale Unstable SIGMAR1 15 47 COc1ccc(CCNC(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000217507181 II For-Sale Unstable MMP13 34 41 COc1ccc(CCNC(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000217507181 II For-Sale Unstable NPY2R 15 47 COc1ccc(CCNC(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000217507181 II For-Sale Unstable CCR3 29 49 COc1ccc(CCNC(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000217507181 II For-Sale Unstable SCN2A 15 40 COc1ccc(CCNC(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000217507181 II For-Sale Unstable CCR5 16 43 COc1ccc(CCNC(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000217507181 II For-Sale Unstable PLA2G4A 51 33 COc1ccc(CCNC(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000217507181 II For-Sale Unstable MTNR1A 82 39 COc1ccc(CCNC(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000217507181 II For-Sale Unstable MTNR1B 75 38 COc1ccc(CCNC(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000217507181 II For-Sale Unstable MMP3 37 53 COc1ccc(CCNC(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000217507181 II For-Sale Unstable FAAH 17 49 COc1ccc(CCNC(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000217507181 II For-Sale Unstable CYP2D6 25 43 COc1ccc(CCNC(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000217507181 II For-Sale Unstable MMP9 32 53 COc1ccc(CCNC(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000217507181 II For-Sale Unstable MMP7 25 53 COc1ccc(CCNC(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000217507181 II For-Sale Unstable HCRTR2 18 40 COc1ccc(CCNC(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000217507181 II For-Sale Unstable MMP1 38 53 COc1ccc(CCNC(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000217507181 II For-Sale Unstable CACNA1G 18 43 COc1ccc(CCNC(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000217507181 II For-Sale Unstable NMUR2 0 58 COc1ccc(CCNC(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000217507181 II For-Sale Unstable NMUR1 0 58 Cc1nc(NCCN)cc(N2CCCC2)n1 ZINC000217507249 BC In-Stock Unstable GALR2 42 35 C[C@@H](c1ccc(F)cc1)N1CCC[C@@H](CN)C1 ZINC000217507251 BF On-Demand Unstable CCR3 41 38 C[C@@](O)(CNC(=O)Cc1c(F)cccc1Cl)c1cc2ccccc2s1 ZINC000217507253 GI In-Stock Unstable P2RX7 33 44 O=C(NCCn1nc(-c2ccccn2)c2c1CCCC2)Nc1cccs1 ZINC000217507255 FH For-Sale Unstable TGFBR1 24 41 CCOCCCNC(=O)NCCc1ccc(OC)cc1 ZINC000217507291 CD On-Demand Unstable SCNN1A 35 40 CCOCCCNC(=O)NCCc1ccc(OC)cc1 ZINC000217507291 CD On-Demand Unstable MTNR1A 70 45 CCOCCCNC(=O)NCCc1ccc(OC)cc1 ZINC000217507291 CD On-Demand Unstable MTNR1B 53 39 CCOCCCNC(=O)NCCc1ccc(OC)cc1 ZINC000217507291 CD On-Demand Unstable CA9 23 47 N[C@@H]1CCCN([C@@H]2CCCN(Cc3ccccc3)C2)C1 ZINC000217507303 CE For-Sale Unstable DRD4 28 40 N[C@@H]1CCCN([C@@H]2CCCN(Cc3ccccc3)C2)C1 ZINC000217507303 CE For-Sale Unstable ACHE 28 42 N[C@@H]1CCCN([C@@H]2CCCN(Cc3ccccc3)C2)C1 ZINC000217507303 CE For-Sale Unstable DRD3 15 40 N[C@@H]1CCCN([C@@H]2CCCN(Cc3ccccc3)C2)C1 ZINC000217507303 CE For-Sale Unstable SIGMAR1 57 48 N[C@@H]1CCCN([C@@H]2CCCN(Cc3ccccc3)C2)C1 ZINC000217507303 CE For-Sale Unstable DPP4 19 40 N[C@@H]1CCCN([C@@H]2CCCN(Cc3ccccc3)C2)C1 ZINC000217507303 CE For-Sale Unstable SLC18A3 23 40 N[C@@H]1CCCN([C@@H]2CCCN(Cc3ccccc3)C2)C1 ZINC000217507303 CE For-Sale Unstable MC3R 15 43 C[C@](O)(CNC(=O)Cc1c(F)cccc1Cl)c1cc2ccccc2s1 ZINC000217507323 GI In-Stock Unstable P2RX7 33 44 Cc1cc(N2CCCCC2)nc(NCCN)n1 ZINC000217507344 BD In-Stock Unstable GALR2 44 37 O=C(NCCn1nc(-c2ccccn2)c2c1CCCC2)NC1CCCCC1 ZINC000217507369 FG For-Sale Unstable EPHX2 18 44 CC(C)c1ccc(NC(=O)c2cc(Br)ccc2I)cc1 ZINC000217507372 IK For-Sale Unstable Q25615_ONCVO 86 50 COc1ccc(CCNC(=O)N2CCCc3ccccc32)cc1 ZINC000217507393 DG For-Sale Unstable DRD4 42 35 COc1ccc(CCNC(=O)N2CCCc3ccccc32)cc1 ZINC000217507393 DG For-Sale Unstable AVPR2 46 47 COc1ccc(CCNC(=O)N2CCCc3ccccc32)cc1 ZINC000217507393 DG For-Sale Unstable AVPR1A 26 40 COc1ccc(CCNC(=O)N2CCCc3ccccc32)cc1 ZINC000217507393 DG For-Sale Unstable NQO2 31 41 COc1ccc(CCNC(=O)N2CCCc3ccccc32)cc1 ZINC000217507393 DG For-Sale Unstable SIGMAR1 15 44 COc1ccc(CCNC(=O)N2CCCc3ccccc32)cc1 ZINC000217507393 DG For-Sale Unstable MTNR1A 73 44 COc1ccc(CCNC(=O)N2CCCc3ccccc32)cc1 ZINC000217507393 DG For-Sale Unstable MTNR1B 68 44 COc1ccc(CCNC(=O)N2CCCc3ccccc32)cc1 ZINC000217507393 DG For-Sale Unstable MMP3 22 44 COc1ccc(CCNC(=O)N2CCCc3ccccc32)cc1 ZINC000217507393 DG For-Sale Unstable MMP9 26 44 COc1ccc(CCNC(=O)N2CCCc3ccccc32)cc1 ZINC000217507393 DG For-Sale Unstable MMP1 33 44 COc1ccc(CCNC(=O)N2CCCc3ccccc32)cc1 ZINC000217507393 DG For-Sale Unstable NOD2 40 42 CCOCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NC1CCCC1 ZINC000217507447 FE In-Stock Unstable AMY2 42 29 CCOCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NC1CCCC1 ZINC000217507447 FE In-Stock Unstable PLA2G4B 40 32 COc1ccc(CCNC(=O)N(C)C2CCN(C)CC2)cc1 ZINC000217507508 DD For-Sale Unstable SIGMAR1 17 46 COc1ccc(CCNC(=O)N(C)C2CCN(C)CC2)cc1 ZINC000217507508 DD For-Sale Unstable MMP13 33 42 COc1ccc(CCNC(=O)N(C)C2CCN(C)CC2)cc1 ZINC000217507508 DD For-Sale Unstable CTSK 18 41 COc1ccc(CCNC(=O)N(C)C2CCN(C)CC2)cc1 ZINC000217507508 DD For-Sale Unstable MTNR1A 68 38 COc1ccc(CCNC(=O)N(C)C2CCN(C)CC2)cc1 ZINC000217507508 DD For-Sale Unstable MTNR1B 59 35 COc1ccc(CCNC(=O)N(C)C2CCN(C)CC2)cc1 ZINC000217507508 DD For-Sale Unstable MMP3 36 42 COc1ccc(CCNC(=O)N(C)C2CCN(C)CC2)cc1 ZINC000217507508 DD For-Sale Unstable MMP8 15 42 COc1ccc(CCNC(=O)N(C)C2CCN(C)CC2)cc1 ZINC000217507508 DD For-Sale Unstable SLC6A5 29 40 COc1ccc(CCNC(=O)N(C)C2CCN(C)CC2)cc1 ZINC000217507508 DD For-Sale Unstable MMP9 30 42 COc1ccc(CCNC(=O)N(C)C2CCN(C)CC2)cc1 ZINC000217507508 DD For-Sale Unstable MMP7 30 42 COc1ccc(CCNC(=O)N(C)C2CCN(C)CC2)cc1 ZINC000217507508 DD For-Sale Unstable MMP1 35 42 COc1ccc(CCNC(=O)N(C)C2CCN(C)CC2)cc1 ZINC000217507508 DD For-Sale Unstable MCHR1 25 46 Clc1cc(CBr)ccc1N1CC[C@@H](N2CCCC2)C1 ZINC000217507558 EH For-Sale Unstable L3MBTL3 86 42 CCOCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NC1CCCCC1 ZINC000217507559 GF In-Stock Unstable AMY2 44 31 Cc1cc(N2CCOCC2)nc(NCCN)n1 ZINC000217507560 BB In-Stock Unstable PIK3CA 16 44 Cc1cc(N2CCOCC2)nc(NCCN)n1 ZINC000217507560 BB In-Stock Unstable SMG1 41 35 Cc1ccccc1NC(=O)NCCn1nc(-c2ccccn2)c2c1CCCC2 ZINC000217507561 GH For-Sale Unstable TGFBR1 26 40 C[C@H]1CN([C@H](C)C(=O)Nc2cccc(CN)c2)CCCO1 ZINC000217507598 CD For-Sale Unstable NOS1 17 41 C[C@H]1CN([C@H](C)C(=O)Nc2cccc(CN)c2)CCCO1 ZINC000217507598 CD For-Sale Unstable TPSAB1 58 40 COc1ccc(CCNC(=O)N2CCN(C(C)=O)CC2)cc1 ZINC000217507609 DD For-Sale Unstable BMP1 59 38 COc1ccc(CCNC(=O)N2CCN(C(C)=O)CC2)cc1 ZINC000217507609 DD For-Sale Unstable NQO2 42 40 COc1ccc(CCNC(=O)N2CCN(C(C)=O)CC2)cc1 ZINC000217507609 DD For-Sale Unstable MMP13 43 44 COc1ccc(CCNC(=O)N2CCN(C(C)=O)CC2)cc1 ZINC000217507609 DD For-Sale Unstable CTSK 20 42 COc1ccc(CCNC(=O)N2CCN(C(C)=O)CC2)cc1 ZINC000217507609 DD For-Sale Unstable CTSL 20 42 COc1ccc(CCNC(=O)N2CCN(C(C)=O)CC2)cc1 ZINC000217507609 DD For-Sale Unstable ADAM17 17 43 COc1ccc(CCNC(=O)N2CCN(C(C)=O)CC2)cc1 ZINC000217507609 DD For-Sale Unstable MMP16 0 40 COc1ccc(CCNC(=O)N2CCN(C(C)=O)CC2)cc1 ZINC000217507609 DD For-Sale Unstable MTNR1A 124 43 COc1ccc(CCNC(=O)N2CCN(C(C)=O)CC2)cc1 ZINC000217507609 DD For-Sale Unstable MTNR1B 105 43 COc1ccc(CCNC(=O)N2CCN(C(C)=O)CC2)cc1 ZINC000217507609 DD For-Sale Unstable MMP2 23 40 COc1ccc(CCNC(=O)N2CCN(C(C)=O)CC2)cc1 ZINC000217507609 DD For-Sale Unstable MMP3 46 53 COc1ccc(CCNC(=O)N2CCN(C(C)=O)CC2)cc1 ZINC000217507609 DD For-Sale Unstable MMP8 26 41 COc1ccc(CCNC(=O)N2CCN(C(C)=O)CC2)cc1 ZINC000217507609 DD For-Sale Unstable MMP9 43 53 COc1ccc(CCNC(=O)N2CCN(C(C)=O)CC2)cc1 ZINC000217507609 DD For-Sale Unstable MMP12 21 41 COc1ccc(CCNC(=O)N2CCN(C(C)=O)CC2)cc1 ZINC000217507609 DD For-Sale Unstable PTGDR 24 40 COc1ccc(CCNC(=O)N2CCN(C(C)=O)CC2)cc1 ZINC000217507609 DD For-Sale Unstable MMP7 39 53 COc1ccc(CCNC(=O)N2CCN(C(C)=O)CC2)cc1 ZINC000217507609 DD For-Sale Unstable CA9 21 48 COc1ccc(CCNC(=O)N2CCN(C(C)=O)CC2)cc1 ZINC000217507609 DD For-Sale Unstable MMP1 53 53 COc1ccc(CCNC(=O)N2CCN(C(C)=O)CC2)cc1 ZINC000217507609 DD For-Sale Unstable PROKR1 60 34 Clc1cc(CBr)ccc1N1CC[C@H](N2CCCC2)C1 ZINC000217507640 EH For-Sale Unstable L3MBTL3 86 42 C[C@@H](CCN)c1ccc(S(C)(=O)=O)cc1F ZINC000217507658 BD For-Sale Unstable PTGS2 27 44 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Cl)cc1 ZINC000217507664 DI For-Sale Unstable LTB4R 0 47 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Cl)cc1 ZINC000217507664 DI For-Sale Unstable HDAC8 16 47 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Cl)cc1 ZINC000217507664 DI For-Sale Unstable MMP2 23 55 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Cl)cc1 ZINC000217507664 DI For-Sale Unstable HDAC1 25 47 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Cl)cc1 ZINC000217507664 DI For-Sale Unstable HDAC2 19 47 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Cl)cc1 ZINC000217507664 DI For-Sale Unstable MMP9 22 55 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Cl)cc1 ZINC000217507664 DI For-Sale Unstable MMP1 26 55 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Cl)cc1 ZINC000217507664 DI For-Sale Unstable TRPM2 0 42 Cc1cccc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)c1 ZINC000217507679 GH For-Sale Unstable CCKAR 26 42 Cc1cccc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)c1 ZINC000217507679 GH For-Sale Unstable CCKBR 39 42 Cc1cccc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)c1 ZINC000217507679 GH For-Sale Unstable TGFBR1 25 44 Cc1cccc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)c1 ZINC000217507679 GH For-Sale Unstable KCNK3 54 34 Cc1cccc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)c1 ZINC000217507679 GH For-Sale Unstable KCNK9 40 34 C[C@H]1CN([C@H](C)C(=O)Nc2ccccc2CN)CCCO1 ZINC000217507707 CD For-Sale Unstable KCNQ2 47 34 COc1ccc(CCNC(=O)N[C@@H](C)C23CC4CC(CC(C4)C2)C3)cc1 ZINC000217507715 FI For-Sale Unstable MTNR1A 51 38 COc1ccc(CCNC(=O)N[C@@H](C)C23CC4CC(CC(C4)C2)C3)cc1 ZINC000217507715 FI For-Sale Unstable MTNR1B 42 35 COc1ccc(CCNC(=O)N[C@@H](C)C23CC4CC(CC(C4)C2)C3)cc1 ZINC000217507715 FI For-Sale Unstable EPHX2 49 59 C[C@H](CCN)c1ccc(S(C)(=O)=O)cc1F ZINC000217507727 BD For-Sale Unstable PTGS2 27 44 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Cl)cc1 ZINC000217507741 DI For-Sale Unstable LTB4R 0 47 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Cl)cc1 ZINC000217507741 DI For-Sale Unstable HDAC8 16 47 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Cl)cc1 ZINC000217507741 DI For-Sale Unstable MMP2 23 55 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Cl)cc1 ZINC000217507741 DI For-Sale Unstable HDAC1 25 47 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Cl)cc1 ZINC000217507741 DI For-Sale Unstable HDAC2 19 47 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Cl)cc1 ZINC000217507741 DI For-Sale Unstable MMP9 22 55 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Cl)cc1 ZINC000217507741 DI For-Sale Unstable MMP1 26 55 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Cl)cc1 ZINC000217507741 DI For-Sale Unstable TRPM2 0 42 Cc1cc(CBr)ccc1N1CC[C@@H](N2CCCC2)C1 ZINC000217507749 DH For-Sale Unstable HRH3 0 44 Cc1cc(CBr)ccc1N1CC[C@@H](N2CCCC2)C1 ZINC000217507749 DH For-Sale Unstable L3MBTL3 80 40 CC[C@H](c1cccc(Cl)c1)N1CCC[C@@H](CN)C1 ZINC000217507759 CG For-Sale Unstable OPRL1 0 48 Cc1cc(N2CCNCC2)nc(NC2CCCCC2)n1 ZINC000217507782 CD In-Stock Unstable HRH4 35 44 Cc1cc(N2CCNCC2)nc(NC2CCCCC2)n1 ZINC000217507782 CD In-Stock Unstable PRKD1 65 47 Cc1cc(N2CCNCC2)nc(NC2CCCCC2)n1 ZINC000217507782 CD In-Stock Unstable TTK 23 42 Cc1cc(N2CCNCC2)nc(NC2CCCCC2)n1 ZINC000217507782 CD In-Stock Unstable PKD2 0 50 Cc1ccc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)cc1 ZINC000217507784 GH For-Sale Unstable TGFBR1 22 44 COc1ccc(CCNC(=O)N[C@H](C)C23CC4CC(CC(C4)C2)C3)cc1 ZINC000217507789 FI For-Sale Unstable MTNR1A 51 38 COc1ccc(CCNC(=O)N[C@H](C)C23CC4CC(CC(C4)C2)C3)cc1 ZINC000217507789 FI For-Sale Unstable MTNR1B 42 35 COc1ccc(CCNC(=O)N[C@H](C)C23CC4CC(CC(C4)C2)C3)cc1 ZINC000217507789 FI For-Sale Unstable EPHX2 49 59 COc1ccc(Cn2nc(C)nc2CC(F)(F)F)cc1 ZINC000217507800 CF In-Stock Unstable NPBWR1 34 41 Cc1cc(CBr)ccc1N1CC[C@H](N2CCCC2)C1 ZINC000217507824 DH For-Sale Unstable HRH3 0 44 Cc1cc(CBr)ccc1N1CC[C@H](N2CCCC2)C1 ZINC000217507824 DH For-Sale Unstable L3MBTL3 80 40 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Br)o1 ZINC000217507831 EH For-Sale Unstable SCAF_EBVB9 15 42 CC[C@@H](c1cccc(Cl)c1)N1CCC[C@@H](CN)C1 ZINC000217507835 CG For-Sale Unstable OPRL1 0 48 O=C(NCCn1nc(-c2ccccn2)c2c1CCCC2)Nc1ccc(F)cc1 ZINC000217507892 GH For-Sale Unstable TGFBR1 16 42 Cc1ccc(Nc2nc(C)cc(N3CCNCC3)n2)cc1 ZINC000217507894 CE In-Stock Unstable ROCK1 0 47 Cc1ccc(Nc2nc(C)cc(N3CCNCC3)n2)cc1 ZINC000217507894 CE In-Stock Unstable PRKD1 46 37 Cc1ccc(Nc2nc(C)cc(N3CCNCC3)n2)cc1 ZINC000217507894 CE In-Stock Unstable GALR2 49 44 Cc1ccc(Nc2nc(C)cc(N3CCNCC3)n2)cc1 ZINC000217507894 CE In-Stock Unstable KARS 57 38 COc1ccc(CCNC(=O)Nc2cccc3c(O)cccc23)cc1 ZINC000217507906 EH For-Sale Unstable CA2 15 47 COc1ccc(CCNC(=O)Nc2cccc3c(O)cccc23)cc1 ZINC000217507906 EH For-Sale Unstable BMP1 28 44 COc1ccc(CCNC(=O)Nc2cccc3c(O)cccc23)cc1 ZINC000217507906 EH For-Sale Unstable NQO2 48 44 COc1ccc(CCNC(=O)Nc2cccc3c(O)cccc23)cc1 ZINC000217507906 EH For-Sale Unstable CA1 23 47 COc1ccc(CCNC(=O)Nc2cccc3c(O)cccc23)cc1 ZINC000217507906 EH For-Sale Unstable TRPV1 27 67 COc1ccc(CCNC(=O)Nc2cccc3c(O)cccc23)cc1 ZINC000217507906 EH For-Sale Unstable MTNR1A 110 48 COc1ccc(CCNC(=O)Nc2cccc3c(O)cccc23)cc1 ZINC000217507906 EH For-Sale Unstable MTNR1B 90 44 COc1ccc(CCNC(=O)Nc2cccc3c(O)cccc23)cc1 ZINC000217507906 EH For-Sale Unstable CA12 18 47 COc1ccc(CCNC(=O)Nc2cccc3c(O)cccc23)cc1 ZINC000217507906 EH For-Sale Unstable PTGDR 23 42 COc1ccc(CCNC(=O)Nc2cccc3c(O)cccc23)cc1 ZINC000217507906 EH For-Sale Unstable CA9 23 46 COc1ccc(CCNC(=O)Nc2cccc3c(O)cccc23)cc1 ZINC000217507906 EH For-Sale Unstable NCE103 32 45 COc1ccc(CCNC(=O)Nc2cccc3c(O)cccc23)cc1 ZINC000217507906 EH For-Sale Unstable P96878_MYCTU 17 42 COc1ccc(CCNC(=O)Nc2cccc3c(O)cccc23)cc1 ZINC000217507906 EH For-Sale Unstable CAN2 0 42 BrCc1ccccc1N1CC[C@@H](N2CCCC2)C1 ZINC000217507922 DG For-Sale Unstable L3MBTL3 87 44 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Br)o1 ZINC000217507924 EH For-Sale Unstable SCAF_EBVB9 15 42 BrCc1ccccc1N1CC[C@H](N2CCCC2)C1 ZINC000217507992 DG For-Sale Unstable L3MBTL3 87 44 Cc1cc(Nc2ccc(N)cc2)nc(N2CCCC2)n1 ZINC000217508002 CF In-Stock Unstable GALR2 53 52 C[C@H](O)c1ccccc1NC(=O)/C=C\c1cccc(Br)c1 ZINC000217508005 EI For-Sale Unstable HDAC8 47 43 C[C@H](O)c1ccccc1NC(=O)/C=C\c1cccc(Br)c1 ZINC000217508005 EI For-Sale Unstable MMP2 22 51 C[C@H](O)c1ccccc1NC(=O)/C=C\c1cccc(Br)c1 ZINC000217508005 EI For-Sale Unstable HDAC1 20 40 C[C@H](O)c1ccccc1NC(=O)/C=C\c1cccc(Br)c1 ZINC000217508005 EI For-Sale Unstable HDAC6 34 43 C[C@H](O)c1ccccc1NC(=O)/C=C\c1cccc(Br)c1 ZINC000217508005 EI For-Sale Unstable MMP9 21 51 C[C@H](O)c1ccccc1NC(=O)/C=C\c1cccc(Br)c1 ZINC000217508005 EI For-Sale Unstable MMP1 25 51 C[C@H](O)c1ccccc1NC(=O)/C=C\c1cccc(Br)c1 ZINC000217508005 EI For-Sale Unstable TRPM8 0 57 COc1ccc(CCNC(=O)NCCCCCC(=O)O)cc1 ZINC000217508027 DE On-Demand Unstable SCNN1A 44 42 COc1ccc(CCNC(=O)NCCCCCC(=O)O)cc1 ZINC000217508027 DE On-Demand Unstable LTB4R 29 40 COc1ccc(CCNC(=O)NCCCCCC(=O)O)cc1 ZINC000217508027 DE On-Demand Unstable MTNR1A 62 43 COc1ccc(CCNC(=O)NCCCCCC(=O)O)cc1 ZINC000217508027 DE On-Demand Unstable MTNR1B 49 39 COc1ccc(CCNC(=O)NCCCCCC(=O)O)cc1 ZINC000217508027 DE On-Demand Unstable SLC2A1 0 40 COc1ccc(CCNC(=O)NCCCCCC(=O)O)cc1 ZINC000217508027 DE On-Demand Unstable PLA2G4B 41 32 COc1ccc(CCNC(=O)NCCCCCC(=O)O)cc1 ZINC000217508027 DE On-Demand Unstable EPHX2 34 45 COc1ccc(CCNC(=O)NCCCCCC(=O)O)cc1 ZINC000217508027 DE On-Demand Unstable FFAR1 47 38 COc1ccc(CCNC(=O)NCCCCCC(=O)O)cc1 ZINC000217508027 DE On-Demand Unstable HT1 0 40 COc1ccc(CCNC(=O)NCCCCCC(=O)O)cc1 ZINC000217508027 DE On-Demand Unstable FFAR4 47 42 COc1ccc(CCNC(=O)NCCCCCC(=O)O)cc1 ZINC000217508027 DE On-Demand Unstable LMGT2 0 40 CC(C)(N)Cc1ccc(S(C)(=O)=O)cc1F ZINC000217508038 BD For-Sale Unstable PTGS2 32 41 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1cccc(Br)c1 ZINC000217508097 EI For-Sale Unstable HDAC8 47 43 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1cccc(Br)c1 ZINC000217508097 EI For-Sale Unstable MMP2 22 51 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1cccc(Br)c1 ZINC000217508097 EI For-Sale Unstable HDAC1 20 40 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1cccc(Br)c1 ZINC000217508097 EI For-Sale Unstable HDAC6 34 43 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1cccc(Br)c1 ZINC000217508097 EI For-Sale Unstable MMP9 21 51 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1cccc(Br)c1 ZINC000217508097 EI For-Sale Unstable MMP1 25 51 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1cccc(Br)c1 ZINC000217508097 EI For-Sale Unstable TRPM8 0 57 BrCc1ccc(N2CC[C@@H](N3CCCC3)C2)nc1 ZINC000217508115 DF For-Sale Unstable HRH3 25 43 BrCc1ccc(N2CC[C@@H](N3CCCC3)C2)nc1 ZINC000217508115 DF For-Sale Unstable L3MBTL3 79 41 CCOCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCc1ccccc1 ZINC000217508125 GF In-Stock Unstable PLA2G4B 50 33 CCOCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCc1ccccc1 ZINC000217508125 GF In-Stock Unstable CCR8 20 41 NC[C@@H]1CCCN([C@@H]2CCc3ccccc32)C1 ZINC000217508142 BE For-Sale Unstable SLC6A1 0 43 COc1ccc(CCNC(=O)N[C@@H](C)c2ccc(OC)cc2)cc1 ZINC000217508175 EG On-Demand Unstable ANPEP 23 48 COc1ccc(CCNC(=O)N[C@@H](C)c2ccc(OC)cc2)cc1 ZINC000217508175 EG On-Demand Unstable BMP1 38 48 COc1ccc(CCNC(=O)N[C@@H](C)c2ccc(OC)cc2)cc1 ZINC000217508175 EG On-Demand Unstable ACACA 26 49 COc1ccc(CCNC(=O)N[C@@H](C)c2ccc(OC)cc2)cc1 ZINC000217508175 EG On-Demand Unstable ACACB 41 48 COc1ccc(CCNC(=O)N[C@@H](C)c2ccc(OC)cc2)cc1 ZINC000217508175 EG On-Demand Unstable MTNR1A 69 43 COc1ccc(CCNC(=O)N[C@@H](C)c2ccc(OC)cc2)cc1 ZINC000217508175 EG On-Demand Unstable MTNR1B 52 39 COc1ccc(CCNC(=O)N[C@@H](C)c2ccc(OC)cc2)cc1 ZINC000217508175 EG On-Demand Unstable MMP1 22 40 BrCc1ccc(N2CC[C@H](N3CCCC3)C2)nc1 ZINC000217508211 DF For-Sale Unstable HRH3 25 43 BrCc1ccc(N2CC[C@H](N3CCCC3)C2)nc1 ZINC000217508211 DF For-Sale Unstable L3MBTL3 79 41 Cc1nc(N2CCCCC2)cc(N2CCNCC2)n1 ZINC000217508224 CD In-Stock Unstable PRKD1 48 36 COc1ccc(CCNC(=O)N[C@H](C)c2ccc(OC)cc2)cc1 ZINC000217508252 EG On-Demand Unstable ANPEP 23 48 COc1ccc(CCNC(=O)N[C@H](C)c2ccc(OC)cc2)cc1 ZINC000217508252 EG On-Demand Unstable BMP1 38 48 COc1ccc(CCNC(=O)N[C@H](C)c2ccc(OC)cc2)cc1 ZINC000217508252 EG On-Demand Unstable ACACA 26 49 COc1ccc(CCNC(=O)N[C@H](C)c2ccc(OC)cc2)cc1 ZINC000217508252 EG On-Demand Unstable ACACB 41 48 COc1ccc(CCNC(=O)N[C@H](C)c2ccc(OC)cc2)cc1 ZINC000217508252 EG On-Demand Unstable MTNR1A 69 43 COc1ccc(CCNC(=O)N[C@H](C)c2ccc(OC)cc2)cc1 ZINC000217508252 EG On-Demand Unstable MTNR1B 52 39 COc1ccc(CCNC(=O)N[C@H](C)c2ccc(OC)cc2)cc1 ZINC000217508252 EG On-Demand Unstable MMP1 22 40 Fc1cc(CBr)ccc1N1CC[C@@H](N2CCCC2)C1 ZINC000217508312 EG For-Sale Unstable L3MBTL3 79 41 Cc1ccc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)cc1C ZINC000217508329 GI For-Sale Unstable TGFBR1 22 46 Cc1nc(N2CCNCC2)cc(N2CCOCC2)n1 ZINC000217508339 CC In-Stock Unstable PRKD1 46 37 Cc1nc(N2CCNCC2)cc(N2CCOCC2)n1 ZINC000217508339 CC In-Stock Unstable PIK3CB 51 39 C[C@@H]1CN(C[C@@H](O)COc2ccccc2CN)CCCO1 ZINC000217508350 CC For-Sale Unstable ADRB2 43 48 C[C@@H]1CN(C[C@@H](O)COc2ccccc2CN)CCCO1 ZINC000217508350 CC For-Sale Unstable ADRB3 44 48 C[C@@H]1CN(C[C@@H](O)COc2ccccc2CN)CCCO1 ZINC000217508350 CC For-Sale Unstable ABCB1 73 45 CCCCCc1ccccc1/C=C/C(=O)O ZINC000217508356 BH For-Sale Unstable PTGER2 25 55 CCCCCc1ccccc1/C=C/C(=O)O ZINC000217508356 BH For-Sale Unstable PTGER4 27 44 CCCCCc1ccccc1/C=C/C(=O)O ZINC000217508356 BH For-Sale Unstable PTGER3 25 55 CCOc1ccc(C)cc1[C@@H](C)NC(=O)NCCc1ccc(OC)cc1 ZINC000217508360 FI For-Sale Unstable MTNR1A 60 51 CCOc1ccc(C)cc1[C@@H](C)NC(=O)NCCc1ccc(OC)cc1 ZINC000217508360 FI For-Sale Unstable MTNR1B 48 51 Fc1cc(CBr)ccc1N1CC[C@H](N2CCCC2)C1 ZINC000217508407 EG For-Sale Unstable L3MBTL3 79 41 C[C@H]1CN(C[C@@H](O)COc2ccccc2CN)CCCO1 ZINC000217508430 CC For-Sale Unstable ADRB2 43 48 C[C@H]1CN(C[C@@H](O)COc2ccccc2CN)CCCO1 ZINC000217508430 CC For-Sale Unstable ADRB3 44 48 C[C@H]1CN(C[C@@H](O)COc2ccccc2CN)CCCO1 ZINC000217508430 CC For-Sale Unstable ABCB1 73 45 Cc1ccc(Nc2cc(N3CCNCC3)nc(C)n2)cc1 ZINC000217508435 CE In-Stock Unstable PRKD1 50 42 Cc1ccc(Nc2cc(N3CCNCC3)nc(C)n2)cc1 ZINC000217508435 CE In-Stock Unstable GALR2 50 42 Cc1ccc(Nc2cc(N3CCNCC3)nc(C)n2)cc1 ZINC000217508435 CE In-Stock Unstable PKD2 0 48 Cc1ccc(Nc2cc(N3CCNCC3)nc(C)n2)cc1 ZINC000217508435 CE In-Stock Unstable KARS 65 40 CCOc1ccc(C)cc1[C@H](C)NC(=O)NCCc1ccc(OC)cc1 ZINC000217508438 FI For-Sale Unstable MTNR1A 60 51 CCOc1ccc(C)cc1[C@H](C)NC(=O)NCCc1ccc(OC)cc1 ZINC000217508438 FI For-Sale Unstable MTNR1B 48 51 Cc1cc(C)cc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)c1 ZINC000217508441 GI For-Sale Unstable TGFBR1 21 43 CCOCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccccc1 ZINC000217508460 HF In-Stock Unstable CCR8 16 43 O=C(COCC(F)(F)C(F)F)N1CCCC[C@@H]1c1ccccn1 ZINC000217508493 EG In-Stock Unstable COLA 143 48 O=C(COCC(F)(F)C(F)F)N1CCCC[C@@H]1c1ccccn1 ZINC000217508493 EG In-Stock Unstable CPT1A 123 48 O=C(COCC(F)(F)C(F)F)N1CCCC[C@@H]1c1ccccn1 ZINC000217508493 EG In-Stock Unstable CPT2 44 34 Cc1nc(N2CCNCC2)cc(-n2ccnc2C)n1 ZINC000217508525 CC In-Stock Unstable PRKD1 47 35 CC[C@@H](NC(=O)NCCc1ccc(OC)cc1)c1ccc2c(c1)CCCC2 ZINC000217508543 FJ For-Sale Unstable MTR1B_CHICK 0 40 CC[C@@H](NC(=O)NCCc1ccc(OC)cc1)c1ccc2c(c1)CCCC2 ZINC000217508543 FJ For-Sale Unstable MTNR1A 66 38 CC[C@@H](NC(=O)NCCc1ccc(OC)cc1)c1ccc2c(c1)CCCC2 ZINC000217508543 FJ For-Sale Unstable MTNR1B 54 36 CCOCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)cc1 ZINC000217508560 IF In-Stock Unstable PLA2G4B 44 34 CCOCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)cc1 ZINC000217508560 IF In-Stock Unstable AKR1C3 18 43 COc1cccc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)c1 ZINC000217508566 GH For-Sale Unstable DRD4 47 37 COc1cccc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)c1 ZINC000217508566 GH For-Sale Unstable HRH2 26 45 COc1cccc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)c1 ZINC000217508566 GH For-Sale Unstable CCR3 36 44 COc1cccc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)c1 ZINC000217508566 GH For-Sale Unstable TGFBR1 24 43 COc1cccc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)c1 ZINC000217508566 GH For-Sale Unstable BUB1 45 33 O=C(COCC(F)(F)C(F)F)N1CCCC[C@H]1c1ccccn1 ZINC000217508574 EG In-Stock Unstable COLA 143 48 O=C(COCC(F)(F)C(F)F)N1CCCC[C@H]1c1ccccn1 ZINC000217508574 EG In-Stock Unstable CPT1A 123 48 O=C(COCC(F)(F)C(F)F)N1CCCC[C@H]1c1ccccn1 ZINC000217508574 EG In-Stock Unstable CPT2 44 34 CC[C@H](NC(=O)NCCc1ccc(OC)cc1)c1ccc2c(c1)CCCC2 ZINC000217508617 FJ For-Sale Unstable MTR1B_CHICK 0 40 CC[C@H](NC(=O)NCCc1ccc(OC)cc1)c1ccc2c(c1)CCCC2 ZINC000217508617 FJ For-Sale Unstable MTNR1A 66 38 CC[C@H](NC(=O)NCCc1ccc(OC)cc1)c1ccc2c(c1)CCCC2 ZINC000217508617 FJ For-Sale Unstable MTNR1B 54 36 COc1ccc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)cc1 ZINC000217508673 GH For-Sale Unstable DRD4 40 31 COc1ccc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)cc1 ZINC000217508673 GH For-Sale Unstable HRH2 16 42 COc1ccc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)cc1 ZINC000217508673 GH For-Sale Unstable TGFBR1 22 43 COc1ccc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)cc1 ZINC000217508673 GH For-Sale Unstable BUB1 44 33 CCOCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)c(OC)c1 ZINC000217508682 JF In-Stock Unstable PTGDR 22 42 CCOCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)c(OC)c1 ZINC000217508682 JF In-Stock Unstable IAP 0 41 CCOCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)c(OC)c1 ZINC000217508682 JF In-Stock Unstable SCMU_MYCTU 0 47 O=C(O)COc1ccccc1CN1CCN(CCO)C[C@@H](O)C1 ZINC000217508689 DB In-Stock Unstable PLA2G1B 51 36 O=C(O)COc1ccccc1CN1CCN(CCO)C[C@@H](O)C1 ZINC000217508689 DB In-Stock Unstable PLA2G2A 43 37 O=C(O)COc1ccccc1CN1CCN(CCO)C[C@@H](O)C1 ZINC000217508689 DB In-Stock Unstable PTGDR2 18 42 BrCc1cnc(N2CC[C@@H](N3CCCC3)C2)nc1 ZINC000217508698 DE For-Sale Unstable HRH3 18 40 BrCc1cnc(N2CC[C@@H](N3CCCC3)C2)nc1 ZINC000217508698 DE For-Sale Unstable L3MBTL3 63 41 CCc1ccc([C@@H](C)NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217508724 EH On-Demand Unstable ADRB2 15 43 CCc1ccc([C@@H](C)NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217508724 EH On-Demand Unstable ADRB3 18 40 CCc1ccc([C@@H](C)NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217508724 EH On-Demand Unstable BMP1 25 45 CCc1ccc([C@@H](C)NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217508724 EH On-Demand Unstable NQO2 23 40 CCc1ccc([C@@H](C)NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217508724 EH On-Demand Unstable ACACA 25 47 CCc1ccc([C@@H](C)NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217508724 EH On-Demand Unstable ACACB 36 47 CCc1ccc([C@@H](C)NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217508724 EH On-Demand Unstable MTNR1A 70 41 CCc1ccc([C@@H](C)NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217508724 EH On-Demand Unstable MTNR1B 55 41 CCc1ccc([C@@H](C)NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217508724 EH On-Demand Unstable CA9 15 44 BrCc1cnc(N2CC[C@H](N3CCCC3)C2)nc1 ZINC000217508787 DE For-Sale Unstable HRH3 18 40 BrCc1cnc(N2CC[C@H](N3CCCC3)C2)nc1 ZINC000217508787 DE For-Sale Unstable L3MBTL3 63 41 CCc1ccc([C@H](C)NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217508801 EH On-Demand Unstable ADRB2 15 43 CCc1ccc([C@H](C)NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217508801 EH On-Demand Unstable ADRB3 18 40 CCc1ccc([C@H](C)NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217508801 EH On-Demand Unstable BMP1 25 45 CCc1ccc([C@H](C)NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217508801 EH On-Demand Unstable NQO2 23 40 CCc1ccc([C@H](C)NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217508801 EH On-Demand Unstable ACACA 25 47 CCc1ccc([C@H](C)NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217508801 EH On-Demand Unstable ACACB 36 47 CCc1ccc([C@H](C)NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217508801 EH On-Demand Unstable MTNR1A 70 41 CCc1ccc([C@H](C)NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217508801 EH On-Demand Unstable MTNR1B 55 41 CCc1ccc([C@H](C)NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217508801 EH On-Demand Unstable CA9 15 44 COc1ccccc1C[C@@H](C)N1CCC[C@@H](N)C1 ZINC000217508807 BE For-Sale Unstable DPP4 16 40 Cc1cc(C)cc(N2CCN(C(=O)c3nc4ccc(F)cc4[nH]3)CC2=O)c1 ZINC000217508822 FF In-Stock Unstable GRIN2B 21 42 Cc1cc(C)cc(N2CCN(C(=O)c3nc4ccc(F)cc4[nH]3)CC2=O)c1 ZINC000217508822 FF In-Stock Unstable P2RX7 19 42 COc1cccc([C@@H](C)N2CCC[C@@H](CN)C2)c1 ZINC000217508845 BE On-Demand Unstable CHRNA10 34 43 C[C@H](O)c1ccccc1NC(=O)/C=C\c1cccc(F)c1 ZINC000217508852 CH For-Sale Unstable HDAC8 35 40 C[C@H](O)c1ccccc1NC(=O)/C=C\c1cccc(F)c1 ZINC000217508852 CH For-Sale Unstable MMP2 22 54 C[C@H](O)c1ccccc1NC(=O)/C=C\c1cccc(F)c1 ZINC000217508852 CH For-Sale Unstable NR1H4 22 40 C[C@H](O)c1ccccc1NC(=O)/C=C\c1cccc(F)c1 ZINC000217508852 CH For-Sale Unstable HDAC6 22 40 C[C@H](O)c1ccccc1NC(=O)/C=C\c1cccc(F)c1 ZINC000217508852 CH For-Sale Unstable MMP9 22 54 C[C@H](O)c1ccccc1NC(=O)/C=C\c1cccc(F)c1 ZINC000217508852 CH For-Sale Unstable IMPDH2 0 46 C[C@H](O)c1ccccc1NC(=O)/C=C\c1cccc(F)c1 ZINC000217508852 CH For-Sale Unstable MMP1 26 54 COc1ccccc1C[C@H](C)N1CCC[C@@H](N)C1 ZINC000217508881 BE For-Sale Unstable DPP4 16 40 O=C(NCCn1nc(-c2ccccn2)c2c1CCCC2)Nc1ccc(Cl)cc1 ZINC000217508888 GI For-Sale Unstable TGFBR1 18 43 Cc1cc(N2CC[C@@H](N3CCCC3)C2)ccc1CBr ZINC000217508898 DH For-Sale Unstable HRH3 27 43 Cc1cc(N2CC[C@@H](N3CCCC3)C2)ccc1CBr ZINC000217508898 DH For-Sale Unstable L3MBTL3 77 46 COc1ccc(CCNC(=O)N[C@@H](C)c2ccc3c(c2)CCCC3)cc1 ZINC000217508902 FI For-Sale Unstable MTNR1A 67 38 COc1ccc(CCNC(=O)N[C@@H](C)c2ccc3c(c2)CCCC3)cc1 ZINC000217508902 FI For-Sale Unstable MTNR1B 56 38 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1cccc(F)c1 ZINC000217508933 CH For-Sale Unstable HDAC8 35 40 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1cccc(F)c1 ZINC000217508933 CH For-Sale Unstable MMP2 22 54 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1cccc(F)c1 ZINC000217508933 CH For-Sale Unstable NR1H4 22 40 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1cccc(F)c1 ZINC000217508933 CH For-Sale Unstable HDAC6 22 40 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1cccc(F)c1 ZINC000217508933 CH For-Sale Unstable MMP9 22 54 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1cccc(F)c1 ZINC000217508933 CH For-Sale Unstable IMPDH2 0 46 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1cccc(F)c1 ZINC000217508933 CH For-Sale Unstable MMP1 26 54 COc1cccc([C@H](C)N2CCC[C@@H](CN)C2)c1 ZINC000217508939 BE On-Demand Unstable CHRNA10 34 43 Cc1cc(N2CC[C@H](N3CCCC3)C2)ccc1CBr ZINC000217508983 DH For-Sale Unstable HRH3 27 43 Cc1cc(N2CC[C@H](N3CCCC3)C2)ccc1CBr ZINC000217508983 DH For-Sale Unstable L3MBTL3 77 46 COc1ccc(CCNC(=O)N[C@H](C)c2ccc3c(c2)CCCC3)cc1 ZINC000217508986 FI For-Sale Unstable MTNR1A 67 38 COc1ccc(CCNC(=O)N[C@H](C)c2ccc3c(c2)CCCC3)cc1 ZINC000217508986 FI For-Sale Unstable MTNR1B 56 38 O=C(NCCn1nc(-c2ccccn2)c2c1CCCC2)Nc1cccc(Cl)c1 ZINC000217508999 GI For-Sale Unstable TGFBR1 17 42 C[C@H](O)c1ccccc1NC(=O)/C=C\c1cccnc1 ZINC000217509018 CF For-Sale Unstable MMP2 0 47 C[C@H](O)c1ccccc1NC(=O)/C=C\c1cccnc1 ZINC000217509018 CF For-Sale Unstable HDAC1 0 41 C[C@H](O)c1ccccc1NC(=O)/C=C\c1cccnc1 ZINC000217509018 CF For-Sale Unstable MMP9 0 47 C[C@H](O)c1ccccc1NC(=O)/C=C\c1cccnc1 ZINC000217509018 CF For-Sale Unstable MMP1 0 47 CCC(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217509047 CE For-Sale Unstable NPY5R 50 54 NC(=O)[C@H]1Cc2ccccc2CN1C(=O)C1CNC1 ZINC000217509058 CB On-Demand Unstable OPRD1 60 36 NC(=O)[C@H]1Cc2ccccc2CN1C(=O)C1CNC1 ZINC000217509058 CB On-Demand Unstable PREP 24 44 BrCc1ccc(Br)cc1N1CC[C@@H](N2CCCC2)C1 ZINC000217509088 GI For-Sale Unstable L3MBTL1 0 40 BrCc1ccc(Br)cc1N1CC[C@@H](N2CCCC2)C1 ZINC000217509088 GI For-Sale Unstable L3MBTL3 88 40 BrCc1ccc(Br)cc1N1CC[C@@H](N2CCCC2)C1 ZINC000217509088 GI For-Sale Unstable MBTD1 0 40 CN(C)[C@@H]1[C@H]2CC[C@@H]1CN(Cc1ccccc1OCCN1CCOCC1)C2 ZINC000217509101 FE In-Stock Unstable DRD5 0 54 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1cccnc1 ZINC000217509106 CF For-Sale Unstable MMP2 0 47 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1cccnc1 ZINC000217509106 CF For-Sale Unstable HDAC1 0 41 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1cccnc1 ZINC000217509106 CF For-Sale Unstable MMP9 0 47 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1cccnc1 ZINC000217509106 CF For-Sale Unstable MMP1 0 47 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable CA2 24 59 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable ADRB2 24 48 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable ADRB1 52 48 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable TSHR 41 32 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable HRH2 22 47 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable SRD5A2 0 43 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable PDGFRB 24 40 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable ADRB3 63 48 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable LTA4H 63 46 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable BMP1 31 45 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable NQO2 36 40 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable TACR2 22 46 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable CA1 59 59 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable MMP13 30 42 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable CCR3 25 42 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable SCN2A 25 47 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable HDAC8 17 47 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable RAF1 71 49 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable KDR 23 41 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable MMP16 0 41 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable MTNR1A 98 49 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable MTNR1B 90 58 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable MMP2 29 44 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable MMP3 33 43 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable MMP8 18 41 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable ROCK2 25 57 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable MMP14 15 41 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable SLC2A1 0 40 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable FAAH 30 45 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable NPY5R 34 57 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable MMP9 28 44 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable EPHX2 20 43 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable MMP12 21 41 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable F7 15 45 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable CA12 33 59 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable PDGFRA 52 41 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable PTGDR 25 45 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable CA9 38 59 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable MMP1 29 41 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable AMP1_PLAFQ 35 41 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable MCHR1 15 53 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable Q8MMZ8_EIMTE 76 49 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable F13A1 15 40 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable TAAR1 26 41 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable FFAR1 21 48 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable AKR1C3 16 40 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable YOPH 0 41 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable HT1 0 40 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable NCE103 43 59 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable ABCG2 17 43 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable CRTM 57 36 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable AKR1C2 35 40 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable MTCA1 15 47 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable P96878_MYCTU 25 47 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable ACAT 0 51 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable NAMPT 28 53 COc1ccc(CCNC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1 ZINC000217509113 FJ For-Sale Unstable LMGT2 0 40 O=C1OC2(CCN(C(=O)C3CCC3)CC2)c2ccccc21 ZINC000217509147 CE For-Sale Unstable NPY5R 62 53 Cc1nc(N(C)CC(=O)O)cc(N2CCOCC2)n1 ZINC000217509160 CC In-Stock Unstable PIK3CB 62 37 BrCc1ccc(Br)cc1N1CC[C@H](N2CCCC2)C1 ZINC000217509169 GI For-Sale Unstable L3MBTL1 0 40 BrCc1ccc(Br)cc1N1CC[C@H](N2CCCC2)C1 ZINC000217509169 GI For-Sale Unstable L3MBTL3 88 40 BrCc1ccc(Br)cc1N1CC[C@H](N2CCCC2)C1 ZINC000217509169 GI For-Sale Unstable MBTD1 0 40 CCc1c(C)c2ccc(OC(=O)[C@@H]3CC[C@@H](CNC(=O)OC(C)(C)C)CC3)cc2oc1=O ZINC000217509220 IJ In-Stock Unstable MAP2K1 0 43 COc1ccc(CCNC(=O)Nc2cc([N+](=O)[O-])ccc2Cl)cc1 ZINC000217509228 EH For-Sale Unstable BMP1 24 40 COc1ccc(CCNC(=O)Nc2cc([N+](=O)[O-])ccc2Cl)cc1 ZINC000217509228 EH For-Sale Unstable RAF1 39 42 COc1ccc(CCNC(=O)Nc2cc([N+](=O)[O-])ccc2Cl)cc1 ZINC000217509228 EH For-Sale Unstable MTNR1A 42 39 COc1ccc(CCNC(=O)Nc2cc([N+](=O)[O-])ccc2Cl)cc1 ZINC000217509228 EH For-Sale Unstable U38 0 43 COc1ccc(CCNC(=O)Nc2cc([N+](=O)[O-])ccc2Cl)cc1 ZINC000217509228 EH For-Sale Unstable Q8MMZ8_EIMTE 29 42 COc1ccc(CCNC(=O)Nc2cc([N+](=O)[O-])ccc2Cl)cc1 ZINC000217509228 EH For-Sale Unstable ABHD6 0 41 C=CCCC(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217509263 CF For-Sale Unstable NPY5R 41 48 BrCc1ccc(N2CC[C@@H](N3CCCC3)C2)cc1 ZINC000217509269 DG For-Sale Unstable HRH3 0 40 BrCc1ccc(N2CC[C@@H](N3CCCC3)C2)cc1 ZINC000217509269 DG For-Sale Unstable L3MBTL1 0 45 BrCc1ccc(N2CC[C@@H](N3CCCC3)C2)cc1 ZINC000217509269 DG For-Sale Unstable L3MBTL3 111 61 BrCc1ccc(N2CC[C@@H](N3CCCC3)C2)cc1 ZINC000217509269 DG For-Sale Unstable L3MBTL4 0 45 BrCc1ccc(N2CC[C@@H](N3CCCC3)C2)cc1 ZINC000217509269 DG For-Sale Unstable MBTD1 0 45 BrCc1ccc(N2CC[C@@H](N3CCCC3)C2)cc1 ZINC000217509269 DG For-Sale Unstable TP53BP1 0 45 O=C(NCCn1nc(-c2ccccn2)c2c1CCCC2)Nc1ccc2c(c1)OCO2 ZINC000217509270 HG For-Sale Unstable TGFBR1 24 44 COc1ccc(CCNC(=O)NCCCCl)cc1 ZINC000217509341 CE For-Sale Unstable CA2 15 50 COc1ccc(CCNC(=O)NCCCCl)cc1 ZINC000217509341 CE For-Sale Unstable SCNN1A 54 42 COc1ccc(CCNC(=O)NCCCCl)cc1 ZINC000217509341 CE For-Sale Unstable BMP1 33 40 COc1ccc(CCNC(=O)NCCCCl)cc1 ZINC000217509341 CE For-Sale Unstable CA1 16 50 COc1ccc(CCNC(=O)NCCCCl)cc1 ZINC000217509341 CE For-Sale Unstable MMP13 17 44 COc1ccc(CCNC(=O)NCCCCl)cc1 ZINC000217509341 CE For-Sale Unstable CTSL 16 42 COc1ccc(CCNC(=O)NCCCCl)cc1 ZINC000217509341 CE For-Sale Unstable MTNR1A 102 46 COc1ccc(CCNC(=O)NCCCCl)cc1 ZINC000217509341 CE For-Sale Unstable MTNR1B 82 46 COc1ccc(CCNC(=O)NCCCCl)cc1 ZINC000217509341 CE For-Sale Unstable MMP9 15 41 COc1ccc(CCNC(=O)NCCCCl)cc1 ZINC000217509341 CE For-Sale Unstable PTGDR 23 40 COc1ccc(CCNC(=O)NCCCCl)cc1 ZINC000217509341 CE For-Sale Unstable CA9 22 50 COc1ccc(CCNC(=O)NCCCCl)cc1 ZINC000217509341 CE For-Sale Unstable MMP1 17 41 COc1ccc(CCNC(=O)NCCCCl)cc1 ZINC000217509341 CE For-Sale Unstable NCE103 25 40 COc1ccc(CCNC(=O)NCCCCl)cc1 ZINC000217509341 CE For-Sale Unstable PROKR1 62 35 COc1ccc(CCNC(=O)NCCCCl)cc1 ZINC000217509341 CE For-Sale Unstable CAN2 0 40 BrCc1ccc(N2CC[C@H](N3CCCC3)C2)cc1 ZINC000217509345 DG For-Sale Unstable HRH3 0 40 BrCc1ccc(N2CC[C@H](N3CCCC3)C2)cc1 ZINC000217509345 DG For-Sale Unstable L3MBTL1 0 45 BrCc1ccc(N2CC[C@H](N3CCCC3)C2)cc1 ZINC000217509345 DG For-Sale Unstable L3MBTL3 111 61 BrCc1ccc(N2CC[C@H](N3CCCC3)C2)cc1 ZINC000217509345 DG For-Sale Unstable L3MBTL4 0 45 BrCc1ccc(N2CC[C@H](N3CCCC3)C2)cc1 ZINC000217509345 DG For-Sale Unstable MBTD1 0 45 BrCc1ccc(N2CC[C@H](N3CCCC3)C2)cc1 ZINC000217509345 DG For-Sale Unstable TP53BP1 0 45 CCOc1ccc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)cc1 ZINC000217509371 HI For-Sale Unstable TGFBR1 16 43 CCCCC(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217509380 CF For-Sale Unstable NPY5R 47 50 CSC[C@@](C)(O)CNc1ccc([N+](=O)[O-])c2nonc12 ZINC000217509387 CD On-Demand Unstable GSTM2 107 50 CSC[C@@](C)(O)CNc1ccc([N+](=O)[O-])c2nonc12 ZINC000217509387 CD On-Demand Unstable GSTP1 82 50 CSC[C@@](C)(O)CNc1ccc([N+](=O)[O-])c2nonc12 ZINC000217509387 CD On-Demand Unstable MYC 0 46 CSC[C@@](C)(O)CNc1ccc([N+](=O)[O-])c2nonc12 ZINC000217509387 CD On-Demand Unstable EPAS1 47 31 COc1ccc(CCNC(=O)NCCCl)cc1 ZINC000217509442 CD For-Sale Unstable CA2 15 52 COc1ccc(CCNC(=O)NCCCl)cc1 ZINC000217509442 CD For-Sale Unstable SCNN1A 31 40 COc1ccc(CCNC(=O)NCCCl)cc1 ZINC000217509442 CD For-Sale Unstable BMP1 31 41 COc1ccc(CCNC(=O)NCCCl)cc1 ZINC000217509442 CD For-Sale Unstable NQO2 31 41 COc1ccc(CCNC(=O)NCCCl)cc1 ZINC000217509442 CD For-Sale Unstable CA1 17 52 COc1ccc(CCNC(=O)NCCCl)cc1 ZINC000217509442 CD For-Sale Unstable MMP13 18 46 COc1ccc(CCNC(=O)NCCCl)cc1 ZINC000217509442 CD For-Sale Unstable CTSL 15 41 COc1ccc(CCNC(=O)NCCCl)cc1 ZINC000217509442 CD For-Sale Unstable MTNR1A 100 47 COc1ccc(CCNC(=O)NCCCl)cc1 ZINC000217509442 CD For-Sale Unstable MTNR1B 77 41 COc1ccc(CCNC(=O)NCCCl)cc1 ZINC000217509442 CD For-Sale Unstable MMP9 20 43 COc1ccc(CCNC(=O)NCCCl)cc1 ZINC000217509442 CD For-Sale Unstable MMP12 15 46 COc1ccc(CCNC(=O)NCCCl)cc1 ZINC000217509442 CD For-Sale Unstable PTGDR 24 42 COc1ccc(CCNC(=O)NCCCl)cc1 ZINC000217509442 CD For-Sale Unstable CA9 23 52 COc1ccc(CCNC(=O)NCCCl)cc1 ZINC000217509442 CD For-Sale Unstable MMP1 24 43 COc1ccc(CCNC(=O)NCCCl)cc1 ZINC000217509442 CD For-Sale Unstable NCE103 23 42 COc1ccc(CCNC(=O)NCCCl)cc1 ZINC000217509442 CD For-Sale Unstable PROKR1 64 37 C[C@H](c1ccc2c(c1)OCO2)N1CCC[C@@H](CN)C1 ZINC000217509447 CE For-Sale Unstable SSTR3 98 34 CSC[C@](C)(O)CNc1ccc([N+](=O)[O-])c2nonc12 ZINC000217509457 CD On-Demand Unstable GSTM2 87 46 CSC[C@](C)(O)CNc1ccc([N+](=O)[O-])c2nonc12 ZINC000217509457 CD On-Demand Unstable GSTP1 82 50 CSC[C@](C)(O)CNc1ccc([N+](=O)[O-])c2nonc12 ZINC000217509457 CD On-Demand Unstable MYC 0 46 CSC[C@](C)(O)CNc1ccc([N+](=O)[O-])c2nonc12 ZINC000217509457 CD On-Demand Unstable EPAS1 47 31 CC(C)(C)C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217509492 CF For-Sale Unstable AVPR1A 15 52 CC(C)(C)C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217509492 CF For-Sale Unstable NPY5R 53 54 CCOc1ccccc1NC(=O)NCCn1nc(-c2ccccn2)c2c1CCCC2 ZINC000217509499 HI For-Sale Unstable BUB1 47 36 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1Cl ZINC000217509549 DI For-Sale Unstable CXCL8 43 39 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1Cl ZINC000217509549 DI For-Sale Unstable KCNQ2 41 46 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1Cl ZINC000217509549 DI For-Sale Unstable UL26 19 42 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1Cl ZINC000217509549 DI For-Sale Unstable MMP1 0 51 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1Cl ZINC000217509549 DI For-Sale Unstable U53 0 42 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1Cl ZINC000217509549 DI For-Sale Unstable SCAF_EBVB9 15 42 C[C@@H](c1ccc2c(c1)OCO2)N1CCC[C@@H](CN)C1 ZINC000217509553 CE For-Sale Unstable SSTR3 98 34 CCCCOC(=O)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217509558 FI For-Sale Unstable BMP1 22 41 CCCCOC(=O)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217509558 FI For-Sale Unstable CA1 20 43 CCCCOC(=O)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217509558 FI For-Sale Unstable MTNR1A 68 43 CCCCOC(=O)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217509558 FI For-Sale Unstable MTNR1B 56 42 CCCCOC(=O)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217509558 FI For-Sale Unstable SLC6A5 24 48 CCCCOC(=O)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217509558 FI For-Sale Unstable CAPN2 22 41 CCCCOC(=O)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217509558 FI For-Sale Unstable CA12 15 44 CCCCOC(=O)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217509558 FI For-Sale Unstable CA9 20 42 CCCCOC(=O)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217509558 FI For-Sale Unstable ABCG2 15 42 CCCCOC(=O)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217509558 FI For-Sale Unstable ACAT 0 44 COc1ccc(CNC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)cc1 ZINC000217509596 HG For-Sale Unstable DRD4 40 31 COc1ccc(CNC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)cc1 ZINC000217509596 HG For-Sale Unstable TGFBR1 18 43 CCOCC(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217509599 CD For-Sale Unstable NPY5R 44 49 C[C@@](O)(CNC(=O)c1noc2c1CCCC2)c1cc2ccccc2s1 ZINC000217509611 FG In-Stock Unstable PANC 57 40 CN(CC(=O)O)c1nccc(N2CCCC2)n1 ZINC000217509619 BC In-Stock Unstable SORD 81 39 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1Cl ZINC000217509632 DI For-Sale Unstable CXCL8 43 39 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1Cl ZINC000217509632 DI For-Sale Unstable KCNQ2 41 46 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1Cl ZINC000217509632 DI For-Sale Unstable UL26 19 42 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1Cl ZINC000217509632 DI For-Sale Unstable MMP1 0 51 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1Cl ZINC000217509632 DI For-Sale Unstable U53 0 42 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1Cl ZINC000217509632 DI For-Sale Unstable SCAF_EBVB9 15 42 CCCCCNc1ccc(C(=O)O)cc1S(=O)(=O)NCCCOCC ZINC000217509662 FF In-Stock Unstable PLA2G4B 50 36 COc1ccc(CCNC(=O)Nc2ccccc2Sc2ccccc2)cc1 ZINC000217509668 GK For-Sale Unstable BMP1 42 44 COc1ccc(CCNC(=O)Nc2ccccc2Sc2ccccc2)cc1 ZINC000217509668 GK For-Sale Unstable NQO2 26 40 COc1ccc(CCNC(=O)Nc2ccccc2Sc2ccccc2)cc1 ZINC000217509668 GK For-Sale Unstable MTNR1A 71 41 COc1ccc(CCNC(=O)Nc2ccccc2Sc2ccccc2)cc1 ZINC000217509668 GK For-Sale Unstable MTNR1B 58 37 COc1ccc(CCNC(=O)Nc2ccccc2Sc2ccccc2)cc1 ZINC000217509668 GK For-Sale Unstable MMP3 25 40 COc1ccc(CCNC(=O)Nc2ccccc2Sc2ccccc2)cc1 ZINC000217509668 GK For-Sale Unstable MMP9 20 40 COc1ccc(CCNC(=O)Nc2ccccc2Sc2ccccc2)cc1 ZINC000217509668 GK For-Sale Unstable CA9 18 41 COc1ccc(CCNC(=O)Nc2ccccc2Sc2ccccc2)cc1 ZINC000217509668 GK For-Sale Unstable MMP1 22 40 C[C@](O)(CNC(=O)c1noc2c1CCCC2)c1cc2ccccc2s1 ZINC000217509690 FG In-Stock Unstable PANC 57 40 CC(C)(C)CC(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217509715 DG For-Sale Unstable NPY5R 46 50 C[C@H](O)c1ccccc1NC(=O)/C=C\c1cccc(Cl)c1 ZINC000217509716 DI For-Sale Unstable HDAC8 36 40 C[C@H](O)c1ccccc1NC(=O)/C=C\c1cccc(Cl)c1 ZINC000217509716 DI For-Sale Unstable MMP2 22 54 C[C@H](O)c1ccccc1NC(=O)/C=C\c1cccc(Cl)c1 ZINC000217509716 DI For-Sale Unstable NR1H4 22 41 C[C@H](O)c1ccccc1NC(=O)/C=C\c1cccc(Cl)c1 ZINC000217509716 DI For-Sale Unstable HDAC6 24 40 C[C@H](O)c1ccccc1NC(=O)/C=C\c1cccc(Cl)c1 ZINC000217509716 DI For-Sale Unstable MMP9 22 54 C[C@H](O)c1ccccc1NC(=O)/C=C\c1cccc(Cl)c1 ZINC000217509716 DI For-Sale Unstable MMP1 27 54 C[C@H](O)c1ccccc1NC(=O)/C=C\c1cccc(Cl)c1 ZINC000217509716 DI For-Sale Unstable SCAF_EBVB9 15 43 C[C@H](O)c1ccccc1NC(=O)/C=C\c1cccc(Cl)c1 ZINC000217509716 DI For-Sale Unstable TRPM8 0 57 C[C@H](O)c1ccccc1NC(=O)/C=C\c1cccc(Cl)c1 ZINC000217509716 DI For-Sale Unstable TUBA4A 0 42 C[C@@H]1CCC[C@@]([C@@H](O)Cc2cc(F)ccc2F)(N(C)C)C1 ZINC000217509728 CG For-Sale Unstable DPP4 20 42 CN(CC(=O)O)c1nccc(N2CCOCC2)n1 ZINC000217509737 CB In-Stock Unstable PIK3CA 33 42 CN(CC(=O)O)c1nccc(N2CCOCC2)n1 ZINC000217509737 CB In-Stock Unstable SORD 71 37 CN(CC(=O)O)c1nccc(N2CCOCC2)n1 ZINC000217509737 CB In-Stock Unstable PIK3CB 52 35 CN(CC(=O)O)c1nccc(N2CCOCC2)n1 ZINC000217509737 CB In-Stock Unstable EPHB4 75 36 CN(CC(=O)O)c1nccc(N2CCOCC2)n1 ZINC000217509737 CB In-Stock Unstable SMG1 45 37 COc1cc([C@@H]2N3CCc4ccccc4[C@H]3CN2S(=O)(=O)c2ccc(C)cc2)ccc1OS(=O)(=O)c1ccc(C)cc1 ZINC000217509769 KK In-Stock Unstable FKBP1A 15 43 COc1ccc(CCNC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)cc1 ZINC000217509779 FJ For-Sale Unstable BMP1 17 43 COc1ccc(CCNC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)cc1 ZINC000217509779 FJ For-Sale Unstable CA1 16 42 COc1ccc(CCNC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)cc1 ZINC000217509779 FJ For-Sale Unstable TRPV1 19 61 COc1ccc(CCNC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)cc1 ZINC000217509779 FJ For-Sale Unstable GUAB 0 42 COc1ccc(CCNC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)cc1 ZINC000217509779 FJ For-Sale Unstable RAF1 87 64 COc1ccc(CCNC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)cc1 ZINC000217509779 FJ For-Sale Unstable KDR 16 54 COc1ccc(CCNC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)cc1 ZINC000217509779 FJ For-Sale Unstable MTNR1A 47 37 COc1ccc(CCNC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)cc1 ZINC000217509779 FJ For-Sale Unstable EPHX2 29 47 COc1ccc(CCNC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)cc1 ZINC000217509779 FJ For-Sale Unstable PTGDR 15 43 COc1ccc(CCNC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)cc1 ZINC000217509779 FJ For-Sale Unstable MCHR1 17 46 COc1ccc(CCNC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)cc1 ZINC000217509779 FJ For-Sale Unstable Q8MMZ8_EIMTE 110 64 COc1ccc(CCNC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)cc1 ZINC000217509779 FJ For-Sale Unstable BRAF 17 47 COc1ccc(CCNC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)cc1 ZINC000217509779 FJ For-Sale Unstable NCE103 31 42 COc1ccc(CCNC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)cc1 ZINC000217509779 FJ For-Sale Unstable ROS1 18 54 COc1ccc(CCNC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)cc1 ZINC000217509779 FJ For-Sale Unstable IMDH_CRYPV 28 44 COc1ccc(CCNC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)cc1 ZINC000217509779 FJ For-Sale Unstable BLM 0 44 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1cccc(Cl)c1 ZINC000217509820 DI For-Sale Unstable HDAC8 36 40 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1cccc(Cl)c1 ZINC000217509820 DI For-Sale Unstable MMP2 22 54 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1cccc(Cl)c1 ZINC000217509820 DI For-Sale Unstable NR1H4 22 41 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1cccc(Cl)c1 ZINC000217509820 DI For-Sale Unstable HDAC6 24 40 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1cccc(Cl)c1 ZINC000217509820 DI For-Sale Unstable MMP9 22 54 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1cccc(Cl)c1 ZINC000217509820 DI For-Sale Unstable MMP1 27 54 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1cccc(Cl)c1 ZINC000217509820 DI For-Sale Unstable SCAF_EBVB9 15 43 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1cccc(Cl)c1 ZINC000217509820 DI For-Sale Unstable TRPM8 0 57 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1cccc(Cl)c1 ZINC000217509820 DI For-Sale Unstable TUBA4A 0 42 Clc1ccc(CBr)c(N2CC[C@@H](N3CCCC3)C2)c1 ZINC000217509822 EH For-Sale Unstable L3MBTL3 66 43 O=C1OC2(CCN(C(=O)c3ccccc3)CC2)c2ccccc21 ZINC000217509827 DF For-Sale Unstable AVPR1A 17 55 O=C1OC2(CCN(C(=O)c3ccccc3)CC2)c2ccccc21 ZINC000217509827 DF For-Sale Unstable NPY5R 56 58 Cc1cc(N2CCOCC2)nc(N(C)CC(=O)O)n1 ZINC000217509869 CC In-Stock Unstable PIK3CB 64 37 C[C@@H]1CCC[C@]([C@@H](O)Cc2cc(F)ccc2F)(N(C)C)C1 ZINC000217509870 CG For-Sale Unstable DPP4 20 42 COc1ccc(CCNC(=O)Nc2ccc(N)cc2Cl)cc1 ZINC000217509901 DG For-Sale Unstable CA2 15 50 COc1ccc(CCNC(=O)Nc2ccc(N)cc2Cl)cc1 ZINC000217509901 DG For-Sale Unstable BMP1 23 41 COc1ccc(CCNC(=O)Nc2ccc(N)cc2Cl)cc1 ZINC000217509901 DG For-Sale Unstable CA1 18 50 COc1ccc(CCNC(=O)Nc2ccc(N)cc2Cl)cc1 ZINC000217509901 DG For-Sale Unstable TRPV1 24 54 COc1ccc(CCNC(=O)Nc2ccc(N)cc2Cl)cc1 ZINC000217509901 DG For-Sale Unstable RAF1 42 45 COc1ccc(CCNC(=O)Nc2ccc(N)cc2Cl)cc1 ZINC000217509901 DG For-Sale Unstable FLT1 19 43 COc1ccc(CCNC(=O)Nc2ccc(N)cc2Cl)cc1 ZINC000217509901 DG For-Sale Unstable MTNR1A 74 42 COc1ccc(CCNC(=O)Nc2ccc(N)cc2Cl)cc1 ZINC000217509901 DG For-Sale Unstable MTNR1B 55 39 COc1ccc(CCNC(=O)Nc2ccc(N)cc2Cl)cc1 ZINC000217509901 DG For-Sale Unstable CA12 15 50 COc1ccc(CCNC(=O)Nc2ccc(N)cc2Cl)cc1 ZINC000217509901 DG For-Sale Unstable PTGDR 17 40 COc1ccc(CCNC(=O)Nc2ccc(N)cc2Cl)cc1 ZINC000217509901 DG For-Sale Unstable CA9 26 50 COc1ccc(CCNC(=O)Nc2ccc(N)cc2Cl)cc1 ZINC000217509901 DG For-Sale Unstable Q8MMZ8_EIMTE 33 45 COc1ccc(CCNC(=O)Nc2ccc(N)cc2Cl)cc1 ZINC000217509901 DG For-Sale Unstable NCE103 27 42 COc1ccc(CCNC(=O)Nc2ccc(N)cc2Cl)cc1 ZINC000217509901 DG For-Sale Unstable PROKR1 60 34 COc1ccc(CCNC(=O)Nc2ccc(N)cc2Cl)cc1 ZINC000217509901 DG For-Sale Unstable CAN2 0 42 CC(C)(C)c1ccc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)cc1 ZINC000217509914 HJ For-Sale Unstable TGFBR1 16 44 CC(C)(C)c1ccc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)cc1 ZINC000217509914 HJ For-Sale Unstable DOT1L 50 33 Clc1ccc(CBr)c(N2CC[C@H](N3CCCC3)C2)c1 ZINC000217509926 EH For-Sale Unstable L3MBTL3 66 43 O=C1OC2(CCN(C(=O)c3ccncc3)CC2)c2ccccc21 ZINC000217509929 DE For-Sale Unstable AVPR1A 23 53 O=C1OC2(CCN(C(=O)c3ccncc3)CC2)c2ccccc21 ZINC000217509929 DE For-Sale Unstable NPY5R 60 55 O=C1OC2(CCN(C(=O)c3ccncc3)CC2)c2ccccc21 ZINC000217509929 DE For-Sale Unstable CCR8 24 41 COc1ccc(CCNC(=O)Nc2ccc(N)c(Cl)c2)cc1 ZINC000217510006 DG For-Sale Unstable CA2 18 46 COc1ccc(CCNC(=O)Nc2ccc(N)c(Cl)c2)cc1 ZINC000217510006 DG For-Sale Unstable BMP1 18 45 COc1ccc(CCNC(=O)Nc2ccc(N)c(Cl)c2)cc1 ZINC000217510006 DG For-Sale Unstable CA1 36 46 COc1ccc(CCNC(=O)Nc2ccc(N)c(Cl)c2)cc1 ZINC000217510006 DG For-Sale Unstable TRPV1 0 48 COc1ccc(CCNC(=O)Nc2ccc(N)c(Cl)c2)cc1 ZINC000217510006 DG For-Sale Unstable RAF1 54 46 COc1ccc(CCNC(=O)Nc2ccc(N)c(Cl)c2)cc1 ZINC000217510006 DG For-Sale Unstable MTNR1A 64 39 COc1ccc(CCNC(=O)Nc2ccc(N)c(Cl)c2)cc1 ZINC000217510006 DG For-Sale Unstable MTNR1B 54 36 COc1ccc(CCNC(=O)Nc2ccc(N)c(Cl)c2)cc1 ZINC000217510006 DG For-Sale Unstable CA12 24 46 COc1ccc(CCNC(=O)Nc2ccc(N)c(Cl)c2)cc1 ZINC000217510006 DG For-Sale Unstable PTGDR 22 45 COc1ccc(CCNC(=O)Nc2ccc(N)c(Cl)c2)cc1 ZINC000217510006 DG For-Sale Unstable CA9 27 46 COc1ccc(CCNC(=O)Nc2ccc(N)c(Cl)c2)cc1 ZINC000217510006 DG For-Sale Unstable Q8MMZ8_EIMTE 50 46 COc1ccc(CCNC(=O)Nc2ccc(N)c(Cl)c2)cc1 ZINC000217510006 DG For-Sale Unstable NCE103 44 46 COc1ccc(CCNC(=O)Nc2ccc(N)c(Cl)c2)cc1 ZINC000217510006 DG For-Sale Unstable PROKR1 68 36 COc1ccc(CCNC(=O)Nc2ccc(N)c(Cl)c2)cc1 ZINC000217510006 DG For-Sale Unstable P96878_MYCTU 19 41 COc1ccc(CCNC(=O)Nc2ccc(N)c(Cl)c2)cc1 ZINC000217510006 DG For-Sale Unstable CAN2 0 41 COc1ccc(CCNC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)cc1 ZINC000217510031 HG For-Sale Unstable DRD4 40 31 COc1ccc(CCNC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)cc1 ZINC000217510031 HG For-Sale Unstable TGFBR1 17 43 Clc1ccc(N2CC[C@@H](N3CCCC3)C2)c(CBr)c1 ZINC000217510033 EH For-Sale Unstable L3MBTL3 68 40 O=C1OC2(CCN(C(=O)c3cccnc3)CC2)c2ccccc21 ZINC000217510046 DE In-Stock Unstable AVPR1A 22 49 O=C1OC2(CCN(C(=O)c3cccnc3)CC2)c2ccccc21 ZINC000217510046 DE In-Stock Unstable NPY5R 61 54 C[C@@H](CO)S(=O)(=O)NCc1ccccc1Cl ZINC000217510054 CD For-Sale Unstable CXCL8 51 33 Clc1ccc(N2CC[C@H](N3CCCC3)C2)c(CBr)c1 ZINC000217510107 EH For-Sale Unstable L3MBTL3 68 40 COc1ccc(CCNC(=O)Nc2ccc(I)cc2C)cc1 ZINC000217510117 HH On-Demand Unstable BMP1 20 40 COc1ccc(CCNC(=O)Nc2ccc(I)cc2C)cc1 ZINC000217510117 HH On-Demand Unstable RAF1 40 43 COc1ccc(CCNC(=O)Nc2ccc(I)cc2C)cc1 ZINC000217510117 HH On-Demand Unstable MTNR1A 73 42 COc1ccc(CCNC(=O)Nc2ccc(I)cc2C)cc1 ZINC000217510117 HH On-Demand Unstable MTNR1B 54 39 COc1ccc(CCNC(=O)Nc2ccc(I)cc2C)cc1 ZINC000217510117 HH On-Demand Unstable CA9 16 43 COc1ccc(CCNC(=O)Nc2ccc(I)cc2C)cc1 ZINC000217510117 HH On-Demand Unstable Q8MMZ8_EIMTE 31 43 C[C@H](CO)S(=O)(=O)NCc1ccccc1Cl ZINC000217510129 CD For-Sale Unstable CXCL8 51 33 Cc1n[nH]c([C@@H]2CCCN2C(=O)CCN2Cc3ccccc3C2=O)n1 ZINC000217510144 ED In-Stock Unstable PRCP 40 41 Cc1n[nH]c([C@@H]2CCCN2C(=O)CCN2Cc3ccccc3C2=O)n1 ZINC000217510144 ED In-Stock Unstable COLA 122 48 Cc1n[nH]c([C@@H]2CCCN2C(=O)CCN2Cc3ccccc3C2=O)n1 ZINC000217510144 ED In-Stock Unstable CPT1A 110 48 Cc1n[nH]c([C@@H]2CCCN2C(=O)CCN2Cc3ccccc3C2=O)n1 ZINC000217510144 ED In-Stock Unstable PREP 20 52 O=C(NCCn1nc(-c2ccccn2)c2c1CCCC2)NC12CC3CC(CC(C3)C1)C2 ZINC000217510154 HI For-Sale Unstable EPHX2 87 44 O=C1OC2(CCN(C(=O)c3ccccn3)CC2)c2ccccc21 ZINC000217510156 DE In-Stock Unstable AVPR1A 24 53 O=C1OC2(CCN(C(=O)c3ccccn3)CC2)c2ccccc21 ZINC000217510156 DE In-Stock Unstable NPY5R 61 53 CN(Cc1cccc(F)c1)C(=O)c1cc(Br)ccc1I ZINC000217510174 II For-Sale Unstable HSP90AB1 25 48 CN(Cc1cccc(F)c1)C(=O)c1cc(Br)ccc1I ZINC000217510174 II For-Sale Unstable HSD17B2 24 44 NC[C@@H]1CC[C@@H](c2ccccc2)C[C@@H]1N1CCCOCC1 ZINC000217510192 CF For-Sale Unstable SLC18A3 48 38 Cc1n[nH]c([C@H]2CCCN2C(=O)CCN2Cc3ccccc3C2=O)n1 ZINC000217510227 ED In-Stock Unstable PRCP 40 41 Cc1n[nH]c([C@H]2CCCN2C(=O)CCN2Cc3ccccc3C2=O)n1 ZINC000217510227 ED In-Stock Unstable COLA 122 48 Cc1n[nH]c([C@H]2CCCN2C(=O)CCN2Cc3ccccc3C2=O)n1 ZINC000217510227 ED In-Stock Unstable CPT1A 110 48 Cc1n[nH]c([C@H]2CCCN2C(=O)CCN2Cc3ccccc3C2=O)n1 ZINC000217510227 ED In-Stock Unstable PREP 20 52 C=CCN(CC=C)C(=O)NCCc1ccc(OC)cc1 ZINC000217510244 CF On-Demand Unstable MMP16 0 42 C=CCN(CC=C)C(=O)NCCc1ccc(OC)cc1 ZINC000217510244 CF On-Demand Unstable MTNR1A 54 37 C=CCN(CC=C)C(=O)NCCc1ccc(OC)cc1 ZINC000217510244 CF On-Demand Unstable MTNR1B 44 37 C=CCN(CC=C)C(=O)NCCc1ccc(OC)cc1 ZINC000217510244 CF On-Demand Unstable CA9 18 47 COc1ccc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)cc1OC ZINC000217510257 HH For-Sale Unstable TGFBR1 18 45 COc1ccc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)cc1OC ZINC000217510257 HH For-Sale Unstable QPCT 20 48 COc1ccc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)cc1OC ZINC000217510257 HH For-Sale Unstable ENPP1 70 36 COc1ccc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)cc1OC ZINC000217510257 HH For-Sale Unstable BUB1 46 35 NC[C@H]1CC[C@@H](c2ccccc2)C[C@@H]1N1CCCOCC1 ZINC000217510265 CF For-Sale Unstable SLC18A3 48 38 O=C1OC2(CCN(C(=O)c3cnccn3)CC2)c2ccccc21 ZINC000217510270 DD For-Sale Unstable AVPR1A 23 51 O=C1OC2(CCN(C(=O)c3cnccn3)CC2)c2ccccc21 ZINC000217510270 DD For-Sale Unstable NPY5R 60 53 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Br)s1 ZINC000217510281 FI For-Sale Unstable UL26 18 42 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Br)s1 ZINC000217510281 FI For-Sale Unstable U53 0 42 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Br)s1 ZINC000217510281 FI For-Sale Unstable SCAF_EBVB9 24 42 COc1ccc(CCNC(=O)NC2CCCCCCCCCCC2)cc1 ZINC000217510325 FK For-Sale Unstable ADRB1 26 41 COc1ccc(CCNC(=O)NC2CCCCCCCCCCC2)cc1 ZINC000217510325 FK For-Sale Unstable CNR1 20 49 COc1ccc(CCNC(=O)NC2CCCCCCCCCCC2)cc1 ZINC000217510325 FK For-Sale Unstable HRH2 20 46 COc1ccc(CCNC(=O)NC2CCCCCCCCCCC2)cc1 ZINC000217510325 FK For-Sale Unstable CNR2 27 47 COc1ccc(CCNC(=O)NC2CCCCCCCCCCC2)cc1 ZINC000217510325 FK For-Sale Unstable BMP1 22 53 COc1ccc(CCNC(=O)NC2CCCCCCCCCCC2)cc1 ZINC000217510325 FK For-Sale Unstable NQO2 35 41 COc1ccc(CCNC(=O)NC2CCCCCCCCCCC2)cc1 ZINC000217510325 FK For-Sale Unstable MMP13 27 42 COc1ccc(CCNC(=O)NC2CCCCCCCCCCC2)cc1 ZINC000217510325 FK For-Sale Unstable CTSK 20 55 COc1ccc(CCNC(=O)NC2CCCCCCCCCCC2)cc1 ZINC000217510325 FK For-Sale Unstable CTSL 15 55 COc1ccc(CCNC(=O)NC2CCCCCCCCCCC2)cc1 ZINC000217510325 FK For-Sale Unstable CACNA1B 15 41 COc1ccc(CCNC(=O)NC2CCCCCCCCCCC2)cc1 ZINC000217510325 FK For-Sale Unstable CCR3 22 41 COc1ccc(CCNC(=O)NC2CCCCCCCCCCC2)cc1 ZINC000217510325 FK For-Sale Unstable MTNR1A 99 40 COc1ccc(CCNC(=O)NC2CCCCCCCCCCC2)cc1 ZINC000217510325 FK For-Sale Unstable MTNR1B 80 43 COc1ccc(CCNC(=O)NC2CCCCCCCCCCC2)cc1 ZINC000217510325 FK For-Sale Unstable MMP3 34 43 COc1ccc(CCNC(=O)NC2CCCCCCCCCCC2)cc1 ZINC000217510325 FK For-Sale Unstable FAAH 30 44 COc1ccc(CCNC(=O)NC2CCCCCCCCCCC2)cc1 ZINC000217510325 FK For-Sale Unstable EPHX2 49 69 COc1ccc(CCNC(=O)NC2CCCCCCCCCCC2)cc1 ZINC000217510325 FK For-Sale Unstable CA9 18 46 COc1ccc(CCNC(=O)NC2CCCCCCCCCCC2)cc1 ZINC000217510325 FK For-Sale Unstable MCHR1 18 45 COc1ccc(CCNC(=O)NC2CCCCCCCCCCC2)cc1 ZINC000217510325 FK For-Sale Unstable BIRC2 29 42 COc1cc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)cc(OC)c1 ZINC000217510358 HH For-Sale Unstable DRD4 42 33 COc1cc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)cc(OC)c1 ZINC000217510358 HH For-Sale Unstable ZAP70 40 33 COc1cc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)cc(OC)c1 ZINC000217510358 HH For-Sale Unstable TGFBR1 21 43 NC[C@@H]1CC[C@H](c2ccccc2)C[C@@H]1N1CCCOCC1 ZINC000217510360 CF For-Sale Unstable SLC18A3 48 38 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Br)s1 ZINC000217510365 FI For-Sale Unstable UL26 18 42 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Br)s1 ZINC000217510365 FI For-Sale Unstable U53 0 42 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Br)s1 ZINC000217510365 FI For-Sale Unstable SCAF_EBVB9 24 42 Cc1cc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)no1 ZINC000217510368 DE For-Sale Unstable AVPR1A 23 53 Cc1cc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)no1 ZINC000217510368 DE For-Sale Unstable NPY5R 50 50 O=C(NCCCCl)Nc1cc(F)ccc1F ZINC000217510377 BF For-Sale Unstable CCR3 25 45 CN(Cc1cccc(F)c1)C(=O)c1cc(I)ccc1O ZINC000217510387 GG On-Demand Unstable HSP90AB1 52 53 CN(Cc1cccc(F)c1)C(=O)c1cc(I)ccc1O ZINC000217510387 GG On-Demand Unstable HSD17B2 28 47 CN(Cc1cccc(F)c1)C(=O)c1cc(I)ccc1O ZINC000217510387 GG On-Demand Unstable LIMK2 27 41 CCCCNc1ccc(C(=O)O)cc1S(=O)(=O)NCCCOC(C)C ZINC000217510428 FF In-Stock Unstable PLA2G4B 41 34 COc1ccc(CCNC(=O)N2CCN(CCN)CC2)cc1 ZINC000217510433 DC For-Sale Unstable DRD4 47 36 COc1ccc(CCNC(=O)N2CCN(CCN)CC2)cc1 ZINC000217510433 DC For-Sale Unstable HTR2A 17 52 COc1ccc(CCNC(=O)N2CCN(CCN)CC2)cc1 ZINC000217510433 DC For-Sale Unstable DRD3 40 38 COc1ccc(CCNC(=O)N2CCN(CCN)CC2)cc1 ZINC000217510433 DC For-Sale Unstable SIGMAR1 21 56 COc1ccc(CCNC(=O)N2CCN(CCN)CC2)cc1 ZINC000217510433 DC For-Sale Unstable MMP13 25 45 COc1ccc(CCNC(=O)N2CCN(CCN)CC2)cc1 ZINC000217510433 DC For-Sale Unstable MTNR1A 52 38 COc1ccc(CCNC(=O)N2CCN(CCN)CC2)cc1 ZINC000217510433 DC For-Sale Unstable MTNR1B 46 38 COc1ccc(CCNC(=O)N2CCN(CCN)CC2)cc1 ZINC000217510433 DC For-Sale Unstable MMP3 22 48 COc1ccc(CCNC(=O)N2CCN(CCN)CC2)cc1 ZINC000217510433 DC For-Sale Unstable MMP9 25 48 COc1ccc(CCNC(=O)N2CCN(CCN)CC2)cc1 ZINC000217510433 DC For-Sale Unstable MMP7 28 48 COc1ccc(CCNC(=O)N2CCN(CCN)CC2)cc1 ZINC000217510433 DC For-Sale Unstable CA9 18 45 COc1ccc(CCNC(=O)N2CCN(CCN)CC2)cc1 ZINC000217510433 DC For-Sale Unstable MMP1 26 48 COc1ccc(CCNC(=O)N2CCN(CCN)CC2)cc1 ZINC000217510433 DC For-Sale Unstable PROKR1 60 35 NC[C@H]1CC[C@H](c2ccccc2)C[C@@H]1N1CCCOCC1 ZINC000217510434 CF For-Sale Unstable SLC18A3 48 38 NC(=O)Cc1nc([C@@H]2Cc3ccccc3O2)n(Cc2ccc3c(c2)OCO3)n1 ZINC000217510471 GD In-Stock Unstable NOS2 75 33 O=C1OC2(CCN(C(=O)c3cccs3)CC2)c2ccccc21 ZINC000217510474 DG For-Sale Unstable AVPR1A 15 51 O=C1OC2(CCN(C(=O)c3cccs3)CC2)c2ccccc21 ZINC000217510474 DG For-Sale Unstable NPY5R 45 51 COc1cccc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)c1OC ZINC000217510476 HH For-Sale Unstable TGFBR1 17 41 COc1ccc(CCNC(=O)NCCN2CCNCC2)cc1 ZINC000217510530 DC On-Demand Unstable DRD4 49 38 COc1ccc(CCNC(=O)NCCN2CCNCC2)cc1 ZINC000217510530 DC On-Demand Unstable MMP13 17 43 COc1ccc(CCNC(=O)NCCN2CCNCC2)cc1 ZINC000217510530 DC On-Demand Unstable CCR3 26 40 COc1ccc(CCNC(=O)NCCN2CCNCC2)cc1 ZINC000217510530 DC On-Demand Unstable MTNR1A 48 40 COc1ccc(CCNC(=O)NCCN2CCNCC2)cc1 ZINC000217510530 DC On-Demand Unstable MTNR1B 48 36 COc1ccc(CCNC(=O)NCCN2CCNCC2)cc1 ZINC000217510530 DC On-Demand Unstable CA9 15 44 COc1ccc(CCNC(=O)NCCN2CCNCC2)cc1 ZINC000217510530 DC On-Demand Unstable MMP1 20 43 NC(=O)Cc1nc([C@H]2Cc3ccccc3O2)n(Cc2ccc3c(c2)OCO3)n1 ZINC000217510564 GD In-Stock Unstable NOS2 75 33 O=C1OC2(CCN(C(=O)CC3CCCC3)CC2)c2ccccc21 ZINC000217510579 DG For-Sale Unstable NPY5R 56 48 COc1ccc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)c(OC)c1 ZINC000217510596 HH For-Sale Unstable DRD4 42 33 COc1ccc(CCNC(=O)NCCCN2CCOCC2)cc1 ZINC000217510653 DD On-Demand Unstable HTR1A 27 41 COc1ccc(CCNC(=O)NCCCN2CCOCC2)cc1 ZINC000217510653 DD On-Demand Unstable DRD2 31 42 COc1ccc(CCNC(=O)NCCCN2CCOCC2)cc1 ZINC000217510653 DD On-Demand Unstable CNR1 15 45 COc1ccc(CCNC(=O)NCCCN2CCOCC2)cc1 ZINC000217510653 DD On-Demand Unstable DRD1 16 40 COc1ccc(CCNC(=O)NCCCN2CCOCC2)cc1 ZINC000217510653 DD On-Demand Unstable DRD4 44 34 COc1ccc(CCNC(=O)NCCCN2CCOCC2)cc1 ZINC000217510653 DD On-Demand Unstable ACHE 15 41 COc1ccc(CCNC(=O)NCCCN2CCOCC2)cc1 ZINC000217510653 DD On-Demand Unstable HRH2 24 40 COc1ccc(CCNC(=O)NCCCN2CCOCC2)cc1 ZINC000217510653 DD On-Demand Unstable HTR2A 25 45 COc1ccc(CCNC(=O)NCCCN2CCOCC2)cc1 ZINC000217510653 DD On-Demand Unstable HTR2C 23 41 COc1ccc(CCNC(=O)NCCCN2CCOCC2)cc1 ZINC000217510653 DD On-Demand Unstable DRD3 45 40 COc1ccc(CCNC(=O)NCCCN2CCOCC2)cc1 ZINC000217510653 DD On-Demand Unstable THRB 0 43 COc1ccc(CCNC(=O)NCCCN2CCOCC2)cc1 ZINC000217510653 DD On-Demand Unstable HTR7 25 40 COc1ccc(CCNC(=O)NCCCN2CCOCC2)cc1 ZINC000217510653 DD On-Demand Unstable TACR2 34 55 COc1ccc(CCNC(=O)NCCCN2CCOCC2)cc1 ZINC000217510653 DD On-Demand Unstable HRH3 18 49 COc1ccc(CCNC(=O)NCCCN2CCOCC2)cc1 ZINC000217510653 DD On-Demand Unstable SIGMAR1 25 47 COc1ccc(CCNC(=O)NCCCN2CCOCC2)cc1 ZINC000217510653 DD On-Demand Unstable MMP13 29 44 COc1ccc(CCNC(=O)NCCCN2CCOCC2)cc1 ZINC000217510653 DD On-Demand Unstable BCHE 28 40 COc1ccc(CCNC(=O)NCCCN2CCOCC2)cc1 ZINC000217510653 DD On-Demand Unstable CCR3 30 48 COc1ccc(CCNC(=O)NCCCN2CCOCC2)cc1 ZINC000217510653 DD On-Demand Unstable CHRNA7 21 48 COc1ccc(CCNC(=O)NCCCN2CCOCC2)cc1 ZINC000217510653 DD On-Demand Unstable ADAM17 21 45 COc1ccc(CCNC(=O)NCCCN2CCOCC2)cc1 ZINC000217510653 DD On-Demand Unstable MTNR1A 58 41 COc1ccc(CCNC(=O)NCCCN2CCOCC2)cc1 ZINC000217510653 DD On-Demand Unstable MTNR1B 48 38 COc1ccc(CCNC(=O)NCCCN2CCOCC2)cc1 ZINC000217510653 DD On-Demand Unstable MMP3 23 41 COc1ccc(CCNC(=O)NCCCN2CCOCC2)cc1 ZINC000217510653 DD On-Demand Unstable ABCB1 15 43 COc1ccc(CCNC(=O)NCCCN2CCOCC2)cc1 ZINC000217510653 DD On-Demand Unstable MMP9 28 41 COc1ccc(CCNC(=O)NCCCN2CCOCC2)cc1 ZINC000217510653 DD On-Demand Unstable PTGDS 33 46 COc1ccc(CCNC(=O)NCCCN2CCOCC2)cc1 ZINC000217510653 DD On-Demand Unstable EPHX2 22 45 COc1ccc(CCNC(=O)NCCCN2CCOCC2)cc1 ZINC000217510653 DD On-Demand Unstable PTGDR 0 42 COc1ccc(CCNC(=O)NCCCN2CCOCC2)cc1 ZINC000217510653 DD On-Demand Unstable CA9 18 45 COc1ccc(CCNC(=O)NCCCN2CCOCC2)cc1 ZINC000217510653 DD On-Demand Unstable MMP1 32 46 COc1ccc(CCNC(=O)NCCCN2CCOCC2)cc1 ZINC000217510653 DD On-Demand Unstable MCHR1 19 40 O=C1OC2(CCN(C(=O)c3ccccc3F)CC2)c2ccccc21 ZINC000217510690 EG For-Sale Unstable AVPR1A 24 60 O=C1OC2(CCN(C(=O)c3ccccc3F)CC2)c2ccccc21 ZINC000217510690 EG For-Sale Unstable NPY5R 49 52 CCN(C(=O)NCCc1ccc(OC)cc1)c1ccccc1 ZINC000217510773 CG For-Sale Unstable BMP1 32 43 CCN(C(=O)NCCc1ccc(OC)cc1)c1ccccc1 ZINC000217510773 CG For-Sale Unstable NQO2 26 40 CCN(C(=O)NCCc1ccc(OC)cc1)c1ccccc1 ZINC000217510773 CG For-Sale Unstable MMP16 0 40 CCN(C(=O)NCCc1ccc(OC)cc1)c1ccccc1 ZINC000217510773 CG For-Sale Unstable MTNR1A 101 40 CCN(C(=O)NCCc1ccc(OC)cc1)c1ccccc1 ZINC000217510773 CG For-Sale Unstable MTNR1B 84 39 CCN(C(=O)NCCc1ccc(OC)cc1)c1ccccc1 ZINC000217510773 CG For-Sale Unstable MMP2 18 40 CCN(C(=O)NCCc1ccc(OC)cc1)c1ccccc1 ZINC000217510773 CG For-Sale Unstable MMP3 24 41 CCN(C(=O)NCCc1ccc(OC)cc1)c1ccccc1 ZINC000217510773 CG For-Sale Unstable MMP8 16 40 CCN(C(=O)NCCc1ccc(OC)cc1)c1ccccc1 ZINC000217510773 CG For-Sale Unstable NPY5R 17 43 CCN(C(=O)NCCc1ccc(OC)cc1)c1ccccc1 ZINC000217510773 CG For-Sale Unstable MMP9 27 41 CCN(C(=O)NCCc1ccc(OC)cc1)c1ccccc1 ZINC000217510773 CG For-Sale Unstable PTGDR 19 40 CCN(C(=O)NCCc1ccc(OC)cc1)c1ccccc1 ZINC000217510773 CG For-Sale Unstable CA9 18 45 CCN(C(=O)NCCc1ccc(OC)cc1)c1ccccc1 ZINC000217510773 CG For-Sale Unstable MMP1 26 41 CCN(C(=O)NCCc1ccc(OC)cc1)c1ccccc1 ZINC000217510773 CG For-Sale Unstable PROKR1 54 35 O=C1OC2(CCN(C(=O)c3ccc(F)cc3)CC2)c2ccccc21 ZINC000217510795 EG For-Sale Unstable AVPR1A 16 54 O=C1OC2(CCN(C(=O)c3ccc(F)cc3)CC2)c2ccccc21 ZINC000217510795 EG For-Sale Unstable INHA 20 49 O=C1OC2(CCN(C(=O)c3ccc(F)cc3)CC2)c2ccccc21 ZINC000217510795 EG For-Sale Unstable NPY5R 52 60 CC1(C)OC(=O)Nc2ccc(OCc3ccccc3)cc21 ZINC000217510796 CI For-Sale Unstable MAOA 30 45 CC1(C)OC(=O)Nc2ccc(OCc3ccccc3)cc21 ZINC000217510796 CI For-Sale Unstable MAOB 84 53 CC1(C)OC(=O)Nc2ccc(OCc3ccccc3)cc21 ZINC000217510796 CI For-Sale Unstable GRM1 23 42 CC1(C)OC(=O)Nc2ccc(OCc3ccccc3)cc21 ZINC000217510796 CI For-Sale Unstable FFAR1 23 40 Cc1ccccc1CN(C)C(=O)c1ccc(O)cc1O ZINC000217510797 CF On-Demand Unstable HSP90AB1 51 55 COc1ccc(Cl)cc1NC(=O)NCCn1nc(-c2ccccn2)c2c1CCCC2 ZINC000217510800 II For-Sale Unstable CPT1A 44 32 COc1ccc(CCNC(=O)NCc2cccc(CN)c2)cc1 ZINC000217510871 DE For-Sale Unstable ANPEP 25 43 COc1ccc(CCNC(=O)NCc2cccc(CN)c2)cc1 ZINC000217510871 DE For-Sale Unstable BMP1 25 40 COc1ccc(CCNC(=O)NCc2cccc(CN)c2)cc1 ZINC000217510871 DE For-Sale Unstable NQO2 39 43 COc1ccc(CCNC(=O)NCc2cccc(CN)c2)cc1 ZINC000217510871 DE For-Sale Unstable CA1 16 46 COc1ccc(CCNC(=O)NCc2cccc(CN)c2)cc1 ZINC000217510871 DE For-Sale Unstable TRPV1 0 47 COc1ccc(CCNC(=O)NCc2cccc(CN)c2)cc1 ZINC000217510871 DE For-Sale Unstable MMP13 26 42 COc1ccc(CCNC(=O)NCc2cccc(CN)c2)cc1 ZINC000217510871 DE For-Sale Unstable ROCK1 24 41 COc1ccc(CCNC(=O)NCc2cccc(CN)c2)cc1 ZINC000217510871 DE For-Sale Unstable MTNR1A 107 47 COc1ccc(CCNC(=O)NCc2cccc(CN)c2)cc1 ZINC000217510871 DE For-Sale Unstable MTNR1B 87 49 COc1ccc(CCNC(=O)NCc2cccc(CN)c2)cc1 ZINC000217510871 DE For-Sale Unstable ROCK2 35 45 COc1ccc(CCNC(=O)NCc2cccc(CN)c2)cc1 ZINC000217510871 DE For-Sale Unstable PTGDR 24 40 COc1ccc(CCNC(=O)NCc2cccc(CN)c2)cc1 ZINC000217510871 DE For-Sale Unstable CA9 22 46 COc1ccc(CCNC(=O)NCc2cccc(CN)c2)cc1 ZINC000217510871 DE For-Sale Unstable NCE103 26 42 COc1ccc(CCNC(=O)NCc2cccc(CN)c2)cc1 ZINC000217510871 DE For-Sale Unstable PROKR1 47 32 COc1ccc(CCNC(=O)NCc2cccc(CN)c2)cc1 ZINC000217510871 DE For-Sale Unstable CAN2 0 42 O=C1OC2(CCN(C(=O)Cc3cccs3)CC2)c2ccccc21 ZINC000217510892 EF For-Sale Unstable NPY5R 40 49 COc1ccc(CCNC(=O)Nc2cc(Cl)ccc2O)cc1 ZINC000217510992 DG For-Sale Unstable THRA 28 48 COc1ccc(CCNC(=O)Nc2cc(Cl)ccc2O)cc1 ZINC000217510992 DG For-Sale Unstable ADRB3 29 44 COc1ccc(CCNC(=O)Nc2cc(Cl)ccc2O)cc1 ZINC000217510992 DG For-Sale Unstable THRB 37 48 COc1ccc(CCNC(=O)Nc2cc(Cl)ccc2O)cc1 ZINC000217510992 DG For-Sale Unstable NQO2 30 41 COc1ccc(CCNC(=O)Nc2cc(Cl)ccc2O)cc1 ZINC000217510992 DG For-Sale Unstable CA1 19 45 COc1ccc(CCNC(=O)Nc2cc(Cl)ccc2O)cc1 ZINC000217510992 DG For-Sale Unstable TRPV1 31 52 COc1ccc(CCNC(=O)Nc2cc(Cl)ccc2O)cc1 ZINC000217510992 DG For-Sale Unstable S1PR4 22 40 COc1ccc(CCNC(=O)Nc2cc(Cl)ccc2O)cc1 ZINC000217510992 DG For-Sale Unstable RAF1 40 43 COc1ccc(CCNC(=O)Nc2cc(Cl)ccc2O)cc1 ZINC000217510992 DG For-Sale Unstable MTNR1A 71 43 COc1ccc(CCNC(=O)Nc2cc(Cl)ccc2O)cc1 ZINC000217510992 DG For-Sale Unstable MTNR1B 54 43 COc1ccc(CCNC(=O)Nc2cc(Cl)ccc2O)cc1 ZINC000217510992 DG For-Sale Unstable KCNMA1 27 43 COc1ccc(CCNC(=O)Nc2cc(Cl)ccc2O)cc1 ZINC000217510992 DG For-Sale Unstable CA12 17 45 COc1ccc(CCNC(=O)Nc2cc(Cl)ccc2O)cc1 ZINC000217510992 DG For-Sale Unstable PTGDR 27 40 COc1ccc(CCNC(=O)Nc2cc(Cl)ccc2O)cc1 ZINC000217510992 DG For-Sale Unstable CA9 24 45 COc1ccc(CCNC(=O)Nc2cc(Cl)ccc2O)cc1 ZINC000217510992 DG For-Sale Unstable U38 0 45 COc1ccc(CCNC(=O)Nc2cc(Cl)ccc2O)cc1 ZINC000217510992 DG For-Sale Unstable Q8MMZ8_EIMTE 30 43 COc1ccc(CCNC(=O)Nc2cc(Cl)ccc2O)cc1 ZINC000217510992 DG For-Sale Unstable NCE103 42 47 COc1ccc(CCNC(=O)Nc2cc(Cl)ccc2O)cc1 ZINC000217510992 DG For-Sale Unstable PROKR1 43 34 COc1ccc(CCNC(=O)Nc2cc(Cl)ccc2O)cc1 ZINC000217510992 DG For-Sale Unstable CAN2 0 47 COc1ccc(CCNC(=O)Nc2cc(Cl)ccc2O)cc1 ZINC000217510992 DG For-Sale Unstable PQSD 0 40 Cc1ccccc1CN(C)C(=O)c1cc(I)ccc1O ZINC000217510998 GH On-Demand Unstable HSP90AB1 43 50 N#Cc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217510999 EF For-Sale Unstable NPY5R 38 49 O=C(NCCn1nc(-c2ccccn2)c2c1CCCC2)Nc1cccc(C(F)(F)F)c1 ZINC000217511015 IJ For-Sale Unstable CCR3 18 43 O=C(NCCn1nc(-c2ccccn2)c2c1CCCC2)Nc1cccc(C(F)(F)F)c1 ZINC000217511015 IJ For-Sale Unstable KDR 18 40 O=C(NCCn1nc(-c2ccccn2)c2c1CCCC2)Nc1cccc(C(F)(F)F)c1 ZINC000217511015 IJ For-Sale Unstable TGFBR1 15 42 O=C(NCCn1nc(-c2ccccn2)c2c1CCCC2)Nc1cccc(C(F)(F)F)c1 ZINC000217511015 IJ For-Sale Unstable BRAF 40 41 CC(C)(C)OC(=O)N1CC[C@H](CNCc2cc(Cl)cc(Cl)c2)C1 ZINC000217511098 FI For-Sale Unstable CACNA1I 79 44 CC(C)(C)OC(=O)N1CC[C@H](CNCc2cc(Cl)cc(Cl)c2)C1 ZINC000217511098 FI For-Sale Unstable GPR119 44 42 CC[C@@H](C)[C@H](c1ccccc1)[C@@H](Br)c1ccc(OC)cc1 ZINC000217511102 EK For-Sale Unstable AOC3 18 40 CC[C@@H](C)[C@H](c1ccccc1)[C@@H](Br)c1ccc(OC)cc1 ZINC000217511102 EK For-Sale Unstable GPR88 0 41 COc1ccc(CCNC(=O)Nc2cc(S(=O)(=O)N3CCOCC3)ccc2Cl)cc1 ZINC000217511112 JF For-Sale Unstable CA2 15 43 COc1ccc(CCNC(=O)Nc2cc(S(=O)(=O)N3CCOCC3)ccc2Cl)cc1 ZINC000217511112 JF For-Sale Unstable LPL 40 40 COc1ccc(CCNC(=O)Nc2cc(S(=O)(=O)N3CCOCC3)ccc2Cl)cc1 ZINC000217511112 JF For-Sale Unstable BMP1 85 42 COc1ccc(CCNC(=O)Nc2cc(S(=O)(=O)N3CCOCC3)ccc2Cl)cc1 ZINC000217511112 JF For-Sale Unstable CA1 16 43 COc1ccc(CCNC(=O)Nc2cc(S(=O)(=O)N3CCOCC3)ccc2Cl)cc1 ZINC000217511112 JF For-Sale Unstable MMP13 55 41 COc1ccc(CCNC(=O)Nc2cc(S(=O)(=O)N3CCOCC3)ccc2Cl)cc1 ZINC000217511112 JF For-Sale Unstable MMP3 52 40 COc1ccc(CCNC(=O)Nc2cc(S(=O)(=O)N3CCOCC3)ccc2Cl)cc1 ZINC000217511112 JF For-Sale Unstable MMP9 40 41 COc1ccc(CCNC(=O)Nc2cc(S(=O)(=O)N3CCOCC3)ccc2Cl)cc1 ZINC000217511112 JF For-Sale Unstable TGM2 28 45 COc1ccc(CCNC(=O)Nc2cc(S(=O)(=O)N3CCOCC3)ccc2Cl)cc1 ZINC000217511112 JF For-Sale Unstable CA12 15 43 COc1ccc(CCNC(=O)Nc2cc(S(=O)(=O)N3CCOCC3)ccc2Cl)cc1 ZINC000217511112 JF For-Sale Unstable MMP7 46 40 COc1ccc(CCNC(=O)Nc2cc(S(=O)(=O)N3CCOCC3)ccc2Cl)cc1 ZINC000217511112 JF For-Sale Unstable CA9 22 43 COc1ccc(CCNC(=O)Nc2cc(S(=O)(=O)N3CCOCC3)ccc2Cl)cc1 ZINC000217511112 JF For-Sale Unstable MMP1 49 41 COc1ccc(CCNC(=O)Nc2cc(S(=O)(=O)N3CCOCC3)ccc2Cl)cc1 ZINC000217511112 JF For-Sale Unstable MURF 0 43 COc1ccc(CCNC(=O)Nc2cc(S(=O)(=O)N3CCOCC3)ccc2Cl)cc1 ZINC000217511112 JF For-Sale Unstable NAMPT 31 43 O=C1OC2(CCN(C(=O)CCc3ccccc3)CC2)c2ccccc21 ZINC000217511117 EG For-Sale Unstable SIGMAR1 26 62 O=C1OC2(CCN(C(=O)CCc3ccccc3)CC2)c2ccccc21 ZINC000217511117 EG For-Sale Unstable NPY5R 48 53 O=C(NCCn1nc(-c2ccccn2)c2c1CCCC2)Nc1ccc(C(F)(F)F)cc1 ZINC000217511121 IJ For-Sale Unstable TRPV1 15 40 O=C(NCCn1nc(-c2ccccn2)c2c1CCCC2)Nc1ccc(C(F)(F)F)cc1 ZINC000217511121 IJ For-Sale Unstable EPHX2 26 48 O=C(Nc1ccccc1)[C@@H]1CCCN(C[C@@H](O)COC[C@@H]2CCCO2)C1 ZINC000217511147 FD On-Demand Unstable SLC6A1 96 39 CC[C@H](C)[C@H](c1ccccc1)[C@@H](Br)c1ccc(OC)cc1 ZINC000217511173 EK For-Sale Unstable AOC3 18 40 CC[C@H](C)[C@H](c1ccccc1)[C@@H](Br)c1ccc(OC)cc1 ZINC000217511173 EK For-Sale Unstable GPR88 0 41 CC(C)OCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NC1CCCC1 ZINC000217511191 GF In-Stock Unstable AMY2 46 31 Cc1cccc(CC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217511223 EG In-Stock Unstable NPY5R 37 46 COc1ccc(CCNC(=O)Nc2ncccn2)cc1 ZINC000217511231 CD For-Sale Unstable BMP1 24 45 COc1ccc(CCNC(=O)Nc2ncccn2)cc1 ZINC000217511231 CD For-Sale Unstable NQO2 28 42 COc1ccc(CCNC(=O)Nc2ncccn2)cc1 ZINC000217511231 CD For-Sale Unstable CA1 15 47 COc1ccc(CCNC(=O)Nc2ncccn2)cc1 ZINC000217511231 CD For-Sale Unstable TRPV1 0 60 COc1ccc(CCNC(=O)Nc2ncccn2)cc1 ZINC000217511231 CD For-Sale Unstable CTSL 16 43 COc1ccc(CCNC(=O)Nc2ncccn2)cc1 ZINC000217511231 CD For-Sale Unstable RAF1 40 40 COc1ccc(CCNC(=O)Nc2ncccn2)cc1 ZINC000217511231 CD For-Sale Unstable MTNR1A 94 43 COc1ccc(CCNC(=O)Nc2ncccn2)cc1 ZINC000217511231 CD For-Sale Unstable MTNR1B 78 40 COc1ccc(CCNC(=O)Nc2ncccn2)cc1 ZINC000217511231 CD For-Sale Unstable ROCK2 16 54 COc1ccc(CCNC(=O)Nc2ncccn2)cc1 ZINC000217511231 CD For-Sale Unstable PTGDR 24 44 COc1ccc(CCNC(=O)Nc2ncccn2)cc1 ZINC000217511231 CD For-Sale Unstable CA9 22 47 COc1ccc(CCNC(=O)Nc2ncccn2)cc1 ZINC000217511231 CD For-Sale Unstable Q8MMZ8_EIMTE 27 40 COc1ccc(CCNC(=O)Nc2ncccn2)cc1 ZINC000217511231 CD For-Sale Unstable PROKR1 60 34 O=C(NCCn1nc(-c2ccccn2)c2c1CCCC2)Nc1ccc(Cl)c(Cl)c1 ZINC000217511248 IJ For-Sale Unstable TGFBR1 18 47 O=C(NCCn1nc(-c2ccccn2)c2c1CCCC2)Nc1ccc(Cl)c(Cl)c1 ZINC000217511248 IJ For-Sale Unstable SHH 22 41 O=C(NCCn1nc(-c2ccccn2)c2c1CCCC2)Nc1ccc(Cl)c(Cl)c1 ZINC000217511248 IJ For-Sale Unstable IMDH_CRYPV 20 41 CC[C@@H](C)[C@@H](c1ccccc1)[C@@H](Br)c1ccc(OC)cc1 ZINC000217511258 EK For-Sale Unstable AOC3 18 40 CC[C@@H](C)[C@@H](c1ccccc1)[C@@H](Br)c1ccc(OC)cc1 ZINC000217511258 EK For-Sale Unstable GPR88 0 41 CC(C)OCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NC1CCCCC1 ZINC000217511291 GG In-Stock Unstable AMY2 48 33 O=C(Nc1ccccc1)[C@@H]1CCCN(C[C@@H](O)COCc2cccs2)C1 ZINC000217511322 FF On-Demand Unstable SLC6A1 85 39 COc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217511328 EF For-Sale Unstable AVPR1A 21 44 COc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217511328 EF For-Sale Unstable NPY5R 42 54 CC[C@H](C)[C@@H](c1ccccc1)[C@@H](Br)c1ccc(OC)cc1 ZINC000217511342 EK For-Sale Unstable AOC3 18 40 CC[C@H](C)[C@@H](c1ccccc1)[C@@H](Br)c1ccc(OC)cc1 ZINC000217511342 EK For-Sale Unstable GPR88 0 41 COc1ccc(-c2coc3cc(OCCN4C[C@@H]5C[C@H](C4)c4cccc(=O)n4C5)ccc3c2=O)cc1 ZINC000217511344 JI In-Stock Unstable ALDH2 111 46 COc1ccc(-c2coc3cc(OCCN4C[C@@H]5C[C@H](C4)c4cccc(=O)n4C5)ccc3c2=O)cc1 ZINC000217511344 JI In-Stock Unstable IL2 27 44 COc1ccc(-c2coc3cc(OCCN4C[C@@H]5C[C@H](C4)c4cccc(=O)n4C5)ccc3c2=O)cc1 ZINC000217511344 JI In-Stock Unstable CHRNA4 36 48 COc1ccc(CCNC(=O)N2CCCC2)cc1 ZINC000217511347 BE For-Sale Unstable DRD4 41 32 COc1ccc(CCNC(=O)N2CCCC2)cc1 ZINC000217511347 BE For-Sale Unstable HRH2 17 45 COc1ccc(CCNC(=O)N2CCCC2)cc1 ZINC000217511347 BE For-Sale Unstable BMP1 42 36 COc1ccc(CCNC(=O)N2CCCC2)cc1 ZINC000217511347 BE For-Sale Unstable NQO2 35 40 COc1ccc(CCNC(=O)N2CCCC2)cc1 ZINC000217511347 BE For-Sale Unstable HRH3 17 55 COc1ccc(CCNC(=O)N2CCCC2)cc1 ZINC000217511347 BE For-Sale Unstable SIGMAR1 17 50 COc1ccc(CCNC(=O)N2CCCC2)cc1 ZINC000217511347 BE For-Sale Unstable MMP13 45 44 COc1ccc(CCNC(=O)N2CCCC2)cc1 ZINC000217511347 BE For-Sale Unstable CTSK 18 43 COc1ccc(CCNC(=O)N2CCCC2)cc1 ZINC000217511347 BE For-Sale Unstable CTSL 17 43 COc1ccc(CCNC(=O)N2CCCC2)cc1 ZINC000217511347 BE For-Sale Unstable MMP16 0 41 COc1ccc(CCNC(=O)N2CCCC2)cc1 ZINC000217511347 BE For-Sale Unstable MTNR1A 107 40 COc1ccc(CCNC(=O)N2CCCC2)cc1 ZINC000217511347 BE For-Sale Unstable MTNR1B 95 41 COc1ccc(CCNC(=O)N2CCCC2)cc1 ZINC000217511347 BE For-Sale Unstable MMP2 24 41 COc1ccc(CCNC(=O)N2CCCC2)cc1 ZINC000217511347 BE For-Sale Unstable MMP3 46 52 COc1ccc(CCNC(=O)N2CCCC2)cc1 ZINC000217511347 BE For-Sale Unstable MMP8 27 44 COc1ccc(CCNC(=O)N2CCCC2)cc1 ZINC000217511347 BE For-Sale Unstable MMP9 43 52 COc1ccc(CCNC(=O)N2CCCC2)cc1 ZINC000217511347 BE For-Sale Unstable EPHX2 15 48 COc1ccc(CCNC(=O)N2CCCC2)cc1 ZINC000217511347 BE For-Sale Unstable MMP12 20 44 COc1ccc(CCNC(=O)N2CCCC2)cc1 ZINC000217511347 BE For-Sale Unstable DPP7 42 50 COc1ccc(CCNC(=O)N2CCCC2)cc1 ZINC000217511347 BE For-Sale Unstable PTGDR 27 40 COc1ccc(CCNC(=O)N2CCCC2)cc1 ZINC000217511347 BE For-Sale Unstable MMP7 36 52 COc1ccc(CCNC(=O)N2CCCC2)cc1 ZINC000217511347 BE For-Sale Unstable CA9 24 49 COc1ccc(CCNC(=O)N2CCCC2)cc1 ZINC000217511347 BE For-Sale Unstable MMP1 51 52 COc1ccc(CCNC(=O)N2CCCC2)cc1 ZINC000217511347 BE For-Sale Unstable PROKR1 61 35 CCCCOc1ccc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)cc1 ZINC000217511366 IJ For-Sale Unstable HRH2 23 41 CCCCOc1ccc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)cc1 ZINC000217511366 IJ For-Sale Unstable TGFBR1 19 42 CCCCOc1ccc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)cc1 ZINC000217511366 IJ For-Sale Unstable BUB1 43 30 CN(Cc1cccs1)C(=O)c1ccc(O)cc1O ZINC000217511376 CE On-Demand Unstable HSP90AB1 47 39 CN(Cc1cccs1)C(=O)c1ccc(O)cc1O ZINC000217511376 CE On-Demand Unstable HSD17B2 23 42 BrCc1ccccc1N1CC[C@@H](N2CCCCC2)C1 ZINC000217511399 DH For-Sale Unstable L3MBTL3 79 43 O=C(Nc1ccccc1)[C@H]1CCCN(C[C@@H](O)COCc2cccs2)C1 ZINC000217511403 FF On-Demand Unstable SLC6A1 85 39 O=C1OC2(CCN(C(=O)COc3ccccc3)CC2)c2ccccc21 ZINC000217511438 EF In-Stock Unstable CPT1A 99 38 O=C1OC2(CCN(C(=O)COc3ccccc3)CC2)c2ccccc21 ZINC000217511438 EF In-Stock Unstable CPT2 48 37 O=C1OC2(CCN(C(=O)COc3ccccc3)CC2)c2ccccc21 ZINC000217511438 EF In-Stock Unstable NPY5R 57 54 CCCCN(CCC)C(=O)NCCc1ccc(OC)cc1 ZINC000217511469 CG For-Sale Unstable INHA 52 36 CCCCN(CCC)C(=O)NCCc1ccc(OC)cc1 ZINC000217511469 CG For-Sale Unstable BMP1 20 40 CCCCN(CCC)C(=O)NCCc1ccc(OC)cc1 ZINC000217511469 CG For-Sale Unstable MTNR1A 73 41 CCCCN(CCC)C(=O)NCCc1ccc(OC)cc1 ZINC000217511469 CG For-Sale Unstable MTNR1B 57 41 CCCCN(CCC)C(=O)NCCc1ccc(OC)cc1 ZINC000217511469 CG For-Sale Unstable CA9 15 45 CCCCN(CCC)C(=O)NCCc1ccc(OC)cc1 ZINC000217511469 CG For-Sale Unstable PLM2_PLAFA 43 41 BrCc1ccccc1N1CC[C@H](N2CCCCC2)C1 ZINC000217511482 DH For-Sale Unstable L3MBTL3 79 43 CC1(C)[C@@H]2C[C@@H]1CC=C2COC[C@@H](O)CN1CCC[C@@H](C(=O)Nc2ccccc2)C1 ZINC000217511491 HH On-Demand Unstable SLC6A1 50 36 CC1(C)[C@@H]2C[C@@H]1CC=C2COC[C@@H](O)CN1CCC[C@@H](C(=O)Nc2ccccc2)C1 ZINC000217511491 HH On-Demand Unstable CXCR3 30 42 Cc1cccc(=O)n1CCCNC(=O)c1cnc2ccccc2c1 ZINC000217511503 DF In-Stock Unstable HTR1A 18 43 Cc1cccc(=O)n1CCCNC(=O)c1cnc2ccccc2c1 ZINC000217511503 DF In-Stock Unstable HTR2A 33 43 Cc1cccc(=O)n1CCCNC(=O)c1cnc2ccccc2c1 ZINC000217511503 DF In-Stock Unstable HTR2C 34 46 Cc1cccc(=O)n1CCCNC(=O)c1cnc2ccccc2c1 ZINC000217511503 DF In-Stock Unstable DRD3 42 43 Cc1cccc(=O)n1CCCNC(=O)c1cnc2ccccc2c1 ZINC000217511503 DF In-Stock Unstable PLD2 32 46 COc1ccccc1C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217511558 EF In-Stock Unstable AVPR1A 16 54 COc1ccccc1C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217511558 EF In-Stock Unstable KCNA3 19 40 COc1ccccc1C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217511558 EF In-Stock Unstable NPY5R 42 60 COc1ccccc1C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217511558 EF In-Stock Unstable CCR8 24 41 CN(Cc1cccs1)C(=O)c1cc(I)ccc1O ZINC000217511577 FG On-Demand Unstable HSP90AB1 43 35 BrCc1ccc(N2CC[C@@H](N3CCCCC3)C2)nc1 ZINC000217511583 DG For-Sale Unstable HRH3 29 42 BrCc1ccc(N2CC[C@@H](N3CCCCC3)C2)nc1 ZINC000217511583 DG For-Sale Unstable L3MBTL3 71 42 CCCCCNC(=O)NCCc1ccc(OC)cc1 ZINC000217511591 CF On-Demand Unstable CNR1 0 63 CCCCCNC(=O)NCCc1ccc(OC)cc1 ZINC000217511591 CF On-Demand Unstable TRPV1 0 48 CCCCCNC(=O)NCCc1ccc(OC)cc1 ZINC000217511591 CF On-Demand Unstable SLC2A1 25 40 CCCCCNC(=O)NCCc1ccc(OC)cc1 ZINC000217511591 CF On-Demand Unstable EPHX2 43 40 CCCCCNC(=O)NCCc1ccc(OC)cc1 ZINC000217511591 CF On-Demand Unstable PTGDR 34 40 CCCCCNC(=O)NCCc1ccc(OC)cc1 ZINC000217511591 CF On-Demand Unstable PLM2_PLAFA 55 37 CCCCCNC(=O)NCCc1ccc(OC)cc1 ZINC000217511591 CF On-Demand Unstable HT1 23 40 CCCCCNC(=O)NCCc1ccc(OC)cc1 ZINC000217511591 CF On-Demand Unstable LMGT2 25 40 COc1cc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)cc(OC)c1OC ZINC000217511604 JH For-Sale Unstable PTK2 36 40 COc1cc(NC(=O)NCCn2nc(-c3ccccn3)c3c2CCCC3)cc(OC)c1OC ZINC000217511604 JH For-Sale Unstable TGFBR1 19 43 Cc1cc(Nc2ccc(N)cc2)nc(N2CCOCC2)n1 ZINC000217511662 CD In-Stock Unstable PIK3CA 29 51 Cc1cc(Nc2ccc(N)cc2)nc(N2CCOCC2)n1 ZINC000217511662 CD In-Stock Unstable MTOR 0 41 Cc1cc(Nc2ccc(N)cc2)nc(N2CCOCC2)n1 ZINC000217511662 CD In-Stock Unstable PIK3CB 22 43 Cc1cc(Nc2ccc(N)cc2)nc(N2CCOCC2)n1 ZINC000217511662 CD In-Stock Unstable EPHB4 40 33 Cc1cc(Nc2ccc(N)cc2)nc(N2CCOCC2)n1 ZINC000217511662 CD In-Stock Unstable STAT6 47 32 COc1cccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217511663 EF For-Sale Unstable DRD4 46 36 COc1cccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217511663 EF For-Sale Unstable AVPR1A 15 49 COc1cccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217511663 EF For-Sale Unstable NPY5R 47 61 BrCc1ccc(N2CC[C@H](N3CCCCC3)C2)nc1 ZINC000217511667 DG For-Sale Unstable HRH3 29 42 BrCc1ccc(N2CC[C@H](N3CCCCC3)C2)nc1 ZINC000217511667 DG For-Sale Unstable L3MBTL3 71 42 COc1ccc(NC[C@@](C)(O)CSC)c([N+](=O)[O-])c1 ZINC000217511685 CE For-Sale Unstable TAAR1 20 44 COc1ccc(NC[C@@](C)(O)CSC)c([N+](=O)[O-])c1 ZINC000217511685 CE For-Sale Unstable AKR1C2 24 49 COc1ccc(CCNC(=O)Nc2ccc(CC(=O)O)cc2)cc1 ZINC000217511709 EF For-Sale Unstable ADRB1 29 47 COc1ccc(CCNC(=O)Nc2ccc(CC(=O)O)cc2)cc1 ZINC000217511709 EF For-Sale Unstable ADRB3 39 42 COc1ccc(CCNC(=O)Nc2ccc(CC(=O)O)cc2)cc1 ZINC000217511709 EF For-Sale Unstable BMP1 24 43 COc1ccc(CCNC(=O)Nc2ccc(CC(=O)O)cc2)cc1 ZINC000217511709 EF For-Sale Unstable CA1 42 54 COc1ccc(CCNC(=O)Nc2ccc(CC(=O)O)cc2)cc1 ZINC000217511709 EF For-Sale Unstable PDE4B 0 41 COc1ccc(CCNC(=O)Nc2ccc(CC(=O)O)cc2)cc1 ZINC000217511709 EF For-Sale Unstable PDE4D 0 41 COc1ccc(CCNC(=O)Nc2ccc(CC(=O)O)cc2)cc1 ZINC000217511709 EF For-Sale Unstable RAF1 41 41 COc1ccc(CCNC(=O)Nc2ccc(CC(=O)O)cc2)cc1 ZINC000217511709 EF For-Sale Unstable MTNR1A 66 42 COc1ccc(CCNC(=O)Nc2ccc(CC(=O)O)cc2)cc1 ZINC000217511709 EF For-Sale Unstable MTNR1B 53 38 COc1ccc(CCNC(=O)Nc2ccc(CC(=O)O)cc2)cc1 ZINC000217511709 EF For-Sale Unstable CA12 28 54 COc1ccc(CCNC(=O)Nc2ccc(CC(=O)O)cc2)cc1 ZINC000217511709 EF For-Sale Unstable PTGDR 0 44 COc1ccc(CCNC(=O)Nc2ccc(CC(=O)O)cc2)cc1 ZINC000217511709 EF For-Sale Unstable CA9 32 52 COc1ccc(CCNC(=O)Nc2ccc(CC(=O)O)cc2)cc1 ZINC000217511709 EF For-Sale Unstable Q8MMZ8_EIMTE 32 41 COc1ccc(CCNC(=O)Nc2ccc(CC(=O)O)cc2)cc1 ZINC000217511709 EF For-Sale Unstable NCE103 43 54 Cc1ccc(CN(C)C(=O)c2cc(Br)ccc2I)cc1 ZINC000217511723 IJ For-Sale Unstable HSP90AB1 20 43 Nc1nccc(C2CCN(C(=O)CCCN3Cc4ccccc4C3)CC2)n1 ZINC000217511759 FF In-Stock Unstable HTR7 23 40 Nc1nccc(C2CCN(C(=O)CCCN3Cc4ccccc4C3)CC2)n1 ZINC000217511759 FF In-Stock Unstable ETHR 57 35 CCNc1cc(Nc2ccc(N)cc2)nc(C)n1 ZINC000217511763 BF In-Stock Unstable AGPAT2 61 38 COc1nn(C)cc1C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217511765 ED For-Sale Unstable AVPR1A 22 52 COc1nn(C)cc1C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217511765 ED For-Sale Unstable NPY5R 42 50 COc1ccc(NC[C@](C)(O)CSC)c([N+](=O)[O-])c1 ZINC000217511768 CE For-Sale Unstable TAAR1 20 44 COc1ccc(NC[C@](C)(O)CSC)c([N+](=O)[O-])c1 ZINC000217511768 CE For-Sale Unstable AKR1C2 24 49 O=C(NCCn1nc(-c2ccccn2)c2c1CCCC2)NC1CCCCCC1 ZINC000217511833 GH For-Sale Unstable EPHX2 18 44 COc1ccc(CCNC(=O)NCc2ccc(C(=O)O)cc2)cc1 ZINC000217511840 EE On-Demand Unstable CA2 15 47 COc1ccc(CCNC(=O)NCc2ccc(C(=O)O)cc2)cc1 ZINC000217511840 EE On-Demand Unstable BMP1 28 40 COc1ccc(CCNC(=O)NCc2ccc(C(=O)O)cc2)cc1 ZINC000217511840 EE On-Demand Unstable CA1 18 47 COc1ccc(CCNC(=O)NCc2ccc(C(=O)O)cc2)cc1 ZINC000217511840 EE On-Demand Unstable KCNA5 16 42 COc1ccc(CCNC(=O)NCc2ccc(C(=O)O)cc2)cc1 ZINC000217511840 EE On-Demand Unstable TRPV1 0 46 COc1ccc(CCNC(=O)NCc2ccc(C(=O)O)cc2)cc1 ZINC000217511840 EE On-Demand Unstable MMP13 35 51 COc1ccc(CCNC(=O)NCc2ccc(C(=O)O)cc2)cc1 ZINC000217511840 EE On-Demand Unstable CTSL 18 43 COc1ccc(CCNC(=O)NCc2ccc(C(=O)O)cc2)cc1 ZINC000217511840 EE On-Demand Unstable MTNR1A 76 43 COc1ccc(CCNC(=O)NCc2ccc(C(=O)O)cc2)cc1 ZINC000217511840 EE On-Demand Unstable MTNR1B 61 39 COc1ccc(CCNC(=O)NCc2ccc(C(=O)O)cc2)cc1 ZINC000217511840 EE On-Demand Unstable PTGDR 27 41 COc1ccc(CCNC(=O)NCc2ccc(C(=O)O)cc2)cc1 ZINC000217511840 EE On-Demand Unstable CA9 24 47 COc1ccc(CCNC(=O)NCc2ccc(C(=O)O)cc2)cc1 ZINC000217511840 EE On-Demand Unstable MMP1 22 40 COc1ccc(CCNC(=O)NCc2ccc(C(=O)O)cc2)cc1 ZINC000217511840 EE On-Demand Unstable PROKR1 59 34 Cc1cc(C)cc(OC[C@@H](O)CN2CCC[C@@H](C(=O)Nc3ccccc3)C2)c1 ZINC000217511866 GG On-Demand Unstable ADRB1 40 38 Cc1cc(C)cc(OC[C@@H](O)CN2CCC[C@@H](C(=O)Nc3ccccc3)C2)c1 ZINC000217511866 GG On-Demand Unstable SLC6A1 141 38 Cc1cc(C)cc(OC[C@@H](O)CN2CCC[C@@H](C(=O)Nc3ccccc3)C2)c1 ZINC000217511866 GG On-Demand Unstable ACOX1 58 41 Cc1cc(C)cc(OC[C@@H](O)CN2CCC[C@@H](C(=O)Nc3ccccc3)C2)c1 ZINC000217511866 GG On-Demand Unstable CCR3 22 45 Cc1cc(C)cc(OC[C@@H](O)CN2CCC[C@@H](C(=O)Nc3ccccc3)C2)c1 ZINC000217511866 GG On-Demand Unstable ABCB1 73 42 Cc1cc(C)cc(OC[C@@H](O)CN2CCC[C@@H](C(=O)Nc3ccccc3)C2)c1 ZINC000217511866 GG On-Demand Unstable EPHX2 29 41 Cc1cc(C)cc(OC[C@@H](O)CN2CCC[C@@H](C(=O)Nc3ccccc3)C2)c1 ZINC000217511866 GG On-Demand Unstable ALK 15 41 Cc1nc(NCCN)cc(N2CCCCC2)n1 ZINC000217511874 BD In-Stock Unstable GALR2 44 37 C[C@H](O)c1ccccc1NC(=O)/C=C\c1cnn(C)c1 ZINC000217511875 CE For-Sale Unstable MMP2 18 44 C[C@H](O)c1ccccc1NC(=O)/C=C\c1cnn(C)c1 ZINC000217511875 CE For-Sale Unstable MMP9 15 44 O=C1OC2(CCN(C(=O)CCC3CCCCC3)CC2)c2ccccc21 ZINC000217511888 EI For-Sale Unstable NPY5R 51 45 Cc1ccc(CN(C)C(=O)c2cc(I)ccc2O)cc1 ZINC000217511922 GH On-Demand Unstable HSP90AB1 49 48 CN1[C@H](c2ccccc2)[C@@H]2CCC[C@@H]([C@H]2O)[C@@H]1c1ccccc1 ZINC000217511936 DI In-Stock Unstable SLC18A3 23 40 Cc1cc(C)cc(OC[C@H](O)CN2CCC[C@@H](C(=O)Nc3ccccc3)C2)c1 ZINC000217511944 GG On-Demand Unstable ADRB1 40 38 Cc1cc(C)cc(OC[C@H](O)CN2CCC[C@@H](C(=O)Nc3ccccc3)C2)c1 ZINC000217511944 GG On-Demand Unstable SLC6A1 141 38 Cc1cc(C)cc(OC[C@H](O)CN2CCC[C@@H](C(=O)Nc3ccccc3)C2)c1 ZINC000217511944 GG On-Demand Unstable ACOX1 58 41 Cc1cc(C)cc(OC[C@H](O)CN2CCC[C@@H](C(=O)Nc3ccccc3)C2)c1 ZINC000217511944 GG On-Demand Unstable CCR3 22 45 Cc1cc(C)cc(OC[C@H](O)CN2CCC[C@@H](C(=O)Nc3ccccc3)C2)c1 ZINC000217511944 GG On-Demand Unstable ABCB1 73 42 Cc1cc(C)cc(OC[C@H](O)CN2CCC[C@@H](C(=O)Nc3ccccc3)C2)c1 ZINC000217511944 GG On-Demand Unstable EPHX2 29 41 Cc1cc(C)cc(OC[C@H](O)CN2CCC[C@@H](C(=O)Nc3ccccc3)C2)c1 ZINC000217511944 GG On-Demand Unstable ALK 15 41 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1cnn(C)c1 ZINC000217511948 CE For-Sale Unstable MMP2 18 44 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1cnn(C)c1 ZINC000217511948 CE For-Sale Unstable MMP9 15 44 COc1ccc(CCNC(=O)N2C(C)(C)CC(N)CC2(C)C)cc1 ZINC000217511961 EF For-Sale Unstable MTNR1A 46 35 COc1ccc(CCNC(=O)N2C(C)(C)CC(N)CC2(C)C)cc1 ZINC000217511961 EF For-Sale Unstable PROKR1 54 34 NCCNc1cc(N2CCCC2)ncn1 ZINC000217511983 BC In-Stock Unstable HRH4 18 56 O=C1OC2(CCN(C(=O)c3ccc(Cl)cc3)CC2)c2ccccc21 ZINC000217512004 EH For-Sale Unstable AVPR1A 25 63 O=C1OC2(CCN(C(=O)c3ccc(Cl)cc3)CC2)c2ccccc21 ZINC000217512004 EH For-Sale Unstable NPY5R 47 60 O=C1OC2(CCN(C(=O)c3ccc(Cl)cc3)CC2)c2ccccc21 ZINC000217512004 EH For-Sale Unstable CCR8 18 42 CC(C)OCCCNS(=O)(=O)c1cc(C(=O)O)ccc1N[C@@H](C)c1ccccc1 ZINC000217512025 HH In-Stock Unstable PLA2G4A 40 33 N#Cc1cccc(C#N)c1-c1ccccn1 ZINC000217512033 BE For-Sale Mild METAP1 19 52 N#Cc1cccc(C#N)c1-c1ccccn1 ZINC000217512033 BE For-Sale Mild GRM5 20 45 Cc1ccc(/C=C\C(=O)Nc2ccccc2[C@@H](C)O)s1 ZINC000217512039 CH For-Sale Unstable UL26 24 42 Cc1ccc(/C=C\C(=O)Nc2ccccc2[C@@H](C)O)s1 ZINC000217512039 CH For-Sale Unstable SCAF_EBVB9 37 42 COc1ccc(CCNC(=O)Nc2cc(C)ccc2O)cc1 ZINC000217512065 DG For-Sale Unstable THRA 28 48 COc1ccc(CCNC(=O)Nc2cc(C)ccc2O)cc1 ZINC000217512065 DG For-Sale Unstable ADRB3 26 44 COc1ccc(CCNC(=O)Nc2cc(C)ccc2O)cc1 ZINC000217512065 DG For-Sale Unstable THRB 32 48 COc1ccc(CCNC(=O)Nc2cc(C)ccc2O)cc1 ZINC000217512065 DG For-Sale Unstable BMP1 24 40 COc1ccc(CCNC(=O)Nc2cc(C)ccc2O)cc1 ZINC000217512065 DG For-Sale Unstable CA1 18 46 COc1ccc(CCNC(=O)Nc2cc(C)ccc2O)cc1 ZINC000217512065 DG For-Sale Unstable TRPV1 25 53 COc1ccc(CCNC(=O)Nc2cc(C)ccc2O)cc1 ZINC000217512065 DG For-Sale Unstable RAF1 42 44 COc1ccc(CCNC(=O)Nc2cc(C)ccc2O)cc1 ZINC000217512065 DG For-Sale Unstable MTNR1A 76 43 COc1ccc(CCNC(=O)Nc2cc(C)ccc2O)cc1 ZINC000217512065 DG For-Sale Unstable MTNR1B 56 43 COc1ccc(CCNC(=O)Nc2cc(C)ccc2O)cc1 ZINC000217512065 DG For-Sale Unstable CA12 16 46 COc1ccc(CCNC(=O)Nc2cc(C)ccc2O)cc1 ZINC000217512065 DG For-Sale Unstable PTGDR 20 41 COc1ccc(CCNC(=O)Nc2cc(C)ccc2O)cc1 ZINC000217512065 DG For-Sale Unstable CA9 22 46 COc1ccc(CCNC(=O)Nc2cc(C)ccc2O)cc1 ZINC000217512065 DG For-Sale Unstable Q8MMZ8_EIMTE 37 41 COc1ccc(CCNC(=O)Nc2cc(C)ccc2O)cc1 ZINC000217512065 DG For-Sale Unstable NCE103 32 42 COc1ccc(CCNC(=O)Nc2cc(C)ccc2O)cc1 ZINC000217512065 DG For-Sale Unstable CAN2 0 42 COc1ccc(CCNC(=O)Nc2cc(C)ccc2O)cc1 ZINC000217512065 DG For-Sale Unstable PQSD 0 41 NCCNc1cc(N2CCCCC2)ncn1 ZINC000217512097 BC In-Stock Unstable HRH4 17 55 Cc1cccc(NC23CC4CC(CC(C4)C2)C3)c1 ZINC000217512103 BI For-Sale Unstable EPHX2 29 63 CC(C)OCCCNS(=O)(=O)c1cc(C(=O)O)ccc1N[C@H](C)c1ccccc1 ZINC000217512114 HH In-Stock Unstable PLA2G4A 40 33 CCCc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217512116 EH For-Sale Unstable AGTR1B 27 41 CCCc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217512116 EH For-Sale Unstable NPY5R 37 48 Cc1ccc(/C=C\C(=O)Nc2ccccc2[C@H](C)O)s1 ZINC000217512123 CH For-Sale Unstable UL26 24 42 Cc1ccc(/C=C\C(=O)Nc2ccccc2[C@H](C)O)s1 ZINC000217512123 CH For-Sale Unstable SCAF_EBVB9 37 42 CC[C@@H]1CC[C@H](O)[C@H](c2ccccc2)C1 ZINC000217512143 BG For-Sale Unstable SLC18A3 20 40 COc1ccc(CCNC(=O)N2CCN(CCO)CC2)cc1 ZINC000217512177 DC For-Sale Unstable HTR1A 29 40 COc1ccc(CCNC(=O)N2CCN(CCO)CC2)cc1 ZINC000217512177 DC For-Sale Unstable DRD4 46 35 COc1ccc(CCNC(=O)N2CCN(CCO)CC2)cc1 ZINC000217512177 DC For-Sale Unstable HTR2A 18 52 COc1ccc(CCNC(=O)N2CCN(CCO)CC2)cc1 ZINC000217512177 DC For-Sale Unstable DRD3 42 39 COc1ccc(CCNC(=O)N2CCN(CCO)CC2)cc1 ZINC000217512177 DC For-Sale Unstable SIGMAR1 23 57 COc1ccc(CCNC(=O)N2CCN(CCO)CC2)cc1 ZINC000217512177 DC For-Sale Unstable MMP13 30 46 COc1ccc(CCNC(=O)N2CCN(CCO)CC2)cc1 ZINC000217512177 DC For-Sale Unstable MTNR1A 55 38 COc1ccc(CCNC(=O)N2CCN(CCO)CC2)cc1 ZINC000217512177 DC For-Sale Unstable MTNR1B 49 39 COc1ccc(CCNC(=O)N2CCN(CCO)CC2)cc1 ZINC000217512177 DC For-Sale Unstable MMP3 24 49 COc1ccc(CCNC(=O)N2CCN(CCO)CC2)cc1 ZINC000217512177 DC For-Sale Unstable FAAH 15 50 COc1ccc(CCNC(=O)N2CCN(CCO)CC2)cc1 ZINC000217512177 DC For-Sale Unstable MMP9 31 49 COc1ccc(CCNC(=O)N2CCN(CCO)CC2)cc1 ZINC000217512177 DC For-Sale Unstable MMP7 29 49 COc1ccc(CCNC(=O)N2CCN(CCO)CC2)cc1 ZINC000217512177 DC For-Sale Unstable MMP1 31 49 BrCc1cnc(N2CC[C@@H](N3CCCCC3)C2)nc1 ZINC000217512192 EE For-Sale Unstable HRH3 28 40 BrCc1cnc(N2CC[C@@H](N3CCCCC3)C2)nc1 ZINC000217512192 EE For-Sale Unstable L3MBTL3 57 40 NCCNc1cc(N2CCOCC2)ncn1 ZINC000217512225 BB In-Stock Unstable SMG1 40 33 Cc1cc(C)c(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c(C)c1 ZINC000217512233 EH For-Sale Unstable AVPR1A 15 52 Cc1cc(C)c(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c(C)c1 ZINC000217512233 EH For-Sale Unstable NPY5R 43 48 Brc1ccc(Br)c(-c2ccccn2)c1 ZINC000217512247 DI For-Sale Anodyne METAP2 41 39 Cc1cc(S(=O)(=O)NC[C@](C)(O)c2cc3ccccc3s2)ccc1F ZINC000217512254 GH In-Stock Unstable LEF 63 40 BrCc1cnc(N2CC[C@H](N3CCCCC3)C2)nc1 ZINC000217512274 EE For-Sale Unstable HRH3 28 40 BrCc1cnc(N2CC[C@H](N3CCCCC3)C2)nc1 ZINC000217512274 EE For-Sale Unstable L3MBTL3 57 40 COC(=O)c1ccc(C(=O)OC)c(NC(=O)NCCc2ccc(OC)cc2)c1 ZINC000217512309 GF For-Sale Unstable MTNR1A 68 41 COC(=O)c1ccc(C(=O)OC)c(NC(=O)NCCc2ccc(OC)cc2)c1 ZINC000217512309 GF For-Sale Unstable MTNR1B 52 39 COC(=O)c1ccc(C(=O)OC)c(NC(=O)NCCc2ccc(OC)cc2)c1 ZINC000217512309 GF For-Sale Unstable PTGDR 23 42 COC(=O)c1ccc(C(=O)OC)c(NC(=O)NCCc2ccc(OC)cc2)c1 ZINC000217512309 GF For-Sale Unstable CA9 15 42 CC[C@@H]1CC[C@@H](O)[C@H](c2ccccc2)C1 ZINC000217512311 BG For-Sale Unstable SLC18A3 20 40 CN1CCN(c2cc(N3CCNCC3)ncn2)CC1 ZINC000217512325 CB In-Stock Unstable ADRA2A 15 44 CN1CCN(c2cc(N3CCNCC3)ncn2)CC1 ZINC000217512325 CB In-Stock Unstable HRH4 47 60 COc1ccc(CCNc2ccc(C(=O)O)cc2S(=O)(=O)NCCCOC(C)C)cc1 ZINC000217512332 JG In-Stock Unstable AKR1C3 20 43 CN(C)c1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217512345 FG For-Sale Unstable NPY5R 40 49 Cc1cc(S(=O)(=O)NC[C@@](C)(O)c2cc3ccccc3s2)ccc1F ZINC000217512353 GH In-Stock Unstable LEF 63 40 CCCCN(CCCC)C(=O)NCCc1ccc(OC)cc1 ZINC000217512419 DH On-Demand Unstable INHA 67 37 CCCCN(CCCC)C(=O)NCCc1ccc(OC)cc1 ZINC000217512419 DH On-Demand Unstable BMP1 25 42 CCCCN(CCCC)C(=O)NCCc1ccc(OC)cc1 ZINC000217512419 DH On-Demand Unstable SCN2A 24 40 CCCCN(CCCC)C(=O)NCCc1ccc(OC)cc1 ZINC000217512419 DH On-Demand Unstable MTNR1A 88 42 CCCCN(CCCC)C(=O)NCCc1ccc(OC)cc1 ZINC000217512419 DH On-Demand Unstable MTNR1B 70 42 CCCCN(CCCC)C(=O)NCCc1ccc(OC)cc1 ZINC000217512419 DH On-Demand Unstable MMP3 18 40 CCCCN(CCCC)C(=O)NCCc1ccc(OC)cc1 ZINC000217512419 DH On-Demand Unstable S1PR2 42 37 CCCCN(CCCC)C(=O)NCCc1ccc(OC)cc1 ZINC000217512419 DH On-Demand Unstable MMP9 15 42 CCCCN(CCCC)C(=O)NCCc1ccc(OC)cc1 ZINC000217512419 DH On-Demand Unstable CA9 21 47 CCCCN(CCCC)C(=O)NCCc1ccc(OC)cc1 ZINC000217512419 DH On-Demand Unstable MMP1 16 42 CCCCN(CCCC)C(=O)NCCc1ccc(OC)cc1 ZINC000217512419 DH On-Demand Unstable PLM2_PLAFA 45 42 Nc1ccc(Nc2cc(N3CCCC3)ncn2)cc1 ZINC000217512427 CE In-Stock Unstable GALR2 50 40 COc1ccc(CCNc2ccc(C(=O)O)cc2S(=O)(=O)NCCCOC(C)C)cc1OC ZINC000217512438 JG In-Stock Unstable PTGDR 19 42 COc1ccc(CCNc2ccc(C(=O)O)cc2S(=O)(=O)NCCCOC(C)C)cc1OC ZINC000217512438 JG In-Stock Unstable IAP 0 41 COc1ccc(CCNc2ccc(C(=O)O)cc2S(=O)(=O)NCCCOC(C)C)cc1OC ZINC000217512438 JG In-Stock Unstable SCMU_MYCTU 0 47 CN(C)c1cccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217512452 FG For-Sale Unstable AVPR1A 15 49 CN(C)c1cccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217512452 FG For-Sale Unstable ACACA 52 36 CN(C)c1cccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217512452 FG For-Sale Unstable NPY5R 37 47 CC(=O)N/N=C1\C(=O)N(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)c2ccccc21 ZINC000217512504 HD In-Stock Unstable CHRNA4 31 52 COc1ccc(CCNC(=O)N(c2ccccc2)c2ccc(N)cc2)cc1 ZINC000217512557 FI For-Sale Unstable BMP1 29 45 COc1ccc(CCNC(=O)N(c2ccccc2)c2ccc(N)cc2)cc1 ZINC000217512557 FI For-Sale Unstable MMP16 0 43 COc1ccc(CCNC(=O)N(c2ccccc2)c2ccc(N)cc2)cc1 ZINC000217512557 FI For-Sale Unstable MTNR1A 72 39 COc1ccc(CCNC(=O)N(c2ccccc2)c2ccc(N)cc2)cc1 ZINC000217512557 FI For-Sale Unstable MTNR1B 62 37 COc1ccc(CCNC(=O)N(c2ccccc2)c2ccc(N)cc2)cc1 ZINC000217512557 FI For-Sale Unstable MMP9 15 43 COc1ccc(CCNC(=O)N(c2ccccc2)c2ccc(N)cc2)cc1 ZINC000217512557 FI For-Sale Unstable CA9 21 45 COc1ccc(CCNC(=O)N(c2ccccc2)c2ccc(N)cc2)cc1 ZINC000217512557 FI For-Sale Unstable MMP1 15 43 O=C1OC2(CCN(C(=O)c3ccc4c(c3)OCO4)CC2)c2ccccc21 ZINC000217512558 FF For-Sale Unstable AVPR1A 18 50 O=C1OC2(CCN(C(=O)c3ccc4c(c3)OCO4)CC2)c2ccccc21 ZINC000217512558 FF For-Sale Unstable NPY5R 38 52 Nc1ccc(Nc2cc(N3CCOCC3)ncn2)cc1 ZINC000217512648 CD In-Stock Unstable MAPKAPK5 45 34 Nc1ccc(Nc2cc(N3CCOCC3)ncn2)cc1 ZINC000217512648 CD In-Stock Unstable MAPK10 23 44 Nc1ccc(Nc2cc(N3CCOCC3)ncn2)cc1 ZINC000217512648 CD In-Stock Unstable TNIK 33 41 Nc1ccc(Nc2cc(N3CCOCC3)ncn2)cc1 ZINC000217512648 CD In-Stock Unstable SMG1 48 41 Cc1oc2cc(OCCN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)ccc2c(=O)c1-c1ccccc1 ZINC000217512654 JI In-Stock Unstable CHRNA4 37 48 COc1ccc(CC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217512666 FF For-Sale Unstable SIGMAR1 21 50 COc1ccc(CC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217512666 FF For-Sale Unstable NPY5R 37 51 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable CA2 24 59 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable EPHX1 0 40 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable ADRB2 27 46 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable ADRB1 49 47 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable TSHR 41 32 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable ADRB3 56 46 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable LTA4H 42 37 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable BMP1 34 43 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable NQO2 37 40 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable CA1 57 59 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable CCR3 28 42 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable SCN2A 24 41 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable HDAC8 19 47 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable RAF1 44 41 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable KDR 15 45 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable MTNR1A 96 46 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable MTNR1B 88 46 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable MMP2 25 44 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable MMP3 36 43 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable ROCK2 20 57 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable FAAH 20 46 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable NPY5R 25 45 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable MMP9 22 44 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable EPHX2 23 41 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable CA12 33 59 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable PTGDR 24 48 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable CA9 37 59 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable FPR1 18 40 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable Q8MMZ8_EIMTE 38 41 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable AKR1C3 29 48 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable NCE103 43 59 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable ABCG2 17 43 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable AKR1C2 58 46 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable ACAT 0 54 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable NAMPT 18 42 COc1ccc(CCNC(=O)Nc2ccc(Nc3ccccc3)cc2)cc1 ZINC000217512677 FJ For-Sale Unstable P95276_MYCTO 0 40 Nc1ccc(Nc2cc(N3CCCCC3)ncn2)cc1 ZINC000217512755 CF In-Stock Unstable GALR2 52 42 O=C([C@H](O)c1ccccc1)N1CCCN(C2CCCCC2)CC1 ZINC000217512760 DF In-Stock Unstable HRH3 26 46 O=C([C@H](O)c1ccccc1)N1CCCN(C2CCCCC2)CC1 ZINC000217512760 DF In-Stock Unstable CCR3 29 42 O=C([C@H](O)c1ccccc1)N1CCCN(C2CCCCC2)CC1 ZINC000217512760 DF In-Stock Unstable NMUR2 0 50 O=C([C@H](O)c1ccccc1)N1CCCN(C2CCCCC2)CC1 ZINC000217512760 DF In-Stock Unstable NMUR1 0 50 O=C([C@H](O)c1ccccc1)N1CCCN(C2CCCCC2)CC1 ZINC000217512760 DF In-Stock Unstable L3MBTL1 0 47 O=C([C@H](O)c1ccccc1)N1CCCN(C2CCCCC2)CC1 ZINC000217512760 DF In-Stock Unstable L3MBTL3 77 43 O=C([C@H](O)c1ccccc1)N1CCCN(C2CCCCC2)CC1 ZINC000217512760 DF In-Stock Unstable MBTD1 0 40 O=C([C@H](O)c1ccccc1)N1CCCN(C2CCCCC2)CC1 ZINC000217512760 DF In-Stock Unstable TP53BP1 0 43 Cc1ccc(/C=C\C(=O)Nc2ccccc2[C@@H](C)O)cc1 ZINC000217512763 CH For-Sale Unstable LTB4R 0 51 Cc1ccc(/C=C\C(=O)Nc2ccccc2[C@@H](C)O)cc1 ZINC000217512763 CH For-Sale Unstable HDAC8 19 40 Cc1ccc(/C=C\C(=O)Nc2ccccc2[C@@H](C)O)cc1 ZINC000217512763 CH For-Sale Unstable MMP2 23 56 Cc1ccc(/C=C\C(=O)Nc2ccccc2[C@@H](C)O)cc1 ZINC000217512763 CH For-Sale Unstable HDAC1 28 51 Cc1ccc(/C=C\C(=O)Nc2ccccc2[C@@H](C)O)cc1 ZINC000217512763 CH For-Sale Unstable HDAC6 15 40 Cc1ccc(/C=C\C(=O)Nc2ccccc2[C@@H](C)O)cc1 ZINC000217512763 CH For-Sale Unstable MMP9 22 56 Cc1ccc(/C=C\C(=O)Nc2ccccc2[C@@H](C)O)cc1 ZINC000217512763 CH For-Sale Unstable MMP1 26 56 Cc1ccc(/C=C\C(=O)Nc2ccccc2[C@@H](C)O)cc1 ZINC000217512763 CH For-Sale Unstable TRPM8 0 50 BrCc1ccc(N2CC[C@@H](N3CCCCC3)C2)cc1 ZINC000217512769 DH For-Sale Unstable L3MBTL1 0 44 BrCc1ccc(N2CC[C@@H](N3CCCCC3)C2)cc1 ZINC000217512769 DH For-Sale Unstable L3MBTL3 107 59 BrCc1ccc(N2CC[C@@H](N3CCCCC3)C2)cc1 ZINC000217512769 DH For-Sale Unstable L3MBTL4 0 44 BrCc1ccc(N2CC[C@@H](N3CCCCC3)C2)cc1 ZINC000217512769 DH For-Sale Unstable MBTD1 0 44 BrCc1ccc(N2CC[C@@H](N3CCCCC3)C2)cc1 ZINC000217512769 DH For-Sale Unstable TP53BP1 0 44 CCOc1ccccc1C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217512775 FG For-Sale Unstable AVPR1A 20 54 CCOc1ccccc1C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217512775 FG For-Sale Unstable NPY5R 43 52 CCOc1ccccc1C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217512775 FG For-Sale Unstable HCN1 79 42 CCOc1ccccc1C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217512775 FG For-Sale Unstable HCN4 60 40 COc1ccc(CCNC(=O)NC(C)(C)CC(C)(C)C)cc1 ZINC000217512782 DH For-Sale Unstable CTSL 20 45 COc1ccc(CCNC(=O)NC(C)(C)CC(C)(C)C)cc1 ZINC000217512782 DH For-Sale Unstable MTNR1A 78 41 COc1ccc(CCNC(=O)NC(C)(C)CC(C)(C)C)cc1 ZINC000217512782 DH For-Sale Unstable MTNR1B 67 39 COc1ccc(CCNC(=O)NC(C)(C)CC(C)(C)C)cc1 ZINC000217512782 DH For-Sale Unstable PTGDR 24 40 COc1ccc(CCNC(=O)NC(C)(C)CC(C)(C)C)cc1 ZINC000217512782 DH For-Sale Unstable CA9 19 47 COc1ccc(CCNC(=O)NC(C)(C)CC(C)(C)C)cc1 ZINC000217512782 DH For-Sale Unstable PROKR1 60 34 Cc1ccc(/C=C\C(=O)Nc2ccccc2[C@H](C)O)cc1 ZINC000217512847 CH For-Sale Unstable LTB4R 0 51 Cc1ccc(/C=C\C(=O)Nc2ccccc2[C@H](C)O)cc1 ZINC000217512847 CH For-Sale Unstable HDAC8 19 40 Cc1ccc(/C=C\C(=O)Nc2ccccc2[C@H](C)O)cc1 ZINC000217512847 CH For-Sale Unstable MMP2 23 56 Cc1ccc(/C=C\C(=O)Nc2ccccc2[C@H](C)O)cc1 ZINC000217512847 CH For-Sale Unstable HDAC1 28 51 Cc1ccc(/C=C\C(=O)Nc2ccccc2[C@H](C)O)cc1 ZINC000217512847 CH For-Sale Unstable HDAC6 15 40 Cc1ccc(/C=C\C(=O)Nc2ccccc2[C@H](C)O)cc1 ZINC000217512847 CH For-Sale Unstable MMP9 22 56 Cc1ccc(/C=C\C(=O)Nc2ccccc2[C@H](C)O)cc1 ZINC000217512847 CH For-Sale Unstable MMP1 26 56 Cc1ccc(/C=C\C(=O)Nc2ccccc2[C@H](C)O)cc1 ZINC000217512847 CH For-Sale Unstable TRPM8 0 50 BrCc1ccc(N2CC[C@H](N3CCCCC3)C2)cc1 ZINC000217512853 DH For-Sale Unstable L3MBTL1 0 44 BrCc1ccc(N2CC[C@H](N3CCCCC3)C2)cc1 ZINC000217512853 DH For-Sale Unstable L3MBTL3 107 59 BrCc1ccc(N2CC[C@H](N3CCCCC3)C2)cc1 ZINC000217512853 DH For-Sale Unstable L3MBTL4 0 44 BrCc1ccc(N2CC[C@H](N3CCCCC3)C2)cc1 ZINC000217512853 DH For-Sale Unstable MBTD1 0 44 BrCc1ccc(N2CC[C@H](N3CCCCC3)C2)cc1 ZINC000217512853 DH For-Sale Unstable TP53BP1 0 44 O=C(O)[C@@H]1CS[C@H](c2ccccc2)N1C(=O)c1ccc(Cl)cc1 ZINC000217512862 EH In-Stock Unstable THYX_PBCV1 0 40 O=C(O)[C@@H]1CS[C@H](c2ccccc2)N1C(=O)c1ccc(Cl)cc1 ZINC000217512862 EH In-Stock Unstable FPTA 43 36 CCOc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217512883 FG For-Sale Unstable AVPR1A 20 46 CCOc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217512883 FG For-Sale Unstable NPY5R 43 49 COc1ccc(CCNC(=O)N(C(C)=O)c2cccc(N)c2)cc1 ZINC000217512893 EF For-Sale Unstable NQO2 29 40 COc1ccc(CCNC(=O)N(C(C)=O)c2cccc(N)c2)cc1 ZINC000217512893 EF For-Sale Unstable MTNR1A 78 46 COc1ccc(CCNC(=O)N(C(C)=O)c2cccc(N)c2)cc1 ZINC000217512893 EF For-Sale Unstable MTNR1B 61 38 COc1ccc(CCNC(=O)N(C(C)=O)c2cccc(N)c2)cc1 ZINC000217512893 EF For-Sale Unstable PTGDR 25 40 Clc1ccc(Cl)c(OCCN2CCN(Cc3ccccn3)CC2)c1 ZINC000217512926 FH On-Demand Unstable DRD2 16 44 Clc1ccc(Cl)c(OCCN2CCN(Cc3ccccn3)CC2)c1 ZINC000217512926 FH On-Demand Unstable ERBB2 24 41 Clc1ccc(Cl)c(OCCN2CCN(Cc3ccccn3)CC2)c1 ZINC000217512926 FH On-Demand Unstable HRP1_PLAFA 64 32 Clc1ccc(Cl)c(OCCN2CCN(Cc3ccccn3)CC2)c1 ZINC000217512926 FH On-Demand Unstable HNMT 45 31 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1F ZINC000217512931 CH For-Sale Unstable KCNQ2 55 42 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1F ZINC000217512931 CH For-Sale Unstable MMP1 0 51 O=C(O)[C@H]1CS[C@H](c2ccccc2)N1C(=O)c1ccc(Cl)cc1 ZINC000217512950 EH In-Stock Unstable THYX_PBCV1 0 40 O=C(O)[C@H]1CS[C@H](c2ccccc2)N1C(=O)c1ccc(Cl)cc1 ZINC000217512950 EH In-Stock Unstable FPTA 43 36 C[C@@H](CN1CCC[C@@H](N)C1)C(N)=O ZINC000217512955 AB For-Sale Unstable XPNPEP1 54 32 C[C@@H](CN1CCC[C@@H](N)C1)C(N)=O ZINC000217512955 AB For-Sale Unstable XPNPEP2 54 32 COc1cccc(CC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217512999 FF For-Sale Unstable DRD4 40 31 COc1cccc(CC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217512999 FF For-Sale Unstable SIGMAR1 21 53 COc1cccc(CC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217512999 FF For-Sale Unstable NPY5R 46 58 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1F ZINC000217513019 CH For-Sale Unstable KCNQ2 55 42 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1F ZINC000217513019 CH For-Sale Unstable MMP1 0 51 O=C(O)[C@@H]1CS[C@@H](c2ccccc2)N1C(=O)c1ccc(Cl)cc1 ZINC000217513035 EH In-Stock Unstable THYX_PBCV1 0 40 O=C(O)[C@@H]1CS[C@@H](c2ccccc2)N1C(=O)c1ccc(Cl)cc1 ZINC000217513035 EH In-Stock Unstable FPTA 43 36 C[C@H](CN1CCC[C@@H](N)C1)C(N)=O ZINC000217513039 AB For-Sale Unstable XPNPEP1 54 32 C[C@H](CN1CCC[C@@H](N)C1)C(N)=O ZINC000217513039 AB For-Sale Unstable XPNPEP2 54 32 C[C@H](c1cccc(F)c1)N1CCC[C@@H](CN)C1 ZINC000217513093 BF On-Demand Unstable CHRNA10 49 42 Cc1ccccc1OCC(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217513105 FG For-Sale Unstable NPY5R 43 52 O=C(O)[C@H]1CS[C@@H](c2ccccc2)N1C(=O)c1ccc(Cl)cc1 ZINC000217513122 EH In-Stock Unstable THYX_PBCV1 0 40 O=C(O)[C@H]1CS[C@@H](c2ccccc2)N1C(=O)c1ccc(Cl)cc1 ZINC000217513122 EH In-Stock Unstable FPTA 43 36 COCCN1CCN(CC(=O)NC[C@@H](c2ccccc2Cl)N2CCCC2)CC1 ZINC000217513178 HD On-Demand Unstable DRD4 44 37 COCCN1CCN(CC(=O)NC[C@@H](c2ccccc2Cl)N2CCCC2)CC1 ZINC000217513178 HD On-Demand Unstable DRD3 41 38 COCCN1CCN(CC(=O)NC[C@@H](c2ccccc2Cl)N2CCCC2)CC1 ZINC000217513178 HD On-Demand Unstable HTR4 50 38 C[C@@H](c1cccc(F)c1)N1CCC[C@@H](CN)C1 ZINC000217513182 BF On-Demand Unstable CHRNA10 49 42 C[C@@H]1CCC[C@@]([C@@H](O)Cc2ccc(Cl)cc2Cl)(N(C)C)C1 ZINC000217513211 EI For-Sale Unstable UGCG 20 41 Cc1cccc(OCC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217513214 FG For-Sale Unstable NPY5R 46 51 COCCN1CCN(CC(=O)NC[C@H](c2ccccc2Cl)N2CCCC2)CC1 ZINC000217513267 HD On-Demand Unstable DRD4 44 37 COCCN1CCN(CC(=O)NC[C@H](c2ccccc2Cl)N2CCCC2)CC1 ZINC000217513267 HD On-Demand Unstable DRD3 41 38 COCCN1CCN(CC(=O)NC[C@H](c2ccccc2Cl)N2CCCC2)CC1 ZINC000217513267 HD On-Demand Unstable HTR4 50 38 CSc1ccccc1C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217513315 FH For-Sale Unstable AVPR1A 17 54 CSc1ccccc1C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217513315 FH For-Sale Unstable NPY5R 41 53 C[C@@H]1CCC[C@]([C@@H](O)Cc2ccc(Cl)cc2Cl)(N(C)C)C1 ZINC000217513392 EI For-Sale Unstable UGCG 20 41 CCCCCNc1ccc(C(=O)O)cc1S(=O)(=O)NCCCOC(C)C ZINC000217513406 GG In-Stock Unstable PLA2G4B 43 36 CSc1ncccc1C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217513437 FG For-Sale Unstable AVPR1A 24 53 CSc1ncccc1C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217513437 FG For-Sale Unstable NPY5R 56 48 CCN(CCc1ccncc1)C(=O)NCCc1ccc(OC)cc1 ZINC000217513446 EF For-Sale Unstable PTGDR 24 41 CCN(CCc1ccncc1)C(=O)NCCc1ccc(OC)cc1 ZINC000217513446 EF For-Sale Unstable PROKR1 52 32 O=S(=O)(NCCF)c1ccc(Cl)cc1 ZINC000217513502 BD On-Demand Unstable TBXA2R 55 44 O=S(=O)(NCCF)c1ccc(Cl)cc1 ZINC000217513502 BD On-Demand Unstable TBXAS1 37 41 O=S(=O)(NCCF)c1ccc(Cl)cc1 ZINC000217513502 BD On-Demand Unstable CCR1 18 46 O=C1OC2(CCN(C(=O)COc3ccc(F)cc3)CC2)c2ccccc21 ZINC000217513543 FF For-Sale Unstable NPY5R 50 56 COc1ccc(CCNC(=O)Nc2ccc(N3CCCCC3)cc2)cc1 ZINC000217513567 FI On-Demand Unstable GYRB 0 41 COc1ccc(CCNC(=O)Nc2ccc(N3CCCCC3)cc2)cc1 ZINC000217513567 FI On-Demand Unstable ADRB1 20 40 COc1ccc(CCNC(=O)Nc2ccc(N3CCCCC3)cc2)cc1 ZINC000217513567 FI On-Demand Unstable DRD4 43 36 COc1ccc(CCNC(=O)Nc2ccc(N3CCCCC3)cc2)cc1 ZINC000217513567 FI On-Demand Unstable HRH2 28 52 COc1ccc(CCNC(=O)Nc2ccc(N3CCCCC3)cc2)cc1 ZINC000217513567 FI On-Demand Unstable BMP1 17 46 COc1ccc(CCNC(=O)Nc2ccc(N3CCCCC3)cc2)cc1 ZINC000217513567 FI On-Demand Unstable KCNQ2 17 41 COc1ccc(CCNC(=O)Nc2ccc(N3CCCCC3)cc2)cc1 ZINC000217513567 FI On-Demand Unstable CA1 18 46 COc1ccc(CCNC(=O)Nc2ccc(N3CCCCC3)cc2)cc1 ZINC000217513567 FI On-Demand Unstable CTSK 18 42 COc1ccc(CCNC(=O)Nc2ccc(N3CCCCC3)cc2)cc1 ZINC000217513567 FI On-Demand Unstable CTSL 25 42 COc1ccc(CCNC(=O)Nc2ccc(N3CCCCC3)cc2)cc1 ZINC000217513567 FI On-Demand Unstable CCR3 28 43 COc1ccc(CCNC(=O)Nc2ccc(N3CCCCC3)cc2)cc1 ZINC000217513567 FI On-Demand Unstable MTNR1A 52 36 COc1ccc(CCNC(=O)Nc2ccc(N3CCCCC3)cc2)cc1 ZINC000217513567 FI On-Demand Unstable MTNR1B 45 40 COc1ccc(CCNC(=O)Nc2ccc(N3CCCCC3)cc2)cc1 ZINC000217513567 FI On-Demand Unstable GALR2 42 33 COc1ccc(CCNC(=O)Nc2ccc(N3CCCCC3)cc2)cc1 ZINC000217513567 FI On-Demand Unstable EPHX2 32 45 COc1ccc(CCNC(=O)Nc2ccc(N3CCCCC3)cc2)cc1 ZINC000217513567 FI On-Demand Unstable CA9 20 41 COc1ccc(CCNC(=O)Nc2ccc(N3CCCCC3)cc2)cc1 ZINC000217513567 FI On-Demand Unstable MCHR1 17 62 COc1ccc(CCNC(=O)Nc2ccc(N3CCCCC3)cc2)cc1 ZINC000217513567 FI On-Demand Unstable NAMPT 15 43 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Br)cc1 ZINC000217513645 EI For-Sale Unstable LTB4R 0 47 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Br)cc1 ZINC000217513645 EI For-Sale Unstable MMP2 22 51 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Br)cc1 ZINC000217513645 EI For-Sale Unstable HDAC2 18 43 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Br)cc1 ZINC000217513645 EI For-Sale Unstable HDAC6 18 43 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Br)cc1 ZINC000217513645 EI For-Sale Unstable MMP9 21 51 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Br)cc1 ZINC000217513645 EI For-Sale Unstable MMP1 25 51 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Br)cc1 ZINC000217513645 EI For-Sale Unstable TRPM2 0 42 O=C(O)CC[C@H](NC(=O)CC(=O)N[C@@H](CCC(=O)O)C(=O)O)C(=O)O ZINC000217513646 FA In-Stock Unstable TYMS 47 34 O=C(O)CC[C@H](NC(=O)CC(=O)N[C@@H](CCC(=O)O)C(=O)O)C(=O)O ZINC000217513646 FA In-Stock Unstable FOLH1 90 56 O=C(O)CC[C@H](NC(=O)CC(=O)N[C@@H](CCC(=O)O)C(=O)O)C(=O)O ZINC000217513646 FA In-Stock Unstable FOLR1 49 31 O=C(O)CC[C@H](NC(=O)CC(=O)N[C@@H](CCC(=O)O)C(=O)O)C(=O)O ZINC000217513646 FA In-Stock Unstable NAALAD2 89 72 O=C(O)CC[C@H](NC(=O)CC(=O)N[C@@H](CCC(=O)O)C(=O)O)C(=O)O ZINC000217513646 FA In-Stock Unstable GRIK3 15 43 O=C(O)CC[C@H](NC(=O)CC(=O)N[C@@H](CCC(=O)O)C(=O)O)C(=O)O ZINC000217513646 FA In-Stock Unstable PAM 0 41 O=C(O)CC[C@H](NC(=O)CC(=O)N[C@@H](CCC(=O)O)C(=O)O)C(=O)O ZINC000217513646 FA In-Stock Unstable GGH 0 50 O=C(O)CC[C@H](NC(=O)CC(=O)N[C@@H](CCC(=O)O)C(=O)O)C(=O)O ZINC000217513646 FA In-Stock Unstable GART 66 33 O=C(O)CC[C@H](NC(=O)CC(=O)N[C@@H](CCC(=O)O)C(=O)O)C(=O)O ZINC000217513646 FA In-Stock Unstable GNPAT 0 55 O=C(O)CC[C@H](NC(=O)CC(=O)N[C@@H](CCC(=O)O)C(=O)O)C(=O)O ZINC000217513646 FA In-Stock Unstable CPG2 0 46 O=C(O)CC[C@H](NC(=O)CC(=O)N[C@@H](CCC(=O)O)C(=O)O)C(=O)O ZINC000217513646 FA In-Stock Unstable DLG4 57 31 O=C(O)CC[C@H](NC(=O)CC(=O)N[C@@H](CCC(=O)O)C(=O)O)C(=O)O ZINC000217513646 FA In-Stock Unstable NOD1 93 49 O=C(O)CC[C@H](NC(=O)CC(=O)N[C@@H](CCC(=O)O)C(=O)O)C(=O)O ZINC000217513646 FA In-Stock Unstable KDM4E 22 41 O=C(O)CC[C@H](NC(=O)CC(=O)N[C@@H](CCC(=O)O)C(=O)O)C(=O)O ZINC000217513646 FA In-Stock Unstable SLC46A1 56 31 O=C(O)CC[C@H](NC(=O)CC(=O)N[C@@H](CCC(=O)O)C(=O)O)C(=O)O ZINC000217513646 FA In-Stock Unstable KDM2A 36 41 O=C(O)CC[C@H](NC(=O)CC(=O)N[C@@H](CCC(=O)O)C(=O)O)C(=O)O ZINC000217513646 FA In-Stock Unstable PHF8 0 41 O=C(O)CC[C@H](NC(=O)CC(=O)N[C@@H](CCC(=O)O)C(=O)O)C(=O)O ZINC000217513646 FA In-Stock Unstable KDM5C 0 41 O=S(=O)(C[C@@H]1CCCN1)c1ccccc1F ZINC000217513656 BD For-Sale Unstable CHRNA10 33 45 COc1ccc(CCNC(=O)Nc2ccc(SC#N)cc2)cc1 ZINC000217513657 EH For-Sale Unstable ADRB1 21 43 COc1ccc(CCNC(=O)Nc2ccc(SC#N)cc2)cc1 ZINC000217513657 EH For-Sale Unstable BMP1 16 47 COc1ccc(CCNC(=O)Nc2ccc(SC#N)cc2)cc1 ZINC000217513657 EH For-Sale Unstable CA1 25 46 COc1ccc(CCNC(=O)Nc2ccc(SC#N)cc2)cc1 ZINC000217513657 EH For-Sale Unstable CTSL 15 41 COc1ccc(CCNC(=O)Nc2ccc(SC#N)cc2)cc1 ZINC000217513657 EH For-Sale Unstable MTNR1A 43 39 COc1ccc(CCNC(=O)Nc2ccc(SC#N)cc2)cc1 ZINC000217513657 EH For-Sale Unstable CA12 18 46 COc1ccc(CCNC(=O)Nc2ccc(SC#N)cc2)cc1 ZINC000217513657 EH For-Sale Unstable PTGDR 17 43 COc1ccc(CCNC(=O)Nc2ccc(SC#N)cc2)cc1 ZINC000217513657 EH For-Sale Unstable CA9 21 42 COc1ccc(CCNC(=O)Nc2ccc(SC#N)cc2)cc1 ZINC000217513657 EH For-Sale Unstable NCE103 28 46 O=C1OC2(CCN(C(=O)Cc3ccc(Cl)cc3)CC2)c2ccccc21 ZINC000217513668 FH For-Sale Unstable AVPR1A 26 57 O=C1OC2(CCN(C(=O)Cc3ccc(Cl)cc3)CC2)c2ccccc21 ZINC000217513668 FH For-Sale Unstable SIGMAR1 17 55 O=C1OC2(CCN(C(=O)Cc3ccc(Cl)cc3)CC2)c2ccccc21 ZINC000217513668 FH For-Sale Unstable NPY5R 42 57 O=S(=O)(C[C@H]1CCCN1)c1ccccc1F ZINC000217513722 BD For-Sale Unstable CHRNA10 33 45 COc1ccc(CCS(=O)(=O)NC[C@@](C)(O)c2cc3ccccc3s2)cc1 ZINC000217513732 HG In-Stock Unstable MMP12 18 48 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Br)cc1 ZINC000217513741 EI For-Sale Unstable LTB4R 0 47 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Br)cc1 ZINC000217513741 EI For-Sale Unstable MMP2 22 51 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Br)cc1 ZINC000217513741 EI For-Sale Unstable HDAC2 18 43 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Br)cc1 ZINC000217513741 EI For-Sale Unstable HDAC6 18 43 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Br)cc1 ZINC000217513741 EI For-Sale Unstable MMP9 21 51 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Br)cc1 ZINC000217513741 EI For-Sale Unstable MMP1 25 51 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Br)cc1 ZINC000217513741 EI For-Sale Unstable TRPM2 0 42 O=C1OC2(CCN(C(=O)Cc3ccccc3Cl)CC2)c2ccccc21 ZINC000217513773 FH For-Sale Unstable AVPR1A 15 50 O=C1OC2(CCN(C(=O)Cc3ccccc3Cl)CC2)c2ccccc21 ZINC000217513773 FH For-Sale Unstable NPY5R 47 56 COc1ccc(CCNC(=O)N(Cc2ccccc2)c2ccccc2)cc1 ZINC000217513774 FJ For-Sale Unstable BMP1 49 45 COc1ccc(CCNC(=O)N(Cc2ccccc2)c2ccccc2)cc1 ZINC000217513774 FJ For-Sale Unstable NQO2 25 40 COc1ccc(CCNC(=O)N(Cc2ccccc2)c2ccccc2)cc1 ZINC000217513774 FJ For-Sale Unstable TSPO 40 32 COc1ccc(CCNC(=O)N(Cc2ccccc2)c2ccccc2)cc1 ZINC000217513774 FJ For-Sale Unstable SIGMAR1 15 42 COc1ccc(CCNC(=O)N(Cc2ccccc2)c2ccccc2)cc1 ZINC000217513774 FJ For-Sale Unstable MMP16 0 40 COc1ccc(CCNC(=O)N(Cc2ccccc2)c2ccccc2)cc1 ZINC000217513774 FJ For-Sale Unstable MTNR1A 86 42 COc1ccc(CCNC(=O)N(Cc2ccccc2)c2ccccc2)cc1 ZINC000217513774 FJ For-Sale Unstable MTNR1B 74 39 COc1ccc(CCNC(=O)N(Cc2ccccc2)c2ccccc2)cc1 ZINC000217513774 FJ For-Sale Unstable MMP2 23 42 COc1ccc(CCNC(=O)N(Cc2ccccc2)c2ccccc2)cc1 ZINC000217513774 FJ For-Sale Unstable MMP3 31 42 COc1ccc(CCNC(=O)N(Cc2ccccc2)c2ccccc2)cc1 ZINC000217513774 FJ For-Sale Unstable MMP8 20 42 COc1ccc(CCNC(=O)N(Cc2ccccc2)c2ccccc2)cc1 ZINC000217513774 FJ For-Sale Unstable NR1H4 28 40 COc1ccc(CCNC(=O)N(Cc2ccccc2)c2ccccc2)cc1 ZINC000217513774 FJ For-Sale Unstable NPY5R 19 40 COc1ccc(CCNC(=O)N(Cc2ccccc2)c2ccccc2)cc1 ZINC000217513774 FJ For-Sale Unstable MMP9 34 42 COc1ccc(CCNC(=O)N(Cc2ccccc2)c2ccccc2)cc1 ZINC000217513774 FJ For-Sale Unstable MMP12 23 42 COc1ccc(CCNC(=O)N(Cc2ccccc2)c2ccccc2)cc1 ZINC000217513774 FJ For-Sale Unstable PTGDR 22 41 COc1ccc(CCNC(=O)N(Cc2ccccc2)c2ccccc2)cc1 ZINC000217513774 FJ For-Sale Unstable CA9 18 44 COc1ccc(CCNC(=O)N(Cc2ccccc2)c2ccccc2)cc1 ZINC000217513774 FJ For-Sale Unstable MMP1 33 42 COc1ccc(CCS(=O)(=O)NC[C@](C)(O)c2cc3ccccc3s2)cc1 ZINC000217513822 HG In-Stock Unstable MMP12 18 48 COc1ccc(CCNC(=O)N(C)c2ccc(O)cc2)cc1 ZINC000217513889 DF For-Sale Unstable ADRB2 21 42 COc1ccc(CCNC(=O)N(C)c2ccc(O)cc2)cc1 ZINC000217513889 DF For-Sale Unstable ADRB1 27 43 COc1ccc(CCNC(=O)N(C)c2ccc(O)cc2)cc1 ZINC000217513889 DF For-Sale Unstable ADRB3 23 46 COc1ccc(CCNC(=O)N(C)c2ccc(O)cc2)cc1 ZINC000217513889 DF For-Sale Unstable MTNR1A 72 38 COc1ccc(CCNC(=O)N(C)c2ccc(O)cc2)cc1 ZINC000217513889 DF For-Sale Unstable MTNR1B 61 38 COc1ccc(CCNC(=O)N(C)c2ccc(O)cc2)cc1 ZINC000217513889 DF For-Sale Unstable SLC6A5 16 46 COc1ccc(CCNC(=O)N(C)c2ccc(O)cc2)cc1 ZINC000217513889 DF For-Sale Unstable PTGDR 22 40 COc1ccc(CCNC(=O)N(C)c2ccc(O)cc2)cc1 ZINC000217513889 DF For-Sale Unstable CA9 18 46 COc1ccc(CCNC(=O)N(C)c2ccc(O)cc2)cc1 ZINC000217513889 DF For-Sale Unstable NCE103 18 40 CCCc1nnsc1C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217513896 FF For-Sale Unstable NPY5R 42 49 COc1ccc(CCNC(=O)N(C=O)CCCN)cc1 ZINC000217514001 CC For-Sale Unstable MTNR1A 53 36 COc1ccc(CCNC(=O)N(C=O)CCCN)cc1 ZINC000217514001 CC For-Sale Unstable MTNR1B 45 34 COc1ccc(CCNC(=O)N(C=O)CCCN)cc1 ZINC000217514001 CC For-Sale Unstable CA9 18 45 COc1ccc(CCNC(=O)N(C=O)CCCN)cc1 ZINC000217514001 CC For-Sale Unstable PROKR1 59 33 O=C1OC2(CCN(C(=O)c3cnc4ccccc4n3)CC2)c2ccccc21 ZINC000217514004 FF For-Sale Unstable AVPR1A 21 50 O=C1OC2(CCN(C(=O)c3cnc4ccccc4n3)CC2)c2ccccc21 ZINC000217514004 FF For-Sale Unstable NPY5R 56 55 COc1ccc2c3c1O[C@@H]1[C@@H](O)C=C[C@H]4[C@H](C2)[N+](C)(C)CC[C@]314 ZINC000217514010 DD In-Stock Unstable OPRM1 0 63 COc1ccc2c3c1O[C@@H]1[C@@H](O)C=C[C@H]4[C@H](C2)[N+](C)(C)CC[C@]314 ZINC000217514010 DD In-Stock Unstable OPRL1 0 59 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCCC ZINC000217514017 EF In-Stock Unstable PLA2G4B 43 36 O=S(=O)(C[C@@H]1CCCN1)c1cccc(F)c1 ZINC000217514041 BD For-Sale Unstable HTR6 33 40 O=S(=O)(C[C@@H]1CCCN1)c1cccc(F)c1 ZINC000217514041 BD For-Sale Unstable CHRNA10 46 52 COc1ccc2c3c1O[C@@H]1[C@@H](O)C=C[C@H]4[C@H](C2)[N+](C)(C)CC[C@@]314 ZINC000217514095 DD In-Stock Unstable OPRM1 0 63 COc1ccc2c3c1O[C@@H]1[C@@H](O)C=C[C@H]4[C@H](C2)[N+](C)(C)CC[C@@]314 ZINC000217514095 DD In-Stock Unstable OPRL1 0 59 O=C1OC2(CCN(C(=O)c3ccc(F)cc3Cl)CC2)c2ccccc21 ZINC000217514107 FH For-Sale Unstable AVPR1A 24 59 O=C1OC2(CCN(C(=O)c3ccc(F)cc3Cl)CC2)c2ccccc21 ZINC000217514107 FH For-Sale Unstable P2RX7 24 48 O=C1OC2(CCN(C(=O)c3ccc(F)cc3Cl)CC2)c2ccccc21 ZINC000217514107 FH For-Sale Unstable NPY5R 48 54 COc1ccc(CCNC(=O)NCCCNC=O)cc1 ZINC000217514117 CC For-Sale Unstable ADRB1 17 40 COc1ccc(CCNC(=O)NCCCNC=O)cc1 ZINC000217514117 CC For-Sale Unstable SCNN1A 34 40 COc1ccc(CCNC(=O)NCCCNC=O)cc1 ZINC000217514117 CC For-Sale Unstable MTNR1A 78 44 COc1ccc(CCNC(=O)NCCCNC=O)cc1 ZINC000217514117 CC For-Sale Unstable MTNR1B 64 41 COc1ccc(CCNC(=O)NCCCNC=O)cc1 ZINC000217514117 CC For-Sale Unstable SLC2A1 0 40 COc1ccc(CCNC(=O)NCCCNC=O)cc1 ZINC000217514117 CC For-Sale Unstable SLC6A5 16 47 COc1ccc(CCNC(=O)NCCCNC=O)cc1 ZINC000217514117 CC For-Sale Unstable CA9 18 47 COc1ccc(CCNC(=O)NCCCNC=O)cc1 ZINC000217514117 CC For-Sale Unstable LMGT2 0 40 O=S(=O)(C[C@H]1CCCN1)c1cccc(F)c1 ZINC000217514122 BD For-Sale Unstable HTR6 33 40 O=S(=O)(C[C@H]1CCCN1)c1cccc(F)c1 ZINC000217514122 BD For-Sale Unstable CHRNA10 46 52 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NC(C)C ZINC000217514126 EF In-Stock Unstable PLA2G4B 41 34 CC(C)c1nccn1[C@@H](C)C(=O)NCCc1noc(-c2ccccc2)n1 ZINC000217514130 FF In-Stock Unstable CASP3 41 35 COc1ccc(Cl)cc1S(=O)(=O)NC[C@@](C)(O)c1cc2ccccc2s1 ZINC000217514160 HH In-Stock Unstable COLA 60 40 COc1ccc(Cl)cc1S(=O)(=O)NC[C@@](C)(O)c1cc2ccccc2s1 ZINC000217514160 HH In-Stock Unstable CPT1A 61 40 COc1ccc(Cl)cc1S(=O)(=O)NC[C@@](C)(O)c1cc2ccccc2s1 ZINC000217514160 HH In-Stock Unstable CPT1B 64 35 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(F)cc1 ZINC000217514176 CH For-Sale Unstable LTB4R 0 47 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(F)cc1 ZINC000217514176 CH For-Sale Unstable HDAC8 15 40 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(F)cc1 ZINC000217514176 CH For-Sale Unstable MMP2 23 55 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(F)cc1 ZINC000217514176 CH For-Sale Unstable HDAC1 27 45 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(F)cc1 ZINC000217514176 CH For-Sale Unstable HDAC2 15 40 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(F)cc1 ZINC000217514176 CH For-Sale Unstable MMP9 22 55 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(F)cc1 ZINC000217514176 CH For-Sale Unstable MMP1 26 55 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCCCC ZINC000217514210 EG In-Stock Unstable PLA2G4B 43 36 Cc1nc2ccccn2c1C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217514216 FF For-Sale Unstable NPY5R 41 48 CC(C)c1nccn1[C@H](C)C(=O)NCCc1noc(-c2ccccc2)n1 ZINC000217514223 FF In-Stock Unstable CASP3 41 35 c1nnc(N2CCNCC2)cc1N1CCCC1 ZINC000217514228 BC In-Stock Unstable CHRNA4 44 49 Cc1cc(NC(=O)c2cc(Br)ccc2I)ccc1Br ZINC000217514232 JK For-Sale Unstable Q25615_ONCVO 70 47 Cc1cc(NC(=O)c2cc(Br)ccc2I)ccc1Br ZINC000217514232 JK For-Sale Unstable KCNK3 41 36 CC1=C(/C=C\C(C)=C/C=C/C(C)=C/C(=O)Oc2c(C)c(C)c3c(c2C)CC[C@@](C)(CCC[C@H](C)CCC[C@H](C)CCCC(C)C)O3)C(C)(C)CCC1 ZINC000217514244 KK In-Stock Unstable RBP4 40 46 COc1ccc(Cl)cc1S(=O)(=O)NC[C@](C)(O)c1cc2ccccc2s1 ZINC000217514250 HH In-Stock Unstable COLA 60 40 COc1ccc(Cl)cc1S(=O)(=O)NC[C@](C)(O)c1cc2ccccc2s1 ZINC000217514250 HH In-Stock Unstable CPT1A 61 40 COc1ccc(Cl)cc1S(=O)(=O)NC[C@](C)(O)c1cc2ccccc2s1 ZINC000217514250 HH In-Stock Unstable CPT1B 64 35 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(F)cc1 ZINC000217514252 CH For-Sale Unstable LTB4R 0 47 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(F)cc1 ZINC000217514252 CH For-Sale Unstable HDAC8 15 40 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(F)cc1 ZINC000217514252 CH For-Sale Unstable MMP2 23 55 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(F)cc1 ZINC000217514252 CH For-Sale Unstable HDAC1 27 45 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(F)cc1 ZINC000217514252 CH For-Sale Unstable HDAC2 15 40 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(F)cc1 ZINC000217514252 CH For-Sale Unstable MMP9 22 55 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(F)cc1 ZINC000217514252 CH For-Sale Unstable MMP1 26 55 CC1=C(/C=C\C(C)=C/C=C/C(C)=C\C(=O)Oc2c(C)c(C)c3c(c2C)CC[C@@](C)(CCC[C@H](C)CCC[C@H](C)CCCC(C)C)O3)C(C)(C)CCC1 ZINC000217514319 KK In-Stock Unstable RBP4 40 46 O=C1OC2(CCN(C(=O)c3cc(-c4ccco4)on3)CC2)c2ccccc21 ZINC000217514321 FG For-Sale Unstable AVPR1A 15 49 O=C1OC2(CCN(C(=O)c3cc(-c4ccco4)on3)CC2)c2ccccc21 ZINC000217514321 FG For-Sale Unstable NPY5R 41 46 Cc1nc(/C=C\C(=O)Nc2ccccc2[C@@H](C)O)cs1 ZINC000217514328 CG For-Sale Unstable UL26 93 40 Cc1nc(/C=C\C(=O)Nc2ccccc2[C@@H](C)O)cs1 ZINC000217514328 CG For-Sale Unstable U53 0 40 Cc1nc(/C=C\C(=O)Nc2ccccc2[C@@H](C)O)cs1 ZINC000217514328 CG For-Sale Unstable SCAF_EBVB9 83 37 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1cccnc1 ZINC000217514329 EF For-Sale Unstable DRD4 40 31 C[C@@H](NC(=O)CN1CCC[C@@H](N)C1)c1ccccc1 ZINC000217514362 CD On-Demand Unstable SLC6A1 70 38 C[C@@H](NC(=O)CN1CCC[C@@H](N)C1)c1ccccc1 ZINC000217514362 CD On-Demand Unstable PRCP 25 44 C[C@@H](NC(=O)CN1CCC[C@@H](N)C1)c1ccccc1 ZINC000217514362 CD On-Demand Unstable XIAP 59 39 C[C@@H](NC(=O)CN1CCC[C@@H](N)C1)c1ccccc1 ZINC000217514362 CD On-Demand Unstable BIRC2 56 43 C[C@@H](NC(=O)CN1CCC[C@@H](N)C1)c1ccccc1 ZINC000217514362 CD On-Demand Unstable BIRC8 54 34 COCCNc1nc2cc(C(=O)N(C)C[C@@H]3COCCO3)ccc2n1C ZINC000217514380 FD In-Stock Unstable ITK 40 37 COc1ccc(CCNC(=O)N2C[C@@]3(C)C[C@H]2CC(C)(C)C3)cc1 ZINC000217514388 EH On-Demand Unstable AVPR2 17 45 COc1ccc(CCNC(=O)N2C[C@@]3(C)C[C@H]2CC(C)(C)C3)cc1 ZINC000217514388 EH On-Demand Unstable AVPR1A 35 41 COc1ccc(CCNC(=O)N2C[C@@]3(C)C[C@H]2CC(C)(C)C3)cc1 ZINC000217514388 EH On-Demand Unstable PROKR1 60 33 Cc1nc(/C=C\C(=O)Nc2ccccc2[C@H](C)O)cs1 ZINC000217514420 CG For-Sale Unstable UL26 93 40 Cc1nc(/C=C\C(=O)Nc2ccccc2[C@H](C)O)cs1 ZINC000217514420 CG For-Sale Unstable U53 0 40 Cc1nc(/C=C\C(=O)Nc2ccccc2[C@H](C)O)cs1 ZINC000217514420 CG For-Sale Unstable SCAF_EBVB9 83 37 COC(=O)c1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217514432 FF For-Sale Unstable NPY5R 53 59 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1[C@H]2C=C[C@@]3(CN(Cc4ccc5c(c4)OCO5)C(=O)[C@H]13)O2 ZINC000217514438 JF In-Stock Unstable BRS3 22 43 C[C@H](NC(=O)CN1CCC[C@@H](N)C1)c1ccccc1 ZINC000217514444 CD On-Demand Unstable SLC6A1 70 38 C[C@H](NC(=O)CN1CCC[C@@H](N)C1)c1ccccc1 ZINC000217514444 CD On-Demand Unstable PRCP 25 44 C[C@H](NC(=O)CN1CCC[C@@H](N)C1)c1ccccc1 ZINC000217514444 CD On-Demand Unstable XIAP 59 39 C[C@H](NC(=O)CN1CCC[C@@H](N)C1)c1ccccc1 ZINC000217514444 CD On-Demand Unstable BIRC2 56 43 C[C@H](NC(=O)CN1CCC[C@@H](N)C1)c1ccccc1 ZINC000217514444 CD On-Demand Unstable BIRC8 54 34 COCCNc1nc2cc(C(=O)N(C)C[C@H]3COCCO3)ccc2n1C ZINC000217514464 FD In-Stock Unstable ITK 40 37 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Cl)s1 ZINC000217514498 DI For-Sale Unstable UL26 15 42 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Cl)s1 ZINC000217514498 DI For-Sale Unstable U53 0 42 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Cl)s1 ZINC000217514498 DI For-Sale Unstable SCAF_EBVB9 24 42 C[C@H](c1ccc(OC(F)(F)F)cc1)N1CCC[C@@H](CN)C1 ZINC000217514500 DG On-Demand Unstable HCRTR1 0 40 C[C@H](c1ccc(OC(F)(F)F)cc1)N1CCC[C@@H](CN)C1 ZINC000217514500 DG On-Demand Unstable HCRTR2 0 40 O=C(NCCc1c[nH]c2ccccc12)[C@H]1[C@H]2C=C[C@@]3(CN(Cc4ccc5c(c4)OCO5)C(=O)[C@H]13)O2 ZINC000217514523 JF In-Stock Unstable BRS3 22 43 O=C1OC2(CCN(C(=O)c3ccc4nsnc4c3)CC2)c2ccccc21 ZINC000217514556 FF In-Stock Unstable AVPR1A 15 48 O=C1OC2(CCN(C(=O)c3ccc4nsnc4c3)CC2)c2ccccc21 ZINC000217514556 FF In-Stock Unstable NPY5R 44 51 Cc1nc(N2CCN(c3ccccn3)CC2)nc(C)c1N ZINC000217514567 CD In-Stock Unstable DRD4 33 42 Cc1nc(N2CCN(c3ccccn3)CC2)nc(C)c1N ZINC000217514567 CD In-Stock Unstable EBP 30 44 Cc1nc(N2CCN(c3ccccn3)CC2)nc(C)c1N ZINC000217514567 CD In-Stock Unstable SORD 54 38 Cc1nc(N2CCN(c3ccccn3)CC2)nc(C)c1N ZINC000217514567 CD In-Stock Unstable SLC6A7 0 41 COc1ccc(CCNC(=O)Nc2cccc(N(C)C)c2)cc1 ZINC000217514576 DG For-Sale Unstable ADRB1 16 40 COc1ccc(CCNC(=O)Nc2cccc(N(C)C)c2)cc1 ZINC000217514576 DG For-Sale Unstable BMP1 27 47 COc1ccc(CCNC(=O)Nc2cccc(N(C)C)c2)cc1 ZINC000217514576 DG For-Sale Unstable NQO2 40 43 COc1ccc(CCNC(=O)Nc2cccc(N(C)C)c2)cc1 ZINC000217514576 DG For-Sale Unstable CA1 23 44 COc1ccc(CCNC(=O)Nc2cccc(N(C)C)c2)cc1 ZINC000217514576 DG For-Sale Unstable TRPV1 0 53 COc1ccc(CCNC(=O)Nc2cccc(N(C)C)c2)cc1 ZINC000217514576 DG For-Sale Unstable CCKAR 0 43 COc1ccc(CCNC(=O)Nc2cccc(N(C)C)c2)cc1 ZINC000217514576 DG For-Sale Unstable CCR3 37 43 COc1ccc(CCNC(=O)Nc2cccc(N(C)C)c2)cc1 ZINC000217514576 DG For-Sale Unstable RAF1 44 43 COc1ccc(CCNC(=O)Nc2cccc(N(C)C)c2)cc1 ZINC000217514576 DG For-Sale Unstable MTNR1A 119 50 COc1ccc(CCNC(=O)Nc2cccc(N(C)C)c2)cc1 ZINC000217514576 DG For-Sale Unstable MTNR1B 99 50 COc1ccc(CCNC(=O)Nc2cccc(N(C)C)c2)cc1 ZINC000217514576 DG For-Sale Unstable ROCK2 24 56 COc1ccc(CCNC(=O)Nc2cccc(N(C)C)c2)cc1 ZINC000217514576 DG For-Sale Unstable FLT4 19 40 COc1ccc(CCNC(=O)Nc2cccc(N(C)C)c2)cc1 ZINC000217514576 DG For-Sale Unstable CA12 15 44 COc1ccc(CCNC(=O)Nc2cccc(N(C)C)c2)cc1 ZINC000217514576 DG For-Sale Unstable PTGDR 22 52 COc1ccc(CCNC(=O)Nc2cccc(N(C)C)c2)cc1 ZINC000217514576 DG For-Sale Unstable CA9 17 44 COc1ccc(CCNC(=O)Nc2cccc(N(C)C)c2)cc1 ZINC000217514576 DG For-Sale Unstable Q8MMZ8_EIMTE 33 43 COc1ccc(CCNC(=O)Nc2cccc(N(C)C)c2)cc1 ZINC000217514576 DG For-Sale Unstable NCE103 26 44 COc1ccc(CCNC(=O)Nc2cccc(N(C)C)c2)cc1 ZINC000217514576 DG For-Sale Unstable ACAT 0 43 COc1ccc(CCNC(=O)Nc2cccc(N(C)C)c2)cc1 ZINC000217514576 DG For-Sale Unstable PSBA 0 43 C[C@@H](c1ccc(OC(F)(F)F)cc1)N1CCC[C@@H](CN)C1 ZINC000217514577 DG On-Demand Unstable HCRTR1 0 40 C[C@@H](c1ccc(OC(F)(F)F)cc1)N1CCC[C@@H](CN)C1 ZINC000217514577 DG On-Demand Unstable HCRTR2 0 40 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Cl)s1 ZINC000217514586 DI For-Sale Unstable UL26 15 42 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Cl)s1 ZINC000217514586 DI For-Sale Unstable U53 0 42 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(Cl)s1 ZINC000217514586 DI For-Sale Unstable SCAF_EBVB9 24 42 COc1ccc(-c2c(C)oc3cc(OCCN4C[C@@H]5C[C@H](C4)c4cccc(=O)n4C5)ccc3c2=O)cc1 ZINC000217514615 JI In-Stock Unstable CHRNA4 35 47 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NC(C)(C)C ZINC000217514625 EG In-Stock Unstable PLA2G4B 42 35 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(O)cc1 ZINC000217514667 CG For-Sale Unstable HDAC8 18 47 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(O)cc1 ZINC000217514667 CG For-Sale Unstable F3 26 43 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(O)cc1 ZINC000217514667 CG For-Sale Unstable MMP2 27 68 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(O)cc1 ZINC000217514667 CG For-Sale Unstable HDAC1 25 41 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(O)cc1 ZINC000217514667 CG For-Sale Unstable MMP9 24 68 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(O)cc1 ZINC000217514667 CG For-Sale Unstable MMP1 29 68 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccc(O)cc1 ZINC000217514667 CG For-Sale Unstable TRPM2 0 45 CC(C)Oc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217514672 FH For-Sale Unstable NPY5R 42 47 COc1ccc(CCNC(=O)NC(=O)c2ccccc2N)cc1 ZINC000217514705 DD For-Sale Unstable BMP1 22 40 COc1ccc(CCNC(=O)NC(=O)c2ccccc2N)cc1 ZINC000217514705 DD For-Sale Unstable CA1 15 49 COc1ccc(CCNC(=O)NC(=O)c2ccccc2N)cc1 ZINC000217514705 DD For-Sale Unstable CTSL 16 40 COc1ccc(CCNC(=O)NC(=O)c2ccccc2N)cc1 ZINC000217514705 DD For-Sale Unstable MTNR1A 73 40 COc1ccc(CCNC(=O)NC(=O)c2ccccc2N)cc1 ZINC000217514705 DD For-Sale Unstable MTNR1B 61 38 COc1ccc(CCNC(=O)NC(=O)c2ccccc2N)cc1 ZINC000217514705 DD For-Sale Unstable SLC6A5 21 46 COc1ccc(CCNC(=O)NC(=O)c2ccccc2N)cc1 ZINC000217514705 DD For-Sale Unstable CA9 22 49 COc1ccc(CCNC(=O)NC(=O)c2ccccc2N)cc1 ZINC000217514705 DD For-Sale Unstable NCE103 23 43 COc1ccc(CCNC(=O)NC(=O)c2ccccc2N)cc1 ZINC000217514705 DD For-Sale Unstable PROKR1 42 30 BrCc1ccccc1N1CC[C@@H](N2CCOCC2)C1 ZINC000217514729 EE For-Sale Unstable L3MBTL3 29 40 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(O)cc1 ZINC000217514752 CG For-Sale Unstable HDAC8 18 47 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(O)cc1 ZINC000217514752 CG For-Sale Unstable F3 26 43 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(O)cc1 ZINC000217514752 CG For-Sale Unstable MMP2 27 68 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(O)cc1 ZINC000217514752 CG For-Sale Unstable HDAC1 25 41 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(O)cc1 ZINC000217514752 CG For-Sale Unstable MMP9 24 68 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(O)cc1 ZINC000217514752 CG For-Sale Unstable MMP1 29 68 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccc(O)cc1 ZINC000217514752 CG For-Sale Unstable TRPM2 0 45 COC(=O)c1cc(OC)c(N)c(I)c1Cl ZINC000217514755 EE For-Sale Unstable HTR4 57 38 COc1ccc(CCC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217514790 FG For-Sale Unstable SIGMAR1 19 48 COc1ccc(CCC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217514790 FG For-Sale Unstable NPY5R 37 52 COc1ccc(CCNC(=O)Nc2ccccc2C(N)=O)cc1 ZINC000217514819 DE For-Sale Unstable CA2 18 48 COc1ccc(CCNC(=O)Nc2ccccc2C(N)=O)cc1 ZINC000217514819 DE For-Sale Unstable BMP1 30 40 COc1ccc(CCNC(=O)Nc2ccccc2C(N)=O)cc1 ZINC000217514819 DE For-Sale Unstable CA1 27 48 COc1ccc(CCNC(=O)Nc2ccccc2C(N)=O)cc1 ZINC000217514819 DE For-Sale Unstable TRPV1 0 58 COc1ccc(CCNC(=O)Nc2ccccc2C(N)=O)cc1 ZINC000217514819 DE For-Sale Unstable MTNR1A 79 44 COc1ccc(CCNC(=O)Nc2ccccc2C(N)=O)cc1 ZINC000217514819 DE For-Sale Unstable MTNR1B 64 39 COc1ccc(CCNC(=O)Nc2ccccc2C(N)=O)cc1 ZINC000217514819 DE For-Sale Unstable MAPK10 18 43 COc1ccc(CCNC(=O)Nc2ccccc2C(N)=O)cc1 ZINC000217514819 DE For-Sale Unstable SLC6A5 23 48 COc1ccc(CCNC(=O)Nc2ccccc2C(N)=O)cc1 ZINC000217514819 DE For-Sale Unstable CA12 22 48 COc1ccc(CCNC(=O)Nc2ccccc2C(N)=O)cc1 ZINC000217514819 DE For-Sale Unstable PTGDR 16 40 COc1ccc(CCNC(=O)Nc2ccccc2C(N)=O)cc1 ZINC000217514819 DE For-Sale Unstable CA9 24 48 COc1ccc(CCNC(=O)Nc2ccccc2C(N)=O)cc1 ZINC000217514819 DE For-Sale Unstable HCAR2 19 50 COc1ccc(CCNC(=O)Nc2ccccc2C(N)=O)cc1 ZINC000217514819 DE For-Sale Unstable NCE103 27 48 COc1ccc(CCNC(=O)Nc2ccccc2C(N)=O)cc1 ZINC000217514819 DE For-Sale Unstable PAGA 0 43 COc1ccc(CCNC(=O)Nc2ccccc2C(N)=O)cc1 ZINC000217514819 DE For-Sale Unstable PROKR1 55 34 BrCc1ccccc1N1CC[C@H](N2CCOCC2)C1 ZINC000217514828 EE For-Sale Unstable L3MBTL3 29 40 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NC1CC1 ZINC000217514845 EE In-Stock Unstable PLA2G4B 42 35 O=C(NCc1ccccc1Cl)c1cc(Br)ccc1O ZINC000217514862 EH For-Sale Unstable THRA 22 43 O=C(NCc1ccccc1Cl)c1cc(Br)ccc1O ZINC000217514862 EH For-Sale Unstable GRIN1 15 46 O=C(NCc1ccccc1Cl)c1cc(Br)ccc1O ZINC000217514862 EH For-Sale Unstable THRB 22 46 O=C(NCc1ccccc1Cl)c1cc(Br)ccc1O ZINC000217514862 EH For-Sale Unstable P2RX7 25 41 O=C(NCc1ccccc1Cl)c1cc(Br)ccc1O ZINC000217514862 EH For-Sale Unstable SCN10A 23 44 O=C(NCc1ccccc1Cl)c1cc(Br)ccc1O ZINC000217514862 EH For-Sale Unstable NCE103 25 43 O=C(NCc1ccccc1Cl)c1cc(Br)ccc1O ZINC000217514862 EH For-Sale Unstable PYK 88 42 O=C(NCc1ccccc1Cl)c1cc(Br)ccc1O ZINC000217514862 EH For-Sale Unstable P96878_MYCTU 17 43 Cc1ccccc1C(=O)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217514898 FH For-Sale Unstable FABP4 46 36 CCOc1ccc(CC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217514903 FG For-Sale Unstable NPY5R 38 46 CCN1CCN(C(=O)NCCc2ccc(OC)cc2)CC1 ZINC000217514922 CD On-Demand Unstable DRD4 42 32 CCN1CCN(C(=O)NCCc2ccc(OC)cc2)CC1 ZINC000217514922 CD On-Demand Unstable BMP1 42 34 CCN1CCN(C(=O)NCCc2ccc(OC)cc2)CC1 ZINC000217514922 CD On-Demand Unstable MMP13 32 44 CCN1CCN(C(=O)NCCc2ccc(OC)cc2)CC1 ZINC000217514922 CD On-Demand Unstable MTNR1A 59 38 CCN1CCN(C(=O)NCCc2ccc(OC)cc2)CC1 ZINC000217514922 CD On-Demand Unstable MTNR1B 50 42 CCN1CCN(C(=O)NCCc2ccc(OC)cc2)CC1 ZINC000217514922 CD On-Demand Unstable MMP3 38 51 CCN1CCN(C(=O)NCCc2ccc(OC)cc2)CC1 ZINC000217514922 CD On-Demand Unstable MMP9 37 51 CCN1CCN(C(=O)NCCc2ccc(OC)cc2)CC1 ZINC000217514922 CD On-Demand Unstable MMP7 31 51 CCN1CCN(C(=O)NCCc2ccc(OC)cc2)CC1 ZINC000217514922 CD On-Demand Unstable MMP1 32 42 CCN1CCN(C(=O)NCCc2ccc(OC)cc2)CC1 ZINC000217514922 CD On-Demand Unstable ABHD6 0 41 CCN1CCN(C(=O)NCCc2ccc(OC)cc2)CC1 ZINC000217514922 CD On-Demand Unstable PROKR1 44 31 BrCc1ccc(N2CC[C@@H](N3CCOCC3)C2)nc1 ZINC000217514937 ED For-Sale Unstable L3MBTL3 34 43 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NC1CCCC1 ZINC000217514965 FG In-Stock Unstable PLA2G4B 43 36 CN1[C@@H]2CC[C@@H]1CC(Oc1ncccc1N)C2 ZINC000217514969 BD In-Stock Unstable GLRA1 53 43 O=C1OC2(CCN(C(=O)C34CC5CC(CC(C5)C3)C4)CC2)c2ccccc21 ZINC000217515013 FH For-Sale Unstable NPY5R 52 51 Cc1cccc(C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)c1 ZINC000217515015 FH For-Sale Unstable DRD4 48 39 Cc1cccc(C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)c1 ZINC000217515015 FH For-Sale Unstable CCR2 42 37 Cc1cccc(C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)c1 ZINC000217515015 FH For-Sale Unstable KCNK3 43 36 Cc1cccc(C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)c1 ZINC000217515015 FH For-Sale Unstable KCNK9 41 35 BrCc1ccc(N2CC[C@H](N3CCOCC3)C2)nc1 ZINC000217515033 ED For-Sale Unstable L3MBTL3 34 43 CN1[C@H]2CC[C@@H]1CC(Oc1ncccc1N)C2 ZINC000217515043 BD In-Stock Unstable GLRA1 53 43 CCOc1ccc(CCNC(=O)NCCc2ccc(OC)cc2)cc1OCC ZINC000217515050 GH For-Sale Unstable INHA 40 34 CCOc1ccc(CCNC(=O)NCCc2ccc(OC)cc2)cc1OCC ZINC000217515050 GH For-Sale Unstable CNR2 41 42 CCOc1ccc(CCNC(=O)NCCc2ccc(OC)cc2)cc1OCC ZINC000217515050 GH For-Sale Unstable TRPV1 0 45 CCOc1ccc(CCNC(=O)NCCc2ccc(OC)cc2)cc1OCC ZINC000217515050 GH For-Sale Unstable SSTR5 44 35 CCOc1ccc(CCNC(=O)NCCc2ccc(OC)cc2)cc1OCC ZINC000217515050 GH For-Sale Unstable CTSL 16 40 CCOc1ccc(CCNC(=O)NCCc2ccc(OC)cc2)cc1OCC ZINC000217515050 GH For-Sale Unstable RAF1 22 41 CCOc1ccc(CCNC(=O)NCCc2ccc(OC)cc2)cc1OCC ZINC000217515050 GH For-Sale Unstable MTNR1A 116 54 CCOc1ccc(CCNC(=O)NCCc2ccc(OC)cc2)cc1OCC ZINC000217515050 GH For-Sale Unstable MTNR1B 94 54 CCOc1ccc(CCNC(=O)NCCc2ccc(OC)cc2)cc1OCC ZINC000217515050 GH For-Sale Unstable PTGDR 31 41 CCOc1ccc(CCNC(=O)NCCc2ccc(OC)cc2)cc1OCC ZINC000217515050 GH For-Sale Unstable CA9 18 46 CCOc1ccc(CCNC(=O)NCCc2ccc(OC)cc2)cc1OCC ZINC000217515050 GH For-Sale Unstable Q8MMZ8_EIMTE 25 41 CCOc1ccc(CCNC(=O)NCCc2ccc(OC)cc2)cc1OCC ZINC000217515050 GH For-Sale Unstable CAN2 0 44 C[C@@H]1[C@H](CC(=O)O)C[C@@H]1NC(=O)OC(C)(C)C ZINC000217515059 BE For-Sale Unstable NAAA 16 41 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NC1CCCCC1 ZINC000217515097 FH In-Stock Unstable CNR2 17 42 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NC1CCCCC1 ZINC000217515097 FH In-Stock Unstable PLA2G4B 43 36 O=C(NCc1cccc(Cl)c1)c1cc(Br)ccc1I ZINC000217515103 JJ On-Demand Unstable U38 0 40 COc1cc(OC)cc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217515130 FG For-Sale Unstable AVPR1A 15 51 COc1cc(OC)cc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217515130 FG For-Sale Unstable ACACA 50 36 COc1cc(OC)cc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217515130 FG For-Sale Unstable NPY5R 42 55 CN1[C@H]2CC[C@H]1CC(Oc1ncccc1N)C2 ZINC000217515131 BD In-Stock Unstable GLRA1 53 43 CN1[C@H]2CC[C@H]1CC(Oc1ncccc1N)C2 ZINC000217515131 BD In-Stock Unstable GPR119 17 41 COc1ccc(CCNC(=O)Nc2nc[nH]n2)cc1 ZINC000217515159 CD For-Sale Unstable ADRB1 17 41 COc1ccc(CCNC(=O)Nc2nc[nH]n2)cc1 ZINC000217515159 CD For-Sale Unstable BMP1 21 43 COc1ccc(CCNC(=O)Nc2nc[nH]n2)cc1 ZINC000217515159 CD For-Sale Unstable RAF1 42 40 COc1ccc(CCNC(=O)Nc2nc[nH]n2)cc1 ZINC000217515159 CD For-Sale Unstable MTNR1A 67 42 COc1ccc(CCNC(=O)Nc2nc[nH]n2)cc1 ZINC000217515159 CD For-Sale Unstable MTNR1B 52 37 COc1ccc(CCNC(=O)Nc2nc[nH]n2)cc1 ZINC000217515159 CD For-Sale Unstable PTGDR 24 42 COc1ccc(CCNC(=O)Nc2nc[nH]n2)cc1 ZINC000217515159 CD For-Sale Unstable CA9 19 47 COc1ccc(CCNC(=O)Nc2nc[nH]n2)cc1 ZINC000217515159 CD For-Sale Unstable Q8MMZ8_EIMTE 27 40 COc1ccc(CCNC(=O)Nc2nc[nH]n2)cc1 ZINC000217515159 CD For-Sale Unstable PROKR1 48 32 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1 ZINC000217515211 CG For-Sale Unstable HDAC8 41 43 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1 ZINC000217515211 CG For-Sale Unstable F3 18 43 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1 ZINC000217515211 CG For-Sale Unstable MMP2 26 64 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1 ZINC000217515211 CG For-Sale Unstable HDAC1 25 40 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1 ZINC000217515211 CG For-Sale Unstable HDAC6 29 51 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1 ZINC000217515211 CG For-Sale Unstable MMP9 22 64 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1 ZINC000217515211 CG For-Sale Unstable MMP1 27 63 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1 ZINC000217515211 CG For-Sale Unstable TRPM8 0 56 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1 ZINC000217515211 CG For-Sale Unstable TRPM2 0 45 CCCCC[C@@H](C)NC(=O)CN1CCC[C@@H](N)C1 ZINC000217515212 CD On-Demand Unstable NOD1 70 35 COc1cccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1OC ZINC000217515225 FG For-Sale Unstable AVPR1A 16 53 COc1cccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1OC ZINC000217515225 FG For-Sale Unstable NPY5R 36 56 COc1cccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1OC ZINC000217515225 FG For-Sale Unstable CCR8 20 40 C[C@H]1[C@@H](NC(=O)OC(C)(C)C)C[C@@H]1CC(=O)O ZINC000217515242 BE For-Sale Unstable NAAA 16 41 Cc1cc(S(=O)(=O)NCC(=O)N2CCC[C@@H]2c2ccccn2)ccc1F ZINC000217515258 GE In-Stock Unstable COLA 95 40 Cc1cc(S(=O)(=O)NCC(=O)N2CCC[C@@H]2c2ccccn2)ccc1F ZINC000217515258 GE In-Stock Unstable CPT1A 88 39 Cc1cc(S(=O)(=O)NCC(=O)N2CCC[C@@H]2c2ccccn2)ccc1F ZINC000217515258 GE In-Stock Unstable FAP 0 44 Cc1cc(S(=O)(=O)NCC(=O)N2CCC[C@@H]2c2ccccn2)ccc1F ZINC000217515258 GE In-Stock Unstable LEF 64 41 Cc1cc(S(=O)(=O)NCC(=O)N2CCC[C@@H]2c2ccccn2)ccc1F ZINC000217515258 GE In-Stock Unstable SFRP1 75 35 Cc1cc(S(=O)(=O)NCC(=O)N2CCC[C@@H]2c2ccccn2)ccc1F ZINC000217515258 GE In-Stock Unstable WNT3 61 34 COc1ccc(CCNC(=O)NCC(OC)OC)cc1 ZINC000217515262 CD For-Sale Unstable ADRB2 17 44 COc1ccc(CCNC(=O)NCC(OC)OC)cc1 ZINC000217515262 CD For-Sale Unstable ADRB1 21 40 COc1ccc(CCNC(=O)NCC(OC)OC)cc1 ZINC000217515262 CD For-Sale Unstable ADRB3 24 43 COc1ccc(CCNC(=O)NCC(OC)OC)cc1 ZINC000217515262 CD For-Sale Unstable NQO2 26 41 COc1ccc(CCNC(=O)NCC(OC)OC)cc1 ZINC000217515262 CD For-Sale Unstable MTNR1A 85 44 COc1ccc(CCNC(=O)NCC(OC)OC)cc1 ZINC000217515262 CD For-Sale Unstable MTNR1B 68 38 COc1ccc(CCNC(=O)NCC(OC)OC)cc1 ZINC000217515262 CD For-Sale Unstable MMP9 17 41 COc1ccc(CCNC(=O)NCC(OC)OC)cc1 ZINC000217515262 CD For-Sale Unstable PTGDR 24 40 COc1ccc(CCNC(=O)NCC(OC)OC)cc1 ZINC000217515262 CD For-Sale Unstable CA9 21 49 COc1ccc(CCNC(=O)NCC(OC)OC)cc1 ZINC000217515262 CD For-Sale Unstable MMP1 20 41 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1 ZINC000217515284 CG For-Sale Unstable HDAC8 41 43 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1 ZINC000217515284 CG For-Sale Unstable F3 18 43 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1 ZINC000217515284 CG For-Sale Unstable MMP2 26 64 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1 ZINC000217515284 CG For-Sale Unstable HDAC1 25 40 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1 ZINC000217515284 CG For-Sale Unstable HDAC6 29 51 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1 ZINC000217515284 CG For-Sale Unstable MMP9 22 64 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1 ZINC000217515284 CG For-Sale Unstable MMP1 27 63 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1 ZINC000217515284 CG For-Sale Unstable TRPM8 0 56 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1 ZINC000217515284 CG For-Sale Unstable TRPM2 0 45 CCCCC[C@H](C)NC(=O)CN1CCC[C@@H](N)C1 ZINC000217515292 CD On-Demand Unstable NOD1 70 35 COc1cccc(OC)c1C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217515324 FG For-Sale Unstable NPY5R 45 61 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCCO ZINC000217515341 ED In-Stock Unstable PLA2G4B 41 35 Cc1cc(S(=O)(=O)NCC(=O)N2CCC[C@H]2c2ccccn2)ccc1F ZINC000217515347 GE In-Stock Unstable COLA 95 40 Cc1cc(S(=O)(=O)NCC(=O)N2CCC[C@H]2c2ccccn2)ccc1F ZINC000217515347 GE In-Stock Unstable CPT1A 91 40 Cc1cc(S(=O)(=O)NCC(=O)N2CCC[C@H]2c2ccccn2)ccc1F ZINC000217515347 GE In-Stock Unstable FAP 0 44 Cc1cc(S(=O)(=O)NCC(=O)N2CCC[C@H]2c2ccccn2)ccc1F ZINC000217515347 GE In-Stock Unstable LEF 64 41 Cc1cc(S(=O)(=O)NCC(=O)N2CCC[C@H]2c2ccccn2)ccc1F ZINC000217515347 GE In-Stock Unstable SFRP1 87 35 Cc1cc(S(=O)(=O)NCC(=O)N2CCC[C@H]2c2ccccn2)ccc1F ZINC000217515347 GE In-Stock Unstable WNT3 69 34 COc1ccc(CCNC(=O)Nc2cc(C(F)(F)F)cc(C(F)(F)F)c2)cc1 ZINC000217515381 HK For-Sale Unstable PPARA 17 44 COc1ccc(CCNC(=O)Nc2cc(C(F)(F)F)cc(C(F)(F)F)c2)cc1 ZINC000217515381 HK For-Sale Unstable TACR1 17 44 COc1ccc(CCNC(=O)Nc2cc(C(F)(F)F)cc(C(F)(F)F)c2)cc1 ZINC000217515381 HK For-Sale Unstable BMP1 20 45 COc1ccc(CCNC(=O)Nc2cc(C(F)(F)F)cc(C(F)(F)F)c2)cc1 ZINC000217515381 HK For-Sale Unstable CSNK1D 18 43 COc1ccc(CCNC(=O)Nc2cc(C(F)(F)F)cc(C(F)(F)F)c2)cc1 ZINC000217515381 HK For-Sale Unstable CTSL 15 40 COc1ccc(CCNC(=O)Nc2cc(C(F)(F)F)cc(C(F)(F)F)c2)cc1 ZINC000217515381 HK For-Sale Unstable RAF1 69 50 COc1ccc(CCNC(=O)Nc2cc(C(F)(F)F)cc(C(F)(F)F)c2)cc1 ZINC000217515381 HK For-Sale Unstable MTNR1A 73 45 COc1ccc(CCNC(=O)Nc2cc(C(F)(F)F)cc(C(F)(F)F)c2)cc1 ZINC000217515381 HK For-Sale Unstable MTNR1B 60 45 COc1ccc(CCNC(=O)Nc2cc(C(F)(F)F)cc(C(F)(F)F)c2)cc1 ZINC000217515381 HK For-Sale Unstable EPHX2 25 45 COc1ccc(CCNC(=O)Nc2cc(C(F)(F)F)cc(C(F)(F)F)c2)cc1 ZINC000217515381 HK For-Sale Unstable PTGDR 23 44 COc1ccc(CCNC(=O)Nc2cc(C(F)(F)F)cc(C(F)(F)F)c2)cc1 ZINC000217515381 HK For-Sale Unstable CA9 16 44 COc1ccc(CCNC(=O)Nc2cc(C(F)(F)F)cc(C(F)(F)F)c2)cc1 ZINC000217515381 HK For-Sale Unstable Q8MMZ8_EIMTE 68 50 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccccc1F ZINC000217515383 FG For-Sale Unstable FABP4 51 38 N#Cc1ccc(-c2ccncc2)cc1C#N ZINC000217515389 BE For-Sale Mild XDH 58 44 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCCCO ZINC000217515422 ED In-Stock Unstable PLA2G4B 42 36 C[C@H](C(=O)O)C1CC(NC(=O)OC(C)(C)C)C1 ZINC000217515425 BE For-Sale Unstable PAPA1_CARPA 41 33 COc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1OC ZINC000217515458 FG For-Sale Unstable AVPR1A 24 49 COc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1OC ZINC000217515458 FG For-Sale Unstable ACACA 51 42 COc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1OC ZINC000217515458 FG For-Sale Unstable ACACB 33 42 COc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1OC ZINC000217515458 FG For-Sale Unstable NPY5R 47 57 Cc1nc(O)nc(C)c1CCC(=O)N1CCCN(Cc2cccnc2)CC1 ZINC000217515471 FD In-Stock Unstable C3AR1 48 44 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc(F)cc1 ZINC000217515492 FG For-Sale Unstable BCHE 23 44 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc(F)cc1 ZINC000217515492 FG For-Sale Unstable PLD1 43 38 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc(F)cc1 ZINC000217515492 FG For-Sale Unstable PLD2 61 40 COc1ccc(CCNC(=O)NC(=O)c2ccc(N)cc2)cc1 ZINC000217515501 DD For-Sale Unstable CA2 15 51 COc1ccc(CCNC(=O)NC(=O)c2ccc(N)cc2)cc1 ZINC000217515501 DD For-Sale Unstable NQO2 25 40 COc1ccc(CCNC(=O)NC(=O)c2ccc(N)cc2)cc1 ZINC000217515501 DD For-Sale Unstable CA1 15 51 COc1ccc(CCNC(=O)NC(=O)c2ccc(N)cc2)cc1 ZINC000217515501 DD For-Sale Unstable MTNR1A 56 39 COc1ccc(CCNC(=O)NC(=O)c2ccc(N)cc2)cc1 ZINC000217515501 DD For-Sale Unstable MTNR1B 45 36 COc1ccc(CCNC(=O)NC(=O)c2ccc(N)cc2)cc1 ZINC000217515501 DD For-Sale Unstable CA12 15 51 COc1ccc(CCNC(=O)NC(=O)c2ccc(N)cc2)cc1 ZINC000217515501 DD For-Sale Unstable PTGDR 16 42 COc1ccc(CCNC(=O)NC(=O)c2ccc(N)cc2)cc1 ZINC000217515501 DD For-Sale Unstable CA9 25 51 COc1ccc(CCNC(=O)NC(=O)c2ccc(N)cc2)cc1 ZINC000217515501 DD For-Sale Unstable CYNT 18 41 COc1ccc(CCNC(=O)NC(=O)c2ccc(N)cc2)cc1 ZINC000217515501 DD For-Sale Unstable PROKR1 48 33 COc1ccc(CCNC(=O)NC(=O)c2ccc(N)cc2)cc1 ZINC000217515501 DD For-Sale Unstable A6YCJ1_9METZ 15 43 C[C@@H](C(=O)O)C1CC(NC(=O)OC(C)(C)C)C1 ZINC000217515511 BE For-Sale Unstable PAPA1_CARPA 41 33 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCCOC ZINC000217515534 ED In-Stock Unstable PLA2G4B 50 38 BrCc1cnc(N2CC[C@@H](N3CCOCC3)C2)nc1 ZINC000217515543 ED For-Sale Unstable L3MBTL3 30 43 O=C(Nc1ccc(F)cc1Cl)c1ccc(=O)[nH]n1 ZINC000217515564 CD For-Sale Anodyne PYGL 25 43 O=C(Nc1ccc(F)cc1Cl)c1ccc(=O)[nH]n1 ZINC000217515564 CD For-Sale Anodyne ALPL 53 32 COc1ccccc1OCC(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217515577 FF For-Sale Unstable NPY5R 44 60 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1cccc(F)c1 ZINC000217515599 FG For-Sale Unstable DRD4 44 35 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1cccc(F)c1 ZINC000217515599 FG For-Sale Unstable PLD2 52 38 CCOC(=O)c1ccccc1NC(=O)[C@@H]1C[C@@H]1c1ccccc1Cl ZINC000217515609 EI On-Demand Unstable KCNK2 0 40 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCCCOC ZINC000217515622 FE In-Stock Unstable PLA2G4B 49 37 BrCc1cnc(N2CC[C@H](N3CCOCC3)C2)nc1 ZINC000217515628 ED For-Sale Unstable L3MBTL3 30 43 COc1ccc(CCNC(=O)Nc2ccc(F)c(Cl)c2)cc1 ZINC000217515630 DH On-Demand Unstable CA2 17 46 COc1ccc(CCNC(=O)Nc2ccc(F)c(Cl)c2)cc1 ZINC000217515630 DH On-Demand Unstable BMP1 19 45 COc1ccc(CCNC(=O)Nc2ccc(F)c(Cl)c2)cc1 ZINC000217515630 DH On-Demand Unstable CA1 28 46 COc1ccc(CCNC(=O)Nc2ccc(F)c(Cl)c2)cc1 ZINC000217515630 DH On-Demand Unstable CTSL 17 40 COc1ccc(CCNC(=O)Nc2ccc(F)c(Cl)c2)cc1 ZINC000217515630 DH On-Demand Unstable CCR3 26 41 COc1ccc(CCNC(=O)Nc2ccc(F)c(Cl)c2)cc1 ZINC000217515630 DH On-Demand Unstable RAF1 61 46 COc1ccc(CCNC(=O)Nc2ccc(F)c(Cl)c2)cc1 ZINC000217515630 DH On-Demand Unstable KDR 19 42 COc1ccc(CCNC(=O)Nc2ccc(F)c(Cl)c2)cc1 ZINC000217515630 DH On-Demand Unstable MTNR1A 63 39 COc1ccc(CCNC(=O)Nc2ccc(F)c(Cl)c2)cc1 ZINC000217515630 DH On-Demand Unstable MTNR1B 55 40 COc1ccc(CCNC(=O)Nc2ccc(F)c(Cl)c2)cc1 ZINC000217515630 DH On-Demand Unstable EPHX2 23 45 COc1ccc(CCNC(=O)Nc2ccc(F)c(Cl)c2)cc1 ZINC000217515630 DH On-Demand Unstable CA12 24 45 COc1ccc(CCNC(=O)Nc2ccc(F)c(Cl)c2)cc1 ZINC000217515630 DH On-Demand Unstable PTGDR 22 45 COc1ccc(CCNC(=O)Nc2ccc(F)c(Cl)c2)cc1 ZINC000217515630 DH On-Demand Unstable CA9 26 45 COc1ccc(CCNC(=O)Nc2ccc(F)c(Cl)c2)cc1 ZINC000217515630 DH On-Demand Unstable MCHR1 23 43 COc1ccc(CCNC(=O)Nc2ccc(F)c(Cl)c2)cc1 ZINC000217515630 DH On-Demand Unstable TAAR1 16 46 COc1ccc(CCNC(=O)Nc2ccc(F)c(Cl)c2)cc1 ZINC000217515630 DH On-Demand Unstable NCE103 39 44 COc1ccc(CCNC(=O)Nc2ccc(F)c(Cl)c2)cc1 ZINC000217515630 DH On-Demand Unstable P96878_MYCTU 21 41 CC[S@](=O)CCN1C[C@@H](C)NC[C@@H]1c1ccccc1 ZINC000217515653 CD For-Sale Unstable CACNA1B 28 43 CCC[C@@H](C)NC(=O)CN1CCC[C@@H](N)C1 ZINC000217515664 BC For-Sale Unstable NOD1 48 31 CCOC(=O)c1ccccc1NC(=O)[C@H]1C[C@@H]1c1ccccc1Cl ZINC000217515685 EI On-Demand Unstable KCNK2 0 40 COc1cccc(OCC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217515700 FF For-Sale Unstable DRD4 40 31 COc1cccc(OCC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217515700 FF For-Sale Unstable NPY5R 48 61 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCc1ccccc1 ZINC000217515719 GG In-Stock Unstable PLA2G4B 58 35 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCc1ccccc1 ZINC000217515719 GG In-Stock Unstable CTRB_BOVIN 45 31 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCc1ccccc1 ZINC000217515719 GG In-Stock Unstable AKR1C3 15 44 CCN(CC)c1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217515748 EH For-Sale Unstable CA2 16 49 CCN(CC)c1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217515748 EH For-Sale Unstable ADRB1 24 41 CCN(CC)c1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217515748 EH For-Sale Unstable BMP1 23 52 CCN(CC)c1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217515748 EH For-Sale Unstable CA1 34 49 CCN(CC)c1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217515748 EH For-Sale Unstable MTNR1A 62 40 CCN(CC)c1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217515748 EH For-Sale Unstable MTNR1B 54 39 CCN(CC)c1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217515748 EH For-Sale Unstable NPY5R 16 42 CCN(CC)c1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217515748 EH For-Sale Unstable CA12 23 49 CCN(CC)c1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217515748 EH For-Sale Unstable PTGDR 15 45 CCN(CC)c1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217515748 EH For-Sale Unstable CA9 25 49 CCN(CC)c1ccc(NC(=O)NCCc2ccc(OC)cc2)cc1 ZINC000217515748 EH For-Sale Unstable NCE103 30 49 CCC[C@H](C)NC(=O)CN1CCC[C@@H](N)C1 ZINC000217515767 BC For-Sale Unstable NOD1 48 31 CCOC(=O)c1ccccc1NC(=O)[C@@H]1C[C@H]1c1ccccc1Cl ZINC000217515773 EI On-Demand Unstable KCNK2 0 40 O=C1OC2(CCN(C(=O)CSCc3ccccc3)CC2)c2ccccc21 ZINC000217515811 FH In-Stock Unstable SIGMAR1 15 49 O=C1OC2(CCN(C(=O)CSCc3ccccc3)CC2)c2ccccc21 ZINC000217515811 FH In-Stock Unstable NPY5R 43 51 CCOC(=O)c1ccccc1NC(=O)[C@H]1C[C@H]1c1ccccc1Cl ZINC000217515855 EI On-Demand Unstable KCNK2 0 40 C[C@@](O)(CNS(=O)(=O)c1cccc2nsnc12)c1cc2ccccc2s1 ZINC000217515862 HG In-Stock Unstable CCKAR 0 41 COc1ccc(CCNC(=O)N(CC(C)C)CC(C)C)cc1 ZINC000217515870 DH On-Demand Unstable ANPEP 16 42 COc1ccc(CCNC(=O)N(CC(C)C)CC(C)C)cc1 ZINC000217515870 DH On-Demand Unstable BMP1 44 40 COc1ccc(CCNC(=O)N(CC(C)C)CC(C)C)cc1 ZINC000217515870 DH On-Demand Unstable MMP16 0 42 COc1ccc(CCNC(=O)N(CC(C)C)CC(C)C)cc1 ZINC000217515870 DH On-Demand Unstable MTNR1A 60 43 COc1ccc(CCNC(=O)N(CC(C)C)CC(C)C)cc1 ZINC000217515870 DH On-Demand Unstable MTNR1B 50 37 COc1ccc(CCNC(=O)N(CC(C)C)CC(C)C)cc1 ZINC000217515870 DH On-Demand Unstable MMP2 17 42 COc1ccc(CCNC(=O)N(CC(C)C)CC(C)C)cc1 ZINC000217515870 DH On-Demand Unstable MMP8 18 42 COc1ccc(CCNC(=O)N(CC(C)C)CC(C)C)cc1 ZINC000217515870 DH On-Demand Unstable MMP9 20 41 COc1ccc(CCNC(=O)N(CC(C)C)CC(C)C)cc1 ZINC000217515870 DH On-Demand Unstable MMP12 25 42 COc1ccc(CCNC(=O)N(CC(C)C)CC(C)C)cc1 ZINC000217515870 DH On-Demand Unstable CA9 19 48 COc1ccc(CCNC(=O)N(CC(C)C)CC(C)C)cc1 ZINC000217515870 DH On-Demand Unstable MMP1 26 42 CCN(CC)C(=O)c1ccc2c(c1)CC[C@H](C)N2 ZINC000217515879 BF In-Stock Unstable OPRM1 25 42 CCN(CC)C(=O)c1ccc2c(c1)CC[C@H](C)N2 ZINC000217515879 BF In-Stock Unstable OPRD1 37 41 C[C@](O)(CNS(=O)(=O)c1cccc2nsnc12)c1cc2ccccc2s1 ZINC000217515912 HG In-Stock Unstable CCKAR 0 41 COC(=O)[C@@H](NC(=O)Cc1coc2ccc3ccc(OC)cc3c12)C(C)C ZINC000217515920 FG For-Sale Unstable NQO2 38 46 COC(=O)[C@@H](NC(=O)Cc1coc2ccc3ccc(OC)cc3c12)C(C)C ZINC000217515920 FG For-Sale Unstable MTNR1A 72 48 COC(=O)[C@@H](NC(=O)Cc1coc2ccc3ccc(OC)cc3c12)C(C)C ZINC000217515920 FG For-Sale Unstable MTNR1B 53 46 CCSc1ccccc1C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217515933 FI In-Stock Unstable NPY5R 36 51 CCN(CC)C(=O)c1ccc2c(c1)CC[C@@H](C)N2 ZINC000217515959 BF In-Stock Unstable OPRM1 25 42 CCN(CC)C(=O)c1ccc2c(c1)CC[C@@H](C)N2 ZINC000217515959 BF In-Stock Unstable OPRD1 37 41 COc1ccc(CCNC(=O)N2CCN(C=O)CC2)cc1 ZINC000217515971 CC For-Sale Unstable ADRB1 17 41 COc1ccc(CCNC(=O)N2CCN(C=O)CC2)cc1 ZINC000217515971 CC For-Sale Unstable ADRB3 15 41 COc1ccc(CCNC(=O)N2CCN(C=O)CC2)cc1 ZINC000217515971 CC For-Sale Unstable MMP13 30 41 COc1ccc(CCNC(=O)N2CCN(C=O)CC2)cc1 ZINC000217515971 CC For-Sale Unstable MTNR1A 68 39 COc1ccc(CCNC(=O)N2CCN(C=O)CC2)cc1 ZINC000217515971 CC For-Sale Unstable MTNR1B 63 39 COc1ccc(CCNC(=O)N2CCN(C=O)CC2)cc1 ZINC000217515971 CC For-Sale Unstable MMP3 33 52 COc1ccc(CCNC(=O)N2CCN(C=O)CC2)cc1 ZINC000217515971 CC For-Sale Unstable MMP9 31 52 COc1ccc(CCNC(=O)N2CCN(C=O)CC2)cc1 ZINC000217515971 CC For-Sale Unstable DPP7 15 41 COc1ccc(CCNC(=O)N2CCN(C=O)CC2)cc1 ZINC000217515971 CC For-Sale Unstable MMP7 30 52 COc1ccc(CCNC(=O)N2CCN(C=O)CC2)cc1 ZINC000217515971 CC For-Sale Unstable CA9 15 44 COc1ccc(CCNC(=O)N2CCN(C=O)CC2)cc1 ZINC000217515971 CC For-Sale Unstable MMP1 35 52 COc1ccc(CCNC(=O)N2CCN(C=O)CC2)cc1 ZINC000217515971 CC For-Sale Unstable GPR183 0 40 C[C@@H](CN1CCC[C@@H](N)C1)C(=O)O ZINC000217515972 AC For-Sale Unstable ACE 17 40 O=C1OC2(CCN(C(=O)CCSc3ccccc3)CC2)c2ccccc21 ZINC000217516021 FH For-Sale Unstable NPY5R 41 48 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccccc1 ZINC000217516027 GH In-Stock Unstable RARB 17 40 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccccc1 ZINC000217516027 GH In-Stock Unstable PLA2G4B 50 33 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccccc1 ZINC000217516027 GH In-Stock Unstable CTRB_BOVIN 54 32 CCN(CCNCc1cncn1C1CC1)C1CC1 ZINC000217516052 BD For-Sale Unstable CAMC 0 45 C[C@@H]1CCc2cc(C(=O)N3CCCC3)ccc2N1 ZINC000217516064 BF In-Stock Unstable L3MBTL1 0 45 C[C@@H]1CCc2cc(C(=O)N3CCCC3)ccc2N1 ZINC000217516064 BF In-Stock Unstable L3MBTL3 87 45 C[C@@H]1CCc2cc(C(=O)N3CCCC3)ccc2N1 ZINC000217516064 BF In-Stock Unstable MBTD1 0 41 C[C@@H]1CCc2cc(C(=O)N3CCCC3)ccc2N1 ZINC000217516064 BF In-Stock Unstable HPGD 44 38 C[C@@H]1CCc2cc(C(=O)N3CCCC3)ccc2N1 ZINC000217516064 BF In-Stock Unstable TP53BP1 0 42 C[C@H](CN1CCC[C@@H](N)C1)C(=O)O ZINC000217516066 AC For-Sale Unstable ACE 17 40 COc1ccc(CCNC(=O)Nc2cc(Cl)cc(Cl)c2)cc1 ZINC000217516082 EI On-Demand Unstable BMP1 25 46 COc1ccc(CCNC(=O)Nc2cc(Cl)cc(Cl)c2)cc1 ZINC000217516082 EI On-Demand Unstable CA1 21 46 COc1ccc(CCNC(=O)Nc2cc(Cl)cc(Cl)c2)cc1 ZINC000217516082 EI On-Demand Unstable TRPV1 0 50 COc1ccc(CCNC(=O)Nc2cc(Cl)cc(Cl)c2)cc1 ZINC000217516082 EI On-Demand Unstable RAF1 48 43 COc1ccc(CCNC(=O)Nc2cc(Cl)cc(Cl)c2)cc1 ZINC000217516082 EI On-Demand Unstable MTNR1A 94 43 COc1ccc(CCNC(=O)Nc2cc(Cl)cc(Cl)c2)cc1 ZINC000217516082 EI On-Demand Unstable MTNR1B 77 39 COc1ccc(CCNC(=O)Nc2cc(Cl)cc(Cl)c2)cc1 ZINC000217516082 EI On-Demand Unstable CA12 17 46 COc1ccc(CCNC(=O)Nc2cc(Cl)cc(Cl)c2)cc1 ZINC000217516082 EI On-Demand Unstable PDGFRA 19 42 COc1ccc(CCNC(=O)Nc2cc(Cl)cc(Cl)c2)cc1 ZINC000217516082 EI On-Demand Unstable PTGDR 24 46 COc1ccc(CCNC(=O)Nc2cc(Cl)cc(Cl)c2)cc1 ZINC000217516082 EI On-Demand Unstable CA9 20 46 COc1ccc(CCNC(=O)Nc2cc(Cl)cc(Cl)c2)cc1 ZINC000217516082 EI On-Demand Unstable U38 0 40 COc1ccc(CCNC(=O)Nc2cc(Cl)cc(Cl)c2)cc1 ZINC000217516082 EI On-Demand Unstable MCHR1 15 44 COc1ccc(CCNC(=O)Nc2cc(Cl)cc(Cl)c2)cc1 ZINC000217516082 EI On-Demand Unstable Q8MMZ8_EIMTE 37 43 COc1ccc(CCNC(=O)Nc2cc(Cl)cc(Cl)c2)cc1 ZINC000217516082 EI On-Demand Unstable NCE103 37 45 COc1ccc(CCNC(=O)Nc2cc(Cl)cc(Cl)c2)cc1 ZINC000217516082 EI On-Demand Unstable PROKR1 60 34 COc1ccc(CCNC(=O)Nc2cc(Cl)cc(Cl)c2)cc1 ZINC000217516082 EI On-Demand Unstable P96878_MYCTU 15 45 COc1ccc(CCNC(=O)Nc2cc(Cl)cc(Cl)c2)cc1 ZINC000217516082 EI On-Demand Unstable CAN2 0 45 BrCc1ccc(N2CC[C@@H](N3CCOCC3)C2)cc1 ZINC000217516114 EE For-Sale Unstable L3MBTL3 50 56 O=C1OC2(CCN(C(=O)CSc3ccc(F)cc3)CC2)c2ccccc21 ZINC000217516135 FH In-Stock Unstable NPY5R 44 55 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)cc1 ZINC000217516145 HH In-Stock Unstable TBXA2R 17 41 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)cc1 ZINC000217516145 HH In-Stock Unstable TBXAS1 15 41 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)cc1 ZINC000217516145 HH In-Stock Unstable PLA2G4A 44 40 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)cc1 ZINC000217516145 HH In-Stock Unstable PLA2G4B 60 38 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)cc1 ZINC000217516145 HH In-Stock Unstable ALOX15 46 39 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)cc1 ZINC000217516145 HH In-Stock Unstable PTGDR 40 40 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)cc1 ZINC000217516145 HH In-Stock Unstable IAP 0 41 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)cc1 ZINC000217516145 HH In-Stock Unstable AKR1C3 21 45 C[C@H]1CCc2cc(C(=O)N3CCCC3)ccc2N1 ZINC000217516149 BF In-Stock Unstable L3MBTL1 0 45 C[C@H]1CCc2cc(C(=O)N3CCCC3)ccc2N1 ZINC000217516149 BF In-Stock Unstable L3MBTL3 87 45 C[C@H]1CCc2cc(C(=O)N3CCCC3)ccc2N1 ZINC000217516149 BF In-Stock Unstable MBTD1 0 41 C[C@H]1CCc2cc(C(=O)N3CCCC3)ccc2N1 ZINC000217516149 BF In-Stock Unstable HPGD 44 38 C[C@H]1CCc2cc(C(=O)N3CCCC3)ccc2N1 ZINC000217516149 BF In-Stock Unstable TP53BP1 0 42 CC(C)CCC[C@@H](C)NC(=O)CN1CCC[C@@H](N)C1 ZINC000217516206 CD On-Demand Unstable BIRC2 40 33 COc1ccc(CCNC(=O)N(CCN)C(C)=O)cc1 ZINC000217516207 CC For-Sale Unstable BMP1 18 40 COc1ccc(CCNC(=O)N(CCN)C(C)=O)cc1 ZINC000217516207 CC For-Sale Unstable MTNR1A 77 38 COc1ccc(CCNC(=O)N(CCN)C(C)=O)cc1 ZINC000217516207 CC For-Sale Unstable MTNR1B 61 38 COc1ccc(CCNC(=O)N(CCN)C(C)=O)cc1 ZINC000217516207 CC For-Sale Unstable CA9 21 48 COc1ccc(CCNC(=O)N(CCN)C(C)=O)cc1 ZINC000217516207 CC For-Sale Unstable PROKR1 53 33 COc1ccc([C@@H](CN)N2CCCO[C@@H](C)C2)cc1OC ZINC000217516212 CD For-Sale Unstable UTS2R 35 40 BrCc1ccc(N2CC[C@H](N3CCOCC3)C2)cc1 ZINC000217516213 EE For-Sale Unstable L3MBTL3 50 56 C[C@@](O)(CNS(=O)(=O)c1ccc(OCC(N)=O)cc1)c1cc2ccccc2s1 ZINC000217516217 HD In-Stock Unstable PRTN3 52 32 O=C(Nc1c(F)cccc1F)c1cc(Br)ccc1I ZINC000217516225 IJ On-Demand Anodyne Q25615_ONCVO 39 40 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)c(OC)c1 ZINC000217516244 JH In-Stock Unstable PLA2G4B 36 41 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)c(OC)c1 ZINC000217516244 JH In-Stock Unstable PTGDR 29 44 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)c(OC)c1 ZINC000217516244 JH In-Stock Unstable IAP 0 42 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)c(OC)c1 ZINC000217516244 JH In-Stock Unstable PTGDR2 18 43 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)c(OC)c1 ZINC000217516244 JH In-Stock Unstable SCMU_MYCTU 0 49 O=C1OC2(CCN(C(=O)COc3ccc(Cl)cc3)CC2)c2ccccc21 ZINC000217516249 FG For-Sale Unstable AVPR1A 15 52 O=C1OC2(CCN(C(=O)COc3ccc(Cl)cc3)CC2)c2ccccc21 ZINC000217516249 FG For-Sale Unstable NPY5R 43 56 C[C@@H]1CCc2cc(C(=O)NC3CC3)ccc2N1 ZINC000217516252 BE In-Stock Unstable MAPK14 49 44 C[C@@H]1CCc2cc(C(=O)NC3CC3)ccc2N1 ZINC000217516252 BE In-Stock Unstable MAPK13 52 38 CC(=O)CCc1cn(C)cn1 ZINC000217516261 AC For-Sale Unstable CPB2 16 43 CC(C)CCC[C@H](C)NC(=O)CN1CCC[C@@H](N)C1 ZINC000217516289 CD On-Demand Unstable BIRC2 40 33 C[C@](O)(CNS(=O)(=O)c1ccc(OCC(N)=O)cc1)c1cc2ccccc2s1 ZINC000217516297 HD In-Stock Unstable PRTN3 52 32 CCN(C(=O)NCCc1ccc(OC)cc1)C(C)(C)C ZINC000217516321 CG For-Sale Unstable CTSL 16 43 CCN(C(=O)NCCc1ccc(OC)cc1)C(C)(C)C ZINC000217516321 CG For-Sale Unstable MMP16 0 42 CCN(C(=O)NCCc1ccc(OC)cc1)C(C)(C)C ZINC000217516321 CG For-Sale Unstable MTNR1A 85 39 CCN(C(=O)NCCc1ccc(OC)cc1)C(C)(C)C ZINC000217516321 CG For-Sale Unstable MTNR1B 68 38 CCN(C(=O)NCCc1ccc(OC)cc1)C(C)(C)C ZINC000217516321 CG For-Sale Unstable MMP9 18 42 CCN(C(=O)NCCc1ccc(OC)cc1)C(C)(C)C ZINC000217516321 CG For-Sale Unstable PTGDR 23 41 CCN(C(=O)NCCc1ccc(OC)cc1)C(C)(C)C ZINC000217516321 CG For-Sale Unstable CA9 18 47 CCN(C(=O)NCCc1ccc(OC)cc1)C(C)(C)C ZINC000217516321 CG For-Sale Unstable MMP1 21 42 CCN(C(=O)NCCc1ccc(OC)cc1)C(C)(C)C ZINC000217516321 CG For-Sale Unstable PROKR1 60 34 N#Cc1cccc(C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)c1 ZINC000217516327 FG For-Sale Unstable DRD4 44 35 C[C@H]1CCc2cc(C(=O)NC3CC3)ccc2N1 ZINC000217516338 BE In-Stock Unstable MAPK14 49 44 C[C@H]1CCc2cc(C(=O)NC3CC3)ccc2N1 ZINC000217516338 BE In-Stock Unstable MAPK13 52 38 O=S(=O)(Cl)CCc1cc2ccncc2o1 ZINC000217516353 BD For-Sale Unstable NAMPT 19 40 COc1ccc(Cl)cc1C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217516376 FH For-Sale Unstable AVPR1A 27 65 COc1ccc(Cl)cc1C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217516376 FH For-Sale Unstable NPY5R 38 53 CCO[C@@H]1C[C@@H](Nc2nc3ccccc3o2)C1(C)C ZINC000217516396 CG For-Sale Unstable SSTR5 50 45 COc1ccc(CCNC(=O)Nc2ccc(-c3nc4ccc(C)cc4s3)cc2)cc1 ZINC000217516438 HK For-Sale Unstable CA2 17 40 COc1ccc(CCNC(=O)Nc2ccc(-c3nc4ccc(C)cc4s3)cc2)cc1 ZINC000217516438 HK For-Sale Unstable LDHA 44 46 COc1ccc(CCNC(=O)Nc2ccc(-c3nc4ccc(C)cc4s3)cc2)cc1 ZINC000217516438 HK For-Sale Unstable CA1 15 40 COc1ccc(CCNC(=O)Nc2ccc(-c3nc4ccc(C)cc4s3)cc2)cc1 ZINC000217516438 HK For-Sale Unstable CSNK1D 35 44 COc1ccc(CCNC(=O)Nc2ccc(-c3nc4ccc(C)cc4s3)cc2)cc1 ZINC000217516438 HK For-Sale Unstable PIK3CA 0 44 COc1ccc(CCNC(=O)Nc2ccc(-c3nc4ccc(C)cc4s3)cc2)cc1 ZINC000217516438 HK For-Sale Unstable APP 30 52 COc1ccc(CCNC(=O)Nc2ccc(-c3nc4ccc(C)cc4s3)cc2)cc1 ZINC000217516438 HK For-Sale Unstable RAF1 44 42 COc1ccc(CCNC(=O)Nc2ccc(-c3nc4ccc(C)cc4s3)cc2)cc1 ZINC000217516438 HK For-Sale Unstable ROCK2 20 51 COc1ccc(CCNC(=O)Nc2ccc(-c3nc4ccc(C)cc4s3)cc2)cc1 ZINC000217516438 HK For-Sale Unstable PIK3CG 17 44 COc1ccc(CCNC(=O)Nc2ccc(-c3nc4ccc(C)cc4s3)cc2)cc1 ZINC000217516438 HK For-Sale Unstable PTGDR 25 41 COc1ccc(CCNC(=O)Nc2ccc(-c3nc4ccc(C)cc4s3)cc2)cc1 ZINC000217516438 HK For-Sale Unstable Q8MMZ8_EIMTE 41 42 COc1ccc(CCNC(=O)Nc2ccc(-c3nc4ccc(C)cc4s3)cc2)cc1 ZINC000217516438 HK For-Sale Unstable LUCI_PHOPE 36 47 COc1ccc(CCNC(=O)Nc2ccc(-c3nc4ccc(C)cc4s3)cc2)cc1 ZINC000217516438 HK For-Sale Unstable PRMT3 62 35 COc1ccc(CCNC(=O)Nc2ccc(-c3nc4ccc(C)cc4s3)cc2)cc1 ZINC000217516438 HK For-Sale Unstable PORCN 0 42 COc1ccc(CCNC(=O)Nc2ccc(-c3nc4ccc(C)cc4s3)cc2)cc1 ZINC000217516438 HK For-Sale Unstable ETHR 20 49 CC(C)(C)OC(=O)CCCCC[C@@H](N)C(=O)O ZINC000217516457 BD For-Sale Unstable GRIA3 15 41 CC(C)(C)OC(=O)CCCCC[C@@H](N)C(=O)O ZINC000217516457 BD For-Sale Unstable GRM8 25 41 CC(C)(C)OC(=O)CCCCC[C@@H](N)C(=O)O ZINC000217516457 BD For-Sale Unstable GRIK3 36 41 CC(C)(C)OC(=O)CCCCC[C@@H](N)C(=O)O ZINC000217516457 BD For-Sale Unstable GRIK5 20 41 CC(C)(C)OC(=O)CCCCC[C@@H](N)C(=O)O ZINC000217516457 BD For-Sale Unstable GRIK2 26 41 CC(C)(C)OC(=O)CCCCC[C@@H](N)C(=O)O ZINC000217516457 BD For-Sale Unstable BHMT 60 41 CC(C)(C)OC(=O)CCCCC[C@@H](N)C(=O)O ZINC000217516457 BD For-Sale Unstable NOD1 81 41 C[C@@H]1CCc2cc(C(=O)N3CCOCC3)ccc2N1 ZINC000217516461 CD In-Stock Unstable L3MBTL3 61 37 CCO[C@H]1C[C@@H](Nc2nc3ccccc3o2)C1(C)C ZINC000217516468 CG For-Sale Unstable SSTR5 50 45 O=C1OC2(CCN(C(=O)c3ccc(C(F)(F)F)cc3)CC2)c2ccccc21 ZINC000217516476 GI For-Sale Unstable NPY5R 41 52 O=C1OC2(CCN(C(=O)c3ccc(C(F)(F)F)cc3)CC2)c2ccccc21 ZINC000217516476 GI For-Sale Unstable MLYCD 18 40 O=C1OC2(CCN(C(=O)c3ccc(C(F)(F)F)cc3)CC2)c2ccccc21 ZINC000217516476 GI For-Sale Unstable TRPM8 21 41 C[C@H]1CCc2cc(C(=O)N3CCOCC3)ccc2N1 ZINC000217516540 CD In-Stock Unstable L3MBTL1 0 43 C[C@H]1CCc2cc(C(=O)N3CCOCC3)ccc2N1 ZINC000217516540 CD In-Stock Unstable L3MBTL3 61 37 CCO[C@@H]1C[C@H](Nc2nc3ccccc3o2)C1(C)C ZINC000217516542 CG For-Sale Unstable SSTR5 50 45 COc1ccc(CCNC(=O)NC(=O)C2CCNCC2)cc1 ZINC000217516549 DD For-Sale Unstable NQO2 36 45 COc1ccc(CCNC(=O)NC(=O)C2CCNCC2)cc1 ZINC000217516549 DD For-Sale Unstable MTNR1A 104 47 COc1ccc(CCNC(=O)NC(=O)C2CCNCC2)cc1 ZINC000217516549 DD For-Sale Unstable MTNR1B 86 40 COc1ccc(CCNC(=O)NC(=O)C2CCNCC2)cc1 ZINC000217516549 DD For-Sale Unstable MMP3 23 42 COc1ccc(CCNC(=O)NC(=O)C2CCNCC2)cc1 ZINC000217516549 DD For-Sale Unstable MMP9 17 42 COc1ccc(CCNC(=O)NC(=O)C2CCNCC2)cc1 ZINC000217516549 DD For-Sale Unstable MMP7 28 42 COc1ccc(CCNC(=O)NC(=O)C2CCNCC2)cc1 ZINC000217516549 DD For-Sale Unstable MMP1 21 42 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1Br ZINC000217516552 EI For-Sale Unstable UL26 15 41 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1Br ZINC000217516552 EI For-Sale Unstable U53 0 41 C[C@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1Br ZINC000217516552 EI For-Sale Unstable SCAF_EBVB9 19 41 O=C1OC2(CCN(C(=O)c3ccccc3C(F)(F)F)CC2)c2ccccc21 ZINC000217516591 GI For-Sale Unstable AVPR1A 16 54 O=C1OC2(CCN(C(=O)c3ccccc3C(F)(F)F)CC2)c2ccccc21 ZINC000217516591 GI For-Sale Unstable NPY5R 42 60 O=C1OC2(CCN(C(=O)c3ccccc3C(F)(F)F)CC2)c2ccccc21 ZINC000217516591 GI For-Sale Unstable RBP4 57 39 O=C1OC2(CCN(C(=O)c3ccccc3C(F)(F)F)CC2)c2ccccc21 ZINC000217516591 GI For-Sale Unstable SCD1 21 43 O=C1OC2(CCN(C(=O)c3ccccc3C(F)(F)F)CC2)c2ccccc21 ZINC000217516591 GI For-Sale Unstable SCD 19 42 CCO[C@H]1C[C@H](Nc2nc3ccccc3o2)C1(C)C ZINC000217516619 CG For-Sale Unstable SSTR5 50 45 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1N1CCCC1 ZINC000217516628 EE In-Stock Unstable KCNQ2 64 33 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1Br ZINC000217516648 EI For-Sale Unstable UL26 15 41 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1Br ZINC000217516648 EI For-Sale Unstable U53 0 41 C[C@@H](O)c1ccccc1NC(=O)/C=C\c1ccccc1Br ZINC000217516648 EI For-Sale Unstable SCAF_EBVB9 19 41 O=C(CCc1ccccc1)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217516664 FH For-Sale Unstable FABP4 45 34 O=C(CCc1ccccc1)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217516664 FH For-Sale Unstable VIPR1 22 40 COc1ccc(CCNC(=O)Nc2ccc(C)cc2O)cc1 ZINC000217516681 DG For-Sale Unstable BMP1 23 40 COc1ccc(CCNC(=O)Nc2ccc(C)cc2O)cc1 ZINC000217516681 DG For-Sale Unstable CA1 17 46 COc1ccc(CCNC(=O)Nc2ccc(C)cc2O)cc1 ZINC000217516681 DG For-Sale Unstable TRPV1 23 53 COc1ccc(CCNC(=O)Nc2ccc(C)cc2O)cc1 ZINC000217516681 DG For-Sale Unstable RAF1 39 42 COc1ccc(CCNC(=O)Nc2ccc(C)cc2O)cc1 ZINC000217516681 DG For-Sale Unstable MTNR1A 78 43 COc1ccc(CCNC(=O)Nc2ccc(C)cc2O)cc1 ZINC000217516681 DG For-Sale Unstable MTNR1B 58 40 COc1ccc(CCNC(=O)Nc2ccc(C)cc2O)cc1 ZINC000217516681 DG For-Sale Unstable CA12 15 46 COc1ccc(CCNC(=O)Nc2ccc(C)cc2O)cc1 ZINC000217516681 DG For-Sale Unstable PTGDR 20 41 COc1ccc(CCNC(=O)Nc2ccc(C)cc2O)cc1 ZINC000217516681 DG For-Sale Unstable CA9 22 46 COc1ccc(CCNC(=O)Nc2ccc(C)cc2O)cc1 ZINC000217516681 DG For-Sale Unstable Q8MMZ8_EIMTE 32 41 COc1ccc(CCNC(=O)Nc2ccc(C)cc2O)cc1 ZINC000217516681 DG For-Sale Unstable NCE103 24 40 COc1ccc(CCNC(=O)Nc2ccc(C)cc2O)cc1 ZINC000217516681 DG For-Sale Unstable CAN2 0 40 O=C1OC2(CCN(C(=O)c3cc(=O)c4ccccc4o3)CC2)c2ccccc21 ZINC000217516706 GG In-Stock Unstable NPY5R 37 47 O=C1OC2(CCN(C(=O)c3cc(=O)c4ccccc4o3)CC2)c2ccccc21 ZINC000217516706 GG In-Stock Unstable TNKS 30 43 CC[S@](=O)CCN1C[C@@H](Cc2ccccc2)NC[C@@H]1C ZINC000217516717 CD For-Sale Unstable CACNA1B 22 40 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1N1CCCCC1 ZINC000217516749 FF In-Stock Unstable KCNQ2 49 33 Cc1cccc(/C=C\C(=O)Nc2ccccc2[C@@H](C)O)c1 ZINC000217516752 CH For-Sale Unstable LTB4R 0 40 Cc1cccc(/C=C\C(=O)Nc2ccccc2[C@@H](C)O)c1 ZINC000217516752 CH For-Sale Unstable HDAC8 49 42 Cc1cccc(/C=C\C(=O)Nc2ccccc2[C@@H](C)O)c1 ZINC000217516752 CH For-Sale Unstable MMP2 24 56 Cc1cccc(/C=C\C(=O)Nc2ccccc2[C@@H](C)O)c1 ZINC000217516752 CH For-Sale Unstable HDAC1 19 40 Cc1cccc(/C=C\C(=O)Nc2ccccc2[C@@H](C)O)c1 ZINC000217516752 CH For-Sale Unstable HDAC6 34 42 Cc1cccc(/C=C\C(=O)Nc2ccccc2[C@@H](C)O)c1 ZINC000217516752 CH For-Sale Unstable MMP9 22 56 Cc1cccc(/C=C\C(=O)Nc2ccccc2[C@@H](C)O)c1 ZINC000217516752 CH For-Sale Unstable MMP1 27 56 Cc1cccc(/C=C\C(=O)Nc2ccccc2[C@@H](C)O)c1 ZINC000217516752 CH For-Sale Unstable TRPM8 24 60 O=C(CS(=O)(=O)Cl)c1cccc(F)c1 ZINC000217516780 BD In-Stock Unstable KMO 0 51 COc1ccc(CCNC(=O)Nc2ccc(Cl)cc2C(F)(F)F)cc1 ZINC000217516788 FJ For-Sale Unstable TRPV1 25 49 COc1ccc(CCNC(=O)Nc2ccc(Cl)cc2C(F)(F)F)cc1 ZINC000217516788 FJ For-Sale Unstable RAF1 61 44 COc1ccc(CCNC(=O)Nc2ccc(Cl)cc2C(F)(F)F)cc1 ZINC000217516788 FJ For-Sale Unstable MTNR1A 53 40 COc1ccc(CCNC(=O)Nc2ccc(Cl)cc2C(F)(F)F)cc1 ZINC000217516788 FJ For-Sale Unstable MTNR1B 40 37 COc1ccc(CCNC(=O)Nc2ccc(Cl)cc2C(F)(F)F)cc1 ZINC000217516788 FJ For-Sale Unstable CA9 16 41 COc1ccc(CCNC(=O)Nc2ccc(Cl)cc2C(F)(F)F)cc1 ZINC000217516788 FJ For-Sale Unstable Q8MMZ8_EIMTE 59 51 O=C1OC2(CCN(C(=O)c3cc4ccccc4oc3=O)CC2)c2ccccc21 ZINC000217516818 GG For-Sale Unstable AVPR1A 16 54 O=C1OC2(CCN(C(=O)c3cc4ccccc4oc3=O)CC2)c2ccccc21 ZINC000217516818 GG For-Sale Unstable NPY5R 44 51 Cc1cccc(/C=C\C(=O)Nc2ccccc2[C@H](C)O)c1 ZINC000217516835 CH For-Sale Unstable LTB4R 0 40 Cc1cccc(/C=C\C(=O)Nc2ccccc2[C@H](C)O)c1 ZINC000217516835 CH For-Sale Unstable HDAC8 49 42 Cc1cccc(/C=C\C(=O)Nc2ccccc2[C@H](C)O)c1 ZINC000217516835 CH For-Sale Unstable MMP2 24 56 Cc1cccc(/C=C\C(=O)Nc2ccccc2[C@H](C)O)c1 ZINC000217516835 CH For-Sale Unstable HDAC1 19 40 Cc1cccc(/C=C\C(=O)Nc2ccccc2[C@H](C)O)c1 ZINC000217516835 CH For-Sale Unstable HDAC6 34 42 Cc1cccc(/C=C\C(=O)Nc2ccccc2[C@H](C)O)c1 ZINC000217516835 CH For-Sale Unstable MMP9 22 56 Cc1cccc(/C=C\C(=O)Nc2ccccc2[C@H](C)O)c1 ZINC000217516835 CH For-Sale Unstable MMP1 27 56 Cc1cccc(/C=C\C(=O)Nc2ccccc2[C@H](C)O)c1 ZINC000217516835 CH For-Sale Unstable TRPM8 24 60 CC(C)(C)OC(=O)N1CC[C@@H](CNCc2ccc(Cl)cc2Cl)C1 ZINC000217516881 FI For-Sale Unstable MC4R 42 40 CC(C)(C)OC(=O)N1CC[C@@H](CNCc2ccc(Cl)cc2Cl)C1 ZINC000217516881 FI For-Sale Unstable P2RX7 40 42 CC(C)(C)OC(=O)N1CC[C@@H](CNCc2ccc(Cl)cc2Cl)C1 ZINC000217516881 FI For-Sale Unstable EPHX2 27 50 CC(C)(C)OC(=O)N1CC[C@@H](CNCc2ccc(Cl)cc2Cl)C1 ZINC000217516881 FI For-Sale Unstable CACNA1I 61 39 CC(C)(C)OC(=O)N1CC[C@@H](CNCc2ccc(Cl)cc2Cl)C1 ZINC000217516881 FI For-Sale Unstable GPR119 42 43 O=C(CS(=O)(=O)Cl)c1ccccc1Cl ZINC000217516888 CE In-Stock Unstable ECR 48 38 COc1ccc(CCNC(=O)Nc2c(C)cc(C)cc2Cl)cc1 ZINC000217516902 EI On-Demand Unstable RAF1 38 44 COc1ccc(CCNC(=O)Nc2c(C)cc(C)cc2Cl)cc1 ZINC000217516902 EI On-Demand Unstable MTNR1A 57 39 COc1ccc(CCNC(=O)Nc2c(C)cc(C)cc2Cl)cc1 ZINC000217516902 EI On-Demand Unstable MTNR1B 44 37 COc1ccc(CCNC(=O)Nc2c(C)cc(C)cc2Cl)cc1 ZINC000217516902 EI On-Demand Unstable CA9 16 42 COc1ccc(CCNC(=O)Nc2c(C)cc(C)cc2Cl)cc1 ZINC000217516902 EI On-Demand Unstable Q8MMZ8_EIMTE 27 44 COc1ccc(CCNC(=O)Nc2c(C)cc(C)cc2Cl)cc1 ZINC000217516902 EI On-Demand Unstable NCE103 25 41 COc1ccc(CCNC(=O)Nc2c(C)cc(C)cc2Cl)cc1 ZINC000217516902 EI On-Demand Unstable FFAR4 30 40 COc1ccc(CCNC(=O)Nc2c(C)cc(C)cc2Cl)cc1 ZINC000217516902 EI On-Demand Unstable ACAT 0 43 COc1ccc(CCNC(=O)Nc2c(C)cc(C)cc2Cl)cc1 ZINC000217516902 EI On-Demand Unstable CAN2 0 41 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCCCOCC ZINC000217516931 FF In-Stock Unstable PLA2G4B 50 36 COc1cccc2cc(C(=O)N3CCC4(CC3)OC(=O)c3ccccc34)oc12 ZINC000217516940 GH For-Sale Unstable NPY5R 34 52 COc1ccc(S(=O)(=O)Nc2ncc(Cc3cccc(C(F)(F)F)c3)s2)cc1[N+](=O)[O-] ZINC000217516947 JI On-Demand Unstable SCN9A 0 42 COc1ccc(S(=O)(=O)Nc2ncc(Cc3cccc(C(F)(F)F)c3)s2)cc1[N+](=O)[O-] ZINC000217516947 JI On-Demand Unstable SCD1 38 44 COc1ccc(S(=O)(=O)Nc2ncc(Cc3cccc(C(F)(F)F)c3)s2)cc1[N+](=O)[O-] ZINC000217516947 JI On-Demand Unstable SCD 40 53 Cc1ccc(C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc1C ZINC000217516976 FH For-Sale Unstable DRD4 41 32 Cc1ccc(C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc1C ZINC000217516976 FH For-Sale Unstable PLD2 41 32 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCCCOC(C)C ZINC000217517004 GG In-Stock Unstable PLA2G4B 43 36 C[C@@H](NC(=O)CN1CCC[C@@H](N)C1)c1cccs1 ZINC000217517006 CD On-Demand Unstable BIRC2 41 33 COc1ccc(CCNC(=O)Nc2c(Cl)cccc2Cl)cc1 ZINC000217517036 EI For-Sale Unstable DRD4 43 34 COc1ccc(CCNC(=O)Nc2c(Cl)cccc2Cl)cc1 ZINC000217517036 EI For-Sale Unstable BMP1 31 44 COc1ccc(CCNC(=O)Nc2c(Cl)cccc2Cl)cc1 ZINC000217517036 EI For-Sale Unstable NQO2 31 42 COc1ccc(CCNC(=O)Nc2c(Cl)cccc2Cl)cc1 ZINC000217517036 EI For-Sale Unstable TRPV1 0 56 COc1ccc(CCNC(=O)Nc2c(Cl)cccc2Cl)cc1 ZINC000217517036 EI For-Sale Unstable RAF1 41 41 COc1ccc(CCNC(=O)Nc2c(Cl)cccc2Cl)cc1 ZINC000217517036 EI For-Sale Unstable MTNR1A 100 45 COc1ccc(CCNC(=O)Nc2c(Cl)cccc2Cl)cc1 ZINC000217517036 EI For-Sale Unstable MTNR1B 86 42 COc1ccc(CCNC(=O)Nc2c(Cl)cccc2Cl)cc1 ZINC000217517036 EI For-Sale Unstable PTGDR 23 44 COc1ccc(CCNC(=O)Nc2c(Cl)cccc2Cl)cc1 ZINC000217517036 EI For-Sale Unstable CA9 22 46 COc1ccc(CCNC(=O)Nc2c(Cl)cccc2Cl)cc1 ZINC000217517036 EI For-Sale Unstable Q8MMZ8_EIMTE 30 41 COc1ccc(CCNC(=O)Nc2c(Cl)cccc2Cl)cc1 ZINC000217517036 EI For-Sale Unstable NCE103 30 47 COc1ccc(CCNC(=O)Nc2c(Cl)cccc2Cl)cc1 ZINC000217517036 EI For-Sale Unstable PROKR1 60 33 COc1ccc(CCNC(=O)Nc2c(Cl)cccc2Cl)cc1 ZINC000217517036 EI For-Sale Unstable ACAT 0 50 COc1ccc(CCNC(=O)Nc2c(Cl)cccc2Cl)cc1 ZINC000217517036 EI For-Sale Unstable CAN2 0 47 O=S(=O)(Nc1ncc(Cc2cccc(C(F)(F)F)c2)s1)c1ccccc1Br ZINC000217517040 JK On-Demand Unstable SCD1 31 47 O=S(=O)(Nc1ncc(Cc2cccc(C(F)(F)F)c2)s1)c1ccccc1Br ZINC000217517040 JK On-Demand Unstable SCD 29 47 O=C1OC2(CCN(C(=O)Cn3c(=O)oc4ccccc43)CC2)c2ccccc21 ZINC000217517041 GE In-Stock Unstable NPY5R 32 44 O=C(CS(=O)(=O)Cl)c1cccc(Cl)c1 ZINC000217517044 CE In-Stock Unstable KMO 0 54 C[C@H](NC(=O)CN1CCC[C@@H](N)C1)c1cccs1 ZINC000217517077 CD On-Demand Unstable BIRC2 41 33 CC(C)CNC(=O)c1cc(I)ccc1O ZINC000217517110 DE On-Demand Unstable F3 60 34 CCCCCNc1ccc(C(=O)O)cc1S(=O)(=O)NCCCCC ZINC000217517134 FG In-Stock Unstable PLA2G4B 44 37 Cc1ccc(S(=O)(=O)Nc2ncc(Cc3cccc(C(F)(F)F)c3)s2)cc1[N+](=O)[O-] ZINC000217517147 JJ On-Demand Unstable SCD1 25 45 Cc1ccc(S(=O)(=O)Nc2ncc(Cc3cccc(C(F)(F)F)c3)s2)cc1[N+](=O)[O-] ZINC000217517147 JJ On-Demand Unstable SCD 26 45 Cc1cccc(C(=O)CS(=O)(=O)Cl)c1 ZINC000217517152 BD In-Stock Unstable KCNK3 48 44 Cc1cccc(C(=O)CS(=O)(=O)Cl)c1 ZINC000217517152 BD In-Stock Unstable KCNK9 48 44 CCN(CC)c1ccc(NC(=O)NCCc2ccc(OC)cc2)c(C)c1 ZINC000217517153 FI For-Sale Unstable RAF1 37 41 CCN(CC)c1ccc(NC(=O)NCCc2ccc(OC)cc2)c(C)c1 ZINC000217517153 FI For-Sale Unstable MTNR1A 60 41 CCN(CC)c1ccc(NC(=O)NCCc2ccc(OC)cc2)c(C)c1 ZINC000217517153 FI For-Sale Unstable MTNR1B 43 36 CCCCOc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217517154 GI For-Sale Unstable AVPR1A 22 48 CCCCOc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217517154 GI For-Sale Unstable PLA2G4B 73 37 CCCCOc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217517154 GI For-Sale Unstable NPY5R 38 48 COc1ccc(C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc1 ZINC000217517175 FG For-Sale Unstable DRD4 47 37 COc1ccc(C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc1 ZINC000217517175 FG For-Sale Unstable GCGR 45 39 COc1ccc(C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc1 ZINC000217517175 FG For-Sale Unstable BCHE 40 35 COc1ccc(C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc1 ZINC000217517175 FG For-Sale Unstable GIPR 52 37 C[C@@H](NC(=O)CN1CCC[C@@H](N)C1)c1ccco1 ZINC000217517176 CC For-Sale Unstable BIRC2 41 33 Cc1nn(C)c(C)c1S(=O)(=O)Nc1ncc(Cc2cccc(C(F)(F)F)c2)s1 ZINC000217517251 IH On-Demand Unstable SCD1 29 46 Cc1nn(C)c(C)c1S(=O)(=O)Nc1ncc(Cc2cccc(C(F)(F)F)c2)s1 ZINC000217517251 IH On-Demand Unstable SCD 31 46 COc1ccc(CCNC(=O)Nc2cc(C)c(Cl)cc2OC)cc1 ZINC000217517252 EI On-Demand Unstable TRPV1 34 50 COc1ccc(CCNC(=O)Nc2cc(C)c(Cl)cc2OC)cc1 ZINC000217517252 EI On-Demand Unstable RAF1 54 67 COc1ccc(CCNC(=O)Nc2cc(C)c(Cl)cc2OC)cc1 ZINC000217517252 EI On-Demand Unstable FLT1 18 40 COc1ccc(CCNC(=O)Nc2cc(C)c(Cl)cc2OC)cc1 ZINC000217517252 EI On-Demand Unstable MTNR1A 66 41 COc1ccc(CCNC(=O)Nc2cc(C)c(Cl)cc2OC)cc1 ZINC000217517252 EI On-Demand Unstable MTNR1B 52 38 COc1ccc(CCNC(=O)Nc2cc(C)c(Cl)cc2OC)cc1 ZINC000217517252 EI On-Demand Unstable CA9 16 41 COc1ccc(CCNC(=O)Nc2cc(C)c(Cl)cc2OC)cc1 ZINC000217517252 EI On-Demand Unstable Q8MMZ8_EIMTE 43 67 COc1ccc(CCNC(=O)Nc2cc(C)c(Cl)cc2OC)cc1 ZINC000217517252 EI On-Demand Unstable NCE103 23 42 COc1ccc(CCNC(=O)Nc2cc(C)c(Cl)cc2OC)cc1 ZINC000217517252 EI On-Demand Unstable CAN2 0 42 O=C(Nc1ccc(Cl)cc1I)c1cc(Cl)ccc1Cl ZINC000217517254 IK On-Demand Anodyne F10 40 42 O=C(Nc1ccc(Cl)cc1I)c1cc(Cl)ccc1Cl ZINC000217517254 IK On-Demand Anodyne PYGL 15 41 O=C(Nc1ccc(Cl)cc1I)c1cc(Cl)ccc1Cl ZINC000217517254 IK On-Demand Anodyne KCNMA1 32 54 O=C(Nc1ccc(Cl)cc1I)c1cc(Cl)ccc1Cl ZINC000217517254 IK On-Demand Anodyne ACPS 0 44 O=C(Nc1ccc(Cl)cc1I)c1cc(Cl)ccc1Cl ZINC000217517254 IK On-Demand Anodyne Q25615_ONCVO 74 41 C[C@H](NC(=O)CN1CCC[C@@H](N)C1)c1ccco1 ZINC000217517258 CC For-Sale Unstable BIRC2 41 33 CC(C)c1ccc(OCC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217517267 GH For-Sale Unstable NPY5R 39 46 O=C(CS(=O)(=O)Cl)c1ccc(Cl)c(Cl)c1 ZINC000217517296 CF In-Stock Unstable CA6 0 40 O=C(CS(=O)(=O)Cl)c1ccc(Cl)c(Cl)c1 ZINC000217517296 CF In-Stock Unstable CA7 19 40 O=C(CS(=O)(=O)Cl)c1ccc(Cl)c(Cl)c1 ZINC000217517296 CF In-Stock Unstable CA13 37 40 O=C(CS(=O)(=O)Cl)c1ccc(Cl)c(Cl)c1 ZINC000217517296 CF In-Stock Unstable KMO 0 56 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1[C@@H]2C=C[C@]3(CN(CCc4ccccc4)C(=O)[C@@H]13)O2 ZINC000217517357 IF In-Stock Unstable MC4R 25 50 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1[C@@H]2C=C[C@]3(CN(CCc4ccccc4)C(=O)[C@@H]13)O2 ZINC000217517357 IF In-Stock Unstable BRS3 26 40 CCN(C(=O)NCCc1ccc(OC)cc1)c1cccc(C)c1 ZINC000217517358 DH For-Sale Unstable NQO2 28 40 CCN(C(=O)NCCc1ccc(OC)cc1)c1cccc(C)c1 ZINC000217517358 DH For-Sale Unstable CTSL 22 40 CCN(C(=O)NCCc1ccc(OC)cc1)c1cccc(C)c1 ZINC000217517358 DH For-Sale Unstable MTNR1A 97 41 CCN(C(=O)NCCc1ccc(OC)cc1)c1cccc(C)c1 ZINC000217517358 DH For-Sale Unstable MTNR1B 78 40 CCN(C(=O)NCCc1ccc(OC)cc1)c1cccc(C)c1 ZINC000217517358 DH For-Sale Unstable NR1H4 31 40 COc1ccccc1C(=O)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217517367 FG For-Sale Unstable HTR1A 19 41 COc1ccccc1C(=O)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217517367 FG For-Sale Unstable DRD2 28 49 COc1ccccc1C(=O)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217517367 FG For-Sale Unstable DRD4 42 32 COc1ccccc1C(=O)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217517367 FG For-Sale Unstable FABP4 46 40 COc1ccccc1C(=O)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217517367 FG For-Sale Unstable KCNA3 42 39 COc1ccccc1C(=O)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217517367 FG For-Sale Unstable HCN1 63 41 COc1ccccc1C(=O)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217517367 FG For-Sale Unstable HCN4 49 37 O=C(CS(=O)(=O)Cl)c1ccc(Cl)cc1Cl ZINC000217517392 CF In-Stock Unstable ALPL 44 36 O=C(CS(=O)(=O)Cl)c1ccc(Cl)cc1Cl ZINC000217517392 CF In-Stock Unstable FEN1 0 56 CCOc1ccc(OCC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217517401 GG For-Sale Unstable CPT1A 21 41 CCOc1ccc(OCC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217517401 GG For-Sale Unstable CPT2 32 41 CCOc1ccc(OCC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217517401 GG For-Sale Unstable NPY5R 43 48 COc1cccc(C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)c1 ZINC000217517458 FG For-Sale Unstable DRD4 66 51 COc1cccc(C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)c1 ZINC000217517458 FG For-Sale Unstable DRD3 27 51 COc1ccc(CCNC(=O)Nc2ccc(C)cc2Br)cc1 ZINC000217517473 FI On-Demand Unstable BMP1 37 41 COc1ccc(CCNC(=O)Nc2ccc(C)cc2Br)cc1 ZINC000217517473 FI On-Demand Unstable CA1 17 48 COc1ccc(CCNC(=O)Nc2ccc(C)cc2Br)cc1 ZINC000217517473 FI On-Demand Unstable RAF1 37 41 COc1ccc(CCNC(=O)Nc2ccc(C)cc2Br)cc1 ZINC000217517473 FI On-Demand Unstable MTNR1A 73 42 COc1ccc(CCNC(=O)Nc2ccc(C)cc2Br)cc1 ZINC000217517473 FI On-Demand Unstable MTNR1B 53 39 COc1ccc(CCNC(=O)Nc2ccc(C)cc2Br)cc1 ZINC000217517473 FI On-Demand Unstable CA12 15 48 COc1ccc(CCNC(=O)Nc2ccc(C)cc2Br)cc1 ZINC000217517473 FI On-Demand Unstable CA9 26 48 O=C1OC2(CCN(C(=O)C3(c4cccs4)CCCC3)CC2)c2ccccc21 ZINC000217517509 GI For-Sale Unstable NPY5R 35 48 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1N[C@@H](C)COC ZINC000217517525 FE In-Stock Unstable PLA2G4B 42 35 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1N[C@H](C)COC ZINC000217517584 FE In-Stock Unstable PLA2G4B 42 35 O=C(CS(=O)(=O)Cl)N1CCc2ccccc21 ZINC000217517623 CD In-Stock Unstable AVPR2 30 40 O=C(CS(=O)(=O)Cl)N1CCc2ccccc21 ZINC000217517623 CD In-Stock Unstable HSD17B3 17 44 O=C(CS(=O)(=O)Cl)N1CCc2ccccc21 ZINC000217517623 CD In-Stock Unstable EIF2AK3 45 36 CS(=O)(=O)N1CCC(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)CC1 ZINC000217517633 GD For-Sale Unstable NPY5R 67 48 NC(=O)C1CCN(C(=O)c2cc(I)ccc2O)CC1 ZINC000217517651 FD On-Demand Unstable L3MBTL3 58 36 CC1(C)Cc2cccc(OCC(=O)N3CCC4(CC3)OC(=O)c3ccccc34)c2O1 ZINC000217517754 HG For-Sale Unstable NPY5R 30 47 O=C(Nc1ccc(Cl)cc1F)c1ccc(=O)[nH]n1 ZINC000217517775 CD On-Demand Anodyne ALPL 50 35 O=C1OC2(CCN(C(=O)C3c4ccccc4Oc4ccccc43)CC2)c2ccccc21 ZINC000217517850 HJ For-Sale Unstable NPY5R 50 49 N[C@@H]1CCCN(C/C=C\c2ccccc2)C1 ZINC000217517877 BE On-Demand Unstable SLC6A1 51 35 CC[C@@H](C)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217517928 EJ For-Sale Unstable BMP1 35 43 CC[C@@H](C)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217517928 EJ For-Sale Unstable NQO2 26 42 CC[C@@H](C)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217517928 EJ For-Sale Unstable MTNR1A 77 42 CC[C@@H](C)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217517928 EJ For-Sale Unstable MTNR1B 63 37 CC[C@@H](C)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217517928 EJ For-Sale Unstable MMP3 23 42 CC[C@@H](C)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217517928 EJ For-Sale Unstable SOAT1 25 44 CC[C@@H](C)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217517928 EJ For-Sale Unstable MMP9 17 42 CC[C@@H](C)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217517928 EJ For-Sale Unstable CA9 20 41 CC[C@@H](C)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217517928 EJ For-Sale Unstable MMP1 22 42 CC[C@@H](C)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217517928 EJ For-Sale Unstable ACAT 0 50 CC[C@@H](C)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217517928 EJ For-Sale Unstable AO-ACHE 0 41 O=C(O)[C@@]12C[C@@H]3C[C@@H](C[C@@](n4ncc(NCc5ccc6c(c5)OCO6)c(Cl)c4=O)(C3)C1)C2 ZINC000217517952 JH In-Stock Unstable NOS2 50 31 CN(C)S(=O)(=O)c1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217517965 HE For-Sale Unstable NPY5R 33 46 Cc1ccc(F)cc1NC(=O)c1ccc(=O)[nH]n1 ZINC000217517967 BD On-Demand Unstable PLA2G7 25 46 Cc1nc2ccccc2cc1C(=O)Nc1cccc(S(=O)(=O)NC2=NCCC2)c1 ZINC000217517991 HG On-Demand Unstable KCNK3 53 35 Cc1nc2ccccc2cc1C(=O)Nc1cccc(S(=O)(=O)NC2=NCCC2)c1 ZINC000217517991 HG On-Demand Unstable KCNK9 47 34 CC(=O)Nc1ccc(N2C[C@@]34C=C[C@H](O3)[C@@H](C(=O)NCc3cccnc3)[C@@H]4C2=O)cc1 ZINC000217518000 HD In-Stock Unstable NAMPT 63 41 CC[C@H](C)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217518013 EJ For-Sale Unstable BMP1 35 43 CC[C@H](C)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217518013 EJ For-Sale Unstable NQO2 26 42 CC[C@H](C)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217518013 EJ For-Sale Unstable MTNR1A 77 42 CC[C@H](C)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217518013 EJ For-Sale Unstable MTNR1B 63 37 CC[C@H](C)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217518013 EJ For-Sale Unstable MMP3 23 42 CC[C@H](C)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217518013 EJ For-Sale Unstable SOAT1 25 44 CC[C@H](C)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217518013 EJ For-Sale Unstable MMP9 17 42 CC[C@H](C)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217518013 EJ For-Sale Unstable CA9 20 41 CC[C@H](C)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217518013 EJ For-Sale Unstable MMP1 22 42 CC[C@H](C)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217518013 EJ For-Sale Unstable ACAT 0 50 CC[C@H](C)c1ccccc1NC(=O)NCCc1ccc(OC)cc1 ZINC000217518013 EJ For-Sale Unstable AO-ACHE 0 41 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccccc1Cl ZINC000217518032 FH For-Sale Unstable FABP4 46 36 COc1ccc(Br)c(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217518072 HH In-Stock Unstable ACACA 15 41 COc1ccc(Br)c(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217518072 HH In-Stock Unstable NPY5R 34 54 CC(=O)Nc1ccc(N2C[C@@]34C=C[C@H](O3)[C@@H](C(=O)NCc3cccnc3)[C@H]4C2=O)cc1 ZINC000217518082 HD In-Stock Unstable NAMPT 63 41 COc1ccc(CCNC(=O)Nc2cc(C)ccc2N)cc1 ZINC000217518110 CF For-Sale Unstable CA1 17 45 COc1ccc(CCNC(=O)Nc2cc(C)ccc2N)cc1 ZINC000217518110 CF For-Sale Unstable RAF1 25 43 COc1ccc(CCNC(=O)Nc2cc(C)ccc2N)cc1 ZINC000217518110 CF For-Sale Unstable MTNR1A 72 42 COc1ccc(CCNC(=O)Nc2cc(C)ccc2N)cc1 ZINC000217518110 CF For-Sale Unstable MTNR1B 54 39 COc1ccc(CCNC(=O)Nc2cc(C)ccc2N)cc1 ZINC000217518110 CF For-Sale Unstable CA9 22 45 COc1ccc(CCNC(=O)Nc2cc(C)ccc2N)cc1 ZINC000217518110 CF For-Sale Unstable Q8MMZ8_EIMTE 34 41 COc1ccc(CCNC(=O)Nc2cc(C)ccc2N)cc1 ZINC000217518110 CF For-Sale Unstable PROKR1 59 33 C#Cc1c(N)c(OC)cc(C(=O)OC)c1Cl ZINC000217518114 BD For-Sale Unstable HTR4 46 36 O=C(Nc1nc2c(s1)CCCC2)[C@@H]1C[C@@H]1c1ccccc1C(F)(F)F ZINC000217518123 FJ On-Demand Unstable RBP4 78 35 O=C(Nc1nc2c(s1)CCCC2)[C@@H]1C[C@@H]1c1ccccc1C(F)(F)F ZINC000217518123 FJ On-Demand Unstable SLC27A1 32 43 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1cccc(Cl)c1 ZINC000217518135 FH For-Sale Unstable DRD4 48 40 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1cccc(Cl)c1 ZINC000217518135 FH For-Sale Unstable CCR2 23 40 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1cccc(Cl)c1 ZINC000217518135 FH For-Sale Unstable PLD2 45 38 CC(=O)Nc1ccc(N2C[C@]34C=C[C@H](O3)[C@@H](C(=O)NCc3cccnc3)[C@H]4C2=O)cc1 ZINC000217518137 HD In-Stock Unstable NAMPT 63 41 Cc1onc(-c2ccccc2Cl)c1C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217518162 HJ For-Sale Unstable AVPR1A 15 48 Cc1onc(-c2ccccc2Cl)c1C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217518162 HJ For-Sale Unstable NPY5R 43 53 Cc1onc(-c2ccccc2Cl)c1C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217518162 HJ For-Sale Unstable GPBAR1 38 48 Cc1ncccc1Oc1ncnc(N2CCn3nc(CO)cc3C2)c1C ZINC000217518174 FD In-Stock Unstable GPR119 19 44 O=C(Nc1nc2c(s1)CCCC2)[C@H]1C[C@@H]1c1ccccc1C(F)(F)F ZINC000217518205 FJ On-Demand Unstable RBP4 78 35 O=C(Nc1nc2c(s1)CCCC2)[C@H]1C[C@@H]1c1ccccc1C(F)(F)F ZINC000217518205 FJ On-Demand Unstable SLC27A1 32 43 COc1ccc(CCNC(=O)Nc2ccc(C)cc2N)cc1 ZINC000217518236 CF For-Sale Unstable CA1 18 45 COc1ccc(CCNC(=O)Nc2ccc(C)cc2N)cc1 ZINC000217518236 CF For-Sale Unstable TRPV1 0 52 COc1ccc(CCNC(=O)Nc2ccc(C)cc2N)cc1 ZINC000217518236 CF For-Sale Unstable RAF1 23 41 COc1ccc(CCNC(=O)Nc2ccc(C)cc2N)cc1 ZINC000217518236 CF For-Sale Unstable MTNR1A 74 42 COc1ccc(CCNC(=O)Nc2ccc(C)cc2N)cc1 ZINC000217518236 CF For-Sale Unstable MTNR1B 54 39 COc1ccc(CCNC(=O)Nc2ccc(C)cc2N)cc1 ZINC000217518236 CF For-Sale Unstable CA9 22 45 COc1ccc(CCNC(=O)Nc2ccc(C)cc2N)cc1 ZINC000217518236 CF For-Sale Unstable Q8MMZ8_EIMTE 31 41 COc1ccc(CCNC(=O)Nc2ccc(C)cc2N)cc1 ZINC000217518236 CF For-Sale Unstable PROKR1 41 31 CC(C)S(=O)(=O)c1ccc(CC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217518275 IG For-Sale Unstable NPY5R 31 44 O=C(Nc1nc2c(s1)CCCC2)[C@@H]1C[C@H]1c1ccccc1C(F)(F)F ZINC000217518282 FJ On-Demand Unstable RBP4 78 35 O=C(Nc1nc2c(s1)CCCC2)[C@@H]1C[C@H]1c1ccccc1C(F)(F)F ZINC000217518282 FJ On-Demand Unstable SLC27A1 32 43 CN(C)CCSc1ccc(-c2ccccc2)cc1 ZINC000217518288 CI On-Demand Unstable DRD2 16 53 CN(C)CCSc1ccc(-c2ccccc2)cc1 ZINC000217518288 CI On-Demand Unstable UTS2 50 38 COc1ccc(CCNC(=O)N2CCCC[C@@H]2CCO)cc1 ZINC000217518338 DE On-Demand Unstable FKBP1A 46 43 COc1ccc(CCNC(=O)N2CCCC[C@@H]2CCO)cc1 ZINC000217518338 DE On-Demand Unstable SLC18A2 53 49 COc1ccc(CCNC(=O)N2CCCC[C@@H]2CCO)cc1 ZINC000217518338 DE On-Demand Unstable CTSK 15 44 COc1ccc(CCNC(=O)N2CCCC[C@@H]2CCO)cc1 ZINC000217518338 DE On-Demand Unstable CCR3 17 41 COc1ccc(CCNC(=O)N2CCCC[C@@H]2CCO)cc1 ZINC000217518338 DE On-Demand Unstable NOS2 15 47 COc1ccc(CCNC(=O)N2CCCC[C@@H]2CCO)cc1 ZINC000217518338 DE On-Demand Unstable MMP3 16 41 COc1ccc(CCNC(=O)N2CCCC[C@@H]2CCO)cc1 ZINC000217518338 DE On-Demand Unstable MMP9 16 41 COc1ccc(CCNC(=O)N2CCCC[C@@H]2CCO)cc1 ZINC000217518338 DE On-Demand Unstable MMP7 22 41 COc1ccc(CCNC(=O)N2CCCC[C@@H]2CCO)cc1 ZINC000217518338 DE On-Demand Unstable MMP1 17 41 O=C(Nc1nc2c(s1)CCCC2)[C@H]1C[C@H]1c1ccccc1C(F)(F)F ZINC000217518365 FJ On-Demand Unstable RBP4 78 35 O=C(Nc1nc2c(s1)CCCC2)[C@H]1C[C@H]1c1ccccc1C(F)(F)F ZINC000217518365 FJ On-Demand Unstable SLC27A1 32 43 O=C1OC2(CCN(C(=O)c3ccc(S(=O)(=O)N4CCOCC4)cc3)CC2)c2ccccc21 ZINC000217518393 JE For-Sale Unstable NPY5R 29 45 COc1ccc(CCNC(=O)N2CCCC[C@H]2CCO)cc1 ZINC000217518406 DE On-Demand Unstable FKBP1A 46 43 COc1ccc(CCNC(=O)N2CCCC[C@H]2CCO)cc1 ZINC000217518406 DE On-Demand Unstable SLC18A2 53 49 COc1ccc(CCNC(=O)N2CCCC[C@H]2CCO)cc1 ZINC000217518406 DE On-Demand Unstable CTSK 15 44 COc1ccc(CCNC(=O)N2CCCC[C@H]2CCO)cc1 ZINC000217518406 DE On-Demand Unstable CCR3 17 41 COc1ccc(CCNC(=O)N2CCCC[C@H]2CCO)cc1 ZINC000217518406 DE On-Demand Unstable NOS2 15 47 COc1ccc(CCNC(=O)N2CCCC[C@H]2CCO)cc1 ZINC000217518406 DE On-Demand Unstable MMP3 16 41 COc1ccc(CCNC(=O)N2CCCC[C@H]2CCO)cc1 ZINC000217518406 DE On-Demand Unstable MMP9 16 41 COc1ccc(CCNC(=O)N2CCCC[C@H]2CCO)cc1 ZINC000217518406 DE On-Demand Unstable MMP7 22 41 COc1ccc(CCNC(=O)N2CCCC[C@H]2CCO)cc1 ZINC000217518406 DE On-Demand Unstable MMP1 17 41 Nc1nc(NC2CC2)cc(N2CCCn3nc(CO)cc3C2)n1 ZINC000217518451 DC In-Stock Unstable HRH4 40 48 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCc1cnc(C(C)(C)C)s1 ZINC000217518465 DJ For-Sale Unstable TRPM8 0 40 O=[N+]([O-])c1cccc(S(=O)(=O)NCc2ccc(OC(F)(F)F)cc2)c1 ZINC000217518471 GF On-Demand Unstable CACNA1D 59 36 O=[N+]([O-])c1cccc(S(=O)(=O)NCc2ccc(OC(F)(F)F)cc2)c1 ZINC000217518471 GF On-Demand Unstable MMP8 16 40 Cn1nc(-c2ccc(F)cc2)cc1C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217518489 HH For-Sale Unstable NPY5R 54 55 COc1ccc(CCNC(=O)NC(C)(C)CO)cc1 ZINC000217518521 CD For-Sale Unstable CTSL 19 43 COc1ccc(CCNC(=O)NC(C)(C)CO)cc1 ZINC000217518521 CD For-Sale Unstable MTNR1A 75 42 COc1ccc(CCNC(=O)NC(C)(C)CO)cc1 ZINC000217518521 CD For-Sale Unstable MTNR1B 62 39 COc1ccc(CCNC(=O)NC(C)(C)CO)cc1 ZINC000217518521 CD For-Sale Unstable MMP9 16 40 COc1ccc(CCNC(=O)NC(C)(C)CO)cc1 ZINC000217518521 CD For-Sale Unstable PTGDR 24 41 COc1ccc(CCNC(=O)NC(C)(C)CO)cc1 ZINC000217518521 CD For-Sale Unstable CA9 19 48 COc1ccc(CCNC(=O)NC(C)(C)CO)cc1 ZINC000217518521 CD For-Sale Unstable MMP1 26 40 COc1ccc(CCNC(=O)NC(C)(C)CO)cc1 ZINC000217518521 CD For-Sale Unstable PROKR1 61 34 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCc1cnc(C(C)(C)C)s1 ZINC000217518549 DJ For-Sale Unstable TRPM8 0 40 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc(F)c(F)c1 ZINC000217518552 FG For-Sale Unstable PLD1 36 40 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc(F)c(F)c1 ZINC000217518552 FG For-Sale Unstable PLD2 55 40 COCC(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217518608 CD In-Stock Unstable NPY5R 49 52 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCc1cnc(C(C)(C)C)s1 ZINC000217518628 DJ For-Sale Unstable TRPM8 0 40 COC(=O)CCNC(=O)NCCc1ccc(OC)cc1 ZINC000217518630 CD For-Sale Unstable BMP1 36 40 COC(=O)CCNC(=O)NCCc1ccc(OC)cc1 ZINC000217518630 CD For-Sale Unstable NQO2 31 40 COC(=O)CCNC(=O)NCCc1ccc(OC)cc1 ZINC000217518630 CD For-Sale Unstable CA1 15 51 COC(=O)CCNC(=O)NCCc1ccc(OC)cc1 ZINC000217518630 CD For-Sale Unstable MTNR1A 96 46 COC(=O)CCNC(=O)NCCc1ccc(OC)cc1 ZINC000217518630 CD For-Sale Unstable MTNR1B 75 40 COC(=O)CCNC(=O)NCCc1ccc(OC)cc1 ZINC000217518630 CD For-Sale Unstable MMP9 15 42 COC(=O)CCNC(=O)NCCc1ccc(OC)cc1 ZINC000217518630 CD For-Sale Unstable CA9 22 51 COC(=O)CCNC(=O)NCCc1ccc(OC)cc1 ZINC000217518630 CD For-Sale Unstable MMP1 19 42 COC(=O)CCNC(=O)NCCc1ccc(OC)cc1 ZINC000217518630 CD For-Sale Unstable PROKR1 59 34 O=C(NC1CCCCCCC1)c1cc(Br)ccc1I ZINC000217518656 IJ For-Sale Unstable CNR1 24 47 O=C(NC1CCCCCCC1)c1cc(Br)ccc1I ZINC000217518656 IJ For-Sale Unstable CNR2 32 49 O=C(NC1CCCCCCC1)c1cc(Br)ccc1I ZINC000217518656 IJ For-Sale Unstable EPHX2 23 41 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1cc2ccccc2o1 ZINC000217518662 GH For-Sale Unstable BCHE 46 38 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCc1cnc(C(C)(C)C)s1 ZINC000217518702 DJ For-Sale Unstable TRPM8 0 40 Cc1ccc(C)c(S(=O)(=O)NCC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217518723 IE For-Sale Unstable NPY5R 34 48 COC(=O)CNC(=O)NCCc1ccc(OC)cc1 ZINC000217518725 CC For-Sale Unstable BMP1 29 41 COC(=O)CNC(=O)NCCc1ccc(OC)cc1 ZINC000217518725 CC For-Sale Unstable NQO2 33 40 COC(=O)CNC(=O)NCCc1ccc(OC)cc1 ZINC000217518725 CC For-Sale Unstable CA1 15 51 COC(=O)CNC(=O)NCCc1ccc(OC)cc1 ZINC000217518725 CC For-Sale Unstable MMP13 16 45 COC(=O)CNC(=O)NCCc1ccc(OC)cc1 ZINC000217518725 CC For-Sale Unstable CTSL 15 43 COC(=O)CNC(=O)NCCc1ccc(OC)cc1 ZINC000217518725 CC For-Sale Unstable MTNR1A 94 46 COC(=O)CNC(=O)NCCc1ccc(OC)cc1 ZINC000217518725 CC For-Sale Unstable MTNR1B 74 40 COC(=O)CNC(=O)NCCc1ccc(OC)cc1 ZINC000217518725 CC For-Sale Unstable MMP9 17 42 COC(=O)CNC(=O)NCCc1ccc(OC)cc1 ZINC000217518725 CC For-Sale Unstable CA9 22 51 COC(=O)CNC(=O)NCCc1ccc(OC)cc1 ZINC000217518725 CC For-Sale Unstable MMP1 22 42 COC(=O)CNC(=O)NCCc1ccc(OC)cc1 ZINC000217518725 CC For-Sale Unstable PROKR1 59 34 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc(Cl)s1 ZINC000217518783 GH For-Sale Unstable F10 17 40 CN(CCN1CCCC1)c1ccc(F)cc1CBr ZINC000217518796 DG For-Sale Unstable MPO 19 41 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCc1cc(F)c(F)c(F)c1 ZINC000217518806 CJ For-Sale Unstable TRPM8 16 42 O=C1OC2(CCN(C(=O)c3ccc(-c4ccsc4)cc3)CC2)c2ccccc21 ZINC000217518824 GJ For-Sale Unstable NPY5R 43 49 COc1ccc(CCNC(=O)NCc2ccc(CO)cc2)cc1 ZINC000217518837 DE On-Demand Unstable MMP13 20 40 COc1ccc(CCNC(=O)NCc2ccc(CO)cc2)cc1 ZINC000217518837 DE On-Demand Unstable CTSL 16 42 COc1ccc(CCNC(=O)NCc2ccc(CO)cc2)cc1 ZINC000217518837 DE On-Demand Unstable MTNR1A 82 47 COc1ccc(CCNC(=O)NCc2ccc(CO)cc2)cc1 ZINC000217518837 DE On-Demand Unstable MTNR1B 63 40 COc1ccc(CCNC(=O)NCc2ccc(CO)cc2)cc1 ZINC000217518837 DE On-Demand Unstable CA9 22 49 COc1ccc(CCNC(=O)NCc2ccc(CO)cc2)cc1 ZINC000217518837 DE On-Demand Unstable MMP1 15 41 COc1ccc(CCNC(=O)NCc2ccc(CO)cc2)cc1 ZINC000217518837 DE On-Demand Unstable U38 0 40 COc1ccc(CCNC(=O)NCc2ccc(CO)cc2)cc1 ZINC000217518837 DE On-Demand Unstable PROKR1 61 35 N[C@@H]1CCCN(C[C@@H]2COc3ccccc3O2)C1 ZINC000217518838 BD On-Demand Unstable ADRA2B 26 49 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCc1cc(F)c(F)c(F)c1 ZINC000217518900 CJ For-Sale Unstable TRPM8 16 42 O=C(CCCc1ccccc1)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217518904 GH For-Sale Unstable FABP4 44 33 O=C(CCCc1ccccc1)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217518904 GH For-Sale Unstable PREP 42 34 O=C1OC2(CCN(C(=O)c3ccc(NS(=O)(=O)c4cccc(F)c4)cc3)CC2)c2ccccc21 ZINC000217518927 JH For-Sale Unstable NPY5R 36 51 COc1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217518949 GH On-Demand Unstable CA2 16 52 COc1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217518949 GH On-Demand Unstable BMP1 42 44 COc1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217518949 GH On-Demand Unstable NQO2 31 41 COc1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217518949 GH On-Demand Unstable CA1 18 52 COc1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217518949 GH On-Demand Unstable MMP13 34 46 COc1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217518949 GH On-Demand Unstable MMP16 0 45 COc1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217518949 GH On-Demand Unstable MTNR1A 103 49 COc1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217518949 GH On-Demand Unstable MTNR1B 80 41 COc1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217518949 GH On-Demand Unstable MMP2 20 45 COc1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217518949 GH On-Demand Unstable MMP8 20 46 COc1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217518949 GH On-Demand Unstable MMP9 39 45 COc1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217518949 GH On-Demand Unstable MMP12 23 46 COc1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217518949 GH On-Demand Unstable PTGDR 29 40 COc1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217518949 GH On-Demand Unstable CA9 23 52 COc1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217518949 GH On-Demand Unstable MMP1 42 45 COc1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217518949 GH On-Demand Unstable PROKR1 60 34 COc1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217518949 GH On-Demand Unstable LIG1 0 41 COc1ccc(N2C[C@@]34C=C[C@@H](O3)[C@@H](C(=O)NCCc3c[nH]c5ccccc35)[C@@H]4C2=O)cc1 ZINC000217518990 IF In-Stock Unstable MTNR1A 27 40 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCc1cc(F)c(F)c(F)c1 ZINC000217518998 CJ For-Sale Unstable TRPM8 16 42 CN(CCN1CCCC1)c1cccc(Cl)c1CBr ZINC000217519013 EH For-Sale Unstable SIGMAR1 18 44 O=C1OC2(CCN(C(=O)CNS(=O)(=O)c3cccc(Cl)c3)CC2)c2ccccc21 ZINC000217519057 IE For-Sale Unstable NPY5R 33 56 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCc1cc(F)c(F)c(F)c1 ZINC000217519074 CJ For-Sale Unstable TRPM8 16 42 COc1ccc(CCNC(=O)Nc2ccc(Br)cn2)cc1 ZINC000217519075 FG For-Sale Unstable BMP1 20 41 COc1ccc(CCNC(=O)Nc2ccc(Br)cn2)cc1 ZINC000217519075 FG For-Sale Unstable CTSK 23 42 COc1ccc(CCNC(=O)Nc2ccc(Br)cn2)cc1 ZINC000217519075 FG For-Sale Unstable CTSL 18 46 COc1ccc(CCNC(=O)Nc2ccc(Br)cn2)cc1 ZINC000217519075 FG For-Sale Unstable RAF1 37 41 COc1ccc(CCNC(=O)Nc2ccc(Br)cn2)cc1 ZINC000217519075 FG For-Sale Unstable MTNR1A 46 38 COc1ccc(CCNC(=O)Nc2ccc(Br)cn2)cc1 ZINC000217519075 FG For-Sale Unstable PTGDR 23 41 COc1ccc(CCNC(=O)Nc2ccc(Br)cn2)cc1 ZINC000217519075 FG For-Sale Unstable CA9 18 43 COc1ccc(CCNC(=O)Nc2ccc(Br)cn2)cc1 ZINC000217519075 FG For-Sale Unstable Q8MMZ8_EIMTE 26 41 COc1ccc(CCNC(=O)Nc2ccc(Br)cn2)cc1 ZINC000217519075 FG For-Sale Unstable LUCI_LUCLA 18 41 Cc1cc2c(c(C)c1Br)C=C(C(=O)O)[C@H](C(F)(F)F)O2 ZINC000217519088 FH Annotated Unstable PTGS1 17 56 Cc1cc2c(c(C)c1Br)C=C(C(=O)O)[C@H](C(F)(F)F)O2 ZINC000217519088 FH Annotated Unstable PTGS2 21 73 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCc1ccc(O)c(Br)c1 ZINC000217519166 EJ For-Sale Unstable TRPM8 16 41 Cc1cc2c(c(C)c1Br)C=C(C(=O)O)[C@@H](C(F)(F)F)O2 ZINC000217519174 FH Annotated Unstable PTGS1 17 56 Cc1cc2c(c(C)c1Br)C=C(C(=O)O)[C@@H](C(F)(F)F)O2 ZINC000217519174 FH Annotated Unstable PTGS2 21 73 O=C1OC2(CCN(C(=O)CNS(=O)(=O)c3cccc(F)c3)CC2)c2ccccc21 ZINC000217519176 HD For-Sale Unstable NPY5R 43 54 COc1ccc(CCNC(=O)Nc2cc(Cl)ccn2)cc1 ZINC000217519186 DG On-Demand Unstable NQO2 22 40 COc1ccc(CCNC(=O)Nc2cc(Cl)ccn2)cc1 ZINC000217519186 DG On-Demand Unstable CTSK 16 40 COc1ccc(CCNC(=O)Nc2cc(Cl)ccn2)cc1 ZINC000217519186 DG On-Demand Unstable CTSL 17 41 COc1ccc(CCNC(=O)Nc2cc(Cl)ccn2)cc1 ZINC000217519186 DG On-Demand Unstable RAF1 47 44 COc1ccc(CCNC(=O)Nc2cc(Cl)ccn2)cc1 ZINC000217519186 DG On-Demand Unstable MTNR1A 49 38 COc1ccc(CCNC(=O)Nc2cc(Cl)ccn2)cc1 ZINC000217519186 DG On-Demand Unstable MTNR1B 43 39 COc1ccc(CCNC(=O)Nc2cc(Cl)ccn2)cc1 ZINC000217519186 DG On-Demand Unstable PDGFRA 43 38 COc1ccc(CCNC(=O)Nc2cc(Cl)ccn2)cc1 ZINC000217519186 DG On-Demand Unstable PTGDR 27 43 COc1ccc(CCNC(=O)Nc2cc(Cl)ccn2)cc1 ZINC000217519186 DG On-Demand Unstable CA9 16 42 COc1ccc(CCNC(=O)Nc2cc(Cl)ccn2)cc1 ZINC000217519186 DG On-Demand Unstable Q8MMZ8_EIMTE 40 44 COc1ccc(CCNC(=O)Nc2cc(Cl)ccn2)cc1 ZINC000217519186 DG On-Demand Unstable PROKR1 53 33 CC[C@H](C(=O)NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccccc1 ZINC000217519246 GI For-Sale Unstable KCNQ2 45 38 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCc1ccc(O)c(Br)c1 ZINC000217519259 EJ For-Sale Unstable TRPM8 16 41 CCOC(=O)[C@@H]1CCCN(C(=O)c2cc(I)ccc2O)C1 ZINC000217519264 HE On-Demand Unstable FDFT1 21 40 Cc1cc(C)c(C)c(S(=O)(=O)NCC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1C ZINC000217519286 JF For-Sale Unstable NPY5R 36 46 COc1ccc(CCNC(=O)Nc2cc(Br)ccn2)cc1 ZINC000217519306 FG On-Demand Unstable RAF1 47 40 COc1ccc(CCNC(=O)Nc2cc(Br)ccn2)cc1 ZINC000217519306 FG On-Demand Unstable MTNR1A 47 38 COc1ccc(CCNC(=O)Nc2cc(Br)ccn2)cc1 ZINC000217519306 FG On-Demand Unstable MTNR1B 41 39 COc1ccc(CCNC(=O)Nc2cc(Br)ccn2)cc1 ZINC000217519306 FG On-Demand Unstable PDGFRA 40 37 COc1ccc(CCNC(=O)Nc2cc(Br)ccn2)cc1 ZINC000217519306 FG On-Demand Unstable PTGDR 24 43 COc1ccc(CCNC(=O)Nc2cc(Br)ccn2)cc1 ZINC000217519306 FG On-Demand Unstable Q8MMZ8_EIMTE 40 40 NC[C@@H]1CCCN([C@@H]2CCSc3ccccc32)C1 ZINC000217519316 CF For-Sale Unstable SLC6A1 0 43 CC[C@@H](C(=O)NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccccc1 ZINC000217519329 GI For-Sale Unstable KCNQ2 45 38 CCOC(=O)[C@H]1CCCN(C(=O)c2cc(I)ccc2O)C1 ZINC000217519338 HE On-Demand Unstable FDFT1 21 40 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCc1ccc(O)c(Br)c1 ZINC000217519339 EJ For-Sale Unstable TRPM8 16 41 O=C(/C=C\c1cccc(Cl)c1)N[C@@H]1CCC(=O)NC1=O ZINC000217519364 CD On-Demand Unstable MMP1 0 44 O=C(/C=C\c1cccc(Cl)c1)N[C@@H]1CCC(=O)NC1=O ZINC000217519364 CD On-Demand Unstable TUBA4A 0 43 CC(C)CCNS(=O)(=O)c1cc(C(=O)O)ccc1NCc1ccccc1 ZINC000217519384 GG In-Stock Unstable AKR1C3 15 44 CC(C)(C)c1ccc(S(=O)(=O)NCC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217519411 JF For-Sale Unstable NPY5R 29 46 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCc1ccc(O)c(Br)c1 ZINC000217519412 EJ For-Sale Unstable TRPM8 16 41 CCOC(CNC(=O)NCCc1ccc(OC)cc1)OCC ZINC000217519424 DD For-Sale Unstable ADRB2 15 42 CCOC(CNC(=O)NCCc1ccc(OC)cc1)OCC ZINC000217519424 DD For-Sale Unstable ADRB3 15 41 CCOC(CNC(=O)NCCc1ccc(OC)cc1)OCC ZINC000217519424 DD For-Sale Unstable MTNR1A 74 44 CCOC(CNC(=O)NCCc1ccc(OC)cc1)OCC ZINC000217519424 DD For-Sale Unstable MTNR1B 57 40 CCOC(CNC(=O)NCCc1ccc(OC)cc1)OCC ZINC000217519424 DD For-Sale Unstable CA9 18 46 CN(C)c1ccc(C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc1 ZINC000217519434 GG For-Sale Unstable GIPR 42 33 O=C(/C=C\c1cccc(Cl)c1)N[C@H]1CCC(=O)NC1=O ZINC000217519452 CD On-Demand Unstable MMP1 0 44 O=C(/C=C\c1cccc(Cl)c1)N[C@H]1CCC(=O)NC1=O ZINC000217519452 CD On-Demand Unstable TUBA4A 0 43 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCCC(C)(C)C ZINC000217519491 BI For-Sale Unstable TRPM8 15 44 CC(C)CCNS(=O)(=O)c1cc(C(=O)O)ccc1N[C@@H](C)c1ccccc1 ZINC000217519501 GH In-Stock Unstable LDHB 0 42 O=C1OC2(CCN(C(=O)c3ccc(NS(=O)(=O)c4ccccc4F)cc3)CC2)c2ccccc21 ZINC000217519518 JH For-Sale Unstable NPY5R 32 49 CCN(Cc1ccccc1)C(=O)c1cc(Br)ccc1I ZINC000217519528 IJ For-Sale Unstable TSPO 27 42 CCN(Cc1ccccc1)C(=O)c1cc(Br)ccc1I ZINC000217519528 IJ For-Sale Unstable LIMK2 21 45 COc1ccc(CCNC(=O)NCCC#N)cc1 ZINC000217519533 BD On-Demand Unstable CTSK 27 45 COc1ccc(CCNC(=O)NCCC#N)cc1 ZINC000217519533 BD On-Demand Unstable CTSL 23 47 COc1ccc(CCNC(=O)NCCC#N)cc1 ZINC000217519533 BD On-Demand Unstable MTNR1B 49 38 COc1ccc(CCNC(=O)NCCC#N)cc1 ZINC000217519533 BD On-Demand Unstable CA9 24 49 COc1ccc(CCNC(=O)NCCC#N)cc1 ZINC000217519533 BD On-Demand Unstable PROKR1 54 33 CN(C)c1cccc(C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)c1 ZINC000217519544 GG For-Sale Unstable DRD4 44 35 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCCC(C)(C)C ZINC000217519578 BI For-Sale Unstable TRPM8 15 44 CC(C)CCNS(=O)(=O)c1cc(C(=O)O)ccc1N[C@H](C)c1ccccc1 ZINC000217519589 GH In-Stock Unstable LDHB 0 42 O=C(Nc1ccc(N2CCOCC2)cc1N1CCOCC1)[C@@H]1C[C@@H]1c1ccccc1Cl ZINC000217519616 IH On-Demand Unstable CSF1R 15 43 O=C(Nc1ccc(N2CCOCC2)cc1N1CCOCC1)[C@@H]1C[C@@H]1c1ccccc1Cl ZINC000217519616 IH On-Demand Unstable AKR1C3 27 42 O=C1OC2(CCN(C(=O)CNS(=O)(=O)c3ccccc3F)CC2)c2ccccc21 ZINC000217519618 HD For-Sale Unstable NPY5R 40 52 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc2c(c1)OCO2 ZINC000217519653 GF For-Sale Unstable NOS2 44 31 CCOC(=O)N(CCN)C(=O)NCCc1ccc(OC)cc1 ZINC000217519658 DD For-Sale Unstable NQO2 23 40 CCOC(=O)N(CCN)C(=O)NCCc1ccc(OC)cc1 ZINC000217519658 DD For-Sale Unstable MTNR1A 51 36 CCOC(=O)N(CCN)C(=O)NCCc1ccc(OC)cc1 ZINC000217519658 DD For-Sale Unstable CA9 18 45 CCOC(=O)N(CCN)C(=O)NCCc1ccc(OC)cc1 ZINC000217519658 DD For-Sale Unstable PROKR1 42 32 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCCC(C)(C)C ZINC000217519663 BI For-Sale Unstable TRPM8 15 44 O=C(Cc1c[nH]c(=O)[nH]c1=O)N1CCC(N2CCc3ccccc3C2)CC1 ZINC000217519678 FC In-Stock Unstable CALCRL 42 34 O=C(Nc1ccc(N2CCOCC2)cc1N1CCOCC1)[C@H]1C[C@@H]1c1ccccc1Cl ZINC000217519706 IH On-Demand Unstable CSF1R 15 43 O=C(Nc1ccc(N2CCOCC2)cc1N1CCOCC1)[C@H]1C[C@@H]1c1ccccc1Cl ZINC000217519706 IH On-Demand Unstable AKR1C3 27 42 CN(CCN1CCCC1)c1ccc(CBr)cc1Cl ZINC000217519712 EH For-Sale Unstable HRH3 15 42 CN(CCN1CCCC1)c1ccc(CBr)cc1Cl ZINC000217519712 EH For-Sale Unstable SIGMAR1 28 58 O=C1OC2(CCN(C(=O)CCNS(=O)(=O)c3ccccc3F)CC2)c2ccccc21 ZINC000217519716 IE For-Sale Unstable NPY5R 34 50 CCN(Cc1ccccc1)C(=O)c1cc(I)ccc1O ZINC000217519739 GH On-Demand Unstable TSPO 30 43 CCN(Cc1ccccc1)C(=O)c1cc(I)ccc1O ZINC000217519739 GH On-Demand Unstable LIMK2 21 46 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCCC(C)(C)C ZINC000217519748 BI For-Sale Unstable TRPM8 15 44 COc1ccc(CC(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc1 ZINC000217519760 GG For-Sale Unstable DRD4 41 32 COc1ccc(CC(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc1 ZINC000217519760 GG For-Sale Unstable CA9 16 41 O=C(Nc1ccc(N2CCOCC2)cc1N1CCOCC1)[C@@H]1C[C@H]1c1ccccc1Cl ZINC000217519779 IH On-Demand Unstable CSF1R 15 43 O=C(Nc1ccc(N2CCOCC2)cc1N1CCOCC1)[C@@H]1C[C@H]1c1ccccc1Cl ZINC000217519779 IH On-Demand Unstable AKR1C3 27 42 CCOC(=O)NCCNC(=O)NCCc1ccc(OC)cc1 ZINC000217519781 DD For-Sale Unstable CA2 17 51 CCOC(=O)NCCNC(=O)NCCc1ccc(OC)cc1 ZINC000217519781 DD For-Sale Unstable CA1 20 51 CCOC(=O)NCCNC(=O)NCCc1ccc(OC)cc1 ZINC000217519781 DD For-Sale Unstable MTNR1A 85 46 CCOC(=O)NCCNC(=O)NCCc1ccc(OC)cc1 ZINC000217519781 DD For-Sale Unstable MTNR1B 66 42 CCOC(=O)NCCNC(=O)NCCc1ccc(OC)cc1 ZINC000217519781 DD For-Sale Unstable CA12 17 51 CCOC(=O)NCCNC(=O)NCCc1ccc(OC)cc1 ZINC000217519781 DD For-Sale Unstable PTGDR 20 41 CCOC(=O)NCCNC(=O)NCCc1ccc(OC)cc1 ZINC000217519781 DD For-Sale Unstable CA9 23 51 CCOC(=O)NCCNC(=O)NCCc1ccc(OC)cc1 ZINC000217519781 DD For-Sale Unstable MMP1 15 42 CCOC(=O)NCCNC(=O)NCCc1ccc(OC)cc1 ZINC000217519781 DD For-Sale Unstable PROKR1 64 37 CC(=O)c1cccc(NC(=O)N[C@@H]2CCN3CCC[C@@H]23)c1 ZINC000217519787 CE For-Sale Unstable CCR3 56 52 CC(=O)c1cccc(NC(=O)N[C@@H]2CCN3CCC[C@@H]23)c1 ZINC000217519787 CE For-Sale Unstable CCKBR 40 40 CC(=O)c1cccc(NC(=O)N[C@@H]2CCN3CCC[C@@H]23)c1 ZINC000217519787 CE For-Sale Unstable EPHX2 34 52 CC(=O)c1cccc(NC(=O)N[C@@H]2CCN3CCC[C@@H]23)c1 ZINC000217519787 CE For-Sale Unstable AKR1C3 26 44 CC(=O)c1cccc(NC(=O)N[C@@H]2CCN3CCC[C@@H]23)c1 ZINC000217519787 CE For-Sale Unstable KCNK3 43 35 COc1ccc(CCNc2ccc(C(=O)O)cc2S(=O)(=O)NCCC(C)C)cc1 ZINC000217519794 HG In-Stock Unstable MMP3 23 40 COc1ccc(CCNc2ccc(C(=O)O)cc2S(=O)(=O)NCCC(C)C)cc1 ZINC000217519794 HG In-Stock Unstable PTGDR 26 40 COc1ccc(CCNc2ccc(C(=O)O)cc2S(=O)(=O)NCCC(C)C)cc1 ZINC000217519794 HG In-Stock Unstable AKR1C3 22 45 C#CCN1[C@H]2CC[C@@H](OC(=O)C(O)(c3ccccc3)c3ccccc3)[C@H]1CC2 ZINC000217519805 GG For-Sale Unstable CHRM2 32 50 C#CCN1[C@H]2CC[C@@H](OC(=O)C(O)(c3ccccc3)c3ccccc3)[C@H]1CC2 ZINC000217519805 GG For-Sale Unstable CHRM1 38 50 C#CCN1[C@H]2CC[C@@H](OC(=O)C(O)(c3ccccc3)c3ccccc3)[C@H]1CC2 ZINC000217519805 GG For-Sale Unstable CHRM3 46 50 C#CCN1[C@H]2CC[C@@H](OC(=O)C(O)(c3ccccc3)c3ccccc3)[C@H]1CC2 ZINC000217519805 GG For-Sale Unstable AMY2 43 29 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1N[C@@H](C)c1ccc(F)cc1O ZINC000217519808 CJ For-Sale Unstable TRPM8 16 44 Cc1cc(CBr)ccc1N(C)CCN1CCCC1 ZINC000217519821 DG For-Sale Unstable HRH3 15 42 Cc1cc(CBr)ccc1N(C)CCN1CCCC1 ZINC000217519821 DG For-Sale Unstable SIGMAR1 18 46 O=C1OC2(CCN(C(=O)CNS(=O)(=O)c3c(Cl)cccc3Cl)CC2)c2ccccc21 ZINC000217519827 JF For-Sale Unstable NPY5R 45 52 O=C(Nc1ccc(N2CCOCC2)cc1N1CCOCC1)[C@H]1C[C@H]1c1ccccc1Cl ZINC000217519864 IH On-Demand Unstable CSF1R 15 43 O=C(Nc1ccc(N2CCOCC2)cc1N1CCOCC1)[C@H]1C[C@H]1c1ccccc1Cl ZINC000217519864 IH On-Demand Unstable AKR1C3 27 42 CCOc1ccccc1C(=O)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217519872 GH For-Sale Unstable FABP4 41 35 CCOc1ccccc1C(=O)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217519872 GH For-Sale Unstable HCN1 79 43 CCOc1ccccc1C(=O)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217519872 GH For-Sale Unstable HCN4 59 40 CCOc1ccccc1C(=O)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217519872 GH For-Sale Unstable KCNK3 26 41 CCOc1ccccc1C(=O)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217519872 GH For-Sale Unstable KCNK9 25 41 CC(=O)c1cccc(NC(=O)N[C@H]2CCN3CCC[C@@H]23)c1 ZINC000217519889 CE For-Sale Unstable CCR3 56 52 CC(=O)c1cccc(NC(=O)N[C@H]2CCN3CCC[C@@H]23)c1 ZINC000217519889 CE For-Sale Unstable CCKBR 40 40 CC(=O)c1cccc(NC(=O)N[C@H]2CCN3CCC[C@@H]23)c1 ZINC000217519889 CE For-Sale Unstable EPHX2 34 52 CC(=O)c1cccc(NC(=O)N[C@H]2CCN3CCC[C@@H]23)c1 ZINC000217519889 CE For-Sale Unstable AKR1C3 26 44 CC(=O)c1cccc(NC(=O)N[C@H]2CCN3CCC[C@@H]23)c1 ZINC000217519889 CE For-Sale Unstable KCNK3 43 35 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1N[C@@H](C)c1ccc(F)cc1O ZINC000217519893 CJ For-Sale Unstable TRPM8 16 44 COc1ccc(CCNC(=O)N(CCN)C(=O)OC(C)(C)C)cc1 ZINC000217519897 EE For-Sale Unstable MTNR1A 46 37 COc1ccc(CCNC(=O)N(CCN)C(=O)OC(C)(C)C)cc1 ZINC000217519897 EE For-Sale Unstable CA9 17 44 COc1ccc(CCNC(=O)N(CCN)C(=O)OC(C)(C)C)cc1 ZINC000217519897 EE For-Sale Unstable PROKR1 44 33 COc1ccc(CCNc2ccc(C(=O)O)cc2S(=O)(=O)NCCC(C)C)cc1OC ZINC000217519903 JG In-Stock Unstable PTGDR 19 44 COc1ccc(CCNc2ccc(C(=O)O)cc2S(=O)(=O)NCCC(C)C)cc1OC ZINC000217519903 JG In-Stock Unstable SCMU_MYCTU 0 49 CCC(CC)NC(=O)c1cc(Br)ccc1O ZINC000217519915 CG On-Demand Unstable PYK 83 44 CN(CCN1CCCC1)c1ccccc1CBr ZINC000217519924 CG For-Sale Unstable HRH3 15 51 CN(CCN1CCCC1)c1ccccc1CBr ZINC000217519924 CG For-Sale Unstable SIGMAR1 17 47 CN(CCN1CCCC1)c1ccccc1CBr ZINC000217519924 CG For-Sale Unstable HNMT 24 51 O=C1OC2(CCN(C(=O)CCNS(=O)(=O)c3c(Cl)cccc3Cl)CC2)c2ccccc21 ZINC000217519942 JG For-Sale Unstable NPY5R 38 50 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1N[C@@H](C)c1ccc(F)cc1O ZINC000217519969 CJ For-Sale Unstable TRPM8 16 44 CCOc1ccc(C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc1 ZINC000217519987 GH For-Sale Unstable DGAT1 17 57 CC/C=C\C(=O)CCc1ccc(O)c(OC)c1 ZINC000217519996 BF Annotated Unstable NA 0 40 CC/C=C\C(=O)CCc1ccc(O)c(OC)c1 ZINC000217519996 BF Annotated Unstable INHA 47 33 CC/C=C\C(=O)CCc1ccc(O)c(OC)c1 ZINC000217519996 BF Annotated Unstable TRPV1 0 75 CC/C=C\C(=O)CCc1ccc(O)c(OC)c1 ZINC000217519996 BF Annotated Unstable SHBG 19 42 CC/C=C\C(=O)CCc1ccc(O)c(OC)c1 ZINC000217519996 BF Annotated Unstable ALOX15 0 43 CC/C=C\C(=O)CCc1ccc(O)c(OC)c1 ZINC000217519996 BF Annotated Unstable NCE103 21 47 CC/C=C\C(=O)CCc1ccc(O)c(OC)c1 ZINC000217519996 BF Annotated Unstable MTCA1 18 47 CC/C=C\C(=O)CCc1ccc(O)c(OC)c1 ZINC000217519996 BF Annotated Unstable CAN2 0 47 O=C(NCCc1ccc(F)cc1)Nc1cccc(C(=O)O)c1 ZINC000217520003 DF For-Sale Unstable PPIA 25 45 O=C(NCCc1ccc(F)cc1)Nc1cccc(C(=O)O)c1 ZINC000217520003 DF For-Sale Unstable CCR3 95 53 O=C(NCCc1ccc(F)cc1)Nc1cccc(C(=O)O)c1 ZINC000217520003 DF For-Sale Unstable RAF1 35 48 O=C(NCCc1ccc(F)cc1)Nc1cccc(C(=O)O)c1 ZINC000217520003 DF For-Sale Unstable ROCK2 15 47 O=C(NCCc1ccc(F)cc1)Nc1cccc(C(=O)O)c1 ZINC000217520003 DF For-Sale Unstable CCKBR 18 40 O=C(NCCc1ccc(F)cc1)Nc1cccc(C(=O)O)c1 ZINC000217520003 DF For-Sale Unstable EPHX2 34 49 O=C(NCCc1ccc(F)cc1)Nc1cccc(C(=O)O)c1 ZINC000217520003 DF For-Sale Unstable Q8MMZ8_EIMTE 24 48 O=C(NCCc1ccc(F)cc1)Nc1cccc(C(=O)O)c1 ZINC000217520003 DF For-Sale Unstable AKR1C3 41 43 O=C(NCCc1ccc(F)cc1)Nc1cccc(C(=O)O)c1 ZINC000217520003 DF For-Sale Unstable NCE103 21 44 O=C(NCCc1ccc(F)cc1)Nc1cccc(C(=O)O)c1 ZINC000217520003 DF For-Sale Unstable PRMT3 49 41 O=C(NCCc1ccc(F)cc1)Nc1cccc(C(=O)O)c1 ZINC000217520003 DF For-Sale Unstable KDM4E 22 44 O=C(NCCc1ccc(F)cc1)Nc1cccc(C(=O)O)c1 ZINC000217520003 DF For-Sale Unstable KCNK3 76 48 O=C(NCCc1ccc(F)cc1)Nc1cccc(C(=O)O)c1 ZINC000217520003 DF For-Sale Unstable KCNK9 44 36 CC(=O)c1ccc(NC(=O)N[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217520014 CE For-Sale Unstable EPHX2 40 43 CC(=O)c1ccc(NC(=O)N[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217520014 CE For-Sale Unstable L3MBTL3 42 33 CCC(CC)NC(=O)c1cc(I)ccc1O ZINC000217520034 EF For-Sale Unstable PYK 19 40 CCC(CC)NC(=O)c1cc(I)ccc1O ZINC000217520034 EF For-Sale Unstable Q25615_ONCVO 48 35 CN(CCN1CCCC1)c1ccc(CBr)cn1 ZINC000217520056 CF For-Sale Unstable HRH3 20 46 CN(CCN1CCCC1)c1ccc(CBr)cn1 ZINC000217520056 CF For-Sale Unstable SIGMAR1 15 45 CN(CCN1CCCC1)c1ccc(CBr)cn1 ZINC000217520056 CF For-Sale Unstable HNMT 19 42 CN(CCN1CCCC1)c1ccc(CBr)cn1 ZINC000217520056 CF For-Sale Unstable TLR7 17 46 CC(C)[C@H]1CC[C@H](C)C[C@@H]1N[C@@H](C)c1ccc(F)cc1O ZINC000217520057 CJ For-Sale Unstable TRPM8 0 44 COc1ccc(C(=O)NC2CCN(C(=O)N3CCOCC3)CC2)cc1C ZINC000217520064 FD In-Stock Unstable CNR2 15 42 COc1ccc(C(=O)NC2CCN(C(=O)N3CCOCC3)CC2)cc1C ZINC000217520064 FD In-Stock Unstable MAPK11 34 40 COc1ccc(C(=O)NC2CCN(C(=O)N3CCOCC3)CC2)cc1C ZINC000217520064 FD In-Stock Unstable MAPK14 45 44 COc1ccc(C(=O)NC2CCN(C(=O)N3CCOCC3)CC2)cc1C ZINC000217520064 FD In-Stock Unstable MAPK13 53 39 COc1ccc(C(=O)NC2CCN(C(=O)N3CCOCC3)CC2)cc1C ZINC000217520064 FD In-Stock Unstable MCHR1 16 45 COc1ccc(C(=O)NC2CCN(C(=O)N3CCOCC3)CC2)cc1C ZINC000217520064 FD In-Stock Unstable CCR8 17 40 O=C1OC2(CCN(C(=O)CCNS(=O)(=O)c3cccc(Cl)c3)CC2)c2ccccc21 ZINC000217520065 IF For-Sale Unstable NPY5R 30 52 COc1cccc(CC(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)c1 ZINC000217520093 GG For-Sale Unstable DRD4 50 39 COc1cccc(CC(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)c1 ZINC000217520093 GG For-Sale Unstable FABP4 30 43 COc1cccc(CC(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)c1 ZINC000217520093 GG For-Sale Unstable MTNR1A 31 40 COc1cccc(CC(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)c1 ZINC000217520093 GG For-Sale Unstable MTNR1B 30 40 CC(=O)c1ccc(NC(=O)N[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217520111 CE For-Sale Unstable EPHX2 40 43 CC(=O)c1ccc(NC(=O)N[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217520111 CE For-Sale Unstable L3MBTL3 42 33 Fc1ccc(CC2CCNCC2)c(Cl)c1F ZINC000217520148 BG For-Sale Unstable SLC6A2 15 51 CC(C)[C@H]1CC[C@H](C)C[C@H]1N[C@H](C)Cc1ccccc1 ZINC000217520150 CJ For-Sale Unstable TRPM8 18 53 CN(CCN1CCCC1)c1ccc(CBr)cc1F ZINC000217520161 DG For-Sale Unstable SIGMAR1 15 47 Cc1cccc(S(=O)(=O)Nc2ccc(C(=O)N3CCC4(CC3)OC(=O)c3ccccc34)cc2)c1 ZINC000217520166 JI For-Sale Unstable NPY5R 30 44 C[C@@](O)(CNC(=O)C(=O)Nc1ccc(OC(F)(F)F)cc1)c1cc2ccccc2s1 ZINC000217520225 IH In-Stock Unstable P2RY1 60 41 C[C@@](O)(CNC(=O)C(=O)Nc1ccc(OC(F)(F)F)cc1)c1cc2ccccc2s1 ZINC000217520225 IH In-Stock Unstable EPHX2 46 36 CC(=O)c1ccc(Br)cc1N1C[C@@H]2CCCCN2C[C@@H]1C ZINC000217520227 FH For-Sale Unstable L3MBTL3 50 38 O=C(NCCc1ccc(F)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217520230 EE For-Sale Unstable CA2 48 59 O=C(NCCc1ccc(F)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217520230 EE For-Sale Unstable ADRB3 18 42 O=C(NCCc1ccc(F)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217520230 EE For-Sale Unstable CA1 52 59 O=C(NCCc1ccc(F)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217520230 EE For-Sale Unstable CA7 30 50 O=C(NCCc1ccc(F)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217520230 EE For-Sale Unstable CCR3 45 52 O=C(NCCc1ccc(F)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217520230 EE For-Sale Unstable RAF1 27 43 O=C(NCCc1ccc(F)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217520230 EE For-Sale Unstable CA4 30 59 O=C(NCCc1ccc(F)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217520230 EE For-Sale Unstable CA5A 24 50 O=C(NCCc1ccc(F)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217520230 EE For-Sale Unstable CA14 29 50 O=C(NCCc1ccc(F)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217520230 EE For-Sale Unstable CA12 54 56 O=C(NCCc1ccc(F)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217520230 EE For-Sale Unstable CA9 54 53 O=C(NCCc1ccc(F)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217520230 EE For-Sale Unstable Q8MMZ8_EIMTE 0 43 O=C(NCCc1ccc(F)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217520230 EE For-Sale Unstable LEF 41 35 O=C(NCCc1ccc(F)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217520230 EE For-Sale Unstable IDO1 30 44 O=C(NCCc1ccc(F)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217520230 EE For-Sale Unstable NCE103 47 59 O=C(NCCc1ccc(F)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217520230 EE For-Sale Unstable PFK 0 44 O=C(NCCc1ccc(F)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217520230 EE For-Sale Unstable MTCA1 48 51 O=C(NCCc1ccc(F)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217520230 EE For-Sale Unstable P96878_MYCTU 63 51 O=C(NCCc1ccc(F)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217520230 EE For-Sale Unstable NAMPT 48 46 O=C(NCCc1ccc(F)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217520230 EE For-Sale Unstable A6YCJ1_9METZ 15 42 COc1ccc(NS(=O)(=O)[C@@H](C)CO)cc1OC ZINC000217520236 CC For-Sale Unstable ENPP1 75 36 CC(C)[C@H]1CC[C@H](C)C[C@@H]1N[C@@H](C)Cc1ccccc1 ZINC000217520243 CJ For-Sale Unstable TRPM8 18 53 FC(F)c1c(Cl)cccc1C[C@@H]1CCNC1 ZINC000217520253 BG For-Sale Unstable SLC6A2 25 41 Cc1cccc(S(=O)(=O)NCC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217520274 HD For-Sale Unstable NPY5R 32 48 C[C@](O)(CNC(=O)C(=O)Nc1ccc(OC(F)(F)F)cc1)c1cc2ccccc2s1 ZINC000217520299 IH In-Stock Unstable P2RY1 60 41 C[C@](O)(CNC(=O)C(=O)Nc1ccc(OC(F)(F)F)cc1)c1cc2ccccc2s1 ZINC000217520299 IH In-Stock Unstable EPHX2 46 36 COc1ccc(NS(=O)(=O)[C@H](C)CO)cc1OC ZINC000217520312 CC For-Sale Unstable ENPP1 75 36 FC(F)c1c(Cl)cccc1C[C@H]1CCNC1 ZINC000217520329 BG For-Sale Unstable SLC6A2 25 41 O=C(NCCc1ccc(F)cc1)Nc1cccc(S(=O)(=O)O)c1 ZINC000217520341 EE For-Sale Unstable CA2 27 54 O=C(NCCc1ccc(F)cc1)Nc1cccc(S(=O)(=O)O)c1 ZINC000217520341 EE For-Sale Unstable CA1 28 54 O=C(NCCc1ccc(F)cc1)Nc1cccc(S(=O)(=O)O)c1 ZINC000217520341 EE For-Sale Unstable CA7 15 47 O=C(NCCc1ccc(F)cc1)Nc1cccc(S(=O)(=O)O)c1 ZINC000217520341 EE For-Sale Unstable CCR3 85 55 O=C(NCCc1ccc(F)cc1)Nc1cccc(S(=O)(=O)O)c1 ZINC000217520341 EE For-Sale Unstable RAF1 26 48 O=C(NCCc1ccc(F)cc1)Nc1cccc(S(=O)(=O)O)c1 ZINC000217520341 EE For-Sale Unstable CA4 24 54 O=C(NCCc1ccc(F)cc1)Nc1cccc(S(=O)(=O)O)c1 ZINC000217520341 EE For-Sale Unstable CA5A 16 47 O=C(NCCc1ccc(F)cc1)Nc1cccc(S(=O)(=O)O)c1 ZINC000217520341 EE For-Sale Unstable EPHX2 17 41 O=C(NCCc1ccc(F)cc1)Nc1cccc(S(=O)(=O)O)c1 ZINC000217520341 EE For-Sale Unstable CA12 28 49 O=C(NCCc1ccc(F)cc1)Nc1cccc(S(=O)(=O)O)c1 ZINC000217520341 EE For-Sale Unstable CA9 27 46 O=C(NCCc1ccc(F)cc1)Nc1cccc(S(=O)(=O)O)c1 ZINC000217520341 EE For-Sale Unstable Q8MMZ8_EIMTE 0 48 O=C(NCCc1ccc(F)cc1)Nc1cccc(S(=O)(=O)O)c1 ZINC000217520341 EE For-Sale Unstable NCE103 27 48 O=C(NCCc1ccc(F)cc1)Nc1cccc(S(=O)(=O)O)c1 ZINC000217520341 EE For-Sale Unstable NAMPT 27 40 CC(C)[C@H]1CC[C@H](C)C[C@@H]1N[C@H](C)Cc1ccccc1 ZINC000217520343 CJ For-Sale Unstable TRPM8 18 53 CC(C)CCNS(=O)(=O)c1cc(C(=O)O)ccc1N1CCCC1 ZINC000217520344 EE In-Stock Unstable KCNQ2 71 36 O=C(Nc1ccc(N2CCOCC2)cc1N1CCOCC1)[C@@H]1C[C@@H]1c1ccccc1C(F)(F)F ZINC000217520362 JI On-Demand Unstable PTK2 15 40 O=C(Nc1ccc(N2CCOCC2)cc1N1CCOCC1)[C@@H]1C[C@@H]1c1ccccc1C(F)(F)F ZINC000217520362 JI On-Demand Unstable RBP4 87 39 Cc1cccc(S(=O)(=O)NC2(C(=O)N3CCC4(CC3)OC(=O)c3ccccc34)CCCCC2)c1 ZINC000217520388 JH For-Sale Unstable NPY5R 30 42 CC(=O)c1ccc(Br)cc1N1C[C@@H]2CCCN2C[C@@H]1C ZINC000217520413 EG For-Sale Unstable L3MBTL3 50 36 O=C(Nc1ccc(N2CCOCC2)cc1N1CCOCC1)[C@H]1C[C@@H]1c1ccccc1C(F)(F)F ZINC000217520440 JI On-Demand Unstable PTK2 15 40 O=C(Nc1ccc(N2CCOCC2)cc1N1CCOCC1)[C@H]1C[C@@H]1c1ccccc1C(F)(F)F ZINC000217520440 JI On-Demand Unstable RBP4 87 39 O=C(NCCc1ccc(F)cc1)Nc1ccc(C(=O)O)cc1 ZINC000217520463 DF For-Sale Unstable CA2 15 56 O=C(NCCc1ccc(F)cc1)Nc1ccc(C(=O)O)cc1 ZINC000217520463 DF For-Sale Unstable ADRB1 25 42 O=C(NCCc1ccc(F)cc1)Nc1ccc(C(=O)O)cc1 ZINC000217520463 DF For-Sale Unstable LTA4H 23 45 O=C(NCCc1ccc(F)cc1)Nc1ccc(C(=O)O)cc1 ZINC000217520463 DF For-Sale Unstable CA1 19 51 O=C(NCCc1ccc(F)cc1)Nc1ccc(C(=O)O)cc1 ZINC000217520463 DF For-Sale Unstable CCR3 55 47 O=C(NCCc1ccc(F)cc1)Nc1ccc(C(=O)O)cc1 ZINC000217520463 DF For-Sale Unstable RAF1 31 40 O=C(NCCc1ccc(F)cc1)Nc1ccc(C(=O)O)cc1 ZINC000217520463 DF For-Sale Unstable EPHX2 29 45 O=C(NCCc1ccc(F)cc1)Nc1ccc(C(=O)O)cc1 ZINC000217520463 DF For-Sale Unstable CA12 19 51 O=C(NCCc1ccc(F)cc1)Nc1ccc(C(=O)O)cc1 ZINC000217520463 DF For-Sale Unstable CA9 19 56 O=C(NCCc1ccc(F)cc1)Nc1ccc(C(=O)O)cc1 ZINC000217520463 DF For-Sale Unstable PRMT3 39 41 O=C(NCCc1ccc(F)cc1)Nc1ccc(C(=O)O)cc1 ZINC000217520463 DF For-Sale Unstable P96878_MYCTU 19 40 CC(C)CCNS(=O)(=O)c1cc(C(=O)O)ccc1N1CCCCC1 ZINC000217520466 FF In-Stock Unstable KCNQ2 68 36 Cc1cccc(CN[C@H]2C[C@H](C)CC[C@H]2C(C)C)c1C ZINC000217520481 CJ For-Sale Unstable TRPM8 16 43 Cc1cccc(S(=O)(=O)NCCC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217520504 IE For-Sale Unstable NPY5R 29 45 O=C(Nc1ccc(N2CCOCC2)cc1N1CCOCC1)[C@@H]1C[C@H]1c1ccccc1C(F)(F)F ZINC000217520533 JI On-Demand Unstable PTK2 15 40 O=C(Nc1ccc(N2CCOCC2)cc1N1CCOCC1)[C@@H]1C[C@H]1c1ccccc1C(F)(F)F ZINC000217520533 JI On-Demand Unstable RBP4 87 39 Cc1cccc(CN[C@H]2C[C@@H](C)CC[C@H]2C(C)C)c1C ZINC000217520576 CJ For-Sale Unstable TRPM8 16 43 O=C(NCCc1ccc(F)cc1)Nc1cccc(Cl)c1Cl ZINC000217520577 EI On-Demand Unstable TRPV1 15 49 O=C(NCCc1ccc(F)cc1)Nc1cccc(Cl)c1Cl ZINC000217520577 EI On-Demand Unstable CCR3 30 40 NC(=O)[C@@H](O[C@@H]1CCCNC1)c1cccc(Cl)c1 ZINC000217520602 CD In-Stock Unstable SLC6A2 20 41 O=C1OC2(CCN(C(=O)CNS(=O)(=O)c3ccc(F)c(Cl)c3)CC2)c2ccccc21 ZINC000217520613 JE For-Sale Unstable NPY5R 35 47 O=C(Nc1ccc(N2CCOCC2)cc1N1CCOCC1)[C@H]1C[C@H]1c1ccccc1C(F)(F)F ZINC000217520620 JI On-Demand Unstable PTK2 15 40 O=C(Nc1ccc(N2CCOCC2)cc1N1CCOCC1)[C@H]1C[C@H]1c1ccccc1C(F)(F)F ZINC000217520620 JI On-Demand Unstable RBP4 87 39 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1cccc([N+](=O)[O-])c1 ZINC000217520650 GG For-Sale Unstable DRD4 42 33 Cc1ccc(C)c(CN[C@H]2C[C@H](C)CC[C@H]2C(C)C)c1 ZINC000217520664 CJ For-Sale Unstable TRPM8 16 46 NC(=O)[C@H](O[C@@H]1CCCNC1)c1cccc(Cl)c1 ZINC000217520683 CD In-Stock Unstable SLC6A2 20 41 CCOC(=O)c1ccccc1NC(=O)NCCc1ccc(F)cc1 ZINC000217520690 EG For-Sale Unstable CCR3 44 38 CCOC(=O)c1ccccc1NC(=O)NCCc1ccc(F)cc1 ZINC000217520690 EG For-Sale Unstable NCE103 15 41 O=C1OC2(CCN(C(=O)CCNS(=O)(=O)c3ccc(F)c(Cl)c3)CC2)c2ccccc21 ZINC000217520715 JF For-Sale Unstable TBXA2R 41 33 O=C1OC2(CCN(C(=O)CCNS(=O)(=O)c3ccc(F)c(Cl)c3)CC2)c2ccccc21 ZINC000217520715 JF For-Sale Unstable NPY5R 33 49 Cc1nc2ccccc2cc1C(=O)Nc1ccc(N2CCOCC2)cc1N1CCOCC1 ZINC000217520723 IG On-Demand Unstable PIK3CD 28 45 Cc1nc2ccccc2cc1C(=O)Nc1ccc(N2CCOCC2)cc1N1CCOCC1 ZINC000217520723 IG On-Demand Unstable PIK3CB 36 45 Cc1nc2ccccc2cc1C(=O)Nc1ccc(N2CCOCC2)cc1N1CCOCC1 ZINC000217520723 IG On-Demand Unstable CSF1R 21 48 Cc1nc2ccccc2cc1C(=O)Nc1ccc(N2CCOCC2)cc1N1CCOCC1 ZINC000217520723 IG On-Demand Unstable EPHB3 20 43 Cc1nc2ccccc2cc1C(=O)Nc1ccc(N2CCOCC2)cc1N1CCOCC1 ZINC000217520723 IG On-Demand Unstable STAT6 52 32 C[C@H](c1nc2ccccc2n1C)N1CCC[C@@H](CN)C1 ZINC000217520755 CE For-Sale Unstable HRH1 16 41 Cc1ccc(C)c(CN[C@H]2C[C@@H](C)CC[C@H]2C(C)C)c1 ZINC000217520762 CJ For-Sale Unstable TRPM8 16 46 NC(=O)[C@@H](O[C@H]1CCCNC1)c1cccc(Cl)c1 ZINC000217520775 CD In-Stock Unstable SLC6A2 20 41 O=C(NCCc1ccc(F)cc1)Nc1ccc(O)cc1 ZINC000217520777 CF On-Demand Unstable NCE103 26 50 FC(F)c1ccc(Cl)c(C[C@@H]2CCNC2)c1 ZINC000217520801 BG For-Sale Unstable SLC6A2 16 43 Cc1nn(C)c(C)c1CC(=O)Nc1ccc(N2CCOCC2)cc1N1CCOCC1 ZINC000217520830 HD On-Demand Unstable P2RX7 21 42 C[C@@H](c1nc2ccccc2n1C)N1CCC[C@@H](CN)C1 ZINC000217520842 CE For-Sale Unstable HRH1 16 41 O=C1OC2(CCN(C(=O)CCNS(=O)(=O)c3cccc(F)c3)CC2)c2ccccc21 ZINC000217520845 IE For-Sale Unstable NPY5R 38 52 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCC[C@@H](C)c1ccccc1 ZINC000217520853 CK For-Sale Unstable TRPM8 17 46 CN(CCN1CCCC1)c1ccc(CBr)cc1 ZINC000217520858 CG For-Sale Unstable HRH3 18 41 CN(CCN1CCCC1)c1ccc(CBr)cc1 ZINC000217520858 CG For-Sale Unstable SIGMAR1 17 50 Cc1cc(=O)c(C(=O)N2CCC[C@@H](N(C)C)CC2)c[nH]1 ZINC000217520860 CD In-Stock Unstable L3MBTL1 0 42 Cc1cc(=O)c(C(=O)N2CCC[C@@H](N(C)C)CC2)c[nH]1 ZINC000217520860 CD In-Stock Unstable L3MBTL3 33 42 NC(=O)[C@H](O[C@H]1CCCNC1)c1cccc(Cl)c1 ZINC000217520869 CD In-Stock Unstable SLC6A2 20 41 CC(C)(C)OC(=O)NCCNC(=O)c1cc(I)cc(I)c1I ZINC000217520871 KH For-Sale Unstable Q25615_ONCVO 63 35 FC(F)c1ccc(Cl)c(C[C@H]2CCNC2)c1 ZINC000217520878 BG For-Sale Unstable SLC6A2 16 43 O=C(NCCc1ccc(F)cc1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217520891 HI For-Sale Unstable OPRD1 25 52 O=C(NCCc1ccc(F)cc1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217520891 HI For-Sale Unstable OPRK1 0 52 O=C(NCCc1ccc(F)cc1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217520891 HI For-Sale Unstable OPRL1 22 44 O=C(NCCc1ccc(F)cc1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217520891 HI For-Sale Unstable SLC6A3 21 52 O=C(NCCc1ccc(F)cc1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217520891 HI For-Sale Unstable MC4R 41 39 O=C(NCCc1ccc(F)cc1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217520891 HI For-Sale Unstable CCR3 33 44 O=C(NCCc1ccc(F)cc1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217520891 HI For-Sale Unstable DPP8 15 45 O=C(NCCc1ccc(F)cc1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217520891 HI For-Sale Unstable CACNA1G 32 43 O=C(NCCc1ccc(F)cc1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217520891 HI For-Sale Unstable NPSR1 24 42 O=C(NCCc1ccc(F)cc1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217520891 HI For-Sale Unstable NMUR2 0 58 O=C(NCCc1ccc(F)cc1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217520891 HI For-Sale Unstable NMUR1 0 58 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCC[C@@H](C)c1ccccc1 ZINC000217520931 CK For-Sale Unstable TRPM8 17 46 Cc1cc(=O)c(C(=O)N2CCC[C@H](N(C)C)CC2)c[nH]1 ZINC000217520939 CD In-Stock Unstable L3MBTL1 0 42 Cc1cc(=O)c(C(=O)N2CCC[C@H](N(C)C)CC2)c[nH]1 ZINC000217520939 CD In-Stock Unstable L3MBTL3 33 42 Cc1nc2ccccc2cc1C(=O)Nc1cccc(-n2cnnn2)c1 ZINC000217520951 EF On-Demand Unstable SHH 42 37 Cc1nc2ccccc2cc1C(=O)Nc1cccc(-n2cnnn2)c1 ZINC000217520951 EF On-Demand Unstable KCNK3 80 40 Cc1nc2ccccc2cc1C(=O)Nc1cccc(-n2cnnn2)c1 ZINC000217520951 EF On-Demand Unstable KCNK9 77 38 O=C1OC2(CCN(C(=O)CNS(=O)(=O)c3c(F)cccc3F)CC2)c2ccccc21 ZINC000217520954 ID For-Sale Unstable NPY5R 44 52 CSc1ccccc1C(=O)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217520973 GH For-Sale Unstable FABP4 45 34 COC(=O)[C@@H](CC(C)C)NC(=O)CN1CCC[C@@H](N)C1 ZINC000217521005 CC For-Sale Unstable NPR 15 40 CCOCCCNC(=O)NCCc1ccc(F)cc1 ZINC000217521006 CE On-Demand Unstable CNR2 29 40 CCOCCCNC(=O)NCCc1ccc(F)cc1 ZINC000217521006 CE On-Demand Unstable CXCR2 16 40 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCC[C@@H](C)c1ccccc1 ZINC000217521011 CK For-Sale Unstable TRPM8 17 46 O=C1OC2(CCN(C(=O)CCNS(=O)(=O)c3c(F)cccc3F)CC2)c2ccccc21 ZINC000217521077 JE For-Sale Unstable NPY5R 37 46 COC(=O)[C@H](CC(C)C)NC(=O)CN1CCC[C@@H](N)C1 ZINC000217521094 CC For-Sale Unstable NPR 15 40 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCC[C@@H](C)c1ccccc1 ZINC000217521100 CK For-Sale Unstable TRPM8 17 46 O=C(NCCc1ccc(F)cc1)N1CCCc2ccccc21 ZINC000217521130 CH For-Sale Unstable AVPR2 54 46 O=C(NCCc1ccc(F)cc1)N1CCCc2ccccc21 ZINC000217521130 CH For-Sale Unstable AVPR1A 15 41 O=C(NCCc1ccc(F)cc1)N1CCCc2ccccc21 ZINC000217521130 CH For-Sale Unstable KCNQ2 19 41 O=C(NCCc1ccc(F)cc1)N1CCCc2ccccc21 ZINC000217521130 CH For-Sale Unstable CCR3 29 42 O=C(NCCc1ccc(F)cc1)N1CCCc2ccccc21 ZINC000217521130 CH For-Sale Unstable AMP1_PLAFQ 16 43 O=C(O)[C@@H]1Cc2ccccc2CN1C(=O)c1cc(=O)[nH]c2ccc(F)cc12 ZINC000217521182 FE In-Stock Unstable AGTR2 48 43 O=C(O)[C@@H]1Cc2ccccc2CN1C(=O)c1cc(=O)[nH]c2ccc(F)cc12 ZINC000217521182 FE In-Stock Unstable CFTR 52 44 O=C(O)[C@@H]1Cc2ccccc2CN1C(=O)c1cc(=O)[nH]c2ccc(F)cc12 ZINC000217521182 FE In-Stock Unstable NR1D1 35 41 Cc1cc(C)c(C)c(S(=O)(=O)NCCC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1C ZINC000217521185 JG For-Sale Unstable NPY5R 31 46 CS(=O)(=O)c1ccc(Cl)cc1C1(N)CC1 ZINC000217521187 BD For-Sale Unstable AKR1B1 16 45 Cc1cc(C)cc(CN[C@H]2C[C@H](C)CC[C@H]2C(C)C)c1 ZINC000217521190 CJ For-Sale Unstable TRPM8 17 47 CN(CCN1CCCC1)c1cc(Cl)ccc1CBr ZINC000217521213 EH For-Sale Unstable SIGMAR1 17 47 CN(CCN1CCCC1)c1cc(Cl)ccc1CBr ZINC000217521213 EH For-Sale Unstable HNMT 52 42 Clc1ccc(-c2cnco2)c(Cl)c1 ZINC000217521226 BH For-Sale Anodyne ALPL 40 33 CN1CCC(N(C)C(=O)NCCc2ccc(F)cc2)CC1 ZINC000217521237 CE On-Demand Unstable HTR1F 43 34 CN1CCC(N(C)C(=O)NCCc2ccc(F)cc2)CC1 ZINC000217521237 CE On-Demand Unstable CCR3 55 46 CN1CCC(N(C)C(=O)NCCc2ccc(F)cc2)CC1 ZINC000217521237 CE On-Demand Unstable MCHR1 25 44 CN1CCC(N(C)C(=O)NCCc2ccc(F)cc2)CC1 ZINC000217521237 CE On-Demand Unstable CACNA1G 41 43 Cc1cc(C)cc(CN[C@H]2C[C@@H](C)CC[C@H]2C(C)C)c1 ZINC000217521275 CJ For-Sale Unstable TRPM8 17 47 O=C(O)[C@H]1Cc2ccccc2CN1C(=O)c1cc(=O)[nH]c2ccc(F)cc12 ZINC000217521276 FE In-Stock Unstable AGTR2 48 43 O=C(O)[C@H]1Cc2ccccc2CN1C(=O)c1cc(=O)[nH]c2ccc(F)cc12 ZINC000217521276 FE In-Stock Unstable CFTR 52 44 O=C(O)[C@H]1Cc2ccccc2CN1C(=O)c1cc(=O)[nH]c2ccc(F)cc12 ZINC000217521276 FE In-Stock Unstable NR1D1 35 41 O=C(/C=C\c1cc(Cl)ccc1Cl)N[C@@H]1CCC(=O)NC1=O ZINC000217521290 ED On-Demand Unstable BOTA 16 40 CC(C)(C)c1ccc(S(=O)(=O)NCCC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217521293 JG For-Sale Unstable NPY5R 26 43 CN(CCN1CCCC1)c1ccc(Cl)cc1CBr ZINC000217521335 EH For-Sale Unstable SIGMAR1 19 50 CN(CCN1CCCC1)c1ccc(Cl)cc1CBr ZINC000217521335 EH For-Sale Unstable HNMT 52 42 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCc1ccc(Cl)c(F)c1 ZINC000217521357 CK For-Sale Unstable SSTR3 0 40 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCc1ccc(Cl)c(F)c1 ZINC000217521357 CK For-Sale Unstable TRPM8 16 46 C[C@@H](NC(=O)NCCc1ccc(F)cc1)C12CC3CC(CC(C3)C1)C2 ZINC000217521363 EI For-Sale Unstable CCR3 20 43 C[C@@H](NC(=O)NCCc1ccc(F)cc1)C12CC3CC(CC(C3)C1)C2 ZINC000217521363 EI For-Sale Unstable EPHX2 70 61 O=C(/C=C\c1cc(Cl)ccc1Cl)N[C@H]1CCC(=O)NC1=O ZINC000217521369 ED On-Demand Unstable BOTA 16 40 O=C1OC2(CCN(C(=O)c3cccc(NS(=O)(=O)c4ccccc4F)c3)CC2)c2ccccc21 ZINC000217521402 JH For-Sale Unstable NPY5R 34 47 O=C(Cc1ccccc1Cl)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217521410 GH For-Sale Unstable P2RX7 53 37 C[C@H](NC(=O)NCCc1ccc(F)cc1)C12CC3CC(CC(C3)C1)C2 ZINC000217521443 EI For-Sale Unstable CCR3 20 43 C[C@H](NC(=O)NCCc1ccc(F)cc1)C12CC3CC(CC(C3)C1)C2 ZINC000217521443 EI For-Sale Unstable EPHX2 40 61 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCc1ccc(Cl)c(F)c1 ZINC000217521450 CK For-Sale Unstable SSTR3 0 40 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCc1ccc(Cl)c(F)c1 ZINC000217521450 CK For-Sale Unstable TRPM8 16 46 O=C1OC2(CCN(C(=O)c3cccc(NS(=O)(=O)c4cccc(F)c4)c3)CC2)c2ccccc21 ZINC000217521520 JH For-Sale Unstable NPY5R 35 51 C[C@@H](NC(=O)CN1CCC[C@@H](N)C1)c1ccc(F)cc1 ZINC000217521536 CD On-Demand Unstable CCR3 92 38 C[C@@H](NC(=O)CN1CCC[C@@H](N)C1)c1ccc(F)cc1 ZINC000217521536 CD On-Demand Unstable BIRC2 48 40 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1cccc2ccccc12 ZINC000217521537 GI For-Sale Unstable FABP4 54 40 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1cccc2ccccc12 ZINC000217521537 GI For-Sale Unstable POLR1A 42 39 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCc1ccc(Cl)c(F)c1 ZINC000217521542 CK For-Sale Unstable SSTR3 0 40 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCc1ccc(Cl)c(F)c1 ZINC000217521542 CK For-Sale Unstable TRPM8 16 46 O=C(NCCc1ccc(F)cc1)Nc1cccc2c(O)cccc12 ZINC000217521549 DI For-Sale Unstable PLA2G7 26 40 O=C(NCCc1ccc(F)cc1)Nc1cccc2c(O)cccc12 ZINC000217521549 DI For-Sale Unstable CA1 15 46 O=C(NCCc1ccc(F)cc1)Nc1cccc2c(O)cccc12 ZINC000217521549 DI For-Sale Unstable TRPV1 25 54 O=C(NCCc1ccc(F)cc1)Nc1cccc2c(O)cccc12 ZINC000217521549 DI For-Sale Unstable CA12 16 46 O=C(NCCc1ccc(F)cc1)Nc1cccc2c(O)cccc12 ZINC000217521549 DI For-Sale Unstable CA9 15 43 O=C(NCCc1ccc(F)cc1)Nc1cccc2c(O)cccc12 ZINC000217521549 DI For-Sale Unstable NCE103 26 42 C[C@H](c1cccc(Cl)c1)N1CCC[C@@H](CN)C1 ZINC000217521562 CG On-Demand Unstable OPRL1 0 44 C[C@H](NC(=O)CN1CCC[C@@H](N)C1)c1ccc(F)cc1 ZINC000217521620 CD On-Demand Unstable CCR3 92 38 C[C@H](NC(=O)CN1CCC[C@@H](N)C1)c1ccc(F)cc1 ZINC000217521620 CD On-Demand Unstable BIRC2 48 40 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCc1ccc(Cl)c(F)c1 ZINC000217521622 CK For-Sale Unstable SSTR3 0 40 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCc1ccc(Cl)c(F)c1 ZINC000217521622 CK For-Sale Unstable TRPM8 16 46 C[C@@H](c1cccc(Cl)c1)N1CCC[C@@H](CN)C1 ZINC000217521636 CG On-Demand Unstable OPRL1 0 44 COc1ccc(Br)cc1CCC(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217521639 II For-Sale Unstable NPY5R 29 49 CN1CCc2cc(S(=O)(=O)Cl)ccc2C1 ZINC000217521641 BD For-Sale Unstable DRD1 17 41 CN1CCc2cc(S(=O)(=O)Cl)ccc2C1 ZINC000217521641 BD For-Sale Unstable DRD5 40 41 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc2ccccc2c1 ZINC000217521650 GI For-Sale Unstable DRD4 43 33 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc2ccccc2c1 ZINC000217521650 GI For-Sale Unstable DRD3 19 44 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc2ccccc2c1 ZINC000217521650 GI For-Sale Unstable KCNJ11 52 34 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc2ccccc2c1 ZINC000217521650 GI For-Sale Unstable PLD1 38 41 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc2ccccc2c1 ZINC000217521650 GI For-Sale Unstable PLD2 66 42 Cc1cc(O)ccc1NC(=O)NCCc1ccc(F)cc1 ZINC000217521671 CG On-Demand Unstable TRPV1 0 50 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCc1ccc(O)c(Cl)c1 ZINC000217521718 CJ For-Sale Unstable TRPM8 18 48 COc1ccc([C@@H](C)NC(=O)NCCc2ccc(F)cc2)cc1 ZINC000217521757 DG On-Demand Unstable BMP1 24 44 COc1ccc([C@@H](C)NC(=O)NCCc2ccc(F)cc2)cc1 ZINC000217521757 DG On-Demand Unstable ACACA 23 45 COc1ccc([C@@H](C)NC(=O)NCCc2ccc(F)cc2)cc1 ZINC000217521757 DG On-Demand Unstable ACACB 31 44 COc1ccc([C@@H](C)NC(=O)NCCc2ccc(F)cc2)cc1 ZINC000217521757 DG On-Demand Unstable MTNR1A 49 39 COc1ccc([C@@H](C)NC(=O)NCCc2ccc(F)cc2)cc1 ZINC000217521757 DG On-Demand Unstable LEF 46 40 O=C1OC2(CCN(C(=O)CCc3ccc(Br)cc3)CC2)c2ccccc21 ZINC000217521760 HI For-Sale Unstable NPY5R 35 47 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1cnc2ccccc2n1 ZINC000217521762 GG For-Sale Unstable HTR3A 15 48 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCc1ccc(O)c(Cl)c1 ZINC000217521789 CJ For-Sale Unstable TRPM8 18 48 COc1ccc([C@H](C)NC(=O)NCCc2ccc(F)cc2)cc1 ZINC000217521862 DG On-Demand Unstable BMP1 24 44 COc1ccc([C@H](C)NC(=O)NCCc2ccc(F)cc2)cc1 ZINC000217521862 DG On-Demand Unstable ACACA 23 45 COc1ccc([C@H](C)NC(=O)NCCc2ccc(F)cc2)cc1 ZINC000217521862 DG On-Demand Unstable ACACB 31 44 COc1ccc([C@H](C)NC(=O)NCCc2ccc(F)cc2)cc1 ZINC000217521862 DG On-Demand Unstable MTNR1A 49 39 COc1ccc([C@H](C)NC(=O)NCCc2ccc(F)cc2)cc1 ZINC000217521862 DG On-Demand Unstable LEF 46 40 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCc1ccc(O)c(Cl)c1 ZINC000217521871 CJ For-Sale Unstable TRPM8 18 48 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc(F)cc1Cl ZINC000217521875 GI For-Sale Unstable P2RX7 52 41 CCCOc1ccc(CCC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217521882 GI For-Sale Unstable NPY5R 29 45 NCC1CCC(Nc2nc3ccccc3s2)CC1 ZINC000217521893 CG For-Sale Unstable ITK 17 44 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCc1ccc(O)c(Cl)c1 ZINC000217521943 CJ For-Sale Unstable TRPM8 18 48 O=C1OC2(CCN(C(=O)CCc3cccc(Cl)c3)CC2)c2ccccc21 ZINC000217521990 FH For-Sale Unstable NPY5R 34 48 Cc1cc(CN[C@H]2C[C@H](C)CC[C@H]2C(C)C)c(C)s1 ZINC000217522029 CJ For-Sale Unstable TRPM8 15 41 O=C1OC2(CCN(C(=O)CCc3ccc(Cl)cc3Cl)CC2)c2ccccc21 ZINC000217522097 HJ For-Sale Unstable AVPR1A 22 54 O=C1OC2(CCN(C(=O)CCc3ccc(Cl)cc3Cl)CC2)c2ccccc21 ZINC000217522097 HJ For-Sale Unstable MC4R 31 42 O=C1OC2(CCN(C(=O)CCc3ccc(Cl)cc3Cl)CC2)c2ccccc21 ZINC000217522097 HJ For-Sale Unstable NPY5R 41 52 Cc1cc(CN[C@H]2C[C@@H](C)CC[C@H]2C(C)C)c(C)s1 ZINC000217522102 CJ For-Sale Unstable TRPM8 15 41 C[C@@](O)(CNC(=O)Nc1ccccc1Cl)c1cc2ccccc2s1 ZINC000217522145 FJ In-Stock Unstable MAPK14 19 43 C[C@H](c1ccccc1Cl)N1CCC[C@@H](CN)C1 ZINC000217522161 CG On-Demand Unstable OPRL1 31 42 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1N[C@H](c1cccs1)C1CC1 ZINC000217522181 CK For-Sale Unstable TRPM8 15 41 C[C@@H](NC(=O)CN1CCC[C@@H](N)C1)c1ccccc1Cl ZINC000217522187 CD On-Demand Unstable SLC6A1 56 35 C[C@@H](NC(=O)CN1CCC[C@@H](N)C1)c1ccccc1Cl ZINC000217522187 CD On-Demand Unstable OPRL1 33 41 C[C@@H](NC(=O)CN1CCC[C@@H](N)C1)c1ccccc1Cl ZINC000217522187 CD On-Demand Unstable BIRC2 44 36 O=C1OC2(CCN(C(=O)CCc3c(Cl)cccc3Cl)CC2)c2ccccc21 ZINC000217522210 HJ For-Sale Unstable NPY5R 46 54 C[C@](O)(CNC(=O)Nc1ccccc1Cl)c1cc2ccccc2s1 ZINC000217522223 FJ In-Stock Unstable MAPK14 19 43 C[C@@H](c1ccccc1Cl)N1CCC[C@@H](CN)C1 ZINC000217522237 CG On-Demand Unstable OPRL1 31 42 C[C@H](NC(=O)CN1CCC[C@@H](N)C1)c1ccccc1Cl ZINC000217522256 CD On-Demand Unstable SLC6A1 56 35 C[C@H](NC(=O)CN1CCC[C@@H](N)C1)c1ccccc1Cl ZINC000217522256 CD On-Demand Unstable OPRL1 33 41 C[C@H](NC(=O)CN1CCC[C@@H](N)C1)c1ccccc1Cl ZINC000217522256 CD On-Demand Unstable BIRC2 44 36 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1N[C@H](c1cccs1)C1CC1 ZINC000217522260 CK For-Sale Unstable TRPM8 15 41 CC(=O)Nc1ccc(N2C[C@@]34C=C[C@@H](O3)[C@@H](C(=O)NCCc3c[nH]c5ccccc35)[C@@H]4C2=O)cc1 ZINC000217522268 JF In-Stock Unstable NMBR 46 30 COc1ccc(CCC(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc1 ZINC000217522313 GH For-Sale Unstable VIPR1 18 43 O=C1OC2(CCN(C(=O)CCc3ccc(Cl)c(Cl)c3)CC2)c2ccccc21 ZINC000217522334 HJ For-Sale Unstable SIGMAR1 15 51 O=C1OC2(CCN(C(=O)CCc3ccc(Cl)c(Cl)c3)CC2)c2ccccc21 ZINC000217522334 HJ For-Sale Unstable NPY5R 45 51 C[C@@](O)(CNC(=O)NCCCc1ccccc1)c1cc2ccccc2s1 ZINC000217522340 FI In-Stock Unstable MTNR1B 27 41 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1N[C@H](c1cccs1)C1CC1 ZINC000217522342 CK For-Sale Unstable TRPM8 15 41 CC(=O)Nc1ccc(N2C[C@]34C=C[C@@H](O3)[C@@H](C(=O)NCCc3c[nH]c5ccccc35)[C@@H]4C2=O)cc1 ZINC000217522352 JF In-Stock Unstable NMBR 46 30 CCc1ccc([C@@H](C)NC(=O)NCCc2ccc(F)cc2)cc1 ZINC000217522353 DH On-Demand Unstable ACACA 36 41 CCc1ccc([C@@H](C)NC(=O)NCCc2ccc(F)cc2)cc1 ZINC000217522353 DH On-Demand Unstable ACACB 16 41 C[C@](O)(CNC(=O)NCCCc1ccccc1)c1cc2ccccc2s1 ZINC000217522422 FI In-Stock Unstable MTNR1B 27 41 CC(C)[C@H]1CC[C@H](C)C[C@@H]1N[C@H](c1cccs1)C1CC1 ZINC000217522423 CK For-Sale Unstable TRPM8 15 41 CC(=O)Nc1ccc(N2C[C@]34C=C[C@@H](O3)[C@@H](C(=O)NCCc3c[nH]c5ccccc35)[C@H]4C2=O)cc1 ZINC000217522438 JF In-Stock Unstable NMBR 46 30 CCc1ccc([C@H](C)NC(=O)NCCc2ccc(F)cc2)cc1 ZINC000217522441 DH On-Demand Unstable ACACA 36 41 CCc1ccc([C@H](C)NC(=O)NCCc2ccc(F)cc2)cc1 ZINC000217522441 DH On-Demand Unstable ACACB 16 41 CCOc1ccccc1CCC(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217522446 GH For-Sale Unstable NPY5R 38 50 CCOc1ccccc1CCC(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217522446 GH For-Sale Unstable HCN1 48 33 CCOc1ccccc1CCC(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217522446 GH For-Sale Unstable HCN4 40 31 COc1cc2nc(N3CCn4nc(CO)cc4C3)nc(N)c2cc1OC ZINC000217522467 FC In-Stock Unstable ADRA1D 15 47 COc1cc2nc(N3CCn4nc(CO)cc4C3)nc(N)c2cc1OC ZINC000217522467 FC In-Stock Unstable ADRA1B 41 50 COc1cc2nc(N3CCn4nc(CO)cc4C3)nc(N)c2cc1OC ZINC000217522467 FC In-Stock Unstable EHMT2 49 33 N[C@H]1CS(=O)(=O)C[C@H]1c1ccc(Cl)cc1 ZINC000217522492 BD For-Sale Unstable SLC6A3 17 40 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCc1cccc(Br)c1O ZINC000217522519 EJ For-Sale Unstable TRPM8 17 44 C[C@@H]1Cc2ccccc2N1C(=O)CN1CCC[C@@H](N)C1 ZINC000217522551 CD On-Demand Unstable DRD4 39 57 C[C@@H]1Cc2ccccc2N1C(=O)CN1CCC[C@@H](N)C1 ZINC000217522551 CD On-Demand Unstable TPP2 59 36 O=C1OC2(CCN(C(=O)CCc3ccccc3F)CC2)c2ccccc21 ZINC000217522566 FG For-Sale Unstable NPY5R 41 48 N[C@H]1CS(=O)(=O)C[C@@H]1c1ccc(Cl)cc1 ZINC000217522583 BD For-Sale Unstable SLC6A3 17 40 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCc1cccc(Br)c1O ZINC000217522605 EJ For-Sale Unstable TRPM8 17 44 CC(C)COCCCNC[C@@H](O)c1ccc(C#N)cc1 ZINC000217522612 CE For-Sale Unstable ADRB1 25 40 CC(C)COCCCNC[C@@H](O)c1ccc(C#N)cc1 ZINC000217522612 CE For-Sale Unstable ADRB3 21 40 C[C@H]1Cc2ccccc2N1C(=O)CN1CCC[C@@H](N)C1 ZINC000217522632 CD On-Demand Unstable DRD4 39 57 C[C@H]1Cc2ccccc2N1C(=O)CN1CCC[C@@H](N)C1 ZINC000217522632 CD On-Demand Unstable TPP2 59 36 O=C1CCN(C(=O)C2CCN(C(=O)c3ccccc3Cl)CC2)CCN1 ZINC000217522636 FD In-Stock Unstable L3MBTL1 0 43 O=C1CCN(C(=O)C2CCN(C(=O)c3ccccc3Cl)CC2)CCN1 ZINC000217522636 FD In-Stock Unstable L3MBTL3 48 38 O=C1CCN(C(=O)C2CCN(C(=O)c3ccccc3Cl)CC2)CCN1 ZINC000217522636 FD In-Stock Unstable TP53BP1 0 43 N[C@@H]1CS(=O)(=O)C[C@H]1c1ccc(Cl)cc1 ZINC000217522661 BD For-Sale Unstable SLC6A3 17 40 COc1ccc2ccccc2c1CCC(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217522676 HI For-Sale Unstable NPY5R 31 50 CC(C)COCCCNC[C@H](O)c1ccc(C#N)cc1 ZINC000217522687 CE For-Sale Unstable ADRB1 25 40 CC(C)COCCCNC[C@H](O)c1ccc(C#N)cc1 ZINC000217522687 CE For-Sale Unstable ADRB3 21 40 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCc1cccc(Br)c1O ZINC000217522691 EJ For-Sale Unstable TRPM8 17 44 NC[C@@H]1CCCN([C@@H]2CCOc3ccccc32)C1 ZINC000217522724 BE For-Sale Unstable SLC6A1 0 41 Cc1[nH]c2ccccc2c1CC(=O)N1C[C@@H]2CC[C@H](C1)[C@@H]2O ZINC000217522741 CE In-Stock Unstable EDNRA 30 40 N[C@@H]1CS(=O)(=O)C[C@@H]1c1ccc(Cl)cc1 ZINC000217522742 BD For-Sale Unstable SLC6A3 17 40 C[C@@H](c1ccccc1)N(C)C(=O)CN1CCC[C@@H](N)C1 ZINC000217522752 CD On-Demand Unstable SLC6A1 80 39 C[C@@H](c1ccccc1)N(C)C(=O)CN1CCC[C@@H](N)C1 ZINC000217522752 CD On-Demand Unstable OPRM1 0 40 C[C@@H](c1ccccc1)N(C)C(=O)CN1CCC[C@@H](N)C1 ZINC000217522752 CD On-Demand Unstable OPRD1 0 40 C[C@@H](c1ccccc1)N(C)C(=O)CN1CCC[C@@H](N)C1 ZINC000217522752 CD On-Demand Unstable OPRK1 32 44 C[C@@H](c1ccccc1)N(C)C(=O)CN1CCC[C@@H](N)C1 ZINC000217522752 CD On-Demand Unstable CCR5 41 41 C[C@@H](c1ccccc1)N(C)C(=O)CN1CCC[C@@H](N)C1 ZINC000217522752 CD On-Demand Unstable BIRC2 45 33 O=C(NCCc1ccc(F)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217522759 FJ For-Sale Unstable CA2 23 59 O=C(NCCc1ccc(F)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217522759 FJ For-Sale Unstable ADRB2 20 47 O=C(NCCc1ccc(F)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217522759 FJ For-Sale Unstable ADRB1 50 47 O=C(NCCc1ccc(F)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217522759 FJ For-Sale Unstable SRD5A2 0 43 O=C(NCCc1ccc(F)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217522759 FJ For-Sale Unstable ADRB3 48 47 O=C(NCCc1ccc(F)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217522759 FJ For-Sale Unstable LTA4H 60 46 O=C(NCCc1ccc(F)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217522759 FJ For-Sale Unstable TACR2 22 41 O=C(NCCc1ccc(F)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217522759 FJ For-Sale Unstable CA1 54 59 O=C(NCCc1ccc(F)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217522759 FJ For-Sale Unstable CCR3 44 47 O=C(NCCc1ccc(F)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217522759 FJ For-Sale Unstable SCN2A 15 47 O=C(NCCc1ccc(F)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217522759 FJ For-Sale Unstable RAF1 67 41 O=C(NCCc1ccc(F)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217522759 FJ For-Sale Unstable MTNR1B 15 46 O=C(NCCc1ccc(F)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217522759 FJ For-Sale Unstable MMP2 17 42 O=C(NCCc1ccc(F)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217522759 FJ For-Sale Unstable ROCK2 16 54 O=C(NCCc1ccc(F)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217522759 FJ For-Sale Unstable NPY5R 29 55 O=C(NCCc1ccc(F)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217522759 FJ For-Sale Unstable S1PR1 0 41 O=C(NCCc1ccc(F)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217522759 FJ For-Sale Unstable EPHX2 23 45 O=C(NCCc1ccc(F)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217522759 FJ For-Sale Unstable CA12 31 59 O=C(NCCc1ccc(F)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217522759 FJ For-Sale Unstable CA9 34 59 O=C(NCCc1ccc(F)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217522759 FJ For-Sale Unstable FABH 0 40 O=C(NCCc1ccc(F)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217522759 FJ For-Sale Unstable AMP1_PLAFQ 40 38 O=C(NCCc1ccc(F)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217522759 FJ For-Sale Unstable Q8MMZ8_EIMTE 71 41 O=C(NCCc1ccc(F)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217522759 FJ For-Sale Unstable F13A1 23 40 O=C(NCCc1ccc(F)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217522759 FJ For-Sale Unstable TAAR1 18 41 O=C(NCCc1ccc(F)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217522759 FJ For-Sale Unstable FFAR1 15 48 O=C(NCCc1ccc(F)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217522759 FJ For-Sale Unstable YOPH 0 41 O=C(NCCc1ccc(F)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217522759 FJ For-Sale Unstable NCE103 39 59 O=C(NCCc1ccc(F)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217522759 FJ For-Sale Unstable CRTM 56 36 O=C(NCCc1ccc(F)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217522759 FJ For-Sale Unstable MTCA1 15 47 O=C(NCCc1ccc(F)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217522759 FJ For-Sale Unstable P96878_MYCTU 22 47 O=C(NCCc1ccc(F)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217522759 FJ For-Sale Unstable ACAT 0 42 O=C(NCCc1ccc(F)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217522759 FJ For-Sale Unstable UPPS 0 41 O=C(NCCc1ccc(F)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217522759 FJ For-Sale Unstable NAMPT 28 53 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCc1cccc(Br)c1O ZINC000217522768 EJ For-Sale Unstable TRPM8 17 44 Cc1ccccc1CCC(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217522790 EH For-Sale Unstable NPY5R 36 47 C[C@H](c1ccccc1)N(C)C(=O)CN1CCC[C@@H](N)C1 ZINC000217522826 CD On-Demand Unstable SLC6A1 80 39 C[C@H](c1ccccc1)N(C)C(=O)CN1CCC[C@@H](N)C1 ZINC000217522826 CD On-Demand Unstable OPRM1 0 40 C[C@H](c1ccccc1)N(C)C(=O)CN1CCC[C@@H](N)C1 ZINC000217522826 CD On-Demand Unstable OPRD1 0 40 C[C@H](c1ccccc1)N(C)C(=O)CN1CCC[C@@H](N)C1 ZINC000217522826 CD On-Demand Unstable OPRK1 32 44 C[C@H](c1ccccc1)N(C)C(=O)CN1CCC[C@@H](N)C1 ZINC000217522826 CD On-Demand Unstable CCR5 41 41 C[C@H](c1ccccc1)N(C)C(=O)CN1CCC[C@@H](N)C1 ZINC000217522826 CD On-Demand Unstable BIRC2 45 33 CC(=O)c1ccc(Br)cc1O[C@@H]1C[C@H]2CC[C@@]1(C)C2(C)C ZINC000217522834 FK For-Sale Unstable ELANE 16 44 CN1CCC2(CC1)C[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccc(C(F)(F)F)cc1)c1ccccc1O2 ZINC000217522873 IJ On-Demand Unstable EPHX2 15 42 CN1CCC2(CC1)C[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccc(C(F)(F)F)cc1)c1ccccc1O2 ZINC000217522873 IJ On-Demand Unstable TRPM8 57 42 O=C(NCCc1ccc(F)cc1)Nc1cc([N+](=O)[O-])ccc1Cl ZINC000217522881 EH For-Sale Unstable CCR3 15 45 O=C(NCCc1ccc(F)cc1)Nc1cc([N+](=O)[O-])ccc1Cl ZINC000217522881 EH For-Sale Unstable WDR5 30 40 Cc1cccc(CCC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217522893 EH For-Sale Unstable NPY5R 34 46 C[C@@](O)(CNC(=O)NCc1ccc(Cl)cc1)c1cc2ccccc2s1 ZINC000217522896 FI In-Stock Unstable U38 0 42 CC(=O)c1ccc(Br)cc1O[C@H]1C[C@H]2CC[C@@]1(C)C2(C)C ZINC000217522909 FK For-Sale Unstable ELANE 16 44 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCc1c[nH]c2ccccc12 ZINC000217522920 CJ For-Sale Unstable SSTR3 26 48 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCc1c[nH]c2ccccc12 ZINC000217522920 CJ For-Sale Unstable TRPM8 15 42 CCOCCOc1ccccc1C(=O)N1CCN(C)[C@@H](c2ccccc2)C1 ZINC000217522961 FG In-Stock Unstable HRH2 15 40 CCOCCOc1ccccc1C(=O)N1CCN(C)[C@@H](c2ccccc2)C1 ZINC000217522961 FG In-Stock Unstable HRH1 18 41 CCOCCOc1ccccc1C(=O)N1CCN(C)[C@@H](c2ccccc2)C1 ZINC000217522961 FG In-Stock Unstable HCN1 46 34 CCOCCOc1ccccc1C(=O)N1CCN(C)[C@@H](c2ccccc2)C1 ZINC000217522961 FG In-Stock Unstable HCN4 42 32 C[C@](O)(CNC(=O)NCc1ccc(Cl)cc1)c1cc2ccccc2s1 ZINC000217522982 FI In-Stock Unstable U38 0 42 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCc1c[nH]c2ccccc12 ZINC000217522983 CJ For-Sale Unstable SSTR3 26 48 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCc1c[nH]c2ccccc12 ZINC000217522983 CJ For-Sale Unstable TRPM8 15 42 O=C(NCCCCl)NCCc1ccc(F)cc1 ZINC000217522988 CE For-Sale Unstable CCR3 26 43 CNC(=O)[C@@H](C)[C@@H]1CCCCN1 ZINC000217523006 AC In-Stock Unstable SLC6A1 0 42 CSc1ccc(CCC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217523008 GI For-Sale Unstable NPY5R 31 45 Cc1cccc(C(=O)N2C[C@H]3CNC[C@@H](C3)C2)c1 ZINC000217523024 BD For-Sale Unstable CHRNA7 30 54 CN1CCC2(CC1)C[C@H](NC(=O)[C@H]1C[C@@H]1c1ccc(C(F)(F)F)cc1)c1ccccc1O2 ZINC000217523039 IJ On-Demand Unstable EPHX2 15 42 CN1CCC2(CC1)C[C@H](NC(=O)[C@H]1C[C@@H]1c1ccc(C(F)(F)F)cc1)c1ccccc1O2 ZINC000217523039 IJ On-Demand Unstable TRPM8 57 42 CCOCCOc1ccccc1C(=O)N1CCN(C)[C@H](c2ccccc2)C1 ZINC000217523041 FG In-Stock Unstable HRH2 15 40 CCOCCOc1ccccc1C(=O)N1CCN(C)[C@H](c2ccccc2)C1 ZINC000217523041 FG In-Stock Unstable HRH1 18 41 CCOCCOc1ccccc1C(=O)N1CCN(C)[C@H](c2ccccc2)C1 ZINC000217523041 FG In-Stock Unstable HCN1 46 34 CCOCCOc1ccccc1C(=O)N1CCN(C)[C@H](c2ccccc2)C1 ZINC000217523041 FG In-Stock Unstable HCN4 42 32 CCO[C@@H]1C[C@@H](Nc2ncnc3ccccc23)C1(C)C ZINC000217523042 CG For-Sale Unstable EGFR 17 43 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCc1c[nH]c2ccccc12 ZINC000217523070 CJ For-Sale Unstable SSTR3 26 48 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCc1c[nH]c2ccccc12 ZINC000217523070 CJ For-Sale Unstable TRPM8 15 42 CNC(=O)[C@H](C)[C@@H]1CCCCN1 ZINC000217523092 AC In-Stock Unstable SLC6A1 0 42 C[C@@](O)(CNC(=O)NC12CC3CC(CC(C3)C1)C2)c1cc2ccccc2s1 ZINC000217523096 GI In-Stock Unstable EPHX2 99 47 Cc1ccsc1CCC(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217523118 FH In-Stock Unstable NPY5R 32 45 CCO[C@H]1C[C@@H](Nc2ncnc3ccccc23)C1(C)C ZINC000217523123 CG For-Sale Unstable EGFR 17 43 C[C@@]1(c2ccccc2)OC[C@@H](CN2CCC[C@@H](N)C2)O1 ZINC000217523129 CD For-Sale Unstable ADRA1D 16 40 C[C@@]1(c2ccccc2)OC[C@@H](CN2CCC[C@@H](N)C2)O1 ZINC000217523129 CD For-Sale Unstable ADRA1B 15 40 COc1cc(OC)cc(C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)c1 ZINC000217523133 GG For-Sale Unstable DRD4 50 39 CC(=O)c1cc(Br)ccc1O[C@@H]1C[C@H]2CC[C@@]1(C)C2(C)C ZINC000217523136 FK For-Sale Unstable ELANE 16 44 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCc1c[nH]c2ccccc12 ZINC000217523155 CJ For-Sale Unstable SSTR3 26 48 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCc1c[nH]c2ccccc12 ZINC000217523155 CJ For-Sale Unstable TRPM8 15 42 CNC(=O)[C@@H](C)[C@H]1CCCCN1 ZINC000217523181 AC In-Stock Unstable SLC6A1 0 42 C[C@](O)(CNC(=O)NC12CC3CC(CC(C3)C1)C2)c1cc2ccccc2s1 ZINC000217523183 GI In-Stock Unstable EPHX2 99 47 CCO[C@@H]1C[C@H](Nc2ncnc3ccccc23)C1(C)C ZINC000217523206 CG For-Sale Unstable EGFR 17 43 C[C@]1(c2ccccc2)OC[C@@H](CN2CCC[C@@H](N)C2)O1 ZINC000217523209 CD For-Sale Unstable ADRA1D 16 40 C[C@]1(c2ccccc2)OC[C@@H](CN2CCC[C@@H](N)C2)O1 ZINC000217523209 CD For-Sale Unstable ADRA1B 15 40 CS(=O)(=O)NCCCNC[C@@H](O)c1ccc(C#N)cc1 ZINC000217523212 CC For-Sale Unstable ADRB3 22 44 CC(=O)c1cc(Br)ccc1O[C@H]1C[C@H]2CC[C@@]1(C)C2(C)C ZINC000217523221 FK For-Sale Unstable ELANE 16 44 CN1CCC2(CC1)C[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1C(F)(F)F)c1ccccc1O2 ZINC000217523226 IJ On-Demand Unstable RBP4 81 37 CCCCOC(=O)c1ccccc1NC(=O)NCCc1ccc(F)cc1 ZINC000217523227 FI For-Sale Unstable CNR2 26 40 CCCCOC(=O)c1ccccc1NC(=O)NCCc1ccc(F)cc1 ZINC000217523227 FI For-Sale Unstable ACAT 0 43 Cc1cc(F)ccc1CN[C@H]1C[C@H](C)CC[C@H]1C(C)C ZINC000217523230 CJ For-Sale Unstable TRPM8 15 42 COc1cccc(C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)c1OC ZINC000217523243 GG For-Sale Unstable DRD2 33 41 COc1cccc(C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)c1OC ZINC000217523243 GG For-Sale Unstable DRD4 41 32 COc1cccc(C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)c1OC ZINC000217523243 GG For-Sale Unstable DRD3 32 47 COc1cccc(C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)c1OC ZINC000217523243 GG For-Sale Unstable FABP4 46 40 O=C1OC2(CCN(C(=O)CCc3cccc4ccccc34)CC2)c2ccccc21 ZINC000217523253 GI For-Sale Unstable NPY5R 35 47 CNC(=O)[C@H](C)[C@H]1CCCCN1 ZINC000217523257 AC In-Stock Unstable SLC6A1 0 42 Cc1ccc(C(=O)N2C[C@H]3CNC[C@@H](C3)C2)cc1 ZINC000217523276 BD For-Sale Unstable L3MBTL3 47 38 CCO[C@H]1C[C@H](Nc2ncnc3ccccc23)C1(C)C ZINC000217523293 CG For-Sale Unstable EGFR 17 43 COc1cccc(NC(=O)NC[C@@](C)(O)c2cc3ccccc3s2)c1OC ZINC000217523296 GH In-Stock Unstable TRPV1 27 40 C[C@@]1(c2ccccc2)OC[C@H](CN2CCC[C@@H](N)C2)O1 ZINC000217523297 CD For-Sale Unstable ADRA1D 16 40 C[C@@]1(c2ccccc2)OC[C@H](CN2CCC[C@@H](N)C2)O1 ZINC000217523297 CD For-Sale Unstable ADRA1B 15 40 CS(=O)(=O)NCCCNC[C@H](O)c1ccc(C#N)cc1 ZINC000217523303 CC For-Sale Unstable ADRB3 22 44 Cc1cc(F)ccc1CN[C@H]1C[C@@H](C)CC[C@H]1C(C)C ZINC000217523321 CJ For-Sale Unstable TRPM8 15 42 O=C(NCCc1ccc(F)cc1)Nc1ccccc1Sc1ccccc1 ZINC000217523337 FK For-Sale Unstable CCR3 24 40 COc1ccc(CNS(=O)(=O)c2[nH]ncc2CO)cc1 ZINC000217523352 CC For-Sale Unstable CA9 16 43 COc1ccc(CNS(=O)(=O)c2[nH]ncc2CO)cc1 ZINC000217523352 CC For-Sale Unstable PROKR1 43 30 COc1cccc(OC)c1C(=O)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217523365 GG For-Sale Unstable HTR1A 19 40 COc1cccc(OC)c1C(=O)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217523365 GG For-Sale Unstable DRD2 28 41 COc1cccc(OC)c1C(=O)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217523365 GG For-Sale Unstable DRD4 44 35 O=C1OC2(CCN(C(=O)CCc3ccc(C(F)(F)F)cc3)CC2)c2ccccc21 ZINC000217523367 HI For-Sale Unstable NPY5R 32 49 CN1CCC2(CC1)C[C@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1C(F)(F)F)c1ccccc1O2 ZINC000217523375 IJ On-Demand Unstable RBP4 81 37 COc1cccc(NC(=O)NC[C@](C)(O)c2cc3ccccc3s2)c1OC ZINC000217523380 GH In-Stock Unstable TRPV1 27 40 C[C@]1(c2ccccc2)OC[C@H](CN2CCC[C@@H](N)C2)O1 ZINC000217523386 CD For-Sale Unstable ADRA1D 16 40 C[C@]1(c2ccccc2)OC[C@H](CN2CCC[C@@H](N)C2)O1 ZINC000217523386 CD For-Sale Unstable ADRA1B 15 40 Cc1cc(CN[C@H]2C[C@H](C)CC[C@H]2C(C)C)ccc1F ZINC000217523415 CJ For-Sale Unstable TRPM8 16 44 O=C1/C(=C\c2ccccc2)c2ccc(Cl)cc2N1CN1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217523437 JI In-Stock Unstable CHRNA4 37 52 NC1(CS(=O)(=O)c2cccc(Cl)c2)CC1 ZINC000217523447 BD For-Sale Unstable FBP1 16 40 O=C(NCCc1ccc(F)cc1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217523448 FJ For-Sale Unstable TRPV1 15 57 O=C(NCCc1ccc(F)cc1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217523448 FJ For-Sale Unstable P2RX7 26 46 O=C(NCCc1ccc(F)cc1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217523448 FJ For-Sale Unstable CCR3 48 44 O=C(NCCc1ccc(F)cc1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217523448 FJ For-Sale Unstable RAF1 66 64 O=C(NCCc1ccc(F)cc1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217523448 FJ For-Sale Unstable EPHX2 23 46 O=C(NCCc1ccc(F)cc1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217523448 FJ For-Sale Unstable ENV 42 33 O=C(NCCc1ccc(F)cc1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217523448 FJ For-Sale Unstable Q8MMZ8_EIMTE 85 64 O=C(NCCc1ccc(F)cc1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217523448 FJ For-Sale Unstable BRAF 17 43 O=C(NCCc1ccc(F)cc1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217523448 FJ For-Sale Unstable PTPA 0 45 O=C(NCCc1ccc(F)cc1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217523448 FJ For-Sale Unstable IMDH_CRYPV 18 45 O=C(NCCc1ccc(F)cc1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217523448 FJ For-Sale Unstable BLM 0 47 C[C@@H](CNCc1c[nH]c2ccccc12)N(C)C1CC1 ZINC000217523464 CF For-Sale Unstable HTR1D 19 40 C[C@@H](CNCc1c[nH]c2ccccc12)N(C)C1CC1 ZINC000217523464 CF For-Sale Unstable HTR1B 16 44 C[C@@H](CNCc1c[nH]c2ccccc12)N(C)C1CC1 ZINC000217523464 CF For-Sale Unstable MPO 29 40 CC(C)(C)c1cc(NC(=O)Oc2ccccc2)n(-c2ccc(O)c(Cl)c2)n1 ZINC000217523465 GK For-Sale Unstable TNF 50 37 CC(C)(C)c1cc(NC(=O)Oc2ccccc2)n(-c2ccc(O)c(Cl)c2)n1 ZINC000217523465 GK For-Sale Unstable MAPK14 31 52 CC(C)(C)c1cc(NC(=O)Oc2ccccc2)n(-c2ccc(O)c(Cl)c2)n1 ZINC000217523465 GK For-Sale Unstable PTK2B 34 41 CC(C)(C)c1cc(NC(=O)Oc2ccccc2)n(-c2ccc(O)c(Cl)c2)n1 ZINC000217523465 GK For-Sale Unstable DDR2 37 46 CC(C)(C)c1cc(NC(=O)Oc2ccccc2)n(-c2ccc(O)c(Cl)c2)n1 ZINC000217523465 GK For-Sale Unstable RPA1 58 34 COc1ccc(CCC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c(OC)c1OC ZINC000217523467 IG For-Sale Unstable NPY5R 27 50 COc1ccc(C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)c(OC)c1 ZINC000217523470 GG For-Sale Unstable DRD4 46 36 COc1ccc(Cl)cc1NC(=O)NC[C@@](C)(O)c1cc2ccccc2s1 ZINC000217523480 GJ In-Stock Unstable CSNK1D 16 41 COc1ccc(Cl)cc1NC(=O)NC[C@@](C)(O)c1cc2ccccc2s1 ZINC000217523480 GJ In-Stock Unstable CPT1A 43 30 COc1ccc(Cl)cc1NC(=O)NC[C@@](C)(O)c1cc2ccccc2s1 ZINC000217523480 GJ In-Stock Unstable RBP4 24 42 Cc1cc(CN[C@H]2C[C@@H](C)CC[C@H]2C(C)C)ccc1F ZINC000217523481 CJ For-Sale Unstable TRPM8 16 44 CCNC(=O)[C@@H](C)[C@@H]1CCCCN1 ZINC000217523538 AC In-Stock Unstable SLC6A1 0 41 C[C@H](CNCc1c[nH]c2ccccc12)N(C)C1CC1 ZINC000217523549 CF For-Sale Unstable HTR1D 19 40 C[C@H](CNCc1c[nH]c2ccccc12)N(C)C1CC1 ZINC000217523549 CF For-Sale Unstable HTR1B 16 44 C[C@H](CNCc1c[nH]c2ccccc12)N(C)C1CC1 ZINC000217523549 CF For-Sale Unstable MPO 29 40 COc1ccc(Cl)cc1NC(=O)NC[C@](C)(O)c1cc2ccccc2s1 ZINC000217523562 GJ In-Stock Unstable CSNK1D 16 41 COc1ccc(Cl)cc1NC(=O)NC[C@](C)(O)c1cc2ccccc2s1 ZINC000217523562 GJ In-Stock Unstable CPT1A 43 30 COc1ccc(Cl)cc1NC(=O)NC[C@](C)(O)c1cc2ccccc2s1 ZINC000217523562 GJ In-Stock Unstable RBP4 24 42 Nc1ccc(NC(=O)NCCc2ccc(F)cc2)c(Cl)c1 ZINC000217523566 DG For-Sale Unstable CA2 15 47 Nc1ccc(NC(=O)NCCc2ccc(F)cc2)c(Cl)c1 ZINC000217523566 DG For-Sale Unstable CA1 15 47 Nc1ccc(NC(=O)NCCc2ccc(F)cc2)c(Cl)c1 ZINC000217523566 DG For-Sale Unstable CCR3 31 41 COc1cc(OC)c(CCC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c(OC)c1 ZINC000217523576 IG For-Sale Unstable NPY5R 35 53 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCc1cc(Br)c(Br)o1 ZINC000217523580 GK For-Sale Unstable TRPM8 15 40 COc1ccc(C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc1OC ZINC000217523588 GG For-Sale Unstable DRD2 20 41 COc1ccc(C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc1OC ZINC000217523588 GG For-Sale Unstable DRD4 45 35 COc1ccc(C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc1OC ZINC000217523588 GG For-Sale Unstable DRD3 28 41 COc1ccc(C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc1OC ZINC000217523588 GG For-Sale Unstable SLC5A7 31 40 CCNC(=O)[C@H](C)[C@@H]1CCCCN1 ZINC000217523613 AC In-Stock Unstable SLC6A1 0 41 NC[C@@H]1CCCN([C@@H]2CCCc3ccccc32)C1 ZINC000217523623 BF On-Demand Unstable SLC6A1 0 46 NC[C@@H]1CCCN([C@@H]2CCCc3ccccc32)C1 ZINC000217523623 BF On-Demand Unstable HTR3B 0 44 Cc1cc(Cl)cc(C(=O)Nc2ccc(Cl)nc2)c1 ZINC000217523653 CH On-Demand Unstable SCN10A 41 45 Cc1cc(Cl)cc(C(=O)Nc2ccc(Cl)nc2)c1 ZINC000217523653 CH On-Demand Unstable CSF1R 29 51 Cc1cc(Cl)cc(C(=O)Nc2ccc(Cl)nc2)c1 ZINC000217523653 CH On-Demand Unstable BTK 17 40 Cc1cc(Cl)cc(C(=O)Nc2ccc(Cl)nc2)c1 ZINC000217523653 CH On-Demand Unstable KCNK3 76 47 Cc1cc(Cl)cc(C(=O)Nc2ccc(Cl)nc2)c1 ZINC000217523653 CH On-Demand Unstable KCNK9 47 47 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCc1cc(Br)c(Br)o1 ZINC000217523656 GK For-Sale Unstable TRPM8 15 40 C[C@@](O)(CNC(=O)Nc1ccccc1C(F)(F)F)c1cc2ccccc2s1 ZINC000217523663 GJ In-Stock Unstable KCNJ11 46 33 C[C@@](O)(CNC(=O)Nc1ccccc1C(F)(F)F)c1cc2ccccc2s1 ZINC000217523663 GJ In-Stock Unstable TRPV1 19 50 COc1ccccc1CCNc1ccc([N+](=O)[O-])nc1 ZINC000217523671 CF On-Demand Unstable PRKCQ 19 43 Nc1ccc(NC(=O)NCCc2ccc(F)cc2)cc1Cl ZINC000217523674 DG For-Sale Unstable CCR3 41 37 Nc1ccc(NC(=O)NCCc2ccc(F)cc2)cc1Cl ZINC000217523674 DG For-Sale Unstable RAF1 36 48 Nc1ccc(NC(=O)NCCc2ccc(F)cc2)cc1Cl ZINC000217523674 DG For-Sale Unstable CA12 17 44 Nc1ccc(NC(=O)NCCc2ccc(F)cc2)cc1Cl ZINC000217523674 DG For-Sale Unstable CA9 15 43 Nc1ccc(NC(=O)NCCc2ccc(F)cc2)cc1Cl ZINC000217523674 DG For-Sale Unstable Q8MMZ8_EIMTE 26 48 Nc1ccc(NC(=O)NCCc2ccc(F)cc2)cc1Cl ZINC000217523674 DG For-Sale Unstable NCE103 34 43 Cc1ccnc2ccc(C(=O)N3CCC4(CC3)OC(=O)c3ccccc34)cc12 ZINC000217523678 FH For-Sale Unstable AVPR1A 18 47 Cc1ccnc2ccc(C(=O)N3CCC4(CC3)OC(=O)c3ccccc34)cc12 ZINC000217523678 FH For-Sale Unstable ACACA 79 40 Cc1ccnc2ccc(C(=O)N3CCC4(CC3)OC(=O)c3ccccc34)cc12 ZINC000217523678 FH For-Sale Unstable ACACB 54 34 Cc1ccnc2ccc(C(=O)N3CCC4(CC3)OC(=O)c3ccccc34)cc12 ZINC000217523678 FH For-Sale Unstable NPY5R 47 47 CCNC(=O)[C@@H](C)[C@H]1CCCCN1 ZINC000217523698 AC In-Stock Unstable SLC6A1 0 41 O=C(NCC1C[C@@H]2CC[C@H](C1)N2)c1ccccc1 ZINC000217523703 BD For-Sale Unstable GRIN2B 19 48 O=C(NCC1C[C@@H]2CC[C@H](C1)N2)c1ccccc1 ZINC000217523703 BD For-Sale Unstable CACNA1I 48 33 O=C(NCC1C[C@@H]2CC[C@H](C1)N2)c1ccccc1 ZINC000217523703 BD For-Sale Unstable ACHP_LYMST 17 50 CC[C@@H]1CN[C@@H](Cc2ccccc2)CN1CC[S@@](=O)CC ZINC000217523722 DE For-Sale Unstable CACNA1B 0 42 C[C@](O)(CNC(=O)Nc1ccccc1C(F)(F)F)c1cc2ccccc2s1 ZINC000217523732 GJ In-Stock Unstable KCNJ11 53 33 C[C@](O)(CNC(=O)Nc1ccccc1C(F)(F)F)c1cc2ccccc2s1 ZINC000217523732 GJ In-Stock Unstable TRPV1 21 50 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCc1cc(Br)c(Br)o1 ZINC000217523741 GK For-Sale Unstable TRPM8 15 40 Cc1cc(I)ccc1NC(=O)NCCc1ccc(F)cc1 ZINC000217523763 GI On-Demand Unstable LEF 52 38 CCNC(=O)[C@H](C)[C@H]1CCCCN1 ZINC000217523776 AC In-Stock Unstable SLC6A1 0 41 O=C1OC2(CCN(C(=O)CCc3ccc(F)c(Cl)c3)CC2)c2ccccc21 ZINC000217523793 GI In-Stock Unstable NPY5R 34 49 COc1cccc(OCC(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)c1 ZINC000217523800 GF For-Sale Unstable DRD4 47 37 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCc1cc(Br)c(Br)o1 ZINC000217523825 GK For-Sale Unstable TRPM8 15 40 O=C(NCCc1ccc(F)cc1)N1CCN(Cc2ccccc2)CC1 ZINC000217523876 EF On-Demand Unstable DRD2 28 43 O=C(NCCc1ccc(F)cc1)N1CCN(Cc2ccccc2)CC1 ZINC000217523876 EF On-Demand Unstable DRD4 57 47 O=C(NCCc1ccc(F)cc1)N1CCN(Cc2ccccc2)CC1 ZINC000217523876 EF On-Demand Unstable ACHE 28 42 O=C(NCCc1ccc(F)cc1)N1CCN(Cc2ccccc2)CC1 ZINC000217523876 EF On-Demand Unstable SLC6A4 26 43 O=C(NCCc1ccc(F)cc1)N1CCN(Cc2ccccc2)CC1 ZINC000217523876 EF On-Demand Unstable DRD3 26 53 O=C(NCCc1ccc(F)cc1)N1CCN(Cc2ccccc2)CC1 ZINC000217523876 EF On-Demand Unstable SLC6A3 29 43 O=C(NCCc1ccc(F)cc1)N1CCN(Cc2ccccc2)CC1 ZINC000217523876 EF On-Demand Unstable MC4R 0 43 O=C(NCCc1ccc(F)cc1)N1CCN(Cc2ccccc2)CC1 ZINC000217523876 EF On-Demand Unstable SIGMAR1 76 53 O=C(NCCc1ccc(F)cc1)N1CCN(Cc2ccccc2)CC1 ZINC000217523876 EF On-Demand Unstable CCR1 24 41 O=C(NCCc1ccc(F)cc1)N1CCN(Cc2ccccc2)CC1 ZINC000217523876 EF On-Demand Unstable CCR3 50 39 O=C(NCCc1ccc(F)cc1)N1CCN(Cc2ccccc2)CC1 ZINC000217523876 EF On-Demand Unstable BRS3 25 43 O=C(NCCc1ccc(F)cc1)N1CCN(Cc2ccccc2)CC1 ZINC000217523876 EF On-Demand Unstable MLNR 59 45 O=C(NCCc1ccc(F)cc1)N1CCN(Cc2ccccc2)CC1 ZINC000217523876 EF On-Demand Unstable FAAH 29 51 O=C(NCCc1ccc(F)cc1)N1CCN(Cc2ccccc2)CC1 ZINC000217523876 EF On-Demand Unstable CXCR3 24 42 O=C(NCCc1ccc(F)cc1)N1CCN(Cc2ccccc2)CC1 ZINC000217523876 EF On-Demand Unstable MCHR1 22 42 O=C(NCCc1ccc(F)cc1)N1CCN(Cc2ccccc2)CC1 ZINC000217523876 EF On-Demand Unstable CACNA1G 54 47 O=C(NCCc1ccc(F)cc1)N1CCN(Cc2ccccc2)CC1 ZINC000217523876 EF On-Demand Unstable MGLL 0 48 O=C(NCCc1ccc(F)cc1)N1CCN(Cc2ccccc2)CC1 ZINC000217523876 EF On-Demand Unstable NPSR1 26 43 O=C(NCCc1ccc(F)cc1)N1CCN(Cc2ccccc2)CC1 ZINC000217523876 EF On-Demand Unstable ABHD6 0 40 O=C(NCCc1ccc(F)cc1)N1CCN(Cc2ccccc2)CC1 ZINC000217523876 EF On-Demand Unstable NPFFR1 56 39 CC[C@@H]1CN[C@H](Cc2ccccc2)CN1CC[S@@](=O)CC ZINC000217523894 DE For-Sale Unstable CACNA1B 0 42 Cc1ccccc1[C@@H](C)NC(=O)CN1CCC[C@@H](N)C1 ZINC000217523914 CD For-Sale Unstable DRD4 0 41 Cc1ccccc1[C@@H](C)NC(=O)CN1CCC[C@@H](N)C1 ZINC000217523914 CD For-Sale Unstable SLC6A1 51 42 Cc1ccccc1[C@@H](C)NC(=O)CN1CCC[C@@H](N)C1 ZINC000217523914 CD For-Sale Unstable BIRC2 49 35 Cc1ccc(CCC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1C ZINC000217523915 FH For-Sale Unstable NPY5R 32 46 O=C(NCCc1ccc(F)cc1)NC1CCCCCCCCCCC1 ZINC000217523971 EK For-Sale Unstable CNR1 17 52 O=C(NCCc1ccc(F)cc1)NC1CCCCCCCCCCC1 ZINC000217523971 EK For-Sale Unstable CNR2 22 52 O=C(NCCc1ccc(F)cc1)NC1CCCCCCCCCCC1 ZINC000217523971 EK For-Sale Unstable CCR3 65 62 O=C(NCCc1ccc(F)cc1)NC1CCCCCCCCCCC1 ZINC000217523971 EK For-Sale Unstable MC5R 0 40 O=C(NCCc1ccc(F)cc1)NC1CCCCCCCCCCC1 ZINC000217523971 EK For-Sale Unstable MMP2 18 40 O=C(NCCc1ccc(F)cc1)NC1CCCCCCCCCCC1 ZINC000217523971 EK For-Sale Unstable SSTR3 19 42 O=C(NCCc1ccc(F)cc1)NC1CCCCCCCCCCC1 ZINC000217523971 EK For-Sale Unstable FAAH 0 44 O=C(NCCc1ccc(F)cc1)NC1CCCCCCCCCCC1 ZINC000217523971 EK For-Sale Unstable EPHX2 41 74 O=C(NCCc1ccc(F)cc1)NC1CCCCCCCCCCC1 ZINC000217523971 EK For-Sale Unstable GPBAR1 22 42 O=C(NCCc1ccc(F)cc1)NC1CCCCCCCCCCC1 ZINC000217523971 EK For-Sale Unstable BIRC2 17 41 Cc1ccccc1[C@H](C)NC(=O)CN1CCC[C@@H](N)C1 ZINC000217524011 CD For-Sale Unstable DRD4 0 41 Cc1ccccc1[C@H](C)NC(=O)CN1CCC[C@@H](N)C1 ZINC000217524011 CD For-Sale Unstable SLC6A1 51 42 Cc1ccccc1[C@H](C)NC(=O)CN1CCC[C@@H](N)C1 ZINC000217524011 CD For-Sale Unstable BIRC2 49 35 O=C1OC2(CCN(C(=O)CCc3ccc(Cl)c(F)c3)CC2)c2ccccc21 ZINC000217524027 GI For-Sale Unstable NPY5R 33 49 NCCN1CCN(C(=O)NCCc2ccc(F)cc2)CC1 ZINC000217524100 CC For-Sale Unstable HTR2A 22 46 NCCN1CCN(C(=O)NCCc2ccc(F)cc2)CC1 ZINC000217524100 CC For-Sale Unstable SIGMAR1 19 57 NCCN1CCN(C(=O)NCCc2ccc(F)cc2)CC1 ZINC000217524100 CC For-Sale Unstable CCR3 35 47 NCCN1CCN(C(=O)NCCc2ccc(F)cc2)CC1 ZINC000217524100 CC For-Sale Unstable CACNA1G 22 41 CC(C)OCC1CCN(C(=O)[C@@H](c2ccc(F)cc2)N(C)C)CC1 ZINC000217524105 EG In-Stock Unstable DPP4 15 41 Cc1ccc(CCC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1F ZINC000217524132 FH For-Sale Unstable NPY5R 35 46 COc1ccc2c(c1)CCC[C@H]2N1CCC[C@@H](CN)C1 ZINC000217524140 CF For-Sale Unstable DRD1 19 50 COc1ccc2c(c1)CCC[C@H]2N1CCC[C@@H](CN)C1 ZINC000217524140 CF For-Sale Unstable SLC6A1 0 50 COc1ccc2c(c1)CCC[C@H]2N1CCC[C@@H](CN)C1 ZINC000217524140 CF For-Sale Unstable SLC6A4 19 50 COc1ccc2c(c1)CCC[C@H]2N1CCC[C@@H](CN)C1 ZINC000217524140 CF For-Sale Unstable HRH3 15 42 COc1ccc2c(c1)CCC[C@H]2N1CCC[C@@H](CN)C1 ZINC000217524140 CF For-Sale Unstable EBP 33 48 CC(C)OCC1CCN(C(=O)[C@H](c2ccc(F)cc2)N(C)C)CC1 ZINC000217524184 EG In-Stock Unstable DPP4 15 41 O=C(NCCc1ccc(F)cc1)NCCN1CCNCC1 ZINC000217524204 CC On-Demand Unstable SIGMAR1 15 42 O=C(NCCc1ccc(F)cc1)NCCN1CCNCC1 ZINC000217524204 CC On-Demand Unstable CCR3 60 57 O=C(NCCc1ccc(F)cc1)NCCN1CCNCC1 ZINC000217524204 CC On-Demand Unstable PLD2 60 36 O=C(NCCc1ccc(F)cc1)NCCN1CCNCC1 ZINC000217524204 CC On-Demand Unstable CACNA1G 29 40 O=C(NCCc1ccc(F)cc1)NCCN1CCNCC1 ZINC000217524204 CC On-Demand Unstable LEF 16 40 COc1ccc2c(c1)CCC[C@@H]2N1CCC[C@@H](CN)C1 ZINC000217524220 CF For-Sale Unstable DRD1 19 50 COc1ccc2c(c1)CCC[C@@H]2N1CCC[C@@H](CN)C1 ZINC000217524220 CF For-Sale Unstable SLC6A1 0 50 COc1ccc2c(c1)CCC[C@@H]2N1CCC[C@@H](CN)C1 ZINC000217524220 CF For-Sale Unstable SLC6A4 19 50 COc1ccc2c(c1)CCC[C@@H]2N1CCC[C@@H](CN)C1 ZINC000217524220 CF For-Sale Unstable HRH3 15 42 COc1ccc2c(c1)CCC[C@@H]2N1CCC[C@@H](CN)C1 ZINC000217524220 CF For-Sale Unstable EBP 33 48 Cc1cc(CCC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)ccc1F ZINC000217524242 FH For-Sale Unstable NPY5R 34 44 CC(C)C1CCC(N[C@H]2C[C@@H](C)CC[C@@H]2C(C)C)CC1 ZINC000217524287 CK For-Sale Unstable TRPM8 15 41 C[C@@H](NC(=O)CN1CCC[C@@H](N)C1)c1ccc(Br)cc1 ZINC000217524322 EE On-Demand Unstable SDH1 0 49 C[C@@H](NC(=O)CN1CCC[C@@H](N)C1)c1ccc(Br)cc1 ZINC000217524322 EE On-Demand Unstable BIRC2 43 40 COc1ccc2nc(C)cc(OCC(=O)Nc3cc(F)cc(F)c3)c2c1 ZINC000217524345 FH On-Demand Unstable OPRL1 0 40 COc1ccc2nc(C)cc(OCC(=O)Nc3cc(F)cc(F)c3)c2c1 ZINC000217524345 FH On-Demand Unstable PDGFRA 45 44 COc1ccc2nc(C)cc(OCC(=O)Nc3cc(F)cc(F)c3)c2c1 ZINC000217524345 FH On-Demand Unstable MCHR1 16 40 COc1ccc2nc(C)cc(OCC(=O)Nc3cc(F)cc(F)c3)c2c1 ZINC000217524345 FH On-Demand Unstable MCHR2 40 40 COc1ccc2nc(C)cc(OCC(=O)Nc3cc(F)cc(F)c3)c2c1 ZINC000217524345 FH On-Demand Unstable DRTS_TRYCR 45 31 Cc1cc(CCC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)ccc1Cl ZINC000217524353 GI For-Sale Unstable NPY5R 33 51 CC(C)C1CCC(N[C@H]2C[C@H](C)CC[C@@H]2C(C)C)CC1 ZINC000217524377 CK For-Sale Unstable TRPM8 15 41 CN(Cc1ccccc1)C(=O)NCCc1ccc(F)cc1 ZINC000217524382 CG On-Demand Unstable MAOA 16 48 CN(Cc1ccccc1)C(=O)NCCc1ccc(F)cc1 ZINC000217524382 CG On-Demand Unstable TSPO 26 44 CN(Cc1ccccc1)C(=O)NCCc1ccc(F)cc1 ZINC000217524382 CG On-Demand Unstable CA5B 15 40 CN(Cc1ccccc1)C(=O)NCCc1ccc(F)cc1 ZINC000217524382 CG On-Demand Unstable AMP1_PLAFQ 29 42 CN(Cc1ccccc1)C(=O)NCCc1ccc(F)cc1 ZINC000217524382 CG On-Demand Unstable LIMK2 48 52 C[C@H](NC(=O)CN1CCC[C@@H](N)C1)c1ccc(Br)cc1 ZINC000217524405 EE On-Demand Unstable SDH1 0 49 C[C@H](NC(=O)CN1CCC[C@@H](N)C1)c1ccc(Br)cc1 ZINC000217524405 EE On-Demand Unstable BIRC2 43 40 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCc1csc2ccccc12 ZINC000217524466 DK For-Sale Unstable TRPM8 15 40 O=C(Cc1cccc2ccccc12)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217524475 HI For-Sale Unstable FABP4 45 39 O=C(Cc1cccc2ccccc12)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217524475 HI For-Sale Unstable P2RX7 29 40 COc1c2ccc(C(=O)N3CCC4(CC3)OC(=O)c3ccccc34)cc2nn1C ZINC000217524477 GF For-Sale Unstable ACACA 48 39 COc1c2ccc(C(=O)N3CCC4(CC3)OC(=O)c3ccccc34)cc2nn1C ZINC000217524477 GF For-Sale Unstable NPY5R 33 49 NCc1cccc(CNC(=O)NCCc2ccc(F)cc2)c1 ZINC000217524494 DE For-Sale Unstable TPSAB1 28 42 CC(C)[C@@H](NC(=O)CN1CCC[C@@H](N)C1)c1cccs1 ZINC000217524496 CD For-Sale Unstable BIRC2 42 34 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCc1csc2ccccc12 ZINC000217524554 DK For-Sale Unstable TRPM8 15 40 O[C@@H]1[C@H]2CC[C@@H]1CN(Cc1ccccc1OCc1ccccc1)C2 ZINC000217524566 DG In-Stock Unstable PTGER2 25 40 O[C@@H]1[C@H]2CC[C@@H]1CN(Cc1ccccc1OCc1ccccc1)C2 ZINC000217524566 DG In-Stock Unstable PTGER1 26 40 Cn1nc2cc(Br)ccc2c1C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217524579 IH For-Sale Unstable AVPR1A 15 49 Cn1nc2cc(Br)ccc2c1C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217524579 IH For-Sale Unstable NPY5R 34 51 CC(C)[C@H](NC(=O)CN1CCC[C@@H](N)C1)c1cccs1 ZINC000217524581 CD For-Sale Unstable BIRC2 42 34 O=C(NCCc1ccc(F)cc1)Nc1cc(Cl)ccc1O ZINC000217524610 DH For-Sale Unstable CCR3 20 51 O=C(NCCc1ccc(F)cc1)Nc1cc(Cl)ccc1O ZINC000217524610 DH For-Sale Unstable KCNMA1 21 46 O=C(NCCc1ccc(F)cc1)Nc1cc(Cl)ccc1O ZINC000217524610 DH For-Sale Unstable LEF 51 35 O=C(NCCc1ccc(F)cc1)Nc1cc(Cl)ccc1O ZINC000217524610 DH For-Sale Unstable NCE103 35 42 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCc1csc2ccccc12 ZINC000217524632 DK For-Sale Unstable TRPM8 15 40 CCC[C@@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1NCc1ccccc1 ZINC000217524681 GG In-Stock Unstable TMPRSS11D 41 35 CCCn1c(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc2c(=O)n(C)c(=O)n(C)c21 ZINC000217524692 JD For-Sale Unstable NPY5R 26 40 COc1ccc(Cl)cc1C(=O)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217524706 HH For-Sale Unstable DRD2 16 46 COc1ccc(Cl)cc1C(=O)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217524706 HH For-Sale Unstable DRD4 43 37 COc1ccc(Cl)cc1C(=O)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217524706 HH For-Sale Unstable DRD3 18 41 COc1ccc(Cl)cc1C(=O)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217524706 HH For-Sale Unstable HTR4 17 43 COc1ccc(Cl)cc1C(=O)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217524706 HH For-Sale Unstable CNR2 15 40 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCc1csc2ccccc12 ZINC000217524715 DK For-Sale Unstable TRPM8 15 40 O=C(NCCc1ccc(F)cc1)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217524730 IF For-Sale Unstable CA1 15 45 O=C(NCCc1ccc(F)cc1)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217524730 IF For-Sale Unstable CCR3 32 41 O=C(NCCc1ccc(F)cc1)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217524730 IF For-Sale Unstable MURF 0 43 O=C(NCCc1ccc(F)cc1)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217524730 IF For-Sale Unstable NAMPT 38 43 C[C@@H](CNC(=O)CN1CCC[C@@H](N)C1)c1ccccc1 ZINC000217524737 CD For-Sale Unstable SLC6A1 71 37 C[C@@H](CNC(=O)CN1CCC[C@@H](N)C1)c1ccccc1 ZINC000217524737 CD For-Sale Unstable BIRC2 52 40 C[C@@H](CNC(=O)CN1CCC[C@@H](N)C1)c1ccccc1 ZINC000217524737 CD For-Sale Unstable BIRC8 44 32 CCC[C@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1NCc1ccccc1 ZINC000217524782 GG In-Stock Unstable TMPRSS11D 41 35 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1N[C@@H](C)C1CCCC1 ZINC000217524793 CJ For-Sale Unstable TRPM8 15 40 O=C(NCc1ccncc1)[C@@H]1[C@H]2C=C[C@@]3(CN(c4ccc5c(c4)OCO5)C(=O)[C@H]13)O2 ZINC000217524795 HD In-Stock Unstable NOS2 64 31 O=C(NCC[C@@H](O)c1ccsc1)c1ccsc1 ZINC000217524808 CF In-Stock Unstable ITGAV 18 40 CCCn1c(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc2c(=O)n3ccccc3nc21 ZINC000217524812 JG For-Sale Unstable NPY5R 27 41 C[C@H](CNC(=O)CN1CCC[C@@H](N)C1)c1ccccc1 ZINC000217524821 CD For-Sale Unstable SLC6A1 71 37 C[C@H](CNC(=O)CN1CCC[C@@H](N)C1)c1ccccc1 ZINC000217524821 CD For-Sale Unstable BIRC2 52 40 C[C@H](CNC(=O)CN1CCC[C@@H](N)C1)c1ccccc1 ZINC000217524821 CD For-Sale Unstable BIRC8 44 32 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1cc(-c2ccccc2)on1 ZINC000217524831 HH For-Sale Unstable HDAC10 15 46 O=C(NCCc1ccc(F)cc1)Nc1ncccn1 ZINC000217524859 CD For-Sale Unstable NCE103 15 40 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1N[C@@H](C)C1CCCC1 ZINC000217524882 CJ For-Sale Unstable TRPM8 15 40 O=C(NCc1ccncc1)[C@H]1[C@H]2C=C[C@@]3(CN(c4ccc5c(c4)OCO5)C(=O)[C@H]13)O2 ZINC000217524884 HD In-Stock Unstable NOS2 64 31 O=C(NCC[C@H](O)c1ccsc1)c1ccsc1 ZINC000217524893 CF In-Stock Unstable ITGAV 18 40 COCCn1c(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc2c(=O)n3ccccc3nc21 ZINC000217524929 JF For-Sale Unstable NPY5R 25 41 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1cccc(C(F)(F)F)c1 ZINC000217524957 HI For-Sale Unstable DRD4 44 35 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1cccc(C(F)(F)F)c1 ZINC000217524957 HI For-Sale Unstable CCR2 89 44 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1N[C@@H](C)C1CCCC1 ZINC000217524978 CJ For-Sale Unstable TRPM8 15 40 CCCCN(CCC)C(=O)NCCc1ccc(F)cc1 ZINC000217524983 CH For-Sale Unstable TSPO 21 40 CCCCN(CCC)C(=O)NCCc1ccc(F)cc1 ZINC000217524983 CH For-Sale Unstable PLM2_PLAFA 76 39 CCCCn1c(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc2c(=O)n3ccccc3nc21 ZINC000217525044 JH For-Sale Unstable NPY5R 25 40 Cc1ccc(NCc2cc(=O)n(C)c(=O)n2C)cc1S(=O)(=O)N1CCCCC1 ZINC000217525056 HD On-Demand Unstable CNR2 17 47 O=C(CN1CCC(c2ccccc2)CC1)NCCCn1ccccc1=O ZINC000217525058 FE In-Stock Unstable DRD4 31 47 O=C(CN1CCC(c2ccccc2)CC1)NCCCn1ccccc1=O ZINC000217525058 FE In-Stock Unstable ADRA1D 48 55 O=C(CN1CCC(c2ccccc2)CC1)NCCCn1ccccc1=O ZINC000217525058 FE In-Stock Unstable ADRA1A 34 42 O=C(CN1CCC(c2ccccc2)CC1)NCCCn1ccccc1=O ZINC000217525058 FE In-Stock Unstable ADRA1B 29 42 O=C(CN1CCC(c2ccccc2)CC1)NCCCn1ccccc1=O ZINC000217525058 FE In-Stock Unstable PRCP 24 44 O=C(CN1CCC(c2ccccc2)CC1)NCCCn1ccccc1=O ZINC000217525058 FE In-Stock Unstable MCHR1 22 42 CC(C)[C@H]1CC[C@H](C)C[C@@H]1N[C@@H](C)C1CCCC1 ZINC000217525091 CJ For-Sale Unstable TRPM8 15 40 O=C(O)Cc1ccc(NC(=O)NCCc2ccc(F)cc2)cc1 ZINC000217525095 DF For-Sale Unstable CA2 15 51 O=C(O)Cc1ccc(NC(=O)NCCc2ccc(F)cc2)cc1 ZINC000217525095 DF For-Sale Unstable ADRB1 21 42 O=C(O)Cc1ccc(NC(=O)NCCc2ccc(F)cc2)cc1 ZINC000217525095 DF For-Sale Unstable CA1 18 51 O=C(O)Cc1ccc(NC(=O)NCCc2ccc(F)cc2)cc1 ZINC000217525095 DF For-Sale Unstable CCR3 42 45 O=C(O)Cc1ccc(NC(=O)NCCc2ccc(F)cc2)cc1 ZINC000217525095 DF For-Sale Unstable CA12 18 51 O=C(O)Cc1ccc(NC(=O)NCCc2ccc(F)cc2)cc1 ZINC000217525095 DF For-Sale Unstable CA9 18 51 O=C(O)Cc1ccc(NC(=O)NCCc2ccc(F)cc2)cc1 ZINC000217525095 DF For-Sale Unstable NCE103 24 51 O=C(O)Cc1ccc(NC(=O)NCCc2ccc(F)cc2)cc1 ZINC000217525095 DF For-Sale Unstable P96878_MYCTU 17 40 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccccc1C(F)(F)F ZINC000217525152 HI For-Sale Unstable FABP4 43 42 O=C1OC2(CCN(C(=O)CCc3ccc([N+](=O)[O-])cc3)CC2)c2ccccc21 ZINC000217525153 GG For-Sale Unstable NPY5R 35 49 O=C1OC2(CCN(C(=O)CCc3ccc([N+](=O)[O-])cc3)CC2)c2ccccc21 ZINC000217525153 GG For-Sale Unstable KCNJ1 29 43 CCOc1ccc(NC(=O)c2ccc(NCc3cc(=O)n(C)c(=O)n3C)cc2)cc1 ZINC000217525155 HE On-Demand Unstable PRNP 48 43 CCOc1ccc(NC(=O)c2ccc(NCc3cc(=O)n(C)c(=O)n3C)cc2)cc1 ZINC000217525155 HE On-Demand Unstable DGAT1 17 40 CCOc1ccc(NC(=O)c2ccc(NCc3cc(=O)n(C)c(=O)n3C)cc2)cc1 ZINC000217525155 HE On-Demand Unstable NOD2 34 45 CC[C@@H](N[C@@H]1C[C@@H](C)CC[C@@H]1C(C)C)c1ccco1 ZINC000217525183 CJ For-Sale Unstable TRPM8 15 40 C[C@@H](O)CCN(C)C[C@@H](O)c1ccc(C#N)cc1 ZINC000217525192 BD On-Demand Unstable AOC3 15 40 N#Cc1ccc(C(=O)NCC[C@H](O)c2ccsc2)cc1 ZINC000217525208 CE In-Stock Unstable CTRB_BOVIN 46 34 O=C(NCCc1ccc(F)cc1)NCc1ccc(C(=O)O)cc1 ZINC000217525209 DF On-Demand Unstable CA1 16 47 O=C(NCCc1ccc(F)cc1)NCc1ccc(C(=O)O)cc1 ZINC000217525209 DF On-Demand Unstable CCR3 17 48 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1cc(=O)c2ccccc2o1 ZINC000217525262 HG For-Sale Unstable BCHE 52 51 CC[C@H](N[C@@H]1C[C@@H](C)CC[C@@H]1C(C)C)c1ccco1 ZINC000217525263 CJ For-Sale Unstable TRPM8 15 40 N#Cc1ccc(CCC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217525266 FG For-Sale Unstable NPY5R 29 45 N#Cc1ccc(C(=O)NCC[C@@H](O)c2ccsc2)cc1 ZINC000217525282 CE In-Stock Unstable CTRB_BOVIN 46 34 CCC[C@@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccccc1 ZINC000217525290 GH In-Stock Unstable CTSG 26 40 CCC[C@@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccccc1 ZINC000217525290 GH In-Stock Unstable CTRB1 34 40 CCC[C@@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccccc1 ZINC000217525290 GH In-Stock Unstable CELA2A 26 40 C[C@H](O)CCN(C)C[C@@H](O)c1ccc(C#N)cc1 ZINC000217525294 BD On-Demand Unstable AOC3 15 40 CC1(C)CC(N)CC(C)(C)N1C(=O)NCCc1ccc(F)cc1 ZINC000217525325 DG For-Sale Unstable CCR3 26 41 CCOCCNc1ccncc1CN ZINC000217525350 AC In-Stock Unstable AMO_PEA 0 50 CC[C@@H](N[C@H]1C[C@@H](C)CC[C@@H]1C(C)C)c1ccco1 ZINC000217525352 CJ For-Sale Unstable TRPM8 15 40 CCC[C@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccccc1 ZINC000217525380 GH In-Stock Unstable CTSG 26 40 CCC[C@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccccc1 ZINC000217525380 GH In-Stock Unstable CTRB1 34 40 CCC[C@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccccc1 ZINC000217525380 GH In-Stock Unstable CELA2A 26 40 O=C1OC2(CCN(C(=O)c3cc4cc(F)ccc4s3)CC2)c2ccccc21 ZINC000217525382 GI In-Stock Unstable NPY5R 45 53 O=C(/C=C/c1ccccc1)NCC[C@H](O)c1ccsc1 ZINC000217525385 CG In-Stock Unstable MMP2 19 51 O=C(/C=C/c1ccccc1)NCC[C@H](O)c1ccsc1 ZINC000217525385 CG In-Stock Unstable MMP9 16 51 O=C(/C=C/c1ccccc1)NCC[C@H](O)c1ccsc1 ZINC000217525385 CG In-Stock Unstable MMP1 0 40 CC[C@H](N[C@H]1C[C@@H](C)CC[C@@H]1C(C)C)c1ccco1 ZINC000217525436 CJ For-Sale Unstable TRPM8 15 40 Cc1ccc(O)c(NC(=O)NCCc2ccc(F)cc2)c1 ZINC000217525441 CG For-Sale Unstable RAF1 39 43 CN(C)CCNc1ccncc1CN ZINC000217525469 AC In-Stock Unstable AOC1 40 49 CN(C)CCNc1ccncc1CN ZINC000217525469 AC In-Stock Unstable AMO_PEA 0 49 O=C(/C=C/c1ccccc1)NCC[C@@H](O)c1ccsc1 ZINC000217525470 CG In-Stock Unstable MMP2 19 51 O=C(/C=C/c1ccccc1)NCC[C@@H](O)c1ccsc1 ZINC000217525470 CG In-Stock Unstable MMP9 16 51 O=C(/C=C/c1ccccc1)NCC[C@@H](O)c1ccsc1 ZINC000217525470 CG In-Stock Unstable MMP1 0 40 CCC[C@@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)cc1 ZINC000217525485 HH In-Stock Unstable AKR1C3 21 40 CC(=O)Nc1ccc(CC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217525508 GF In-Stock Unstable NPY5R 53 51 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1N[C@@H]1CCCc2sccc21 ZINC000217525524 CK For-Sale Unstable TRPM8 0 40 O=C(NCCc1ccc(F)cc1)N1CCN(CCO)CC1 ZINC000217525556 CC On-Demand Unstable HTR2A 23 46 O=C(NCCc1ccc(F)cc1)N1CCN(CCO)CC1 ZINC000217525556 CC On-Demand Unstable MLNR 24 40 O=C(NCCc1ccc(F)cc1)N1CCN(CCO)CC1 ZINC000217525556 CC On-Demand Unstable CACNA1G 24 42 CCC[C@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)cc1 ZINC000217525561 HH In-Stock Unstable AKR1C3 21 40 NCc1cnccc1NCC1CC1 ZINC000217525575 AD In-Stock Unstable AOC1 29 46 COc1ccc(C(S[C@@H](C)C(=O)O)(c2ccccc2)c2ccccc2)cc1 ZINC000217525602 GK For-Sale Unstable KIF11 40 60 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1N[C@@H]1CCCc2sccc21 ZINC000217525612 CK For-Sale Unstable TRPM8 0 40 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1cc(Cl)cc(Cl)c1 ZINC000217525618 HJ For-Sale Unstable CACNA1H 27 43 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1cc(Cl)cc(Cl)c1 ZINC000217525618 HJ For-Sale Unstable CACNA1I 61 37 Cc1nc2ccc(C(=O)N3CCC4(CC3)OC(=O)c3ccccc34)cc2s1 ZINC000217525623 GH For-Sale Unstable ACACA 85 39 Cc1nc2ccc(C(=O)N3CCC4(CC3)OC(=O)c3ccccc34)cc2s1 ZINC000217525623 GH For-Sale Unstable ACACB 59 36 Cc1nc2ccc(C(=O)N3CCC4(CC3)OC(=O)c3ccccc34)cc2s1 ZINC000217525623 GH For-Sale Unstable NPY5R 39 48 CCC[C@@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)c(OC)c1 ZINC000217525659 JH In-Stock Unstable PTGDR 24 43 CCC[C@@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)c(OC)c1 ZINC000217525659 JH In-Stock Unstable SCMU_MYCTU 0 48 COc1ccc(C(S[C@H](C)C(=O)O)(c2ccccc2)c2ccccc2)cc1 ZINC000217525675 GK For-Sale Unstable KIF11 40 60 CCN(Cc1ccccc1)C(=O)NCCc1ccc(F)cc1 ZINC000217525679 DH On-Demand Unstable OPRD1 23 47 CCN(Cc1ccccc1)C(=O)NCCc1ccc(F)cc1 ZINC000217525679 DH On-Demand Unstable TSPO 32 51 CCN(Cc1ccccc1)C(=O)NCCc1ccc(F)cc1 ZINC000217525679 DH On-Demand Unstable PLM2_PLAFA 36 41 CCN(Cc1ccccc1)C(=O)NCCc1ccc(F)cc1 ZINC000217525679 DH On-Demand Unstable AMP1_PLAFQ 29 40 CCN(Cc1ccccc1)C(=O)NCCc1ccc(F)cc1 ZINC000217525679 DH On-Demand Unstable PTGES 19 47 CCN(Cc1ccccc1)C(=O)NCCc1ccc(F)cc1 ZINC000217525679 DH On-Demand Unstable LIMK2 42 45 CCN(Cc1ccccc1)C(=O)NCCc1ccc(F)cc1 ZINC000217525679 DH On-Demand Unstable ACAT 0 42 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1N[C@@H]1CCCc2sccc21 ZINC000217525694 CK For-Sale Unstable TRPM8 0 40 CCCCCCCNC[C@@H](C)N(C)C1CC1 ZINC000217525709 BG For-Sale Unstable Q8WS26_TRYCR 35 41 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1cc(Cl)ccc1Cl ZINC000217525730 HJ For-Sale Unstable CNR1 52 32 CNCCCN1CCC(c2cccc(OC)c2)CC1 ZINC000217525738 CE On-Demand Unstable HTR1A 36 44 CNCCCN1CCC(c2cccc(OC)c2)CC1 ZINC000217525738 CE On-Demand Unstable DRD2 38 53 CNCCCN1CCC(c2cccc(OC)c2)CC1 ZINC000217525738 CE On-Demand Unstable DRD4 47 36 CNCCCN1CCC(c2cccc(OC)c2)CC1 ZINC000217525738 CE On-Demand Unstable ADRA1D 33 43 CNCCCN1CCC(c2cccc(OC)c2)CC1 ZINC000217525738 CE On-Demand Unstable HTR2A 24 46 CNCCCN1CCC(c2cccc(OC)c2)CC1 ZINC000217525738 CE On-Demand Unstable SLC6A4 20 48 CNCCCN1CCC(c2cccc(OC)c2)CC1 ZINC000217525738 CE On-Demand Unstable ADRA1B 27 44 CNCCCN1CCC(c2cccc(OC)c2)CC1 ZINC000217525738 CE On-Demand Unstable DRD3 33 45 CNCCCN1CCC(c2cccc(OC)c2)CC1 ZINC000217525738 CE On-Demand Unstable HTR7 33 47 CNCCCN1CCC(c2cccc(OC)c2)CC1 ZINC000217525738 CE On-Demand Unstable HRH3 31 48 CNCCCN1CCC(c2cccc(OC)c2)CC1 ZINC000217525738 CE On-Demand Unstable SIGMAR1 32 46 CNCCCN1CCC(c2cccc(OC)c2)CC1 ZINC000217525738 CE On-Demand Unstable NPY1R 15 49 CNCCCN1CCC(c2cccc(OC)c2)CC1 ZINC000217525738 CE On-Demand Unstable CCR3 21 45 CNCCCN1CCC(c2cccc(OC)c2)CC1 ZINC000217525738 CE On-Demand Unstable CCR5 21 42 CNCCCN1CCC(c2cccc(OC)c2)CC1 ZINC000217525738 CE On-Demand Unstable EBP 67 46 CNCCCN1CCC(c2cccc(OC)c2)CC1 ZINC000217525738 CE On-Demand Unstable MCHR1 38 50 CNCCCN1CCC(c2cccc(OC)c2)CC1 ZINC000217525738 CE On-Demand Unstable CARM1 73 44 CCC[C@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)c(OC)c1 ZINC000217525743 JH In-Stock Unstable PTGDR 24 43 CCC[C@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)c(OC)c1 ZINC000217525743 JH In-Stock Unstable SCMU_MYCTU 0 48 CCc1nc2ccc(C(=O)N3CCC4(CC3)OC(=O)c3ccccc34)cc2s1 ZINC000217525749 GI In-Stock Unstable ACACA 69 35 CCc1nc2ccc(C(=O)N3CCC4(CC3)OC(=O)c3ccccc34)cc2s1 ZINC000217525749 GI In-Stock Unstable ACACB 46 35 CCc1nc2ccc(C(=O)N3CCC4(CC3)OC(=O)c3ccccc34)cc2s1 ZINC000217525749 GI In-Stock Unstable NPY5R 34 47 Cc1nc2ccccc2cc1C(=O)Nc1ccc2c(c1)OC(F)(F)O2 ZINC000217525755 EI On-Demand Unstable KIT 33 53 Cc1nc2ccccc2cc1C(=O)Nc1ccc2c(c1)OC(F)(F)O2 ZINC000217525755 EI On-Demand Unstable BRAF 40 53 Cc1nc2ccccc2cc1C(=O)Nc1ccc2c(c1)OC(F)(F)O2 ZINC000217525755 EI On-Demand Unstable NR2E3 59 35 Cc1nc2ccccc2cc1C(=O)Nc1ccc2c(c1)OC(F)(F)O2 ZINC000217525755 EI On-Demand Unstable SHH 46 41 Cc1nc2ccccc2cc1C(=O)Nc1ccc2c(c1)OC(F)(F)O2 ZINC000217525755 EI On-Demand Unstable KCNK3 55 35 Cc1nc2ccccc2cc1C(=O)Nc1ccc2c(c1)OC(F)(F)O2 ZINC000217525755 EI On-Demand Unstable KCNK9 47 33 CC(C)[C@H]1CC[C@H](C)C[C@@H]1N[C@@H]1CCCc2sccc21 ZINC000217525775 CK For-Sale Unstable TRPM8 0 40 CCCCCCCNC[C@H](C)N(C)C1CC1 ZINC000217525787 BG For-Sale Unstable Q8WS26_TRYCR 35 41 O=C(NCCc1ccc(F)cc1)N(Cc1ccccc1)Cc1ccccc1 ZINC000217525805 FJ On-Demand Unstable TSPO 25 44 O=C(NCCc1ccc(F)cc1)N(Cc1ccccc1)Cc1ccccc1 ZINC000217525805 FJ On-Demand Unstable CPA1 24 40 O=C(NCCc1ccc(F)cc1)N(Cc1ccccc1)Cc1ccccc1 ZINC000217525805 FJ On-Demand Unstable CA5B 16 42 O=C(NCCc1ccc(F)cc1)N(Cc1ccccc1)Cc1ccccc1 ZINC000217525805 FJ On-Demand Unstable AMP1_PLAFQ 30 40 O=C(NCCc1ccc(F)cc1)N(Cc1ccccc1)Cc1ccccc1 ZINC000217525805 FJ On-Demand Unstable PTGES 20 48 O=C(NCCc1ccc(F)cc1)N(Cc1ccccc1)Cc1ccccc1 ZINC000217525805 FJ On-Demand Unstable LIMK2 42 45 O=C(NCCc1ccc(F)cc1)N(Cc1ccccc1)Cc1ccccc1 ZINC000217525805 FJ On-Demand Unstable ACAT 0 43 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc(Cl)cc1Cl ZINC000217525842 HJ For-Sale Unstable CNR1 51 32 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc(Cl)cc1Cl ZINC000217525842 HJ For-Sale Unstable SLC6A9 47 35 CC(=O)Nc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217525857 FF In-Stock Unstable AVPR1A 15 48 CC(=O)Nc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217525857 FF In-Stock Unstable NPY5R 61 56 Cc1cc(CN[C@H]2C[C@H](C)CC[C@H]2C(C)C)c(C)n1C ZINC000217525888 CI For-Sale Unstable TRPM8 15 40 Cc1cc(-c2ccc(Cn3ccnc3)cn2)ccc1O ZINC000217525900 CG In-Stock Unstable CYP19A1 22 42 Cc1cc(-c2ccc(Cn3ccnc3)cn2)ccc1O ZINC000217525900 CG In-Stock Unstable CYP11B1 68 71 Cc1cc(-c2ccc(Cn3ccnc3)cn2)ccc1O ZINC000217525900 CG In-Stock Unstable TBXAS1 29 43 Cc1cc(-c2ccc(Cn3ccnc3)cn2)ccc1O ZINC000217525900 CG In-Stock Unstable CYP11B2 61 75 Cc1cc(-c2ccc(Cn3ccnc3)cn2)ccc1O ZINC000217525900 CG In-Stock Unstable CYP17A1 40 51 O=C(NCCc1ccc(F)cc1)N(CCO)Cc1ccccc1 ZINC000217525907 DF On-Demand Unstable LIMK2 38 46 O=C(NCCc1ccc(F)cc1)N(CCO)Cc1ccccc1 ZINC000217525907 DF On-Demand Unstable ACAT 0 44 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc(Cl)c(Cl)c1 ZINC000217525948 HJ For-Sale Unstable DRD4 43 33 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc(Cl)c(Cl)c1 ZINC000217525948 HJ For-Sale Unstable PLD1 28 40 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc(Cl)c(Cl)c1 ZINC000217525948 HJ For-Sale Unstable PLD2 45 40 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc(Cl)c(Cl)c1 ZINC000217525948 HJ For-Sale Unstable RPA1 40 33 COCCOc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217525981 GG For-Sale Unstable AVPR1A 16 46 COCCOc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217525981 GG For-Sale Unstable NPY5R 37 49 Cc1cc(CN[C@H]2C[C@@H](C)CC[C@H]2C(C)C)c(C)n1C ZINC000217525984 CI For-Sale Unstable TRPM8 15 40 COc1ccccc1C(=O)NCC[C@H](O)c1ccsc1 ZINC000217526001 CF In-Stock Unstable KCNA3 38 51 COc1ccccc1C(=O)NCC[C@H](O)c1ccsc1 ZINC000217526001 CF In-Stock Unstable HCN1 56 40 COc1ccccc1C(=O)NCC[C@H](O)c1ccsc1 ZINC000217526001 CF In-Stock Unstable KCNK3 35 40 COc1ccccc1C(=O)NCC[C@H](O)c1ccsc1 ZINC000217526001 CF In-Stock Unstable KCNK9 30 40 O=C(NCCCO)NCCc1ccc(F)cc1 ZINC000217526014 BD On-Demand Unstable CA5A 15 40 O=C(NCCCO)NCCc1ccc(F)cc1 ZINC000217526014 BD On-Demand Unstable LEF 40 37 COc1cccc2cc(C(=O)NCCn3nc(C(F)(F)F)c4c3CCCC4)oc12 ZINC000217526059 HH For-Sale Unstable DRD2 16 49 COc1cccc2cc(C(=O)NCCn3nc(C(F)(F)F)c4c3CCCC4)oc12 ZINC000217526059 HH For-Sale Unstable DRD4 40 31 COc1cccc2cc(C(=O)NCCn3nc(C(F)(F)F)c4c3CCCC4)oc12 ZINC000217526059 HH For-Sale Unstable DRD3 27 49 COc1cccc2cc(C(=O)NCCn3nc(C(F)(F)F)c4c3CCCC4)oc12 ZINC000217526059 HH For-Sale Unstable BCHE 52 37 Cc1ccc(O)c(CN[C@H]2C[C@H](C)CC[C@H]2C(C)C)c1 ZINC000217526078 CI For-Sale Unstable TRPM8 16 47 COc1ccccc1C(=O)NCC[C@@H](O)c1ccsc1 ZINC000217526081 CF In-Stock Unstable KCNA3 38 51 COc1ccccc1C(=O)NCC[C@@H](O)c1ccsc1 ZINC000217526081 CF In-Stock Unstable HCN1 56 40 COc1ccccc1C(=O)NCC[C@@H](O)c1ccsc1 ZINC000217526081 CF In-Stock Unstable KCNK3 35 40 COc1ccccc1C(=O)NCC[C@@H](O)c1ccsc1 ZINC000217526081 CF In-Stock Unstable KCNK9 30 40 O=C1OC2(CCN(C(=O)CCCCCN3C(=O)c4ccccc4C3=O)CC2)c2ccccc21 ZINC000217526095 IH For-Sale Unstable NPY5R 40 47 Cc1ccc(O)c(CN[C@H]2C[C@@H](C)CC[C@H]2C(C)C)c1 ZINC000217526168 CI For-Sale Unstable TRPM8 16 47 O=C(/C=C/c1ccc2c(c1)OCO2)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217526182 HG For-Sale Unstable DYRK2 48 32 COc1cccc(C(=O)NCC[C@H](O)c2ccsc2)c1 ZINC000217526203 CF In-Stock Unstable DRD4 59 45 O=C1OC2(CCN(C(=O)Cn3nnc(N4CCOCC4)n3)CC2)c2ccccc21 ZINC000217526204 GC For-Sale Unstable NPY5R 39 46 O=C1C[C@]2(C[C@H]3C=C[C@@H]2C3)C(=O)N1c1ccc(Cl)c(Cl)c1 ZINC000217526205 DH In-Stock Unstable BCL2A1 55 38 O=C(/C=C\c1ccc(Cl)c(Cl)c1)NCC1CC(O)C1 ZINC000217526235 DF For-Sale Unstable HDAC8 23 42 O=C(/C=C\c1ccc(Cl)c(Cl)c1)NCC1CC(O)C1 ZINC000217526235 DF For-Sale Unstable HDAC1 23 42 COC(=O)c1ccc(C(=O)OC)c(NC(=O)NCCc2ccc(F)cc2)c1 ZINC000217526245 FF For-Sale Unstable CCR3 33 41 CC(C)CNC(=O)[C@@H](C)N1CCC[C@@H](N)C1 ZINC000217526253 BC On-Demand Unstable TPP2 19 40 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1N[C@@H](C)c1ccc(Br)s1 ZINC000217526266 EK For-Sale Unstable TRPM8 15 42 COc1cccc(C(=O)NCC[C@@H](O)c2ccsc2)c1 ZINC000217526271 CF In-Stock Unstable DRD4 59 45 CNC(=O)[C@H](c1ccccc1)[C@@H]1CCCCN1 ZINC000217526272 BD In-Stock Unstable SLC6A1 26 73 CNC(=O)[C@H](c1ccccc1)[C@@H]1CCCCN1 ZINC000217526272 BD In-Stock Unstable SLC6A3 15 71 CNC(=O)[C@H](c1ccccc1)[C@@H]1CCCCN1 ZINC000217526272 BD In-Stock Unstable BIRC8 41 32 NC[C@@H]1CCCN([C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217526297 CD For-Sale Unstable DRD2 22 48 NC[C@@H]1CCCN([C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217526297 CD For-Sale Unstable DRD4 40 43 NC[C@@H]1CCCN([C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217526297 CD For-Sale Unstable ACHE 38 44 NC[C@@H]1CCCN([C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217526297 CD For-Sale Unstable DRD3 28 45 NC[C@@H]1CCCN([C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217526297 CD For-Sale Unstable SIGMAR1 60 44 NC[C@@H]1CCCN([C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217526297 CD For-Sale Unstable CCR3 16 43 NC[C@@H]1CCCN([C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217526297 CD For-Sale Unstable SLC18A3 26 45 O=[N+]([O-])c1cncc(B(O)O)c1 ZINC000217526303 AA For-Sale Reactive APR 0 55 COc1cccc(C(=O)NCC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217526326 GE In-Stock Unstable DRD4 54 42 COc1cccc(C(=O)NCC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217526326 GE In-Stock Unstable NPY5R 45 57 CNC(=O)[C@@H](c1ccccc1)[C@@H]1CCCCN1 ZINC000217526348 BD In-Stock Unstable SLC6A1 26 73 CNC(=O)[C@@H](c1ccccc1)[C@@H]1CCCCN1 ZINC000217526348 BD In-Stock Unstable SLC6A3 15 71 CNC(=O)[C@@H](c1ccccc1)[C@@H]1CCCCN1 ZINC000217526348 BD In-Stock Unstable BIRC8 41 32 CC(C)CNC(=O)[C@H](C)N1CCC[C@@H](N)C1 ZINC000217526352 BC On-Demand Unstable TPP2 19 40 CCO[C@@H]1C[C@@H](Nc2ccnc3ccccc23)C1(C)C ZINC000217526353 CH For-Sale Unstable HNMT 48 37 CCCCN(CCCC)C(=O)NCCc1ccc(F)cc1 ZINC000217526360 CH On-Demand Unstable THRA 0 41 CCCCN(CCCC)C(=O)NCCc1ccc(F)cc1 ZINC000217526360 CH On-Demand Unstable CNR2 24 41 CCCCN(CCCC)C(=O)NCCc1ccc(F)cc1 ZINC000217526360 CH On-Demand Unstable TSPO 24 42 CCCCN(CCCC)C(=O)NCCc1ccc(F)cc1 ZINC000217526360 CH On-Demand Unstable S1PR2 41 38 CCCCN(CCCC)C(=O)NCCc1ccc(F)cc1 ZINC000217526360 CH On-Demand Unstable PLM2_PLAFA 41 40 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1N[C@@H](C)c1ccc(Br)s1 ZINC000217526372 EK For-Sale Unstable TRPM8 15 42 Cn1cccc(C(=O)NCC[C@H](O)c2ccsc2)c1=O ZINC000217526373 CD In-Stock Unstable POLR1A 50 31 CCC[C@@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1N1CCCC1 ZINC000217526401 EE In-Stock Unstable KCNQ2 52 39 CNC(=O)[C@H](c1ccccc1)[C@H]1CCCCN1 ZINC000217526428 BD In-Stock Unstable SLC6A1 26 73 CNC(=O)[C@H](c1ccccc1)[C@H]1CCCCN1 ZINC000217526428 BD In-Stock Unstable SLC6A3 15 71 CNC(=O)[C@H](c1ccccc1)[C@H]1CCCCN1 ZINC000217526428 BD In-Stock Unstable BIRC8 41 32 C[C@@H](C(=O)Nc1ccccc1)N1CCC[C@@H](N)C1 ZINC000217526438 BD On-Demand Unstable ACE 31 43 C[C@@H](C(=O)Nc1ccccc1)N1CCC[C@@H](N)C1 ZINC000217526438 BD On-Demand Unstable XIAP 42 35 C[C@@H](C(=O)Nc1ccccc1)N1CCC[C@@H](N)C1 ZINC000217526438 BD On-Demand Unstable BIRC2 51 37 CN1CCC(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)CC1 ZINC000217526443 EE For-Sale Unstable NPY5R 60 51 CCO[C@H]1C[C@@H](Nc2ccnc3ccccc23)C1(C)C ZINC000217526449 CH For-Sale Unstable HNMT 48 37 Cn1cccc(C(=O)NCC[C@@H](O)c2ccsc2)c1=O ZINC000217526458 CD In-Stock Unstable POLR1A 50 31 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1N[C@@H](C)c1ccc(Br)s1 ZINC000217526461 EK For-Sale Unstable TRPM8 15 42 CCC[C@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1N1CCCC1 ZINC000217526475 EE In-Stock Unstable KCNQ2 52 39 O=C1/C(=C/N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)SC(=S)N1C[C@H]1CCCO1 ZINC000217526494 HE In-Stock Unstable CHRNA4 25 41 CCCCOc1ccc(C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc1 ZINC000217526509 HI For-Sale Unstable GCGR 38 40 CCCCOc1ccc(C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc1 ZINC000217526509 HI For-Sale Unstable PLA2G4B 49 34 CNC(=O)[C@@H](c1ccccc1)[C@H]1CCCCN1 ZINC000217526511 BD In-Stock Unstable SLC6A1 26 73 CNC(=O)[C@@H](c1ccccc1)[C@H]1CCCCN1 ZINC000217526511 BD In-Stock Unstable SLC6A3 15 71 CNC(=O)[C@@H](c1ccccc1)[C@H]1CCCCN1 ZINC000217526511 BD In-Stock Unstable BIRC8 41 32 CCO[C@@H]1C[C@H](Nc2ccnc3ccccc23)C1(C)C ZINC000217526536 CH For-Sale Unstable HNMT 48 37 C[C@H](C(=O)Nc1ccccc1)N1CCC[C@@H](N)C1 ZINC000217526545 BD On-Demand Unstable ACE 31 43 C[C@H](C(=O)Nc1ccccc1)N1CCC[C@@H](N)C1 ZINC000217526545 BD On-Demand Unstable XIAP 42 35 C[C@H](C(=O)Nc1ccccc1)N1CCC[C@@H](N)C1 ZINC000217526545 BD On-Demand Unstable BIRC2 51 37 CC(C)[C@H]1CC[C@H](C)C[C@@H]1N[C@@H](C)c1ccc(Br)s1 ZINC000217526549 EK For-Sale Unstable TRPM8 15 42 O=C1OC2(CCN(C(=O)Cn3cc(-c4ccc(F)cc4)cn3)CC2)c2ccccc21 ZINC000217526561 HG For-Sale Unstable NPY5R 53 60 CCC[C@@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1N1CCCCC1 ZINC000217526595 FF In-Stock Unstable KCNQ2 51 39 CCO[C@H]1C[C@H](Nc2ccnc3ccccc23)C1(C)C ZINC000217526619 CH For-Sale Unstable HNMT 48 37 CCNC(=O)[C@H](c1ccccc1)[C@@H]1CCCCN1 ZINC000217526639 BE In-Stock Unstable SLC6A2 18 67 CCNC(=O)[C@H](c1ccccc1)[C@@H]1CCCCN1 ZINC000217526639 BE In-Stock Unstable SLC6A1 30 67 CCNC(=O)[C@H](c1ccccc1)[C@@H]1CCCCN1 ZINC000217526639 BE In-Stock Unstable SLC6A3 16 67 CCNC(=O)[C@H](c1ccccc1)[C@@H]1CCCCN1 ZINC000217526639 BE In-Stock Unstable AMY2 43 30 COc1ccc(Cl)cc1CN[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217526649 DJ For-Sale Unstable TACR1 29 40 COc1ccc(Cl)cc1CN[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217526649 DJ For-Sale Unstable TRPM8 16 48 O=C1OC2(CCN(C(=O)c3n[nH]c4cc(F)ccc34)CC2)c2ccccc21 ZINC000217526660 FG For-Sale Unstable AVPR1A 24 56 O=C1OC2(CCN(C(=O)c3n[nH]c4cc(F)ccc34)CC2)c2ccccc21 ZINC000217526660 FG For-Sale Unstable NPY5R 48 54 CCC[C@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1N1CCCCC1 ZINC000217526686 FF In-Stock Unstable KCNQ2 51 39 CCNC(=O)[C@@H](c1ccccc1)[C@@H]1CCCCN1 ZINC000217526708 BE In-Stock Unstable SLC6A2 18 67 CCNC(=O)[C@@H](c1ccccc1)[C@@H]1CCCCN1 ZINC000217526708 BE In-Stock Unstable SLC6A1 0 67 CCNC(=O)[C@@H](c1ccccc1)[C@@H]1CCCCN1 ZINC000217526708 BE In-Stock Unstable SLC6A3 16 67 CCNC(=O)[C@@H](c1ccccc1)[C@@H]1CCCCN1 ZINC000217526708 BE In-Stock Unstable AMY2 43 30 O=C(NCCc1ccc(F)cc1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217526718 EJ On-Demand Unstable CA2 18 60 O=C(NCCc1ccc(F)cc1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217526718 EJ On-Demand Unstable ADRB2 15 41 O=C(NCCc1ccc(F)cc1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217526718 EJ On-Demand Unstable ADRB1 43 41 O=C(NCCc1ccc(F)cc1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217526718 EJ On-Demand Unstable ADRB3 33 41 O=C(NCCc1ccc(F)cc1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217526718 EJ On-Demand Unstable CA1 28 53 O=C(NCCc1ccc(F)cc1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217526718 EJ On-Demand Unstable CCR3 54 52 O=C(NCCc1ccc(F)cc1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217526718 EJ On-Demand Unstable MMP3 15 43 O=C(NCCc1ccc(F)cc1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217526718 EJ On-Demand Unstable EPHX2 22 43 O=C(NCCc1ccc(F)cc1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217526718 EJ On-Demand Unstable CA12 21 60 O=C(NCCc1ccc(F)cc1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217526718 EJ On-Demand Unstable CA9 22 57 O=C(NCCc1ccc(F)cc1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217526718 EJ On-Demand Unstable NCE103 26 57 O=C(NCCc1ccc(F)cc1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217526718 EJ On-Demand Unstable P96878_MYCTU 21 40 O=C(NCCc1ccc(F)cc1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217526718 EJ On-Demand Unstable ACAT 0 45 O=C(NCCc1ccc(F)cc1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217526718 EJ On-Demand Unstable UPPS 0 41 O=C(NCCc1ccc(F)cc1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217526718 EJ On-Demand Unstable NAMPT 25 40 O=C(NCCc1ccc(F)cc1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217526718 EJ On-Demand Unstable P95276_MYCTO 0 43 COc1ccc(Cl)cc1CN[C@H]1C[C@H](C)CC[C@@H]1C(C)C ZINC000217526739 DJ For-Sale Unstable TACR1 29 40 COc1ccc(Cl)cc1CN[C@H]1C[C@H](C)CC[C@@H]1C(C)C ZINC000217526739 DJ For-Sale Unstable TRPM8 16 48 O=C1OC2(CCN(C(=O)CC34CC5CC(CC(C5)C3)C4)CC2)c2ccccc21 ZINC000217526766 GI For-Sale Unstable NPY5R 45 48 NC[C@@H]1CCCN([C@@H]2CCCN(Cc3ccccc3)C2)C1 ZINC000217526785 CE For-Sale Unstable DRD4 29 40 NC[C@@H]1CCCN([C@@H]2CCCN(Cc3ccccc3)C2)C1 ZINC000217526785 CE For-Sale Unstable ACHE 27 41 NC[C@@H]1CCCN([C@@H]2CCCN(Cc3ccccc3)C2)C1 ZINC000217526785 CE For-Sale Unstable SIGMAR1 54 47 NC[C@@H]1CCCN([C@@H]2CCCN(Cc3ccccc3)C2)C1 ZINC000217526785 CE For-Sale Unstable SLC18A3 24 42 NC[C@@H]1CCCN([C@@H]2CCCN(Cc3ccccc3)C2)C1 ZINC000217526785 CE For-Sale Unstable MC3R 15 43 O=C(NCC[C@H](O)c1ccsc1)c1cccc(Cl)c1 ZINC000217526787 CG In-Stock Unstable CCKBR 0 40 CCNC(=O)[C@H](c1ccccc1)[C@H]1CCCCN1 ZINC000217526799 BE In-Stock Unstable SLC6A2 18 67 CCNC(=O)[C@H](c1ccccc1)[C@H]1CCCCN1 ZINC000217526799 BE In-Stock Unstable SLC6A1 30 67 CCNC(=O)[C@H](c1ccccc1)[C@H]1CCCCN1 ZINC000217526799 BE In-Stock Unstable SLC6A3 16 67 CCNC(=O)[C@H](c1ccccc1)[C@H]1CCCCN1 ZINC000217526799 BE In-Stock Unstable AMY2 43 30 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1N[C@@H]1CCc2cc(Br)ccc21 ZINC000217526827 FK For-Sale Unstable TRPM8 0 40 CC[C@H](C)N1C(=O)/C(=C/N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)SC1=S ZINC000217526839 GF In-Stock Unstable CHRNA4 27 44 O=C(/C=C\c1cccc(Cl)c1)NCC1CC(O)C1 ZINC000217526856 CE For-Sale Unstable HDAC8 53 37 O=C1OC2(CCN(C(=O)c3ccc(-c4cccs4)cc3)CC2)c2ccccc21 ZINC000217526881 GJ In-Stock Unstable NPY5R 48 51 CCNC(=O)[C@@H](c1ccccc1)[C@H]1CCCCN1 ZINC000217526884 BE In-Stock Unstable SLC6A2 18 67 CCNC(=O)[C@@H](c1ccccc1)[C@H]1CCCCN1 ZINC000217526884 BE In-Stock Unstable SLC6A1 30 67 CCNC(=O)[C@@H](c1ccccc1)[C@H]1CCCCN1 ZINC000217526884 BE In-Stock Unstable SLC6A3 16 67 CCNC(=O)[C@@H](c1ccccc1)[C@H]1CCCCN1 ZINC000217526884 BE In-Stock Unstable AMY2 43 30 O=C(NCC[C@@H](O)c1ccsc1)c1cccc(Cl)c1 ZINC000217526893 CG In-Stock Unstable CCKBR 0 40 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1N[C@@H]1CCc2cc(Br)ccc21 ZINC000217526909 FK For-Sale Unstable TRPM8 0 40 C[C@H](c1cccc(OC(F)F)c1)N1CCC[C@@H](CN)C1 ZINC000217526922 CG For-Sale Unstable CHRNA10 40 33 N[C@H](C(=O)O)c1ccc(Br)c(O)c1 ZINC000217526925 BD For-Sale Unstable GRM8 17 53 CC[C@@H](C)N1C(=O)/C(=C/N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)SC1=S ZINC000217526938 GF In-Stock Unstable CHRNA4 27 44 O=C(/C=C\c1ccc(Cl)cc1Cl)NC1CC(O)C1 ZINC000217526965 CF For-Sale Unstable BOTA 36 65 COCCC(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217526996 CD For-Sale Unstable NPY5R 42 51 N[C@@H](C(=O)O)c1ccc(Br)c(O)c1 ZINC000217526997 BD For-Sale Unstable CACNA2D1 27 56 N[C@@H](C(=O)O)c1ccc(Br)c(O)c1 ZINC000217526997 BD For-Sale Unstable SLC7A11 0 53 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1N[C@@H]1CCc2cc(Br)ccc21 ZINC000217526999 FK For-Sale Unstable TRPM8 0 40 O=C(NC1CC1)[C@H](c1ccccc1)[C@@H]1CCCCN1 ZINC000217527002 CE In-Stock Unstable SLC6A1 24 68 O=C(NC1CC1)[C@H](c1ccccc1)[C@@H]1CCCCN1 ZINC000217527002 CE In-Stock Unstable C3AR1 43 45 O=C(NC1CC1)[C@H](c1ccccc1)[C@@H]1CCCCN1 ZINC000217527002 CE In-Stock Unstable EPHX2 24 42 O=C(NC1CC1)[C@H](c1ccccc1)[C@@H]1CCCCN1 ZINC000217527002 CE In-Stock Unstable NMUR2 0 43 O=C(NC1CC1)[C@H](c1ccccc1)[C@@H]1CCCCN1 ZINC000217527002 CE In-Stock Unstable NMUR1 0 43 C[C@@H](c1cccc(OC(F)F)c1)N1CCC[C@@H](CN)C1 ZINC000217527016 CG For-Sale Unstable CHRNA10 40 33 O=C(Nc1ccccc1C(=O)N1CCCC1)[C@@H]1C[C@@H]1c1ccc(C(F)(F)F)cc1 ZINC000217527022 HJ On-Demand Unstable MTTP 30 44 O=C(Nc1ccccc1C(=O)N1CCCC1)[C@@H]1C[C@@H]1c1ccc(C(F)(F)F)cc1 ZINC000217527022 HJ On-Demand Unstable EPHX2 18 44 O=C(Nc1ccccc1C(=O)N1CCCC1)[C@@H]1C[C@@H]1c1ccc(C(F)(F)F)cc1 ZINC000217527022 HJ On-Demand Unstable RBP4 58 39 O=C(Nc1ccccc1C(=O)N1CCCC1)[C@@H]1C[C@@H]1c1ccc(C(F)(F)F)cc1 ZINC000217527022 HJ On-Demand Unstable NPSR1 15 41 O=C(Nc1ccccc1C(=O)N1CCCC1)[C@@H]1C[C@@H]1c1ccc(C(F)(F)F)cc1 ZINC000217527022 HJ On-Demand Unstable TRPM8 51 38 O=C(NCc1nc(-c2ccccc2)n[nH]1)c1ccnc2ccccc12 ZINC000217527044 EF In-Stock Unstable PREP 30 44 O=C(NCc1nc(-c2ccccc2)n[nH]1)c1ccnc2ccccc12 ZINC000217527044 EF In-Stock Unstable TACR3 43 37 O=C(NCc1nc(-c2ccccc2)n[nH]1)c1ccnc2ccccc12 ZINC000217527044 EF In-Stock Unstable FAP 0 47 O=C1/C(=C/N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)SC(=S)N1CCc1ccccc1 ZINC000217527049 IG In-Stock Unstable CHRNA4 30 52 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc(-c2ccccc2)cc1 ZINC000217527073 HJ For-Sale Unstable FABP4 40 34 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc(-c2ccccc2)cc1 ZINC000217527073 HJ For-Sale Unstable BCHE 21 40 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc(-c2ccccc2)cc1 ZINC000217527073 HJ For-Sale Unstable PLD2 41 32 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc(-c2ccccc2)cc1 ZINC000217527073 HJ For-Sale Unstable GIPR 58 35 Cc1cccc(/C=C\C(=O)NC2CC(O)C2)c1 ZINC000217527078 BD For-Sale Unstable HDAC8 61 42 Cc1cccc(/C=C\C(=O)NC2CC(O)C2)c1 ZINC000217527078 BD For-Sale Unstable MMP2 22 49 Cc1cccc(/C=C\C(=O)NC2CC(O)C2)c1 ZINC000217527078 BD For-Sale Unstable HDAC1 24 43 Cc1cccc(/C=C\C(=O)NC2CC(O)C2)c1 ZINC000217527078 BD For-Sale Unstable HDAC6 40 43 Cc1cccc(/C=C\C(=O)NC2CC(O)C2)c1 ZINC000217527078 BD For-Sale Unstable MMP9 0 49 Cc1cccc(/C=C\C(=O)NC2CC(O)C2)c1 ZINC000217527078 BD For-Sale Unstable MMP1 22 49 Cc1cccc(/C=C\C(=O)NC2CC(O)C2)c1 ZINC000217527078 BD For-Sale Unstable HDA106 0 43 Cc1cccc(/C=C\C(=O)NC2CC(O)C2)c1 ZINC000217527078 BD For-Sale Unstable HD1B 0 43 CC(C)[C@H]1CC[C@H](C)C[C@@H]1N[C@@H]1CCc2cc(Br)ccc21 ZINC000217527082 FK For-Sale Unstable TRPM8 0 40 O=C(NC1CC1)[C@@H](c1ccccc1)[C@@H]1CCCCN1 ZINC000217527085 CE In-Stock Unstable SLC6A1 24 68 O=C(NC1CC1)[C@@H](c1ccccc1)[C@@H]1CCCCN1 ZINC000217527085 CE In-Stock Unstable C3AR1 43 45 O=C(NC1CC1)[C@@H](c1ccccc1)[C@@H]1CCCCN1 ZINC000217527085 CE In-Stock Unstable EPHX2 24 42 O=C(NC1CC1)[C@@H](c1ccccc1)[C@@H]1CCCCN1 ZINC000217527085 CE In-Stock Unstable NMUR2 0 43 O=C(NC1CC1)[C@@H](c1ccccc1)[C@@H]1CCCCN1 ZINC000217527085 CE In-Stock Unstable NMUR1 0 43 Cn1nc(-c2ccccc2)cc1C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217527108 GG For-Sale Unstable NPY5R 61 59 O=C(Nc1ccccc1C(=O)N1CCCC1)[C@H]1C[C@@H]1c1ccc(C(F)(F)F)cc1 ZINC000217527119 HJ On-Demand Unstable MTTP 30 44 O=C(Nc1ccccc1C(=O)N1CCCC1)[C@H]1C[C@@H]1c1ccc(C(F)(F)F)cc1 ZINC000217527119 HJ On-Demand Unstable EPHX2 18 44 O=C(Nc1ccccc1C(=O)N1CCCC1)[C@H]1C[C@@H]1c1ccc(C(F)(F)F)cc1 ZINC000217527119 HJ On-Demand Unstable RBP4 58 39 O=C(Nc1ccccc1C(=O)N1CCCC1)[C@H]1C[C@@H]1c1ccc(C(F)(F)F)cc1 ZINC000217527119 HJ On-Demand Unstable NPSR1 15 41 O=C(Nc1ccccc1C(=O)N1CCCC1)[C@H]1C[C@@H]1c1ccc(C(F)(F)F)cc1 ZINC000217527119 HJ On-Demand Unstable TRPM8 51 38 CCCN1C(=O)/C(=C/N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)SC1=S ZINC000217527162 GE In-Stock Unstable CHRNA4 37 52 O=C(NC1CC1)[C@H](c1ccccc1)[C@H]1CCCCN1 ZINC000217527170 CE In-Stock Unstable SLC6A1 24 68 O=C(NC1CC1)[C@H](c1ccccc1)[C@H]1CCCCN1 ZINC000217527170 CE In-Stock Unstable C3AR1 43 45 O=C(NC1CC1)[C@H](c1ccccc1)[C@H]1CCCCN1 ZINC000217527170 CE In-Stock Unstable EPHX2 24 42 O=C(NC1CC1)[C@H](c1ccccc1)[C@H]1CCCCN1 ZINC000217527170 CE In-Stock Unstable NMUR2 0 43 O=C(NC1CC1)[C@H](c1ccccc1)[C@H]1CCCCN1 ZINC000217527170 CE In-Stock Unstable NMUR1 0 43 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1cccc(Br)c1 ZINC000217527179 HH For-Sale Unstable DRD4 44 34 CCc1ccc([C@@H](C)N[C@@H]2C[C@@H](C)CC[C@@H]2C(C)C)s1 ZINC000217527189 CK For-Sale Unstable TRPM8 15 40 O=Cc1ccc(Oc2ccc([N+](=O)[O-])cc2)c(Br)c1 ZINC000217527207 DH On-Demand Bother ENR 0 51 O=Cc1ccc(Oc2ccc([N+](=O)[O-])cc2)c(Br)c1 ZINC000217527207 DH On-Demand Bother PPOX1 16 50 O=C(Nc1ccccc1C(=O)N1CCCC1)[C@@H]1C[C@H]1c1ccc(C(F)(F)F)cc1 ZINC000217527221 HJ On-Demand Unstable MTTP 30 44 O=C(Nc1ccccc1C(=O)N1CCCC1)[C@@H]1C[C@H]1c1ccc(C(F)(F)F)cc1 ZINC000217527221 HJ On-Demand Unstable EPHX2 18 44 O=C(Nc1ccccc1C(=O)N1CCCC1)[C@@H]1C[C@H]1c1ccc(C(F)(F)F)cc1 ZINC000217527221 HJ On-Demand Unstable RBP4 58 39 O=C(Nc1ccccc1C(=O)N1CCCC1)[C@@H]1C[C@H]1c1ccc(C(F)(F)F)cc1 ZINC000217527221 HJ On-Demand Unstable NPSR1 15 41 O=C(Nc1ccccc1C(=O)N1CCCC1)[C@@H]1C[C@H]1c1ccc(C(F)(F)F)cc1 ZINC000217527221 HJ On-Demand Unstable TRPM8 51 38 O=C1OC2(CCN(C(=O)CSc3ccncc3)CC2)c2ccccc21 ZINC000217527233 FF For-Sale Unstable NPY5R 53 48 O=C(NC1CC1)[C@@H](c1ccccc1)[C@H]1CCCCN1 ZINC000217527259 CE In-Stock Unstable SLC6A1 24 68 O=C(NC1CC1)[C@@H](c1ccccc1)[C@H]1CCCCN1 ZINC000217527259 CE In-Stock Unstable C3AR1 43 45 O=C(NC1CC1)[C@@H](c1ccccc1)[C@H]1CCCCN1 ZINC000217527259 CE In-Stock Unstable EPHX2 24 42 O=C(NC1CC1)[C@@H](c1ccccc1)[C@H]1CCCCN1 ZINC000217527259 CE In-Stock Unstable NMUR2 0 43 O=C(NC1CC1)[C@@H](c1ccccc1)[C@H]1CCCCN1 ZINC000217527259 CE In-Stock Unstable NMUR1 0 43 COCCCN1C(=O)/C(=C/N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)SC1=S ZINC000217527272 HE In-Stock Unstable CHRNA4 27 43 CCc1ccc([C@H](C)N[C@@H]2C[C@@H](C)CC[C@@H]2C(C)C)s1 ZINC000217527291 CK For-Sale Unstable TRPM8 15 40 O=C(Nc1ccccc1C(=O)N1CCCC1)[C@H]1C[C@H]1c1ccc(C(F)(F)F)cc1 ZINC000217527298 HJ On-Demand Unstable MTTP 30 44 O=C(Nc1ccccc1C(=O)N1CCCC1)[C@H]1C[C@H]1c1ccc(C(F)(F)F)cc1 ZINC000217527298 HJ On-Demand Unstable EPHX2 18 44 O=C(Nc1ccccc1C(=O)N1CCCC1)[C@H]1C[C@H]1c1ccc(C(F)(F)F)cc1 ZINC000217527298 HJ On-Demand Unstable RBP4 58 39 O=C(Nc1ccccc1C(=O)N1CCCC1)[C@H]1C[C@H]1c1ccc(C(F)(F)F)cc1 ZINC000217527298 HJ On-Demand Unstable NPSR1 15 41 O=C(Nc1ccccc1C(=O)N1CCCC1)[C@H]1C[C@H]1c1ccc(C(F)(F)F)cc1 ZINC000217527298 HJ On-Demand Unstable TRPM8 51 38 CCCC(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217527354 CE For-Sale Unstable NPY5R 47 50 CCc1ccc([C@@H](C)N[C@H]2C[C@@H](C)CC[C@@H]2C(C)C)s1 ZINC000217527358 CK For-Sale Unstable TRPM8 15 40 CCN(CCc1ccncc1)C(=O)NCCc1ccc(F)cc1 ZINC000217527372 DG For-Sale Unstable GNRHR 15 40 O=C(/C=C\c1ccc2c(c1)OCO2)NC1CC(O)C1 ZINC000217527393 CD For-Sale Unstable HDAC1 0 52 O=C(/C=C\c1ccc2c(c1)OCO2)NC1CC(O)C1 ZINC000217527393 CD For-Sale Unstable DYRK2 66 35 CCCCN1C(=O)/C(=C/N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)SC1=S ZINC000217527394 GF In-Stock Unstable CHRNA4 37 55 CCc1ccc([C@H](C)N[C@H]2C[C@@H](C)CC[C@@H]2C(C)C)s1 ZINC000217527438 CK For-Sale Unstable TRPM8 15 40 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccccc1Br ZINC000217527439 HH For-Sale Unstable FABP4 42 36 O=C(NCCc1ccc(F)cc1)Nc1ccccc1N1CCOCC1 ZINC000217527475 EG For-Sale Unstable KCNQ2 87 55 O=C(NCCc1ccc(F)cc1)Nc1ccccc1N1CCOCC1 ZINC000217527475 EG For-Sale Unstable CCR3 53 47 O=C(NCCc1ccc(F)cc1)Nc1ccccc1N1CCOCC1 ZINC000217527475 EG For-Sale Unstable MTOR 25 41 O=C(NCCc1ccc(F)cc1)Nc1ccccc1N1CCOCC1 ZINC000217527475 EG For-Sale Unstable CSF1R 0 48 Cc1noc(C)c1CCC(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217527476 FF For-Sale Unstable NPY5R 39 46 CO[C@@H]1CC[C@@H](NC(=O)CCc2cccnc2)CC1 ZINC000217527501 CE In-Stock Unstable GRIN2B 15 45 CO[C@@H]1CC[C@@H](NC(=O)CCc2cccnc2)CC1 ZINC000217527501 CE In-Stock Unstable TBXAS1 36 47 CO[C@@H]1CC[C@@H](NC(=O)CCc2cccnc2)CC1 ZINC000217527501 CE In-Stock Unstable NPY2R 46 36 CO[C@@H]1CC[C@@H](NC(=O)CCc2cccnc2)CC1 ZINC000217527501 CE In-Stock Unstable CHRNA7 37 40 CO[C@@H]1CC[C@@H](NC(=O)CCc2cccnc2)CC1 ZINC000217527501 CE In-Stock Unstable C3AR1 55 48 CO[C@@H]1CC[C@@H](NC(=O)CCc2cccnc2)CC1 ZINC000217527501 CE In-Stock Unstable ACHP_LYMST 21 40 CO[C@@H]1CC[C@@H](NC(=O)CCc2cccnc2)CC1 ZINC000217527501 CE In-Stock Unstable TNKS 50 37 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1N[C@@H]1C[C@@H]2CC[C@@H]1C2 ZINC000217527522 BI For-Sale Unstable TRPM8 0 41 O=C(CCCc1cn(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)c2ccccc12)N1CCCCCC1 ZINC000217527535 JJ In-Stock Unstable CHRNA4 30 52 COc1cc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc(OC)c1OC ZINC000217527586 GG For-Sale Unstable HRH1 24 42 COc1cc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc(OC)c1OC ZINC000217527586 GG For-Sale Unstable AVPR1A 15 52 COc1cc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc(OC)c1OC ZINC000217527586 GG For-Sale Unstable TACR1 21 43 COc1cc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc(OC)c1OC ZINC000217527586 GG For-Sale Unstable TACR2 21 43 COc1cc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc(OC)c1OC ZINC000217527586 GG For-Sale Unstable ACACA 54 40 COc1cc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc(OC)c1OC ZINC000217527586 GG For-Sale Unstable ACACB 34 40 COc1cc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc(OC)c1OC ZINC000217527586 GG For-Sale Unstable NPY5R 43 57 COc1cc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc(OC)c1OC ZINC000217527586 GG For-Sale Unstable ACKR3 40 33 Cc1c(Br)c(C)c2c(c1Br)O[C@H](C(F)(F)F)C(C(=O)O)=C2 ZINC000217527590 IJ Annotated Unstable PTGS1 17 51 N#CSc1ccc(NC(=O)NCCc2ccc(F)cc2)cc1 ZINC000217527600 DH For-Sale Unstable ADRB1 39 41 N#CSc1ccc(NC(=O)NCCc2ccc(F)cc2)cc1 ZINC000217527600 DH For-Sale Unstable CCR3 36 45 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1N[C@@H]1C[C@@H]2CC[C@@H]1C2 ZINC000217527610 BI For-Sale Unstable TRPM8 0 41 Cn1cc(CCNc2ccc(Cl)cc2Br)cn1 ZINC000217527620 DG On-Demand Unstable HNMT 40 33 Cc1c(Br)c(C)c2c(c1Br)O[C@@H](C(F)(F)F)C(C(=O)O)=C2 ZINC000217527672 IJ Annotated Unstable PTGS1 17 51 CN1CCN(C(=O)Cc2cn(CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)c3ccccc23)CC1 ZINC000217527679 JE In-Stock Unstable CHRNA4 31 51 O=C1OC2(CCN(C(=O)c3ccccc3Cl)CC2)c2ccccc21 ZINC000217527690 EH In-Stock Unstable AVPR1A 26 64 O=C1OC2(CCN(C(=O)c3ccccc3Cl)CC2)c2ccccc21 ZINC000217527690 EH In-Stock Unstable NPY5R 57 59 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1N[C@@H]1C[C@@H]2CC[C@@H]1C2 ZINC000217527699 BI For-Sale Unstable TRPM8 0 41 O=C(NCCc1ccc(F)cc1)N(Cc1ccccc1)c1ccccc1 ZINC000217527720 EJ For-Sale Unstable LIMK2 30 40 O=[N+]([O-])c1cccc(CNc2cc(F)cc(Cl)c2)c1 ZINC000217527742 CH On-Demand Unstable CACNA1D 53 37 O=C(NCC[C@H](O)c1ccsc1)c1ccc(Cl)s1 ZINC000217527752 DG In-Stock Unstable F10 0 41 CC(C)[C@H]1CC[C@H](C)C[C@@H]1N[C@@H]1C[C@@H]2CC[C@@H]1C2 ZINC000217527792 BI For-Sale Unstable TRPM8 0 41 O=C1OC2(CCN(C(=O)COc3ccc4ccccc4c3)CC2)c2ccccc21 ZINC000217527806 GH For-Sale Unstable HTR1B 19 43 O=C1OC2(CCN(C(=O)COc3ccc4ccccc4c3)CC2)c2ccccc21 ZINC000217527806 GH For-Sale Unstable NPY5R 45 48 O=C(NCC[C@@H](O)c1ccsc1)c1ccc(Cl)s1 ZINC000217527827 DG In-Stock Unstable F10 0 41 O=C(NCCc1ccc(F)cc1)Nc1ccc2ccccc2c1 ZINC000217527835 DI On-Demand Unstable ADRB1 28 40 O=C(NCCc1ccc(F)cc1)Nc1ccc2ccccc2c1 ZINC000217527835 DI On-Demand Unstable CA1 22 48 O=C(NCCc1ccc(F)cc1)Nc1ccc2ccccc2c1 ZINC000217527835 DI On-Demand Unstable TRPV1 17 48 O=C(NCCc1ccc(F)cc1)Nc1ccc2ccccc2c1 ZINC000217527835 DI On-Demand Unstable CCR3 79 42 O=C(NCCc1ccc(F)cc1)Nc1ccc2ccccc2c1 ZINC000217527835 DI On-Demand Unstable RAF1 37 45 O=C(NCCc1ccc(F)cc1)Nc1ccc2ccccc2c1 ZINC000217527835 DI On-Demand Unstable ECE1 0 42 O=C(NCCc1ccc(F)cc1)Nc1ccc2ccccc2c1 ZINC000217527835 DI On-Demand Unstable EPHX2 15 41 O=C(NCCc1ccc(F)cc1)Nc1ccc2ccccc2c1 ZINC000217527835 DI On-Demand Unstable CA12 18 48 O=C(NCCc1ccc(F)cc1)Nc1ccc2ccccc2c1 ZINC000217527835 DI On-Demand Unstable CA9 17 48 O=C(NCCc1ccc(F)cc1)Nc1ccc2ccccc2c1 ZINC000217527835 DI On-Demand Unstable Q8MMZ8_EIMTE 24 45 O=C(NCCc1ccc(F)cc1)Nc1ccc2ccccc2c1 ZINC000217527835 DI On-Demand Unstable NCE103 28 48 O=C(NCCc1ccc(F)cc1)Nc1ccc2ccccc2c1 ZINC000217527835 DI On-Demand Unstable PRMT3 41 39 O=C(NCCc1ccc(F)cc1)Nc1ccc2ccccc2c1 ZINC000217527835 DI On-Demand Unstable ACAT 0 53 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCc1c(Cl)ccc(Cl)c1Cl ZINC000217527916 EK For-Sale Unstable TRPM8 16 47 NS(=O)(=O)c1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217527920 GD For-Sale Unstable AVPR1A 15 48 NS(=O)(=O)c1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217527920 GD For-Sale Unstable NPY5R 38 48 CC[C@H](C(=O)NCC[C@H](O)c1ccsc1)c1ccccc1 ZINC000217527932 DG In-Stock Unstable KCNQ2 42 41 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCc1c(Cl)ccc(Cl)c1Cl ZINC000217527997 EK For-Sale Unstable TRPM8 16 47 CC[C@@H](C(=O)NCC[C@H](O)c1ccsc1)c1ccccc1 ZINC000217528018 DG In-Stock Unstable KCNQ2 42 41 O=C1OC2(CCN(C(=O)c3cc4ccccc4[nH]3)CC2)c2ccccc21 ZINC000217528036 EG For-Sale Unstable AVPR1A 23 55 O=C1OC2(CCN(C(=O)c3cc4ccccc4[nH]3)CC2)c2ccccc21 ZINC000217528036 EG For-Sale Unstable HRH4 29 56 O=C1OC2(CCN(C(=O)c3cc4ccccc4[nH]3)CC2)c2ccccc21 ZINC000217528036 EG For-Sale Unstable NPY5R 42 51 O=C1OC2(CCN(C(=O)c3cc4ccccc4[nH]3)CC2)c2ccccc21 ZINC000217528036 EG For-Sale Unstable AKR1C3 36 46 CSc1ccc(CC(=O)NCc2ccc3nc(C)[nH]c3c2)cc1 ZINC000217528054 EG In-Stock Unstable TYMS 52 36 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCc1c(Cl)ccc(Cl)c1Cl ZINC000217528087 EK For-Sale Unstable TRPM8 16 47 CC[C@H](C(=O)NCC[C@@H](O)c1ccsc1)c1ccccc1 ZINC000217528100 DG In-Stock Unstable KCNQ2 42 41 O=C1C[C@H]2c3ccccc3[C@@H]1[C@H]1C(=O)N(c3ccc(F)cc3)C(=O)[C@@H]21 ZINC000217528148 EF In-Stock Unstable ME1 0 40 O=C1OC2(CCN(C(=O)Cn3cccn3)CC2)c2ccccc21 ZINC000217528159 DD In-Stock Unstable NPY5R 55 52 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCc1c(Cl)ccc(Cl)c1Cl ZINC000217528168 EK For-Sale Unstable TRPM8 16 47 CC[C@@H](C(=O)NCC[C@@H](O)c1ccsc1)c1ccccc1 ZINC000217528179 DG In-Stock Unstable KCNQ2 42 41 Cn1cc(/C=C2\C(=O)N(CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)c3cc(Cl)ccc32)c2ccccc21 ZINC000217528193 KJ In-Stock Unstable CHRNA4 35 44 O=CNCCCNC(=O)NCCc1ccc(F)cc1 ZINC000217528203 CC For-Sale Unstable LEF 47 37 COc1ccc(CNS(=O)(=O)N(C)CCCO)cc1 ZINC000217528239 CC For-Sale Unstable CA9 18 40 COc1ccccc1N1CCN(c2cnn([C@@]34C[C@@H]5C[C@@H](C[C@@H](C5)C3)[C@H]4C(=O)O)c(=O)c2Cl)CC1 ZINC000217528248 JG In-Stock Unstable HTR1A 72 45 COc1ccccc1N1CCN(c2cnn([C@@]34C[C@@H]5C[C@@H](C[C@@H](C5)C3)[C@H]4C(=O)O)c(=O)c2Cl)CC1 ZINC000217528248 JG In-Stock Unstable DRD2 45 44 COc1ccccc1N1CCN(c2cnn([C@@]34C[C@@H]5C[C@@H](C[C@@H](C5)C3)[C@H]4C(=O)O)c(=O)c2Cl)CC1 ZINC000217528248 JG In-Stock Unstable ADRA1D 59 36 COc1ccccc1N1CCN(c2cnn([C@@]34C[C@@H]5C[C@@H](C[C@@H](C5)C3)[C@H]4C(=O)O)c(=O)c2Cl)CC1 ZINC000217528248 JG In-Stock Unstable HTR2A 28 41 COc1ccccc1N1CCN(c2cnn([C@@]34C[C@@H]5C[C@@H](C[C@@H](C5)C3)[C@H]4C(=O)O)c(=O)c2Cl)CC1 ZINC000217528248 JG In-Stock Unstable ADRA1A 52 39 COc1ccccc1N1CCN(c2cnn([C@@]34C[C@@H]5C[C@@H](C[C@@H](C5)C3)[C@H]4C(=O)O)c(=O)c2Cl)CC1 ZINC000217528248 JG In-Stock Unstable ADRA1B 48 38 COc1ccccc1N1CCN(c2cnn([C@@]34C[C@@H]5C[C@@H](C[C@@H](C5)C3)[C@H]4C(=O)O)c(=O)c2Cl)CC1 ZINC000217528248 JG In-Stock Unstable DRD3 50 36 COc1ccccc1N1CCN(c2cnn([C@@]34C[C@@H]5C[C@@H](C[C@@H](C5)C3)[C@H]4C(=O)O)c(=O)c2Cl)CC1 ZINC000217528248 JG In-Stock Unstable HTR7 41 39 O=C1OC2(CCN(C(=O)/C=C/c3ccc(Cl)cc3)CC2)c2ccccc21 ZINC000217528271 FI For-Sale Unstable NPY5R 38 57 O=C(/C=C\c1ccc(O)cc1)NCC1CC(O)C1 ZINC000217528322 BD On-Demand Unstable HDAC8 0 53 O=C(/C=C\c1ccc(O)cc1)NCC1CC(O)C1 ZINC000217528322 BD On-Demand Unstable F3 25 45 O=C(/C=C\c1ccc(O)cc1)NCC1CC(O)C1 ZINC000217528322 BD On-Demand Unstable MMP2 0 49 O=C(/C=C\c1ccc(O)cc1)NCC1CC(O)C1 ZINC000217528322 BD On-Demand Unstable MMP9 0 49 O=C(/C=C\c1ccc(O)cc1)NCC1CC(O)C1 ZINC000217528322 BD On-Demand Unstable MMP1 22 49 O=C(/C=C\c1ccc(O)cc1)NCC1CC(O)C1 ZINC000217528322 BD On-Demand Unstable IMA1 0 56 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1N[C@@H](C)c1ccc(Br)cc1Br ZINC000217528333 HK For-Sale Unstable TRPM8 15 43 CCCCCNC(=O)[C@@H](C)N1CCC[C@@H](N)C1 ZINC000217528363 BD On-Demand Unstable TPP2 43 45 COc1ncccc1C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217528383 EE In-Stock Unstable NPY5R 55 53 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1N[C@@H](C)c1ccc(Br)cc1Br ZINC000217528420 HK For-Sale Unstable TRPM8 15 43 CCCCCNC(=O)[C@H](C)N1CCC[C@@H](N)C1 ZINC000217528438 BD On-Demand Unstable TPP2 43 45 O=[N+]([O-])c1ccccc1CNc1cc(F)cc(Cl)c1 ZINC000217528440 CH On-Demand Unstable COLA 83 39 O=C(c1cn(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)c2ccccc12)N1CCN(c2cccc(Cl)c2)CC1 ZINC000217528455 KI In-Stock Unstable CHRNA4 36 47 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1N[C@@H](C)c1ccc(Br)cc1Br ZINC000217528473 HK For-Sale Unstable TRPM8 15 43 CC1(C)C[C@H]2C[C@@](C)(CN2C(=O)NCCc2ccc(F)cc2)C1 ZINC000217528493 DH On-Demand Unstable AVPR2 16 42 CC1(C)C[C@H]2C[C@@](C)(CN2C(=O)NCCc2ccc(F)cc2)C1 ZINC000217528493 DH On-Demand Unstable AVPR1A 35 42 CS(=O)(=O)N1CCC(C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)CC1 ZINC000217528507 HD For-Sale Unstable CTSS 41 35 O=C1OC2(CCN(C(=O)c3ccc4cc[nH]c4c3)CC2)c2ccccc21 ZINC000217528516 EG For-Sale Unstable AVPR1A 23 56 O=C1OC2(CCN(C(=O)c3ccc4cc[nH]c4c3)CC2)c2ccccc21 ZINC000217528516 EG For-Sale Unstable INHA 16 48 O=C1OC2(CCN(C(=O)c3ccc4cc[nH]c4c3)CC2)c2ccccc21 ZINC000217528516 EG For-Sale Unstable ACACA 62 38 O=C1OC2(CCN(C(=O)c3ccc4cc[nH]c4c3)CC2)c2ccccc21 ZINC000217528516 EG For-Sale Unstable ACACB 44 35 O=C1OC2(CCN(C(=O)c3ccc4cc[nH]c4c3)CC2)c2ccccc21 ZINC000217528516 EG For-Sale Unstable NPY5R 41 50 CCCCNC(=O)[C@@H](C)N1CCC[C@@H](N)C1 ZINC000217528540 BC On-Demand Unstable TPP2 47 45 N#Cc1ccc(F)cc1CNc1cc(F)cc(Cl)c1 ZINC000217528552 CI For-Sale Unstable MAP3K8 60 34 C[C@@H](c1ccc(F)cc1)N(C)C(=O)CN(C)S(=O)(=O)c1cccc([N+](=O)[O-])c1 ZINC000217528553 HF On-Demand Unstable COLA 42 42 C[C@@H](c1ccc(F)cc1)N(C)C(=O)CN(C)S(=O)(=O)c1cccc([N+](=O)[O-])c1 ZINC000217528553 HF On-Demand Unstable MMP8 19 41 CC(C)[C@H]1CC[C@H](C)C[C@@H]1N[C@@H](C)c1ccc(Br)cc1Br ZINC000217528587 HK For-Sale Unstable TRPM8 15 43 Cc1n[nH]c([C@@H]2CCCN2C(=O)Cn2ncc3ccccc32)n1 ZINC000217528602 DD In-Stock Unstable PRCP 37 40 Cc1n[nH]c([C@@H]2CCCN2C(=O)Cn2ncc3ccccc32)n1 ZINC000217528602 DD In-Stock Unstable CPT1A 100 46 O=C1OC2(CCN(C(=O)CCCc3ccccc3)CC2)c2ccccc21 ZINC000217528615 EH For-Sale Unstable GHRHR 43 35 O=C1OC2(CCN(C(=O)CCCc3ccccc3)CC2)c2ccccc21 ZINC000217528615 EH For-Sale Unstable SIGMAR1 30 60 O=C1OC2(CCN(C(=O)CCCc3ccccc3)CC2)c2ccccc21 ZINC000217528615 EH For-Sale Unstable PREP 43 42 O=C1OC2(CCN(C(=O)CCCc3ccccc3)CC2)c2ccccc21 ZINC000217528615 EH For-Sale Unstable FAAH 28 42 O=C1OC2(CCN(C(=O)CCCc3ccccc3)CC2)c2ccccc21 ZINC000217528615 EH For-Sale Unstable NPY5R 46 53 CCCCNC(=O)[C@H](C)N1CCC[C@@H](N)C1 ZINC000217528625 BC On-Demand Unstable TPP2 47 45 COc1ccc(/C=C/C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc1OC ZINC000217528626 HH For-Sale Unstable BCHE 17 44 C[C@H](c1ccc(F)cc1)N(C)C(=O)CN(C)S(=O)(=O)c1cccc([N+](=O)[O-])c1 ZINC000217528648 HF On-Demand Unstable COLA 42 42 C[C@H](c1ccc(F)cc1)N(C)C(=O)CN(C)S(=O)(=O)c1cccc([N+](=O)[O-])c1 ZINC000217528648 HF On-Demand Unstable MMP8 19 41 O=C(CCCc1cn(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)c2ccccc12)N1CCOCC1 ZINC000217528654 JG In-Stock Unstable CHRNA4 30 50 Cc1n[nH]c([C@H]2CCCN2C(=O)Cn2ncc3ccccc32)n1 ZINC000217528682 DD In-Stock Unstable PRCP 37 40 Cc1n[nH]c([C@H]2CCCN2C(=O)Cn2ncc3ccccc32)n1 ZINC000217528682 DD In-Stock Unstable CPT1A 100 46 CN(C)c1cccc(NC(=O)NCCc2ccc(F)cc2)c1 ZINC000217528695 DG For-Sale Unstable CCR3 84 45 CN(C)c1cccc(NC(=O)NCCc2ccc(F)cc2)c1 ZINC000217528695 DG For-Sale Unstable RAF1 33 44 CN(C)c1cccc(NC(=O)NCCc2ccc(F)cc2)c1 ZINC000217528695 DG For-Sale Unstable Q8MMZ8_EIMTE 0 44 CN(C)c1cccc(NC(=O)NCCc2ccc(F)cc2)c1 ZINC000217528695 DG For-Sale Unstable ACAT 0 41 CN(C)c1cccc(NC(=O)NCCc2ccc(F)cc2)c1 ZINC000217528695 DG For-Sale Unstable PSBA 0 41 CC[C@@H](N[C@@H]1C[C@@H](C)CC[C@@H]1C(C)C)c1cccc(Br)c1 ZINC000217528713 FK For-Sale Unstable TRPM8 15 42 COc1ccc(OCC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217528721 FF For-Sale Unstable CPT1A 42 37 COc1ccc(OCC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217528721 FF For-Sale Unstable NPY5R 45 54 Cc1nc2ccccc2cc1C(=O)N[C@@H](C)c1nnc2ccccn12 ZINC000217528778 EG On-Demand Unstable POLR1A 59 37 CC[C@H](N[C@@H]1C[C@@H](C)CC[C@@H]1C(C)C)c1cccc(Br)c1 ZINC000217528794 FK For-Sale Unstable TRPM8 15 42 O=C1OC2(CCN(C(=O)Cc3ccc(Br)cc3)CC2)c2ccccc21 ZINC000217528850 HH For-Sale Unstable NPY5R 39 48 CCOc1ccc(C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc1OCC ZINC000217528854 II For-Sale Unstable DRD4 40 31 Cc1ccn2cc(CNC(=O)c3cc(-c4ccsc4)n[nH]3)nc2c1 ZINC000217528859 EG In-Stock Unstable ALPL 43 32 Cc1nc2ccccc2cc1C(=O)N[C@H](C)c1nnc2ccccn12 ZINC000217528867 EG On-Demand Unstable POLR1A 59 37 C[C@@H](C(N)=O)N1CCC[C@@H](N)C1 ZINC000217528870 AB On-Demand Unstable XPNPEP1 54 31 C[C@@H](C(N)=O)N1CCC[C@@H](N)C1 ZINC000217528870 AB On-Demand Unstable XPNPEP2 53 31 CC[C@@H](N[C@H]1C[C@@H](C)CC[C@@H]1C(C)C)c1cccc(Br)c1 ZINC000217528880 FK For-Sale Unstable TRPM8 15 42 CCCCNc1ccc(C(=O)O)cc1S(=O)(=O)N[C@@H](C)COC ZINC000217528891 ED In-Stock Unstable PLA2G4B 41 34 Cn1cc(CC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c2ccccc21 ZINC000217528936 FG In-Stock Unstable PRKCG 51 36 Cn1cc(CC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c2ccccc21 ZINC000217528936 FG In-Stock Unstable NPY5R 38 46 COc1cc(C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc(OC)c1OC ZINC000217528937 IG For-Sale Unstable DRD4 41 32 COc1cc(C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc(OC)c1OC ZINC000217528937 IG For-Sale Unstable BCHE 29 42 NC(=O)c1ccccc1NC(=O)NCCc1ccc(F)cc1 ZINC000217528939 DE For-Sale Unstable CA2 15 46 NC(=O)c1ccccc1NC(=O)NCCc1ccc(F)cc1 ZINC000217528939 DE For-Sale Unstable CA1 15 46 NC(=O)c1ccccc1NC(=O)NCCc1ccc(F)cc1 ZINC000217528939 DE For-Sale Unstable CCR3 31 45 NC(=O)c1ccccc1NC(=O)NCCc1ccc(F)cc1 ZINC000217528939 DE For-Sale Unstable CA12 16 46 NC(=O)c1ccccc1NC(=O)NCCc1ccc(F)cc1 ZINC000217528939 DE For-Sale Unstable CA9 15 43 NC(=O)c1ccccc1NC(=O)NCCc1ccc(F)cc1 ZINC000217528939 DE For-Sale Unstable HCAR2 15 41 NC(=O)c1ccccc1NC(=O)NCCc1ccc(F)cc1 ZINC000217528939 DE For-Sale Unstable PAGA 0 45 O=C(Cc1cn(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)c2ccccc12)N1CCCCCC1 ZINC000217528950 JH In-Stock Unstable CHRNA4 31 49 O=C(Cc1cn(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)c2ccccc12)N1CCCCCC1 ZINC000217528950 JH In-Stock Unstable PLK1 0 41 C[C@H](C(N)=O)N1CCC[C@@H](N)C1 ZINC000217528955 AB On-Demand Unstable XPNPEP1 54 31 C[C@H](C(N)=O)N1CCC[C@@H](N)C1 ZINC000217528955 AB On-Demand Unstable XPNPEP2 53 31 CC[C@H](N[C@H]1C[C@@H](C)CC[C@@H]1C(C)C)c1cccc(Br)c1 ZINC000217528975 FK For-Sale Unstable TRPM8 15 42 CCCCNc1ccc(C(=O)O)cc1S(=O)(=O)N[C@H](C)COC ZINC000217528978 ED In-Stock Unstable PLA2G4B 41 34 N#Cc1ccccc1N1CCC[C@@H]2CCCC[C@H]21 ZINC000217528991 BH For-Sale Unstable AR 15 47 c1ccc(Cn2nnnc2C[C@@H]2CCCN2)cc1 ZINC000217529004 BD For-Sale Unstable CHRNA10 29 41 O=C1OC2(CCN(C(=O)Cn3cccc3)CC2)c2ccccc21 ZINC000217529035 DE For-Sale Unstable NPY5R 46 51 CCOc1ccc(CCNC(=O)NCCc2ccc(F)cc2)cc1OCC ZINC000217529068 FH On-Demand Unstable CNR2 34 44 N#Cc1ccccc1N1CCC[C@H]2CCCC[C@H]21 ZINC000217529079 BH For-Sale Unstable AR 15 47 c1ccc(Cn2nnnc2C[C@H]2CCCN2)cc1 ZINC000217529091 BD For-Sale Unstable CHRNA10 29 41 CCCCCCC[C@@H](C)N[C@@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217529093 CK For-Sale Unstable ADH1B 0 40 CCCCCCC[C@@H](C)N[C@@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217529093 CK For-Sale Unstable ADH1C 0 40 O=C1C[C@H]2c3ccccc3[C@@H]1[C@H]1C(=O)N(c3ccc(Cl)c(Cl)c3)C(=O)[C@@H]21 ZINC000217529105 GH In-Stock Unstable BCL2A1 44 34 O=C1OC2(CCN(C(=O)c3cncc(Br)c3)CC2)c2ccccc21 ZINC000217529153 GG For-Sale Unstable AVPR1A 18 49 O=C1OC2(CCN(C(=O)c3cncc(Br)c3)CC2)c2ccccc21 ZINC000217529153 GG For-Sale Unstable NPY5R 51 52 Cc1ccc(CN2C(=O)/C(=C/N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)SC2=S)cc1 ZINC000217529159 IG In-Stock Unstable CHRNA4 28 52 O=C(Cc1ccc(-c2ccccc2)cc1)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217529162 IJ For-Sale Unstable FABP4 44 36 CCCCCCC[C@H](C)N[C@@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217529174 CK For-Sale Unstable ADH1B 0 40 CCCCCCC[C@H](C)N[C@@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217529174 CK For-Sale Unstable ADH1C 0 40 CC(C)CN1C(=O)/C(=C/N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)SC1=S ZINC000217529241 GF In-Stock Unstable CHRNA4 27 44 CCCCCCC[C@@H](C)N[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217529245 CK For-Sale Unstable ADH1B 0 40 CCCCCCC[C@@H](C)N[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217529245 CK For-Sale Unstable ADH1C 0 40 O=C1OC2(CCN(C(=O)Cn3cnnn3)CC2)c2ccccc21 ZINC000217529255 DC For-Sale Unstable NPY5R 42 48 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)C(c1ccccc1)c1ccccc1 ZINC000217529271 IJ For-Sale Unstable FABP4 49 38 COC(CNC(=O)NCCc1ccc(F)cc1)OC ZINC000217529298 CD For-Sale Unstable LEF 48 41 CCCCCCC[C@H](C)N[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217529322 CK For-Sale Unstable ADH1B 0 40 CCCCCCC[C@H](C)N[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217529322 CK For-Sale Unstable ADH1C 0 40 O=C1OC2(CCN(C(=O)c3cc(Br)ccc3Cl)CC2)c2ccccc21 ZINC000217529358 HI For-Sale Unstable AVPR1A 25 60 O=C1OC2(CCN(C(=O)c3cc(Br)ccc3Cl)CC2)c2ccccc21 ZINC000217529358 HI For-Sale Unstable NPY5R 40 52 CC(C)CCN1C(=O)/C(=C/N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)SC1=S ZINC000217529364 HG In-Stock Unstable CHRNA4 36 45 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccccc1Oc1ccccc1 ZINC000217529382 IK For-Sale Unstable FABP4 46 35 O=C(NCCc1ccc(F)cc1)Nc1ccc2cn[nH]c2c1 ZINC000217529398 CG For-Sale Unstable CCR3 39 40 O=C(NCCc1ccc(F)cc1)Nc1ccc2cn[nH]c2c1 ZINC000217529398 CG For-Sale Unstable ROCK1 16 67 O=C(NCCc1ccc(F)cc1)Nc1ccc2cn[nH]c2c1 ZINC000217529398 CG For-Sale Unstable RAF1 42 44 O=C(NCCc1ccc(F)cc1)Nc1ccc2cn[nH]c2c1 ZINC000217529398 CG For-Sale Unstable Q8MMZ8_EIMTE 29 44 O=C(NCCc1ccc(F)cc1)Nc1ccc2cn[nH]c2c1 ZINC000217529398 CG For-Sale Unstable PHLPP2 0 50 CC(C)CC(CC(C)C)N[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217529462 CK For-Sale Unstable TRPM8 15 40 O=C1OC2(CCN(C(=O)CCCCc3ccccc3)CC2)c2ccccc21 ZINC000217529463 FI For-Sale Unstable GHRHR 42 34 O=C1OC2(CCN(C(=O)CCCCc3ccccc3)CC2)c2ccccc21 ZINC000217529463 FI For-Sale Unstable SIGMAR1 29 59 O=C1OC2(CCN(C(=O)CCCCc3ccccc3)CC2)c2ccccc21 ZINC000217529463 FI For-Sale Unstable PREP 39 40 O=C1OC2(CCN(C(=O)CCCCc3ccccc3)CC2)c2ccccc21 ZINC000217529463 FI For-Sale Unstable FAAH 56 38 O=C1OC2(CCN(C(=O)CCCCc3ccccc3)CC2)c2ccccc21 ZINC000217529463 FI For-Sale Unstable NPY5R 44 52 O=C1OC2(CCN(C(=O)CCCCc3ccccc3)CC2)c2ccccc21 ZINC000217529463 FI For-Sale Unstable CES1 57 37 CC(C)(C)c1ccc(C(=O)NCC[C@H](O)c2ccsc2)cc1 ZINC000217529479 DH In-Stock Unstable CYNT 25 41 O=C(CCc1cn(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)c2ccccc12)N1CCOCC1 ZINC000217529503 JF In-Stock Unstable CHRNA4 29 46 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc(Oc2ccccc2)cc1 ZINC000217529504 IK For-Sale Unstable DRD4 41 32 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc(Oc2ccccc2)cc1 ZINC000217529504 IK For-Sale Unstable GCGR 40 39 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc(Oc2ccccc2)cc1 ZINC000217529504 IK For-Sale Unstable GIPR 45 35 O=C(NCCc1ccc(F)cc1)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217529506 GK For-Sale Unstable TACR1 21 45 O=C(NCCc1ccc(F)cc1)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217529506 GK For-Sale Unstable CCR3 46 49 O=C(NCCc1ccc(F)cc1)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217529506 GK For-Sale Unstable RAF1 40 49 O=C(NCCc1ccc(F)cc1)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217529506 GK For-Sale Unstable EPHX2 21 40 O=C(NCCc1ccc(F)cc1)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217529506 GK For-Sale Unstable Q8MMZ8_EIMTE 29 49 O=C(NCCc1ccc(F)cc1)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217529506 GK For-Sale Unstable PTPA 0 45 CC(=O)N/N=C/c1ccc(Cl)nc1 ZINC000217529544 AD For-Sale Unstable UREA_CANEN 17 40 CC(C)CC(CC(C)C)N[C@H]1C[C@H](C)CC[C@@H]1C(C)C ZINC000217529550 CK For-Sale Unstable TRPM8 15 40 CC(C)(C)c1ccc(C(=O)NCC[C@@H](O)c2ccsc2)cc1 ZINC000217529556 DH In-Stock Unstable CYNT 25 41 O=[N+]([O-])c1ccc(CNc2cc(F)cc(Cl)c2)cc1 ZINC000217529558 CH On-Demand Unstable EPAS1 19 40 COc1ccc(/C=C/C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1OC ZINC000217529584 GG For-Sale Unstable ITGAL 24 44 COc1ccc(/C=C/C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1OC ZINC000217529584 GG For-Sale Unstable NPY5R 34 53 Nc1ccc(C(=O)NC(=O)NCCc2ccc(F)cc2)cc1 ZINC000217529615 DE For-Sale Unstable CYNT 18 40 Nc1ccc(C(=O)NC(=O)NCCc2ccc(F)cc2)cc1 ZINC000217529615 DE For-Sale Unstable A6YCJ1_9METZ 17 46 O=C1OC2(CCN(C(=O)c3ccc4n[nH]nc4c3)CC2)c2ccccc21 ZINC000217529686 EE For-Sale Unstable AVPR1A 15 52 O=C1OC2(CCN(C(=O)c3ccc4n[nH]nc4c3)CC2)c2ccccc21 ZINC000217529686 EE For-Sale Unstable ACACA 79 39 O=C1OC2(CCN(C(=O)c3ccc4n[nH]nc4c3)CC2)c2ccccc21 ZINC000217529686 EE For-Sale Unstable ACACB 54 38 O=C1OC2(CCN(C(=O)c3ccc4n[nH]nc4c3)CC2)c2ccccc21 ZINC000217529686 EE For-Sale Unstable NPY5R 50 52 CCN(CC)c1ccc(NC(=O)NCCc2ccc(F)cc2)cc1 ZINC000217529741 EI For-Sale Unstable CCR3 51 42 CCOCCCN1C(=O)/C(=C/N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)SC1=S ZINC000217529777 HE In-Stock Unstable CHRNA4 27 42 O=C1OC2(CCN(C(=O)Cn3ccc4ccccc43)CC2)c2ccccc21 ZINC000217529788 FG For-Sale Unstable NPY5R 39 51 O=C(NCC[C@H](O)c1ccsc1)c1nc2ccccc2s1 ZINC000217529845 DG In-Stock Unstable ST14 41 36 O=C(NCC[C@H](O)c1ccsc1)c1nc2ccccc2s1 ZINC000217529845 DG In-Stock Unstable TMPRSS6 67 35 Cc1noc(C)c1CC(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217529903 EF In-Stock Unstable NPY5R 41 46 O=C(NCC[C@@H](O)c1ccsc1)c1nc2ccccc2s1 ZINC000217529933 DG In-Stock Unstable ST14 41 36 O=C(NCC[C@@H](O)c1ccsc1)c1nc2ccccc2s1 ZINC000217529933 DG In-Stock Unstable TMPRSS6 67 35 CC(C)CN(CC(C)C)C(=O)NCCc1ccc(F)cc1 ZINC000217529972 CH On-Demand Unstable LEF 42 35 CC(C)NC[C@@H](O)c1ncccc1Br ZINC000217529981 CD In-Stock Unstable ADRB2 24 49 Cc1noc(C)c1C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217530014 EF In-Stock Unstable AVPR1A 15 48 Cc1noc(C)c1C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217530014 EF In-Stock Unstable NPY5R 46 50 CC(C)NC[C@H](O)c1ncccc1Br ZINC000217530069 CD In-Stock Unstable ADRB2 24 49 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1N[C@@H](C)c1ccsc1 ZINC000217530088 CJ For-Sale Unstable TRPM8 15 42 O=CN1CCN(C(=O)NCCc2ccc(F)cc2)CC1 ZINC000217530092 CC For-Sale Unstable CCR3 17 43 O=CN1CCN(C(=O)NCCc2ccc(F)cc2)CC1 ZINC000217530092 CC For-Sale Unstable NPSR1 23 40 COc1cccc2cc(C(=O)NCCn3nc(C(F)(F)F)c4c3CCCC4)c(=O)oc12 ZINC000217530124 IG For-Sale Unstable DRD3 21 41 CC(=O)N1CCC(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)CC1 ZINC000217530127 FD For-Sale Unstable NPY5R 61 51 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1N[C@@H](C)c1ccsc1 ZINC000217530162 CJ For-Sale Unstable TRPM8 15 42 C[C@H](C(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)c1ccc2c(c1)[nH]c1ccc(Cl)cc12 ZINC000217530173 IJ In-Stock Unstable CHRNA4 31 41 CC(C)(C)NC[C@@H](O)c1ncccc1Br ZINC000217530176 CE In-Stock Unstable ADRB2 33 44 CC(C)(C)NC[C@@H](O)c1ncccc1Br ZINC000217530176 CE In-Stock Unstable ADRB1 0 43 O=C1OC2(CCN(C(=O)CCn3cnc4ccccc4c3=O)CC2)c2ccccc21 ZINC000217530236 HE For-Sale Unstable NPY5R 40 46 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1N[C@@H](C)c1ccsc1 ZINC000217530244 CJ For-Sale Unstable TRPM8 15 42 COc1ccc(Cl)cc1C(=O)NCCSc1nccn1C ZINC000217530252 EF In-Stock Unstable F10 52 37 COc1ccc(Cl)cc1C(=O)NCCSc1nccn1C ZINC000217530252 EF In-Stock Unstable COLA 41 33 C[C@@H](C(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)c1ccc2c(c1)[nH]c1ccc(Cl)cc12 ZINC000217530253 IJ In-Stock Unstable CHRNA4 31 41 CC(C)(C)NC[C@H](O)c1ncccc1Br ZINC000217530270 CE In-Stock Unstable ADRB2 33 44 CC(C)(C)NC[C@H](O)c1ncccc1Br ZINC000217530270 CE In-Stock Unstable ADRB1 0 43 CC(C)[C@H]1CC[C@H](C)C[C@@H]1N[C@@H](C)c1ccsc1 ZINC000217530315 CJ For-Sale Unstable TRPM8 15 42 COC[C@@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1NC1CCCCC1 ZINC000217530355 FE In-Stock Unstable AMY2 44 30 O=C1OC2(CCN(C(=O)Cn3cncn3)CC2)c2ccccc21 ZINC000217530361 DC For-Sale Unstable NPY5R 45 48 O=C(CNc1cc(F)cc(Cl)c1)Nc1ccc(F)cc1 ZINC000217530378 CH On-Demand Unstable IMDH_CRYPV 27 43 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1N[C@@H](C)c1cc(Cl)ccc1Cl ZINC000217530413 EK For-Sale Unstable TRPM8 17 55 COC[C@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1NC1CCCCC1 ZINC000217530429 FE In-Stock Unstable AMY2 44 30 C[C@@H]1Cc2ccccc2N1C(=O)NCCc1ccc(F)cc1 ZINC000217530448 CH On-Demand Unstable DRD4 32 57 C[C@@H]1Cc2ccccc2N1C(=O)NCCc1ccc(F)cc1 ZINC000217530448 CH On-Demand Unstable KCNQ2 15 40 C[C@@H]1Cc2ccccc2N1C(=O)NCCc1ccc(F)cc1 ZINC000217530448 CH On-Demand Unstable CCR3 18 41 C[C@@H]1Cc2ccccc2N1C(=O)NCCc1ccc(F)cc1 ZINC000217530448 CH On-Demand Unstable TPP2 58 38 O=Cc1cc(Br)ccc1Oc1ccc([N+](=O)[O-])cc1 ZINC000217530460 DH For-Sale Bother PPOX1 17 51 O=C1OC2(CCN(C(=O)CCCN3C(=O)c4ccccc4C3=O)CC2)c2ccccc21 ZINC000217530462 HF For-Sale Unstable NPY5R 41 48 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1N[C@@H](C)c1cc(Cl)ccc1Cl ZINC000217530493 EK For-Sale Unstable TRPM8 17 55 C[C@H]1Cc2ccccc2N1C(=O)NCCc1ccc(F)cc1 ZINC000217530531 CH On-Demand Unstable DRD4 32 57 C[C@H]1Cc2ccccc2N1C(=O)NCCc1ccc(F)cc1 ZINC000217530531 CH On-Demand Unstable KCNQ2 15 40 C[C@H]1Cc2ccccc2N1C(=O)NCCc1ccc(F)cc1 ZINC000217530531 CH On-Demand Unstable CCR3 18 41 C[C@H]1Cc2ccccc2N1C(=O)NCCc1ccc(F)cc1 ZINC000217530531 CH On-Demand Unstable TPP2 58 38 O=C1OC2(CCN(C(=O)CCN3C(=O)c4ccccc4C3=O)CC2)c2ccccc21 ZINC000217530548 HE For-Sale Unstable NPY5R 41 48 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1N[C@@H](C)c1cc(Cl)ccc1Cl ZINC000217530572 EK For-Sale Unstable TRPM8 17 55 O=Cc1cc(Br)ccc1Oc1ccc([N+](=O)[O-])cc1Cl ZINC000217530586 FJ For-Sale Bother SNCA 24 41 C[C@@H](Cc1cccnc1)NC(=O)c1ccc(N)nc1 ZINC000217530597 CD In-Stock Unstable TBXAS1 17 41 C[C@@H](Cc1cccnc1)NC(=O)c1ccc(N)nc1 ZINC000217530597 CD In-Stock Unstable PTAFR 28 43 C[C@@H](Cc1cccnc1)NC(=O)c1ccc(N)nc1 ZINC000217530597 CD In-Stock Unstable CPB2 23 41 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)C1c2ccccc2Oc2ccccc21 ZINC000217530635 IJ For-Sale Unstable GRM1 16 41 CC(C)[C@H]1CC[C@H](C)C[C@@H]1N[C@@H](C)c1cc(Cl)ccc1Cl ZINC000217530651 EK For-Sale Unstable TRPM8 17 55 Cc1ccc2nc(-c3ccc(NC(=O)NCCc4ccc(F)cc4)cc3)sc2c1 ZINC000217530671 HK For-Sale Unstable LDHA 44 46 Cc1ccc2nc(-c3ccc(NC(=O)NCCc4ccc(F)cc4)cc3)sc2c1 ZINC000217530671 HK For-Sale Unstable CCR3 44 34 Cc1ccc2nc(-c3ccc(NC(=O)NCCc4ccc(F)cc4)cc3)sc2c1 ZINC000217530671 HK For-Sale Unstable APP 26 53 Cc1ccc2nc(-c3ccc(NC(=O)NCCc4ccc(F)cc4)cc3)sc2c1 ZINC000217530671 HK For-Sale Unstable RAF1 26 43 Cc1ccc2nc(-c3ccc(NC(=O)NCCc4ccc(F)cc4)cc3)sc2c1 ZINC000217530671 HK For-Sale Unstable Q8MMZ8_EIMTE 23 43 Cc1ccc2nc(-c3ccc(NC(=O)NCCc4ccc(F)cc4)cc3)sc2c1 ZINC000217530671 HK For-Sale Unstable LUCI_PHOPE 28 44 Cc1ccc2nc(-c3ccc(NC(=O)NCCc4ccc(F)cc4)cc3)sc2c1 ZINC000217530671 HK For-Sale Unstable PRMT3 65 40 Cc1ccc2nc(-c3ccc(NC(=O)NCCc4ccc(F)cc4)cc3)sc2c1 ZINC000217530671 HK For-Sale Unstable FABK 0 41 Cc1ccc2nc(-c3ccc(NC(=O)NCCc4ccc(F)cc4)cc3)sc2c1 ZINC000217530671 HK For-Sale Unstable PORCN 0 41 C[C@H](Cc1cccnc1)NC(=O)c1ccc(N)nc1 ZINC000217530678 CD In-Stock Unstable TBXAS1 17 41 C[C@H](Cc1cccnc1)NC(=O)c1ccc(N)nc1 ZINC000217530678 CD In-Stock Unstable PTAFR 28 43 C[C@H](Cc1cccnc1)NC(=O)c1ccc(N)nc1 ZINC000217530678 CD In-Stock Unstable CPB2 23 41 O=C1OC2(CCN(C(=O)C3CCCC3)CC2)c2ccccc21 ZINC000217530680 CF For-Sale Unstable NPY5R 62 53 O=C(NCCc1ccc(F)cc1)NC(=O)C1CCNCC1 ZINC000217530787 CD For-Sale Unstable CCR3 30 45 O=C(NCCc1ccc(F)cc1)NC(=O)C1CCNCC1 ZINC000217530787 CD For-Sale Unstable GPBAR1 32 40 O=C1OC2(CCN(C(=O)/C=C/c3ccccc3Cl)CC2)c2ccccc21 ZINC000217530795 FI For-Sale Unstable NPY5R 48 57 O=C(/C=C/c1ccccc1Cl)NCC[C@H](O)c1ccsc1 ZINC000217530823 DH In-Stock Unstable KCNQ2 39 40 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC1CCC(C(C)(C)C)CC1 ZINC000217530845 CK For-Sale Unstable TRPM8 0 40 CCO[C@@H]1C[C@@H](Nc2cc(Cl)nc(N)n2)C1(C)C ZINC000217530847 CE For-Sale Unstable AGPAT2 43 37 CCCN1CCC(NC(=O)NC(=O)/C=C\C(=O)O)CC1 ZINC000217530878 CC For-Sale Unstable EPHX2 22 40 C[C@@H](C(=O)N1CCCCC1)N1CCC[C@@H](N)C1 ZINC000217530902 BC On-Demand Unstable DPP7 42 30 O=C(/C=C/c1ccccc1Cl)NCC[C@@H](O)c1ccsc1 ZINC000217530913 DH In-Stock Unstable KCNQ2 39 40 Cc1ccc(NC(=O)NCCc2ccc(F)cc2)c(O)c1 ZINC000217530914 CG For-Sale Unstable RAF1 38 41 CC(C)(C)OC(=O)N1CCC[C@H](CNN)CC1 ZINC000217530922 BD For-Sale Unstable CACNA1I 41 33 CC(C)(C)OC(=O)N1CCC[C@H](CNN)CC1 ZINC000217530922 BD For-Sale Unstable GPR119 42 42 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC1CCC(C(C)(C)C)CC1 ZINC000217530937 CK For-Sale Unstable TRPM8 0 40 C[C@@H](CCN1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217530938 BF On-Demand Unstable SLC6A1 74 39 CCO[C@H]1C[C@@H](Nc2cc(Cl)nc(N)n2)C1(C)C ZINC000217530947 CE For-Sale Unstable AGPAT2 43 37 O=C1OC2(CCN(C(=O)Cc3c(F)cccc3Cl)CC2)c2ccccc21 ZINC000217530951 FH For-Sale Unstable NPY5R 43 51 C[C@H](C(=O)N1CCCCC1)N1CCC[C@@H](N)C1 ZINC000217530995 BC On-Demand Unstable DPP7 42 30 CC(C)(C)OC(=O)N1CCC[C@@H](CNN)CC1 ZINC000217531004 BD For-Sale Unstable CACNA1I 41 33 CC(C)(C)OC(=O)N1CCC[C@@H](CNN)CC1 ZINC000217531004 BD For-Sale Unstable GPR119 42 42 C[C@H](CCN1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217531016 BF On-Demand Unstable SLC6A1 74 39 O=C(NCC[C@H](O)c1ccsc1)c1cc(-c2ccccc2)on1 ZINC000217531027 EG In-Stock Unstable HDAC10 19 53 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC1CCC(C(C)(C)C)CC1 ZINC000217531034 CK For-Sale Unstable TRPM8 0 40 CCO[C@@H]1C[C@H](Nc2cc(Cl)nc(N)n2)C1(C)C ZINC000217531035 CE For-Sale Unstable AGPAT2 43 37 O=C(NCCc1ccc(F)cc1)Nc1ccc(Cl)cc1C(F)(F)F ZINC000217531042 FJ For-Sale Unstable TRPV1 23 50 O=C(NCCc1ccc(F)cc1)Nc1ccc(Cl)cc1C(F)(F)F ZINC000217531042 FJ For-Sale Unstable CCR3 19 47 O=C(NCCc1ccc(F)cc1)Nc1ccc(Cl)cc1C(F)(F)F ZINC000217531042 FJ For-Sale Unstable RAF1 42 43 O=C(NCCc1ccc(F)cc1)Nc1ccc(Cl)cc1C(F)(F)F ZINC000217531042 FJ For-Sale Unstable Q8MMZ8_EIMTE 31 43 COc1ccc(/C=C\C(=O)NC2CC(O)C2)cc1F ZINC000217531058 CD For-Sale Unstable MMP2 0 53 COc1ccc(/C=C\C(=O)NC2CC(O)C2)cc1F ZINC000217531058 CD For-Sale Unstable HDAC1 15 44 COc1ccc(/C=C\C(=O)NC2CC(O)C2)cc1F ZINC000217531058 CD For-Sale Unstable TUBB1 54 49 COc1ccc(/C=C\C(=O)NC2CC(O)C2)cc1F ZINC000217531058 CD For-Sale Unstable ABCG2 16 42 CCn1cc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c(=O)c2ccc(C)nc21 ZINC000217531062 HG For-Sale Unstable AVPR1A 18 49 CCn1cc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c(=O)c2ccc(C)nc21 ZINC000217531062 HG For-Sale Unstable NPY5R 30 43 O=C(NCC[C@@H](O)c1ccsc1)c1cc(-c2ccccc2)on1 ZINC000217531113 EG In-Stock Unstable HDAC10 19 53 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC1CCC(C(C)(C)C)CC1 ZINC000217531117 CK For-Sale Unstable TRPM8 0 40 CC(C)(C)OC(=O)N1CCC[C@H](CCNN)C1 ZINC000217531119 BD For-Sale Unstable GPR119 29 40 CCO[C@H]1C[C@H](Nc2cc(Cl)nc(N)n2)C1(C)C ZINC000217531124 CE For-Sale Unstable AGPAT2 43 37 Cc1cc(C)c(NC(=O)NCCc2ccc(F)cc2)c(Cl)c1 ZINC000217531148 DI On-Demand Unstable RAF1 36 42 Cc1cc(C)c(NC(=O)NCCc2ccc(F)cc2)c(Cl)c1 ZINC000217531148 DI On-Demand Unstable Q8MMZ8_EIMTE 23 42 Cc1cc(C)c(NC(=O)NCCc2ccc(F)cc2)c(Cl)c1 ZINC000217531148 DI On-Demand Unstable LEF 47 38 Cc1cc(C)c(NC(=O)NCCc2ccc(F)cc2)c(Cl)c1 ZINC000217531148 DI On-Demand Unstable ACAT 0 42 O=C1OC2(CCN(C(=O)c3ccc4noc(-c5ccccc5)c4c3)CC2)c2ccccc21 ZINC000217531156 HJ For-Sale Unstable AVPR1A 15 47 O=C1OC2(CCN(C(=O)c3ccc4noc(-c5ccccc5)c4c3)CC2)c2ccccc21 ZINC000217531156 HJ For-Sale Unstable NPY5R 48 52 CN1CCC(CN(C)c2cc(Cl)ccc2CBr)CC1 ZINC000217531160 EI For-Sale Unstable NOS2 16 49 CN1CCC(CN(C)c2cc(Cl)ccc2CBr)CC1 ZINC000217531160 EI For-Sale Unstable NOS3 19 49 COc1ccc(C(=O)NC2CCN(C(=O)N3CCOCC3)CC2)o1 ZINC000217531191 EC In-Stock Unstable PDK1 49 36 COc1ccc(C(=O)NC2CCN(C(=O)N3CCOCC3)CC2)o1 ZINC000217531191 EC In-Stock Unstable MCHR1 27 40 COc1ccc(C(=O)NC2CCN(C(=O)N3CCOCC3)CC2)o1 ZINC000217531191 EC In-Stock Unstable AKR1C3 30 40 CC(C)(C)OC(=O)N1CCC[C@@H](CCNN)C1 ZINC000217531193 BD For-Sale Unstable GPR119 29 40 COc1ccc(CN[C@H]2C[C@@H](C)CC[C@@H]2C(C)C)cc1F ZINC000217531239 CI For-Sale Unstable TRPM8 16 42 C[C@@H](C(=O)N1CCCCCC1)N1CCC[C@@H](N)C1 ZINC000217531242 CD On-Demand Unstable DPP7 42 30 O=C(NCCc1ccc(F)cc1)Nc1c(Cl)cccc1Cl ZINC000217531256 EI For-Sale Unstable NCE103 24 40 O=C(NCCc1ccc(F)cc1)Nc1c(Cl)cccc1Cl ZINC000217531256 EI For-Sale Unstable ACAT 0 49 O=C(NCCc1ccc(F)cc1)Nc1c(Cl)cccc1Cl ZINC000217531256 EI For-Sale Unstable CAN2 0 40 O=C1OC2(CCN(C(=O)Cn3cnc4ccccc43)CC2)c2ccccc21 ZINC000217531265 FF In-Stock Unstable NPY5R 46 50 CN1CCC(CN(C)c2ccc(Cl)cc2CBr)CC1 ZINC000217531282 EI For-Sale Unstable NOS2 19 52 CN1CCC(CN(C)c2ccc(Cl)cc2CBr)CC1 ZINC000217531282 EI For-Sale Unstable NOS3 22 52 Cc1ccc(/C=C\C(=O)NCC2CC(O)C2)cc1 ZINC000217531289 BD For-Sale Unstable HDAC8 33 40 Cc1ccc(/C=C\C(=O)NCC2CC(O)C2)cc1 ZINC000217531289 BD For-Sale Unstable HDAC1 28 44 Cc1ccc(/C=C\C(=O)NCC2CC(O)C2)cc1 ZINC000217531289 BD For-Sale Unstable HDAC4 23 44 Cc1ccc(/C=C\C(=O)NCC2CC(O)C2)cc1 ZINC000217531289 BD For-Sale Unstable HDAC6 23 41 Cc1ccc(/C=C\C(=O)NCC2CC(O)C2)cc1 ZINC000217531289 BD For-Sale Unstable IMA1 0 43 CC(C)(C)OC(=O)N1CCCCC[C@@H]1CNN ZINC000217531300 BD For-Sale Unstable PREP 15 48 C[C@H](C(=O)N1CCCCCC1)N1CCC[C@@H](N)C1 ZINC000217531329 CD On-Demand Unstable DPP7 42 30 COc1ccc(CN[C@H]2C[C@H](C)CC[C@@H]2C(C)C)cc1F ZINC000217531330 CI For-Sale Unstable TRPM8 16 42 COc1cccc(N2C[C@H](C(=O)NCCn3nc(C(F)(F)F)c4c3CCCC4)CC2=O)c1 ZINC000217531367 JF For-Sale Unstable DRD4 46 35 CCN(CC)c1ccc(NC(=O)NCCc2ccc(F)cc2)c(C)c1 ZINC000217531370 EI For-Sale Unstable LEF 40 36 CC[C@@H](NC(=O)Cc1ccc(O)c(Cl)c1)c1nc2cc(C)ccc2[nH]1 ZINC000217531373 FI In-Stock Unstable PRCP 15 42 CC[C@@H](NC(=O)Cc1ccc(O)c(Cl)c1)c1nc2cc(C)ccc2[nH]1 ZINC000217531373 FI In-Stock Unstable NCE103 29 47 CC[C@@H](NC(=O)Cc1ccc(O)c(Cl)c1)c1nc2cc(C)ccc2[nH]1 ZINC000217531373 FI In-Stock Unstable CAN2 0 47 CC(C)(C)OC(=O)N1CCCCC[C@H]1CNN ZINC000217531382 BD For-Sale Unstable PREP 15 48 COC(=O)c1ccccc1C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217531384 FF For-Sale Unstable AVPR1A 20 54 COC(=O)c1ccccc1C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217531384 FF For-Sale Unstable NPY5R 52 54 CN(C)c1ccc(/C=C\C(=O)NCC2CC(O)C2)cc1 ZINC000217531405 CD For-Sale Unstable HDAC8 24 41 CN(C)c1ccc(/C=C\C(=O)NCC2CC(O)C2)cc1 ZINC000217531405 CD For-Sale Unstable HDAC1 22 41 CN(C)c1ccc(/C=C\C(=O)NCC2CC(O)C2)cc1 ZINC000217531405 CD For-Sale Unstable IMA1 0 41 COc1cccc(N2C[C@@H](C(=O)NCCn3nc(C(F)(F)F)c4c3CCCC4)CC2=O)c1 ZINC000217531452 JF For-Sale Unstable DRD4 46 35 CC[C@H](NC(=O)Cc1ccc(O)c(Cl)c1)c1nc2cc(C)ccc2[nH]1 ZINC000217531455 FI In-Stock Unstable NCE103 29 47 CC[C@H](NC(=O)Cc1ccc(O)c(Cl)c1)c1nc2cc(C)ccc2[nH]1 ZINC000217531455 FI In-Stock Unstable CAN2 0 47 O=C1OC2(CCN(C(=O)c3cccc(F)c3)CC2)c2ccccc21 ZINC000217531502 EG For-Sale Unstable AVPR1A 15 52 O=C1OC2(CCN(C(=O)c3cccc(F)c3)CC2)c2ccccc21 ZINC000217531502 EG For-Sale Unstable INHA 23 52 O=C1OC2(CCN(C(=O)c3cccc(F)c3)CC2)c2ccccc21 ZINC000217531502 EG For-Sale Unstable NPY5R 53 60 COc1ccc(N2C[C@H](C(=O)NCCn3nc(C(F)(F)F)c4c3CCCC4)CC2=O)cc1 ZINC000217531562 JF For-Sale Unstable DRD4 40 31 COc1ccc(N2C[C@H](C(=O)NCCn3nc(C(F)(F)F)c4c3CCCC4)CC2=O)cc1 ZINC000217531562 JF For-Sale Unstable F10 32 40 O=C(NCCc1ccc(F)cc1)NC[C@@H]1COc2ccccc2O1 ZINC000217531607 EF On-Demand Unstable HTR1A 0 44 O=C1OC2(CCN(C(=O)CN3C(=O)c4ccccc4C3=O)CC2)c2ccccc21 ZINC000217531615 GD For-Sale Unstable NPY5R 46 49 COc1cccc2cc(C(=O)NCC[C@H](O)c3ccsc3)oc12 ZINC000217531621 EG In-Stock Unstable DRD3 15 47 COc1ccc(N2C[C@@H](C(=O)NCCn3nc(C(F)(F)F)c4c3CCCC4)CC2=O)cc1 ZINC000217531653 JF For-Sale Unstable DRD4 40 31 COc1ccc(N2C[C@@H](C(=O)NCCn3nc(C(F)(F)F)c4c3CCCC4)CC2=O)cc1 ZINC000217531653 JF For-Sale Unstable F10 32 40 O=C(NCCc1ccc(F)cc1)NC[C@H]1COc2ccccc2O1 ZINC000217531698 EF On-Demand Unstable HTR1A 0 44 COc1cccc2cc(C(=O)NCC[C@@H](O)c3ccsc3)oc12 ZINC000217531702 EG In-Stock Unstable DRD3 15 47 O=C1OC2(CCN(C(=O)Cc3noc4ccccc34)CC2)c2ccccc21 ZINC000217531724 FG For-Sale Unstable NPY5R 40 45 COC[C@@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1N[C@@H](C)c1ccccc1 ZINC000217531740 GF In-Stock Unstable LDHB 0 41 Cc1cc(NC(=O)NCCc2ccc(F)cc2)ccc1Br ZINC000217531802 FI For-Sale Unstable CCR3 56 39 Cc1cc(NC(=O)NCCc2ccc(F)cc2)ccc1Br ZINC000217531802 FI For-Sale Unstable RAF1 39 45 Cc1cc(NC(=O)NCCc2ccc(F)cc2)ccc1Br ZINC000217531802 FI For-Sale Unstable CA12 16 44 Cc1cc(NC(=O)NCCc2ccc(F)cc2)ccc1Br ZINC000217531802 FI For-Sale Unstable LEF 92 42 COc1ccc(CC(=O)NCC[C@H](O)c2ccsc2)cc1OC ZINC000217531807 EF In-Stock Unstable TRPV1 23 43 COc1ccc(CC(=O)NCC[C@H](O)c2ccsc2)cc1OC ZINC000217531807 EF In-Stock Unstable NCE103 17 48 COc1ccc(CC(=O)NCC[C@H](O)c2ccsc2)cc1OC ZINC000217531807 EF In-Stock Unstable CAN2 0 48 COC[C@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1N[C@@H](C)c1ccccc1 ZINC000217531818 GF In-Stock Unstable LDHB 0 41 O=C(NCC(=O)N1CCC2(CC1)OC(=O)c1ccccc12)c1ccccc1 ZINC000217531846 FE For-Sale Unstable NPY5R 48 53 Cc1onc(-c2ccccc2Cl)c1C(=O)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217531879 JJ For-Sale Unstable GPBAR1 36 47 COc1ccc(CC(=O)NCC[C@@H](O)c2ccsc2)cc1OC ZINC000217531890 EF In-Stock Unstable TRPV1 23 43 COc1ccc(CC(=O)NCC[C@@H](O)c2ccsc2)cc1OC ZINC000217531890 EF In-Stock Unstable NCE103 17 48 COc1ccc(CC(=O)NCC[C@@H](O)c2ccsc2)cc1OC ZINC000217531890 EF In-Stock Unstable CAN2 0 48 COC[C@@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1N[C@H](C)c1ccccc1 ZINC000217531904 GF In-Stock Unstable LDHB 0 41 Cc1cc(C)cc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217531954 EH For-Sale Unstable AVPR1A 16 53 Cc1cc(C)cc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217531954 EH For-Sale Unstable INHA 19 40 Cc1cc(C)cc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217531954 EH For-Sale Unstable ACACA 63 36 Cc1cc(C)cc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217531954 EH For-Sale Unstable ACACB 42 35 Cc1cc(C)cc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217531954 EH For-Sale Unstable NPY5R 50 51 COC[C@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1N[C@H](C)c1ccccc1 ZINC000217531987 GF In-Stock Unstable LDHB 0 41 O=C(NCC[C@H](O)c1ccsc1)c1ccc(-c2ccccc2)cc1 ZINC000217532004 EI In-Stock Unstable EPHX2 0 44 O=C(NCC[C@@H](O)c1ccsc1)c1ccc(-c2ccccc2)cc1 ZINC000217532089 EI In-Stock Unstable EPHX2 0 44 CC(C)CC(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217532093 CF For-Sale Unstable NPY5R 46 51 COc1cc(/C=C/C(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc(OC)c1OC ZINC000217532100 JH For-Sale Unstable BCHE 22 41 O=C(NC1CCN(Cc2ccccc2)CC1)c1ccnn1-c1ccccc1 ZINC000217532134 FG On-Demand Unstable CHRM2 18 42 O=C(NC1CCN(Cc2ccccc2)CC1)c1ccnn1-c1ccccc1 ZINC000217532134 FG On-Demand Unstable DRD2 20 57 O=C(NC1CCN(Cc2ccccc2)CC1)c1ccnn1-c1ccccc1 ZINC000217532134 FG On-Demand Unstable DRD4 47 50 O=C(NC1CCN(Cc2ccccc2)CC1)c1ccnn1-c1ccccc1 ZINC000217532134 FG On-Demand Unstable ACHE 40 52 O=C(NC1CCN(Cc2ccccc2)CC1)c1ccnn1-c1ccccc1 ZINC000217532134 FG On-Demand Unstable HRH1 19 40 O=C(NC1CCN(Cc2ccccc2)CC1)c1ccnn1-c1ccccc1 ZINC000217532134 FG On-Demand Unstable DRD3 24 54 O=C(NC1CCN(Cc2ccccc2)CC1)c1ccnn1-c1ccccc1 ZINC000217532134 FG On-Demand Unstable KCNH2 15 41 O=C(NC1CCN(Cc2ccccc2)CC1)c1ccnn1-c1ccccc1 ZINC000217532134 FG On-Demand Unstable CHRM3 22 44 O=C(NC1CCN(Cc2ccccc2)CC1)c1ccnn1-c1ccccc1 ZINC000217532134 FG On-Demand Unstable LTA4H 22 40 O=C(NC1CCN(Cc2ccccc2)CC1)c1ccnn1-c1ccccc1 ZINC000217532134 FG On-Demand Unstable SIGMAR1 64 58 O=C(NC1CCN(Cc2ccccc2)CC1)c1ccnn1-c1ccccc1 ZINC000217532134 FG On-Demand Unstable SSTR5 53 38 O=C(NC1CCN(Cc2ccccc2)CC1)c1ccnn1-c1ccccc1 ZINC000217532134 FG On-Demand Unstable BCHE 17 40 O=C(NC1CCN(Cc2ccccc2)CC1)c1ccnn1-c1ccccc1 ZINC000217532134 FG On-Demand Unstable CCR3 39 45 O=C(NC1CCN(Cc2ccccc2)CC1)c1ccnn1-c1ccccc1 ZINC000217532134 FG On-Demand Unstable UTS2R 15 41 O=C(NC1CCN(Cc2ccccc2)CC1)c1ccnn1-c1ccccc1 ZINC000217532134 FG On-Demand Unstable FAAH 17 41 O=C(NC1CCN(Cc2ccccc2)CC1)c1ccnn1-c1ccccc1 ZINC000217532134 FG On-Demand Unstable SLC6A5 25 46 O=C(NC1CCN(Cc2ccccc2)CC1)c1ccnn1-c1ccccc1 ZINC000217532134 FG On-Demand Unstable PDK1 49 42 O=C(NC1CCN(Cc2ccccc2)CC1)c1ccnn1-c1ccccc1 ZINC000217532134 FG On-Demand Unstable MCHR1 50 49 O=C(NC1CCN(Cc2ccccc2)CC1)c1ccnn1-c1ccccc1 ZINC000217532134 FG On-Demand Unstable CACNA1G 17 44 O=C(NC1CCN(Cc2ccccc2)CC1)c1ccnn1-c1ccccc1 ZINC000217532134 FG On-Demand Unstable NPFFR1 44 33 O=C(O)/C=C\C(=O)NC(=O)Nc1nc2c(s1)CCCC2 ZINC000217532144 CD For-Sale Unstable SLC27A1 33 45 N[C@@H]1CCCN([C@@H]2CCC[C@@H]2O)C1 ZINC000217532197 AC For-Sale Unstable MAN2B1 0 42 N[C@@H]1CCCN([C@@H]2CCC[C@@H]2O)C1 ZINC000217532197 AC For-Sale Unstable MAN2C1 0 42 N[C@@H]1CCCN([C@@H]2CCC[C@@H]2O)C1 ZINC000217532197 AC For-Sale Unstable ALPHA-MAN-IA 0 42 O=C1OC2(CCN(C(=O)c3ccc(Cl)cc3Cl)CC2)c2ccccc21 ZINC000217532210 GI For-Sale Unstable AVPR1A 28 70 O=C1OC2(CCN(C(=O)c3ccc(Cl)cc3Cl)CC2)c2ccccc21 ZINC000217532210 GI For-Sale Unstable NPY5R 44 53 COc1ccc(-c2coc3cc(OCC(=O)N4C[C@@H]5C[C@H](C4)c4cccc(=O)n4C5)ccc3c2=O)cc1 ZINC000217532230 JH In-Stock Unstable ALDH2 110 47 COc1ccc(-c2coc3cc(OCC(=O)N4C[C@@H]5C[C@H](C4)c4cccc(=O)n4C5)ccc3c2=O)cc1 ZINC000217532230 JH In-Stock Unstable IL2 27 43 COc1ccc(-c2coc3cc(OCC(=O)N4C[C@@H]5C[C@H](C4)c4cccc(=O)n4C5)ccc3c2=O)cc1 ZINC000217532230 JH In-Stock Unstable CHRNA4 24 41 COC[C@@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)cc1 ZINC000217532273 HE In-Stock Unstable MMP13 25 40 COC[C@@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)cc1 ZINC000217532273 HE In-Stock Unstable MMP2 19 40 COC[C@@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)cc1 ZINC000217532273 HE In-Stock Unstable MMP9 17 40 COC[C@@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)cc1 ZINC000217532273 HE In-Stock Unstable AKR1C3 20 40 CC[C@@H](C)c1ccccc1NC(=O)NCCc1ccc(F)cc1 ZINC000217532275 DJ For-Sale Unstable CCR3 34 44 CC[C@@H](C)c1ccccc1NC(=O)NCCc1ccc(F)cc1 ZINC000217532275 DJ For-Sale Unstable ACAT 0 51 CC[C@@H](C)c1ccccc1NC(=O)NCCc1ccc(F)cc1 ZINC000217532275 DJ For-Sale Unstable AO-ACHE 0 42 N[C@@H]1CCCN([C@@H]2CCCC[C@@H]2O)C1 ZINC000217532317 AC For-Sale Unstable VACHT_TETCF 0 42 N[C@@H]1CCCN([C@@H]2CCCC[C@@H]2O)C1 ZINC000217532317 AC For-Sale Unstable MAN2B1 0 42 N[C@@H]1CCCN([C@@H]2CCCC[C@@H]2O)C1 ZINC000217532317 AC For-Sale Unstable MAN2C1 0 42 N[C@@H]1CCCN([C@@H]2CCCC[C@@H]2O)C1 ZINC000217532317 AC For-Sale Unstable ALPHA-MAN-IA 0 42 Cc1cccc(NC(=O)CNc2cc(F)cc(Cl)c2)c1 ZINC000217532324 CH On-Demand Unstable F12 0 40 Cc1cccc(NC(=O)CNc2cc(F)cc(Cl)c2)c1 ZINC000217532324 CH On-Demand Unstable SCN10A 18 40 Cc1cccc(NC(=O)CNc2cc(F)cc(Cl)c2)c1 ZINC000217532324 CH On-Demand Unstable PSBA 0 43 Cc1cccc(NC(=O)CNc2cc(F)cc(Cl)c2)c1 ZINC000217532324 CH On-Demand Unstable KCNK3 61 44 Cc1cccc(NC(=O)CNc2cc(F)cc(Cl)c2)c1 ZINC000217532324 CH On-Demand Unstable KCNK9 47 44 O=C1OC2(CCN(C(=O)CSC3CCCC3)CC2)c2ccccc21 ZINC000217532338 EG In-Stock Unstable NPY5R 51 46 COC[C@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)cc1 ZINC000217532347 HE In-Stock Unstable MMP13 25 40 COC[C@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)cc1 ZINC000217532347 HE In-Stock Unstable MMP2 19 40 COC[C@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)cc1 ZINC000217532347 HE In-Stock Unstable MMP9 17 40 COC[C@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)cc1 ZINC000217532347 HE In-Stock Unstable AKR1C3 20 40 CC[C@H](C)c1ccccc1NC(=O)NCCc1ccc(F)cc1 ZINC000217532355 DJ For-Sale Unstable CCR3 34 44 CC[C@H](C)c1ccccc1NC(=O)NCCc1ccc(F)cc1 ZINC000217532355 DJ For-Sale Unstable ACAT 0 51 CC[C@H](C)c1ccccc1NC(=O)NCCc1ccc(F)cc1 ZINC000217532355 DJ For-Sale Unstable AO-ACHE 0 42 CC(=O)Nc1cc(B(O)O)ccc1C ZINC000217532390 AB For-Sale Unstable LDLR 41 33 Cn1cc(/C=C(\NC(=O)c2ccccc2)C(=O)N2C[C@@H]3C[C@H](C2)Cn2c3cccc2=O)c2ccccc21 ZINC000217532424 JH In-Stock Unstable CHRNA4 27 47 COC[C@@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)c(OC)c1 ZINC000217532452 JE In-Stock Unstable PTGDR 19 44 O=C1OC2(CCN(C(=O)CC3CCCCC3)CC2)c2ccccc21 ZINC000217532456 EH For-Sale Unstable NPY5R 55 48 O=C(NCCc1ccc(F)cc1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217532464 GF For-Sale Unstable DRD4 15 43 O=C(NCCc1ccc(F)cc1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217532464 GF For-Sale Unstable KCNH2 18 49 O=C(NCCc1ccc(F)cc1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217532464 GF For-Sale Unstable SIGMAR1 15 65 O=C(NCCc1ccc(F)cc1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217532464 GF For-Sale Unstable CCR3 33 40 O=C(NCCc1ccc(F)cc1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217532464 GF For-Sale Unstable NOS2 92 38 O=C(NCCc1ccc(F)cc1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217532464 GF For-Sale Unstable MLNR 58 39 O=C(NCCc1ccc(F)cc1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217532464 GF For-Sale Unstable SSTR3 50 38 O=C(NCCc1ccc(F)cc1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217532464 GF For-Sale Unstable MCHR1 41 49 COC[C@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1NCCc1ccc(OC)c(OC)c1 ZINC000217532526 JE In-Stock Unstable PTGDR 19 44 c1ccc(CN2CCC[C@@H]2[C@@H]2CO2)cc1 ZINC000217532528 BE In-Stock Unstable DRD2 0 48 c1ccc(CN2CCC[C@@H]2[C@@H]2CO2)cc1 ZINC000217532528 BE In-Stock Unstable SIGMAR1 47 45 c1ccc(CN2CCC[C@@H]2[C@@H]2CO2)cc1 ZINC000217532528 BE In-Stock Unstable SLC18A3 26 43 COc1cc([C@H](N)CO)ccc1Br ZINC000217532530 BD For-Sale Unstable N1L 0 43 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccccc1I ZINC000217532550 JH For-Sale Unstable FABP4 42 36 CCOc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1OCC ZINC000217532562 GH In-Stock Unstable ACACA 45 35 CCOc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1OCC ZINC000217532562 GH In-Stock Unstable NPY5R 43 49 CCOc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1OCC ZINC000217532562 GH In-Stock Unstable HCN1 48 32 CCOc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1OCC ZINC000217532562 GH In-Stock Unstable HCN4 41 32 Cc1ccc(N)c(NC(=O)NCCc2ccc(F)cc2)c1 ZINC000217532574 CG For-Sale Unstable RAF1 38 43 COc1cc([C@@H](N)CO)ccc1Br ZINC000217532600 BD For-Sale Unstable N1L 0 43 c1ccc(CN2CCC[C@H]2[C@@H]2CO2)cc1 ZINC000217532607 BE In-Stock Unstable DRD2 0 48 c1ccc(CN2CCC[C@H]2[C@@H]2CO2)cc1 ZINC000217532607 BE In-Stock Unstable SIGMAR1 47 45 c1ccc(CN2CCC[C@H]2[C@@H]2CO2)cc1 ZINC000217532607 BE In-Stock Unstable SLC18A3 26 43 NC[C@@H]1CCCN(C(=O)/C=C\c2ccccc2)C1 ZINC000217532667 BD On-Demand Unstable CCR2 44 37 NC[C@@H]1CCCN(C(=O)/C=C\c2ccccc2)C1 ZINC000217532667 BD On-Demand Unstable GPR183 0 43 Cc1cnc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cn1 ZINC000217532673 DE In-Stock Unstable AVPR1A 22 51 Cc1cnc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cn1 ZINC000217532673 DE In-Stock Unstable NPY5R 58 53 Cc1cnc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cn1 ZINC000217532673 DE In-Stock Unstable CCR8 18 40 Cc1ccc(NC(=O)NCCc2ccc(F)cc2)c(N)c1 ZINC000217532686 CG For-Sale Unstable CCR3 33 41 Cc1ccc(NC(=O)NCCc2ccc(F)cc2)c(N)c1 ZINC000217532686 CG For-Sale Unstable RAF1 38 41 Cc1ccc(NC(=O)NCCc2ccc(F)cc2)c(N)c1 ZINC000217532686 CG For-Sale Unstable LEF 42 36 O=C(NCCc1nc(-c2ccccc2)cs1)c1ccnnc1 ZINC000217532728 DF In-Stock Unstable GIPR 45 38 O=C(NCCc1nc(-c2ccccc2)cs1)c1ccnnc1 ZINC000217532728 DF In-Stock Unstable KDM4E 22 40 NC[C@H]1CCCN(C(=O)/C=C\c2ccccc2)C1 ZINC000217532745 BD On-Demand Unstable CCR2 44 37 NC[C@H]1CCCN(C(=O)/C=C\c2ccccc2)C1 ZINC000217532745 BD On-Demand Unstable GPR183 0 43 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217532763 JF For-Sale Unstable TGM2 36 43 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217532763 JF For-Sale Unstable NAMPT 50 46 COc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c(OC)c1OC ZINC000217532781 GG For-Sale Unstable AVPR1A 16 53 COc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c(OC)c1OC ZINC000217532781 GG For-Sale Unstable NPY5R 36 56 COC(=O)[C@H](CCSC)NC(=S)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217532801 GD In-Stock Unstable CHRNA4 27 45 O=C(NCCc1ccc(F)cc1)N1CCCC[C@H]1CCO ZINC000217532810 CE On-Demand Unstable HCRTR1 15 41 COC[C@@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1NC[C@@H]1CCCO1 ZINC000217532820 FD In-Stock Unstable TNK2 40 32 CCOC(=O)C[C@@H](C)c1ccc(O)cc1C ZINC000217532841 BF For-Sale Unstable CA7 17 44 CCOC(=O)C[C@@H](C)c1ccc(O)cc1C ZINC000217532841 BF For-Sale Unstable CA14 15 44 NC[C@@H]1CCCN(C(=O)/C=C\c2ccc3c(c2)OCO3)C1 ZINC000217532855 CD On-Demand Unstable SSTR3 97 33 NC[C@@H]1CCCN(C(=O)/C=C\c2ccc3c(c2)OCO3)C1 ZINC000217532855 CD On-Demand Unstable DYRK2 42 34 O=C1OC2(CCN(C(=O)CSc3nc4ccccc4o3)CC2)c2ccccc21 ZINC000217532884 GH For-Sale Unstable NPY5R 44 46 COC[C@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1NC[C@@H]1CCCO1 ZINC000217532898 FD In-Stock Unstable TNK2 40 32 O=C(NCCc1ccc(F)cc1)N1CCCC[C@@H]1CCO ZINC000217532899 CE On-Demand Unstable HCRTR1 15 41 CCOC(=O)C[C@H](C)c1ccc(O)cc1C ZINC000217532935 BF For-Sale Unstable CA7 17 44 CCOC(=O)C[C@H](C)c1ccc(O)cc1C ZINC000217532935 BF For-Sale Unstable CA14 15 44 NC[C@H]1CCCN(C(=O)/C=C\c2ccc3c(c2)OCO3)C1 ZINC000217532936 CD On-Demand Unstable ITGAL 20 40 NC[C@H]1CCCN(C(=O)/C=C\c2ccc3c(c2)OCO3)C1 ZINC000217532936 CD On-Demand Unstable SSTR3 97 33 NC[C@H]1CCCN(C(=O)/C=C\c2ccc3c(c2)OCO3)C1 ZINC000217532936 CD On-Demand Unstable DYRK2 42 34 COC[C@@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1NC[C@H]1CCCO1 ZINC000217532986 FD In-Stock Unstable TNK2 40 32 O=C1OC2(CCN(C(=O)c3ccc(Br)o3)CC2)c2ccccc21 ZINC000217533007 GG For-Sale Unstable NPY5R 41 50 O=C(CNc1cc(F)cc(Cl)c1)Nc1cccc(F)c1 ZINC000217533020 CH On-Demand Unstable PPIA 22 41 O=C(CNc1cc(F)cc(Cl)c1)Nc1cccc(F)c1 ZINC000217533020 CH On-Demand Unstable PSBA 0 45 O=C(CNc1cc(F)cc(Cl)c1)Nc1cccc(F)c1 ZINC000217533020 CH On-Demand Unstable KCNK3 38 41 O=C(CNc1cc(F)cc(Cl)c1)Nc1cccc(F)c1 ZINC000217533020 CH On-Demand Unstable KCNK9 19 41 COC[C@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1NC[C@H]1CCCO1 ZINC000217533056 FD In-Stock Unstable TNK2 40 32 Cc1ccc([C@@H](C)NC(=O)NC(=O)/C=C\C(=O)O)cc1 ZINC000217533065 CD For-Sale Unstable ACACA 52 37 Cc1c(O)ccc2c(CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)cc(=O)oc12 ZINC000217533072 GF In-Stock Unstable CHRNA4 31 51 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000217533081 JG For-Sale Unstable TGM2 32 43 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000217533081 JG For-Sale Unstable NAMPT 49 47 COc1ccc(/C=C\C(=O)N2CCC[C@@H](CN)C2)cc1 ZINC000217533097 CD On-Demand Unstable CCR2 0 46 COc1ccc(/C=C\C(=O)N2CCC[C@@H](CN)C2)cc1 ZINC000217533097 CD On-Demand Unstable GPR183 0 54 O=C1OC2(CCN(C(=O)c3cccc(Br)c3)CC2)c2ccccc21 ZINC000217533123 GH For-Sale Unstable AVPR1A 15 52 O=C1OC2(CCN(C(=O)c3cccc(Br)c3)CC2)c2ccccc21 ZINC000217533123 GH For-Sale Unstable NPY5R 43 49 O=C(/C=C\c1ccccc1F)NC1CC(O)C1 ZINC000217533163 BD For-Sale Unstable KCNQ2 51 38 Cc1ccc([C@H](C)NC(=O)NC(=O)/C=C\C(=O)O)cc1 ZINC000217533166 CD For-Sale Unstable ACACA 52 37 COc1ccc(/C=C\C(=O)N2CCC[C@H](CN)C2)cc1 ZINC000217533196 CD On-Demand Unstable CCR2 0 46 COc1ccc(/C=C\C(=O)N2CCC[C@H](CN)C2)cc1 ZINC000217533196 CD On-Demand Unstable GPR183 0 54 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc(S(=O)(=O)N2CCOCC2)cc1 ZINC000217533210 JE For-Sale Unstable TGM2 32 48 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc(S(=O)(=O)N2CCOCC2)cc1 ZINC000217533210 JE For-Sale Unstable NAMPT 43 46 O=C(O)[C@@H](c1c[nH]c2cc(Br)ccc12)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217533217 IG In-Stock Unstable CHRNA4 26 40 O=C1OC2(CCN(C(=O)c3ccc(Br)cc3)CC2)c2ccccc21 ZINC000217533219 GH For-Sale Unstable AVPR1A 15 52 O=C1OC2(CCN(C(=O)c3ccc(Br)cc3)CC2)c2ccccc21 ZINC000217533219 GH For-Sale Unstable NPY5R 45 52 COC(=O)c1ccc(CNC(=O)NCCc2ccc(F)cc2)cc1 ZINC000217533241 EF On-Demand Unstable LEF 46 38 CN[C@H](CN1CCCO[C@@H](C)C1)c1ccc2c(c1)OCO2 ZINC000217533247 CD For-Sale Unstable SSTR3 53 31 CC(C)c1ccc(/C=C\C(=O)NC2CC(O)C2)cc1 ZINC000217533277 CE For-Sale Unstable MMP2 16 44 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1cc(C2CC2)on1 ZINC000217533326 FG For-Sale Unstable S1PR3 17 42 Cc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c(C)c1 ZINC000217533337 EH For-Sale Unstable AVPR1A 23 56 Cc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c(C)c1 ZINC000217533337 EH For-Sale Unstable NPY5R 40 49 O=C(O)[C@@H](c1c[nH]c2ccc(OCc3ccccc3)cc12)N1C[C@@H]2C[C@H](C1)Cn1c2cccc1=O ZINC000217533340 JI In-Stock Unstable CHRNA4 33 44 O=C(NCCc1ccc(F)cc1)NCc1ccc(CO)cc1 ZINC000217533367 DE For-Sale Unstable Q76353_9HIV1 0 40 O=C(O)[C@H](c1c[nH]c2ccc(OCc3ccccc3)cc12)N1C[C@@H]2C[C@H](C1)Cn1c2cccc1=O ZINC000217533430 JI In-Stock Unstable CHRNA4 33 44 COc1ccc(OC)c(-c2cc(C(=O)NCCn3nc(C(F)(F)F)c4c3CCCC4)n(C)n2)c1 ZINC000217533451 JH For-Sale Unstable DRD4 42 33 Cc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1C ZINC000217533454 EH For-Sale Unstable AVPR1A 15 52 Cc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1C ZINC000217533454 EH For-Sale Unstable INHA 21 45 Cc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1C ZINC000217533454 EH For-Sale Unstable ACACA 80 43 Cc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1C ZINC000217533454 EH For-Sale Unstable ACACB 56 38 Cc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1C ZINC000217533454 EH For-Sale Unstable NPY5R 41 50 O=C(NCCc1ccc(F)cc1)NCCc1ccc(Br)cc1 ZINC000217533485 FH On-Demand Unstable LIG1 0 44 O=C(NCCc1ccc(F)cc1)NCCc1ccc(Br)cc1 ZINC000217533485 FH On-Demand Unstable Q76353_9HIV1 0 45 c1ccc(CN2CC[C@H]([C@@H]3CO3)C2)cc1 ZINC000217533529 BD In-Stock Unstable DRD2 23 49 c1ccc(CN2CC[C@H]([C@@H]3CO3)C2)cc1 ZINC000217533529 BD In-Stock Unstable DRD4 45 49 c1ccc(CN2CC[C@H]([C@@H]3CO3)C2)cc1 ZINC000217533529 BD In-Stock Unstable ACHE 35 43 c1ccc(CN2CC[C@H]([C@@H]3CO3)C2)cc1 ZINC000217533529 BD In-Stock Unstable DRD3 24 49 c1ccc(CN2CC[C@H]([C@@H]3CO3)C2)cc1 ZINC000217533529 BD In-Stock Unstable VACHT_TETCF 0 48 c1ccc(CN2CC[C@H]([C@@H]3CO3)C2)cc1 ZINC000217533529 BD In-Stock Unstable SIGMAR1 88 52 c1ccc(CN2CC[C@H]([C@@H]3CO3)C2)cc1 ZINC000217533529 BD In-Stock Unstable SLC18A3 22 45 O=C(O)[C@@H](c1c[nH]c2cc(Cl)ccc12)N1C[C@@H]2C[C@H](C1)Cn1c2cccc1=O ZINC000217533558 GG In-Stock Unstable CHRNA4 26 42 O=C1OC2(CCN(C(=O)c3ccc(I)cc3)CC2)c2ccccc21 ZINC000217533561 IH For-Sale Unstable AVPR1A 15 52 O=C1OC2(CCN(C(=O)c3ccc(I)cc3)CC2)c2ccccc21 ZINC000217533561 IH For-Sale Unstable NPY5R 46 52 Cc1ccc(NC(=O)NCCc2ccc(F)cc2)cn1 ZINC000217533595 CF On-Demand Unstable CCR3 51 37 Cc1ccc(NC(=O)NCCc2ccc(F)cc2)cn1 ZINC000217533595 CF On-Demand Unstable RAF1 41 44 Cc1ccc(NC(=O)NCCc2ccc(F)cc2)cn1 ZINC000217533595 CF On-Demand Unstable NAMPT 29 47 c1ccc(CN2CC[C@@H]([C@@H]3CO3)C2)cc1 ZINC000217533604 BD In-Stock Unstable DRD2 23 49 c1ccc(CN2CC[C@@H]([C@@H]3CO3)C2)cc1 ZINC000217533604 BD In-Stock Unstable DRD4 45 49 c1ccc(CN2CC[C@@H]([C@@H]3CO3)C2)cc1 ZINC000217533604 BD In-Stock Unstable ACHE 35 43 c1ccc(CN2CC[C@@H]([C@@H]3CO3)C2)cc1 ZINC000217533604 BD In-Stock Unstable DRD3 24 49 c1ccc(CN2CC[C@@H]([C@@H]3CO3)C2)cc1 ZINC000217533604 BD In-Stock Unstable VACHT_TETCF 0 48 c1ccc(CN2CC[C@@H]([C@@H]3CO3)C2)cc1 ZINC000217533604 BD In-Stock Unstable SIGMAR1 88 52 c1ccc(CN2CC[C@@H]([C@@H]3CO3)C2)cc1 ZINC000217533604 BD In-Stock Unstable SLC18A3 22 45 NC[C@@H]1CCCN(C(=O)/C=C\c2ccc(Cl)cc2)C1 ZINC000217533610 CF On-Demand Unstable GPR183 0 40 Cn1c(CCNC(=O)c2cc(=O)[nH]c3ccc(F)cc23)nc2ccccc21 ZINC000217533655 FF In-Stock Unstable PLD2 61 37 Cn1c(CCNC(=O)c2cc(=O)[nH]c3ccc(F)cc23)nc2ccccc21 ZINC000217533655 FF In-Stock Unstable POLR1A 49 30 O=C1OC2(CCN(C(=O)CSc3nc4ccccc4s3)CC2)c2ccccc21 ZINC000217533675 HI For-Sale Unstable NPY5R 45 48 NC[C@H]1CCCN(C(=O)/C=C\c2ccc(Cl)cc2)C1 ZINC000217533693 CF On-Demand Unstable GPR183 0 40 COc1cccc(/C=C\C(=O)NCC2CC(O)C2)c1 ZINC000217533768 CD For-Sale Unstable DRD4 41 32 COc1cccc(/C=C\C(=O)NCC2CC(O)C2)c1 ZINC000217533768 CD For-Sale Unstable HDAC8 55 40 COc1cccc(/C=C\C(=O)NCC2CC(O)C2)c1 ZINC000217533768 CD For-Sale Unstable MTNR1A 63 39 COc1cccc(/C=C\C(=O)NCC2CC(O)C2)c1 ZINC000217533768 CD For-Sale Unstable MTNR1B 56 39 COc1cccc(/C=C\C(=O)NCC2CC(O)C2)c1 ZINC000217533768 CD For-Sale Unstable MMP2 15 45 COc1cccc(/C=C\C(=O)NCC2CC(O)C2)c1 ZINC000217533768 CD For-Sale Unstable HDAC1 27 46 COc1cccc(/C=C\C(=O)NCC2CC(O)C2)c1 ZINC000217533768 CD For-Sale Unstable HDAC6 34 40 Cn1c(=O)c2c(ncn2CC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)n(C)c1=O ZINC000217533783 HC For-Sale Unstable NPY5R 39 45 O=C(O)[C@@H](c1c[nH]c2cc(OCc3ccccc3)ccc12)N1C[C@@H]2C[C@H](C1)Cn1c2cccc1=O ZINC000217533800 JI In-Stock Unstable CHRNA4 26 44 O=C(O)[C@@H](c1c[nH]c2cc(OCc3ccccc3)ccc12)N1C[C@@H]2C[C@H](C1)Cn1c2cccc1=O ZINC000217533800 JI In-Stock Unstable MDH2 0 40 O=C(NCCc1ccc(F)cc1)Nc1ccc(Br)cn1 ZINC000217533812 EG For-Sale Unstable POL 0 59 O=C(O)[C@H](c1c[nH]c2cc(OCc3ccccc3)ccc12)N1C[C@@H]2C[C@H](C1)Cn1c2cccc1=O ZINC000217533883 JI In-Stock Unstable CHRNA4 26 44 O=C(O)[C@H](c1c[nH]c2cc(OCc3ccccc3)ccc12)N1C[C@@H]2C[C@H](C1)Cn1c2cccc1=O ZINC000217533883 JI In-Stock Unstable MDH2 0 40 O=C1OC2(CCN(C(=O)c3ccc4nccnc4c3)CC2)c2ccccc21 ZINC000217533892 FF For-Sale Unstable AVPR1A 18 49 O=C1OC2(CCN(C(=O)c3ccc4nccnc4c3)CC2)c2ccccc21 ZINC000217533892 FF For-Sale Unstable ACACA 50 38 O=C1OC2(CCN(C(=O)c3ccc4nccnc4c3)CC2)c2ccccc21 ZINC000217533892 FF For-Sale Unstable NPY5R 58 52 O=C(NCCc1ccc(F)cc1)Nc1cc(Cl)ccn1 ZINC000217533932 CG For-Sale Unstable CCR3 23 43 C[C@@H]1CC[C@@H](C(=O)N[C@H](C)c2cccc(Br)c2)O1 ZINC000217533968 DG On-Demand Unstable SDH1 0 43 CCOc1cc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc(OCC)c1OCC ZINC000217534000 II For-Sale Unstable ACACA 48 39 CCOc1cc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc(OCC)c1OCC ZINC000217534000 II For-Sale Unstable NPY5R 41 49 CCOc1cc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc(OCC)c1OCC ZINC000217534000 II For-Sale Unstable HCN1 48 32 CCOc1cc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc(OCC)c1OCC ZINC000217534000 II For-Sale Unstable HCN4 41 32 NC[C@@H]1CCCN(C(=O)/C=C\c2cccc([N+](=O)[O-])c2)C1 ZINC000217534008 CD On-Demand Unstable CACNA1D 41 34 NC[C@@H]1CCCN(C(=O)/C=C\c2cccc([N+](=O)[O-])c2)C1 ZINC000217534008 CD On-Demand Unstable TRPM8 0 42 C[C@@H]1CC[C@H](C(=O)N[C@H](C)c2cccc(Br)c2)O1 ZINC000217534043 DG On-Demand Unstable SDH1 0 43 O=C(NCC[C@H](O)c1ccsc1)c1ccc(OC(F)(F)F)cc1 ZINC000217534057 EH In-Stock Unstable GCGR 39 44 O=C(NCC[C@H](O)c1ccsc1)c1ccc(OC(F)(F)F)cc1 ZINC000217534057 EH In-Stock Unstable TRPV1 0 50 O=C(NCC[C@H](O)c1ccsc1)c1ccc(OC(F)(F)F)cc1 ZINC000217534057 EH In-Stock Unstable GIPR 44 41 NC[C@H]1CCCN(C(=O)/C=C\c2cccc([N+](=O)[O-])c2)C1 ZINC000217534106 CD On-Demand Unstable CACNA1D 41 34 NC[C@H]1CCCN(C(=O)/C=C\c2cccc([N+](=O)[O-])c2)C1 ZINC000217534106 CD On-Demand Unstable TRPM8 0 42 CCCCCNc1ccc(C(=O)O)cc1S(=O)(=O)N[C@@H](C)COC ZINC000217534113 FE In-Stock Unstable PLA2G4B 43 36 CC(C)C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217534122 CE For-Sale Unstable NPY5R 49 54 O=C(NCC[C@@H](O)c1ccsc1)c1ccc(OC(F)(F)F)cc1 ZINC000217534137 EH In-Stock Unstable GCGR 39 44 O=C(NCC[C@@H](O)c1ccsc1)c1ccc(OC(F)(F)F)cc1 ZINC000217534137 EH In-Stock Unstable TRPV1 0 50 O=C(NCC[C@@H](O)c1ccsc1)c1ccc(OC(F)(F)F)cc1 ZINC000217534137 EH In-Stock Unstable GIPR 44 41 O=C(NCCCCc1ccccc1)NCCc1ccc(F)cc1 ZINC000217534153 DH On-Demand Unstable HRH2 20 41 O=C(NCCCCc1ccccc1)NCCc1ccc(F)cc1 ZINC000217534153 DH On-Demand Unstable SCNN1A 53 39 O=C(NCCCCc1ccccc1)NCCc1ccc(F)cc1 ZINC000217534153 DH On-Demand Unstable MME 15 40 O=C(NCCCCc1ccccc1)NCCc1ccc(F)cc1 ZINC000217534153 DH On-Demand Unstable CA1 16 49 O=C(NCCCCc1ccccc1)NCCc1ccc(F)cc1 ZINC000217534153 DH On-Demand Unstable SIGMAR1 19 49 O=C(NCCCCc1ccccc1)NCCc1ccc(F)cc1 ZINC000217534153 DH On-Demand Unstable CCR3 30 61 O=C(NCCCCc1ccccc1)NCCc1ccc(F)cc1 ZINC000217534153 DH On-Demand Unstable SCN2A 25 42 O=C(NCCCCc1ccccc1)NCCc1ccc(F)cc1 ZINC000217534153 DH On-Demand Unstable CA5B 16 43 O=C(NCCCCc1ccccc1)NCCc1ccc(F)cc1 ZINC000217534153 DH On-Demand Unstable CA5A 16 49 O=C(NCCCCc1ccccc1)NCCc1ccc(F)cc1 ZINC000217534153 DH On-Demand Unstable MTNR1A 27 42 O=C(NCCCCc1ccccc1)NCCc1ccc(F)cc1 ZINC000217534153 DH On-Demand Unstable MTNR1B 37 42 O=C(NCCCCc1ccccc1)NCCc1ccc(F)cc1 ZINC000217534153 DH On-Demand Unstable MMP2 15 43 O=C(NCCCCc1ccccc1)NCCc1ccc(F)cc1 ZINC000217534153 DH On-Demand Unstable MMP3 20 42 O=C(NCCCCc1ccccc1)NCCc1ccc(F)cc1 ZINC000217534153 DH On-Demand Unstable FAAH 55 45 O=C(NCCCCc1ccccc1)NCCc1ccc(F)cc1 ZINC000217534153 DH On-Demand Unstable S1PR2 22 42 O=C(NCCCCc1ccccc1)NCCc1ccc(F)cc1 ZINC000217534153 DH On-Demand Unstable SLC6A5 29 47 O=C(NCCCCc1ccccc1)NCCc1ccc(F)cc1 ZINC000217534153 DH On-Demand Unstable CES1 61 42 O=C(NCCCCc1ccccc1)NCCc1ccc(F)cc1 ZINC000217534153 DH On-Demand Unstable AMP1_PLAFQ 36 48 O=C(NCCCCc1ccccc1)NCCc1ccc(F)cc1 ZINC000217534153 DH On-Demand Unstable LEF 50 38 O=C(NCCCCc1ccccc1)NCCc1ccc(F)cc1 ZINC000217534153 DH On-Demand Unstable NCE103 27 44 O=C(NCCCCc1ccccc1)NCCc1ccc(F)cc1 ZINC000217534153 DH On-Demand Unstable CRTM 35 42 CCCCCNc1ccc(C(=O)O)cc1S(=O)(=O)N[C@H](C)COC ZINC000217534198 FE In-Stock Unstable PLA2G4B 43 36 CC(C)NCC(=O)O[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217534209 CF For-Sale Unstable TRPM8 0 40 O=C1OC2(CCN(C(=O)c3cccc4ccccc34)CC2)c2ccccc21 ZINC000217534238 FI For-Sale Unstable NPY5R 47 51 CCOc1ccc(/C=C\C(=O)NC2CC(O)C2)cc1 ZINC000217534310 CD For-Sale Unstable HDAC8 29 44 CCOc1ccc(/C=C\C(=O)NC2CC(O)C2)cc1 ZINC000217534310 CD For-Sale Unstable MMP2 0 43 CCOc1ccc(/C=C\C(=O)NC2CC(O)C2)cc1 ZINC000217534310 CD For-Sale Unstable HDAC6 23 44 CC(C)NCC(=O)O[C@H]1C[C@H](C)CC[C@@H]1C(C)C ZINC000217534317 CF For-Sale Unstable TRPM8 0 40 COc1ccc2[nH]cc([C@H](C(=O)O)N3C[C@@H]4C[C@H](C3)Cn3c4cccc3=O)c2c1 ZINC000217534335 GF In-Stock Unstable CHRNA4 25 40 O=C1OC2(CCN(C(=O)COc3cccnc3)CC2)c2ccccc21 ZINC000217534356 EE For-Sale Unstable AVPR1A 16 41 O=C1OC2(CCN(C(=O)COc3cccnc3)CC2)c2ccccc21 ZINC000217534356 EE For-Sale Unstable CPT2 40 32 O=C1OC2(CCN(C(=O)COc3cccnc3)CC2)c2ccccc21 ZINC000217534356 EE For-Sale Unstable NPY5R 59 52 COc1ccc(Br)cc1/C=C\C(=O)NC1CC(O)C1 ZINC000217534412 EE For-Sale Unstable TNFRSF1A 16 55 COc1ccc(Br)cc1/C=C\C(=O)NC1CC(O)C1 ZINC000217534412 EE For-Sale Unstable BOTA 25 41 CC(C)(C)OC(=O)NC[C@@H]1CC[C@@H](C(=O)Oc2cc3oc(=O)c4ccccc4c3cc2Cl)CC1 ZINC000217534420 JK In-Stock Unstable ACACB 27 43 CC(C)(C)OC(=O)NC[C@@H]1CC[C@@H](C(=O)Oc2cc3oc(=O)c4ccccc4c3cc2Cl)CC1 ZINC000217534420 JK In-Stock Unstable RAF1 0 40 COc1ccc2[nH]cc([C@@H](C(=O)O)N3C[C@@H]4C[C@H](C3)Cn3c4cccc3=O)c2c1 ZINC000217534427 GF In-Stock Unstable CHRNA4 25 40 O=C1OC2(CCN(C(=O)Cc3cccc4ccccc34)CC2)c2ccccc21 ZINC000217534469 FI For-Sale Unstable NPY5R 42 49 O=C(O)[C@@H](c1c(-c2ccccc2)[nH]c2ccccc12)N1C[C@@H]2C[C@H](C1)Cn1c2cccc1=O ZINC000217534550 II In-Stock Unstable CHRNA4 29 48 COc1ccc(CNS(=O)(=O)CCCCO)cc1 ZINC000217534559 CC For-Sale Unstable MMP13 43 50 COc1ccc(CNS(=O)(=O)CCCCO)cc1 ZINC000217534559 CC For-Sale Unstable MMP2 22 43 COc1ccc(CNS(=O)(=O)CCCCO)cc1 ZINC000217534559 CC For-Sale Unstable MMP8 23 50 COc1ccc(CNS(=O)(=O)CCCCO)cc1 ZINC000217534559 CC For-Sale Unstable MMP9 43 43 COc1ccc(CNS(=O)(=O)CCCCO)cc1 ZINC000217534559 CC For-Sale Unstable MMP12 29 50 COc1ccc(CNS(=O)(=O)CCCCO)cc1 ZINC000217534559 CC For-Sale Unstable CA9 17 43 COc1ccc(CNS(=O)(=O)CCCCO)cc1 ZINC000217534559 CC For-Sale Unstable MMP1 45 38 O=C1OC2(CCN(C(=O)Cc3c[nH]c4ccccc34)CC2)c2ccccc21 ZINC000217534581 FG For-Sale Unstable AVPR1A 24 56 O=C1OC2(CCN(C(=O)Cc3c[nH]c4ccccc34)CC2)c2ccccc21 ZINC000217534581 FG For-Sale Unstable NPY5R 33 45 O=C1OC2(CCN(C(=O)Cc3c[nH]c4ccccc34)CC2)c2ccccc21 ZINC000217534581 FG For-Sale Unstable SSSIM 27 41 CCOC(=O)NCCNC(=O)NCCc1ccc(F)cc1 ZINC000217534630 CD For-Sale Unstable CA1 15 49 CCOC(=O)NCCNC(=O)NCCc1ccc(F)cc1 ZINC000217534630 CD For-Sale Unstable LEF 49 38 O=C(O)[C@H](c1c(-c2ccccc2)[nH]c2ccccc12)N1C[C@@H]2C[C@H](C1)Cn1c2cccc1=O ZINC000217534643 II In-Stock Unstable CHRNA4 29 48 CCC(CC)C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217534714 DG For-Sale Unstable NPY5R 46 51 Cc1c(O)c(=O)oc2cc(N)ccc12 ZINC000217534722 AD For-Sale Unstable MAOB 44 45 Cc1c(O)c(=O)oc2cc(N)ccc12 ZINC000217534722 AD For-Sale Unstable CCR4 0 45 Cc1c(O)c(=O)oc2cc(N)ccc12 ZINC000217534722 AD For-Sale Unstable HSD17B3 31 56 Cc1c(O)c(=O)oc2cc(N)ccc12 ZINC000217534722 AD For-Sale Unstable NQO1 71 45 O=C(O)[C@@H](c1c[nH]c2cc(F)ccc12)N1C[C@@H]2C[C@H](C1)Cn1c2cccc1=O ZINC000217534761 GF In-Stock Unstable CHRNA4 35 49 CC[C@@H](C)[C@@H](C(=O)N1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217534796 CG For-Sale Unstable CHRM1 17 40 CC[C@@H](C)[C@@H](C(=O)N1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217534796 CG For-Sale Unstable ACE 38 42 CC[C@@H](C)[C@@H](C(=O)N1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217534796 CG For-Sale Unstable REN 16 41 CC[C@@H](C)[C@@H](C(=O)N1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217534796 CG For-Sale Unstable DPP7 61 37 COc1cc(/C=C/C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc(OC)c1OC ZINC000217534831 HG For-Sale Unstable ITGAL 16 40 COc1cc(/C=C/C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc(OC)c1OC ZINC000217534831 HG For-Sale Unstable NPY5R 32 53 O=S(=O)(NCC[C@H](O)c1ccsc1)c1cccnc1 ZINC000217534851 CD In-Stock Unstable ADRB3 64 37 O=C(NCCc1ccc(Br)cc1)Nc1cccc(C(=O)O)c1 ZINC000217534855 FH On-Demand Unstable CCKAR 0 43 O=C(NCCc1ccc(Br)cc1)Nc1cccc(C(=O)O)c1 ZINC000217534855 FH On-Demand Unstable Q8MMZ8_EIMTE 0 43 CC[C@H](C)[C@@H](C(=O)N1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217534870 CG On-Demand Unstable ACE 26 42 CC[C@H](C)[C@@H](C(=O)N1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217534870 CG On-Demand Unstable DPP7 54 34 COC(=O)Cn1nc(-c2cccnc2)cc1N ZINC000217534906 BC In-Stock Unstable CYP2A6 35 43 O=S(=O)(NCC[C@@H](O)c1ccsc1)c1cccnc1 ZINC000217534931 CD In-Stock Unstable ADRB3 64 37 CC[C@@H](C)[C@H](C(=O)N1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217534947 CG For-Sale Unstable CHRM1 17 40 CC[C@@H](C)[C@H](C(=O)N1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217534947 CG For-Sale Unstable ACE 38 42 CC[C@@H](C)[C@H](C(=O)N1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217534947 CG For-Sale Unstable REN 16 41 CC[C@@H](C)[C@H](C(=O)N1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217534947 CG For-Sale Unstable DPP7 61 37 Cc1c(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cnn1-c1ccccc1 ZINC000217534957 GG For-Sale Unstable AVPR1A 21 49 Cc1c(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cnn1-c1ccccc1 ZINC000217534957 GG For-Sale Unstable NPY5R 48 55 O=C(NCCc1ccc(Br)cc1)Nc1ccccc1[N+](=O)[O-] ZINC000217534962 FH For-Sale Unstable COLA 84 39 CC[C@H](C)[C@H](C(=O)N1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217535034 CG On-Demand Unstable ACE 26 42 CC[C@H](C)[C@H](C(=O)N1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217535034 CG On-Demand Unstable DPP7 54 34 O=C(O)CCNC(=O)NCCc1ccc(Br)cc1 ZINC000217535065 DD On-Demand Unstable CA5A 15 40 O=C(O)CCNC(=O)NCCc1ccc(Br)cc1 ZINC000217535065 DD On-Demand Unstable FFAR1 42 49 COc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c(OC)c1 ZINC000217535074 FG For-Sale Unstable OXTR 27 40 COc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c(OC)c1 ZINC000217535074 FG For-Sale Unstable AVPR1A 16 52 COc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c(OC)c1 ZINC000217535074 FG For-Sale Unstable ACACA 21 41 COc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c(OC)c1 ZINC000217535074 FG For-Sale Unstable NPY5R 37 54 O=C(O)[C@@H](c1c[nH]c2ccccc12)N1C[C@@H]2C[C@H](C1)Cn1c2cccc1=O ZINC000217535079 FF In-Stock Unstable CHRNA4 28 46 C/C(=C/Br)c1ccc(Cl)c(Cl)c1 ZINC000217535141 CJ For-Sale Unstable CYSP_TRYCR 16 41 CC(C)(NC(=O)c1ccc(-c2ccccc2Cl)o1)c1nnc(N)s1 ZINC000217535143 FH In-Stock Unstable MAP 0 55 O=C(O)[C@H](c1c[nH]c2ccccc12)N1C[C@@H]2C[C@H](C1)Cn1c2cccc1=O ZINC000217535164 FF In-Stock Unstable CHRNA4 28 46 O=C1OC2(CCN(C(=O)c3ccc4ccccc4c3)CC2)c2ccccc21 ZINC000217535213 FI For-Sale Unstable ACACA 60 36 O=C1OC2(CCN(C(=O)c3ccc4ccccc4c3)CC2)c2ccccc21 ZINC000217535213 FI For-Sale Unstable ACACB 45 33 O=C1OC2(CCN(C(=O)c3ccc4ccccc4c3)CC2)c2ccccc21 ZINC000217535213 FI For-Sale Unstable NPY5R 48 51 NS(=O)(=O)c1ccc(NCCC2=CCCCC2)c(C(=O)O)c1 ZINC000217535248 DE In-Stock Unstable CA2 58 39 NS(=O)(=O)c1ccc(NCCC2=CCCCC2)c(C(=O)O)c1 ZINC000217535248 DE In-Stock Unstable CA1 52 39 NS(=O)(=O)c1ccc(NCCC2=CCCCC2)c(C(=O)O)c1 ZINC000217535248 DE In-Stock Unstable CA7 44 37 NS(=O)(=O)c1ccc(NCCC2=CCCCC2)c(C(=O)O)c1 ZINC000217535248 DE In-Stock Unstable CA5B 44 37 NS(=O)(=O)c1ccc(NCCC2=CCCCC2)c(C(=O)O)c1 ZINC000217535248 DE In-Stock Unstable CA4 57 38 NS(=O)(=O)c1ccc(NCCC2=CCCCC2)c(C(=O)O)c1 ZINC000217535248 DE In-Stock Unstable CA5A 46 37 O=C(NCCc1ccc(Br)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217535297 GG For-Sale Unstable CA2 44 59 O=C(NCCc1ccc(Br)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217535297 GG For-Sale Unstable CA1 48 59 O=C(NCCc1ccc(Br)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217535297 GG For-Sale Unstable CA7 30 50 O=C(NCCc1ccc(Br)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217535297 GG For-Sale Unstable CA4 26 59 O=C(NCCc1ccc(Br)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217535297 GG For-Sale Unstable CA14 30 50 O=C(NCCc1ccc(Br)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217535297 GG For-Sale Unstable CA12 48 52 O=C(NCCc1ccc(Br)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217535297 GG For-Sale Unstable CA9 49 52 O=C(NCCc1ccc(Br)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217535297 GG For-Sale Unstable IDO1 43 48 O=C(NCCc1ccc(Br)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217535297 GG For-Sale Unstable NCE103 29 59 O=C(NCCc1ccc(Br)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217535297 GG For-Sale Unstable PFK 0 44 O=C(NCCc1ccc(Br)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217535297 GG For-Sale Unstable LIG1 0 48 O=C(NCCc1ccc(Br)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217535297 GG For-Sale Unstable MTCA1 48 51 O=C(NCCc1ccc(Br)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217535297 GG For-Sale Unstable P96878_MYCTU 62 51 O=C(NCCc1ccc(Br)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217535297 GG For-Sale Unstable NAMPT 45 46 O=C(NCCc1ccc(Br)cc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217535297 GG For-Sale Unstable A6YCJ1_9METZ 15 42 COc1ccc(/C(C)=C\Br)cc1F ZINC000217535300 BH For-Sale Unstable TUBB1 48 50 O=C1OC2(CCN(C(=O)c3ccc4ccccc4n3)CC2)c2ccccc21 ZINC000217535319 FH For-Sale Unstable AVPR1A 15 51 O=C1OC2(CCN(C(=O)c3ccc4ccccc4n3)CC2)c2ccccc21 ZINC000217535319 FH For-Sale Unstable NPY5R 49 51 NC[C@@H]1CCCN(C(=O)/C=C\c2ccc([N+](=O)[O-])cc2)C1 ZINC000217535339 CD On-Demand Unstable SLC27A4 47 31 C[C@@H](Nc1ccc(S(N)(=O)=O)cc1C(=O)O)c1ccccc1 ZINC000217535366 DE In-Stock Unstable CA2 84 45 C[C@@H](Nc1ccc(S(N)(=O)=O)cc1C(=O)O)c1ccccc1 ZINC000217535366 DE In-Stock Unstable CA1 69 42 C[C@@H](Nc1ccc(S(N)(=O)=O)cc1C(=O)O)c1ccccc1 ZINC000217535366 DE In-Stock Unstable CA7 43 44 C[C@@H](Nc1ccc(S(N)(=O)=O)cc1C(=O)O)c1ccccc1 ZINC000217535366 DE In-Stock Unstable CA5B 53 44 C[C@@H](Nc1ccc(S(N)(=O)=O)cc1C(=O)O)c1ccccc1 ZINC000217535366 DE In-Stock Unstable CA4 84 45 C[C@@H](Nc1ccc(S(N)(=O)=O)cc1C(=O)O)c1ccccc1 ZINC000217535366 DE In-Stock Unstable CA5A 61 44 C[C@@H](Nc1ccc(S(N)(=O)=O)cc1C(=O)O)c1ccccc1 ZINC000217535366 DE In-Stock Unstable CA12 36 41 C[C@@H](Nc1ccc(S(N)(=O)=O)cc1C(=O)O)c1ccccc1 ZINC000217535366 DE In-Stock Unstable CA9 43 41 C[C@@H](Nc1ccc(S(N)(=O)=O)cc1C(=O)O)c1ccccc1 ZINC000217535366 DE In-Stock Unstable P96878_MYCTU 42 38 O=C(NCCc1ccc(Br)cc1)Nc1cccc(S(=O)(=O)O)c1 ZINC000217535399 GG For-Sale Unstable CA2 24 54 O=C(NCCc1ccc(Br)cc1)Nc1cccc(S(=O)(=O)O)c1 ZINC000217535399 GG For-Sale Unstable CA1 25 54 O=C(NCCc1ccc(Br)cc1)Nc1cccc(S(=O)(=O)O)c1 ZINC000217535399 GG For-Sale Unstable CCR3 27 43 O=C(NCCc1ccc(Br)cc1)Nc1cccc(S(=O)(=O)O)c1 ZINC000217535399 GG For-Sale Unstable CA4 21 54 O=C(NCCc1ccc(Br)cc1)Nc1cccc(S(=O)(=O)O)c1 ZINC000217535399 GG For-Sale Unstable CA5A 15 47 O=C(NCCc1ccc(Br)cc1)Nc1cccc(S(=O)(=O)O)c1 ZINC000217535399 GG For-Sale Unstable CA12 22 47 O=C(NCCc1ccc(Br)cc1)Nc1cccc(S(=O)(=O)O)c1 ZINC000217535399 GG For-Sale Unstable CA9 23 45 O=C(NCCc1ccc(Br)cc1)Nc1cccc(S(=O)(=O)O)c1 ZINC000217535399 GG For-Sale Unstable LIG1 0 42 NC[C@H]1CCCN(C(=O)/C=C\c2ccc([N+](=O)[O-])cc2)C1 ZINC000217535427 CD On-Demand Unstable SLC27A4 47 31 Cc1ccc(OCC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217535437 FG For-Sale Unstable NPY5R 44 49 COc1ccc2c(c1OC)C(=O)O[C@@H]2N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217535440 GE In-Stock Unstable CHRNA4 26 42 C[C@H](Nc1ccc(S(N)(=O)=O)cc1C(=O)O)c1ccccc1 ZINC000217535449 DE In-Stock Unstable CA2 84 45 C[C@H](Nc1ccc(S(N)(=O)=O)cc1C(=O)O)c1ccccc1 ZINC000217535449 DE In-Stock Unstable CA1 69 42 C[C@H](Nc1ccc(S(N)(=O)=O)cc1C(=O)O)c1ccccc1 ZINC000217535449 DE In-Stock Unstable CA7 43 44 C[C@H](Nc1ccc(S(N)(=O)=O)cc1C(=O)O)c1ccccc1 ZINC000217535449 DE In-Stock Unstable CA5B 53 44 C[C@H](Nc1ccc(S(N)(=O)=O)cc1C(=O)O)c1ccccc1 ZINC000217535449 DE In-Stock Unstable CA4 84 45 C[C@H](Nc1ccc(S(N)(=O)=O)cc1C(=O)O)c1ccccc1 ZINC000217535449 DE In-Stock Unstable CA5A 61 44 C[C@H](Nc1ccc(S(N)(=O)=O)cc1C(=O)O)c1ccccc1 ZINC000217535449 DE In-Stock Unstable CA12 36 41 C[C@H](Nc1ccc(S(N)(=O)=O)cc1C(=O)O)c1ccccc1 ZINC000217535449 DE In-Stock Unstable CA9 43 41 C[C@H](Nc1ccc(S(N)(=O)=O)cc1C(=O)O)c1ccccc1 ZINC000217535449 DE In-Stock Unstable P96878_MYCTU 42 38 O=C(/C=C\c1cccnc1)NCC1CC(O)C1 ZINC000217535520 BC On-Demand Unstable IMA1 0 41 CC(C)c1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217535522 FJ For-Sale Unstable CA1 16 43 CC(C)c1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217535522 FJ For-Sale Unstable F7 23 48 CC(C)c1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217535522 FJ For-Sale Unstable CA12 15 46 CC(C)c1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217535522 FJ For-Sale Unstable NCE103 24 46 CC(C)c1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217535522 FJ For-Sale Unstable P96878_MYCTU 17 45 COc1ccc2c(c1OC)C(=O)O[C@H]2N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217535523 GE In-Stock Unstable CHRNA4 26 42 O=C1OC2(CCN(C(=O)Cn3ncccc3=O)CC2)c2ccccc21 ZINC000217535534 EC In-Stock Unstable NPY5R 50 48 NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217535556 DD In-Stock Unstable CA2 139 53 NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217535556 DD In-Stock Unstable CA6 25 43 NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217535556 DD In-Stock Unstable CA1 112 51 NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217535556 DD In-Stock Unstable CA7 70 53 NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217535556 DD In-Stock Unstable CA13 37 43 NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217535556 DD In-Stock Unstable CA5B 81 53 NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217535556 DD In-Stock Unstable CA4 122 48 NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217535556 DD In-Stock Unstable CA5A 87 53 NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217535556 DD In-Stock Unstable CA14 45 45 NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217535556 DD In-Stock Unstable CA12 66 50 NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217535556 DD In-Stock Unstable CA9 66 50 NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217535556 DD In-Stock Unstable CAH_METTE 43 36 NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217535556 DD In-Stock Unstable AKR1C3 17 43 NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217535556 DD In-Stock Unstable CYNT 45 35 NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217535556 DD In-Stock Unstable NCE103 46 41 NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217535556 DD In-Stock Unstable ALPI 15 50 NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217535556 DD In-Stock Unstable CA15 26 41 NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217535556 DD In-Stock Unstable MTCA1 38 41 NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217535556 DD In-Stock Unstable P96878_MYCTU 44 41 NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217535556 DD In-Stock Unstable CA 0 42 NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217535556 DD In-Stock Unstable A6YCJ1_9METZ 24 44 NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217535556 DD In-Stock Unstable Q5TU56_ANOGA 0 41 CN1CC[C@@H](CN(C)c2cc(Cl)ccc2CBr)C1 ZINC000217535589 EH For-Sale Unstable NOS2 15 45 CN1CC[C@@H](CN(C)c2cc(Cl)ccc2CBr)C1 ZINC000217535589 EH For-Sale Unstable NOS3 19 45 Cc1cc(S(=O)(=O)NCC[C@H](O)c2ccsc2)ccc1F ZINC000217535614 EF In-Stock Unstable LEF 70 42 O=C1OC2(CCN(C(=O)C3CCCCC3)CC2)c2ccccc21 ZINC000217535635 DG For-Sale Unstable NPY5R 61 53 Cc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1Cl ZINC000217535639 FJ For-Sale Unstable LDHA 25 42 Cc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1Cl ZINC000217535639 FJ For-Sale Unstable RAF1 36 59 Cc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1Cl ZINC000217535639 FJ For-Sale Unstable Q8MMZ8_EIMTE 25 59 Cc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1Cl ZINC000217535639 FJ For-Sale Unstable NCE103 34 42 COc1ccc(CNS(=O)(=O)[C@@H](C)CO)cc1 ZINC000217535653 CC For-Sale Unstable BMP1 55 37 COc1ccc(CNS(=O)(=O)[C@@H](C)CO)cc1 ZINC000217535653 CC For-Sale Unstable MMP13 36 42 COc1ccc(CNS(=O)(=O)[C@@H](C)CO)cc1 ZINC000217535653 CC For-Sale Unstable MMP2 27 40 COc1ccc(CNS(=O)(=O)[C@@H](C)CO)cc1 ZINC000217535653 CC For-Sale Unstable MMP8 24 42 COc1ccc(CNS(=O)(=O)[C@@H](C)CO)cc1 ZINC000217535653 CC For-Sale Unstable MMP9 36 40 COc1ccc(CNS(=O)(=O)[C@@H](C)CO)cc1 ZINC000217535653 CC For-Sale Unstable MMP12 28 42 COc1ccc(CNS(=O)(=O)[C@@H](C)CO)cc1 ZINC000217535653 CC For-Sale Unstable MMP7 27 41 COc1ccc(CNS(=O)(=O)[C@@H](C)CO)cc1 ZINC000217535653 CC For-Sale Unstable CA9 20 44 COc1ccc(CNS(=O)(=O)[C@@H](C)CO)cc1 ZINC000217535653 CC For-Sale Unstable MMP1 42 41 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1 ZINC000217535666 FD In-Stock Unstable CA2 118 55 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1 ZINC000217535666 FD In-Stock Unstable BMP1 81 39 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1 ZINC000217535666 FD In-Stock Unstable CA6 22 43 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1 ZINC000217535666 FD In-Stock Unstable CA1 100 54 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1 ZINC000217535666 FD In-Stock Unstable CA7 64 46 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1 ZINC000217535666 FD In-Stock Unstable MMP13 49 40 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1 ZINC000217535666 FD In-Stock Unstable CA13 22 43 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1 ZINC000217535666 FD In-Stock Unstable CA5B 56 42 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1 ZINC000217535666 FD In-Stock Unstable CA4 83 43 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1 ZINC000217535666 FD In-Stock Unstable CA5A 59 42 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1 ZINC000217535666 FD In-Stock Unstable MMP16 0 48 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1 ZINC000217535666 FD In-Stock Unstable CA14 48 49 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1 ZINC000217535666 FD In-Stock Unstable MMP2 28 45 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1 ZINC000217535666 FD In-Stock Unstable MMP3 49 39 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1 ZINC000217535666 FD In-Stock Unstable MMP9 47 40 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1 ZINC000217535666 FD In-Stock Unstable CA12 63 54 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1 ZINC000217535666 FD In-Stock Unstable PTGDR 24 50 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1 ZINC000217535666 FD In-Stock Unstable MMP7 42 39 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1 ZINC000217535666 FD In-Stock Unstable CA9 68 55 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1 ZINC000217535666 FD In-Stock Unstable MMP1 64 48 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1 ZINC000217535666 FD In-Stock Unstable AKR1C3 28 40 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1 ZINC000217535666 FD In-Stock Unstable CYNT 31 42 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1 ZINC000217535666 FD In-Stock Unstable NCE103 39 40 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1 ZINC000217535666 FD In-Stock Unstable AKR1C2 54 40 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1 ZINC000217535666 FD In-Stock Unstable SCMU_MYCTU 0 41 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1 ZINC000217535666 FD In-Stock Unstable CA 0 40 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1 ZINC000217535666 FD In-Stock Unstable A6YCJ1_9METZ 23 42 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1 ZINC000217535666 FD In-Stock Unstable CHMU_MYCTU 0 43 CN1CC[C@H](CN(C)c2cc(Cl)ccc2CBr)C1 ZINC000217535684 EH For-Sale Unstable NOS2 15 45 CN1CC[C@H](CN(C)c2cc(Cl)ccc2CBr)C1 ZINC000217535684 EH For-Sale Unstable NOS3 19 45 Cc1cc(S(=O)(=O)NCC[C@@H](O)c2ccsc2)ccc1F ZINC000217535688 EF In-Stock Unstable LEF 70 42 CC(C)N(C)CCCNC(=O)c1ccc(Br)c(Cl)c1 ZINC000217535721 EH On-Demand Unstable CA2 21 45 COc1ccc(CNS(=O)(=O)[C@H](C)CO)cc1 ZINC000217535732 CC For-Sale Unstable BMP1 55 37 COc1ccc(CNS(=O)(=O)[C@H](C)CO)cc1 ZINC000217535732 CC For-Sale Unstable MMP13 36 42 COc1ccc(CNS(=O)(=O)[C@H](C)CO)cc1 ZINC000217535732 CC For-Sale Unstable MMP2 27 40 COc1ccc(CNS(=O)(=O)[C@H](C)CO)cc1 ZINC000217535732 CC For-Sale Unstable MMP8 24 42 COc1ccc(CNS(=O)(=O)[C@H](C)CO)cc1 ZINC000217535732 CC For-Sale Unstable MMP9 36 40 COc1ccc(CNS(=O)(=O)[C@H](C)CO)cc1 ZINC000217535732 CC For-Sale Unstable MMP12 28 42 COc1ccc(CNS(=O)(=O)[C@H](C)CO)cc1 ZINC000217535732 CC For-Sale Unstable MMP7 27 41 COc1ccc(CNS(=O)(=O)[C@H](C)CO)cc1 ZINC000217535732 CC For-Sale Unstable CA9 20 44 COc1ccc(CNS(=O)(=O)[C@H](C)CO)cc1 ZINC000217535732 CC For-Sale Unstable MMP1 42 41 Cc1cccc(C(C)C)c1NC(=O)NCCc1ccc(Br)cc1 ZINC000217535746 GK On-Demand Unstable SOAT1 60 48 Cc1cccc(C(C)C)c1NC(=O)NCCc1ccc(Br)cc1 ZINC000217535746 GK On-Demand Unstable ACAT 0 67 Cc1cccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217535753 DG For-Sale Unstable AVPR1A 15 52 Cc1cccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217535753 DG For-Sale Unstable INHA 21 52 Cc1cccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217535753 DG For-Sale Unstable ACACA 55 37 Cc1cccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217535753 DG For-Sale Unstable NPY5R 44 49 Cc1cccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217535753 DG For-Sale Unstable KCNK3 47 35 Cc1cccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217535753 DG For-Sale Unstable KCNK9 40 35 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1OC ZINC000217535772 GD In-Stock Unstable CA2 92 52 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1OC ZINC000217535772 GD In-Stock Unstable CA1 79 53 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1OC ZINC000217535772 GD In-Stock Unstable CA7 48 60 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1OC ZINC000217535772 GD In-Stock Unstable CA5B 50 38 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1OC ZINC000217535772 GD In-Stock Unstable CA4 75 39 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1OC ZINC000217535772 GD In-Stock Unstable CA5A 53 38 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1OC ZINC000217535772 GD In-Stock Unstable CA14 35 60 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1OC ZINC000217535772 GD In-Stock Unstable CA12 46 42 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1OC ZINC000217535772 GD In-Stock Unstable IAP 0 40 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1OC ZINC000217535772 GD In-Stock Unstable CA9 50 44 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1OC ZINC000217535772 GD In-Stock Unstable NCE103 35 43 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1OC ZINC000217535772 GD In-Stock Unstable P96878_MYCTU 26 43 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1OC ZINC000217535772 GD In-Stock Unstable SCMU_MYCTU 0 56 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1OC ZINC000217535772 GD In-Stock Unstable CA 0 41 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1OC ZINC000217535772 GD In-Stock Unstable CAN2 0 43 COc1ccc(CCNc2ccc(S(N)(=O)=O)cc2C(=O)O)cc1OC ZINC000217535772 GD In-Stock Unstable Q5TU56_ANOGA 0 41 CN1CC[C@@H](CN(C)c2ccc(Cl)cc2CBr)C1 ZINC000217535787 EH For-Sale Unstable SLC6A1 33 41 CN1CC[C@@H](CN(C)c2ccc(Cl)cc2CBr)C1 ZINC000217535787 EH For-Sale Unstable NOS2 17 48 CN1CC[C@@H](CN(C)c2ccc(Cl)cc2CBr)C1 ZINC000217535787 EH For-Sale Unstable NOS3 21 48 O=C(NCCc1ccc(Br)cc1)Nc1ccc(C(=O)O)cc1 ZINC000217535856 FH On-Demand Unstable CA1 15 48 O=C(NCCc1ccc(Br)cc1)Nc1ccc(C(=O)O)cc1 ZINC000217535856 FH On-Demand Unstable CA9 16 56 O=C(NCCc1ccc(Br)cc1)Nc1ccc(C(=O)O)cc1 ZINC000217535856 FH On-Demand Unstable IDO1 15 41 O=C(NCCc1ccc(Br)cc1)Nc1ccc(C(=O)O)cc1 ZINC000217535856 FH On-Demand Unstable NCE103 21 51 CCCC(CCC)C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217535858 EH For-Sale Unstable NPY5R 41 49 CN1CC[C@H](CN(C)c2ccc(Cl)cc2CBr)C1 ZINC000217535879 EH For-Sale Unstable SLC6A1 33 41 CN1CC[C@H](CN(C)c2ccc(Cl)cc2CBr)C1 ZINC000217535879 EH For-Sale Unstable NOS2 17 48 CN1CC[C@H](CN(C)c2ccc(Cl)cc2CBr)C1 ZINC000217535879 EH For-Sale Unstable NOS3 21 48 CC(C)OCCCNc1ccc(S(N)(=O)=O)cc1C(=O)O ZINC000217535910 DD In-Stock Unstable CA2 91 43 CC(C)OCCCNc1ccc(S(N)(=O)=O)cc1C(=O)O ZINC000217535910 DD In-Stock Unstable CA1 78 40 CC(C)OCCCNc1ccc(S(N)(=O)=O)cc1C(=O)O ZINC000217535910 DD In-Stock Unstable CA7 51 39 CC(C)OCCCNc1ccc(S(N)(=O)=O)cc1C(=O)O ZINC000217535910 DD In-Stock Unstable CA5B 41 39 CC(C)OCCCNc1ccc(S(N)(=O)=O)cc1C(=O)O ZINC000217535910 DD In-Stock Unstable CA4 85 41 CC(C)OCCCNc1ccc(S(N)(=O)=O)cc1C(=O)O ZINC000217535910 DD In-Stock Unstable CA5A 43 39 CC(C)OCCCNc1ccc(S(N)(=O)=O)cc1C(=O)O ZINC000217535910 DD In-Stock Unstable CA12 35 40 CC(C)OCCCNc1ccc(S(N)(=O)=O)cc1C(=O)O ZINC000217535910 DD In-Stock Unstable CA9 37 40 Cc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217535961 DG For-Sale Unstable AVPR1A 15 52 Cc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217535961 DG For-Sale Unstable INHA 20 49 Cc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217535961 DG For-Sale Unstable ACACA 47 37 Cc1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217535961 DG For-Sale Unstable NPY5R 48 54 Cc1c(Cl)cccc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217535977 FJ For-Sale Unstable TRPV1 0 47 O=S(=O)(NCC[C@H](O)c1ccsc1)c1ccccc1Cl ZINC000217535982 EF In-Stock Unstable ITGAV 15 42 CNS(=O)(=O)c1ccc(NCC(C)C)c(C(=O)O)c1 ZINC000217536037 CD In-Stock Unstable F3 43 30 CNS(=O)(=O)c1ccc(NCC(C)C)c(C(=O)O)c1 ZINC000217536037 CD In-Stock Unstable MTNN 73 34 O=S(=O)(NCC[C@@H](O)c1ccsc1)c1ccccc1Cl ZINC000217536058 EF In-Stock Unstable ITGAV 15 42 CCN(CC)S(=O)(=O)c1ccc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217536070 IG For-Sale Unstable NPY5R 37 46 CCOC(=O)c1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217536083 GH For-Sale Unstable CHRM2 0 41 CCOC(=O)c1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217536083 GH For-Sale Unstable CHRM3 0 41 CCOC(=O)c1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217536083 GH For-Sale Unstable CA1 19 45 CCOC(=O)c1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217536083 GH For-Sale Unstable F7 18 42 CCOC(=O)c1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217536083 GH For-Sale Unstable ACR 64 44 CCOC(=O)c1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217536083 GH For-Sale Unstable CA12 18 50 CCOC(=O)c1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217536083 GH For-Sale Unstable CA9 22 50 CCOC(=O)c1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217536083 GH For-Sale Unstable NOD2 17 41 CCCOc1ccc([C@@H](N)CN2CCCO[C@@H](C)C2)cc1 ZINC000217536129 CF For-Sale Unstable PSMB1 36 41 O=C1OC2(CCN(C(=O)c3ccc(S(=O)(=O)N4CCCCC4)cc3)CC2)c2ccccc21 ZINC000217536177 JG For-Sale Unstable NPY5R 35 46 O=C1OC2(CCN(C(=O)c3ccc(S(=O)(=O)N4CCCCC4)cc3)CC2)c2ccccc21 ZINC000217536177 JG For-Sale Unstable L3MBTL3 35 47 CC(C)c1ccccc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217536181 FJ On-Demand Unstable ANPEP 30 43 CC(C)c1ccccc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217536181 FJ On-Demand Unstable SOAT1 43 43 CC(C)c1ccccc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217536181 FJ On-Demand Unstable AMP1_PLAFQ 27 43 CC(C)c1ccccc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217536181 FJ On-Demand Unstable ACAT 0 61 CCCOc1ccc([C@H](N)CN2CCCO[C@@H](C)C2)cc1 ZINC000217536224 CF For-Sale Unstable PSMB1 36 41 O=C1OC2(CCN(C(=O)CSc3ncccn3)CC2)c2ccccc21 ZINC000217536281 FE For-Sale Unstable NPY5R 60 52 O=C(NCCc1ccc(Br)cc1)Nc1cccc(Cl)c1Cl ZINC000217536293 GK For-Sale Unstable NCE103 20 40 COc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1Cl ZINC000217536403 GI On-Demand Unstable HTR2A 26 42 COc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1Cl ZINC000217536403 GI On-Demand Unstable RAF1 27 46 COc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1Cl ZINC000217536403 GI On-Demand Unstable GRM4 15 45 COc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1Cl ZINC000217536403 GI On-Demand Unstable PDE6A 42 33 COc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1Cl ZINC000217536403 GI On-Demand Unstable Q8MMZ8_EIMTE 34 46 COc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1Cl ZINC000217536403 GI On-Demand Unstable P96878_MYCTU 17 45 COc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1Cl ZINC000217536403 GI On-Demand Unstable CAN2 0 45 O=C1OC2(CCN(C(=O)c3cc(-c4ccc(F)cc4)n[nH]3)CC2)c2ccccc21 ZINC000217536404 GH For-Sale Unstable AVPR1A 15 49 O=C1OC2(CCN(C(=O)c3cc(-c4ccc(F)cc4)n[nH]3)CC2)c2ccccc21 ZINC000217536404 GH For-Sale Unstable TACR3 22 51 O=C1OC2(CCN(C(=O)c3cc(-c4ccc(F)cc4)n[nH]3)CC2)c2ccccc21 ZINC000217536404 GH For-Sale Unstable NPY5R 58 65 O=C(/C=C\c1ccccc1Cl)NC1CC(O)C1 ZINC000217536411 CD For-Sale Unstable KCNQ2 22 46 O=C(/C=C\c1ccccc1Cl)NC1CC(O)C1 ZINC000217536411 CD For-Sale Unstable BOTA 30 43 CNS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217536429 DD In-Stock Unstable CA2 27 40 CNS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217536429 DD In-Stock Unstable CA1 23 42 CNS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217536429 DD In-Stock Unstable TRY2_BOVIN 44 32 CNS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217536429 DD In-Stock Unstable BDKRB1 0 40 CNS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217536429 DD In-Stock Unstable CA5B 31 42 CNS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217536429 DD In-Stock Unstable CA5A 35 42 CNS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217536429 DD In-Stock Unstable ACPS 0 40 Cc1cc(S(=O)(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)ccc1F ZINC000217536459 HG For-Sale Unstable LEF 57 34 N#Cc1ccccc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217536504 EH For-Sale Unstable ADRB1 45 37 O=C1OC2(CCN(C(=O)c3cc(-c4cccs4)[nH]n3)CC2)c2ccccc21 ZINC000217536506 GG For-Sale Unstable AVPR1A 15 49 O=C1OC2(CCN(C(=O)c3cc(-c4cccs4)[nH]n3)CC2)c2ccccc21 ZINC000217536506 GG For-Sale Unstable NPY5R 43 50 C[C@@H]1CCCN([C@H](C)C(=O)c2ccccc2)C1 ZINC000217536527 BF For-Sale Unstable ACE 30 41 C[C@@H]1CCCN([C@H](C)C(=O)c2ccccc2)C1 ZINC000217536527 BF For-Sale Unstable SLC6A1 52 35 CCCCCCCCc1cc(F)c(C#N)cc1O ZINC000217536544 BI For-Sale Unstable INHA 47 33 Cc1nc(-n2cccc2)sc1C(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217536614 GH For-Sale Unstable NPY5R 35 47 CCOC(=O)c1ccccc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217536620 GH For-Sale Unstable NCE103 15 41 Cc1ccc2[nH]cc([C@H](C(=O)O)N3C[C@@H]4C[C@H](C3)Cn3c4cccc3=O)c2c1 ZINC000217536654 GF In-Stock Unstable CHRNA4 34 43 C[C@@H]1CCCN([C@H](C)C(=O)c2cccc(Cl)c2)C1 ZINC000217536667 CH For-Sale Unstable GRM5 18 41 C[C@@H]1CCCN([C@H](C)C(=O)c2cccc(Cl)c2)C1 ZINC000217536667 CH For-Sale Unstable CCKBR 0 40 O=C(NCCc1ccc(Br)cc1)Nc1ccc(O)cc1 ZINC000217536702 EH For-Sale Unstable ADRB1 26 40 O=C(NCCc1ccc(Br)cc1)Nc1ccc(O)cc1 ZINC000217536702 EH For-Sale Unstable ADRB3 22 41 O=C(NCCc1ccc(Br)cc1)Nc1ccc(O)cc1 ZINC000217536702 EH For-Sale Unstable CA1 15 50 O=C(NCCc1ccc(Br)cc1)Nc1ccc(O)cc1 ZINC000217536702 EH For-Sale Unstable CA9 15 50 O=C(NCCc1ccc(Br)cc1)Nc1ccc(O)cc1 ZINC000217536702 EH For-Sale Unstable IDO1 17 40 O=C(NCCc1ccc(Br)cc1)Nc1ccc(O)cc1 ZINC000217536702 EH For-Sale Unstable NCE103 26 50 O=C(NCCc1ccc(Br)cc1)Nc1ccc(O)cc1 ZINC000217536702 EH For-Sale Unstable LIG1 0 40 CNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217536724 ED In-Stock Unstable CA2 32 40 CNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217536724 ED In-Stock Unstable CA1 26 41 CNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217536724 ED In-Stock Unstable CA7 23 41 CNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217536724 ED In-Stock Unstable CA5B 38 41 CNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217536724 ED In-Stock Unstable CA5A 39 41 CNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217536724 ED In-Stock Unstable AKR1C3 25 47 Cc1ccc2[nH]cc([C@@H](C(=O)O)N3C[C@@H]4C[C@H](C3)Cn3c4cccc3=O)c2c1 ZINC000217536732 GF In-Stock Unstable CHRNA4 34 43 COc1cc(-c2cc(C(=O)N3CCC4(CC3)OC(=O)c3ccccc34)[nH]n2)cc(OC)c1OC ZINC000217536747 JG For-Sale Unstable TACR3 29 49 COc1cc(-c2cc(C(=O)N3CCC4(CC3)OC(=O)c3ccccc34)[nH]n2)cc(OC)c1OC ZINC000217536747 JG For-Sale Unstable NPY5R 40 56 COc1ccc(CNS(=O)(=O)c2c[nH]c(CO)c2)cc1 ZINC000217536754 CC For-Sale Unstable MMP13 23 41 COc1ccc(CNS(=O)(=O)c2c[nH]c(CO)c2)cc1 ZINC000217536754 CC For-Sale Unstable MMP9 21 41 COc1ccc(CNS(=O)(=O)c2c[nH]c(CO)c2)cc1 ZINC000217536754 CC For-Sale Unstable CA9 19 41 COc1ccc(CNS(=O)(=O)c2c[nH]c(CO)c2)cc1 ZINC000217536754 CC For-Sale Unstable MMP1 19 41 C[C@@H]1CCCN([C@H](C)C(=O)c2ccc(Cl)cc2)C1 ZINC000217536793 CH For-Sale Unstable SLC6A1 44 48 C[C@@H]1CCCN([C@H](C)C(=O)c2ccc(Cl)cc2)C1 ZINC000217536793 CH For-Sale Unstable SLC6A3 18 48 C[C@@H]1CCCN([C@H](C)C(=O)c2ccc(Cl)cc2)C1 ZINC000217536793 CH For-Sale Unstable CCR1 41 38 CCCCc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217536814 GK For-Sale Unstable SCN2A 15 53 CCCCc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217536814 GK For-Sale Unstable S1PR4 19 41 CCCCc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217536814 GK For-Sale Unstable S1PR3 18 41 CCCCc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217536814 GK For-Sale Unstable S1PR2 42 41 CCCCc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217536814 GK For-Sale Unstable SPHK1 15 43 CCCCc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217536814 GK For-Sale Unstable CA9 15 47 CCCCc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217536814 GK For-Sale Unstable NCE103 27 47 CCCCc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217536814 GK For-Sale Unstable LIG1 0 41 CCCCc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217536814 GK For-Sale Unstable P96878_MYCTU 19 54 CCCCc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217536814 GK For-Sale Unstable ACAT 0 51 CCCCc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217536814 GK For-Sale Unstable PSBA 0 40 COc1cc2c(c(OC)c1OC)NC[C@@H](CN)[C@@H]2O ZINC000217536821 CC In-Stock Unstable DRTS_TOXGO 42 36 O=C([C@H]1CC(=O)N(c2ccc(Cl)cc2)C1)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217536829 HF In-Stock Unstable CHRNA4 28 45 CNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217536851 FD In-Stock Unstable CA2 26 43 CNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217536851 FD In-Stock Unstable BMP1 87 39 CNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217536851 FD In-Stock Unstable CA1 21 42 CNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217536851 FD In-Stock Unstable MMP13 53 39 CNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217536851 FD In-Stock Unstable MMP3 48 40 CNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217536851 FD In-Stock Unstable MMP9 41 40 CNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217536851 FD In-Stock Unstable CA12 16 40 CNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217536851 FD In-Stock Unstable MMP7 44 40 CNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217536851 FD In-Stock Unstable IAP 0 44 CNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217536851 FD In-Stock Unstable CA9 27 46 CNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217536851 FD In-Stock Unstable MMP1 58 39 CNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217536851 FD In-Stock Unstable AKR1C3 30 42 CNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217536851 FD In-Stock Unstable AKR1C2 54 40 O=C1OC2(CCN(C(=O)c3cc(-c4ccco4)[nH]n3)CC2)c2ccccc21 ZINC000217536868 FF For-Sale Unstable AVPR1A 15 50 O=C1OC2(CCN(C(=O)c3cc(-c4ccco4)[nH]n3)CC2)c2ccccc21 ZINC000217536868 FF For-Sale Unstable NPY5R 38 51 COc1ccc(N2C[C@H](C(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)CC2=O)cc1 ZINC000217536908 HD In-Stock Unstable CHRNA4 27 44 COc1cc2c(c(OC)c1OC)NC[C@H](CN)[C@@H]2O ZINC000217536915 CC In-Stock Unstable DRTS_TOXGO 42 36 C[C@@H]1CCCN([C@H](C)C(=O)c2ccc(F)cc2)C1 ZINC000217536925 BG For-Sale Unstable CCR3 42 38 CNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217536967 GD In-Stock Unstable PTGDR 22 41 CNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217536967 GD In-Stock Unstable IAP 0 45 CNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217536967 GD In-Stock Unstable SCMU_MYCTU 0 48 COc1cc2c(c(OC)c1OC)NC[C@@H](CN)[C@H]2O ZINC000217536984 CC In-Stock Unstable DRTS_TOXGO 42 36 O=C1OC2(CCN(C(=O)c3cccc(-n4cnnn4)c3)CC2)c2ccccc21 ZINC000217536989 GD For-Sale Unstable NPY5R 38 52 O=C1OC2(CCN(C(=O)c3cccc(-n4cnnn4)c3)CC2)c2ccccc21 ZINC000217536989 GD For-Sale Unstable KCNJ1 43 35 COc1ccc(N2C[C@@H](C(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)CC2=O)cc1 ZINC000217537002 HD In-Stock Unstable CHRNA4 27 44 CC(=O)Nc1cc(-c2cccc(F)c2)[nH]n1 ZINC000217537049 BE For-Sale Unstable GSK3A 19 46 CC(=O)Nc1cc(-c2cccc(F)c2)[nH]n1 ZINC000217537049 BE For-Sale Unstable HAO2 34 41 O=C(NCCc1ccc(O)cc1)NCCc1ccc(Br)cc1 ZINC000217537058 FG On-Demand Unstable HTT 0 43 O=C(NCCc1ccc(O)cc1)NCCc1ccc(Br)cc1 ZINC000217537058 FG On-Demand Unstable LIG1 0 45 O=C(NCCc1ccc(O)cc1)NCCc1ccc(Br)cc1 ZINC000217537058 FG On-Demand Unstable CAN2 0 41 COc1cc2c(c(OC)c1OC)NC[C@H](CN)[C@H]2O ZINC000217537070 CC In-Stock Unstable DRTS_TOXGO 42 36 CNS(=O)(=O)c1ccc(NC[C@@H]2CCCO2)c(C(=O)O)c1 ZINC000217537083 DC In-Stock Unstable BDKRB1 0 46 CNS(=O)(=O)c1ccc(NC[C@@H]2CCCO2)c(C(=O)O)c1 ZINC000217537083 DC In-Stock Unstable TNK2 35 46 COc1ccc(CCN)c(O)c1Br ZINC000217537089 BD For-Sale Unstable TAAR1 15 49 COc1cccc(-c2cc3ccc(O)c(CN4C[C@@H]5C[C@H](C4)c4cccc(=O)n4C5)c3oc2=O)c1 ZINC000217537098 JH In-Stock Unstable CHRNA4 28 45 O=C1OC2(CCN(C(=O)c3cc(-c4ccc5c(c4)OCO5)n[nH]3)CC2)c2ccccc21 ZINC000217537107 HG For-Sale Unstable AVPR1A 18 47 O=C1OC2(CCN(C(=O)c3cc(-c4ccc5c(c4)OCO5)n[nH]3)CC2)c2ccccc21 ZINC000217537107 HG For-Sale Unstable TACR3 21 42 O=C1OC2(CCN(C(=O)c3cc(-c4ccc5c(c4)OCO5)n[nH]3)CC2)c2ccccc21 ZINC000217537107 HG For-Sale Unstable NPY5R 40 57 CC(C)N(Cc1ccccc1)C(=O)NCCc1ccc(Br)cc1 ZINC000217537150 GJ On-Demand Unstable MME 41 36 CC(C)N(Cc1ccccc1)C(=O)NCCc1ccc(Br)cc1 ZINC000217537150 GJ On-Demand Unstable ANPEP 27 47 CC(C)N(Cc1ccccc1)C(=O)NCCc1ccc(Br)cc1 ZINC000217537150 GJ On-Demand Unstable CA1 15 41 CC(C)N(Cc1ccccc1)C(=O)NCCc1ccc(Br)cc1 ZINC000217537150 GJ On-Demand Unstable CPA1 16 40 CC(C)N(Cc1ccccc1)C(=O)NCCc1ccc(Br)cc1 ZINC000217537150 GJ On-Demand Unstable CA5B 16 41 CC(C)N(Cc1ccccc1)C(=O)NCCc1ccc(Br)cc1 ZINC000217537150 GJ On-Demand Unstable MMP2 28 41 CC(C)N(Cc1ccccc1)C(=O)NCCc1ccc(Br)cc1 ZINC000217537150 GJ On-Demand Unstable MMP3 35 40 CC(C)N(Cc1ccccc1)C(=O)NCCc1ccc(Br)cc1 ZINC000217537150 GJ On-Demand Unstable MMP8 22 40 CC(C)N(Cc1ccccc1)C(=O)NCCc1ccc(Br)cc1 ZINC000217537150 GJ On-Demand Unstable MMP9 20 40 CC(C)N(Cc1ccccc1)C(=O)NCCc1ccc(Br)cc1 ZINC000217537150 GJ On-Demand Unstable MMP1 24 40 CC(C)N(Cc1ccccc1)C(=O)NCCc1ccc(Br)cc1 ZINC000217537150 GJ On-Demand Unstable AMP1_PLAFQ 41 47 CC(C)N(Cc1ccccc1)C(=O)NCCc1ccc(Br)cc1 ZINC000217537150 GJ On-Demand Unstable PTGES 18 44 CC(C)N(Cc1ccccc1)C(=O)NCCc1ccc(Br)cc1 ZINC000217537150 GJ On-Demand Unstable LIMK2 40 36 CC(=O)Nc1n[nH]c(-c2cccc(F)c2)c1I ZINC000217537159 EF For-Sale Unstable GSK3A 26 45 CNS(=O)(=O)c1ccc(NC[C@H]2CCCO2)c(C(=O)O)c1 ZINC000217537167 DC In-Stock Unstable BDKRB1 0 46 CNS(=O)(=O)c1ccc(NC[C@H]2CCCO2)c(C(=O)O)c1 ZINC000217537167 DC In-Stock Unstable TNK2 35 46 O=C(Nc1ccc(I)cc1Cl)c1cccc(Cl)c1F ZINC000217537181 HJ On-Demand Anodyne GRM4 24 46 O=C(Nc1ccc(I)cc1Cl)c1cccc(Cl)c1F ZINC000217537181 HJ On-Demand Anodyne MAP2K1 22 44 O=C(Nc1ccc(I)cc1Cl)c1cccc(Cl)c1F ZINC000217537181 HJ On-Demand Anodyne EPHB3 47 38 O=C(Nc1ccc(I)cc1Cl)c1cccc(Cl)c1F ZINC000217537181 HJ On-Demand Anodyne SMO 17 40 O=C(Nc1ccc(I)cc1Cl)c1cccc(Cl)c1F ZINC000217537181 HJ On-Demand Anodyne Q25615_ONCVO 53 33 O=C(Nc1ccc(I)cc1Cl)c1cccc(Cl)c1F ZINC000217537181 HJ On-Demand Anodyne G2YM83_BOTF4 43 31 COc1ccccc1-c1cc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)[nH]n1 ZINC000217537207 HG For-Sale Unstable AVPR1A 15 48 COc1ccccc1-c1cc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)[nH]n1 ZINC000217537207 HG For-Sale Unstable ACACA 41 40 COc1ccccc1-c1cc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)[nH]n1 ZINC000217537207 HG For-Sale Unstable ACACB 23 40 COc1ccccc1-c1cc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)[nH]n1 ZINC000217537207 HG For-Sale Unstable TACR3 26 48 COc1ccccc1-c1cc(C(=O)N2CCC3(CC2)OC(=O)c2ccccc23)[nH]n1 ZINC000217537207 HG For-Sale Unstable NPY5R 46 58 COc1c(CCN)ccc(O)c1Br ZINC000217537211 BD For-Sale Unstable TAAR1 16 41 COc1cccc(/C=C2\Oc3c(ccc(O)c3CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)C2=O)c1OC ZINC000217537227 KH In-Stock Unstable CHRNA4 27 43 CN(C(=O)NCCc1ccc(Br)cc1)C1CCCCC1 ZINC000217537270 EH On-Demand Unstable GPBAR1 0 42 COc1cc(C(=O)Nc2ccc(I)cc2Cl)ccc1F ZINC000217537311 HI On-Demand Unstable F10 29 43 COc1cc(C(=O)Nc2ccc(I)cc2Cl)ccc1F ZINC000217537311 HI On-Demand Unstable COLA 79 37 COc1cc(C(=O)Nc2ccc(I)cc2Cl)ccc1F ZINC000217537311 HI On-Demand Unstable CPT1A 78 37 COc1cc(C(=O)Nc2ccc(I)cc2Cl)ccc1F ZINC000217537311 HI On-Demand Unstable CPT2 45 34 COc1cc(C(=O)Nc2ccc(I)cc2Cl)ccc1F ZINC000217537311 HI On-Demand Unstable PYGL 19 47 COc1cc(C(=O)Nc2ccc(I)cc2Cl)ccc1F ZINC000217537311 HI On-Demand Unstable KDR 18 40 COc1cc(C(=O)Nc2ccc(I)cc2Cl)ccc1F ZINC000217537311 HI On-Demand Unstable GRM4 26 44 COc1cc(C(=O)Nc2ccc(I)cc2Cl)ccc1F ZINC000217537311 HI On-Demand Unstable MAP2K1 36 42 COc1cc(C(=O)Nc2ccc(I)cc2Cl)ccc1F ZINC000217537311 HI On-Demand Unstable CPT1B 58 36 COc1cc(C(=O)Nc2ccc(I)cc2Cl)ccc1F ZINC000217537311 HI On-Demand Unstable PDGFRA 22 40 COc1cc(C(=O)Nc2ccc(I)cc2Cl)ccc1F ZINC000217537311 HI On-Demand Unstable FABH 0 43 COc1cc(C(=O)Nc2ccc(I)cc2Cl)ccc1F ZINC000217537311 HI On-Demand Unstable TAAR1 21 46 COc1cc(C(=O)Nc2ccc(I)cc2Cl)ccc1F ZINC000217537311 HI On-Demand Unstable SCD1 31 40 COc1cc(C(=O)Nc2ccc(I)cc2Cl)ccc1F ZINC000217537311 HI On-Demand Unstable SCD 20 40 COc1cc(C(=O)Nc2ccc(I)cc2Cl)ccc1F ZINC000217537311 HI On-Demand Unstable GPR35 42 38 O=C1OC2(CCN(C(=O)Cn3nnc4ccccc43)CC2)c2ccccc21 ZINC000217537313 FE For-Sale Unstable NPY5R 44 48 Cc1cc(CCN)c(O)c(Br)c1O ZINC000217537321 BD For-Sale Unstable TAAR1 17 42 NC(=O)c1ccc(/C=C\C(=O)NCC2CC(O)C2)cc1 ZINC000217537330 CC For-Sale Unstable HDAC1 23 40 NC(=O)c1ccc(/C=C\C(=O)NCC2CC(O)C2)cc1 ZINC000217537330 CC For-Sale Unstable IMA1 0 42 O=c1c(-c2ccccc2)coc2c(CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)c(O)ccc12 ZINC000217537358 IH In-Stock Unstable CHRNA4 31 55 COc1ccc(C(=O)[C@@H](C)N2CCC[C@@H](C)C2)cc1 ZINC000217537361 CF For-Sale Unstable ELANE 17 41 COc1ccc(C(=O)[C@@H](C)N2CCC[C@@H](C)C2)cc1 ZINC000217537361 CF For-Sale Unstable RORC 36 42 CC1CCN(C(=O)NCCc2ccc(Br)cc2)CC1 ZINC000217537397 EG On-Demand Unstable GPBAR1 23 43 COc1cccc(-c2cc(C(=O)N3CCC4(CC3)OC(=O)c3ccccc34)n(C)n2)c1 ZINC000217537420 HG For-Sale Unstable NPY5R 47 61 Cc1c(Cl)cccc1S(=O)(=O)NCC[C@H](O)c1ccsc1 ZINC000217537513 EG In-Stock Unstable ITGAV 19 42 O=C(O)C1CCN(C(=O)NCCc2ccc(Br)cc2)CC1 ZINC000217537522 FE On-Demand Unstable GPBAR1 31 44 Cc1ncn(CC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c(=O)c1C ZINC000217537539 FD In-Stock Unstable NPY5R 43 48 O=S(=O)(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc(Cl)s1 ZINC000217537543 HG For-Sale Unstable CCR4 50 33 Cc1c(Cl)cccc1S(=O)(=O)NCC[C@@H](O)c1ccsc1 ZINC000217537595 EG In-Stock Unstable ITGAV 19 42 O=C(NCCc1ccc(Br)cc1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217537631 JK For-Sale Unstable OPRD1 0 46 O=C(NCCc1ccc(Br)cc1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217537631 JK For-Sale Unstable OPRK1 0 46 O=C(NCCc1ccc(Br)cc1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217537631 JK For-Sale Unstable OPRL1 17 46 O=C(NCCc1ccc(Br)cc1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217537631 JK For-Sale Unstable NMUR2 0 58 O=C(NCCc1ccc(Br)cc1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217537631 JK For-Sale Unstable NMUR1 0 58 O=C1OC2(CCN(C(=O)c3cccc(I)c3)CC2)c2ccccc21 ZINC000217537651 IH For-Sale Unstable AVPR1A 15 52 O=C1OC2(CCN(C(=O)c3cccc(I)c3)CC2)c2ccccc21 ZINC000217537651 IH For-Sale Unstable NPY5R 43 50 O=C(O)c1ccccc1CN1CCCn2nc(CO)cc2C1 ZINC000217537659 DD In-Stock Unstable FABP4 45 34 O=C(N[C@@H]1CCN2CCCC[C@@H]12)c1ccc(Br)c(Cl)c1 ZINC000217537689 FG On-Demand Unstable VACHT_TETCF 0 41 O=C(N[C@@H]1CCN2CCCC[C@@H]12)c1ccc(Br)c(Cl)c1 ZINC000217537689 FG On-Demand Unstable SIGMAR1 0 50 O=C(N[C@@H]1CCN2CCCC[C@@H]12)c1ccc(Br)c(Cl)c1 ZINC000217537689 FG On-Demand Unstable L3MBTL3 54 33 CCOC(=O)Cn1nc(-c2ccccc2)cc1NC(C)=O ZINC000217537703 CE On-Demand Unstable P2RY12 57 38 CCOC(=O)Cn1nc(-c2ccccc2)cc1NC(C)=O ZINC000217537703 CE On-Demand Unstable GPR142 21 51 CCCNc1ccc(S(=O)(=O)NCC)cc1C(=O)O ZINC000217537712 CD In-Stock Unstable CASP3 0 41 CCCNc1ccc(S(=O)(=O)NCC)cc1C(=O)O ZINC000217537712 CD In-Stock Unstable BDKRB1 0 40 CCc1cc(N)c(O)c(Br)c1OC ZINC000217537754 BE For-Sale Unstable SLC22A12 44 36 O=C(NCCc1ccc(Br)cc1)N1CCCc2ccccc21 ZINC000217537756 FI For-Sale Unstable AVPR2 41 45 CCOc1ccccc1/C=C\C(=O)NC1CC(O)C1 ZINC000217537757 CD For-Sale Unstable PTGER2 0 40 CCOc1ccccc1/C=C\C(=O)NC1CC(O)C1 ZINC000217537757 CD For-Sale Unstable HCN1 46 30 O=C(N[C@H]1CCN2CCCC[C@@H]12)c1ccc(Br)c(Cl)c1 ZINC000217537765 FG On-Demand Unstable VACHT_TETCF 0 41 O=C(N[C@H]1CCN2CCCC[C@@H]12)c1ccc(Br)c(Cl)c1 ZINC000217537765 FG On-Demand Unstable SIGMAR1 0 50 O=C(N[C@H]1CCN2CCCC[C@@H]12)c1ccc(Br)c(Cl)c1 ZINC000217537765 FG On-Demand Unstable CHRNA7 15 41 O=C(N[C@H]1CCN2CCCC[C@@H]12)c1ccc(Br)c(Cl)c1 ZINC000217537765 FG On-Demand Unstable L3MBTL3 54 33 O=C(NCC(=O)N1CCC2(CC1)OC(=O)c1ccccc12)OCc1ccccc1 ZINC000217537768 GF For-Sale Unstable GHRHR 44 34 O=C(NCC(=O)N1CCC2(CC1)OC(=O)c1ccccc12)OCc1ccccc1 ZINC000217537768 GF For-Sale Unstable NPY5R 39 48 O=C(NCC(=O)N1CCC2(CC1)OC(=O)c1ccccc12)OCc1ccccc1 ZINC000217537768 GF For-Sale Unstable CAPN2 54 31 O=C(NCC(=O)N1CCC2(CC1)OC(=O)c1ccccc12)OCc1ccccc1 ZINC000217537768 GF For-Sale Unstable NPR 62 35 O=C(NCC(=O)N1CCC2(CC1)OC(=O)c1ccccc12)OCc1ccccc1 ZINC000217537768 GF For-Sale Unstable SLC12A5 57 34 CC(=O)c1cccc(S(=O)(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)c1 ZINC000217537785 HF For-Sale Unstable AKR1C3 17 41 Cc1c(-c2ccccc2)c(=O)oc2c(CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)c(O)ccc12 ZINC000217537793 JI In-Stock Unstable CHRNA4 30 52 Cc1ccc(Br)c(C(=O)N[C@@H]2CCN3CCCC[C@@H]23)c1 ZINC000217537852 EG On-Demand Unstable SIGMAR1 0 42 COc1ccc2cc(C(=O)N3CCC4(CC3)OC(=O)c3ccccc34)[nH]c2c1 ZINC000217537871 GG For-Sale Unstable AVPR1A 15 49 COc1ccc2cc(C(=O)N3CCC4(CC3)OC(=O)c3ccccc34)[nH]c2c1 ZINC000217537871 GG For-Sale Unstable GRIN2B 24 46 COc1ccc2cc(C(=O)N3CCC4(CC3)OC(=O)c3ccccc34)[nH]c2c1 ZINC000217537871 GG For-Sale Unstable HRH4 24 43 COc1ccc2cc(C(=O)N3CCC4(CC3)OC(=O)c3ccccc34)[nH]c2c1 ZINC000217537871 GG For-Sale Unstable NPY5R 35 51 COc1ccc2cc(C(=O)N3CCC4(CC3)OC(=O)c3ccccc34)[nH]c2c1 ZINC000217537871 GG For-Sale Unstable TUBB2B 31 40 COc1ccc2cc(C(=O)N3CCC4(CC3)OC(=O)c3ccccc34)[nH]c2c1 ZINC000217537871 GG For-Sale Unstable FPR2 17 41 CCCCOCCCNC(=O)NCCc1ccc(Br)cc1 ZINC000217537882 FG On-Demand Unstable EPHX2 31 40 Cc1ccc(Br)c(C(=O)N[C@H]2CCN3CCCC[C@@H]23)c1 ZINC000217537954 EG On-Demand Unstable SIGMAR1 0 42 COc1cc(NC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc(OC)c1OC ZINC000217537974 HG For-Sale Unstable NPY5R 70 65 CCCCNc1ccc(S(=O)(=O)NCC)cc1C(=O)O ZINC000217537975 DD In-Stock Unstable CASP3 15 42 CCCCNc1ccc(S(=O)(=O)NCC)cc1C(=O)O ZINC000217537975 DD In-Stock Unstable BDKRB1 0 41 O=C(NCCc1ccc(Br)cc1)N1CCC(Cc2ccccc2)CC1 ZINC000217538005 HJ For-Sale Unstable GRIN2B 94 44 O=C(NCCc1ccc(Br)cc1)N1CCC(Cc2ccccc2)CC1 ZINC000217538005 HJ For-Sale Unstable SIGMAR1 36 47 O=C(NCCc1ccc(Br)cc1)N1CCC(Cc2ccccc2)CC1 ZINC000217538005 HJ For-Sale Unstable CCR3 62 54 O=C(NCCc1ccc(Br)cc1)N1CCC(Cc2ccccc2)CC1 ZINC000217538005 HJ For-Sale Unstable EPHX2 19 43 O=C(NCCc1ccc(Br)cc1)N1CCC(Cc2ccccc2)CC1 ZINC000217538005 HJ For-Sale Unstable AMP1_PLAFQ 41 50 O=C(NCCc1ccc(Br)cc1)N1CCC(Cc2ccccc2)CC1 ZINC000217538005 HJ For-Sale Unstable GPBAR1 0 40 CCNS(=O)(=O)c1ccc(NCC(C)C)c(C(=O)O)c1 ZINC000217538067 DD In-Stock Unstable BDKRB1 0 43 CCNS(=O)(=O)c1ccc(NCC(C)C)c(C(=O)O)c1 ZINC000217538067 DD In-Stock Unstable MTNN 61 33 O=C1OC2(CCN(C(=O)Nc3ccc(Cl)c(Cl)c3)CC2)c2ccccc21 ZINC000217538079 GJ For-Sale Unstable CACNA1H 46 39 O=C1OC2(CCN(C(=O)Nc3ccc(Cl)c(Cl)c3)CC2)c2ccccc21 ZINC000217538079 GJ For-Sale Unstable NPY5R 85 66 O=C1OC2(CCN(C(=O)Nc3ccc(Cl)c(Cl)c3)CC2)c2ccccc21 ZINC000217538079 GJ For-Sale Unstable EPHX2 23 48 O=C1OC2(CCN(C(=O)Nc3ccc(Cl)c(Cl)c3)CC2)c2ccccc21 ZINC000217538079 GJ For-Sale Unstable TRPM8 32 45 CN1CCC(N(C)C(=O)NCCc2ccc(Br)cc2)CC1 ZINC000217538113 FF For-Sale Unstable GPBAR1 26 43 C=C1CC[C@@H](O[Si](C)(C)C(C)(C)C)C/C1=C\C=C1/CCC[C@@]2(C)[C@H]1CC[C@@H]2[C@H](C)CCCC(C)C ZINC000217538164 JK For-Sale Unstable VDR 178 69 C=C1CC[C@@H](O[Si](C)(C)C(C)(C)C)C/C1=C\C=C1/CCC[C@@]2(C)[C@H]1CC[C@@H]2[C@H](C)CCCC(C)C ZINC000217538164 JK For-Sale Unstable CDC25A 56 69 C=C1CC[C@@H](O[Si](C)(C)C(C)(C)C)C/C1=C\C=C1/CCC[C@@]2(C)[C@H]1CC[C@@H]2[C@H](C)CCCC(C)C ZINC000217538164 JK For-Sale Unstable CDC25B 51 49 C=C1CC[C@@H](O[Si](C)(C)C(C)(C)C)C/C1=C\C=C1/CCC[C@@]2(C)[C@H]1CC[C@@H]2[C@H](C)CCCC(C)C ZINC000217538164 JK For-Sale Unstable CYP24A1 39 51 O=C1/C(=C/c2ccccc2F)Oc2c1ccc(O)c2CN1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217538186 JH In-Stock Unstable CHRNA4 30 49 O=C1OC2(CCN(C(=O)Nc3ccccc3)CC2)c2ccccc21 ZINC000217538196 DG For-Sale Unstable NPY5R 87 74 O=C1OC2(CCN(C(=O)Nc3ccccc3)CC2)c2ccccc21 ZINC000217538196 DG For-Sale Unstable TRPM8 35 44 C[C@@H](NC(=O)NCCc1ccc(Br)cc1)c1ccccc1 ZINC000217538236 EI On-Demand Unstable MME 45 36 C[C@@H](NC(=O)NCCc1ccc(Br)cc1)c1ccccc1 ZINC000217538236 EI On-Demand Unstable ANPEP 46 45 C[C@@H](NC(=O)NCCc1ccc(Br)cc1)c1ccccc1 ZINC000217538236 EI On-Demand Unstable SDH1 0 46 C[C@@H](NC(=O)NCCc1ccc(Br)cc1)c1ccccc1 ZINC000217538236 EI On-Demand Unstable MMP2 22 42 C[C@@H](NC(=O)NCCc1ccc(Br)cc1)c1ccccc1 ZINC000217538236 EI On-Demand Unstable MMP3 34 42 C[C@@H](NC(=O)NCCc1ccc(Br)cc1)c1ccccc1 ZINC000217538236 EI On-Demand Unstable AMP1_PLAFQ 35 45 O=C1OC2(CCN(C(=O)Nc3ccc(Cl)cc3)CC2)c2ccccc21 ZINC000217538316 FI For-Sale Unstable CACNA1H 58 40 O=C1OC2(CCN(C(=O)Nc3ccc(Cl)cc3)CC2)c2ccccc21 ZINC000217538316 FI For-Sale Unstable NPY5R 79 71 O=C1OC2(CCN(C(=O)Nc3ccc(Cl)cc3)CC2)c2ccccc21 ZINC000217538316 FI For-Sale Unstable EPHX2 36 47 O=C1OC2(CCN(C(=O)Nc3ccc(Cl)cc3)CC2)c2ccccc21 ZINC000217538316 FI For-Sale Unstable TRPM8 36 47 C[C@H](NC(=O)NCCc1ccc(Br)cc1)c1ccccc1 ZINC000217538317 EI On-Demand Unstable MME 45 36 C[C@H](NC(=O)NCCc1ccc(Br)cc1)c1ccccc1 ZINC000217538317 EI On-Demand Unstable ANPEP 46 45 C[C@H](NC(=O)NCCc1ccc(Br)cc1)c1ccccc1 ZINC000217538317 EI On-Demand Unstable SDH1 0 46 C[C@H](NC(=O)NCCc1ccc(Br)cc1)c1ccccc1 ZINC000217538317 EI On-Demand Unstable MMP2 22 42 C[C@H](NC(=O)NCCc1ccc(Br)cc1)c1ccccc1 ZINC000217538317 EI On-Demand Unstable MMP3 34 42 C[C@H](NC(=O)NCCc1ccc(Br)cc1)c1ccccc1 ZINC000217538317 EI On-Demand Unstable AMP1_PLAFQ 35 45 CC(=O)N1CCN(C(=O)NCCc2ccc(Br)cc2)CC1 ZINC000217538420 FD For-Sale Unstable GPBAR1 0 40 CC(=O)N1CCN(C(=O)NCCc2ccc(Br)cc2)CC1 ZINC000217538420 FD For-Sale Unstable LIG1 0 42 CCCNC(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217538431 CE For-Sale Unstable NPY5R 58 56 CN(C)C[C@@]1(O)CCCN(C(=O)c2cccc(N3CCOCC3)c2)C1 ZINC000217538487 ED In-Stock Unstable AKR1C3 22 40 C[C@@H](NC(=O)NCc1ccccc1)C(=O)OC(C)(C)C ZINC000217538488 CE For-Sale Unstable CA2 21 43 C[C@@H](NC(=O)NCc1ccccc1)C(=O)OC(C)(C)C ZINC000217538488 CE For-Sale Unstable SSTR2 17 40 C[C@@H](NC(=O)NCc1ccccc1)C(=O)OC(C)(C)C ZINC000217538488 CE For-Sale Unstable MME 50 40 C[C@@H](NC(=O)NCc1ccccc1)C(=O)OC(C)(C)C ZINC000217538488 CE For-Sale Unstable ANPEP 45 52 C[C@@H](NC(=O)NCc1ccccc1)C(=O)OC(C)(C)C ZINC000217538488 CE For-Sale Unstable CA1 18 46 C[C@@H](NC(=O)NCc1ccccc1)C(=O)OC(C)(C)C ZINC000217538488 CE For-Sale Unstable CTSB 45 44 C[C@@H](NC(=O)NCc1ccccc1)C(=O)OC(C)(C)C ZINC000217538488 CE For-Sale Unstable PAPA1_CARPA 74 43 C[C@@H](NC(=O)NCc1ccccc1)C(=O)OC(C)(C)C ZINC000217538488 CE For-Sale Unstable CTSK 33 48 C[C@@H](NC(=O)NCc1ccccc1)C(=O)OC(C)(C)C ZINC000217538488 CE For-Sale Unstable CTSL 28 44 C[C@@H](NC(=O)NCc1ccccc1)C(=O)OC(C)(C)C ZINC000217538488 CE For-Sale Unstable CTRB1 45 38 C[C@@H](NC(=O)NCc1ccccc1)C(=O)OC(C)(C)C ZINC000217538488 CE For-Sale Unstable TACR3 17 43 C[C@@H](NC(=O)NCc1ccccc1)C(=O)OC(C)(C)C ZINC000217538488 CE For-Sale Unstable CA5B 17 42 C[C@@H](NC(=O)NCc1ccccc1)C(=O)OC(C)(C)C ZINC000217538488 CE For-Sale Unstable CA5A 19 42 C[C@@H](NC(=O)NCc1ccccc1)C(=O)OC(C)(C)C ZINC000217538488 CE For-Sale Unstable CAPNS1 52 33 C[C@@H](NC(=O)NCc1ccccc1)C(=O)OC(C)(C)C ZINC000217538488 CE For-Sale Unstable REN 31 41 C[C@@H](NC(=O)NCc1ccccc1)C(=O)OC(C)(C)C ZINC000217538488 CE For-Sale Unstable FURIN 43 34 C[C@@H](NC(=O)NCc1ccccc1)C(=O)OC(C)(C)C ZINC000217538488 CE For-Sale Unstable CTSS 17 44 C[C@@H](NC(=O)NCc1ccccc1)C(=O)OC(C)(C)C ZINC000217538488 CE For-Sale Unstable CAPN1 61 39 C[C@@H](NC(=O)NCc1ccccc1)C(=O)OC(C)(C)C ZINC000217538488 CE For-Sale Unstable CAPN2 75 38 C[C@@H](NC(=O)NCc1ccccc1)C(=O)OC(C)(C)C ZINC000217538488 CE For-Sale Unstable FPR1 65 42 C[C@@H](NC(=O)NCc1ccccc1)C(=O)OC(C)(C)C ZINC000217538488 CE For-Sale Unstable CTRB_BOVIN 56 37 C[C@@H](NC(=O)NCc1ccccc1)C(=O)OC(C)(C)C ZINC000217538488 CE For-Sale Unstable NPR 72 36 C[C@@H](NC(=O)NCc1ccccc1)C(=O)OC(C)(C)C ZINC000217538488 CE For-Sale Unstable AMP1_PLAFQ 53 41 C[C@@H](NC(=O)NCc1ccccc1)C(=O)OC(C)(C)C ZINC000217538488 CE For-Sale Unstable PDS 57 38 N#Cc1ccc(OC[C@@H](O)CN2CCC[C@@H](CO)C2)cc1 ZINC000217538496 CD On-Demand Unstable MEN1 44 38 O=C(NCCc1ccc(Br)cc1)NCc1ccc2c(c1)OCO2 ZINC000217538521 GG On-Demand Unstable BMP1 42 42 O=C(NCCc1ccc(Br)cc1)NCc1ccc2c(c1)OCO2 ZINC000217538521 GG On-Demand Unstable NOS2 96 36 O=C1OC2(CCN(C(=O)Nc3ccc(C(F)(F)F)cc3)CC2)c2ccccc21 ZINC000217538543 GI In-Stock Unstable TRPV1 20 49 O=C1OC2(CCN(C(=O)Nc3ccc(C(F)(F)F)cc3)CC2)c2ccccc21 ZINC000217538543 GI In-Stock Unstable NPY5R 69 63 O=C1OC2(CCN(C(=O)Nc3ccc(C(F)(F)F)cc3)CC2)c2ccccc21 ZINC000217538543 GI In-Stock Unstable EPHX2 60 50 O=C1OC2(CCN(C(=O)Nc3ccc(C(F)(F)F)cc3)CC2)c2ccccc21 ZINC000217538543 GI In-Stock Unstable TRPM8 81 60 CN(C)C[C@]1(O)CCCN(C(=O)c2cccc(N3CCOCC3)c2)C1 ZINC000217538562 ED In-Stock Unstable AKR1C3 22 40 O=C1/C(=C/c2ccccc2Cl)Oc2c1ccc(O)c2CN1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217538568 JI In-Stock Unstable CHRNA4 29 50 CCNS(=O)(=O)c1ccc(NC2CC2)c(C(=O)O)c1 ZINC000217538589 CD In-Stock Unstable SFRP1 42 33 O=c1cc(CO)n(CCO)cc1O ZINC000217538605 AB For-Sale Unstable COMT 52 49 C[C@@H](NC(=O)NCCc1ccc(Br)cc1)C12CC3CC(CC(C3)C1)C2 ZINC000217538633 HJ For-Sale Unstable EPHX2 38 61 CC(C)(C)NC(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217538666 DF For-Sale Unstable NPY5R 67 59 C[C@H](NC(=O)NCCc1ccc(Br)cc1)C12CC3CC(CC(C3)C1)C2 ZINC000217538710 HJ For-Sale Unstable EPHX2 38 61 COC(=O)c1ccc(/C=C2\Oc3c(ccc(O)c3CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)C2=O)cc1 ZINC000217538750 JH In-Stock Unstable CHRNA4 28 43 COc1cccc(NC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217538778 FG For-Sale Unstable DRD4 40 31 COc1cccc(NC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217538778 FG For-Sale Unstable NPY5R 80 71 COc1cccc(NC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217538778 FG For-Sale Unstable EPHX2 28 40 COc1cccc(NC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217538778 FG For-Sale Unstable TRPM8 28 41 COc1cccc(NC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217538778 FG For-Sale Unstable LIMK2 19 45 O=C(NCCc1ccc(Br)cc1)Nc1cccc2c(O)cccc12 ZINC000217538820 GJ For-Sale Unstable TRPV1 28 54 O=C(NCCc1ccc(Br)cc1)Nc1cccc2c(O)cccc12 ZINC000217538820 GJ For-Sale Unstable NCE103 26 42 COc1ccc(-c2c(C)oc3c(CN4C[C@@H]5C[C@H](C4)c4cccc(=O)n4C5)c(O)ccc3c2=O)cc1 ZINC000217538845 JI In-Stock Unstable CHRNA4 27 44 CC(C)(C)c1ccc(NC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217538891 GJ For-Sale Unstable TRPV1 24 48 CC(C)(C)c1ccc(NC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217538891 GJ For-Sale Unstable NPY5R 75 63 CC(C)(C)c1ccc(NC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217538891 GJ For-Sale Unstable EPHX2 38 41 CC(C)(C)c1ccc(NC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217538891 GJ For-Sale Unstable TRPM8 39 48 CN(CC(=O)NCC1(c2ccccc2)CCOCC1)[C@@H]1CCS(=O)(=O)C1 ZINC000217538909 GC In-Stock Unstable KCNA3 47 36 O=C(/C=C\c1ccc(F)c(Cl)c1)NC1CC(O)C1 ZINC000217538912 CE For-Sale Unstable HDAC8 22 44 O=C(/C=C\c1ccc(F)c(Cl)c1)NC1CC(O)C1 ZINC000217538912 CE For-Sale Unstable HDAC1 28 42 O=C(/C=C\c1ccc(F)c(Cl)c1)NC1CC(O)C1 ZINC000217538912 CE For-Sale Unstable HDAC2 17 45 O=C(/C=C\c1ccc(F)c(Cl)c1)NC1CC(O)C1 ZINC000217538912 CE For-Sale Unstable BOTA 30 43 CN(CC(=O)NCC1(c2ccccc2)CCOCC1)[C@H]1CCS(=O)(=O)C1 ZINC000217538988 GC In-Stock Unstable KCNA3 47 36 O=C1OC2(CCN(C(=O)NCCCl)CC2)c2ccccc21 ZINC000217539002 DE For-Sale Unstable NPY5R 51 56 CCNS(=O)(=O)c1ccc(NCCCO)c(C(=O)O)c1 ZINC000217539030 DC In-Stock Unstable CASP3 15 41 CCNS(=O)(=O)c1ccc(NCCCO)c(C(=O)O)c1 ZINC000217539030 DC In-Stock Unstable BDKRB1 0 41 O=C(O)CNC(=O)NCCc1ccc(Br)cc1 ZINC000217539031 DD For-Sale Unstable LIG1 0 43 COc1ccc(N2C[C@H](C(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)CC2=O)cc1Cl ZINC000217539086 IF In-Stock Unstable CHRNA4 25 41 CCCCOc1ccc(NC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217539118 GJ For-Sale Unstable PDGFRB 42 40 CCCCOc1ccc(NC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217539118 GJ For-Sale Unstable FAAH 27 44 CCCCOc1ccc(NC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217539118 GJ For-Sale Unstable NPY5R 68 60 CCCCOc1ccc(NC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217539118 GJ For-Sale Unstable EPHX2 39 44 CCCCOc1ccc(NC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217539118 GJ For-Sale Unstable TRPM8 29 42 CCNS(=O)(=O)c1ccc(NCCOC)c(C(=O)O)c1 ZINC000217539153 DC In-Stock Unstable BDKRB1 0 42 O=C(NCCc1ccc(Br)cc1)N(CCO)CCO ZINC000217539160 EC For-Sale Unstable LIG1 0 44 CNCCc1ccc(F)c(Br)c1C ZINC000217539163 BF For-Sale Unstable TAAR1 15 52 COc1ccc(N2C[C@@H](C(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)CC2=O)cc1Cl ZINC000217539173 IF In-Stock Unstable CHRNA4 25 41 O=C1OC2(CCN(C(=O)Nc3cccc(Cl)c3)CC2)c2ccccc21 ZINC000217539234 FI For-Sale Unstable CACNA1H 54 42 O=C1OC2(CCN(C(=O)Nc3cccc(Cl)c3)CC2)c2ccccc21 ZINC000217539234 FI For-Sale Unstable NPY5R 77 69 O=C1OC2(CCN(C(=O)Nc3cccc(Cl)c3)CC2)c2ccccc21 ZINC000217539234 FI For-Sale Unstable TRPM8 34 43 C[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539256 DD For-Sale Unstable MME 30 48 C[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539256 DD For-Sale Unstable ANPEP 32 48 C[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539256 DD For-Sale Unstable SLC15A1 0 41 C[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539256 DD For-Sale Unstable AMP1_PLAFQ 16 42 C[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539256 DD For-Sale Unstable SLC15A2 0 43 C[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539256 DD For-Sale Unstable LIG1 0 40 CNCCc1cc(C)c(Br)cc1F ZINC000217539258 BF For-Sale Unstable TAAR1 15 47 CCNS(=O)(=O)c1ccc(NCCCOC)c(C(=O)O)c1 ZINC000217539262 DD In-Stock Unstable BDKRB1 0 43 O=C(/C=C\c1cc(Br)ccc1F)NC1CC(O)C1 ZINC000217539280 DE For-Sale Unstable BOTA 25 44 CCOc1ccc(NC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217539325 FH For-Sale Unstable NPY5R 77 62 CN1CCCN(C[C@@H](O)COCc2ccccc2)CC1 ZINC000217539334 CD On-Demand Unstable MC4R 27 44 CN1CCCN(C[C@@H](O)COCc2ccccc2)CC1 ZINC000217539334 CD On-Demand Unstable PLK1 0 43 CN1CCCN(C[C@@H](O)COCc2ccccc2)CC1 ZINC000217539334 CD On-Demand Unstable CYP2D6 0 41 CN1CCCN(C[C@@H](O)COCc2ccccc2)CC1 ZINC000217539334 CD On-Demand Unstable ABCB1 70 44 CN1CCCN(C[C@@H](O)COCc2ccccc2)CC1 ZINC000217539334 CD On-Demand Unstable HSP90AB1 38 44 C[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539345 DD For-Sale Unstable MME 30 48 C[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539345 DD For-Sale Unstable ANPEP 32 48 C[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539345 DD For-Sale Unstable SLC15A1 0 41 C[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539345 DD For-Sale Unstable AMP1_PLAFQ 16 42 C[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539345 DD For-Sale Unstable SLC15A2 0 43 C[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539345 DD For-Sale Unstable LIG1 0 40 CCNS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217539369 EE In-Stock Unstable GNRHR 16 40 CCNS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217539369 EE In-Stock Unstable AKR1C3 22 42 Cc1ccc(/C=C\C(=O)NC2CC(O)C2)c(C)c1 ZINC000217539406 BD For-Sale Unstable BOTA 27 48 O=C1OC2(CCN(C(=O)Nc3ccccc3Cl)CC2)c2ccccc21 ZINC000217539424 FI For-Sale Unstable NPY5R 79 70 O=C1OC2(CCN(C(=O)Nc3ccccc3Cl)CC2)c2ccccc21 ZINC000217539424 FI For-Sale Unstable EPHB3 42 34 O=C1OC2(CCN(C(=O)Nc3ccccc3Cl)CC2)c2ccccc21 ZINC000217539424 FI For-Sale Unstable TRPM8 26 45 O=C1OC2(CCN(C(=O)Nc3ccccc3Cl)CC2)c2ccccc21 ZINC000217539424 FI For-Sale Unstable SMO 27 44 O=C(O)CCCCCNC(=O)NCCc1ccc(Br)cc1 ZINC000217539432 FF On-Demand Unstable HDAC9 34 49 O=C(O)CCCCCNC(=O)NCCc1ccc(Br)cc1 ZINC000217539432 FF On-Demand Unstable HDA106 0 42 O=C(O)CCCCCNC(=O)NCCc1ccc(Br)cc1 ZINC000217539432 FF On-Demand Unstable FFAR1 24 44 O=C(O)CCCCCNC(=O)NCCc1ccc(Br)cc1 ZINC000217539432 FF On-Demand Unstable LIG1 0 42 C[C@@H]1CN(C[C@@H](N)c2ccc3c(c2)OCO3)CCCO1 ZINC000217539461 CD For-Sale Unstable SSTR3 101 35 CCNS(=O)(=O)c1ccc(N[C@@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217539472 EF In-Stock Unstable BDKRB1 26 41 COc1ccc(C)cc1/C=C\C(=O)NC1CC(O)C1 ZINC000217539513 CD For-Sale Unstable CYSP_PLAFA 42 37 CC[C@@H](O)CCNC(=O)NCc1ccccc1 ZINC000217539521 BD On-Demand Unstable DNPEP 0 42 CC[C@@H](O)CCNC(=O)NCc1ccccc1 ZINC000217539521 BD On-Demand Unstable POL 0 41 Cc1c(C(=O)O)sc2nc(N)nc(Cl)c12 ZINC000217539529 BD For-Sale Unstable CHRM4 30 40 C[C@H]1CN(C[C@@H](N)c2ccc3c(c2)OCO3)CCCO1 ZINC000217539543 CD For-Sale Unstable SSTR3 101 35 COCCNC(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217539545 DD For-Sale Unstable NPY5R 52 56 CC(C)[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539556 EE For-Sale Unstable ANPEP 22 40 CC(C)[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539556 EE For-Sale Unstable MMP2 18 44 CC(C)[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539556 EE For-Sale Unstable MMP3 21 44 CC(C)[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539556 EE For-Sale Unstable LIG1 0 41 CCNS(=O)(=O)c1ccc(N[C@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217539558 EF In-Stock Unstable BDKRB1 26 41 CC[C@H](O)CCNC(=O)NCc1ccccc1 ZINC000217539604 BD On-Demand Unstable DNPEP 0 42 CC[C@H](O)CCNC(=O)NCc1ccccc1 ZINC000217539604 BD On-Demand Unstable POL 0 41 O=C(NCCCn1ccccc1=O)c1ccc2cc[nH]c2c1 ZINC000217539606 CE In-Stock Unstable DRD2 22 41 O=C(NCCCn1ccccc1=O)c1ccc2cc[nH]c2c1 ZINC000217539606 CE In-Stock Unstable DRD4 40 31 O=C(NCCCn1ccccc1=O)c1ccc2cc[nH]c2c1 ZINC000217539606 CE In-Stock Unstable DRD3 44 41 O=C(NCCCn1ccccc1=O)c1ccc2cc[nH]c2c1 ZINC000217539606 CE In-Stock Unstable PLD1 62 41 O=C(NCCCn1ccccc1=O)c1ccc2cc[nH]c2c1 ZINC000217539606 CE In-Stock Unstable HDAC9 15 44 O=C(NCCCn1ccccc1=O)c1ccc2cc[nH]c2c1 ZINC000217539606 CE In-Stock Unstable PLD2 88 42 C[C@@H]1CN([C@@H]2C[C@@H](c3ccccc3)CC[C@@H]2N)CCCO1 ZINC000217539613 CF For-Sale Unstable SLC18A3 49 39 CC(C)[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539652 EE For-Sale Unstable ANPEP 22 40 CC(C)[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539652 EE For-Sale Unstable MMP2 18 44 CC(C)[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539652 EE For-Sale Unstable MMP3 21 44 CC(C)[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539652 EE For-Sale Unstable LIG1 0 41 O=C1OC2(CCN(C(=O)NC3CCCC3)CC2)c2ccccc21 ZINC000217539658 DF For-Sale Unstable NPY5R 65 58 O=C1OC2(CCN(C(=O)NC3CCCC3)CC2)c2ccccc21 ZINC000217539658 DF For-Sale Unstable EPHX2 23 52 CCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217539672 EE In-Stock Unstable CA2 27 40 CCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217539672 EE In-Stock Unstable TBXA2R 50 39 CCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217539672 EE In-Stock Unstable CA4 20 40 CCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217539672 EE In-Stock Unstable AKR1C3 16 51 CSCC[C@@H](O)C(=O)NCCc1cccnc1 ZINC000217539769 CC In-Stock Unstable TBXAS1 35 40 CSCC[C@@H](O)C(=O)NCCc1cccnc1 ZINC000217539769 CC In-Stock Unstable PTAFR 30 42 O=C(O)CCCNC(=O)NCCc1ccc(Br)cc1 ZINC000217539771 EE On-Demand Unstable FFAR1 35 47 O=C(O)CCCNC(=O)NCCc1ccc(Br)cc1 ZINC000217539771 EE On-Demand Unstable LIG1 0 44 Cc1ccc(NC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1C ZINC000217539774 FH For-Sale Unstable NPY5R 80 62 CCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217539776 GE In-Stock Unstable CA2 21 41 CCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217539776 GE In-Stock Unstable TBXA2R 34 42 CCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217539776 GE In-Stock Unstable BMP1 63 38 CCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217539776 GE In-Stock Unstable CA1 22 44 CCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217539776 GE In-Stock Unstable MMP13 57 41 CCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217539776 GE In-Stock Unstable MMP2 35 41 CCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217539776 GE In-Stock Unstable MMP3 45 37 CCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217539776 GE In-Stock Unstable MMP8 27 41 CCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217539776 GE In-Stock Unstable MMP14 16 41 CCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217539776 GE In-Stock Unstable MMP9 49 41 CCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217539776 GE In-Stock Unstable MMP12 26 41 CCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217539776 GE In-Stock Unstable PTGDR 25 43 CCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217539776 GE In-Stock Unstable CA9 25 44 CCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217539776 GE In-Stock Unstable MMP1 51 38 CCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217539776 GE In-Stock Unstable AKR1C3 30 45 CCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217539776 GE In-Stock Unstable AKR1C2 52 38 CSCC[C@H](O)C(=O)NCCc1cccnc1 ZINC000217539853 CC In-Stock Unstable TBXAS1 43 40 CSCC[C@H](O)C(=O)NCCc1cccnc1 ZINC000217539853 CC In-Stock Unstable PTAFR 33 42 O=S(=O)(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc2ccccc2c1 ZINC000217539863 HH For-Sale Unstable HTR7 25 51 O=S(=O)(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc2ccccc2c1 ZINC000217539863 HH For-Sale Unstable NPY1R 21 42 O=S(=O)(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1ccc2ccccc2c1 ZINC000217539863 HH For-Sale Unstable TRY2_BOVIN 61 39 CC(C)C[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539888 FF For-Sale Unstable ACE 25 42 CC(C)C[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539888 FF For-Sale Unstable FOLH1 43 53 CC(C)C[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539888 FF For-Sale Unstable MME 55 45 CC(C)C[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539888 FF For-Sale Unstable LTA4H 27 42 CC(C)C[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539888 FF For-Sale Unstable ANPEP 59 50 CC(C)C[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539888 FF For-Sale Unstable RNPEP 25 42 CC(C)C[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539888 FF For-Sale Unstable CTSB 25 42 CC(C)C[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539888 FF For-Sale Unstable CTSK 28 48 CC(C)C[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539888 FF For-Sale Unstable CTSL 25 42 CC(C)C[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539888 FF For-Sale Unstable NAALAD2 44 39 CC(C)C[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539888 FF For-Sale Unstable CAPNS1 49 40 CC(C)C[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539888 FF For-Sale Unstable MMP2 24 47 CC(C)C[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539888 FF For-Sale Unstable MMP3 44 47 CC(C)C[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539888 FF For-Sale Unstable PAM 0 40 CC(C)C[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539888 FF For-Sale Unstable CAPN1 53 42 CC(C)C[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539888 FF For-Sale Unstable CAPN2 75 40 CC(C)C[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539888 FF For-Sale Unstable LAP3 18 42 CC(C)C[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539888 FF For-Sale Unstable MMP1 22 41 CC(C)C[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539888 FF For-Sale Unstable FPR1 74 49 CC(C)C[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539888 FF For-Sale Unstable NPR 75 41 CC(C)C[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539888 FF For-Sale Unstable AMP1_PLAFQ 37 47 CC(C)C[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539888 FF For-Sale Unstable AMPX_VIBPR 0 42 CC(C)C[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539888 FF For-Sale Unstable SLC15A2 0 40 COc1cc(NC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc(OC)c1 ZINC000217539890 GG For-Sale Unstable NPY5R 78 65 COc1cc(NC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc(OC)c1 ZINC000217539890 GG For-Sale Unstable S1PR2 29 41 COc1cc(NC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc(OC)c1 ZINC000217539890 GG For-Sale Unstable TRPM8 27 40 CCNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217539893 HE In-Stock Unstable PTGDR 20 40 CCNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217539893 HE In-Stock Unstable IAP 0 46 CCNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217539893 HE In-Stock Unstable SCMU_MYCTU 0 46 Cn1c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)nc2cc([N+](=O)[O-])ccc21 ZINC000217539917 GE In-Stock Unstable CHRNA4 30 49 CCOC(=O)[C@@H]1CNc2c(OC)cccc2[C@@H]1O ZINC000217539946 CD In-Stock Unstable DHFR-TS 0 46 CC(C)C[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539970 FF For-Sale Unstable ACE 25 42 CC(C)C[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539970 FF For-Sale Unstable FOLH1 43 53 CC(C)C[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539970 FF For-Sale Unstable MME 55 45 CC(C)C[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539970 FF For-Sale Unstable LTA4H 27 42 CC(C)C[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539970 FF For-Sale Unstable ANPEP 59 50 CC(C)C[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539970 FF For-Sale Unstable RNPEP 25 42 CC(C)C[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539970 FF For-Sale Unstable CTSB 25 42 CC(C)C[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539970 FF For-Sale Unstable CTSK 28 48 CC(C)C[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539970 FF For-Sale Unstable CTSL 25 42 CC(C)C[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539970 FF For-Sale Unstable NAALAD2 44 39 CC(C)C[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539970 FF For-Sale Unstable CAPNS1 49 40 CC(C)C[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539970 FF For-Sale Unstable MMP2 24 47 CC(C)C[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539970 FF For-Sale Unstable MMP3 44 47 CC(C)C[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539970 FF For-Sale Unstable PAM 0 40 CC(C)C[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539970 FF For-Sale Unstable CAPN1 53 42 CC(C)C[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539970 FF For-Sale Unstable CAPN2 75 40 CC(C)C[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539970 FF For-Sale Unstable LAP3 18 42 CC(C)C[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539970 FF For-Sale Unstable MMP1 22 41 CC(C)C[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539970 FF For-Sale Unstable FPR1 74 49 CC(C)C[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539970 FF For-Sale Unstable NPR 75 41 CC(C)C[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539970 FF For-Sale Unstable AMP1_PLAFQ 37 47 CC(C)C[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539970 FF For-Sale Unstable AMPX_VIBPR 0 42 CC(C)C[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217539970 FF For-Sale Unstable SLC15A2 0 40 O=S(=O)(NCCn1nc(C(F)(F)F)c2c1CCCC2)c1cccc2ccccc12 ZINC000217539976 HH For-Sale Unstable NPY2R 40 41 COc1ccc(NC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217540001 FG For-Sale Unstable PDGFRB 39 40 COc1ccc(NC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217540001 FG For-Sale Unstable NPY5R 76 63 COc1ccc(NC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217540001 FG For-Sale Unstable TRPM8 33 46 CCOC(=O)[C@H]1CNc2c(OC)cccc2[C@@H]1O ZINC000217540030 CD In-Stock Unstable DHFR-TS 0 46 O=C1CCc2cc(S(=O)(=O)NCC[C@@H](O)c3ccsc3)cc3c2N1CC3 ZINC000217540035 GD In-Stock Unstable CYP11B1 27 42 O=C1CCc2cc(S(=O)(=O)NCC[C@@H](O)c3ccsc3)cc3c2N1CC3 ZINC000217540035 GD In-Stock Unstable CYP11B2 27 42 CSCC[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217540083 GE For-Sale Unstable FOLH1 56 48 CSCC[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217540083 GE For-Sale Unstable MME 17 50 CSCC[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217540083 GE For-Sale Unstable LTA4H 0 40 CSCC[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217540083 GE For-Sale Unstable NAALAD2 54 36 CSCC[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217540083 GE For-Sale Unstable PAM 0 46 CSCC[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217540083 GE For-Sale Unstable FPR1 41 39 CSCC[C@@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217540083 GE For-Sale Unstable SLC15A2 0 43 CCNS(=O)(=O)c1ccc(NC[C@@H]2CCCO2)c(C(=O)O)c1 ZINC000217540110 ED In-Stock Unstable BDKRB1 23 44 O=C1CCc2cc(S(=O)(=O)NCC[C@H](O)c3ccsc3)cc3c2N1CC3 ZINC000217540113 GD In-Stock Unstable CYP11B1 27 42 O=C1CCc2cc(S(=O)(=O)NCC[C@H](O)c3ccsc3)cc3c2N1CC3 ZINC000217540113 GD In-Stock Unstable CYP11B2 27 42 CCOC(=O)[C@@H]1CNc2c(OC)cccc2[C@H]1O ZINC000217540117 CD In-Stock Unstable DHFR-TS 0 46 COc1ccc(CNC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217540118 FG For-Sale Unstable MMP13 21 43 COc1ccc(CNC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217540118 FG For-Sale Unstable NPY5R 47 56 COc1ccc(CNC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217540118 FG For-Sale Unstable MMP9 15 43 CCNS(=O)(=O)c1ccc(NC[C@H]2CCCO2)c(C(=O)O)c1 ZINC000217540182 ED In-Stock Unstable BDKRB1 23 44 CSCC[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217540188 GE For-Sale Unstable FOLH1 56 48 CSCC[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217540188 GE For-Sale Unstable MME 17 50 CSCC[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217540188 GE For-Sale Unstable LTA4H 0 40 CSCC[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217540188 GE For-Sale Unstable NAALAD2 54 36 CSCC[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217540188 GE For-Sale Unstable PAM 0 46 CSCC[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217540188 GE For-Sale Unstable FPR1 41 39 CSCC[C@H](NC(=O)NCCc1ccc(Br)cc1)C(=O)O ZINC000217540188 GE For-Sale Unstable SLC15A2 0 43 CCOC(=O)[C@H]1CNc2c(OC)cccc2[C@H]1O ZINC000217540190 CD In-Stock Unstable DHFR-TS 0 46 Cc1ccc(NC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217540198 EH For-Sale Unstable NPY5R 83 69 Cc1ccc(NC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217540198 EH For-Sale Unstable EPHX2 32 41 Cc1ccc(NC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217540198 EH For-Sale Unstable TRPM8 31 52 C[C@H]1C[C@@H](C)CN([C@H](C)C(=O)c2ccc(Cl)cc2)C1 ZINC000217540209 CH For-Sale Unstable SLC6A1 25 43 O=C1CCN(C(=O)[C@@H]2CCc3ccccc3C2)CCN1 ZINC000217540220 CD In-Stock Unstable PREP 45 43 COc1ccc([C@@H](C)NC(=O)NCCc2ccc(Br)cc2)cc1OC ZINC000217540288 HI On-Demand Unstable SDH1 0 43 COc1ccc([C@@H](C)NC(=O)NCCc2ccc(Br)cc2)cc1OC ZINC000217540288 HI On-Demand Unstable TRPV1 25 40 COc1ccc([C@@H](C)NC(=O)NCCc2ccc(Br)cc2)cc1OC ZINC000217540288 HI On-Demand Unstable CAN2 0 44 C[C@@H]1C[C@@H](C)CN([C@H](C)C(=O)c2ccc(Cl)cc2)C1 ZINC000217540292 CH For-Sale Unstable SLC6A1 25 43 CCNS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217540298 DD In-Stock Unstable KCNQ2 69 34 CCNS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217540298 DD In-Stock Unstable PNMT 15 41 CCNS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217540298 DD In-Stock Unstable SLC6A9 20 46 CCNS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217540298 DD In-Stock Unstable SFRP1 63 33 CCNS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217540298 DD In-Stock Unstable WNT3 54 33 O=C1CCN(C(=O)[C@H]2CCc3ccccc3C2)CCN1 ZINC000217540316 CD In-Stock Unstable PREP 45 43 O=C1OC2(CCN(C(=O)NCCCc3ccccc3)CC2)c2ccccc21 ZINC000217540336 FG For-Sale Unstable GHRHR 44 36 O=C1OC2(CCN(C(=O)NCCCc3ccccc3)CC2)c2ccccc21 ZINC000217540336 FG For-Sale Unstable SIGMAR1 25 56 O=C1OC2(CCN(C(=O)NCCCc3ccccc3)CC2)c2ccccc21 ZINC000217540336 FG For-Sale Unstable NPY5R 50 57 CC(C)(C)OC(=O)N1CCC[C@H](Oc2ccc(C(N)=O)cc2[N+](=O)[O-])C1 ZINC000217540345 FE For-Sale Unstable GPR119 26 45 COc1ccc([C@H](C)NC(=O)NCCc2ccc(Br)cc2)cc1OC ZINC000217540381 HI On-Demand Unstable SDH1 0 43 COc1ccc([C@H](C)NC(=O)NCCc2ccc(Br)cc2)cc1OC ZINC000217540381 HI On-Demand Unstable TRPV1 25 40 COc1ccc([C@H](C)NC(=O)NCCc2ccc(Br)cc2)cc1OC ZINC000217540381 HI On-Demand Unstable CAN2 0 44 CCNS(=O)(=O)c1ccc(NCCCOCC)c(C(=O)O)c1 ZINC000217540401 ED In-Stock Unstable BDKRB1 15 40 CC(=O)Nc1ccc(S(=O)(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc1 ZINC000217540428 IF For-Sale Unstable IDO1 28 40 COc1ccc([C@@H](C)NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217540453 GI On-Demand Unstable SDH1 0 45 COc1ccc([C@@H](C)NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217540453 GI On-Demand Unstable BMP1 34 46 COc1ccc([C@@H](C)NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217540453 GI On-Demand Unstable ACACA 60 45 COc1ccc([C@@H](C)NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217540453 GI On-Demand Unstable ACACB 23 44 COc1ccc([C@@H](C)NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217540453 GI On-Demand Unstable MTNR1A 52 39 COc1ccc([C@@H](C)NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217540453 GI On-Demand Unstable MTNR1B 42 38 COc1ccc([C@@H](C)NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217540453 GI On-Demand Unstable CA9 15 44 COc1ccc([C@@H](C)NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217540453 GI On-Demand Unstable DXR 18 40 COc1ccccc1NC(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217540455 FG For-Sale Unstable NPY5R 75 72 COc1ccccc1NC(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217540455 FG For-Sale Unstable RBP4 26 41 Cc1ccc(OC[C@H](O)CN[C@@H]2CCC[C@@H](C)[C@@H]2C)cc1 ZINC000217540471 CG On-Demand Unstable ADRB2 41 42 Cc1ccc(OC[C@H](O)CN[C@@H]2CCC[C@@H](C)[C@@H]2C)cc1 ZINC000217540471 CG On-Demand Unstable ADRB1 27 42 CCNS(=O)(=O)c1ccc(NCCCOC(C)C)c(C(=O)O)c1 ZINC000217540507 ED In-Stock Unstable BDKRB1 15 40 CN(Cc1nc2ccccc2c(=O)[nH]1)C(=O)c1ccc(C#CC(C)(C)O)cc1 ZINC000217540513 GE In-Stock Unstable WNT3A 18 40 CC(=O)Nc1ccc2c(c1)nc(CN1C[C@@H]3C[C@H](C1)c1cccc(=O)n1C3)n2C ZINC000217540516 GE In-Stock Unstable CHRNA4 31 52 COc1ccc([C@H](C)NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217540531 GI On-Demand Unstable SDH1 0 45 COc1ccc([C@H](C)NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217540531 GI On-Demand Unstable BMP1 34 46 COc1ccc([C@H](C)NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217540531 GI On-Demand Unstable ACACA 60 45 COc1ccc([C@H](C)NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217540531 GI On-Demand Unstable ACACB 23 44 COc1ccc([C@H](C)NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217540531 GI On-Demand Unstable MTNR1A 52 39 COc1ccc([C@H](C)NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217540531 GI On-Demand Unstable MTNR1B 42 38 COc1ccc([C@H](C)NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217540531 GI On-Demand Unstable CA9 15 44 COc1ccc([C@H](C)NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217540531 GI On-Demand Unstable DXR 18 40 C[C@@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217540552 CD On-Demand Unstable SLC6A1 51 37 C[C@@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217540552 CD On-Demand Unstable PRCP 27 45 C[C@@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217540552 CD On-Demand Unstable CCR3 44 34 C[C@@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217540552 CD On-Demand Unstable CCR5 32 40 C[C@@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217540552 CD On-Demand Unstable F11 41 36 C[C@@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217540552 CD On-Demand Unstable XIAP 50 38 C[C@@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217540552 CD On-Demand Unstable BIRC2 56 42 C[C@@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217540552 CD On-Demand Unstable BIRC8 53 33 COc1ccc(NC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c(OC)c1 ZINC000217540581 GG For-Sale Unstable NPY5R 76 66 C[C@@H]1CN(C[C@@H](N)c2ccc(C(C)(C)C)cc2)CCCO1 ZINC000217540589 CG For-Sale Unstable LOC100281352 0 42 C[C@@H]1CN(C[C@@H](N)c2ccc(C(C)(C)C)cc2)CCCO1 ZINC000217540589 CG For-Sale Unstable ZM.86993 0 42 C[C@@H]1CN(C[C@@H](N)c2ccc(C(C)(C)C)cc2)CCCO1 ZINC000217540589 CG For-Sale Unstable Q2TU57_MAIZE 21 42 CCCCCNc1ccc(S(=O)(=O)NCC)cc1C(=O)O ZINC000217540617 DE In-Stock Unstable CASP3 15 43 CCCCCNc1ccc(S(=O)(=O)NCC)cc1C(=O)O ZINC000217540617 DE In-Stock Unstable BDKRB1 0 41 C[C@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217540638 CD On-Demand Unstable SLC6A1 51 37 C[C@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217540638 CD On-Demand Unstable PRCP 27 45 C[C@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217540638 CD On-Demand Unstable CCR3 44 34 C[C@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217540638 CD On-Demand Unstable CCR5 32 40 C[C@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217540638 CD On-Demand Unstable F11 41 36 C[C@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217540638 CD On-Demand Unstable XIAP 50 38 C[C@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217540638 CD On-Demand Unstable BIRC2 56 42 C[C@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217540638 CD On-Demand Unstable BIRC8 53 33 COc1cccc(NC(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1OC ZINC000217540666 GG For-Sale Unstable NPY5R 64 67 C[C@H]1CN(C[C@@H](N)c2ccc(C(C)(C)C)cc2)CCCO1 ZINC000217540685 CG For-Sale Unstable LOC100281352 0 42 C[C@H]1CN(C[C@@H](N)c2ccc(C(C)(C)C)cc2)CCCO1 ZINC000217540685 CG For-Sale Unstable ZM.86993 0 42 C[C@H]1CN(C[C@@H](N)c2ccc(C(C)(C)C)cc2)CCCO1 ZINC000217540685 CG For-Sale Unstable Q2TU57_MAIZE 21 42 CCNS(=O)(=O)c1ccc(NCCC(C)C)c(C(=O)O)c1 ZINC000217540737 DE In-Stock Unstable CASP3 15 42 CCNS(=O)(=O)c1ccc(NCCC(C)C)c(C(=O)O)c1 ZINC000217540737 DE In-Stock Unstable BDKRB1 0 40 O=C1OC2(CCN(S(=O)(=O)C3CC3)CC2)c2ccccc21 ZINC000217540786 DD For-Sale Unstable NPY5R 48 43 Cc1cccc(OC[C@H](O)CN[C@@H]2CCC[C@@H](C)[C@@H]2C)c1 ZINC000217540794 CG On-Demand Unstable ADRB2 39 58 Cc1cccc(OC[C@H](O)CN[C@@H]2CCC[C@@H](C)[C@@H]2C)c1 ZINC000217540794 CG On-Demand Unstable ADRB1 26 58 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NCC)cc1C(=O)O ZINC000217540867 DE In-Stock Unstable CASP3 15 41 CC(C)S(=O)(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217540883 DD For-Sale Unstable NPY5R 34 45 CCC[C@H](C)Nc1ccc(S(=O)(=O)NCC)cc1C(=O)O ZINC000217540954 DE In-Stock Unstable CASP3 15 41 CC(C)CS(=O)(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217540987 DE For-Sale Unstable NPY5R 31 47 N#Cc1ccccc1NC(=O)C(=O)NCC[C@H](O)c1ccsc1 ZINC000217541000 ED In-Stock Unstable ADRB1 40 32 CCc1ccc([C@@H](C)NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217541015 GJ For-Sale Unstable SDH1 0 48 COc1ccc(C(=O)[C@@H](C)N2C[C@@H](C)C[C@@H](C)C2)cc1 ZINC000217541029 CG For-Sale Unstable RORC 27 40 O=C(Nc1ccc2[nH]cc([C@H](C(=O)O)N3C[C@@H]4C[C@H](C3)Cn3c4cccc3=O)c2c1)c1ccccc1 ZINC000217541048 JH In-Stock Unstable CHRNA4 24 42 N#Cc1ccccc1NC(=O)C(=O)NCC[C@@H](O)c1ccsc1 ZINC000217541065 ED In-Stock Unstable ADRB1 40 32 CCCCS(=O)(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217541083 DE For-Sale Unstable NPY5R 30 42 CCc1ccc([C@H](C)NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217541085 GJ For-Sale Unstable SDH1 0 48 COc1ccc(C(=O)[C@@H](C)N2C[C@H](C)C[C@@H](C)C2)cc1 ZINC000217541124 CG For-Sale Unstable RORC 27 40 O=C(Nc1ccc2[nH]cc([C@@H](C(=O)O)N3C[C@@H]4C[C@H](C3)Cn3c4cccc3=O)c2c1)c1ccccc1 ZINC000217541131 JH In-Stock Unstable CHRNA4 24 42 COc1cc(Cl)c(C(=O)[C@H](C)N)cc1OC ZINC000217541153 BD For-Sale Unstable HTR4 42 38 C[C@@H]1CCCCN1C(=O)CN1CCC[C@@H](CN)C1 ZINC000217541154 CD On-Demand Unstable UTS2R 43 30 C[C@@H](NC(=O)NCCc1ccc(Br)cc1)c1ccc2c(c1)CCCC2 ZINC000217541208 HJ For-Sale Unstable SDH1 0 43 Cc1cccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217541213 FF For-Sale Unstable NPY5R 31 46 C[C@H]1CCCCN1C(=O)CN1CCC[C@@H](CN)C1 ZINC000217541221 CD On-Demand Unstable UTS2R 43 30 COc1cc(Cl)c(C(=O)[C@@H](C)N)cc1OC ZINC000217541235 BD For-Sale Unstable HTR4 42 38 C[C@H](NC(=O)NCCc1ccc(Br)cc1)c1ccc2c(c1)CCCC2 ZINC000217541288 HJ For-Sale Unstable SDH1 0 43 CCCNc1ccc(S(=O)(=O)NCCC)cc1C(=O)O ZINC000217541291 DD In-Stock Unstable CASP3 16 44 CCCNc1ccc(S(=O)(=O)NCCC)cc1C(=O)O ZINC000217541291 DD In-Stock Unstable BDKRB1 0 43 O=C1OC2(CCN(S(=O)(=O)c3ccccc3F)CC2)c2ccccc21 ZINC000217541322 FF For-Sale Unstable NPY5R 37 51 O=C1OC2(CCN(S(=O)(=O)c3ccccc3F)CC2)c2ccccc21 ZINC000217541322 FF For-Sale Unstable PKM 23 47 CCCCC[C@@H](C)NC(=O)CN1CCC[C@@H](CN)C1 ZINC000217541340 CD On-Demand Unstable NOD1 81 38 c1ccc(N2CCN([C@@H]3CCOC3)CC2)cc1 ZINC000217541356 BD On-Demand Unstable SLC18A3 18 43 c1ccc(N2CCN([C@@H]3CCOC3)CC2)cc1 ZINC000217541356 BD On-Demand Unstable L3MBTL3 27 41 O=C(/C=C\c1ccccc1)NCC1CC(O)C1 ZINC000217541365 BD On-Demand Unstable HDAC8 66 38 O=C(/C=C\c1ccccc1)NCC1CC(O)C1 ZINC000217541365 BD On-Demand Unstable MMP2 22 55 O=C(/C=C\c1ccccc1)NCC1CC(O)C1 ZINC000217541365 BD On-Demand Unstable HDAC1 35 40 O=C(/C=C\c1ccccc1)NCC1CC(O)C1 ZINC000217541365 BD On-Demand Unstable HDAC2 22 40 O=C(/C=C\c1ccccc1)NCC1CC(O)C1 ZINC000217541365 BD On-Demand Unstable HDAC6 48 56 O=C(/C=C\c1ccccc1)NCC1CC(O)C1 ZINC000217541365 BD On-Demand Unstable HDAC9 32 40 O=C(/C=C\c1ccccc1)NCC1CC(O)C1 ZINC000217541365 BD On-Demand Unstable HDAC7 48 40 O=C(/C=C\c1ccccc1)NCC1CC(O)C1 ZINC000217541365 BD On-Demand Unstable MMP1 0 44 O=C(/C=C\c1ccccc1)NCC1CC(O)C1 ZINC000217541365 BD On-Demand Unstable IMA1 0 55 CCc1cccc(CC)c1NC(=O)NCCc1ccc(Br)cc1 ZINC000217541406 GJ On-Demand Unstable MTNR1A 37 40 CCc1cccc(CC)c1NC(=O)NCCc1ccc(Br)cc1 ZINC000217541406 GJ On-Demand Unstable ACAT 0 51 CCCNS(=O)(=O)c1ccc(NC(C)C)c(C(=O)O)c1 ZINC000217541413 DD In-Stock Unstable CASP3 16 42 CCCCC[C@H](C)NC(=O)CN1CCC[C@@H](CN)C1 ZINC000217541426 CD On-Demand Unstable NOD1 81 38 O=C1OC2(CCN(S(=O)(=O)c3ccc(F)cc3)CC2)c2ccccc21 ZINC000217541435 FF For-Sale Unstable NPY5R 39 49 O=C1OC2(CCN(S(=O)(=O)c3ccc(F)cc3)CC2)c2ccccc21 ZINC000217541435 FF For-Sale Unstable PKM 42 45 C[C@@H]1CCCCN1C[C@@H](O)CO ZINC000217541443 AC On-Demand Unstable SLC18A2 40 33 C[C@H]1CCCCN1C[C@@H](O)CO ZINC000217541525 AC On-Demand Unstable SLC18A2 40 33 CCCCNc1ccc(S(=O)(=O)NCCC)cc1C(=O)O ZINC000217541526 DE In-Stock Unstable CASP3 15 44 CCCCNc1ccc(S(=O)(=O)NCCC)cc1C(=O)O ZINC000217541526 DE In-Stock Unstable BDKRB1 0 43 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217541539 HK For-Sale Unstable CA2 20 59 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217541539 HK For-Sale Unstable ADRB2 17 47 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217541539 HK For-Sale Unstable ADRB1 43 47 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217541539 HK For-Sale Unstable SRD5A2 0 43 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217541539 HK For-Sale Unstable ADRB3 47 47 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217541539 HK For-Sale Unstable LTA4H 53 46 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217541539 HK For-Sale Unstable CA1 53 59 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217541539 HK For-Sale Unstable SCN2A 15 47 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217541539 HK For-Sale Unstable RAF1 42 40 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217541539 HK For-Sale Unstable MMP2 16 44 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217541539 HK For-Sale Unstable NPY5R 26 43 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217541539 HK For-Sale Unstable CA12 27 59 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217541539 HK For-Sale Unstable CA9 30 59 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217541539 HK For-Sale Unstable AMP1_PLAFQ 42 41 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217541539 HK For-Sale Unstable Q8MMZ8_EIMTE 51 40 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217541539 HK For-Sale Unstable F13A1 15 40 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217541539 HK For-Sale Unstable FFAR1 15 48 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217541539 HK For-Sale Unstable NCE103 39 59 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217541539 HK For-Sale Unstable CRTM 56 36 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217541539 HK For-Sale Unstable P96878_MYCTU 20 47 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217541539 HK For-Sale Unstable NAMPT 24 53 Cc1noc(C)c1S(=O)(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217541553 FE For-Sale Unstable NPY5R 32 44 C[C@@H]1CCCCN1C[C@@H](O)COc1ccc(C#N)cc1 ZINC000217541608 CE In-Stock Unstable ADRB2 15 43 C[C@@H]1CCCCN1C[C@@H](O)COc1ccc(C#N)cc1 ZINC000217541608 CE In-Stock Unstable HRH3 34 47 C[C@@H]1CCCCN1C[C@@H](O)COc1ccc(C#N)cc1 ZINC000217541608 CE In-Stock Unstable ABCB1 0 40 C[C@@H]1Cc2ccccc2N(c2ccc(Cl)cc2CBr)C1 ZINC000217541610 FK For-Sale Unstable DRD4 18 41 CCCNS(=O)(=O)c1ccc(NCC(C)C)c(C(=O)O)c1 ZINC000217541649 DE In-Stock Unstable CASP3 16 43 CCCNS(=O)(=O)c1ccc(NCC(C)C)c(C(=O)O)c1 ZINC000217541649 DE In-Stock Unstable BDKRB1 0 46 CCCNS(=O)(=O)c1ccc(NCC(C)C)c(C(=O)O)c1 ZINC000217541649 DE In-Stock Unstable MTNN 45 32 Cc1ccc(Cl)cc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217541652 FJ For-Sale Unstable RAF1 37 42 Cc1ccc(Cl)cc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217541652 FJ For-Sale Unstable Q8MMZ8_EIMTE 25 42 Cc1ccc(Cl)cc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217541652 FJ For-Sale Unstable LEF 44 35 Cc1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)s1 ZINC000217541659 FF For-Sale Unstable NPY5R 31 45 C[C@H]1Cc2ccccc2N(c2ccc(Cl)cc2CBr)C1 ZINC000217541699 FK For-Sale Unstable DRD4 18 41 COc1ccc2c(CC(=O)NC[C@H]3CC[C@@H](C(=O)O)CC3)cc(=O)oc2c1 ZINC000217541721 FE In-Stock Unstable MAOA 40 39 COc1ccc2c(CC(=O)NC[C@H]3CC[C@@H](C(=O)O)CC3)cc(=O)oc2c1 ZINC000217541721 FE In-Stock Unstable MAOB 29 50 COc1ccc2c(CC(=O)NC[C@H]3CC[C@@H](C(=O)O)CC3)cc(=O)oc2c1 ZINC000217541721 FE In-Stock Unstable MTR1B_CHICK 0 41 COc1ccc2c(CC(=O)NC[C@H]3CC[C@@H](C(=O)O)CC3)cc(=O)oc2c1 ZINC000217541721 FE In-Stock Unstable MTNR1A 58 43 COc1ccc2c(CC(=O)NC[C@H]3CC[C@@H](C(=O)O)CC3)cc(=O)oc2c1 ZINC000217541721 FE In-Stock Unstable VCP 30 42 CCCNS(=O)(=O)c1ccc(N[C@@H](C)CC)c(C(=O)O)c1 ZINC000217541753 DE In-Stock Unstable CASP3 16 41 COc1ccc(OC)c(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217541767 GH On-Demand Unstable TRPV1 23 49 COc1ccc(OC)c(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217541767 GH On-Demand Unstable RAF1 45 46 COc1ccc(OC)c(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217541767 GH On-Demand Unstable MTNR1A 87 43 COc1ccc(OC)c(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217541767 GH On-Demand Unstable MTNR1B 73 43 COc1ccc(OC)c(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217541767 GH On-Demand Unstable CA9 15 40 COc1ccc(OC)c(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217541767 GH On-Demand Unstable Q8MMZ8_EIMTE 35 46 COc1ccc(OC)c(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217541767 GH On-Demand Unstable AKR1C2 38 43 O=C(O)CCC(=O)Nc1ccc2c([C@H](C(=O)O)N3C[C@@H]4C[C@H](C3)Cn3c4cccc3=O)c[nH]c2c1 ZINC000217541769 JE In-Stock Unstable CHRNA4 31 40 CCc1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217541776 FG For-Sale Unstable NPY5R 30 43 C[C@@H]1CN(c2ccc(F)cc2CBr)CCN1C ZINC000217541800 DF For-Sale Unstable ADRA2B 0 43 C[C@@H]1CN(c2ccc(F)cc2CBr)CCN1C ZINC000217541800 DF For-Sale Unstable ADRA2C 0 43 CCCNS(=O)(=O)c1ccc(N[C@H](C)CC)c(C(=O)O)c1 ZINC000217541833 DE In-Stock Unstable CASP3 16 41 CCc1cccc(C)c1NC(=O)NCCc1ccc(Br)cc1 ZINC000217541868 FJ On-Demand Unstable ACAT 0 50 Cc1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1C ZINC000217541873 FG For-Sale Unstable NPY5R 31 50 C[C@H]1CN(c2ccc(F)cc2CBr)CCN1C ZINC000217541894 DF For-Sale Unstable ADRA2B 0 43 C[C@H]1CN(c2ccc(F)cc2CBr)CCN1C ZINC000217541894 DF For-Sale Unstable ADRA2C 0 43 CCCNS(=O)(=O)c1ccc(NC(C)(C)C)c(C(=O)O)c1 ZINC000217541938 DE In-Stock Unstable CASP3 15 42 CCCNS(=O)(=O)c1ccc(NC(C)(C)C)c(C(=O)O)c1 ZINC000217541938 DE In-Stock Unstable PRTN3 45 33 CCCNS(=O)(=O)c1ccc(NC(C)(C)C)c(C(=O)O)c1 ZINC000217541938 DE In-Stock Unstable AKR1C3 20 40 CC[C@H](CSC)N1C(=O)[C@H](C2CC2)NC(=O)[C@@H]1C(C)C ZINC000217541960 CD For-Sale Unstable OXTR 45 33 Cc1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c(C)c1 ZINC000217541979 FG For-Sale Unstable NPY5R 31 50 Cc1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c(C)c1 ZINC000217541979 FG For-Sale Unstable EPHX2 16 44 Cc1cc(C)c(NC(=O)NCCc2ccc(Br)cc2)c(C)c1 ZINC000217541989 FJ On-Demand Unstable ACAT 0 45 CC(C)(C)c1ccc(C(=O)N2CCC(C(=O)N[C@@H]3CCOC3)CC2)cc1 ZINC000217542010 FF In-Stock Unstable EPHX2 31 55 CC(C)(C)c1ccc(C(=O)N2CCC(C(=O)N[C@@H]3CCOC3)CC2)cc1 ZINC000217542010 FF In-Stock Unstable L3MBTL1 0 43 CC(C)(C)c1ccc(C(=O)N2CCC(C(=O)N[C@@H]3CCOC3)CC2)cc1 ZINC000217542010 FF In-Stock Unstable L3MBTL3 72 38 COc1ccc(Cl)cc1S(=O)(=O)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217542035 IG For-Sale Unstable CPT1A 66 37 COc1ccc(Cl)cc1S(=O)(=O)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217542035 IG For-Sale Unstable CPT2 45 35 COc1ccc(Cl)cc1S(=O)(=O)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217542035 IG For-Sale Unstable CPT1B 61 34 C=CCNc1ccc(S(=O)(=O)NCCC)cc1C(=O)O ZINC000217542040 CD In-Stock Unstable CASP3 0 42 CC(C)(C)c1ccc(C(=O)N2CCC(C(=O)N[C@H]3CCOC3)CC2)cc1 ZINC000217542077 FF In-Stock Unstable EPHX2 31 55 CC(C)(C)c1ccc(C(=O)N2CCC(C(=O)N[C@H]3CCOC3)CC2)cc1 ZINC000217542077 FF In-Stock Unstable L3MBTL1 0 43 CC(C)(C)c1ccc(C(=O)N2CCC(C(=O)N[C@H]3CCOC3)CC2)cc1 ZINC000217542077 FF In-Stock Unstable L3MBTL3 72 38 O=C1OC2(CCN(S(=O)(=O)CCc3ccccc3)CC2)c2ccccc21 ZINC000217542090 FF For-Sale Unstable SIGMAR1 24 62 O=C1OC2(CCN(S(=O)(=O)CCc3ccccc3)CC2)c2ccccc21 ZINC000217542090 FF For-Sale Unstable NPY5R 32 43 COC(=O)c1ccccc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217542112 GH For-Sale Unstable SLC6A5 23 40 COC(=O)c1ccccc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217542112 GH For-Sale Unstable NCE103 19 41 COC(=O)c1ccccc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217542112 GH For-Sale Unstable FAS 54 44 Cc1cc(=O)cc(C(=O)N2CCCN(C3Cc4ccccc4C3)CC2)o1 ZINC000217542195 FE In-Stock Unstable L3MBTL1 0 41 Cc1cc(=O)cc(C(=O)N2CCCN(C3Cc4ccccc4C3)CC2)o1 ZINC000217542195 FE In-Stock Unstable L3MBTL3 58 41 C[C@@H]1CN(c2cccc(Cl)c2CBr)CCN1C ZINC000217542199 DG For-Sale Unstable DRD3 15 41 C[C@@H]1CN(c2cccc(Cl)c2CBr)CCN1C ZINC000217542199 DG For-Sale Unstable ADRA2B 0 41 C[C@@H]1CN(c2cccc(Cl)c2CBr)CCN1C ZINC000217542199 DG For-Sale Unstable ADRA2C 0 41 Cc1ccc(C)c(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217542205 FG For-Sale Unstable NPY5R 32 51 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217542222 GI For-Sale Unstable BLM 0 48 CCCNS(=O)(=O)c1ccc(NC2CCCC2)c(C(=O)O)c1 ZINC000217542258 EE In-Stock Unstable CASP3 0 44 Cc1ccc(/C=C\C(=O)NC2CC(O)C2)c(Br)c1 ZINC000217542277 DE For-Sale Unstable BOTA 27 41 C[C@H]1CN(c2cccc(Cl)c2CBr)CCN1C ZINC000217542282 DG For-Sale Unstable DRD3 15 41 C[C@H]1CN(c2cccc(Cl)c2CBr)CCN1C ZINC000217542282 DG For-Sale Unstable ADRA2B 0 41 C[C@H]1CN(c2cccc(Cl)c2CBr)CCN1C ZINC000217542282 DG For-Sale Unstable ADRA2C 0 41 O=C(O)Cn1cc([C@H](C(=O)O)N2C[C@@H]3C[C@H](C2)Cn2c3cccc2=O)c2ccccc21 ZINC000217542302 HE In-Stock Unstable CHRNA4 30 48 COc1cc([N+](=O)[O-])ccc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217542314 GH For-Sale Unstable KCNMA1 23 50 COc1cc([N+](=O)[O-])ccc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217542314 GH For-Sale Unstable Q8MMZ8_EIMTE 0 49 Cc1cccc(CS(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217542320 FF For-Sale Unstable NPY5R 30 44 CCCNS(=O)(=O)c1ccc(NC2CCCCC2)c(C(=O)O)c1 ZINC000217542372 EF In-Stock Unstable CASP3 0 43 O=C(O)Cn1cc([C@@H](C(=O)O)N2C[C@@H]3C[C@H](C2)Cn2c3cccc2=O)c2ccccc21 ZINC000217542383 HE In-Stock Unstable CHRNA4 30 48 O=C(NCCc1ccc(Br)cc1)Nc1ccc([N+](=O)[O-])cc1 ZINC000217542396 FH On-Demand Unstable PPIA 15 40 O=C(NCCc1ccc(Br)cc1)Nc1ccc([N+](=O)[O-])cc1 ZINC000217542396 FH On-Demand Unstable CA5A 15 61 O=C(NCCc1ccc(Br)cc1)Nc1ccc([N+](=O)[O-])cc1 ZINC000217542396 FH On-Demand Unstable MMP2 15 43 O=C(NCCc1ccc(Br)cc1)Nc1ccc([N+](=O)[O-])cc1 ZINC000217542396 FH On-Demand Unstable MMP8 33 43 O=C(NCCc1ccc(Br)cc1)Nc1ccc([N+](=O)[O-])cc1 ZINC000217542396 FH On-Demand Unstable MMP9 16 43 O=C(NCCc1ccc(Br)cc1)Nc1ccc([N+](=O)[O-])cc1 ZINC000217542396 FH On-Demand Unstable CA12 15 45 O=C(NCCc1ccc(Br)cc1)Nc1ccc([N+](=O)[O-])cc1 ZINC000217542396 FH On-Demand Unstable MMP1 30 43 O=C(NCCc1ccc(Br)cc1)Nc1ccc([N+](=O)[O-])cc1 ZINC000217542396 FH On-Demand Unstable NCE103 28 48 O=C(NCCc1ccc(Br)cc1)Nc1ccc([N+](=O)[O-])cc1 ZINC000217542396 FH On-Demand Unstable PRMT3 18 47 O=C(NCCc1ccc(Br)cc1)Nc1ccc([N+](=O)[O-])cc1 ZINC000217542396 FH On-Demand Unstable P96878_MYCTU 15 40 Cc1cc(CCN)c(C)c(F)c1Br ZINC000217542415 BF For-Sale Unstable TAAR1 16 40 COc1cccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217542421 FF For-Sale Unstable NPY5R 31 52 COc1cccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217542421 FF For-Sale Unstable PKM 38 54 COc1cccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217542421 FF For-Sale Unstable AKR1C3 18 41 Cc1ccc(/C=C\C(=O)NC2CC(O)C2)cc1Cl ZINC000217542488 CE For-Sale Unstable HDAC2 15 42 Cc1ccc(/C=C\C(=O)NC2CC(O)C2)cc1Cl ZINC000217542488 CE For-Sale Unstable CCR2 16 44 O=C(NCCc1ccc(Br)cc1)Nc1cccc([N+](=O)[O-])c1 ZINC000217542500 FH On-Demand Unstable PPIA 17 44 O=C(NCCc1ccc(Br)cc1)Nc1cccc([N+](=O)[O-])c1 ZINC000217542500 FH On-Demand Unstable CA5A 17 49 O=C(NCCc1ccc(Br)cc1)Nc1cccc([N+](=O)[O-])c1 ZINC000217542500 FH On-Demand Unstable NCE103 21 48 O=C(NCCc1ccc(Br)cc1)Nc1cccc([N+](=O)[O-])c1 ZINC000217542500 FH On-Demand Unstable TRPM8 0 46 O=C(NCCc1ccc(Br)cc1)Nc1cccc([N+](=O)[O-])c1 ZINC000217542500 FH On-Demand Unstable PRMT3 17 42 Cc1c(F)cc(Br)c(C)c1CCN ZINC000217542512 BF For-Sale Unstable TAAR1 16 41 NC[C@@H]1CCCN(C/C=C\c2ccccc2)C1 ZINC000217542523 BE On-Demand Unstable SLC6A1 47 34 COc1ccccc1S(=O)(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217542536 FF For-Sale Unstable NPY5R 33 53 CCCNS(=O)(=O)c1ccc(NCCO)c(C(=O)O)c1 ZINC000217542589 DC In-Stock Unstable CASP3 15 42 CCCNS(=O)(=O)c1ccc(NCCO)c(C(=O)O)c1 ZINC000217542589 DC In-Stock Unstable BDKRB1 0 41 NC[C@H]1CCCN(C/C=C\c2ccccc2)C1 ZINC000217542614 BE On-Demand Unstable SLC6A1 47 34 O=C1OC2(CCN(S(=O)(=O)Cc3cccc(F)c3)CC2)c2ccccc21 ZINC000217542646 GF For-Sale Unstable SIGMAR1 15 56 O=C1OC2(CCN(S(=O)(=O)Cc3cccc(F)c3)CC2)c2ccccc21 ZINC000217542646 GF For-Sale Unstable NPY5R 39 48 CCCNS(=O)(=O)c1ccc(NCCCO)c(C(=O)O)c1 ZINC000217542696 DC In-Stock Unstable CASP3 16 45 CCCNS(=O)(=O)c1ccc(NCCCO)c(C(=O)O)c1 ZINC000217542696 DC In-Stock Unstable BDKRB1 0 42 O=C(NCCCCl)NCCc1ccc(Br)cc1 ZINC000217542712 DF For-Sale Unstable LIG1 0 42 Cc1cc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)ccc1F ZINC000217542762 GF For-Sale Unstable NPY5R 32 45 Cc1cc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)ccc1F ZINC000217542762 GF For-Sale Unstable PKM 49 42 CCCNS(=O)(=O)c1ccc(NCCOC)c(C(=O)O)c1 ZINC000217542816 DD In-Stock Unstable CASP3 15 40 CCCNS(=O)(=O)c1ccc(NCCOC)c(C(=O)O)c1 ZINC000217542816 DD In-Stock Unstable BDKRB1 0 43 O=C(NCCCl)NCCc1ccc(Br)cc1 ZINC000217542825 DF For-Sale Unstable LIG1 0 44 O=C(O)CCC(=O)Nc1ccc2[nH]cc([C@H](C(=O)O)N3C[C@@H]4C[C@H](C3)Cn3c4cccc3=O)c2c1 ZINC000217542847 JE In-Stock Unstable CHRNA4 31 40 O=C1OC2(CCN(S(=O)(=O)Cc3ccc(F)cc3)CC2)c2ccccc21 ZINC000217542878 GF For-Sale Unstable NPY5R 37 48 CCCNS(=O)(=O)c1ccc(NCCCOC)c(C(=O)O)c1 ZINC000217542920 ED In-Stock Unstable CASP3 22 41 O=C(NCCc1ccc(Br)cc1)N1CCN(c2ccc(F)cc2)CC1 ZINC000217542930 HH On-Demand Unstable AKR1C3 0 45 CCc1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)s1 ZINC000217542982 GG For-Sale Unstable NPY5R 29 40 O=C(O)Cn1cc([C@H](C(=O)O)N2C[C@@H]3C[C@H](C2)Cn2c3cccc2=O)c2ccc(Br)cc21 ZINC000217542997 KF In-Stock Unstable CHRNA4 26 41 Cc1cccc([C@@H]2N[C@H](c3cccc(C)c3)[C@H]([N+](=O)[O-])C(C)(C)[C@H]2[N+](=O)[O-])c1 ZINC000217543025 GI In-Stock Unstable CACNA1D 51 32 CCCNS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217543041 EF In-Stock Unstable GNRHR 16 41 CCCNS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217543041 EF In-Stock Unstable TBXA2R 42 37 CCCNS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217543041 EF In-Stock Unstable CASP3 18 40 CCCNS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217543041 EF In-Stock Unstable AKR1C3 16 45 CCCCOC(=O)c1ccccc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217543054 HJ For-Sale Unstable ACAT 0 42 O=C1OC2(CCN(S(=O)(=O)c3cccc(Cl)c3)CC2)c2ccccc21 ZINC000217543086 GG For-Sale Unstable NPY5R 31 49 COc1cccc(-c2cccc(C(=O)NCCSc3nncn3C)c2)c1 ZINC000217543103 FG In-Stock Unstable DRD4 58 45 COc1cccc(-c2cccc(C(=O)NCCSc3nncn3C)c2)c1 ZINC000217543103 FG In-Stock Unstable DRD3 16 43 COc1cccc(-c2cccc(C(=O)NCCSc3nncn3C)c2)c1 ZINC000217543103 FG In-Stock Unstable MTNR1A 26 45 Cc1cccc([C@H]2N[C@H](c3cccc(C)c3)[C@H]([N+](=O)[O-])C(C)(C)[C@@H]2[N+](=O)[O-])c1 ZINC000217543112 GI In-Stock Unstable CACNA1D 58 33 CCCNS(=O)(=O)c1ccc(N[C@@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217543141 FG In-Stock Unstable CASP3 19 40 CC(=O)c1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217543160 FI On-Demand Unstable CA9 16 47 CC(=O)c1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217543160 FI On-Demand Unstable DNAB 0 48 CC(=O)c1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217543160 FI On-Demand Unstable P96878_MYCTU 16 43 Cc1cccc([C@H]2N[C@H](c3cccc(C)c3)[C@H]([N+](=O)[O-])C(C)(C)[C@H]2[N+](=O)[O-])c1 ZINC000217543196 GI In-Stock Unstable CACNA1D 51 32 CCCNS(=O)(=O)c1ccc(N[C@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217543215 FG In-Stock Unstable CASP3 19 40 O=C1OC2(CCN(S(=O)(=O)c3ccccc3Cl)CC2)c2ccccc21 ZINC000217543216 GG For-Sale Unstable NPY5R 40 52 O=C(NCC[C@H](O)c1ccsc1)C(=O)Nc1ccc(F)c(Cl)c1 ZINC000217543242 FF In-Stock Unstable ENV 40 31 CC(=O)c1cccc(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217543276 FI On-Demand Unstable CCR3 42 48 CC(=O)c1cccc(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217543276 FI On-Demand Unstable GUAB 0 48 CC(=O)c1cccc(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217543276 FI On-Demand Unstable RAF1 31 45 CC(=O)c1cccc(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217543276 FI On-Demand Unstable EPHX2 15 43 CC(=O)c1cccc(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217543276 FI On-Demand Unstable Q8MMZ8_EIMTE 0 45 CC(=O)c1cccc(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217543276 FI On-Demand Unstable AKR1C3 26 43 CC(=O)c1cccc(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217543276 FI On-Demand Unstable IMDH_CRYPV 26 40 CC(=O)c1cccc(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217543276 FI On-Demand Unstable KCNK3 71 35 O=C(/C=C\c1ccc(Cl)cc1)NCC1CC(O)C1 ZINC000217543301 CE On-Demand Unstable HDAC8 19 49 O=C(/C=C\c1ccc(Cl)cc1)NCC1CC(O)C1 ZINC000217543301 CE On-Demand Unstable HDAC1 20 44 O=C1OC2(CCN(S(=O)(=O)c3ccc(F)c(F)c3)CC2)c2ccccc21 ZINC000217543308 GF For-Sale Unstable NPY5R 33 50 O=C1OC2(CCN(S(=O)(=O)c3ccc(F)c(F)c3)CC2)c2ccccc21 ZINC000217543308 GF For-Sale Unstable PKM 49 44 CCCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217543309 FF In-Stock Unstable TBXA2R 52 41 O=C(NCC[C@@H](O)c1ccsc1)C(=O)Nc1ccc(F)c(Cl)c1 ZINC000217543335 FF In-Stock Unstable ENV 40 31 O=C(NCCc1ccc(Br)cc1)Nc1ccccc1Sc1ccccc1 ZINC000217543388 IK For-Sale Unstable AMP1_PLAFQ 29 40 CNCC(=O)O[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217543407 BE For-Sale Unstable TRPM8 0 41 CCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217543412 GF In-Stock Unstable CA2 20 41 CCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217543412 GF In-Stock Unstable TBXA2R 50 43 CCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217543412 GF In-Stock Unstable TBXAS1 17 42 CCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217543412 GF In-Stock Unstable BMP1 60 37 CCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217543412 GF In-Stock Unstable CA1 20 44 CCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217543412 GF In-Stock Unstable MMP13 53 40 CCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217543412 GF In-Stock Unstable ALOX15B 0 41 CCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217543412 GF In-Stock Unstable MMP2 32 40 CCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217543412 GF In-Stock Unstable MMP3 41 37 CCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217543412 GF In-Stock Unstable MMP8 24 40 CCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217543412 GF In-Stock Unstable MMP14 15 40 CCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217543412 GF In-Stock Unstable ALOX15 48 41 CCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217543412 GF In-Stock Unstable MMP9 46 40 CCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217543412 GF In-Stock Unstable MMP12 26 40 CCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217543412 GF In-Stock Unstable PTGDR 25 43 CCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217543412 GF In-Stock Unstable IAP 0 46 CCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217543412 GF In-Stock Unstable CA9 23 44 CCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217543412 GF In-Stock Unstable MMP1 48 39 CCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217543412 GF In-Stock Unstable AKR1C3 30 47 CCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217543412 GF In-Stock Unstable AKR1C2 51 38 Cc1ccccc1/C=C\C(=O)NC1CC(O)C1 ZINC000217543415 BD For-Sale Unstable BOTA 20 40 O=C1OC2(CCN(S(=O)(=O)c3cc(F)ccc3F)CC2)c2ccccc21 ZINC000217543416 GF For-Sale Unstable NPY5R 38 50 CNCC(=O)O[C@H]1C[C@H](C)CC[C@@H]1C(C)C ZINC000217543491 BE For-Sale Unstable TRPM8 0 41 CCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217543511 HF In-Stock Unstable TBXA2R 44 40 CCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217543511 HF In-Stock Unstable IAP 0 47 CCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217543511 HF In-Stock Unstable AKR1C3 15 43 CCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217543511 HF In-Stock Unstable SCMU_MYCTU 0 46 O=C1OC2(CCN(S(=O)(=O)c3ccc(Cl)s3)CC2)c2ccccc21 ZINC000217543536 GG For-Sale Unstable NPY5R 31 45 Cc1ccc(NC(=O)NCCc2ccc(Br)cc2)c(C)c1 ZINC000217543595 EI On-Demand Unstable RAF1 32 40 CC(=O)c1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217543645 GF For-Sale Unstable NPY5R 36 44 CC(C)CCC[C@@H](C)NC(=O)CN1CCC[C@@H](CN)C1 ZINC000217543666 CD On-Demand Unstable BIRC2 40 32 Cc1ccc(N[C@H]2C[C@H](C)CC[C@H]2C(C)C)cc1I ZINC000217543680 FK For-Sale Unstable TRPM8 15 42 COc1ccc2c(c1)c([C@H](C(=O)O)N1C[C@@H]3C[C@H](C1)Cn1c3cccc1=O)cn2CC(=O)O ZINC000217543682 JE In-Stock Unstable CHRNA4 32 42 COc1ccc(C)cc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217543693 FI On-Demand Unstable TRPV1 0 42 COc1ccc(C)cc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217543693 FI On-Demand Unstable RAF1 39 48 COc1ccc(C)cc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217543693 FI On-Demand Unstable Q8MMZ8_EIMTE 30 48 COc1ccccc1/C=C\C(=O)NCC1CC(O)C1 ZINC000217543722 CD For-Sale Unstable DRD3 15 50 CCCNS(=O)(=O)c1ccc(NC[C@@H]2CCCO2)c(C(=O)O)c1 ZINC000217543731 ED In-Stock Unstable BDKRB1 28 41 CC(=O)c1cccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217543746 GF For-Sale Unstable NPY5R 41 43 CC(=O)c1cccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217543746 GF For-Sale Unstable AKR1C3 64 43 CC(C)CCC[C@H](C)NC(=O)CN1CCC[C@@H](CN)C1 ZINC000217543752 CD On-Demand Unstable BIRC2 40 32 Cc1ccc(N[C@H]2C[C@@H](C)CC[C@H]2C(C)C)cc1I ZINC000217543769 FK For-Sale Unstable TRPM8 15 42 COc1ccc2c(c1)c([C@@H](C(=O)O)N1C[C@@H]3C[C@H](C1)Cn1c3cccc1=O)cn2CC(=O)O ZINC000217543783 JE In-Stock Unstable CHRNA4 32 42 C[C@H]1Cc2ccccc2N(C[C@@H](O)c2ccccc2)C1 ZINC000217543793 CG On-Demand Unstable SLC18A3 15 40 C[C@H]1Cc2ccccc2N(C[C@@H](O)c2ccccc2)C1 ZINC000217543793 CG On-Demand Unstable TPP2 51 31 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217543809 HK For-Sale Unstable GUAB 0 42 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217543809 HK For-Sale Unstable RAF1 63 61 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217543809 HK For-Sale Unstable EPHX2 15 45 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217543809 HK For-Sale Unstable Q8MMZ8_EIMTE 79 61 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217543809 HK For-Sale Unstable BRAF 16 42 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217543809 HK For-Sale Unstable PTPA 0 44 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217543809 HK For-Sale Unstable IMDH_CRYPV 20 44 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217543809 HK For-Sale Unstable BLM 0 47 CCCNS(=O)(=O)c1ccc(NC[C@H]2CCCO2)c(C(=O)O)c1 ZINC000217543818 ED In-Stock Unstable BDKRB1 0 41 O=C(/C=C\c1cccc(Br)c1)NCC1CC(O)C1 ZINC000217543849 DE For-Sale Unstable HDAC8 58 39 O=C(/C=C\c1cccc(Br)c1)NCC1CC(O)C1 ZINC000217543849 DE For-Sale Unstable HDAC6 41 41 O=C(/C=C\c1cccc(Br)c1)NCC1CC(O)C1 ZINC000217543849 DE For-Sale Unstable IMA1 0 41 CCCc1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217543861 GG For-Sale Unstable NPY5R 29 41 C[C@@H]1Cc2ccccc2N(C[C@@H](O)c2ccccc2)C1 ZINC000217543876 CG On-Demand Unstable SLC18A3 15 40 C[C@@H]1Cc2ccccc2N(C[C@@H](O)c2ccccc2)C1 ZINC000217543876 CG On-Demand Unstable TPP2 51 31 C[C@@H]1CN(c2ccc(CBr)cn2)CCN1C ZINC000217543879 CE For-Sale Unstable SORD 56 35 CCCNS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217543930 DD In-Stock Unstable KCNQ2 69 35 CCCNS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217543930 DD In-Stock Unstable SLC6A9 18 43 CCCNS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217543930 DD In-Stock Unstable SFRP1 60 33 CCCNS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217543930 DD In-Stock Unstable WNT3 42 33 C[C@H]1CN(c2ccc(CBr)cn2)CCN1C ZINC000217543965 CE For-Sale Unstable SORD 56 35 Cc1cc(C)c(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c(C)c1 ZINC000217543988 GG For-Sale Unstable NPY5R 31 48 Cc1cc(C)c(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c(C)c1 ZINC000217543988 GG For-Sale Unstable EPHX2 19 41 COc1ccc2c(c1)C[C@@H](C(=O)NCCc1nnc(C)s1)CO2 ZINC000217543996 ED In-Stock Unstable MTNR1A 40 41 COc1ccc2c(c1)C[C@@H](C(=O)NCCc1nnc(C)s1)CO2 ZINC000217543996 ED In-Stock Unstable ROCK2 35 49 COc1ccc2c(c1)C[C@@H](C(=O)NCCc1nnc(C)s1)CO2 ZINC000217543996 ED In-Stock Unstable CDC42BPA 0 44 CCOC(=O)[C@@H](C)N1C[C@@H](C)Cc2ccccc21 ZINC000217544000 BF For-Sale Unstable ACE 29 42 CCOC(=O)[C@@H](C)N1C[C@@H](C)Cc2ccccc21 ZINC000217544000 BF For-Sale Unstable TPP2 71 39 Nc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1Cl ZINC000217544014 FI For-Sale Unstable RAF1 27 46 Nc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1Cl ZINC000217544014 FI For-Sale Unstable NCE103 34 43 CCCNS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217544041 EE In-Stock Unstable KCNQ2 68 35 CCCNS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217544041 EE In-Stock Unstable SLC6A9 18 45 CCCNS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217544041 EE In-Stock Unstable SFRP1 59 32 CCCNS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217544041 EE In-Stock Unstable WNT3 44 32 CCOC(=O)[C@H](C)N1C[C@@H](C)Cc2ccccc21 ZINC000217544075 BF For-Sale Unstable ACE 29 42 CCOC(=O)[C@H](C)N1C[C@@H](C)Cc2ccccc21 ZINC000217544075 BF For-Sale Unstable TPP2 71 39 COc1ccc2c(c1)C[C@H](C(=O)NCCc1nnc(C)s1)CO2 ZINC000217544077 ED In-Stock Unstable MTNR1A 40 41 COc1ccc2c(c1)C[C@H](C(=O)NCCc1nnc(C)s1)CO2 ZINC000217544077 ED In-Stock Unstable ROCK2 35 49 COc1ccc2c(c1)C[C@H](C(=O)NCCc1nnc(C)s1)CO2 ZINC000217544077 ED In-Stock Unstable CDC42BPA 0 44 Cc1cc(C)c(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1C ZINC000217544102 GG For-Sale Unstable NPY5R 32 54 CCCNS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1 ZINC000217544153 EC In-Stock Unstable SLC6A9 21 48 CC[C@H](C(N)=O)N1C[C@@H](C)Cc2ccccc21 ZINC000217544161 BD For-Sale Unstable TPP2 63 40 CC(C)c1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217544212 GH For-Sale Unstable NPY5R 30 43 CC(C)(C)NC(=O)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217544225 EF For-Sale Unstable CACNA1H 29 40 Cc1cc(O)c(Cl)c(C)c1C[C@H](N)C(=O)O ZINC000217544236 BD For-Sale Unstable OPRM1 23 45 Cc1cc(O)c(Cl)c(C)c1C[C@H](N)C(=O)O ZINC000217544236 BD For-Sale Unstable OPRD1 17 45 Cc1cc(O)c(Cl)c(C)c1C[C@H](N)C(=O)O ZINC000217544236 BD For-Sale Unstable GRIA3 58 40 Cc1cc(O)c(Cl)c(C)c1C[C@H](N)C(=O)O ZINC000217544236 BD For-Sale Unstable GRIA1 39 40 Cc1cc(O)c(Cl)c(C)c1C[C@H](N)C(=O)O ZINC000217544236 BD For-Sale Unstable GRIA2 48 40 Cc1cc(O)c(Cl)c(C)c1C[C@H](N)C(=O)O ZINC000217544236 BD For-Sale Unstable GRIA4 48 40 Cc1cc(O)c(Cl)c(C)c1C[C@H](N)C(=O)O ZINC000217544236 BD For-Sale Unstable GRIK1 39 40 O=C(NCC[C@@H](O)c1ccsc1)C(=O)Nc1cc2c3c(c1)CCN3C(=O)CC2 ZINC000217544238 GD In-Stock Unstable CYP11B1 26 40 O=C(NCC[C@@H](O)c1ccsc1)C(=O)Nc1cc2c3c(c1)CCN3C(=O)CC2 ZINC000217544238 GD In-Stock Unstable CYP11B2 25 40 CC[C@@H](C(N)=O)N1C[C@@H](C)Cc2ccccc21 ZINC000217544248 BD For-Sale Unstable TPP2 63 40 O=C(NCCc1ccc(Br)cc1)N1CCN(Cc2ccccc2)CC1 ZINC000217544250 HH On-Demand Unstable DRD4 50 45 O=C(NCCc1ccc(Br)cc1)N1CCN(Cc2ccccc2)CC1 ZINC000217544250 HH On-Demand Unstable ACHE 35 42 O=C(NCCc1ccc(Br)cc1)N1CCN(Cc2ccccc2)CC1 ZINC000217544250 HH On-Demand Unstable HRH2 15 42 O=C(NCCc1ccc(Br)cc1)N1CCN(Cc2ccccc2)CC1 ZINC000217544250 HH On-Demand Unstable DRD3 17 42 O=C(NCCc1ccc(Br)cc1)N1CCN(Cc2ccccc2)CC1 ZINC000217544250 HH On-Demand Unstable SIGMAR1 69 53 O=C(NCCc1ccc(Br)cc1)N1CCN(Cc2ccccc2)CC1 ZINC000217544250 HH On-Demand Unstable NPFFR2 34 44 O=C(NCCc1ccc(Br)cc1)N1CCN(Cc2ccccc2)CC1 ZINC000217544250 HH On-Demand Unstable FAAH 29 52 O=C(NCCc1ccc(Br)cc1)N1CCN(Cc2ccccc2)CC1 ZINC000217544250 HH On-Demand Unstable CXCR3 27 43 O=C(NCCc1ccc(Br)cc1)N1CCN(Cc2ccccc2)CC1 ZINC000217544250 HH On-Demand Unstable MGLL 0 48 O=C(NCCc1ccc(Br)cc1)N1CCN(Cc2ccccc2)CC1 ZINC000217544250 HH On-Demand Unstable ABHD6 0 40 O=C(NCCc1ccc(Br)cc1)N1CCN(Cc2ccccc2)CC1 ZINC000217544250 HH On-Demand Unstable NPFFR1 57 44 O=C(NCCc1ccc(Br)cc1)N1CCN(Cc2ccccc2)CC1 ZINC000217544250 HH On-Demand Unstable GPR183 0 40 CCCNS(=O)(=O)c1ccc(NCCCOCC)c(C(=O)O)c1 ZINC000217544262 ED In-Stock Unstable CASP3 0 42 O=C(O)[C@@H]1Cc2ccccc2CN1C(=O)c1cc(Cl)c[nH]c1=O ZINC000217544315 ED In-Stock Unstable OPRD1 26 40 O=C(O)[C@@H]1Cc2ccccc2CN1C(=O)c1cc(Cl)c[nH]c1=O ZINC000217544315 ED In-Stock Unstable AGTR2 60 47 O=C(O)[C@@H]1Cc2ccccc2CN1C(=O)c1cc(Cl)c[nH]c1=O ZINC000217544315 ED In-Stock Unstable CFTR 51 38 CCOc1ccccc1S(=O)(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217544322 GF For-Sale Unstable NPY5R 32 44 O=C(NCC[C@H](O)c1ccsc1)C(=O)Nc1cc2c3c(c1)CCN3C(=O)CC2 ZINC000217544323 GD In-Stock Unstable CYP11B1 26 40 O=C(NCC[C@H](O)c1ccsc1)C(=O)Nc1cc2c3c(c1)CCN3C(=O)CC2 ZINC000217544323 GD In-Stock Unstable CYP11B2 25 40 Cc1cc(O)c(Cl)c(C)c1C[C@@H](N)C(=O)O ZINC000217544326 BD For-Sale Unstable OPRM1 23 45 Cc1cc(O)c(Cl)c(C)c1C[C@@H](N)C(=O)O ZINC000217544326 BD For-Sale Unstable OPRD1 17 45 Cc1cc(O)c(Cl)c(C)c1C[C@@H](N)C(=O)O ZINC000217544326 BD For-Sale Unstable GRIA3 58 40 Cc1cc(O)c(Cl)c(C)c1C[C@@H](N)C(=O)O ZINC000217544326 BD For-Sale Unstable GRIA1 39 40 Cc1cc(O)c(Cl)c(C)c1C[C@@H](N)C(=O)O ZINC000217544326 BD For-Sale Unstable GRIA2 48 40 Cc1cc(O)c(Cl)c(C)c1C[C@@H](N)C(=O)O ZINC000217544326 BD For-Sale Unstable GRIA4 48 40 Cc1cc(O)c(Cl)c(C)c1C[C@@H](N)C(=O)O ZINC000217544326 BD For-Sale Unstable GRIK1 39 40 O=C(/C=C\c1ccc(Br)cc1)NC1CC(O)C1 ZINC000217544348 CE For-Sale Unstable HDAC8 42 41 O=C(/C=C\c1ccc(Br)cc1)NC1CC(O)C1 ZINC000217544348 CE For-Sale Unstable HDAC1 40 41 O=C(/C=C\c1ccc(Br)cc1)NC1CC(O)C1 ZINC000217544348 CE For-Sale Unstable HDAC2 17 45 O=C(/C=C\c1ccc(Br)cc1)NC1CC(O)C1 ZINC000217544348 CE For-Sale Unstable HDAC6 30 45 O=C(/C=C\c1ccc(Br)cc1)NC1CC(O)C1 ZINC000217544348 CE For-Sale Unstable BOTA 20 40 CN1CCN(C(=O)NCCc2ccc(Br)cc2)CC1 ZINC000217544367 ED On-Demand Unstable GPBAR1 22 40 CN1CCN(C(=O)NCCc2ccc(Br)cc2)CC1 ZINC000217544367 ED On-Demand Unstable LIG1 0 42 CCCNS(=O)(=O)c1ccc(NCCCOC(C)C)c(C(=O)O)c1 ZINC000217544369 FE In-Stock Unstable CASP3 0 42 O=C(O)[C@H]1Cc2ccccc2CN1C(=O)c1cc(Cl)c[nH]c1=O ZINC000217544389 ED In-Stock Unstable OPRD1 26 40 O=C(O)[C@H]1Cc2ccccc2CN1C(=O)c1cc(Cl)c[nH]c1=O ZINC000217544389 ED In-Stock Unstable AGTR2 60 47 O=C(O)[C@H]1Cc2ccccc2CN1C(=O)c1cc(Cl)c[nH]c1=O ZINC000217544389 ED In-Stock Unstable CFTR 51 38 Cn1cc([C@H](C(=O)O)N2C[C@@H]3C[C@H](C2)Cn2c3cccc2=O)c2ccc(C(=O)O)cc21 ZINC000217544396 HE In-Stock Unstable CHRNA4 27 44 COc1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1C ZINC000217544440 GF For-Sale Unstable NPY5R 29 46 C[C@@H](NC(=O)CN1CCC[C@@H](CN)C1)c1cccs1 ZINC000217544460 CD On-Demand Unstable BIRC2 41 34 O=C(NCCc1ccc(Br)cc1)N1CCCCC1 ZINC000217544474 DG On-Demand Unstable DPP7 54 41 O=C(NCCc1ccc(Br)cc1)N1CCCCC1 ZINC000217544474 DG On-Demand Unstable GPBAR1 24 43 O=C(NCCc1ccc(Br)cc1)N1CCCCC1 ZINC000217544474 DG On-Demand Unstable LIG1 0 40 CCCCCNc1ccc(S(=O)(=O)NCCC)cc1C(=O)O ZINC000217544478 EF In-Stock Unstable CASP3 17 45 Cn1cc([C@@H](C(=O)O)N2C[C@@H]3C[C@H](C2)Cn2c3cccc2=O)c2ccc(C(=O)O)cc21 ZINC000217544480 HE In-Stock Unstable CHRNA4 27 44 O=C(NCCc1ccc(Br)cc1)NC1CCCCCCCCCCC1 ZINC000217544540 HK For-Sale Unstable CNR2 16 41 O=C(NCCc1ccc(Br)cc1)NC1CCCCCCCCCCC1 ZINC000217544540 HK For-Sale Unstable EPHX2 33 74 O=C(NCCc1ccc(Br)cc1)NC1CCCCCCCCCCC1 ZINC000217544540 HK For-Sale Unstable GPBAR1 0 42 O=C(NCCc1ccc(Br)cc1)NC1CCCCCCCCCCC1 ZINC000217544540 HK For-Sale Unstable TRAR 18 40 C[C@H](NC(=O)CN1CCC[C@@H](CN)C1)c1cccs1 ZINC000217544542 CD On-Demand Unstable BIRC2 41 34 COc1ccc(C)cc1S(=O)(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217544549 GF For-Sale Unstable NPY5R 32 47 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)Nc1ccccc1 ZINC000217544566 FH For-Sale Unstable FABP4 40 35 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)Nc1ccccc1 ZINC000217544566 FH For-Sale Unstable EPHX2 16 44 O=C(/C=C\c1cccc([N+](=O)[O-])c1)NC1CC(O)C1 ZINC000217544575 CD For-Sale Unstable CACNA1D 40 35 O=C(/C=C\c1cccc([N+](=O)[O-])c1)NC1CC(O)C1 ZINC000217544575 CD For-Sale Unstable MMP2 0 41 O=C(/C=C\c1cccc([N+](=O)[O-])c1)NC1CC(O)C1 ZINC000217544575 CD For-Sale Unstable TRPM8 22 58 CCCNS(=O)(=O)c1ccc(NCCC(C)C)c(C(=O)O)c1 ZINC000217544598 EF In-Stock Unstable CASP3 16 44 NCCN1CCN(C(=O)NCCc2ccc(Br)cc2)CC1 ZINC000217544654 FD For-Sale Unstable LIG1 0 41 COc1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c(C)c1 ZINC000217544671 GF For-Sale Unstable NPY5R 33 56 C[C@@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccco1 ZINC000217544683 CD For-Sale Unstable CCR3 41 33 C[C@@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccco1 ZINC000217544683 CD For-Sale Unstable BIRC2 41 34 CCCNS(=O)(=O)c1ccc(N[C@@H](C)CCC)c(C(=O)O)c1 ZINC000217544718 EF In-Stock Unstable CASP3 16 44 Cc1cc(N2CCN(C)[C@@H](C)C2)ccc1CBr ZINC000217544729 CG For-Sale Unstable ADRA2A 0 44 Cc1cc(N2CCN(C)[C@@H](C)C2)ccc1CBr ZINC000217544729 CG For-Sale Unstable ADRA2B 24 44 Cc1cc(N2CCN(C)[C@@H](C)C2)ccc1CBr ZINC000217544729 CG For-Sale Unstable ADRA2C 22 44 C[C@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccco1 ZINC000217544766 CD For-Sale Unstable CCR3 41 33 C[C@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccco1 ZINC000217544766 CD For-Sale Unstable BIRC2 41 34 COc1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1F ZINC000217544780 GF For-Sale Unstable NPY5R 30 44 COc1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1F ZINC000217544780 GF For-Sale Unstable PKM 47 40 CCCNS(=O)(=O)c1ccc(N[C@H](C)CCC)c(C(=O)O)c1 ZINC000217544791 EF In-Stock Unstable CASP3 16 44 CCc1ccc(/C=C\C(=O)NC2CC(O)C2)cc1 ZINC000217544800 BD For-Sale Unstable HDAC8 56 44 CCc1ccc(/C=C\C(=O)NC2CC(O)C2)cc1 ZINC000217544800 BD For-Sale Unstable MMP2 0 46 CCc1ccc(/C=C\C(=O)NC2CC(O)C2)cc1 ZINC000217544800 BD For-Sale Unstable HDAC1 40 39 CCc1ccc(/C=C\C(=O)NC2CC(O)C2)cc1 ZINC000217544800 BD For-Sale Unstable HDAC6 37 40 COc1ccc(C(=O)[C@H](C)N)c(Cl)c1OC ZINC000217544817 BD For-Sale Unstable PDE4D 15 40 CCN(C(=O)NCCc1ccc(Br)cc1)c1ccccc1 ZINC000217544884 EI For-Sale Unstable AMP1_PLAFQ 23 41 Cc1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1Cl ZINC000217544885 GG For-Sale Unstable NPY5R 31 47 COc1ccc(C(=O)[C@@H](C)N)c(Cl)c1OC ZINC000217544900 BD For-Sale Unstable PDE4D 15 40 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)NCc1ccccc1 ZINC000217544912 FG For-Sale Unstable FABP4 47 35 Cc1ccc(Cl)cc1S(=O)(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217544977 GG For-Sale Unstable NPY5R 33 53 NCc1cccc(CNC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217545006 FF For-Sale Unstable TPSAB1 22 42 CCOC(=O)[C@@H]1CCCCN1C[C@@H](O)COC(C)C ZINC000217545043 CD On-Demand Unstable FKBP12.6 0 43 CCCNc1ccc(S(=O)(=O)NC(C)C)cc1C(=O)O ZINC000217545075 DD In-Stock Unstable LEF 49 35 O=C1OC2(CCN(S(=O)(=O)Cc3ccccc3Cl)CC2)c2ccccc21 ZINC000217545091 GG In-Stock Unstable NPY5R 34 47 CCOC(=O)[C@H]1CCCCN1C[C@@H](O)COC(C)C ZINC000217545109 CD On-Demand Unstable FKBP12.6 0 43 N#Cc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217545116 EH On-Demand Unstable IDO1 19 48 N#Cc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217545116 EH On-Demand Unstable P96878_MYCTU 15 45 N#Cc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217545116 EH On-Demand Unstable BLM 0 40 Cc1cccc(NC(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)c1 ZINC000217545160 FH For-Sale Unstable CCKAR 22 41 Cc1cccc(NC(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)c1 ZINC000217545160 FH For-Sale Unstable KCNK3 41 35 Cc1cccc(NC(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)c1 ZINC000217545160 FH For-Sale Unstable KCNK9 40 33 CC(C)Nc1ccc(S(=O)(=O)NC(C)C)cc1C(=O)O ZINC000217545191 DD In-Stock Unstable MMP13 23 40 CC(C)Nc1ccc(S(=O)(=O)NC(C)C)cc1C(=O)O ZINC000217545191 DD In-Stock Unstable MMP2 19 40 CC(C)Nc1ccc(S(=O)(=O)NC(C)C)cc1C(=O)O ZINC000217545191 DD In-Stock Unstable MMP12 50 39 CC(C)Nc1ccc(S(=O)(=O)NC(C)C)cc1C(=O)O ZINC000217545191 DD In-Stock Unstable LEF 46 36 O=C1OC2(CCN(S(=O)(=O)Cc3cccc(Cl)c3)CC2)c2ccccc21 ZINC000217545194 GG For-Sale Unstable SIGMAR1 15 57 O=C1OC2(CCN(S(=O)(=O)Cc3cccc(Cl)c3)CC2)c2ccccc21 ZINC000217545194 GG For-Sale Unstable NPY5R 31 48 O=C(NCC1C[C@@H]2CC[C@H](C1)N2)c1cccnc1 ZINC000217545211 BD For-Sale Unstable GRIN2B 15 44 O=C(NCC1C[C@@H]2CC[C@H](C1)N2)c1cccnc1 ZINC000217545211 BD For-Sale Unstable GLRA1 31 56 O=C(NCCc1ccc(Br)cc1)Nc1cc(Cl)ccc1O ZINC000217545229 FI For-Sale Unstable KCNMA1 21 46 O=C(NCCc1ccc(Br)cc1)Nc1cc(Cl)ccc1O ZINC000217545229 FI For-Sale Unstable NCE103 35 42 O=C(NCCc1ccc(Br)cc1)Nc1cc(Cl)ccc1O ZINC000217545229 FI For-Sale Unstable CAN2 0 42 Cc1ccc(NC(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc1 ZINC000217545266 FH For-Sale Unstable EPHX2 17 45 Cn1cc([C@H](C(=O)O)N2C[C@@H]3C[C@H](C2)Cn2c3cccc2=O)c2cc(C(=O)O)ccc21 ZINC000217545274 HE In-Stock Unstable CHRNA4 27 43 CCCCNc1ccc(S(=O)(=O)NC(C)C)cc1C(=O)O ZINC000217545300 DE In-Stock Unstable LEF 45 38 O=C1OC2(CCN(S(=O)(=O)c3cccc4ccccc34)CC2)c2ccccc21 ZINC000217545306 GH For-Sale Unstable HTR6 16 43 O=C1OC2(CCN(S(=O)(=O)c3cccc4ccccc34)CC2)c2ccccc21 ZINC000217545306 GH For-Sale Unstable NPY5R 35 49 Cn1cc([C@@H](C(=O)O)N2C[C@@H]3C[C@H](C2)Cn2c3cccc2=O)c2cc(C(=O)O)ccc21 ZINC000217545359 HE In-Stock Unstable CHRNA4 27 43 CCOc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1OCC ZINC000217545375 HJ On-Demand Unstable AGPAT2 40 43 CC(C)CNc1ccc(S(=O)(=O)NC(C)C)cc1C(=O)O ZINC000217545399 DE In-Stock Unstable BDKRB1 0 40 CC(C)CNc1ccc(S(=O)(=O)NC(C)C)cc1C(=O)O ZINC000217545399 DE In-Stock Unstable MMP12 40 36 CC(C)CNc1ccc(S(=O)(=O)NC(C)C)cc1C(=O)O ZINC000217545399 DE In-Stock Unstable MTNN 75 35 CC(C)CNc1ccc(S(=O)(=O)NC(C)C)cc1C(=O)O ZINC000217545399 DE In-Stock Unstable LEF 48 34 O=C1OC2(CCN(S(=O)(=O)c3ccc4c(c3)CCCC4)CC2)c2ccccc21 ZINC000217545424 GG For-Sale Unstable NPY5R 29 42 O=C1OC2(CCN(S(=O)(=O)c3ccc4c(c3)CCCC4)CC2)c2ccccc21 ZINC000217545424 GG For-Sale Unstable AKR1C3 43 36 CCOC(=O)[C@@H]1CCCCN1C[C@@H](O)c1ccccc1 ZINC000217545429 CE On-Demand Unstable SLC6A3 27 47 CCOC(=O)[C@@H]1CCCCN1C[C@@H](O)c1ccccc1 ZINC000217545429 CE On-Demand Unstable AMY2 46 32 CCOC(=O)[C@@H]1CCCCN1C[C@@H](O)c1ccccc1 ZINC000217545429 CE On-Demand Unstable FKBP12.6 0 48 CCOC(=O)[C@@H]1CCCCN1C[C@@H](O)c1ccccc1 ZINC000217545429 CE On-Demand Unstable POL 0 44 CCOC(=O)[C@@H]1CCCCN1C[C@@H](O)c1ccccc1 ZINC000217545429 CE On-Demand Unstable Q8WSF8_APLCA 24 40 c1ccc(-c2ccc(N[C@H]3C[C@@H]4CC[C@H]3C4)cc2)cc1 ZINC000217545476 CJ For-Sale Unstable BRS3 24 41 CSc1cccc(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217545481 FJ On-Demand Unstable CCR3 27 51 CSc1cccc(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217545481 FJ On-Demand Unstable RAF1 23 42 CCOC(=O)[C@H]1CCCCN1C[C@@H](O)c1ccccc1 ZINC000217545502 CE On-Demand Unstable SLC6A3 27 47 CCOC(=O)[C@H]1CCCCN1C[C@@H](O)c1ccccc1 ZINC000217545502 CE On-Demand Unstable AMY2 46 32 CCOC(=O)[C@H]1CCCCN1C[C@@H](O)c1ccccc1 ZINC000217545502 CE On-Demand Unstable FKBP12.6 0 48 CCOC(=O)[C@H]1CCCCN1C[C@@H](O)c1ccccc1 ZINC000217545502 CE On-Demand Unstable POL 0 44 CCOC(=O)[C@H]1CCCCN1C[C@@H](O)c1ccccc1 ZINC000217545502 CE On-Demand Unstable Q8WSF8_APLCA 24 40 CC[C@@H](C)Nc1ccc(S(=O)(=O)NC(C)C)cc1C(=O)O ZINC000217545520 DE In-Stock Unstable LEF 46 38 CC(C)(C)c1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217545530 GH For-Sale Unstable HSD11B1 20 52 CC(C)(C)c1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217545530 GH For-Sale Unstable NPY5R 31 45 c1ccc(-c2ccc(N[C@H]3C[C@H]4CC[C@H]3C4)cc2)cc1 ZINC000217545571 CJ For-Sale Unstable BRS3 24 41 CC[C@H](C)Nc1ccc(S(=O)(=O)NC(C)C)cc1C(=O)O ZINC000217545606 DE In-Stock Unstable LEF 46 38 O=C(NCCc1ccc(Br)cc1)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217545607 KG For-Sale Unstable MURF 0 43 O=C(NCCc1ccc(Br)cc1)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217545607 KG For-Sale Unstable NAMPT 35 43 O=C(NCCc1ccccc1)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217545608 GG For-Sale Unstable FABP4 45 34 C[C@@H]1CN(c2cc(Cl)ccc2CBr)CCN1C ZINC000217545617 DG For-Sale Unstable ADRA2B 0 45 C[C@@H]1CN(c2cc(Cl)ccc2CBr)CCN1C ZINC000217545617 DG For-Sale Unstable ADRA2C 0 45 CC(=O)Nc1ccc(CN2CCN(C)[C@@H](c3ccccc3)C2)cc1 ZINC000217545636 DG In-Stock Unstable TSHR 48 32 CC(=O)Nc1ccc(CN2CCN(C)[C@@H](c3ccccc3)C2)cc1 ZINC000217545636 DG In-Stock Unstable DRD4 41 41 CC(=O)Nc1ccc(CN2CCN(C)[C@@H](c3ccccc3)C2)cc1 ZINC000217545636 DG In-Stock Unstable DRD3 0 42 CC(=O)Nc1ccc(CN2CCN(C)[C@@H](c3ccccc3)C2)cc1 ZINC000217545636 DG In-Stock Unstable LTA4H 25 42 CC(=O)Nc1ccc(CN2CCN(C)[C@@H](c3ccccc3)C2)cc1 ZINC000217545636 DG In-Stock Unstable SIGMAR1 33 40 CC(=O)Nc1ccc(CN2CCN(C)[C@@H](c3ccccc3)C2)cc1 ZINC000217545636 DG In-Stock Unstable PRNP 40 36 CC(=O)Nc1ccc(CN2CCN(C)[C@@H](c3ccccc3)C2)cc1 ZINC000217545636 DG In-Stock Unstable MCHR1 35 43 CC(=O)Nc1ccc(CN2CCN(C)[C@@H](c3ccccc3)C2)cc1 ZINC000217545636 DG In-Stock Unstable NOD1 31 40 CC(=O)Nc1ccc(CN2CCN(C)[C@@H](c3ccccc3)C2)cc1 ZINC000217545636 DG In-Stock Unstable NOD2 47 40 Cc1cc(C)c(C)c(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1C ZINC000217545647 GH For-Sale Unstable NPY5R 31 48 NS(=O)(=O)c1ccc(CNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217545684 HE On-Demand Unstable CA2 148 65 NS(=O)(=O)c1ccc(CNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217545684 HE On-Demand Unstable CA6 24 45 NS(=O)(=O)c1ccc(CNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217545684 HE On-Demand Unstable CA1 128 65 NS(=O)(=O)c1ccc(CNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217545684 HE On-Demand Unstable CA7 77 65 NS(=O)(=O)c1ccc(CNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217545684 HE On-Demand Unstable CA13 36 45 NS(=O)(=O)c1ccc(CNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217545684 HE On-Demand Unstable CA5B 63 54 NS(=O)(=O)c1ccc(CNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217545684 HE On-Demand Unstable CA4 98 65 NS(=O)(=O)c1ccc(CNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217545684 HE On-Demand Unstable CA5A 65 54 NS(=O)(=O)c1ccc(CNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217545684 HE On-Demand Unstable CA14 62 65 NS(=O)(=O)c1ccc(CNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217545684 HE On-Demand Unstable CA12 99 65 NS(=O)(=O)c1ccc(CNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217545684 HE On-Demand Unstable CA9 110 65 NS(=O)(=O)c1ccc(CNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217545684 HE On-Demand Unstable CAH_METTE 30 44 NS(=O)(=O)c1ccc(CNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217545684 HE On-Demand Unstable IDO1 15 42 NS(=O)(=O)c1ccc(CNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217545684 HE On-Demand Unstable CYNT 41 51 NS(=O)(=O)c1ccc(CNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217545684 HE On-Demand Unstable NCE103 47 55 NS(=O)(=O)c1ccc(CNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217545684 HE On-Demand Unstable ALPI 24 54 NS(=O)(=O)c1ccc(CNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217545684 HE On-Demand Unstable LIG1 0 64 NS(=O)(=O)c1ccc(CNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217545684 HE On-Demand Unstable CA15 18 45 NS(=O)(=O)c1ccc(CNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217545684 HE On-Demand Unstable MTCA1 55 51 NS(=O)(=O)c1ccc(CNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217545684 HE On-Demand Unstable P96878_MYCTU 69 51 NS(=O)(=O)c1ccc(CNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217545684 HE On-Demand Unstable CA 0 47 NS(=O)(=O)c1ccc(CNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217545684 HE On-Demand Unstable A6YCJ1_9METZ 30 58 NS(=O)(=O)c1ccc(CNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217545684 HE On-Demand Unstable Q5TU56_ANOGA 0 45 C[C@H]1CN(c2cc(Cl)ccc2CBr)CCN1C ZINC000217545689 DG For-Sale Unstable ADRA2B 0 45 C[C@H]1CN(c2cc(Cl)ccc2CBr)CCN1C ZINC000217545689 DG For-Sale Unstable ADRA2C 0 45 Cc1ccc(NC(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc1C ZINC000217545697 GI For-Sale Unstable EPHX2 16 42 CC(C)NS(=O)(=O)c1ccc(NC(C)(C)C)c(C(=O)O)c1 ZINC000217545717 DE In-Stock Unstable PRTN3 52 35 CC(C)NS(=O)(=O)c1ccc(NC(C)(C)C)c(C(=O)O)c1 ZINC000217545717 DE In-Stock Unstable MMP12 46 37 CC(C)NS(=O)(=O)c1ccc(NC(C)(C)C)c(C(=O)O)c1 ZINC000217545717 DE In-Stock Unstable LEF 41 34 CC(=O)Nc1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217545745 HE For-Sale Unstable LPL 43 33 CC(=O)Nc1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217545745 HE For-Sale Unstable NPY5R 53 47 CC(=O)Nc1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217545745 HE For-Sale Unstable TGM2 65 39 CC(=O)Nc1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217545745 HE For-Sale Unstable F13A1 92 40 CC(=O)Nc1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217545745 HE For-Sale Unstable NAMPT 26 40 C[C@@H]1C[C@@H](C)CN(C(=O)NCCc2ccc(Br)cc2)C1 ZINC000217545800 EH On-Demand Unstable GPBAR1 22 43 C=CCNc1ccc(S(=O)(=O)NC(C)C)cc1C(=O)O ZINC000217545816 CD In-Stock Unstable ADAMTS4 44 34 C[C@@H]1CN(c2ccc(Cl)cc2CBr)CCN1C ZINC000217545821 DG For-Sale Unstable ADRA2B 0 43 C[C@@H]1CN(c2ccc(Cl)cc2CBr)CCN1C ZINC000217545821 DG For-Sale Unstable ADRA2C 0 43 O=C1OC2(CCN(S(=O)(=O)c3ccc4c(c3)OCCO4)CC2)c2ccccc21 ZINC000217545846 HE In-Stock Unstable NPY5R 29 45 O=C1OC2(CCN(S(=O)(=O)c3ccc4c(c3)OCCO4)CC2)c2ccccc21 ZINC000217545846 HE In-Stock Unstable PKM 54 60 C[C@H]1C[C@@H](C)CN(C(=O)NCCc2ccc(Br)cc2)C1 ZINC000217545876 EH On-Demand Unstable GPBAR1 22 43 C[C@H]1CN(c2ccc(Cl)cc2CBr)CCN1C ZINC000217545878 DG For-Sale Unstable ADRA2B 0 43 C[C@H]1CN(c2ccc(Cl)cc2CBr)CCN1C ZINC000217545878 DG For-Sale Unstable ADRA2C 0 43 C[C@@H]1CCC[C@@](NC(=O)/C=C\c2ccccc2)(C(=O)O)C1 ZINC000217545882 CF For-Sale Unstable MMP2 16 40 C[C@@H]1CCC[C@@](NC(=O)/C=C\c2ccccc2)(C(=O)O)C1 ZINC000217545882 CF For-Sale Unstable HDAC6 24 43 O=C(NCC[C@H](O)c1ccsc1)Nc1ccccc1Cl ZINC000217545888 DH In-Stock Unstable CXCL8 41 35 CC(C)NS(=O)(=O)c1ccc(NC2CC2)c(C(=O)O)c1 ZINC000217545907 CD In-Stock Unstable MMP2 17 40 CC(C)NS(=O)(=O)c1ccc(NC2CC2)c(C(=O)O)c1 ZINC000217545907 CD In-Stock Unstable LEF 40 41 COc1cccc(NC(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)c1 ZINC000217545916 GH For-Sale Unstable DRD4 47 37 COc1cccc(NC(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)c1 ZINC000217545916 GH For-Sale Unstable HRH2 23 46 COc1cccc(NC(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)c1 ZINC000217545916 GH For-Sale Unstable CCR3 45 47 COc1cccc(NC(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)c1 ZINC000217545916 GH For-Sale Unstable EPHX2 29 42 COc1cccc(NC(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)c1 ZINC000217545916 GH For-Sale Unstable TAAR1 44 42 C[C@H]1C[C@H](C)CN(C(=O)NCCc2ccc(Br)cc2)C1 ZINC000217545949 EH On-Demand Unstable GPBAR1 22 43 C[C@H]1CCC[C@@](NC(=O)/C=C\c2ccccc2)(C(=O)O)C1 ZINC000217545950 CF For-Sale Unstable MMP2 16 40 C[C@H]1CCC[C@@](NC(=O)/C=C\c2ccccc2)(C(=O)O)C1 ZINC000217545950 CF For-Sale Unstable HDAC6 24 43 COc1cc(C)c(C)cc1S(=O)(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217545953 HG For-Sale Unstable NPY5R 31 51 O=C(NCC[C@@H](O)c1ccsc1)Nc1ccccc1Cl ZINC000217545968 DH In-Stock Unstable CXCL8 41 35 O=C(COCc1ccccc1)N1CCn2nc(CO)cc2C1 ZINC000217546002 DC In-Stock Unstable GRM5 0 53 CC(C)NS(=O)(=O)c1ccc(NC2CCCC2)c(C(=O)O)c1 ZINC000217546009 EE In-Stock Unstable MMP13 19 41 CC(C)NS(=O)(=O)c1ccc(NC2CCCC2)c(C(=O)O)c1 ZINC000217546009 EE In-Stock Unstable LEF 34 43 COc1ccc(NC(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc1 ZINC000217546023 GH For-Sale Unstable EPHX2 28 43 O=C(NCCc1ccc(Br)cc1)Nc1ncccn1 ZINC000217546052 DF For-Sale Unstable NCE103 15 40 CCOc1ccc(C)cc1S(=O)(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217546061 HG For-Sale Unstable NPY5R 30 44 CC(C)NS(=O)(=O)c1ccc(NC2CCCCC2)c(C(=O)O)c1 ZINC000217546114 EF In-Stock Unstable MMP13 18 43 CC(C)NS(=O)(=O)c1ccc(NC2CCCCC2)c(C(=O)O)c1 ZINC000217546114 EF In-Stock Unstable LEF 34 44 O=C(/C=C\c1ccc(Cl)c(Cl)c1)NC1CC(O)C1 ZINC000217546148 CF For-Sale Unstable PYGL 32 56 O=C(/C=C\c1ccc(Cl)c(Cl)c1)NC1CC(O)C1 ZINC000217546148 CF For-Sale Unstable HDAC8 22 45 O=C(/C=C\c1ccc(Cl)c(Cl)c1)NC1CC(O)C1 ZINC000217546148 CF For-Sale Unstable MMP2 0 41 O=C(/C=C\c1ccc(Cl)c(Cl)c1)NC1CC(O)C1 ZINC000217546148 CF For-Sale Unstable HDAC1 36 45 O=C(/C=C\c1ccc(Cl)c(Cl)c1)NC1CC(O)C1 ZINC000217546148 CF For-Sale Unstable HDAC2 0 45 O=C(/C=C\c1ccc(Cl)c(Cl)c1)NC1CC(O)C1 ZINC000217546148 CF For-Sale Unstable CCR2 0 45 CN(C(=O)NCCc1ccc(Br)cc1)c1ccccc1 ZINC000217546149 EH For-Sale Unstable AMP1_PLAFQ 28 43 O=[N+]([O-])c1ccc(OCCOCc2ccccc2)c(C(F)(F)F)c1 ZINC000217546160 EI In-Stock Unstable S1PR4 18 42 O=[N+]([O-])c1ccc(OCCOCc2ccccc2)c(C(F)(F)F)c1 ZINC000217546160 EI In-Stock Unstable F2RL3 40 41 CN1CC[C@@H](NC(=S)Nc2ccccc2)C1=O ZINC000217546164 BD On-Demand Unstable EPHX1 0 42 CCOc1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1C ZINC000217546169 HG For-Sale Unstable PDE5A 35 41 CCOc1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1C ZINC000217546169 HG For-Sale Unstable NPY5R 28 42 CCCCCCCCNC[C@@H](C)N(C)C1CC1 ZINC000217546207 BG For-Sale Unstable Q8WS26_TRYCR 35 41 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)Nc1ccc(Cl)cc1 ZINC000217546226 GI For-Sale Unstable EPHX2 22 46 O=C(NCCc1ccc(Br)cc1)N1CCCCCC1 ZINC000217546248 EH On-Demand Unstable DPP7 54 41 O=C(NCCc1ccc(Br)cc1)N1CCCCCC1 ZINC000217546248 EH On-Demand Unstable GPBAR1 24 43 O=C(NCCc1ccc(Br)cc1)N1CCCCCC1 ZINC000217546248 EH On-Demand Unstable LIG1 0 40 CN1CC[C@H](NC(=S)Nc2ccccc2)C1=O ZINC000217546256 BD On-Demand Unstable EPHX1 0 42 O=C(O)c1ccc2c(c1)c([C@H](C(=O)O)N1C[C@@H]3C[C@H](C1)Cn1c3cccc1=O)cn2Cc1ccccc1 ZINC000217546270 JH In-Stock Unstable CHRNA4 27 49 COc1c(C)cc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1C ZINC000217546289 HG For-Sale Unstable NPY5R 29 45 CCCCCCCCNC[C@H](C)N(C)C1CC1 ZINC000217546291 BG For-Sale Unstable Q8WS26_TRYCR 35 41 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)Nc1cccc(Cl)c1 ZINC000217546327 GI For-Sale Unstable EPHX2 20 44 CC(C)NS(=O)(=O)c1ccc(NCCO)c(C(=O)O)c1 ZINC000217546339 DC In-Stock Unstable LEF 48 33 O=C(O)c1ccc2c(c1)c([C@@H](C(=O)O)N1C[C@@H]3C[C@H](C1)Cn1c3cccc1=O)cn2Cc1ccccc1 ZINC000217546363 JH In-Stock Unstable CHRNA4 27 49 CCCCN(CCC)C(=O)NCCc1ccc(Br)cc1 ZINC000217546366 EI For-Sale Unstable LIG1 0 40 Cc1ccc(/C=C\C(=O)NC2CC(O)C2)cc1 ZINC000217546394 BD For-Sale Unstable HDAC8 58 43 Cc1ccc(/C=C\C(=O)NC2CC(O)C2)cc1 ZINC000217546394 BD For-Sale Unstable MMP2 0 46 Cc1ccc(/C=C\C(=O)NC2CC(O)C2)cc1 ZINC000217546394 BD For-Sale Unstable HDAC1 33 47 Cc1ccc(/C=C\C(=O)NC2CC(O)C2)cc1 ZINC000217546394 BD For-Sale Unstable HDAC2 0 40 Cc1ccc(/C=C\C(=O)NC2CC(O)C2)cc1 ZINC000217546394 BD For-Sale Unstable HDAC4 25 47 Cc1ccc(/C=C\C(=O)NC2CC(O)C2)cc1 ZINC000217546394 BD For-Sale Unstable HDAC6 38 44 Cc1ccc(/C=C\C(=O)NC2CC(O)C2)cc1 ZINC000217546394 BD For-Sale Unstable HK2 0 42 Cc1ccc(/C=C\C(=O)NC2CC(O)C2)cc1 ZINC000217546394 BD For-Sale Unstable MMP9 0 49 Cc1ccc(/C=C\C(=O)NC2CC(O)C2)cc1 ZINC000217546394 BD For-Sale Unstable MMP1 0 49 Cc1ccc(/C=C\C(=O)NC2CC(O)C2)cc1 ZINC000217546394 BD For-Sale Unstable HD1B 0 43 CCc1ccc(OC)c(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217546401 HG For-Sale Unstable NPY5R 30 45 CC(C)NS(=O)(=O)c1ccc(NCCCO)c(C(=O)O)c1 ZINC000217546448 DC In-Stock Unstable LEF 43 32 C[C@H](C(=O)c1cccc(Cl)c1)N1CCC[C@@H](O)C1 ZINC000217546461 CE For-Sale Unstable GRM5 18 40 O=C(NCCOc1ccccc1)NCC[C@H](O)c1ccsc1 ZINC000217546470 DF In-Stock Unstable ADRB3 15 40 COc1ccc2c(c1OC)O[C@@H](C(=O)O)C2 ZINC000217546472 BD In-Stock Unstable AGTR2 53 37 COc1ccc2c(c1OC)O[C@@H](C(=O)O)C2 ZINC000217546472 BD In-Stock Unstable MT-ND4 40 31 CCCCCNC(=O)NCCc1ccc(Br)cc1 ZINC000217546488 DG On-Demand Unstable S1PR2 48 41 CCCCCNC(=O)NCCc1ccc(Br)cc1 ZINC000217546488 DG On-Demand Unstable EPHX2 37 42 CCCCCNC(=O)NCCc1ccc(Br)cc1 ZINC000217546488 DG On-Demand Unstable ASAH1 74 37 CCCCCNC(=O)NCCc1ccc(Br)cc1 ZINC000217546488 DG On-Demand Unstable LIG1 0 41 CCCCCNC(=O)NCCc1ccc(Br)cc1 ZINC000217546488 DG On-Demand Unstable ACAT 0 52 COc1ccc(CCS(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217546518 HF For-Sale Unstable NPY5R 30 42 C[C@@H](C(=O)c1cccc(Cl)c1)N1CCC[C@@H](O)C1 ZINC000217546537 CE For-Sale Unstable GRM5 18 40 COCCNc1ccc(S(=O)(=O)NC(C)C)cc1C(=O)O ZINC000217546538 DD In-Stock Unstable LEF 43 33 O=C(NCCOc1ccccc1)NCC[C@@H](O)c1ccsc1 ZINC000217546553 DF In-Stock Unstable ADRB3 15 40 COc1ccc2c(c1OC)O[C@H](C(=O)O)C2 ZINC000217546556 BD In-Stock Unstable AGTR2 53 37 COc1ccc2c(c1OC)O[C@H](C(=O)O)C2 ZINC000217546556 BD In-Stock Unstable MT-ND4 40 31 O=C(O)c1ccc2c([C@H](C(=O)O)N3C[C@@H]4C[C@H](C3)Cn3c4cccc3=O)cn(Cc3ccccc3)c2c1 ZINC000217546601 JH In-Stock Unstable CHRNA4 28 50 O=C(O)Cc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217546604 GG On-Demand Unstable CA1 15 51 O=C(O)Cc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217546604 GG On-Demand Unstable CA9 15 51 O=C(O)Cc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217546604 GG On-Demand Unstable IDO1 18 44 O=C(O)Cc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217546604 GG On-Demand Unstable NCE103 24 51 O=C(O)Cc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217546604 GG On-Demand Unstable P96878_MYCTU 15 40 OC[C@H]1O[C@@H](O)[C@H](F)[C@H]1O ZINC000217546613 AA For-Sale Unstable CDA 49 42 COc1ccc(OC)c(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c1 ZINC000217546630 HF For-Sale Unstable NPY5R 34 51 C[C@H](C(=O)c1ccc(Cl)cc1)N1CCC[C@@H](O)C1 ZINC000217546642 CE For-Sale Unstable SLC6A1 44 48 C[C@H](C(=O)c1ccc(Cl)cc1)N1CCC[C@@H](O)C1 ZINC000217546642 CE For-Sale Unstable SLC6A3 18 48 C[C@H](C(=O)c1ccc(Cl)cc1)N1CCC[C@@H](O)C1 ZINC000217546642 CE For-Sale Unstable CCR1 41 38 COCCCNc1ccc(S(=O)(=O)NC(C)C)cc1C(=O)O ZINC000217546649 ED In-Stock Unstable BDKRB1 15 40 CC[C@H](C)[C@@H]1NC(=O)[C@@H](C(C)C)N(CC[S@@](=O)CC)C1=O ZINC000217546659 DD For-Sale Unstable GALR1 47 37 COc1ccc(CCNC(=O)NCC[C@H](O)c2ccsc2)cc1 ZINC000217546671 EF In-Stock Unstable ADRB2 15 47 COc1ccc(CCNC(=O)NCC[C@H](O)c2ccsc2)cc1 ZINC000217546671 EF In-Stock Unstable ADRB3 22 41 O=C(NCCCc1ccccc1)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217546674 GH For-Sale Unstable FABP4 44 33 O=C(O)c1ccc2c([C@@H](C(=O)O)N3C[C@@H]4C[C@H](C3)Cn3c4cccc3=O)cn(Cc3ccccc3)c2c1 ZINC000217546680 JH In-Stock Unstable CHRNA4 28 50 COc1ccc(OC)c2c1C[C@H](C(=O)O)O2 ZINC000217546683 BD In-Stock Unstable MT-ND4 54 34 C[C@@H](C(=O)c1ccc(Cl)cc1)N1CCC[C@@H](O)C1 ZINC000217546724 CE For-Sale Unstable SLC6A1 44 48 C[C@@H](C(=O)c1ccc(Cl)cc1)N1CCC[C@@H](O)C1 ZINC000217546724 CE For-Sale Unstable SLC6A3 18 48 C[C@@H](C(=O)c1ccc(Cl)cc1)N1CCC[C@@H](O)C1 ZINC000217546724 CE For-Sale Unstable CCR1 41 38 O=C(NCCc1ccc(Br)cc1)NCc1ccc(C(=O)O)cc1 ZINC000217546727 GG On-Demand Unstable LIG1 0 40 COc1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1OC ZINC000217546739 HF For-Sale Unstable NPY5R 30 46 COc1ccc(CCNC(=O)NCC[C@@H](O)c2ccsc2)cc1 ZINC000217546744 EF In-Stock Unstable ADRB2 15 47 COc1ccc(CCNC(=O)NCC[C@@H](O)c2ccsc2)cc1 ZINC000217546744 EF In-Stock Unstable ADRB3 22 41 COc1ccc(OC)c2c1C[C@@H](C(=O)O)O2 ZINC000217546753 BD In-Stock Unstable MT-ND4 54 34 CC(C)NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217546772 EF In-Stock Unstable TRY2_BOVIN 56 34 CC(C)NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217546772 EF In-Stock Unstable MMP9 23 40 CC(C)NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217546772 EF In-Stock Unstable MMP12 50 40 CC(C)NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217546772 EF In-Stock Unstable ADAMTS4 56 38 CC(C)NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217546772 EF In-Stock Unstable ACPS 0 40 CC(C)NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217546772 EF In-Stock Unstable LEF 40 37 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)Nc1ccc2c(c1)OCO2 ZINC000217546798 GG For-Sale Unstable NOS2 57 31 N#Cc1cccc(/C=C\C(=O)NC2CC(O)C2)c1 ZINC000217546816 BD For-Sale Unstable HDAC8 43 35 N#Cc1cccc(/C=C\C(=O)NC2CC(O)C2)c1 ZINC000217546816 BD For-Sale Unstable MMP2 0 41 CCc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217546834 EI For-Sale Unstable CA1 17 46 CCc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217546834 EI For-Sale Unstable CA12 17 49 CCc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217546834 EI For-Sale Unstable CA9 19 49 CCc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217546834 EI For-Sale Unstable IDO1 20 40 CCc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217546834 EI For-Sale Unstable NCE103 27 49 CCc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217546834 EI For-Sale Unstable LIG1 0 40 CCc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217546834 EI For-Sale Unstable P96878_MYCTU 17 41 CCOc1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1F ZINC000217546841 HG For-Sale Unstable NPY5R 31 42 CCOc1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1F ZINC000217546841 HG For-Sale Unstable PKM 40 38 O=C(NCC[C@@H](O)c1ccsc1)NC12CC3CC(CC(C3)C1)C2 ZINC000217546847 EG In-Stock Unstable EPHX2 99 51 COc1ccc(C(=O)[C@@H](C)N2CCC[C@@H](O)C2)cc1 ZINC000217546861 CD For-Sale Unstable GRM3 18 54 CC(C)NS(=O)(=O)c1ccc(N[C@@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217546878 FG In-Stock Unstable LEF 30 42 O=C(NCC[C@H](O)c1ccsc1)NC12CC3CC(CC(C3)C1)C2 ZINC000217546912 EG In-Stock Unstable EPHX2 99 51 COc1ccc(C(=O)[C@H](C)N2CCC[C@@H](O)C2)cc1 ZINC000217546924 CD For-Sale Unstable GRM3 18 54 COC(=O)c1sccc1S(=O)(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217546951 HE For-Sale Unstable NPY5R 40 49 CCOc1ccc(NC(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc1 ZINC000217546953 GI For-Sale Unstable EPHX2 27 42 CC(C)NS(=O)(=O)c1ccc(N[C@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217546965 FG In-Stock Unstable LEF 30 42 CN(C)c1ccc(/C=C\C(=O)NC2CC(O)C2)cc1 ZINC000217547039 CD For-Sale Unstable HDAC8 26 43 CN(C)c1ccc(/C=C\C(=O)NC2CC(O)C2)cc1 ZINC000217547039 CD For-Sale Unstable MMP2 0 44 CN(C)c1ccc(/C=C\C(=O)NC2CC(O)C2)cc1 ZINC000217547039 CD For-Sale Unstable HDAC1 42 41 CN(C)c1ccc(/C=C\C(=O)NC2CC(O)C2)cc1 ZINC000217547039 CD For-Sale Unstable HDAC4 0 40 CN(C)c1ccc(/C=C\C(=O)NC2CC(O)C2)cc1 ZINC000217547039 CD For-Sale Unstable HDA106 0 41 CN(C)c1ccc(/C=C\C(=O)NC2CC(O)C2)cc1 ZINC000217547039 CD For-Sale Unstable HD1B 0 40 COc1ccc(Cl)cc1S(=O)(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217547044 HG For-Sale Unstable CPT1A 73 41 COc1ccc(Cl)cc1S(=O)(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217547044 HG For-Sale Unstable CPT2 49 39 COc1ccc(Cl)cc1S(=O)(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217547044 HG For-Sale Unstable NPY5R 31 50 COc1ccc(Cl)cc1S(=O)(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217547044 HG For-Sale Unstable CPT1B 59 39 c1cc(CNC2CC2)c2c(c1)OCC2 ZINC000217547051 AD In-Stock Unstable MTNR1A 33 43 c1cc(CNC2CC2)c2c(c1)OCC2 ZINC000217547051 AD In-Stock Unstable MTNR1B 23 43 CC(C)NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217547062 FF In-Stock Unstable ADRB3 44 38 CC(C)NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217547062 FF In-Stock Unstable TRY2_BOVIN 51 33 CC(C)NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217547062 FF In-Stock Unstable BDKRB1 15 40 CC(C)NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217547062 FF In-Stock Unstable MMP8 17 43 CC(C)NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217547062 FF In-Stock Unstable PRTN3 44 32 CC(C)NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217547062 FF In-Stock Unstable MMP12 44 36 CC(C)NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217547062 FF In-Stock Unstable ADAMTS4 52 35 CC(C)NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217547062 FF In-Stock Unstable AKR1C3 16 47 CC1(C)CC(NC(=O)NCCc2ccc(Br)cc2)CC(C)(C)N1 ZINC000217547069 GH On-Demand Unstable EZH2 52 38 CC1(C)CC(NC(=O)NCCc2ccc(Br)cc2)CC(C)(C)N1 ZINC000217547069 GH On-Demand Unstable HIV1_ENV 0 41 Cc1nonc1CC(=O)N1CCC(Oc2cccc(C(F)(F)F)c2)CC1 ZINC000217547148 FG In-Stock Unstable HRH1 29 42 Cc1nonc1CC(=O)N1CCC(Oc2cccc(C(F)(F)F)c2)CC1 ZINC000217547148 FG In-Stock Unstable PRSS2 45 32 Cc1nonc1CC(=O)N1CCC(Oc2cccc(C(F)(F)F)c2)CC1 ZINC000217547148 FG In-Stock Unstable CCR3 23 43 Cc1nonc1CC(=O)N1CCC(Oc2cccc(C(F)(F)F)c2)CC1 ZINC000217547148 FG In-Stock Unstable BRS3 20 42 Cc1nonc1CC(=O)N1CCC(Oc2cccc(C(F)(F)F)c2)CC1 ZINC000217547148 FG In-Stock Unstable CCR2 48 38 Cc1nonc1CC(=O)N1CCC(Oc2cccc(C(F)(F)F)c2)CC1 ZINC000217547148 FG In-Stock Unstable LIPG 58 38 O=C(NCCOc1ccccc1)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217547150 GG For-Sale Unstable HRH2 24 42 O=C1OC2(CCN(S(=O)(=O)c3cccc(C(F)(F)F)c3)CC2)c2ccccc21 ZINC000217547161 HH For-Sale Unstable CACNA1B 47 45 O=C1OC2(CCN(S(=O)(=O)c3cccc(C(F)(F)F)c3)CC2)c2ccccc21 ZINC000217547161 HH For-Sale Unstable NPY5R 30 52 O=C1OC2(CCN(S(=O)(=O)c3cccc(C(F)(F)F)c3)CC2)c2ccccc21 ZINC000217547161 HH For-Sale Unstable PKM 31 54 Cc1ccc(O)c(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217547172 EH For-Sale Unstable RAF1 30 41 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)C)cc2C(=O)O)cc1 ZINC000217547183 GF In-Stock Unstable CA2 17 42 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)C)cc2C(=O)O)cc1 ZINC000217547183 GF In-Stock Unstable BMP1 95 40 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)C)cc2C(=O)O)cc1 ZINC000217547183 GF In-Stock Unstable CA1 18 43 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)C)cc2C(=O)O)cc1 ZINC000217547183 GF In-Stock Unstable MMP13 78 47 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)C)cc2C(=O)O)cc1 ZINC000217547183 GF In-Stock Unstable MMP2 52 43 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)C)cc2C(=O)O)cc1 ZINC000217547183 GF In-Stock Unstable MMP3 55 43 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)C)cc2C(=O)O)cc1 ZINC000217547183 GF In-Stock Unstable MMP8 37 43 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)C)cc2C(=O)O)cc1 ZINC000217547183 GF In-Stock Unstable PRTN3 44 31 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)C)cc2C(=O)O)cc1 ZINC000217547183 GF In-Stock Unstable MMP9 54 47 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)C)cc2C(=O)O)cc1 ZINC000217547183 GF In-Stock Unstable MMP12 51 40 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)C)cc2C(=O)O)cc1 ZINC000217547183 GF In-Stock Unstable PTGDR 26 43 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)C)cc2C(=O)O)cc1 ZINC000217547183 GF In-Stock Unstable MMP7 41 40 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)C)cc2C(=O)O)cc1 ZINC000217547183 GF In-Stock Unstable IAP 0 40 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)C)cc2C(=O)O)cc1 ZINC000217547183 GF In-Stock Unstable ADAMTS4 61 37 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)C)cc2C(=O)O)cc1 ZINC000217547183 GF In-Stock Unstable CA9 25 43 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)C)cc2C(=O)O)cc1 ZINC000217547183 GF In-Stock Unstable MMP1 54 41 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)C)cc2C(=O)O)cc1 ZINC000217547183 GF In-Stock Unstable AKR1C3 31 42 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)C)cc2C(=O)O)cc1 ZINC000217547183 GF In-Stock Unstable LEF 17 41 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)C)cc2C(=O)O)cc1 ZINC000217547183 GF In-Stock Unstable AKR1C2 51 38 O=C(NCC[C@H](O)c1ccsc1)Nc1cccc(C(F)(F)F)c1 ZINC000217547239 EI In-Stock Unstable CCR3 17 45 O=C1OC2(CCN(S(=O)(=O)c3cc(Cl)ccc3Cl)CC2)c2ccccc21 ZINC000217547269 HH For-Sale Unstable NPY5R 34 55 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)C)cc2C(=O)O)cc1OC ZINC000217547281 HF In-Stock Unstable MMP12 45 34 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)C)cc2C(=O)O)cc1OC ZINC000217547281 HF In-Stock Unstable PTGDR 20 41 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)C)cc2C(=O)O)cc1OC ZINC000217547281 HF In-Stock Unstable IAP 0 42 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)C)cc2C(=O)O)cc1OC ZINC000217547281 HF In-Stock Unstable ADAMTS4 53 33 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)C)cc2C(=O)O)cc1OC ZINC000217547281 HF In-Stock Unstable SCMU_MYCTU 0 46 Cc1cc(C)c(C[C@H](N)C(=O)O)c(O)c1Cl ZINC000217547295 BD For-Sale Unstable OPRM1 19 47 Cc1cc(C)c(C[C@H](N)C(=O)O)c(O)c1Cl ZINC000217547295 BD For-Sale Unstable GRIA3 58 41 Cc1cc(C)c(C[C@H](N)C(=O)O)c(O)c1Cl ZINC000217547295 BD For-Sale Unstable GRIA1 40 41 Cc1cc(C)c(C[C@H](N)C(=O)O)c(O)c1Cl ZINC000217547295 BD For-Sale Unstable GRIA2 48 41 Cc1cc(C)c(C[C@H](N)C(=O)O)c(O)c1Cl ZINC000217547295 BD For-Sale Unstable GRIA4 48 41 Cc1cc(C)c(C[C@H](N)C(=O)O)c(O)c1Cl ZINC000217547295 BD For-Sale Unstable GRIK1 39 41 O=C(NCC[C@@H](O)c1ccsc1)Nc1cccc(C(F)(F)F)c1 ZINC000217547332 EI In-Stock Unstable CCR3 17 45 O=C(/C=C\c1ccc([N+](=O)[O-])cc1)NC1CC(O)C1 ZINC000217547364 CD For-Sale Unstable HDAC8 0 49 O=C(/C=C\c1ccc([N+](=O)[O-])cc1)NC1CC(O)C1 ZINC000217547364 CD For-Sale Unstable HDAC1 23 52 CC(C)COc1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217547376 HH For-Sale Unstable NPY5R 26 41 CC(C)(C)c1ccc(NC(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc1 ZINC000217547377 HJ For-Sale Unstable EPHX2 25 49 CC(C)(C)c1ccc(NC(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc1 ZINC000217547377 HJ For-Sale Unstable DOT1L 57 35 Cc1cc(C)c(C[C@@H](N)C(=O)O)c(O)c1Cl ZINC000217547378 BD For-Sale Unstable OPRM1 19 47 Cc1cc(C)c(C[C@@H](N)C(=O)O)c(O)c1Cl ZINC000217547378 BD For-Sale Unstable GRIA3 58 41 Cc1cc(C)c(C[C@@H](N)C(=O)O)c(O)c1Cl ZINC000217547378 BD For-Sale Unstable GRIA1 40 41 Cc1cc(C)c(C[C@@H](N)C(=O)O)c(O)c1Cl ZINC000217547378 BD For-Sale Unstable GRIA2 48 41 Cc1cc(C)c(C[C@@H](N)C(=O)O)c(O)c1Cl ZINC000217547378 BD For-Sale Unstable GRIA4 48 41 Cc1cc(C)c(C[C@@H](N)C(=O)O)c(O)c1Cl ZINC000217547378 BD For-Sale Unstable GRIK1 39 41 C[C@@H]1CCCN(C(=O)NCCc2ccc(Br)cc2)C1 ZINC000217547401 EG On-Demand Unstable HRH3 33 43 C[C@@H]1CCCN(C(=O)NCCc2ccc(Br)cc2)C1 ZINC000217547401 EG On-Demand Unstable GPBAR1 32 48 COc1ccc(CNC(=O)NCC[C@H](O)c2ccsc2)cc1OC ZINC000217547426 FF In-Stock Unstable MT-ND1 24 40 CC(C)NS(=O)(=O)c1ccc(NC[C@@H]2CCCO2)c(C(=O)O)c1 ZINC000217547473 ED In-Stock Unstable LEF 42 36 C[C@H]1CCCN(C(=O)NCCc2ccc(Br)cc2)C1 ZINC000217547475 EG On-Demand Unstable HRH3 33 43 C[C@H]1CCCN(C(=O)NCCc2ccc(Br)cc2)C1 ZINC000217547475 EG On-Demand Unstable GPBAR1 32 48 CCCOc1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1C ZINC000217547490 HH For-Sale Unstable PDE5A 44 44 CCCOc1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1C ZINC000217547490 HH For-Sale Unstable NPY5R 26 41 COc1ccc(CNC(=O)NCC[C@@H](O)c2ccsc2)cc1OC ZINC000217547519 FF In-Stock Unstable MT-ND1 24 40 CC(C)NS(=O)(=O)c1ccc(NC[C@H]2CCCO2)c(C(=O)O)c1 ZINC000217547563 ED In-Stock Unstable LEF 42 36 Cc1n[nH]c(C)c1CN1CCN(CCN2CCCC2)C[C@@H](C(=O)O)C1 ZINC000217547575 EC In-Stock Unstable SLC6A1 130 38 Cc1cc(I)ccc1N[C@H]1C[C@H](C)CC[C@H]1C(C)C ZINC000217547583 FK For-Sale Unstable TRPM8 15 42 CCN(Cc1ccccc1)C(=O)NCCc1ccc(Br)cc1 ZINC000217547588 FI On-Demand Unstable OPRD1 20 41 CCN(Cc1ccccc1)C(=O)NCCc1ccc(Br)cc1 ZINC000217547588 FI On-Demand Unstable SDH1 0 41 CCN(Cc1ccccc1)C(=O)NCCc1ccc(Br)cc1 ZINC000217547588 FI On-Demand Unstable TSPO 23 42 CCN(Cc1ccccc1)C(=O)NCCc1ccc(Br)cc1 ZINC000217547588 FI On-Demand Unstable PLM2_PLAFA 35 41 CCN(Cc1ccccc1)C(=O)NCCc1ccc(Br)cc1 ZINC000217547588 FI On-Demand Unstable AMP1_PLAFQ 32 43 CCN(Cc1ccccc1)C(=O)NCCc1ccc(Br)cc1 ZINC000217547588 FI On-Demand Unstable PTGES 19 47 CCN(Cc1ccccc1)C(=O)NCCc1ccc(Br)cc1 ZINC000217547588 FI On-Demand Unstable LIMK2 40 36 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)NC12CC3CC(CC(C3)C1)C2 ZINC000217547590 HI For-Sale Unstable EPHX2 82 44 O=C1OC2(CCN(S(=O)(=O)c3ccccc3Br)CC2)c2ccccc21 ZINC000217547598 HG For-Sale Unstable NPY5R 33 47 CC(C)NS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217547663 EE In-Stock Unstable KCNQ2 49 37 CC(C)NS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217547663 EE In-Stock Unstable SLC6A9 21 47 OC[C@H](O)CN1CCC[C@@H]2CCCC[C@@H]21 ZINC000217547665 BC In-Stock Unstable SLC18A2 45 34 Cc1cc(I)ccc1N[C@H]1C[C@@H](C)CC[C@H]1C(C)C ZINC000217547677 FK For-Sale Unstable TRPM8 15 42 COc1ccc(NC(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc1OC ZINC000217547687 HH For-Sale Unstable QPCT 21 49 COc1ccc(NC(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc1OC ZINC000217547687 HH For-Sale Unstable ENPP1 70 33 Cc1cc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)c(Cl)cc1Cl ZINC000217547711 II For-Sale Unstable NPY5R 33 52 C[C@@H]1CCCCN1C(=O)NCCc1ccc(Br)cc1 ZINC000217547713 EH On-Demand Unstable FKBP1A 40 38 C[C@@H]1CCCCN1C(=O)NCCc1ccc(Br)cc1 ZINC000217547713 EH On-Demand Unstable HRH3 31 50 C[C@@H]1CCCCN1C(=O)NCCc1ccc(Br)cc1 ZINC000217547713 EH On-Demand Unstable DPP7 22 43 C[C@@H]1CCCCN1C(=O)NCCc1ccc(Br)cc1 ZINC000217547713 EH On-Demand Unstable GPBAR1 27 45 O[C@@H](CN1CCC[C@@H]2CCCC[C@@H]21)c1ccccc1 ZINC000217547738 CG On-Demand Unstable SLC6A3 18 49 O[C@@H](CN1CCC[C@@H]2CCCC[C@@H]21)c1ccccc1 ZINC000217547738 CG On-Demand Unstable SLC18A3 49 44 CN(C)[C@@H]1[C@H]2CC[C@@H]1CN(C(=O)c1nc3ccccc3[nH]1)C2 ZINC000217547790 CD In-Stock Unstable GRIN2B 27 44 C[C@H]1CCCCN1C(=O)NCCc1ccc(Br)cc1 ZINC000217547793 EH On-Demand Unstable FKBP1A 40 38 C[C@H]1CCCCN1C(=O)NCCc1ccc(Br)cc1 ZINC000217547793 EH On-Demand Unstable HRH3 31 50 C[C@H]1CCCCN1C(=O)NCCc1ccc(Br)cc1 ZINC000217547793 EH On-Demand Unstable DPP7 22 43 C[C@H]1CCCCN1C(=O)NCCc1ccc(Br)cc1 ZINC000217547793 EH On-Demand Unstable GPBAR1 27 45 Nc1nc(=O)c2ncn(COCCC(=O)O)c2[nH]1 ZINC000217547802 CB Annotated Unstable TK 25 47 Nc1nc(=O)c2ncn(COCCC(=O)O)c2[nH]1 ZINC000217547802 CB Annotated Unstable HPRT1 81 51 Nc1nc(=O)c2ncn(COCCC(=O)O)c2[nH]1 ZINC000217547802 CB Annotated Unstable PNP 31 44 O=C1OC2(CCN(S(=O)(=O)c3ccc(Br)s3)CC2)c2ccccc21 ZINC000217547813 IG For-Sale Unstable NPY5R 30 42 COc1ccc(C(=O)NCc2ccc([C@H](O)c3ccccc3)s2)cc1OC ZINC000217547826 GH In-Stock Unstable PPARA 15 41 COc1ccc(C(=O)NCc2ccc([C@H](O)c3ccccc3)s2)cc1OC ZINC000217547826 GH In-Stock Unstable CYSLTR1 40 32 COc1ccc(C(=O)NCc2ccc([C@H](O)c3ccccc3)s2)cc1OC ZINC000217547826 GH In-Stock Unstable PPARD 19 40 COc1ccc(C(=O)NCc2ccc([C@H](O)c3ccccc3)s2)cc1OC ZINC000217547826 GH In-Stock Unstable MT-ND1 24 40 O[C@H](CN1CCC[C@@H]2CCCC[C@@H]21)c1ccccc1 ZINC000217547838 CG On-Demand Unstable SLC18A3 23 44 COc1ccc(C(=O)NCc2ccc([C@@H](O)c3ccccc3)s2)cc1OC ZINC000217547900 GH In-Stock Unstable PPARA 15 41 COc1ccc(C(=O)NCc2ccc([C@@H](O)c3ccccc3)s2)cc1OC ZINC000217547900 GH In-Stock Unstable CYSLTR1 40 32 COc1ccc(C(=O)NCc2ccc([C@@H](O)c3ccccc3)s2)cc1OC ZINC000217547900 GH In-Stock Unstable PPARD 19 40 COc1ccc(C(=O)NCc2ccc([C@@H](O)c3ccccc3)s2)cc1OC ZINC000217547900 GH In-Stock Unstable MT-ND1 24 40 CC[C@@H]1CCCCN1C(=O)NCCc1ccc(Br)cc1 ZINC000217547911 EH On-Demand Unstable FKBP1A 45 37 CC[C@@H]1CCCCN1C(=O)NCCc1ccc(Br)cc1 ZINC000217547911 EH On-Demand Unstable GPBAR1 25 44 Cc1ccc(/C=C/S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217547936 GG For-Sale Unstable NPY5R 29 42 CCCCCNc1ccc(S(=O)(=O)NC(C)C)cc1C(=O)O ZINC000217547981 EF In-Stock Unstable CASP3 0 40 CCCCCNc1ccc(S(=O)(=O)NC(C)C)cc1C(=O)O ZINC000217547981 EF In-Stock Unstable LEF 44 37 CC[C@H]1CCCCN1C(=O)NCCc1ccc(Br)cc1 ZINC000217547993 EH On-Demand Unstable FKBP1A 45 37 CC[C@H]1CCCCN1C(=O)NCCc1ccc(Br)cc1 ZINC000217547993 EH On-Demand Unstable GPBAR1 25 44 COc1ccc(NC(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)c(OC)c1 ZINC000217548035 HH For-Sale Unstable DRD4 40 31 COC(=O)c1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217548062 HE For-Sale Unstable NPY5R 42 55 CC(C)CCNc1ccc(S(=O)(=O)NC(C)C)cc1C(=O)O ZINC000217548091 EF In-Stock Unstable LEF 52 34 O=C(NCCc1ccc(Br)cc1)N(Cc1ccccc1)Cc1ccccc1 ZINC000217548124 HK For-Sale Unstable CPA1 17 40 O=C(NCCc1ccc(Br)cc1)N(Cc1ccccc1)Cc1ccccc1 ZINC000217548124 HK For-Sale Unstable CA5B 16 42 O=C(NCCc1ccc(Br)cc1)N(Cc1ccccc1)Cc1ccccc1 ZINC000217548124 HK For-Sale Unstable AMP1_PLAFQ 36 43 O=C(NCCc1ccc(Br)cc1)N(Cc1ccccc1)Cc1ccccc1 ZINC000217548124 HK For-Sale Unstable PTGES 20 48 O=C(NCCc1ccc(Br)cc1)N(Cc1ccccc1)Cc1ccccc1 ZINC000217548124 HK For-Sale Unstable LIG1 0 42 O=C(NCCc1ccc(Br)cc1)N(Cc1ccccc1)Cc1ccccc1 ZINC000217548124 HK For-Sale Unstable LIMK2 40 37 Cn1cc(/C=C\C(=O)NC2CC(O)C2)cn1 ZINC000217548138 BC For-Sale Unstable HDAC8 47 34 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)NCc1cccc2ccccc12 ZINC000217548146 HI For-Sale Unstable FABP4 44 38 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)NCc1cccc2ccccc12 ZINC000217548146 HI For-Sale Unstable P2RX7 30 41 Cc1noc(C)c1S(=O)(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217548147 ED In-Stock Unstable CHRNA4 30 48 O=C1OC2(CCN(S(=O)(=O)Cc3cc(F)ccc3F)CC2)c2ccccc21 ZINC000217548169 GF In-Stock Unstable NPY5R 37 45 COC(=O)[C@@H](CC(C)C)NC(=O)CN1CCC[C@@H](CN)C1 ZINC000217548173 CC For-Sale Unstable NMT1 20 41 COC(=O)[C@@H](CC(C)C)NC(=O)CN1CCC[C@@H](CN)C1 ZINC000217548173 CC For-Sale Unstable CCR3 41 34 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NC(C)C)cc1C(=O)O ZINC000217548213 EF In-Stock Unstable LEF 48 35 COc1ccc(NC(=O)NCCc2ccc(Br)cc2)c(OC)c1 ZINC000217548237 GH On-Demand Unstable TRPV1 29 49 COc1ccc(NC(=O)NCCc2ccc(Br)cc2)c(OC)c1 ZINC000217548237 GH On-Demand Unstable RAF1 40 43 COc1ccc(NC(=O)NCCc2ccc(Br)cc2)c(OC)c1 ZINC000217548237 GH On-Demand Unstable MTNR1A 94 43 COc1ccc(NC(=O)NCCc2ccc(Br)cc2)c(OC)c1 ZINC000217548237 GH On-Demand Unstable MTNR1B 80 40 COc1ccc(NC(=O)NCCc2ccc(Br)cc2)c(OC)c1 ZINC000217548237 GH On-Demand Unstable ROCK2 15 43 COc1ccc(NC(=O)NCCc2ccc(Br)cc2)c(OC)c1 ZINC000217548237 GH On-Demand Unstable CA9 16 40 COc1ccc(NC(=O)NCCc2ccc(Br)cc2)c(OC)c1 ZINC000217548237 GH On-Demand Unstable Q8MMZ8_EIMTE 29 43 COc1ccc(NC(=O)NCCc2ccc(Br)cc2)c(OC)c1 ZINC000217548237 GH On-Demand Unstable AKR1C2 20 40 COc1ccc(NC(=O)NCCc2ccc(Br)cc2)c(OC)c1 ZINC000217548237 GH On-Demand Unstable ACAT 0 55 COc1ccc(Cl)cc1NC(=O)NCCn1nc(C(F)(F)F)c2c1CCCC2 ZINC000217548245 HI For-Sale Unstable RBP4 25 41 COC(=O)[C@H](CC(C)C)NC(=O)CN1CCC[C@@H](CN)C1 ZINC000217548268 CC For-Sale Unstable NMT1 20 41 COC(=O)[C@H](CC(C)C)NC(=O)CN1CCC[C@@H](CN)C1 ZINC000217548268 CC For-Sale Unstable CCR3 41 34 CCC[C@H](C)Nc1ccc(S(=O)(=O)NC(C)C)cc1C(=O)O ZINC000217548291 EF In-Stock Unstable LEF 48 35 O=C1OC2(CCN(S(=O)(=O)Cc3ccc(C(F)(F)F)cc3)CC2)c2ccccc21 ZINC000217548292 IH For-Sale Unstable NPY5R 28 50 Cc1cc(Cl)ccc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217548354 FJ For-Sale Unstable RAF1 37 41 Cc1cc(Cl)ccc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217548354 FJ For-Sale Unstable Q8MMZ8_EIMTE 24 41 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)Nc1ccccc1C(F)(F)F ZINC000217548360 HJ For-Sale Unstable FABP4 26 40 Cn1nc(-c2ccccc2NC(=O)c2c[nH]c3ccccc23)ccc1=O ZINC000217548371 EG In-Stock Unstable CFTR 35 42 CCCS(=O)(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217548391 DD For-Sale Unstable SLC6A9 50 39 CCCS(=O)(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217548391 DD For-Sale Unstable NPY5R 33 43 CNC(=O)c1cccc(S(=O)(=O)N2CCCn3nc([C@@H](C)O)cc3C2)c1 ZINC000217548469 GC In-Stock Unstable PPARD 0 41 CNC(=O)c1cccc(S(=O)(=O)N2CCCn3nc([C@@H](C)O)cc3C2)c1 ZINC000217548469 GC In-Stock Unstable AKR1C3 65 54 O=C(NCCOCCO)NCCc1ccc(Br)cc1 ZINC000217548477 ED For-Sale Unstable LIG1 0 40 C[C@H](C(=O)c1ccccc1)N1CCC[C@@H](CO)C1 ZINC000217548485 BD For-Sale Unstable ACE 29 41 C[C@H](C(=O)c1ccccc1)N1CCC[C@@H](CO)C1 ZINC000217548485 BD For-Sale Unstable SLC6A1 56 35 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)Nc1cccc(C(F)(F)F)c1 ZINC000217548487 HJ For-Sale Unstable CCR3 25 47 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)Nc1cccc(C(F)(F)F)c1 ZINC000217548487 HJ For-Sale Unstable RAF1 15 43 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)Nc1cccc(C(F)(F)F)c1 ZINC000217548487 HJ For-Sale Unstable KDR 17 40 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)Nc1cccc(C(F)(F)F)c1 ZINC000217548487 HJ For-Sale Unstable EPHX2 19 49 CCOc1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217548491 GF For-Sale Unstable NPY5R 30 41 CNC(=O)c1cccc(S(=O)(=O)N2CCCn3nc([C@H](C)O)cc3C2)c1 ZINC000217548550 GC In-Stock Unstable PPARD 0 41 CNC(=O)c1cccc(S(=O)(=O)N2CCCn3nc([C@H](C)O)cc3C2)c1 ZINC000217548550 GC In-Stock Unstable AKR1C3 65 54 C[C@@H](C(=O)c1ccccc1)N1CCC[C@@H](CO)C1 ZINC000217548557 BD For-Sale Unstable ACE 29 41 C[C@@H](C(=O)c1ccccc1)N1CCC[C@@H](CO)C1 ZINC000217548557 BD For-Sale Unstable SLC6A1 56 35 CCCCNS(=O)(=O)c1ccc(NCCC)c(C(=O)O)c1 ZINC000217548592 DE In-Stock Unstable CASP3 16 46 CCCCNS(=O)(=O)c1ccc(NCCC)c(C(=O)O)c1 ZINC000217548592 DE In-Stock Unstable BDKRB1 0 43 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)Nc1ccc(C(F)(F)F)cc1 ZINC000217548595 HJ For-Sale Unstable EPHX2 31 56 COC(=O)c1ccc(C(=O)OC)c(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217548599 IG For-Sale Unstable FAS 33 43 O=C1OC2(CCN(S(=O)(=O)c3ccc(F)cc3F)CC2)c2ccccc21 ZINC000217548605 GF For-Sale Unstable NPY5R 40 50 COc1cccc(F)c1C(=O)N(C)CC[C@@H]1CCCCO1 ZINC000217548687 CF In-Stock Unstable OXTR 25 42 COc1cccc(F)c1C(=O)N(C)CC[C@@H]1CCCCO1 ZINC000217548687 CF In-Stock Unstable AVPR1A 0 42 COc1cccc(F)c1C(=O)N(C)CC[C@@H]1CCCCO1 ZINC000217548687 CF In-Stock Unstable ACKR3 65 35 CCCCNS(=O)(=O)c1ccc(NC(C)C)c(C(=O)O)c1 ZINC000217548689 DE In-Stock Unstable CASP3 17 45 CCCCNS(=O)(=O)c1ccc(NC(C)C)c(C(=O)O)c1 ZINC000217548689 DE In-Stock Unstable BDKRB1 0 40 CCCCN(CCCC)C(=O)NCCc1ccc(Br)cc1 ZINC000217548699 FJ For-Sale Unstable THRA 0 41 CCCCN(CCCC)C(=O)NCCc1ccc(Br)cc1 ZINC000217548699 FJ For-Sale Unstable PLM2_PLAFA 40 40 CCCCN(CCCC)C(=O)NCCc1ccc(Br)cc1 ZINC000217548699 FJ For-Sale Unstable LIG1 0 42 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)Nc1ccc(Cl)c(Cl)c1 ZINC000217548702 HJ For-Sale Unstable RAF1 25 42 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)Nc1ccc(Cl)c(Cl)c1 ZINC000217548702 HJ For-Sale Unstable EPHX2 17 42 O=C(NCCn1nc(C(F)(F)F)c2c1CCCC2)Nc1ccc(Cl)c(Cl)c1 ZINC000217548702 HJ For-Sale Unstable Q8MMZ8_EIMTE 36 42 O=C1OC2(CCN(S(=O)(=O)Cc3ccccc3)CC2)c2ccccc21 ZINC000217548711 FF For-Sale Unstable SIGMAR1 27 66 O=C1OC2(CCN(S(=O)(=O)Cc3ccccc3)CC2)c2ccccc21 ZINC000217548711 FF For-Sale Unstable NPY5R 37 45 C[C@@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccc(F)cc1 ZINC000217548717 CD On-Demand Unstable CCR3 60 44 C[C@@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccc(F)cc1 ZINC000217548717 CD On-Demand Unstable BIRC2 48 41 O=C(/C=C\c1ccc2c(c1)CCO2)NC1CC(O)C1 ZINC000217548737 CD For-Sale Unstable GPR183 0 42 COc1cccc(F)c1C(=O)N(C)CC[C@H]1CCCCO1 ZINC000217548767 CF In-Stock Unstable OXTR 25 42 COc1cccc(F)c1C(=O)N(C)CC[C@H]1CCCCO1 ZINC000217548767 CF In-Stock Unstable AVPR1A 0 42 COc1cccc(F)c1C(=O)N(C)CC[C@H]1CCCCO1 ZINC000217548767 CF In-Stock Unstable ACKR3 65 35 CCCCNc1ccc(S(=O)(=O)NCCCC)cc1C(=O)O ZINC000217548792 EF In-Stock Unstable CASP3 22 47 C[C@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccc(F)cc1 ZINC000217548803 CD On-Demand Unstable CCR3 60 44 C[C@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccc(F)cc1 ZINC000217548803 CD On-Demand Unstable BIRC2 48 41 CC(=O)N1c2ccccc2[C@H](C=O)C[C@H]1C ZINC000217548807 BE In-Stock Unstable PTGDR2 57 46 CC(=O)N1c2ccccc2[C@H](C=O)C[C@H]1C ZINC000217548807 BE In-Stock Unstable BRD4 41 45 CC(=O)N1c2ccccc2[C@H](C=O)C[C@H]1C ZINC000217548807 BE In-Stock Unstable BRD2 62 45 CCN(CC)CCCNC(=O)NCCc1ccc(Br)cc1 ZINC000217548811 FG On-Demand Unstable PLM2_PLAFA 58 37 CCCCOc1ccc(NC(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc1 ZINC000217548813 HJ For-Sale Unstable HRH2 23 42 CCCCOc1ccc(NC(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc1 ZINC000217548813 HJ For-Sale Unstable EPHX2 29 41 O=C1OC2(CCN(S(=O)(=O)c3cc(F)cc(F)c3)CC2)c2ccccc21 ZINC000217548822 GF For-Sale Unstable NPY5R 37 47 CCOc1ccc2nc(NC(=O)Cn3nc(-n4ccc5ccccc54)ccc3=O)sc2c1 ZINC000217548883 IH In-Stock Unstable CSNK1D 45 49 CCOc1ccc2nc(NC(=O)Cn3nc(-n4ccc5ccccc54)ccc3=O)sc2c1 ZINC000217548883 IH In-Stock Unstable PORCN 0 41 CCOc1ccc2nc(NC(=O)Cn3nc(-n4ccc5ccccc54)ccc3=O)sc2c1 ZINC000217548883 IH In-Stock Unstable ISPD 0 43 CC(=O)N1c2ccccc2[C@H](C=O)C[C@@H]1C ZINC000217548896 BE In-Stock Unstable ECR 0 40 CC(=O)N1c2ccccc2[C@H](C=O)C[C@@H]1C ZINC000217548896 BE In-Stock Unstable PTGDR2 57 46 CC(=O)N1c2ccccc2[C@H](C=O)C[C@@H]1C ZINC000217548896 BE In-Stock Unstable BRD4 46 43 CC(=O)N1c2ccccc2[C@H](C=O)C[C@@H]1C ZINC000217548896 BE In-Stock Unstable BRD2 62 45 CCCCNS(=O)(=O)c1ccc(NCC(C)C)c(C(=O)O)c1 ZINC000217548900 EF In-Stock Unstable CASP3 16 46 CCCCNS(=O)(=O)c1ccc(NCC(C)C)c(C(=O)O)c1 ZINC000217548900 EF In-Stock Unstable MTNN 41 32 Cc1c(Cl)c(=O)oc2cc(OC(=O)[C@@H]3CC[C@@H](CNC(=O)OCc4ccccc4)CC3)ccc12 ZINC000217548912 JK In-Stock Unstable MAOB 54 45 Cc1c(Cl)c(=O)oc2cc(OC(=O)[C@@H]3CC[C@@H](CNC(=O)OCc4ccccc4)CC3)ccc12 ZINC000217548912 JK In-Stock Unstable MAP2K1 0 43 COc1ccc(CNC(=O)NCCn2nc(C(F)(F)F)c3c2CCCC3)cc1OC ZINC000217548925 IG For-Sale Unstable MT-ND1 23 40 OCC[C@@H]1CCCCN1C[C@@H](O)CO ZINC000217548934 BB On-Demand Unstable SLC18A2 64 47 CN(C)CCCNC(=O)NCCc1ccc(Br)cc1 ZINC000217548939 EE On-Demand Unstable LIG1 0 40 O=C1OC2(CCN(S(=O)(=O)c3cnc[nH]3)CC2)c2ccccc21 ZINC000217548940 ED For-Sale Unstable NPY5R 42 44 O=C(CCn1ccc(=O)[nH]c1=O)NCCN1CCNC1=O ZINC000217548941 CA In-Stock Unstable DUT 48 37 O=C(CCn1ccc(=O)[nH]c1=O)NCCN1CCNC1=O ZINC000217548941 CA In-Stock Unstable Q8II92_PLAF7 53 40 CC(=O)N1c2ccccc2[C@@H](C=O)C[C@H]1C ZINC000217548968 BE In-Stock Unstable ECR 0 40 CC(=O)N1c2ccccc2[C@@H](C=O)C[C@H]1C ZINC000217548968 BE In-Stock Unstable PTGDR2 0 46 CC(=O)N1c2ccccc2[C@@H](C=O)C[C@H]1C ZINC000217548968 BE In-Stock Unstable BRD4 41 45 CC(=O)N1c2ccccc2[C@@H](C=O)C[C@H]1C ZINC000217548968 BE In-Stock Unstable BRD2 62 45 OCC[C@H]1CCCCN1C[C@@H](O)CO ZINC000217549006 BB On-Demand Unstable SLC18A2 64 47 CCCCNS(=O)(=O)c1ccc(N[C@@H](C)CC)c(C(=O)O)c1 ZINC000217549011 EF In-Stock Unstable CASP3 16 44 CC(=O)N1c2ccccc2[C@@H](C=O)C[C@@H]1C ZINC000217549048 BE In-Stock Unstable ECR 0 40 CC(=O)N1c2ccccc2[C@@H](C=O)C[C@@H]1C ZINC000217549048 BE In-Stock Unstable PTGDR2 57 46 CC(=O)N1c2ccccc2[C@@H](C=O)C[C@@H]1C ZINC000217549048 BE In-Stock Unstable BRD4 46 43 CC(=O)N1c2ccccc2[C@@H](C=O)C[C@@H]1C ZINC000217549048 BE In-Stock Unstable BRD2 62 45 C[C@@H]1CCC[C@@H](C)N1C(=O)NCCc1ccc(Br)cc1 ZINC000217549060 EH For-Sale Unstable HRH3 0 43 C[C@@H]1CCC[C@@H](C)N1C(=O)NCCc1ccc(Br)cc1 ZINC000217549060 EH For-Sale Unstable GPBAR1 0 43 O=C1OC2(CCN(S(=O)(=O)c3cccc(F)c3)CC2)c2ccccc21 ZINC000217549061 FF For-Sale Unstable NPY5R 36 50 O=C1OC2(CCN(S(=O)(=O)c3cccc(F)c3)CC2)c2ccccc21 ZINC000217549061 FF For-Sale Unstable PKM 46 51 CCCCNS(=O)(=O)c1ccc(N[C@H](C)CC)c(C(=O)O)c1 ZINC000217549092 EF In-Stock Unstable CASP3 16 44 CCCCCCCCCCCC(=O)NCCC(C)(C)N ZINC000217549099 CI For-Sale Unstable CNR1 16 61 CCCCCCCCCCCC(=O)NCCC(C)(C)N ZINC000217549099 CI For-Sale Unstable LPAR1 15 47 CCCCCCCCCCCC(=O)NCCC(C)(C)N ZINC000217549099 CI For-Sale Unstable EPHX2 15 50 CCCCCCCCCCCC(=O)NCCC(C)(C)N ZINC000217549099 CI For-Sale Unstable LPAR3 26 40 CCCCCCCCCCCC(=O)NCCC(C)(C)N ZINC000217549099 CI For-Sale Unstable LASR 40 37 CCCCCCCCCCCC(=O)NCCC(C)(C)N ZINC000217549099 CI For-Sale Unstable NOD1 69 44 CCCCCCCCCCCC(=O)NCCC(C)(C)N ZINC000217549099 CI For-Sale Unstable CQSS 58 37 OCC[C@@H]1CCCCN1C[C@@H](O)COCc1ccccc1 ZINC000217549127 CD On-Demand Unstable SLC18A2 96 48 C[C@H]1CCC[C@@H](C)N1C(=O)NCCc1ccc(Br)cc1 ZINC000217549157 EH For-Sale Unstable HRH3 0 43 C[C@H]1CCC[C@@H](C)N1C(=O)NCCc1ccc(Br)cc1 ZINC000217549157 EH For-Sale Unstable GPBAR1 0 43 O=C1OC2(CCN(S(=O)(=O)c3ccc4ccccc4c3)CC2)c2ccccc21 ZINC000217549173 GH For-Sale Unstable NPY5R 32 46 O=C1OC2(CCN(S(=O)(=O)c3ccc4ccccc4c3)CC2)c2ccccc21 ZINC000217549173 GH For-Sale Unstable PKM 40 48 CCCCNS(=O)(=O)c1ccc(NC(C)(C)C)c(C(=O)O)c1 ZINC000217549182 EF In-Stock Unstable CASP3 16 45 C[C@@H]1C[C@@H](C=O)c2ccccc2N1C(=O)C1CC1 ZINC000217549183 BF In-Stock Unstable PTGDR2 0 41 CCO[C@@H]1C[C@@H](NC(=S)Nc2ccccc2)C1(C)C ZINC000217549187 CG For-Sale Unstable TIMP3 41 32 C[C@@H](Cc1ccccc1)NC[C@@H](C)N(C)C1CC1 ZINC000217549218 BF For-Sale Unstable GALR1 47 38 C[C@H](C(=O)O)c1ccc(S(C)(=O)=O)cc1F ZINC000217549221 BD For-Sale Unstable PTGS1 18 41 C[C@H](C(=O)O)c1ccc(S(C)(=O)=O)cc1F ZINC000217549221 BD For-Sale Unstable PTGS2 33 45 C[C@H](C(=O)O)c1ccc(S(C)(=O)=O)cc1F ZINC000217549221 BD For-Sale Unstable O49150_SOLTU 43 38 C[C@H]1CCC[C@H](C)N1C(=O)NCCc1ccc(Br)cc1 ZINC000217549229 EH For-Sale Unstable HRH3 0 43 C[C@H]1CCC[C@H](C)N1C(=O)NCCc1ccc(Br)cc1 ZINC000217549229 EH For-Sale Unstable GPBAR1 0 43 CCO[C@H]1C[C@@H](NC(=S)Nc2ccccc2)C1(C)C ZINC000217549251 CG For-Sale Unstable TIMP3 41 32 C[C@H]1C[C@@H](C=O)c2ccccc2N1C(=O)C1CC1 ZINC000217549258 BF In-Stock Unstable PTGDR2 53 41 COc1ccc(C(=O)Nc2ccc(N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)nc2)cc1 ZINC000217549260 HG In-Stock Unstable CHRNA4 26 43 COc1ccc(C(=O)Nc2ccc(N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)nc2)cc1 ZINC000217549260 HG In-Stock Unstable DGAT1 41 40 Cc1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217549276 FF For-Sale Unstable NPY5R 32 45 O=C(CCn1ccc(=O)[nH]c1=O)N1CCCC[C@@H]1c1nc2ccccc2[nH]1 ZINC000217549277 FD In-Stock Unstable PRCP 59 49 O=C(CCn1ccc(=O)[nH]c1=O)N1CCCC[C@@H]1c1nc2ccccc2[nH]1 ZINC000217549277 FD In-Stock Unstable COLA 109 40 O=C(CCn1ccc(=O)[nH]c1=O)N1CCCC[C@@H]1c1nc2ccccc2[nH]1 ZINC000217549277 FD In-Stock Unstable CPT1A 93 40 O=C(CCn1ccc(=O)[nH]c1=O)N1CCCC[C@@H]1c1nc2ccccc2[nH]1 ZINC000217549277 FD In-Stock Unstable DUT 82 50 O=C(CCn1ccc(=O)[nH]c1=O)N1CCCC[C@@H]1c1nc2ccccc2[nH]1 ZINC000217549277 FD In-Stock Unstable Q8II92_PLAF7 42 34 C=CCNc1ccc(S(=O)(=O)NCCCC)cc1C(=O)O ZINC000217549284 DE In-Stock Unstable CASP3 0 45 C=CCNc1ccc(S(=O)(=O)NCCCC)cc1C(=O)O ZINC000217549284 DE In-Stock Unstable BDKRB1 0 42 CS[C@@H]1CCN(C(=O)c2c(F)cccc2F)C1 ZINC000217549289 CF In-Stock Unstable L3MBTL3 41 38 C[C@H](Cc1ccccc1)NC[C@@H](C)N(C)C1CC1 ZINC000217549304 BF For-Sale Unstable GALR1 47 38 CCO[C@@H]1C[C@H](NC(=S)Nc2ccccc2)C1(C)C ZINC000217549315 CG For-Sale Unstable TIMP3 41 32 CC[S@](=O)CCN1C(=O)[C@H](C2CC2)NC(=O)[C@@H]1C ZINC000217549317 CB For-Sale Unstable GHRL 40 32 C[C@@H]1C[C@H](C=O)c2ccccc2N1C(=O)C1CC1 ZINC000217549321 BF In-Stock Unstable PTGDR2 53 41 C[C@@H](C(=O)O)c1ccc(S(C)(=O)=O)cc1F ZINC000217549332 BD For-Sale Unstable PTGS1 18 41 C[C@@H](C(=O)O)c1ccc(S(C)(=O)=O)cc1F ZINC000217549332 BD For-Sale Unstable PTGS2 33 45 C[C@@H](C(=O)O)c1ccc(S(C)(=O)=O)cc1F ZINC000217549332 BD For-Sale Unstable O49150_SOLTU 43 38 C[C@@H]1CCCC[C@@H]1NC(=O)NCCc1ccc(Br)cc1 ZINC000217549353 EH On-Demand Unstable TRAR 18 40 O=C1OC2(CCN(S(=O)(=O)c3ccc(Cl)cc3)CC2)c2ccccc21 ZINC000217549358 GG For-Sale Unstable NPY5R 33 49 O=C1OC2(CCN(S(=O)(=O)c3ccc(Cl)cc3)CC2)c2ccccc21 ZINC000217549358 GG For-Sale Unstable PKM 33 45 O=C(CCc1ccccc1)Nc1ccc(N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)nc1 ZINC000217549379 HG In-Stock Unstable CHRNA4 30 48 O=C(CCn1ccc(=O)[nH]c1=O)N1CCCC[C@H]1c1nc2ccccc2[nH]1 ZINC000217549382 FD In-Stock Unstable PRCP 59 49 O=C(CCn1ccc(=O)[nH]c1=O)N1CCCC[C@H]1c1nc2ccccc2[nH]1 ZINC000217549382 FD In-Stock Unstable COLA 109 40 O=C(CCn1ccc(=O)[nH]c1=O)N1CCCC[C@H]1c1nc2ccccc2[nH]1 ZINC000217549382 FD In-Stock Unstable CPT1A 93 40 O=C(CCn1ccc(=O)[nH]c1=O)N1CCCC[C@H]1c1nc2ccccc2[nH]1 ZINC000217549382 FD In-Stock Unstable DUT 82 50 O=C(CCn1ccc(=O)[nH]c1=O)N1CCCC[C@H]1c1nc2ccccc2[nH]1 ZINC000217549382 FD In-Stock Unstable Q8II92_PLAF7 42 34 CS[C@H]1CCN(C(=O)c2c(F)cccc2F)C1 ZINC000217549387 CF In-Stock Unstable L3MBTL3 41 38 C[C@@H](Cc1ccccc1)NC[C@H](C)N(C)C1CC1 ZINC000217549389 BF For-Sale Unstable GALR1 47 38 CCCCNS(=O)(=O)c1ccc(NC2CC2)c(C(=O)O)c1 ZINC000217549399 DE In-Stock Unstable CASP3 15 41 C[C@H]1C[C@H](C=O)c2ccccc2N1C(=O)C1CC1 ZINC000217549401 BF In-Stock Unstable PTGDR2 0 41 CCO[C@H]1C[C@H](NC(=S)Nc2ccccc2)C1(C)C ZINC000217549422 CG For-Sale Unstable TIMP3 41 32 C[C@H]1CCCC[C@@H]1NC(=O)NCCc1ccc(Br)cc1 ZINC000217549440 EH On-Demand Unstable TRAR 18 40 COc1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217549455 FF For-Sale Unstable NPY5R 32 45 COc1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217549455 FF For-Sale Unstable PKM 29 55 CS(=O)(=O)c1ccc(CCC(=O)O)c(F)c1 ZINC000217549460 BD For-Sale Unstable PTGS2 28 41 CS(=O)(=O)c1ccc(CCC(=O)O)c(F)c1 ZINC000217549460 BD For-Sale Unstable TBXA2R 52 42 CS(=O)(=O)c1ccc(CCC(=O)O)c(F)c1 ZINC000217549460 BD For-Sale Unstable FFAR1 38 42 CS(=O)(=O)c1ccc(CCC(=O)O)c(F)c1 ZINC000217549460 BD For-Sale Unstable FFAR4 58 46 C[C@@H](CN[C@H](C)Cc1ccccc1)N(C)C1CC1 ZINC000217549474 BF For-Sale Unstable GALR1 47 38 COc1ccc(C(=O)Nc2ccc(N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)nc2)cc1OC ZINC000217549479 IG In-Stock Unstable CHRNA4 26 43 COc1ccc(C(=O)Nc2ccc(N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)nc2)cc1OC ZINC000217549479 IG In-Stock Unstable DGAT1 31 40 Fc1cc(Cn2cnc3nc(I)nc(Cl)c32)ccc1Cl ZINC000217549500 HH For-Sale Unstable DNAE 69 32 CCCCNS(=O)(=O)c1ccc(NC2CCCC2)c(C(=O)O)c1 ZINC000217549513 EF In-Stock Unstable CASP3 15 40 C[C@@H]1CCCC[C@H]1NC(=O)NCCc1ccc(Br)cc1 ZINC000217549516 EH On-Demand Unstable TRAR 18 40 CC(C)C(=O)N1c2ccccc2[C@H](C=O)C[C@@H]1C ZINC000217549521 BF In-Stock Unstable PTGDR2 0 41 C[C@@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccccc1Cl ZINC000217549552 DE On-Demand Unstable SLC6A1 52 34 C[C@@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccccc1Cl ZINC000217549552 DE On-Demand Unstable PRCP 30 40 C[C@@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccccc1Cl ZINC000217549552 DE On-Demand Unstable BIRC2 44 35 CN(C)c1ccc(C(=O)Nc2ccc(N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)nc2)cc1 ZINC000217549565 IG In-Stock Unstable CHRNA4 26 43 CCCO[C@@H]1CCCN(C(=O)CCn2ccc(=O)[nH]c2=O)C1 ZINC000217549568 DC In-Stock Unstable DUT 74 44 O=C1OC2(CCN(S(=O)(=O)Cc3ccc(Cl)cc3)CC2)c2ccccc21 ZINC000217549569 GG For-Sale Unstable SIGMAR1 18 56 O=C1OC2(CCN(S(=O)(=O)Cc3ccc(Cl)cc3)CC2)c2ccccc21 ZINC000217549569 GG For-Sale Unstable NPY5R 30 48 CS(=O)(=O)c1ccc(CCC(=O)O)cc1F ZINC000217549576 BD For-Sale Unstable TBXA2R 53 42 CS(=O)(=O)c1ccc(CCC(=O)O)cc1F ZINC000217549576 BD For-Sale Unstable TBXAS1 17 40 CS(=O)(=O)c1ccc(CCC(=O)O)cc1F ZINC000217549576 BD For-Sale Unstable TRPV1 15 40 CS(=O)(=O)c1ccc(CCC(=O)O)cc1F ZINC000217549576 BD For-Sale Unstable FFAR1 83 50 CS(=O)(=O)c1ccc(CCC(=O)O)cc1F ZINC000217549576 BD For-Sale Unstable FFAR4 65 37 C[C@H]1CCCC[C@H]1NC(=O)NCCc1ccc(Br)cc1 ZINC000217549595 EH On-Demand Unstable TRAR 18 40 C[C@H]1CCCCN1[C@H](C)C(=O)c1ccccc1 ZINC000217549597 BG For-Sale Unstable SLC6A3 15 46 C[C@H]1CCCCN1[C@H](C)C(=O)c1ccccc1 ZINC000217549597 BG For-Sale Unstable VACHT_TETCF 0 40 CC(C)C(=O)N1c2ccccc2[C@H](C=O)C[C@H]1C ZINC000217549606 BF In-Stock Unstable PTGDR2 0 41 CCCCNS(=O)(=O)c1ccc(NC2CCCCC2)c(C(=O)O)c1 ZINC000217549626 FG In-Stock Unstable CASP3 0 46 CCCO[C@H]1CCCN(C(=O)CCn2ccc(=O)[nH]c2=O)C1 ZINC000217549648 DC In-Stock Unstable DUT 74 44 C[C@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccccc1Cl ZINC000217549650 DE On-Demand Unstable SLC6A1 52 34 C[C@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccccc1Cl ZINC000217549650 DE On-Demand Unstable PRCP 30 40 C[C@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccccc1Cl ZINC000217549650 DE On-Demand Unstable BIRC2 44 35 O=C(Nc1ccc(N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)nc1)c1cc(=O)c2ccccc2o1 ZINC000217549668 JG In-Stock Unstable CHRNA4 23 41 O=C(Nc1ccc(N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)nc1)c1cc(=O)c2ccccc2o1 ZINC000217549668 JG In-Stock Unstable DGAT1 41 45 O=C1OC2(CCN(S(=O)(=O)Cc3cc(F)cc(F)c3)CC2)c2ccccc21 ZINC000217549672 GF For-Sale Unstable SIGMAR1 15 61 O=C1OC2(CCN(S(=O)(=O)Cc3cc(F)cc(F)c3)CC2)c2ccccc21 ZINC000217549672 GF For-Sale Unstable NPY5R 36 45 O=C(O)CCc1ccccc1SCC(F)F ZINC000217549686 BG For-Sale Unstable FFAR1 49 42 O=C(O)CCc1ccccc1SCC(F)F ZINC000217549686 BG For-Sale Unstable FFAR4 48 37 CC(C)C(=O)N1c2ccccc2[C@@H](C=O)C[C@@H]1C ZINC000217549691 BF In-Stock Unstable PTGDR2 52 41 O=C(c1cc(=O)c2ccccc2o1)N1CC[C@H](S(=O)(=O)c2ccc(Cl)cc2)C1 ZINC000217549696 HG In-Stock Unstable TNKS 29 40 C[C@H]1CCCCN1[C@H](C)C(=O)c1cccc(Cl)c1 ZINC000217549715 CH For-Sale Unstable GRM5 22 40 C[C@H]1CCCCN1[C@H](C)C(=O)c1cccc(Cl)c1 ZINC000217549715 CH For-Sale Unstable CCKBR 0 41 Cc1nn(C)c(C)c1S(=O)(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217549770 GD For-Sale Unstable NPY5R 31 43 O=C(c1cc(=O)c2ccccc2o1)N1CC[C@@H](S(=O)(=O)c2ccc(Cl)cc2)C1 ZINC000217549774 HG In-Stock Unstable TNKS 29 40 CC(C)C(=O)N1c2ccccc2[C@@H](C=O)C[C@H]1C ZINC000217549775 BF In-Stock Unstable PTGDR2 0 41 COc1ccc(/C=C/C(=O)Nc2ccc(N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)nc2)cc1OC ZINC000217549791 JH In-Stock Unstable CHRNA4 23 40 COc1ccc(/C=C/C(=O)Nc2ccc(N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)nc2)cc1OC ZINC000217549791 JH In-Stock Unstable IMPDH2 0 47 O=C(O)CCc1ccc(SCC(F)F)cc1 ZINC000217549798 BG For-Sale Unstable FFAR1 82 49 O=C(O)CCc1ccc(SCC(F)F)cc1 ZINC000217549798 BG For-Sale Unstable FFAR4 49 37 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217549823 HK For-Sale Unstable CA2 16 60 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217549823 HK For-Sale Unstable EPHX1 0 43 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217549823 HK For-Sale Unstable ADRB1 24 44 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217549823 HK For-Sale Unstable ADRB3 32 41 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217549823 HK For-Sale Unstable CA1 24 53 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217549823 HK For-Sale Unstable CA12 19 60 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217549823 HK For-Sale Unstable CA9 20 57 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217549823 HK For-Sale Unstable IDO1 24 40 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217549823 HK For-Sale Unstable NCE103 26 57 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217549823 HK For-Sale Unstable P96878_MYCTU 18 40 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217549823 HK For-Sale Unstable P95276_MYCTO 0 43 C[C@H]1CCCCN1[C@H](C)C(=O)c1ccc(Cl)cc1 ZINC000217549835 CH For-Sale Unstable SLC6A1 36 46 C[C@H]1CCCCN1[C@H](C)C(=O)c1ccc(Cl)cc1 ZINC000217549835 CH For-Sale Unstable SLC6A3 15 46 C[C@H]1CCCCN1[C@H](C)C(=O)c1ccc(Cl)cc1 ZINC000217549835 CH For-Sale Unstable CCR1 34 40 C[C@H]1CCCCN1[C@H](C)C(=O)c1ccc(Cl)cc1 ZINC000217549835 CH For-Sale Unstable DPP7 20 41 CCCCNS(=O)(=O)c1ccc(NCCO)c(C(=O)O)c1 ZINC000217549836 DC In-Stock Unstable CASP3 16 45 CCCCNS(=O)(=O)c1ccc(NCCO)c(C(=O)O)c1 ZINC000217549836 DC In-Stock Unstable BDKRB1 0 42 CC[C@H](C)[C@@H]1NC(=O)[C@@H](CC)N(CC[S@@](=O)CC)C1=O ZINC000217549842 DC For-Sale Unstable GALR1 40 37 O=C1OC2(CCN(S(=O)(=O)CCOc3ccccc3)CC2)c2ccccc21 ZINC000217549867 GF For-Sale Unstable NPY5R 39 43 CCC(=O)N1c2ccccc2[C@H](C=O)C[C@@H]1C ZINC000217549888 BF In-Stock Unstable PTGDR2 0 45 CC(=O)Nc1ccc(N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)nc1 ZINC000217549917 DD In-Stock Unstable CHRNA4 30 52 O=C(NCCc1ccc(Br)cc1)N1CCc2ccccc2C1 ZINC000217549926 FH On-Demand Unstable AMP1_PLAFQ 16 45 O=C(NCCc1ccc(Br)cc1)N1CCc2ccccc2C1 ZINC000217549926 FH On-Demand Unstable DPP8 15 42 O=C(NCCc1ccc(Br)cc1)N1CCc2ccccc2C1 ZINC000217549926 FH On-Demand Unstable NOD2 41 34 O=C(NCCc1ccc(Br)cc1)N1CCc2ccccc2C1 ZINC000217549926 FH On-Demand Unstable NAMPT 17 43 C[C@@H](Cc1ccc(O)cc1)NC[C@@H](C)N(C)C1CC1 ZINC000217549934 CE On-Demand Unstable OPRM1 15 40 CCCCNS(=O)(=O)c1ccc(NCCCO)c(C(=O)O)c1 ZINC000217549939 ED In-Stock Unstable CASP3 16 46 CCC(=O)N1c2ccccc2[C@H](C=O)C[C@H]1C ZINC000217549977 BF In-Stock Unstable PTGDR2 0 45 O=C1OC2(CCN(S(=O)(=O)c3ccc4oc(=O)[nH]c4c3)CC2)c2ccccc21 ZINC000217549988 HD For-Sale Unstable NPY5R 31 45 C[C@H](Cc1ccc(O)cc1)NC[C@@H](C)N(C)C1CC1 ZINC000217550003 CE On-Demand Unstable OPRM1 15 40 CC(C)CC(=O)Nc1ccc(N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)nc1 ZINC000217550009 FF In-Stock Unstable CHRNA4 28 46 Cc1cccc(NC(=O)NCCc2ccc(Br)cc2)n1 ZINC000217550024 EH On-Demand Unstable GRM5 19 47 Cc1cccc(NC(=O)NCCc2ccc(Br)cc2)n1 ZINC000217550024 EH On-Demand Unstable SORT1 22 48 C[C@@H]1Cc2ccccc2N1C(=O)CN1CCC[C@@H](CN)C1 ZINC000217550037 CD On-Demand Unstable DRD4 40 57 C[C@@H]1Cc2ccccc2N1C(=O)CN1CCC[C@@H](CN)C1 ZINC000217550037 CD On-Demand Unstable TPP2 58 35 CCC(=O)N1c2ccccc2[C@@H](C=O)C[C@@H]1C ZINC000217550042 BF In-Stock Unstable PTGDR2 55 45 CCCCNS(=O)(=O)c1ccc(NCCOC)c(C(=O)O)c1 ZINC000217550055 ED In-Stock Unstable CASP3 22 43 Cc1nnn([C@@]23C[C@H]4C[C@@H](C2)C[C@](C(=O)NCc2ccc5c(c2)OCO5)(C4)C3)n1 ZINC000217550062 GE In-Stock Unstable NOS2 97 38 COc1ccccc1Oc1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217550091 JI For-Sale Unstable NPY5R 26 46 Cc1ccccc1S(=O)(=O)Nc1cc(F)cc(Cl)c1 ZINC000217550094 CH On-Demand Unstable NR1I2 25 42 C[C@@H](Cc1ccc(O)cc1)NC[C@H](C)N(C)C1CC1 ZINC000217550104 CE On-Demand Unstable OPRM1 15 40 C=C(C)C(=O)Nc1ccc(N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)nc1 ZINC000217550111 FE In-Stock Unstable CHRNA4 28 48 CCC(=O)N1c2ccccc2[C@@H](C=O)C[C@H]1C ZINC000217550122 BF In-Stock Unstable PTGDR2 0 45 C[C@H]1Cc2ccccc2N1C(=O)CN1CCC[C@@H](CN)C1 ZINC000217550123 CD On-Demand Unstable DRD4 40 57 C[C@H]1Cc2ccccc2N1C(=O)CN1CCC[C@@H](CN)C1 ZINC000217550123 CD On-Demand Unstable TPP2 58 35 CCCCNS(=O)(=O)c1ccc(NCCCOC)c(C(=O)O)c1 ZINC000217550173 ED In-Stock Unstable CASP3 22 42 C[C@@H](CN[C@H](C)Cc1ccc(O)cc1)N(C)C1CC1 ZINC000217550186 CE On-Demand Unstable OPRM1 15 40 O=C1OC2(CCN(S(=O)(=O)c3ccc(Oc4ccccc4Cl)cc3)CC2)c2ccccc21 ZINC000217550212 JJ For-Sale Unstable NPY5R 27 42 C[C@@H](O)c1cc2n(n1)CCN(Cc1cc(Cl)ccc1OCC(N)=O)C2 ZINC000217550227 FD In-Stock Unstable PTGER1 40 37 COc1ccc(C(=O)[C@@H](C)N2CCCC[C@@H]2C)cc1 ZINC000217550228 CG For-Sale Unstable CHRM2 31 43 COc1ccc(C(=O)[C@@H](C)N2CCCC[C@@H]2C)cc1 ZINC000217550228 CG For-Sale Unstable CHRM4 17 40 C[C@H](c1ccccc1)N(C)C(=O)CN1CCC[C@@H](CN)C1 ZINC000217550253 CD On-Demand Unstable SLC6A1 63 38 C[C@H](c1ccccc1)N(C)C(=O)CN1CCC[C@@H](CN)C1 ZINC000217550253 CD On-Demand Unstable OPRK1 29 44 C[C@H](c1ccccc1)N(C)C(=O)CN1CCC[C@@H](CN)C1 ZINC000217550253 CD On-Demand Unstable CCR5 45 40 CCCCNS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217550289 FG In-Stock Unstable GNRHR 15 40 CCCCNS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217550289 FG In-Stock Unstable CASP3 18 43 CCCCNS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217550289 FG In-Stock Unstable ALOX15 45 37 CC(C)Oc1ccc(C(=O)Nc2ccc(N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)nc2)cc1 ZINC000217550305 IH In-Stock Unstable CHRNA4 26 42 CC(C)Oc1ccc(C(=O)Nc2ccc(N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)nc2)cc1 ZINC000217550305 IH In-Stock Unstable PRNP 20 41 CC(C)Oc1ccc(C(=O)Nc2ccc(N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)nc2)cc1 ZINC000217550305 IH In-Stock Unstable DGAT1 29 40 C[C@H](O)c1cc2n(n1)CCN(Cc1cc(Cl)ccc1OCC(N)=O)C2 ZINC000217550315 FD In-Stock Unstable PTGER1 40 37 Cc1ccccc1Oc1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217550318 IJ For-Sale Unstable NPY5R 26 41 C[C@@H](c1ccccc1)N(C)C(=O)CN1CCC[C@@H](CN)C1 ZINC000217550331 CD On-Demand Unstable SLC6A1 63 38 C[C@@H](c1ccccc1)N(C)C(=O)CN1CCC[C@@H](CN)C1 ZINC000217550331 CD On-Demand Unstable OPRK1 29 44 C[C@@H](c1ccccc1)N(C)C(=O)CN1CCC[C@@H](CN)C1 ZINC000217550331 CD On-Demand Unstable CCR5 45 40 CC(C)N1C[C@@H](C(=O)Nc2ccc(N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)nc2)CC1=O ZINC000217550396 IE In-Stock Unstable CHRNA4 25 41 O=C1O[C@H](CCl)CN1c1ccc(Br)cc1 ZINC000217550399 CG For-Sale Unstable GRM2 15 46 CCCCNS(=O)(=O)c1ccc(N[C@@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217550411 GH In-Stock Unstable CASP3 19 43 O=C1OC2(CCN(S(=O)(=O)c3c(Cl)cccc3Cl)CC2)c2ccccc21 ZINC000217550429 HH For-Sale Unstable NPY5R 38 48 CC(C)N1C[C@H](C(=O)Nc2ccc(N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)nc2)CC1=O ZINC000217550472 IE In-Stock Unstable CHRNA4 25 41 CCCCNS(=O)(=O)c1ccc(N[C@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217550497 GH In-Stock Unstable CASP3 19 43 CCOc1ccccc1[C@@H](CN1CCCO[C@@H](C)C1)NC ZINC000217550545 CE For-Sale Unstable HCN1 40 31 CCOc1ccccc1[C@@H](CN1CCCO[C@@H](C)C1)NC ZINC000217550545 CE For-Sale Unstable HCN4 40 31 Cc1ccc(-c2ccc(S(=O)(=O)N3CCC4(CC3)OC(=O)c3ccccc34)cc2)cc1 ZINC000217550565 IJ For-Sale Unstable NPY5R 33 44 CCCCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217550587 GG In-Stock Unstable CA2 18 41 CCCCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217550587 GG In-Stock Unstable TBXA2R 50 40 CCCCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217550587 GG In-Stock Unstable CASP3 17 42 CCCCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217550587 GG In-Stock Unstable CA1 15 40 CCCCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217550587 GG In-Stock Unstable ALOX15 55 40 CCOc1ccccc1[C@H](CN1CCCO[C@@H](C)C1)NC ZINC000217550633 CE For-Sale Unstable HCN1 40 31 CCOc1ccccc1[C@H](CN1CCCO[C@@H](C)C1)NC ZINC000217550633 CE For-Sale Unstable HCN4 40 31 C[C@]1(c2ccccc2)OC[C@@H](CN2CCC[C@@H](CN)C2)O1 ZINC000217550666 CD For-Sale Unstable ADRA1D 16 41 C[C@]1(c2ccccc2)OC[C@@H](CN2CCC[C@@H](CN)C2)O1 ZINC000217550666 CD For-Sale Unstable ADRA1B 15 41 O=C1OC2(CCN(S(=O)(=O)c3ccc(-c4ccc(F)cc4)cc3)CC2)c2ccccc21 ZINC000217550682 II For-Sale Unstable NPY5R 40 54 O=C1OC2(CCN(S(=O)(=O)c3ccc(-c4ccc(F)cc4)cc3)CC2)c2ccccc21 ZINC000217550682 II For-Sale Unstable PKM 33 43 Cc1nc(C)c(CC(=O)NCc2cnn(-c3ccccc3C)c2)c(=O)[nH]1 ZINC000217550698 FD In-Stock Unstable P2RX7 28 52 CCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217550702 HG In-Stock Unstable CA2 16 42 CCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217550702 HG In-Stock Unstable TBXA2R 39 42 CCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217550702 HG In-Stock Unstable TBXAS1 28 43 CCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217550702 HG In-Stock Unstable BMP1 55 36 CCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217550702 HG In-Stock Unstable CA1 17 42 CCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217550702 HG In-Stock Unstable MMP13 48 39 CCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217550702 HG In-Stock Unstable ALOX15B 0 43 CCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217550702 HG In-Stock Unstable ALOX15 55 45 CCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217550702 HG In-Stock Unstable MMP9 44 39 CCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217550702 HG In-Stock Unstable PTGDR 29 41 CCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217550702 HG In-Stock Unstable IAP 0 49 CCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217550702 HG In-Stock Unstable CA9 25 42 CCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217550702 HG In-Stock Unstable MMP1 40 38 CCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217550702 HG In-Stock Unstable AKR1C3 29 45 CCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217550702 HG In-Stock Unstable AKR1C2 49 37 C[C@@]1(c2ccccc2)OC[C@@H](CN2CCC[C@@H](CN)C2)O1 ZINC000217550744 CD For-Sale Unstable ADRA1D 16 41 C[C@@]1(c2ccccc2)OC[C@@H](CN2CCC[C@@H](CN)C2)O1 ZINC000217550744 CD For-Sale Unstable ADRA1B 15 41 COc1ccc(-c2ccc(S(=O)(=O)N3CCC4(CC3)OC(=O)c3ccccc34)cc2)cc1 ZINC000217550787 II For-Sale Unstable NPY5R 32 45 COc1ccc(-c2ccc(S(=O)(=O)N3CCC4(CC3)OC(=O)c3ccccc34)cc2)cc1 ZINC000217550787 II For-Sale Unstable PKM 23 51 CCN(CCc1ccncc1)C(=O)NCCc1ccc(Br)cc1 ZINC000217550797 GH For-Sale Unstable LIG1 0 40 CCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217550823 IG In-Stock Unstable TBXAS1 18 44 CCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217550823 IG In-Stock Unstable BDKRB1 0 40 CCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217550823 IG In-Stock Unstable ALOX15 40 37 CCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217550823 IG In-Stock Unstable PTGDR 25 43 CCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217550823 IG In-Stock Unstable IAP 0 50 CCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217550823 IG In-Stock Unstable PTGDR2 17 43 CCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217550823 IG In-Stock Unstable SCMU_MYCTU 0 44 C[C@]1(c2ccccc2)OC[C@H](CN2CCC[C@@H](CN)C2)O1 ZINC000217550835 CD For-Sale Unstable ADRA1D 16 41 C[C@]1(c2ccccc2)OC[C@H](CN2CCC[C@@H](CN)C2)O1 ZINC000217550835 CD For-Sale Unstable ADRA1B 15 41 COC(=O)CS[C@@H]1CCN(C(=O)c2cccnc2)C1 ZINC000217550897 CD In-Stock Unstable SLC18A3 24 48 O=C1OC2(CCN(S(=O)(=O)c3ccc(Oc4ccccc4)cc3)CC2)c2ccccc21 ZINC000217550899 II For-Sale Unstable NPY5R 34 41 O=C(NCCc1ccc(Br)cc1)Nc1ccccc1N1CCOCC1 ZINC000217550919 HH For-Sale Unstable KCNQ2 81 42 O=C(NCCc1ccc(Br)cc1)Nc1ccccc1N1CCOCC1 ZINC000217550919 HH For-Sale Unstable CSF1R 0 48 CCCCNS(=O)(=O)c1ccc(NCc2ccco2)c(C(=O)O)c1 ZINC000217550923 FF In-Stock Unstable CASP3 15 40 C[C@@]1(c2ccccc2)OC[C@H](CN2CCC[C@@H](CN)C2)O1 ZINC000217550927 CD For-Sale Unstable ADRA1D 16 41 C[C@@]1(c2ccccc2)OC[C@H](CN2CCC[C@@H](CN)C2)O1 ZINC000217550927 CD For-Sale Unstable ADRA1B 15 41 COC(=O)CS[C@H]1CCN(C(=O)c2cccnc2)C1 ZINC000217550990 CD In-Stock Unstable SLC18A3 24 48 O=C1OC2(CCN(S(=O)(=O)c3ccc(Br)cc3)CC2)c2ccccc21 ZINC000217551013 HG For-Sale Unstable NPY5R 31 49 CN1CCN(c2ccc(NC(=O)NCCc3ccc(Br)cc3)cc2)CC1 ZINC000217551032 HH For-Sale Unstable HTR1B 15 41 CN1CCN(c2ccc(NC(=O)NCCc3ccc(Br)cc3)cc2)CC1 ZINC000217551032 HH For-Sale Unstable LCK 15 41 CN1CCN(c2ccc(NC(=O)NCCc3ccc(Br)cc3)cc2)CC1 ZINC000217551032 HH For-Sale Unstable CTSK 18 43 CN1CCN(c2ccc(NC(=O)NCCc3ccc(Br)cc3)cc2)CC1 ZINC000217551032 HH For-Sale Unstable PRNP 39 45 CN1CCN(c2ccc(NC(=O)NCCc3ccc(Br)cc3)cc2)CC1 ZINC000217551032 HH For-Sale Unstable MTOR 29 42 CN1CCN(c2ccc(NC(=O)NCCc3ccc(Br)cc3)cc2)CC1 ZINC000217551032 HH For-Sale Unstable HCK 27 41 CN1CCN(c2ccc(NC(=O)NCCc3ccc(Br)cc3)cc2)CC1 ZINC000217551032 HH For-Sale Unstable FLT3 15 45 CCCCNS(=O)(=O)c1ccc(NC[C@@H]2CCCO2)c(C(=O)O)c1 ZINC000217551033 FE In-Stock Unstable BDKRB1 28 40 NC[C@@H]1CCCN(CC(=O)N2CCC[C@@H]2c2cccs2)C1 ZINC000217551066 DE For-Sale Unstable UTS2R 45 30 CCCCNS(=O)(=O)c1ccc(NC[C@H]2CCCO2)c(C(=O)O)c1 ZINC000217551099 FE In-Stock Unstable BDKRB1 28 40 N#Cc1ccccc1S(=O)(=O)N1CCC2(CC1)OC(=O)c1ccccc12 ZINC000217551134 FE For-Sale Unstable NPY5R 30 44 O=C(NCCc1ccc(Br)cc1)Nc1ccc(N2CCCCC2)cc1 ZINC000217551155 HJ On-Demand Unstable GPBAR1 0 42 O=C(NCCc1ccc(Br)cc1)Nc1ccc(N2CCCCC2)cc1 ZINC000217551155 HJ On-Demand Unstable NAMPT 18 45 Cc1c(Cl)nc(C2CC2)nc1N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217551176 DG For-Sale Unstable CHRM3 15 47 CCCCNS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217551210 EE In-Stock Unstable HTR7 23 40 CCCCNS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217551210 EE In-Stock Unstable CASP3 24 43 CCCCNS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217551210 EE In-Stock Unstable KCNQ2 64 34 CCCCNS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217551210 EE In-Stock Unstable HTR6 0 40 CCCCNS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217551210 EE In-Stock Unstable PNMT 15 40 CCCCNS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217551210 EE In-Stock Unstable SFRP1 58 32 NS(=O)(=O)c1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217551259 HD For-Sale Unstable NPY5R 30 43 NS(=O)(=O)c1ccc(S(=O)(=O)N2CCC3(CC2)OC(=O)c2ccccc23)cc1 ZINC000217551259 HD For-Sale Unstable CA12 15 40 Cc1c(Cl)nc(C2CC2)nc1N[C@H]1CCN2CCCC[C@@H]12 ZINC000217551266 DG For-Sale Unstable CHRM3 15 47 N#CSc1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217551279 GI For-Sale Unstable NCE103 15 43 CCCCNS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217551327 EE In-Stock Unstable CASP3 23 42 CCCCNS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217551327 EE In-Stock Unstable KCNQ2 61 33 CCCCNS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217551327 EE In-Stock Unstable SFRP1 50 32 O=C1OC2(CCN(S(=O)(=O)Cc3cccc(C(F)(F)F)c3)CC2)c2ccccc21 ZINC000217551363 IH In-Stock Unstable NPY5R 29 50 COC(=O)c1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217551390 GH On-Demand Unstable ADRB1 30 45 COC(=O)c1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217551390 GH On-Demand Unstable ADRB3 37 45 COC(=O)c1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217551390 GH On-Demand Unstable CA1 15 45 COC(=O)c1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217551390 GH On-Demand Unstable F7 22 45 COC(=O)c1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217551390 GH On-Demand Unstable ACR 61 44 COC(=O)c1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217551390 GH On-Demand Unstable CA9 17 45 COC(=O)c1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217551390 GH On-Demand Unstable IDO1 18 42 COC(=O)c1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217551390 GH On-Demand Unstable NCE103 24 45 CCCCNS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1 ZINC000217551441 ED In-Stock Unstable HTR7 19 40 CCCCNS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1 ZINC000217551441 ED In-Stock Unstable CASP3 23 41 CCCCNS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1 ZINC000217551441 ED In-Stock Unstable SLC6A9 19 46 Cc1cccc(Oc2ccc(S(=O)(=O)N3CCC4(CC3)OC(=O)c3ccccc34)cc2)c1 ZINC000217551476 IJ For-Sale Unstable NPY5R 28 40 COC(=O)CS[C@H]1CCN(C(=O)c2ccccc2C)C1 ZINC000217551481 CE In-Stock Unstable CHRM2 17 45 COC(=O)CS[C@H]1CCN(C(=O)c2ccccc2C)C1 ZINC000217551481 CE In-Stock Unstable SLC6A1 44 35 COC(=O)CS[C@H]1CCN(C(=O)c2ccccc2C)C1 ZINC000217551481 CE In-Stock Unstable CCR8 64 37 O=C(NCCc1ccc(Br)cc1)N(Cc1ccccc1)c1ccccc1 ZINC000217551494 HK For-Sale Unstable AMP1_PLAFQ 29 41 COC(=O)CS[C@@H]1CCN(C(=O)c2ccccc2C)C1 ZINC000217551561 CE In-Stock Unstable CHRM2 17 45 COC(=O)CS[C@@H]1CCN(C(=O)c2ccccc2C)C1 ZINC000217551561 CE In-Stock Unstable SLC6A1 44 35 COC(=O)CS[C@@H]1CCN(C(=O)c2ccccc2C)C1 ZINC000217551561 CE In-Stock Unstable CCR8 64 37 Cc1ccccc1[C@@H](C)NC(=O)CN1CCC[C@@H](CN)C1 ZINC000217551565 CD For-Sale Unstable DRD4 0 40 Cc1ccccc1[C@@H](C)NC(=O)CN1CCC[C@@H](CN)C1 ZINC000217551565 CD For-Sale Unstable SLC6A1 46 41 Cc1ccccc1[C@@H](C)NC(=O)CN1CCC[C@@H](CN)C1 ZINC000217551565 CD For-Sale Unstable CCR3 44 34 Cc1ccccc1[C@@H](C)NC(=O)CN1CCC[C@@H](CN)C1 ZINC000217551565 CD For-Sale Unstable BIRC2 47 36 CCCCNS(=O)(=O)c1ccc(NCCCOCC)c(C(=O)O)c1 ZINC000217551573 FE In-Stock Unstable CASP3 22 44 O=C1OC2(CCN(S(=O)(=O)c3cccc(-c4ccccc4)c3)CC2)c2ccccc21 ZINC000217551596 HI For-Sale Unstable NPY5R 48 51 O=C1OC2(CCN(S(=O)(=O)c3cccc(-c4ccccc4)c3)CC2)c2ccccc21 ZINC000217551596 HI For-Sale Unstable PKM 32 41 O=C1OC2(CCN(S(=O)(=O)c3cccc(-c4ccccc4)c3)CC2)c2ccccc21 ZINC000217551596 HI For-Sale Unstable AKR1C3 47 36 O=C(NCCc1ccc(Br)cc1)Nc1ccc2ccccc2c1 ZINC000217551605 FJ For-Sale Unstable CA1 17 48 O=C(NCCc1ccc(Br)cc1)Nc1ccc2ccccc2c1 ZINC000217551605 FJ For-Sale Unstable GUAB 0 40 O=C(NCCc1ccc(Br)cc1)Nc1ccc2ccccc2c1 ZINC000217551605 FJ For-Sale Unstable RAF1 23 42 O=C(NCCc1ccc(Br)cc1)Nc1ccc2ccccc2c1 ZINC000217551605 FJ For-Sale Unstable Q8MMZ8_EIMTE 0 42 O=C(NCCc1ccc(Br)cc1)Nc1ccc2ccccc2c1 ZINC000217551605 FJ For-Sale Unstable NCE103 28 48 Cc1ccccc1[C@H](C)NC(=O)CN1CCC[C@@H](CN)C1 ZINC000217551638 CD For-Sale Unstable DRD4 0 40 Cc1ccccc1[C@H](C)NC(=O)CN1CCC[C@@H](CN)C1 ZINC000217551638 CD For-Sale Unstable SLC6A1 46 41 Cc1ccccc1[C@H](C)NC(=O)CN1CCC[C@@H](CN)C1 ZINC000217551638 CD For-Sale Unstable CCR3 44 34 Cc1ccccc1[C@H](C)NC(=O)CN1CCC[C@@H](CN)C1 ZINC000217551638 CD For-Sale Unstable BIRC2 47 36 O=C(CCCOCc1ccccc1)N1CCCn2nc(CO)cc2C1 ZINC000217551642 EE In-Stock Unstable PREP 46 37 CCCCNS(=O)(=O)c1ccc(NCCCOC(C)C)c(C(=O)O)c1 ZINC000217551686 FF In-Stock Unstable CASP3 15 43 CCCCNS(=O)(=O)c1ccc(NCCCOC(C)C)c(C(=O)O)c1 ZINC000217551686 FF In-Stock Unstable BDKRB1 16 41 O=C1OC2(CCN(S(=O)(=O)CCCOc3ccccc3)CC2)c2ccccc21 ZINC000217551691 HF For-Sale Unstable NPY5R 38 42 CC(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217551797 BD For-Sale Unstable NPY5R 38 45 CCCCCNc1ccc(S(=O)(=O)NCCCC)cc1C(=O)O ZINC000217551798 EG In-Stock Unstable CASP3 22 48 CCCCCNc1ccc(S(=O)(=O)NCCCC)cc1C(=O)O ZINC000217551798 EG In-Stock Unstable BDKRB1 0 43 COc1cc2c(cc1OC)CN(C(=O)[C@]13C[C@@H]4C[C@@H](C[C@@](Cl)(C4)C1)C3)CC2 ZINC000217551832 GI In-Stock Unstable ABCB1 0 41 CCCN(CCC)C(=O)NCCc1ccc(Br)cc1 ZINC000217551839 EH On-Demand Unstable LIG1 0 43 CC(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217551891 BD For-Sale Unstable NPY5R 38 45 Cc1c(Cl)nc(C2CC2)nc1N[C@@H]1CCN2CCC[C@@H]12 ZINC000217551903 CF For-Sale Unstable CHRM3 0 45 COc1cc2c(cc1OC)CN(C(=O)[C@@]13C[C@@H]4C[C@@H](C[C@](Cl)(C4)C1)C3)CC2 ZINC000217551921 GI In-Stock Unstable ABCB1 0 41 CCCCNS(=O)(=O)c1ccc(NCCC(C)C)c(C(=O)O)c1 ZINC000217551934 EF In-Stock Unstable CASP3 17 47 Cc1c(Cl)nc(C2CC2)nc1N[C@H]1CCN2CCC[C@@H]12 ZINC000217551984 CF For-Sale Unstable CHRM3 0 45 C[C@@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccc(Br)cc1 ZINC000217551985 FE On-Demand Unstable SDH1 0 47 C[C@@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccc(Br)cc1 ZINC000217551985 FE On-Demand Unstable BIRC2 29 41 CN(C)C[C@@]1(O)CCCN(C(=O)CN2CCC(c3ccccc3)CC2)C1 ZINC000217552005 FD In-Stock Unstable CCR5 23 41 CCC(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217552016 CE For-Sale Unstable NPY5R 33 43 CCCCNS(=O)(=O)c1ccc(N[C@@H](C)CCC)c(C(=O)O)c1 ZINC000217552044 EG In-Stock Unstable CASP3 22 48 C[C@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccc(Br)cc1 ZINC000217552051 FE On-Demand Unstable SDH1 0 47 C[C@H](NC(=O)CN1CCC[C@@H](CN)C1)c1ccc(Br)cc1 ZINC000217552051 FE On-Demand Unstable BIRC2 29 41 O=CNCCCNC(=O)NCCc1ccc(Br)cc1 ZINC000217552072 ED For-Sale Unstable LIG1 0 40 CN(C)C[C@]1(O)CCCN(C(=O)CN2CCC(c3ccccc3)CC2)C1 ZINC000217552082 FD In-Stock Unstable CCR5 23 41 CCC(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217552103 CE For-Sale Unstable NPY5R 33 43 CCCCNS(=O)(=O)c1ccc(N[C@H](C)CCC)c(C(=O)O)c1 ZINC000217552136 EG In-Stock Unstable CASP3 22 48 CC(C)[C@@H](NC(=O)CN1CCC[C@@H](CN)C1)c1cccs1 ZINC000217552174 DE For-Sale Unstable BIRC2 42 35 C=CCCC(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217552212 CF For-Sale Unstable NPY5R 25 41 OCCCCCCNCc1ccc(I)cc1 ZINC000217552214 EF On-Demand Unstable LEF 47 33 OCCCCCCNCc1ccc(I)cc1 ZINC000217552214 EF On-Demand Unstable GPM3 0 52 O=C(Nc1ccc(N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)nc1)c1ccc2c(c1)OCCCO2 ZINC000217552217 JG In-Stock Unstable CHRNA4 25 40 CCCCNS(=O)(=O)c1ccc(N[C@@H](C)COC)c(C(=O)O)c1 ZINC000217552250 ED In-Stock Unstable CASP3 16 41 CC(C)[C@H](NC(=O)CN1CCC[C@@H](CN)C1)c1cccs1 ZINC000217552278 DE For-Sale Unstable BIRC2 42 35 C=CCCC(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217552301 CF For-Sale Unstable NPY5R 25 41 CCCCNS(=O)(=O)c1ccc(N[C@H](C)COC)c(C(=O)O)c1 ZINC000217552360 ED In-Stock Unstable CASP3 16 41 CC1(C)C[C@H]2C[C@@](C)(CN2C(=O)NCCc2ccc(Br)cc2)C1 ZINC000217552374 GJ For-Sale Unstable AVPR2 18 42 CC1(C)C[C@H]2C[C@@](C)(CN2C(=O)NCCc2ccc(Br)cc2)C1 ZINC000217552374 GJ For-Sale Unstable AVPR1A 35 42 CCCCC(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217552422 CF For-Sale Unstable NPY5R 28 42 COC(=O)CS[C@@H]1CCN(C(=O)c2ccc(C#N)cc2)C1 ZINC000217552448 DD In-Stock Unstable GRM3 16 44 COC(=O)CS[C@@H]1CCN(C(=O)c2ccc(C#N)cc2)C1 ZINC000217552448 DD In-Stock Unstable L3MBTL3 60 36 C[C@@H](CNC(=O)CN1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217552453 CD For-Sale Unstable SLC6A1 49 36 C[C@@H](CNC(=O)CN1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217552453 CD For-Sale Unstable CCR5 21 41 C[C@@H](CNC(=O)CN1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217552453 CD For-Sale Unstable BIRC2 50 35 CCCNc1ccc(S(=O)(=O)NCC(C)C)cc1C(=O)O ZINC000217552466 DE In-Stock Unstable CASP3 16 41 CCCNc1ccc(S(=O)(=O)NCC(C)C)cc1C(=O)O ZINC000217552466 DE In-Stock Unstable BDKRB1 0 43 CC(C)(C)OC(=O)N1CC[C@@H](F)[C@@H](CN)CC1 ZINC000217552485 BD For-Sale Unstable GPR119 40 43 CCCCC(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217552498 CF For-Sale Unstable NPY5R 28 42 CNC(=O)Nc1ccc(CO)c(Cl)c1 ZINC000217552516 BD For-Sale Unstable P95276_MYCTO 0 47 CNC(=O)Nc1ccc(CO)c(Cl)c1 ZINC000217552516 BD For-Sale Unstable PPX1 0 43 Cc1ccc(C(=O)Nc2ccc(N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)nc2)c(=O)n1C ZINC000217552523 IE In-Stock Unstable CHRNA4 27 43 COC(=O)CS[C@H]1CCN(C(=O)c2ccc(C#N)cc2)C1 ZINC000217552535 DD In-Stock Unstable GRM3 16 44 COC(=O)CS[C@H]1CCN(C(=O)c2ccc(C#N)cc2)C1 ZINC000217552535 DD In-Stock Unstable L3MBTL3 60 36 C[C@H](CNC(=O)CN1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217552539 CD For-Sale Unstable SLC6A1 49 36 C[C@H](CNC(=O)CN1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217552539 CD For-Sale Unstable CCR5 21 41 C[C@H](CNC(=O)CN1CCC[C@@H](CN)C1)c1ccccc1 ZINC000217552539 CD For-Sale Unstable BIRC2 50 35 CN(C)c1cccc(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217552556 FH For-Sale Unstable RAF1 17 40 CN(C)c1cccc(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217552556 FH For-Sale Unstable NCE103 15 40 CC(C)CNS(=O)(=O)c1ccc(NC(C)C)c(C(=O)O)c1 ZINC000217552564 DE In-Stock Unstable F3 66 32 CC(C)CNS(=O)(=O)c1ccc(NC(C)C)c(C(=O)O)c1 ZINC000217552564 DE In-Stock Unstable MTNN 41 33 CC(C)(C)OC(=O)N1CC[C@@H](CN)[C@H](F)CC1 ZINC000217552582 BD For-Sale Unstable GPR119 40 43 CCOCC(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217552616 CD For-Sale Unstable NPY5R 29 41 COC(=O)CS[C@@H]1CCN(C(=O)/C=C/c2ccccc2)C1 ZINC000217552636 DE In-Stock Unstable CCR2 62 37 COC(=O)CS[C@@H]1CCN(C(=O)/C=C/c2ccccc2)C1 ZINC000217552636 DE In-Stock Unstable GPR183 0 45 CN1CCc2nc(NC(=O)NCCc3ccc(Br)cc3)sc2C1 ZINC000217552673 GG For-Sale Unstable F10 25 46 CC(C)(C)OC(=O)N1CC[C@H](F)[C@@H](CN)CC1 ZINC000217552676 BD For-Sale Unstable GPR119 40 43 CCCCNc1ccc(S(=O)(=O)NCC(C)C)cc1C(=O)O ZINC000217552681 EF In-Stock Unstable CASP3 15 42 CCN1c2ccccc2C[C@H]1C=O ZINC000217552683 AD In-Stock Unstable TPP2 52 33 CCOCC(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217552709 CD For-Sale Unstable NPY5R 29 41 COC(=O)CS[C@H]1CCN(C(=O)/C=C/c2ccccc2)C1 ZINC000217552722 DE In-Stock Unstable CCR2 62 37 COC(=O)CS[C@H]1CCN(C(=O)/C=C/c2ccccc2)C1 ZINC000217552722 DE In-Stock Unstable GPR183 0 45 Cn1nnc(-c2ccc(NC(=O)CCN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)cc2)n1 ZINC000217552736 HD In-Stock Unstable CHRNA4 32 53 CCN1c2ccccc2C[C@@H]1C=O ZINC000217552765 AD In-Stock Unstable TPP2 52 33 CC(C)(C)OC(=O)N1CC[C@H](F)[C@H](CN)CC1 ZINC000217552771 BD For-Sale Unstable GPR119 40 43 CC(C)CNc1ccc(S(=O)(=O)NCC(C)C)cc1C(=O)O ZINC000217552796 EE In-Stock Unstable CASP3 19 41 CC(C)CNc1ccc(S(=O)(=O)NCC(C)C)cc1C(=O)O ZINC000217552796 EE In-Stock Unstable MTNN 77 36 Nc1ccccc1C(=O)NC(=O)NCCc1ccc(Br)cc1 ZINC000217552803 FF For-Sale Unstable LIG1 0 40 O=C1O[C@@]2(CCCN(C(=O)c3ccco3)C2)c2ccccc21 ZINC000217552821 CF For-Sale Unstable NPY5R 25 41 COC(=O)CS[C@@H]1CCN(C(=O)Cc2ccc(F)cc2)C1 ZINC000217552823 DD In-Stock Unstable MLNR 44 47 CCCN1c2ccccc2C[C@H]1C=O ZINC000217552875 AE In-Stock Unstable TPP2 55 35 O=C1O[C@]2(CCCN(C(=O)c3ccco3)C2)c2ccccc21 ZINC000217552898 CF For-Sale Unstable NPY5R 25 41 COC(=O)CS[C@H]1CCN(C(=O)Cc2ccc(F)cc2)C1 ZINC000217552901 DD In-Stock Unstable MLNR 44 47 NC(=O)c1ccccc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217552918 FF For-Sale Unstable HCAR2 16 41 NC(=O)c1ccccc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217552918 FF For-Sale Unstable PAGA 0 45 O=C(Nc1ccc(N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)nc1)c1ccc2c(c1)OCO2 ZINC000217552940 IF In-Stock Unstable CHRNA4 25 41 Cc1cn2c(CN(C)C(=O)[C@@H]3C[C@@H]3c3ccccc3C(F)(F)F)c(C)nc2s1 ZINC000217552943 HJ On-Demand Unstable RBP4 70 34 CCCN1c2ccccc2C[C@@H]1C=O ZINC000217552960 AE In-Stock Unstable TPP2 55 35 CC(C)(C)CC(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217553014 DG For-Sale Unstable NPY5R 27 40 Cc1cn2c(CN(C)C(=O)[C@H]3C[C@@H]3c3ccccc3C(F)(F)F)c(C)nc2s1 ZINC000217553023 HJ On-Demand Unstable RBP4 70 34 CCOc1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1OCC ZINC000217553033 II For-Sale Unstable AGPAT2 32 41 CC(C)(C)CC(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217553100 DG For-Sale Unstable NPY5R 27 40 Cc1cn2c(CN(C)C(=O)[C@@H]3C[C@H]3c3ccccc3C(F)(F)F)c(C)nc2s1 ZINC000217553110 HJ On-Demand Unstable RBP4 70 34 CC(C)CNS(=O)(=O)c1ccc(NC(C)(C)C)c(C(=O)O)c1 ZINC000217553127 EF In-Stock Unstable MTNN 44 31 COc1ccc(Br)cc1S(=O)(=O)Nc1cc(F)cc(Cl)c1 ZINC000217553149 GI On-Demand Unstable COLA 0 41 COc1ccc(Br)cc1S(=O)(=O)Nc1cc(F)cc(Cl)c1 ZINC000217553149 GI On-Demand Unstable CPT1A 18 41 COc1ccc(Br)cc1S(=O)(=O)Nc1cc(F)cc(Cl)c1 ZINC000217553149 GI On-Demand Unstable ALPL 28 52 CC[C@H](C)[C@@H]1NC(=O)[C@@H](C)N(CC[S@@](=O)CC)C1=O ZINC000217553152 CC For-Sale Unstable GALR1 40 37 O=C1O[C@@]2(CCCN(C(=O)c3ccccc3)C2)c2ccccc21 ZINC000217553198 DF For-Sale Unstable NPY5R 40 47 Cc1cn2c(CN(C)C(=O)[C@H]3C[C@H]3c3ccccc3C(F)(F)F)c(C)nc2s1 ZINC000217553201 HJ On-Demand Unstable RBP4 70 34 Cc1cccc(C(=O)N2c3ccccc3CC[C@@H]2C)c1I ZINC000217553202 GJ On-Demand Unstable ACE 19 40 Cc1cccc(C(=O)N2c3ccccc3CC[C@@H]2C)c1I ZINC000217553202 GJ On-Demand Unstable PTGDR2 34 43 C=CCNc1ccc(S(=O)(=O)NCC(C)C)cc1C(=O)O ZINC000217553235 DD In-Stock Unstable BDKRB1 0 41 Cc1cccc(C(=O)N2c3ccccc3CC[C@H]2C)c1I ZINC000217553295 GJ On-Demand Unstable ACE 19 40 Cc1cccc(C(=O)N2c3ccccc3CC[C@H]2C)c1I ZINC000217553295 GJ On-Demand Unstable PTGDR2 34 43 O=C1O[C@]2(CCCN(C(=O)c3ccccc3)C2)c2ccccc21 ZINC000217553301 DF For-Sale Unstable NPY5R 40 47 CC(C)CNS(=O)(=O)c1ccc(NC2CC2)c(C(=O)O)c1 ZINC000217553346 DD In-Stock Unstable SFRP1 68 34 CC(C)CNS(=O)(=O)c1ccc(NC2CC2)c(C(=O)O)c1 ZINC000217553346 DD In-Stock Unstable WNT3 41 34 O=C(/C=C\c1ccc(Cl)cc1Cl)N[C@@H]1CC[C@H](C(=O)O)C1 ZINC000217553400 EG For-Sale Unstable BOTA 32 56 O=C1O[C@@]2(CCCN(C(=O)c3ccncc3)C2)c2ccccc21 ZINC000217553422 DE For-Sale Unstable NPY5R 48 44 CC(C)CNS(=O)(=O)c1ccc(NC2CCCC2)c(C(=O)O)c1 ZINC000217553444 EF In-Stock Unstable CASP3 0 42 CC(C)CNS(=O)(=O)c1ccc(NC2CCCC2)c(C(=O)O)c1 ZINC000217553444 EF In-Stock Unstable SFRP1 56 33 CC(C)CNS(=O)(=O)c1ccc(NC2CCCC2)c(C(=O)O)c1 ZINC000217553444 EF In-Stock Unstable WNT3 45 33 O=C(NCCc1ccc(Br)cc1)Nc1ccc2cn[nH]c2c1 ZINC000217553485 FH For-Sale Unstable Q8MMZ8_EIMTE 23 43 O=C1O[C@]2(CCCN(C(=O)c3ccncc3)C2)c2ccccc21 ZINC000217553503 DE For-Sale Unstable NPY5R 48 44 CC(C)CNS(=O)(=O)c1ccc(NC2CCCCC2)c(C(=O)O)c1 ZINC000217553550 FG In-Stock Unstable CASP3 0 41 CC(C)CNS(=O)(=O)c1ccc(NC2CCCCC2)c(C(=O)O)c1 ZINC000217553550 FG In-Stock Unstable SFRP1 50 32 CC(C)CNS(=O)(=O)c1ccc(NC2CCCCC2)c(C(=O)O)c1 ZINC000217553550 FG In-Stock Unstable WNT3 45 32 CC(C)(C)c1ccccc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217553575 GK On-Demand Unstable AMP1_PLAFQ 19 40 O=C1O[C@@]2(CCCN(C(=O)c3cccnc3)C2)c2ccccc21 ZINC000217553608 DE For-Sale Unstable NPY5R 50 44 O=C1O[C@]2(CCCN(C(=O)c3cccnc3)C2)c2ccccc21 ZINC000217553665 DE For-Sale Unstable NPY5R 50 44 Cc1nnc(CN(C)C(=O)c2cc3ccccc3cc2O)o1 ZINC000217553669 CF In-Stock Unstable HSP90AB1 48 39 NS(=O)(=O)c1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217553710 IE On-Demand Unstable CA2 174 64 NS(=O)(=O)c1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217553710 IE On-Demand Unstable CA6 29 49 NS(=O)(=O)c1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217553710 IE On-Demand Unstable CA1 151 64 NS(=O)(=O)c1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217553710 IE On-Demand Unstable CA7 90 60 NS(=O)(=O)c1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217553710 IE On-Demand Unstable CA13 40 49 NS(=O)(=O)c1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217553710 IE On-Demand Unstable CA5B 66 60 NS(=O)(=O)c1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217553710 IE On-Demand Unstable CA4 118 64 NS(=O)(=O)c1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217553710 IE On-Demand Unstable CA5A 68 60 NS(=O)(=O)c1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217553710 IE On-Demand Unstable CA14 70 58 NS(=O)(=O)c1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217553710 IE On-Demand Unstable MMP14 23 40 NS(=O)(=O)c1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217553710 IE On-Demand Unstable CA12 116 64 NS(=O)(=O)c1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217553710 IE On-Demand Unstable CA9 128 64 NS(=O)(=O)c1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217553710 IE On-Demand Unstable CAH_METTE 32 49 NS(=O)(=O)c1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217553710 IE On-Demand Unstable IDO1 19 46 NS(=O)(=O)c1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217553710 IE On-Demand Unstable CYNT 48 56 NS(=O)(=O)c1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217553710 IE On-Demand Unstable NCE103 47 60 NS(=O)(=O)c1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217553710 IE On-Demand Unstable ALPI 25 60 NS(=O)(=O)c1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217553710 IE On-Demand Unstable LIG1 0 70 NS(=O)(=O)c1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217553710 IE On-Demand Unstable CA15 19 49 NS(=O)(=O)c1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217553710 IE On-Demand Unstable MTCA1 59 56 NS(=O)(=O)c1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217553710 IE On-Demand Unstable P96878_MYCTU 74 56 NS(=O)(=O)c1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217553710 IE On-Demand Unstable CA 0 51 NS(=O)(=O)c1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217553710 IE On-Demand Unstable A6YCJ1_9METZ 32 64 NS(=O)(=O)c1ccc(CCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217553710 IE On-Demand Unstable Q5TU56_ANOGA 0 49 COc1cc(/C=C\C(=O)O)ccc1OCc1cnc(C)s1 ZINC000217553741 DG For-Sale Unstable PTGER2 27 52 COc1cc(/C=C\C(=O)O)ccc1OCc1cnc(C)s1 ZINC000217553741 DG For-Sale Unstable APP 20 42 COc1cc(/C=C\C(=O)O)ccc1OCc1cnc(C)s1 ZINC000217553741 DG For-Sale Unstable AKR1C3 34 43 CC(C)CNS(=O)(=O)c1ccc(NCCO)c(C(=O)O)c1 ZINC000217553774 DC In-Stock Unstable CASP3 18 41 CC(C)CNS(=O)(=O)c1ccc(NCCO)c(C(=O)O)c1 ZINC000217553774 DC In-Stock Unstable BDKRB1 0 43 O=C1O[C@@]2(CCCN(C(=O)c3ccccn3)C2)c2ccccc21 ZINC000217553783 DE For-Sale Unstable NPY5R 48 43 COC(=O)CS[C@@H]1CCN(C(=O)Cc2ccccc2Cl)C1 ZINC000217553801 EE In-Stock Unstable DPP7 18 40 O=C(NCCc1ccc(Br)cc1)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217553821 JK For-Sale Unstable RAF1 34 46 O=C(NCCc1ccc(Br)cc1)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217553821 JK For-Sale Unstable EPHX2 15 40 O=C(NCCc1ccc(Br)cc1)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217553821 JK For-Sale Unstable Q8MMZ8_EIMTE 25 46 O=C(NCCc1ccc(Br)cc1)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217553821 JK For-Sale Unstable PTPA 0 44 O=C1O[C@]2(CCCN(C(=O)c3ccccn3)C2)c2ccccc21 ZINC000217553853 DE For-Sale Unstable NPY5R 48 43 COC(=O)CS[C@H]1CCN(C(=O)Cc2ccccc2Cl)C1 ZINC000217553866 EE In-Stock Unstable DPP7 18 40 CC(C)CNS(=O)(=O)c1ccc(NCCCO)c(C(=O)O)c1 ZINC000217553894 ED In-Stock Unstable CASP3 16 41 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable ACE 17 42 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable LHCGR 50 45 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable OPRM1 83 73 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable OPRD1 85 73 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable MME 41 42 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable NPR1 54 43 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable TACR1 16 48 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable HLA-DRB3 18 55 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable MC4R 58 48 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable FCER2 45 34 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable TACR2 21 54 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable GLO1 40 35 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable NPY1R 19 43 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable KLK3 52 38 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable CTSB 50 47 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable PAPA1_CARPA 71 47 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable CCKAR 18 44 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable NTSR1 147 66 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable NTSR2 108 47 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable CTSK 15 47 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable CTSL 29 53 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable PGA 40 45 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable F2R 61 54 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable NPFFR2 74 41 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable C3AR1 44 53 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable HLA-A 110 51 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable TACR3 24 53 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable MC3R 72 45 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable MC5R 70 43 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable CAPNS1 61 39 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable MMP8 19 41 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable GRIA1 104 41 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable GRPR 69 35 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable HLA-DRB1 106 47 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable REN 34 41 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable REN1 43 40 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable F11 15 40 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable PCSK5 41 34 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable FURIN 83 41 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable SORT1 60 43 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable CCKBR 20 47 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable CAPN1 77 45 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable MMP9 15 41 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable CASP1 24 43 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable CAPN2 120 41 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable MC1R 114 48 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable ST14 59 47 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable PROC 33 40 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable MMP1 23 43 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable FPR1 72 39 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable NPR 67 36 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable KISS1R 82 44 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable QRFPR 57 42 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable F2RL1 63 50 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable NPFFR1 70 35 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable Q9NAW4_PLAFA 25 45 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable TMPRSS6 68 47 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable HPN 55 35 CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](N)CCCN=C(N)N)C(=O)NCC(=O)O ZINC000217553909 KA In-Stock Unstable H9B8T9_CAPHI 44 45 CCc1ccccc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217553925 EI On-Demand Unstable ANPEP 15 40 CCc1ccccc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217553925 EI On-Demand Unstable MTNR1A 20 40 CCc1ccccc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217553925 EI On-Demand Unstable AMP1_PLAFQ 23 42 CCc1ccccc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217553925 EI On-Demand Unstable ACAT 0 45 O=C1O[C@@]2(CCCN(C(=O)c3cnccn3)C2)c2ccccc21 ZINC000217553959 DD For-Sale Unstable NPY5R 47 43 C[C@H](C(=O)Nc1ccccc1)N1CCC[C@@H](CN)C1 ZINC000217553976 CD On-Demand Unstable ACE 31 41 C[C@H](C(=O)Nc1ccccc1)N1CCC[C@@H](CN)C1 ZINC000217553976 CD On-Demand Unstable CCR3 49 36 C[C@H](C(=O)Nc1ccccc1)N1CCC[C@@H](CN)C1 ZINC000217553976 CD On-Demand Unstable XIAP 41 33 C[C@H](C(=O)Nc1ccccc1)N1CCC[C@@H](CN)C1 ZINC000217553976 CD On-Demand Unstable BIRC2 48 36 CCCC[C@@H](CC)CNC[C@@H](O)COc1ccccc1 ZINC000217553990 CG For-Sale Unstable ADRB2 56 62 CCCC[C@@H](CC)CNC[C@@H](O)COc1ccccc1 ZINC000217553990 CG For-Sale Unstable ADRB1 70 46 CCCC[C@@H](CC)CNC[C@@H](O)COc1ccccc1 ZINC000217553990 CG For-Sale Unstable ADRB3 45 46 CCCC[C@@H](CC)CNC[C@@H](O)COc1ccccc1 ZINC000217553990 CG For-Sale Unstable ABCB1 16 45 CCCC[C@@H](CC)CNC[C@@H](O)COc1ccccc1 ZINC000217553990 CG For-Sale Unstable PDS 50 37 Nc1ccc(C(=O)NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217554023 FF For-Sale Unstable CYNT 18 40 Nc1ccc(C(=O)NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217554023 FF For-Sale Unstable LIG1 0 41 Nc1ccc(C(=O)NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217554023 FF For-Sale Unstable A6YCJ1_9METZ 17 46 COCCNc1ccc(S(=O)(=O)NCC(C)C)cc1C(=O)O ZINC000217554034 ED In-Stock Unstable BDKRB1 18 45 NCc1nnc2ccc(-c3ccc(Cl)cc3Cl)nn12 ZINC000217554038 CF In-Stock Unstable ALPL 40 35 NCc1nnc2ccc(-c3ccc(Cl)cc3Cl)nn12 ZINC000217554038 CF In-Stock Unstable DPP8 55 33 NCc1nnc2ccc(-c3ccc(Cl)cc3Cl)nn12 ZINC000217554038 CF In-Stock Unstable DPP9 50 34 O=C1O[C@]2(CCCN(C(=O)c3cnccn3)C2)c2ccccc21 ZINC000217554046 DD For-Sale Unstable NPY5R 47 43 C[C@@H](C(=O)Nc1ccccc1)N1CCC[C@@H](CN)C1 ZINC000217554060 CD On-Demand Unstable ACE 31 41 C[C@@H](C(=O)Nc1ccccc1)N1CCC[C@@H](CN)C1 ZINC000217554060 CD On-Demand Unstable CCR3 49 36 C[C@@H](C(=O)Nc1ccccc1)N1CCC[C@@H](CN)C1 ZINC000217554060 CD On-Demand Unstable XIAP 41 33 C[C@@H](C(=O)Nc1ccccc1)N1CCC[C@@H](CN)C1 ZINC000217554060 CD On-Demand Unstable BIRC2 48 36 O=S(=O)(Nc1cc(F)cc(Cl)c1)c1ccccc1Br ZINC000217554071 FI On-Demand Anodyne NR1I2 22 42 CCCC[C@H](CC)CNC[C@@H](O)COc1ccccc1 ZINC000217554103 CG For-Sale Unstable ADRB2 56 62 CCCC[C@H](CC)CNC[C@@H](O)COc1ccccc1 ZINC000217554103 CG For-Sale Unstable ADRB1 70 46 CCCC[C@H](CC)CNC[C@@H](O)COc1ccccc1 ZINC000217554103 CG For-Sale Unstable ADRB3 45 46 CCCC[C@H](CC)CNC[C@@H](O)COc1ccccc1 ZINC000217554103 CG For-Sale Unstable ABCB1 16 45 CCCC[C@H](CC)CNC[C@@H](O)COc1ccccc1 ZINC000217554103 CG For-Sale Unstable PDS 50 37 COCCCNc1ccc(S(=O)(=O)NCC(C)C)cc1C(=O)O ZINC000217554113 ED In-Stock Unstable CASP3 18 40 COCCCNc1ccc(S(=O)(=O)NCC(C)C)cc1C(=O)O ZINC000217554113 ED In-Stock Unstable BDKRB1 22 46 O=C(NCCc1ccc(Br)cc1)Nc1ccc(F)c(Cl)c1 ZINC000217554114 FJ For-Sale Unstable RAF1 31 46 O=C(NCCc1ccc(Br)cc1)Nc1ccc(F)c(Cl)c1 ZINC000217554114 FJ For-Sale Unstable CA12 15 42 O=C(NCCc1ccc(Br)cc1)Nc1ccc(F)c(Cl)c1 ZINC000217554114 FJ For-Sale Unstable ERBB4 44 36 O=C(NCCc1ccc(Br)cc1)Nc1ccc(F)c(Cl)c1 ZINC000217554114 FJ For-Sale Unstable CA9 15 42 O=C(NCCc1ccc(Br)cc1)Nc1ccc(F)c(Cl)c1 ZINC000217554114 FJ For-Sale Unstable Q8MMZ8_EIMTE 22 46 O=C(NCCc1ccc(Br)cc1)Nc1ccc(F)c(Cl)c1 ZINC000217554114 FJ For-Sale Unstable NCE103 29 43 O=C(NCCc1ccc(Br)cc1)Nc1ccc(F)c(Cl)c1 ZINC000217554114 FJ For-Sale Unstable P95276_MYCTO 0 43 COc1ccc(-c2ccc3nnc(CN)n3n2)cc1OC ZINC000217554137 CD In-Stock Unstable PDE4D 49 44 COc1ccc(-c2ccc3nnc(CN)n3n2)cc1OC ZINC000217554137 CD In-Stock Unstable MET 24 46 Cc1cc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)no1 ZINC000217554154 DE For-Sale Unstable NPY5R 32 41 COC(=O)CS[C@@H]1CCN(C(=O)c2ccc(F)cc2Cl)C1 ZINC000217554160 EF In-Stock Unstable P2RX7 34 47 CCCC[C@@H](CC)CNC[C@H](O)COc1ccccc1 ZINC000217554170 CG For-Sale Unstable ADRB2 56 62 CCCC[C@@H](CC)CNC[C@H](O)COc1ccccc1 ZINC000217554170 CG For-Sale Unstable ADRB1 70 46 CCCC[C@@H](CC)CNC[C@H](O)COc1ccccc1 ZINC000217554170 CG For-Sale Unstable ADRB3 45 46 CCCC[C@@H](CC)CNC[C@H](O)COc1ccccc1 ZINC000217554170 CG For-Sale Unstable ABCB1 16 45 CCCC[C@@H](CC)CNC[C@H](O)COc1ccccc1 ZINC000217554170 CG For-Sale Unstable PDS 50 37 CC(C)CNS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217554210 FF In-Stock Unstable ACPS 0 40 CCN(CC)c1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217554213 GJ For-Sale Unstable GHSR 19 41 CCN(CC)c1ccc(NC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217554213 GJ For-Sale Unstable NCE103 18 45 COC(=O)CS[C@H]1CCN(C(=O)c2ccc(F)cc2Cl)C1 ZINC000217554231 EF In-Stock Unstable P2RX7 34 47 Cc1cc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)no1 ZINC000217554233 DE For-Sale Unstable NPY5R 32 41 COc1ccc(OC)c(-c2ccc3nnc(CN)n3n2)c1 ZINC000217554238 CD In-Stock Unstable LRRK2 32 44 CCCC[C@H](CC)CNC[C@H](O)COc1ccccc1 ZINC000217554254 CG For-Sale Unstable ADRB2 56 62 CCCC[C@H](CC)CNC[C@H](O)COc1ccccc1 ZINC000217554254 CG For-Sale Unstable ADRB1 70 46 CCCC[C@H](CC)CNC[C@H](O)COc1ccccc1 ZINC000217554254 CG For-Sale Unstable ADRB3 45 46 CCCC[C@H](CC)CNC[C@H](O)COc1ccccc1 ZINC000217554254 CG For-Sale Unstable ABCB1 16 45 CCCC[C@H](CC)CNC[C@H](O)COc1ccccc1 ZINC000217554254 CG For-Sale Unstable PDS 50 37 CC(C)CNS(=O)(=O)c1ccc(N[C@@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217554301 GG In-Stock Unstable KCNA5 0 41 COc1ccccc1N1CCN(C(=O)NCCc2ccc(Br)cc2)CC1 ZINC000217554318 HH On-Demand Unstable HTR1A 108 53 COc1ccccc1N1CCN(C(=O)NCCc2ccc(Br)cc2)CC1 ZINC000217554318 HH On-Demand Unstable DRD2 88 54 COc1ccccc1N1CCN(C(=O)NCCc2ccc(Br)cc2)CC1 ZINC000217554318 HH On-Demand Unstable DRD1 32 48 COc1ccccc1N1CCN(C(=O)NCCc2ccc(Br)cc2)CC1 ZINC000217554318 HH On-Demand Unstable DRD4 51 51 COc1ccccc1N1CCN(C(=O)NCCc2ccc(Br)cc2)CC1 ZINC000217554318 HH On-Demand Unstable ADRA1D 85 47 COc1ccccc1N1CCN(C(=O)NCCc2ccc(Br)cc2)CC1 ZINC000217554318 HH On-Demand Unstable HTR1D 27 45 COc1ccccc1N1CCN(C(=O)NCCc2ccc(Br)cc2)CC1 ZINC000217554318 HH On-Demand Unstable HTR1B 24 53 COc1ccccc1N1CCN(C(=O)NCCc2ccc(Br)cc2)CC1 ZINC000217554318 HH On-Demand Unstable HTR2A 41 45 COc1ccccc1N1CCN(C(=O)NCCc2ccc(Br)cc2)CC1 ZINC000217554318 HH On-Demand Unstable ADRA1A 80 47 COc1ccccc1N1CCN(C(=O)NCCc2ccc(Br)cc2)CC1 ZINC000217554318 HH On-Demand Unstable ADRA1B 66 47 COc1ccccc1N1CCN(C(=O)NCCc2ccc(Br)cc2)CC1 ZINC000217554318 HH On-Demand Unstable DRD3 96 54 COc1ccccc1N1CCN(C(=O)NCCc2ccc(Br)cc2)CC1 ZINC000217554318 HH On-Demand Unstable PDGFRB 25 42 COc1ccccc1N1CCN(C(=O)NCCc2ccc(Br)cc2)CC1 ZINC000217554318 HH On-Demand Unstable HTR7 68 48 COc1ccccc1N1CCN(C(=O)NCCc2ccc(Br)cc2)CC1 ZINC000217554318 HH On-Demand Unstable TACR3 23 43 COc1ccccc1N1CCN(C(=O)NCCc2ccc(Br)cc2)CC1 ZINC000217554318 HH On-Demand Unstable HSP90AB1 0 44 COc1ccccc1N1CCN(C(=O)NCCc2ccc(Br)cc2)CC1 ZINC000217554318 HH On-Demand Unstable CXCR3 15 41 COc1ccccc1N1CCN(C(=O)NCCc2ccc(Br)cc2)CC1 ZINC000217554318 HH On-Demand Unstable AP2S1 0 51 COc1ccccc1N1CCN(C(=O)NCCc2ccc(Br)cc2)CC1 ZINC000217554318 HH On-Demand Unstable ALPHA-1A 0 48 COC(=O)CS[C@@H]1CCN(C(=O)c2nc3ccccc3s2)C1 ZINC000217554320 EE In-Stock Unstable PRSS3 0 42 COC(=O)CS[C@@H]1CCN(C(=O)c2nc3ccccc3s2)C1 ZINC000217554320 EE In-Stock Unstable TRY1_BOVIN 47 38 COC(=O)CS[C@@H]1CCN(C(=O)c2nc3ccccc3s2)C1 ZINC000217554320 EE In-Stock Unstable TPSAB1 21 42 COC(=O)CS[C@@H]1CCN(C(=O)c2nc3ccccc3s2)C1 ZINC000217554320 EE In-Stock Unstable TMPRSS6 48 32 O=S(=O)(Nc1cc(F)cc(Cl)c1)c1cccnc1Cl ZINC000217554340 DG For-Sale Anodyne SGK1 41 33 NCc1nnc2ccc(-c3cccc(Br)c3)nn12 ZINC000217554345 DE In-Stock Unstable MET 20 42 O=C1O[C@@]2(CCCN(C(=O)c3cccs3)C2)c2ccccc21 ZINC000217554347 DG For-Sale Unstable NPY5R 26 41 COC(=O)CS[C@H]1CCN(C(=O)c2nc3ccccc3s2)C1 ZINC000217554394 EE In-Stock Unstable PRSS3 0 42 COC(=O)CS[C@H]1CCN(C(=O)c2nc3ccccc3s2)C1 ZINC000217554394 EE In-Stock Unstable TRY1_BOVIN 47 38 COC(=O)CS[C@H]1CCN(C(=O)c2nc3ccccc3s2)C1 ZINC000217554394 EE In-Stock Unstable TPSAB1 21 42 COC(=O)CS[C@H]1CCN(C(=O)c2nc3ccccc3s2)C1 ZINC000217554394 EE In-Stock Unstable TMPRSS6 48 32 CC(C)CNS(=O)(=O)c1ccc(N[C@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217554399 GG In-Stock Unstable KCNA5 0 41 O=C1O[C@]2(CCCN(C(=O)c3cccs3)C2)c2ccccc21 ZINC000217554429 DG For-Sale Unstable NPY5R 26 41 C[C@@H](N)c1nnc2ccc(-c3ccc(Cl)cc3Cl)nn12 ZINC000217554471 DG In-Stock Unstable DPP4 26 41 C[C@@H](N)c1nnc2ccc(-c3ccc(Cl)cc3Cl)nn12 ZINC000217554471 DG In-Stock Unstable DPP8 43 33 C[C@@H](N)c1nnc2ccc(-c3ccc(Cl)cc3Cl)nn12 ZINC000217554471 DG In-Stock Unstable DPP9 42 33 CC(C)CNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217554503 GF In-Stock Unstable ADRB3 55 41 CC(C)CNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217554503 GF In-Stock Unstable TBXA2R 48 38 CC(C)CNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217554503 GF In-Stock Unstable SFRP1 15 45 Cn1c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c(O)c1CN1CCN(c2ccc(F)cc2)CC1 ZINC000217554505 KE In-Stock Unstable CHRNA4 38 54 COC(=O)CS[C@@H]1CCN(C(=O)c2ccc(C(=O)OC)cc2)C1 ZINC000217554507 ED In-Stock Unstable L3MBTL3 68 39 COC(=O)CS[C@@H]1CCN(C(=O)c2ccc(C(=O)OC)cc2)C1 ZINC000217554507 ED In-Stock Unstable GPR183 0 40 O=C1O[C@@]2(CCCN(C(=O)c3ccsc3)C2)c2ccccc21 ZINC000217554540 DG For-Sale Unstable NPY5R 24 41 C[C@H](N)c1nnc2ccc(-c3ccc(Cl)cc3Cl)nn12 ZINC000217554544 DG In-Stock Unstable DPP4 26 41 C[C@H](N)c1nnc2ccc(-c3ccc(Cl)cc3Cl)nn12 ZINC000217554544 DG In-Stock Unstable DPP8 43 33 C[C@H](N)c1nnc2ccc(-c3ccc(Cl)cc3Cl)nn12 ZINC000217554544 DG In-Stock Unstable DPP9 42 33 CC(C)CN(CC(C)C)C(=O)NCCc1ccc(Br)cc1 ZINC000217554565 FI For-Sale Unstable AMP1_PLAFQ 30 42 CC(C)CN(CC(C)C)C(=O)NCCc1ccc(Br)cc1 ZINC000217554565 FI For-Sale Unstable LIG1 0 42 C[C@H](C(=O)N1CCCC1)N1CCC[C@@H](CN)C1 ZINC000217554583 BC For-Sale Unstable DPP7 58 42 COC(=O)CS[C@H]1CCN(C(=O)c2ccc(C(=O)OC)cc2)C1 ZINC000217554591 ED In-Stock Unstable L3MBTL3 68 39 COC(=O)CS[C@H]1CCN(C(=O)c2ccc(C(=O)OC)cc2)C1 ZINC000217554591 ED In-Stock Unstable GPR183 0 40 COc1ccc(CCNc2ccc(S(=O)(=O)NCC(C)C)cc2C(=O)O)cc1 ZINC000217554622 HF In-Stock Unstable CA2 17 40 COc1ccc(CCNc2ccc(S(=O)(=O)NCC(C)C)cc2C(=O)O)cc1 ZINC000217554622 HF In-Stock Unstable ADRB2 30 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCC(C)C)cc2C(=O)O)cc1 ZINC000217554622 HF In-Stock Unstable ADRB1 43 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCC(C)C)cc2C(=O)O)cc1 ZINC000217554622 HF In-Stock Unstable ADRB3 51 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCC(C)C)cc2C(=O)O)cc1 ZINC000217554622 HF In-Stock Unstable TBXA2R 28 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCC(C)C)cc2C(=O)O)cc1 ZINC000217554622 HF In-Stock Unstable BMP1 105 38 COc1ccc(CCNc2ccc(S(=O)(=O)NCC(C)C)cc2C(=O)O)cc1 ZINC000217554622 HF In-Stock Unstable CA1 16 44 COc1ccc(CCNc2ccc(S(=O)(=O)NCC(C)C)cc2C(=O)O)cc1 ZINC000217554622 HF In-Stock Unstable MMP13 66 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCC(C)C)cc2C(=O)O)cc1 ZINC000217554622 HF In-Stock Unstable MMP2 43 40 COc1ccc(CCNc2ccc(S(=O)(=O)NCC(C)C)cc2C(=O)O)cc1 ZINC000217554622 HF In-Stock Unstable MMP3 48 40 COc1ccc(CCNc2ccc(S(=O)(=O)NCC(C)C)cc2C(=O)O)cc1 ZINC000217554622 HF In-Stock Unstable MMP8 31 40 COc1ccc(CCNc2ccc(S(=O)(=O)NCC(C)C)cc2C(=O)O)cc1 ZINC000217554622 HF In-Stock Unstable MMP14 19 40 COc1ccc(CCNc2ccc(S(=O)(=O)NCC(C)C)cc2C(=O)O)cc1 ZINC000217554622 HF In-Stock Unstable MMP9 56 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCC(C)C)cc2C(=O)O)cc1 ZINC000217554622 HF In-Stock Unstable MMP12 33 40 COc1ccc(CCNc2ccc(S(=O)(=O)NCC(C)C)cc2C(=O)O)cc1 ZINC000217554622 HF In-Stock Unstable PTGDR 23 42 COc1ccc(CCNc2ccc(S(=O)(=O)NCC(C)C)cc2C(=O)O)cc1 ZINC000217554622 HF In-Stock Unstable MMP7 33 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCC(C)C)cc2C(=O)O)cc1 ZINC000217554622 HF In-Stock Unstable IAP 0 45 COc1ccc(CCNc2ccc(S(=O)(=O)NCC(C)C)cc2C(=O)O)cc1 ZINC000217554622 HF In-Stock Unstable CA9 25 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCC(C)C)cc2C(=O)O)cc1 ZINC000217554622 HF In-Stock Unstable MMP1 56 39 COc1ccc(CCNc2ccc(S(=O)(=O)NCC(C)C)cc2C(=O)O)cc1 ZINC000217554622 HF In-Stock Unstable AKR1C3 30 44 COc1ccc(CCNc2ccc(S(=O)(=O)NCC(C)C)cc2C(=O)O)cc1 ZINC000217554622 HF In-Stock Unstable AKR1C2 50 37 O=C1O[C@]2(CCCN(C(=O)c3ccsc3)C2)c2ccccc21 ZINC000217554628 DG For-Sale Unstable NPY5R 24 41 C[C@@H](C(=O)N1CCCC1)N1CCC[C@@H](CN)C1 ZINC000217554651 BC For-Sale Unstable DPP7 58 42 COc1ccc(-c2ccc3nnc([C@@H](C)N)n3n2)cc1 ZINC000217554654 CD In-Stock Unstable PDE1A 22 40 COc1ccc(-c2ccc3nnc([C@@H](C)N)n3n2)cc1 ZINC000217554654 CD In-Stock Unstable MET 18 44 O=CN1CCN(C(=O)NCCc2ccc(Br)cc2)CC1 ZINC000217554679 ED For-Sale Unstable LIG1 0 40 COC(=O)CS[C@@H]1CCN(C(=O)c2ccc3nsnc3c2)C1 ZINC000217554718 ED In-Stock Unstable L3MBTL3 47 34 O=C1O[C@@]2(CCCN(C(=O)CC3CCCC3)C2)c2ccccc21 ZINC000217554738 DG For-Sale Unstable NPY5R 41 40 COc1ccc(CCNc2ccc(S(=O)(=O)NCC(C)C)cc2C(=O)O)cc1OC ZINC000217554743 IF In-Stock Unstable BDKRB1 0 40 COc1ccc(CCNc2ccc(S(=O)(=O)NCC(C)C)cc2C(=O)O)cc1OC ZINC000217554743 IF In-Stock Unstable IAP 0 47 COc1ccc(CCNc2ccc(S(=O)(=O)NCC(C)C)cc2C(=O)O)cc1OC ZINC000217554743 IF In-Stock Unstable SCMU_MYCTU 0 45 COc1ccc(-c2ccc3nnc([C@H](C)N)n3n2)cc1 ZINC000217554751 CD In-Stock Unstable PDE1A 22 40 COc1ccc(-c2ccc3nnc([C@H](C)N)n3n2)cc1 ZINC000217554751 CD In-Stock Unstable MET 18 44 C[C@@H](N[C@@H](c1ccccc1)C1CC1)C(=O)NC12CC3CC(CC(C3)C1)C2 ZINC000217554769 FI On-Demand Unstable CNR2 17 40 C[C@@H](N[C@@H](c1ccccc1)C1CC1)C(=O)NC12CC3CC(CC(C3)C1)C2 ZINC000217554769 FI On-Demand Unstable EPHX2 79 55 O=C(NCCc1ccc(Br)cc1)NC1CCCCCC1 ZINC000217554775 EI For-Sale Unstable CNR2 16 41 O=C(NCCc1ccc(Br)cc1)NC1CCCCCC1 ZINC000217554775 EI For-Sale Unstable EPHX2 33 74 O=C(NCCc1ccc(Br)cc1)NC1CCCCCC1 ZINC000217554775 EI For-Sale Unstable GPBAR1 0 42 O=C(NCCc1ccc(Br)cc1)NC1CCCCCC1 ZINC000217554775 EI For-Sale Unstable TRAR 18 40 COC(=O)CS[C@H]1CCN(C(=O)c2ccc3nsnc3c2)C1 ZINC000217554800 ED In-Stock Unstable L3MBTL3 47 34 O=C(O)C1C[C@@H]2CC[C@H](C1)N2Cc1cccnc1 ZINC000217554823 BD For-Sale Unstable KCNH2 35 42 O=C(O)C1C[C@@H]2CC[C@H](C1)N2Cc1cccnc1 ZINC000217554823 BD For-Sale Unstable TBXAS1 29 40 O=C(O)C1C[C@@H]2CC[C@H](C1)N2Cc1cccnc1 ZINC000217554823 BD For-Sale Unstable CHRNA7 41 38 O=C1O[C@]2(CCCN(C(=O)CC3CCCC3)C2)c2ccccc21 ZINC000217554824 DG For-Sale Unstable NPY5R 41 40 C[C@H](N[C@@H](c1ccccc1)C1CC1)C(=O)NC12CC3CC(CC(C3)C1)C2 ZINC000217554849 FI On-Demand Unstable CNR2 17 40 C[C@H](N[C@@H](c1ccccc1)C1CC1)C(=O)NC12CC3CC(CC(C3)C1)C2 ZINC000217554849 FI On-Demand Unstable EPHX2 79 55 COc1ccc(-c2ccc3nnc([C@@H](C)N)n3n2)cc1OC ZINC000217554857 CD In-Stock Unstable PRKDC 15 41 COc1ccc(-c2ccc3nnc([C@@H](C)N)n3n2)cc1OC ZINC000217554857 CD In-Stock Unstable PDE1A 22 41 COc1ccc(-c2ccc3nnc([C@@H](C)N)n3n2)cc1OC ZINC000217554857 CD In-Stock Unstable PDE4D 49 44 COc1ccc(-c2ccc3nnc([C@@H](C)N)n3n2)cc1OC ZINC000217554857 CD In-Stock Unstable PDE3B 15 41 COc1ccc(-c2ccc3nnc([C@@H](C)N)n3n2)cc1OC ZINC000217554857 CD In-Stock Unstable MET 20 52 Cc1ccc(C)c(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217554869 EI On-Demand Unstable RAF1 37 45 Cc1ccc(C)c(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217554869 EI On-Demand Unstable Q8MMZ8_EIMTE 26 41 COC(=O)CS[C@H]1CCN(C(=O)c2ccc(OC(C)C)cc2)C1 ZINC000217554922 EF In-Stock Unstable GRM3 15 41 COC(=O)CS[C@H]1CCN(C(=O)c2ccc(OC(C)C)cc2)C1 ZINC000217554922 EF In-Stock Unstable L3MBTL3 56 36 Cc1ccccc1C(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217554932 DG For-Sale Unstable NPY5R 30 42 C[C@@H](N[C@H](c1ccccc1)C1CC1)C(=O)NC12CC3CC(CC(C3)C1)C2 ZINC000217554934 FI On-Demand Unstable CNR2 17 40 C[C@@H](N[C@H](c1ccccc1)C1CC1)C(=O)NC12CC3CC(CC(C3)C1)C2 ZINC000217554934 FI On-Demand Unstable EPHX2 79 55 COc1ccc(-c2ccc3nnc([C@H](C)N)n3n2)cc1OC ZINC000217554952 CD In-Stock Unstable PRKDC 15 41 COc1ccc(-c2ccc3nnc([C@H](C)N)n3n2)cc1OC ZINC000217554952 CD In-Stock Unstable PDE1A 22 41 COc1ccc(-c2ccc3nnc([C@H](C)N)n3n2)cc1OC ZINC000217554952 CD In-Stock Unstable PDE4D 49 44 COc1ccc(-c2ccc3nnc([C@H](C)N)n3n2)cc1OC ZINC000217554952 CD In-Stock Unstable PDE3B 15 41 COc1ccc(-c2ccc3nnc([C@H](C)N)n3n2)cc1OC ZINC000217554952 CD In-Stock Unstable MET 20 52 CC(C)CNS(=O)(=O)c1ccc(NC[C@@H]2CCCO2)c(C(=O)O)c1 ZINC000217554962 FD In-Stock Unstable BDKRB1 0 42 O=C(NCCc1ccc(Br)cc1)Nc1cc(Cl)cc(Cl)c1 ZINC000217554982 GK For-Sale Unstable RAF1 34 42 O=C(NCCc1ccc(Br)cc1)Nc1cc(Cl)cc(Cl)c1 ZINC000217554982 GK For-Sale Unstable Q8MMZ8_EIMTE 22 42 O=C(NCCc1ccc(Br)cc1)Nc1cc(Cl)cc(Cl)c1 ZINC000217554982 GK For-Sale Unstable NCE103 26 42 COC(=O)CS[C@@H]1CCN(C(=O)c2ccc(OC(C)C)cc2)C1 ZINC000217555005 EF In-Stock Unstable GRM3 15 41 COC(=O)CS[C@@H]1CCN(C(=O)c2ccc(OC(C)C)cc2)C1 ZINC000217555005 EF In-Stock Unstable L3MBTL3 56 36 C[C@H](N[C@H](c1ccccc1)C1CC1)C(=O)NC12CC3CC(CC(C3)C1)C2 ZINC000217555021 FI On-Demand Unstable CNR2 17 40 C[C@H](N[C@H](c1ccccc1)C1CC1)C(=O)NC12CC3CC(CC(C3)C1)C2 ZINC000217555021 FI On-Demand Unstable EPHX2 79 55 Cc1ccccc1C(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217555022 DG For-Sale Unstable NPY5R 30 42 CC(C)CNS(=O)(=O)c1ccc(NC[C@H]2CCCO2)c(C(=O)O)c1 ZINC000217555038 FD In-Stock Unstable BDKRB1 0 42 COc1ccc(OC)c(-c2ccc3nnc([C@@H](C)N)n3n2)c1 ZINC000217555063 CD In-Stock Unstable LRRK2 30 44 CCOc1ccccc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217555077 FI On-Demand Unstable ACAT 0 44 O=C(O)C1C[C@@H]2CC[C@H](C1)N2Cc1ccncc1 ZINC000217555087 BD For-Sale Unstable KCNH2 27 40 COC(=O)CS[C@H]1CCN(C(=O)CCc2ccc(OC)cc2)C1 ZINC000217555109 EE In-Stock Unstable MMP13 29 40 COC(=O)CS[C@H]1CCN(C(=O)CCc2ccc(OC)cc2)C1 ZINC000217555109 EE In-Stock Unstable C3AR1 29 42 COC(=O)CS[C@H]1CCN(C(=O)CCc2ccc(OC)cc2)C1 ZINC000217555109 EE In-Stock Unstable MMP3 25 40 COC(=O)CS[C@H]1CCN(C(=O)CCc2ccc(OC)cc2)C1 ZINC000217555109 EE In-Stock Unstable MMP9 25 40 COC(=O)CS[C@H]1CCN(C(=O)CCc2ccc(OC)cc2)C1 ZINC000217555109 EE In-Stock Unstable MMP7 30 40 COC(=O)CS[C@H]1CCN(C(=O)CCc2ccc(OC)cc2)C1 ZINC000217555109 EE In-Stock Unstable MMP1 27 42 CN1CCC(c2[nH]nc(C(=O)O)c2Cl)CC1 ZINC000217555122 BD For-Sale Unstable HTR1F 42 32 CCCNC(=O)[C@@H](C)N1CCC[C@@H](CN)C1 ZINC000217555125 BC On-Demand Unstable HLA-DRB3 46 35 O=C1O[C@@]2(CCCN(C(=O)c3ccc(F)cc3)C2)c2ccccc21 ZINC000217555136 EG For-Sale Unstable NPY5R 36 48 CC(C)CNS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217555148 ED In-Stock Unstable KCNQ2 65 36 CC(C)CNS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217555148 ED In-Stock Unstable SLC6A9 23 43 CC(C)CNS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217555148 ED In-Stock Unstable SFRP1 82 36 CC(C)CNS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217555148 ED In-Stock Unstable WNT3 62 36 COc1ccc(OC)c(-c2ccc3nnc([C@H](C)N)n3n2)c1 ZINC000217555150 CD In-Stock Unstable LRRK2 30 44 Cc1cc(C)cc(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217555174 EI For-Sale Unstable RAF1 30 40 Cc1cc(C)cc(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217555174 EI For-Sale Unstable Q8MMZ8_EIMTE 0 40 Cc1cc(C)cc(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217555174 EI For-Sale Unstable NCE103 26 43 Cc1cc(C)cc(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217555174 EI For-Sale Unstable LIG1 0 40 Cc1cc(C)cc(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217555174 EI For-Sale Unstable P96878_MYCTU 18 41 COC(=O)CS[C@@H]1CCN(C(=O)CCc2ccc(OC)cc2)C1 ZINC000217555205 EE In-Stock Unstable MMP13 29 40 COC(=O)CS[C@@H]1CCN(C(=O)CCc2ccc(OC)cc2)C1 ZINC000217555205 EE In-Stock Unstable C3AR1 29 42 COC(=O)CS[C@@H]1CCN(C(=O)CCc2ccc(OC)cc2)C1 ZINC000217555205 EE In-Stock Unstable MMP3 25 40 COC(=O)CS[C@@H]1CCN(C(=O)CCc2ccc(OC)cc2)C1 ZINC000217555205 EE In-Stock Unstable MMP9 25 40 COC(=O)CS[C@@H]1CCN(C(=O)CCc2ccc(OC)cc2)C1 ZINC000217555205 EE In-Stock Unstable MMP7 30 40 COC(=O)CS[C@@H]1CCN(C(=O)CCc2ccc(OC)cc2)C1 ZINC000217555205 EE In-Stock Unstable MMP1 27 42 CCCNC(=O)[C@H](C)N1CCC[C@@H](CN)C1 ZINC000217555225 BC On-Demand Unstable HLA-DRB3 46 35 O=C1O[C@]2(CCCN(C(=O)c3ccc(F)cc3)C2)c2ccccc21 ZINC000217555228 EG For-Sale Unstable NPY5R 36 48 C[C@@H](N)c1nnc2ccc(-c3ccc(Br)cc3)nn12 ZINC000217555256 DF In-Stock Unstable PDE1A 21 42 CC(C)CNS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217555261 EE In-Stock Unstable KCNQ2 59 35 CC(C)CNS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217555261 EE In-Stock Unstable SLC6A9 22 45 CC(C)CNS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217555261 EE In-Stock Unstable SFRP1 76 36 CC(C)CNS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217555261 EE In-Stock Unstable WNT3 61 36 COc1cc(F)ccc1NC(=O)NC(=O)/C=C\C(=O)O ZINC000217555265 CD For-Sale Unstable PYGL 35 52 COc1ccc(OCCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217555282 GG On-Demand Unstable BMP1 32 40 COc1ccc(OCCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217555282 GG On-Demand Unstable MMP13 22 40 COc1ccc(OCCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217555282 GG On-Demand Unstable MTNR1A 79 43 COc1ccc(OCCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217555282 GG On-Demand Unstable MTNR1B 62 43 COc1ccc(OCCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217555282 GG On-Demand Unstable MMP9 22 41 COc1ccc(OCCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217555282 GG On-Demand Unstable CA9 23 46 COc1ccc(OCCNC(=O)NCCc2ccc(Br)cc2)cc1 ZINC000217555282 GG On-Demand Unstable MMP1 23 41 C[C@@H](N)c1ccc(Br)cc1N1CC[C@@H](c2ccccc2)C1 ZINC000217555309 EI For-Sale Unstable SLC18A3 22 40 C[C@H](N)c1nnc2ccc(-c3ccc(Br)cc3)nn12 ZINC000217555338 DF In-Stock Unstable PDE1A 21 42 O=C1O[C@@]2(CCCN(C(=O)Cc3cccs3)C2)c2ccccc21 ZINC000217555342 EF For-Sale Unstable NPY5R 23 40 CC(C)CNS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1 ZINC000217555379 ED In-Stock Unstable SLC6A9 24 48 CC(=O)N(CCN)C(=O)NCCc1ccc(Br)cc1 ZINC000217555398 ED For-Sale Unstable LIG1 0 40 O=C1O[C@]2(CCCN(C(=O)Cc3cccs3)C2)c2ccccc21 ZINC000217555403 EF For-Sale Unstable NPY5R 23 40 C[C@H](N)c1ccc(Br)cc1N1CC[C@@H](c2ccccc2)C1 ZINC000217555411 EI For-Sale Unstable SLC18A3 22 40 C[C@@H](N)c1nnc2ccc(-c3cccc(Br)c3)nn12 ZINC000217555450 DF In-Stock Unstable PDE1A 23 42 C[C@@H](N)c1nnc2ccc(-c3cccc(Br)c3)nn12 ZINC000217555450 DF In-Stock Unstable MET 19 44 O=c1cccc2n1C[C@H]1C[C@@H]2CN(S(=O)(=O)c2cccc([N+](=O)[O-])c2)C1 ZINC000217555467 GD On-Demand Unstable CHRNA4 29 48 CCOCCCNc1ccc(S(=O)(=O)NCC(C)C)cc1C(=O)O ZINC000217555473 FE In-Stock Unstable CASP3 0 40 COC(=O)CS[C@@H]1CCN(C(=O)CSCc2ccccc2)C1 ZINC000217555478 EE In-Stock Unstable LTA4H 24 41 C[C@@H](N)c1cc(Br)ccc1N1CC[C@@H](c2ccccc2)C1 ZINC000217555494 EI For-Sale Unstable SLC18A3 21 40 N#Cc1ccc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217555514 EF For-Sale Unstable NPY5R 23 40 Cn1c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c(O)c1CN1CCN(Cc2ccccc2)CC1 ZINC000217555525 KE In-Stock Unstable CHRNA4 41 64 C[C@H](N)c1nnc2ccc(-c3cccc(Br)c3)nn12 ZINC000217555530 DF In-Stock Unstable PDE1A 23 42 C[C@H](N)c1nnc2ccc(-c3cccc(Br)c3)nn12 ZINC000217555530 DF In-Stock Unstable MET 19 44 COc1cc(CN2CC[C@@H](N)C2)ccc1OCC=C(C)C ZINC000217555555 CF In-Stock Unstable SSTR5 63 40 NNC(=O)c1ccc2c(c1)CC(=O)N2 ZINC000217555563 AB For-Sale Unstable HDAC9 25 48 COC(=O)CS[C@H]1CCN(C(=O)CSCc2ccccc2)C1 ZINC000217555565 EE In-Stock Unstable LTA4H 24 41 CC(C)CNS(=O)(=O)c1ccc(NCCCOC(C)C)c(C(=O)O)c1 ZINC000217555578 FF In-Stock Unstable CASP3 0 40 CC(C)CNS(=O)(=O)c1ccc(NCCCOC(C)C)c(C(=O)O)c1 ZINC000217555578 FF In-Stock Unstable BDKRB1 0 42 C[C@H](N)c1cc(Br)ccc1N1CC[C@@H](c2ccccc2)C1 ZINC000217555591 EI For-Sale Unstable SLC18A3 21 40 N#Cc1ccc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217555607 EF For-Sale Unstable NPY5R 23 40 O=C(NCCc1ccc(Br)cc1)Nc1cccc2cccnc12 ZINC000217555622 FI On-Demand Unstable TRPV1 15 57 O=C(NCCc1ccc(Br)cc1)Nc1cccc2cccnc12 ZINC000217555622 FI On-Demand Unstable EGLN1 0 47 COc1cc(CN2CC[C@H](N)C2)ccc1OCC=C(C)C ZINC000217555652 CF In-Stock Unstable SSTR5 63 40 COC(=O)CS[C@@H]1CCN(C(=O)CCSc2ccccc2)C1 ZINC000217555672 EF In-Stock Unstable FAS 24 41 CCCCCNc1ccc(S(=O)(=O)NCC(C)C)cc1C(=O)O ZINC000217555677 EF In-Stock Unstable CASP3 16 43 O=C(CN[C@@H](c1ccccc1)C1CC1)N1CCN(c2ccc(F)cc2)CC1 ZINC000217555690 FG On-Demand Unstable HTR7 18 40 O=C1O[C@@]2(CCCN(C(=O)CCc3ccccc3)C2)c2ccccc21 ZINC000217555706 EG For-Sale Unstable NPY5R 28 42 C[C@@H]1Cc2ccccc2N1C(=O)NCCc1ccc(Br)cc1 ZINC000217555739 FI On-Demand Unstable DRD4 28 45 C[C@@H]1Cc2ccccc2N1C(=O)NCCc1ccc(Br)cc1 ZINC000217555739 FI On-Demand Unstable TPP2 58 38 COC(=O)CS[C@H]1CCN(C(=O)CCSc2ccccc2)C1 ZINC000217555759 EF In-Stock Unstable FAS 24 41 O=C(CN[C@H](c1ccccc1)C1CC1)N1CCN(c2ccc(F)cc2)CC1 ZINC000217555771 FG On-Demand Unstable HTR7 18 40 CC(C)CCNc1ccc(S(=O)(=O)NCC(C)C)cc1C(=O)O ZINC000217555793 EF In-Stock Unstable CASP3 17 43 O=C1O[C@]2(CCCN(C(=O)CCc3ccccc3)C2)c2ccccc21 ZINC000217555803 EG For-Sale Unstable NPY5R 28 42 C[C@H]1Cc2ccccc2N1C(=O)NCCc1ccc(Br)cc1 ZINC000217555828 FI On-Demand Unstable DRD4 28 45 C[C@H]1Cc2ccccc2N1C(=O)NCCc1ccc(Br)cc1 ZINC000217555828 FI On-Demand Unstable TPP2 58 38 COC(=O)CS[C@@H]1CCN(C(=O)COc2ccc(Cl)cc2)C1 ZINC000217555874 EE In-Stock Unstable SLC6A1 29 42 COC(=O)CS[C@@H]1CCN(C(=O)COc2ccc(Cl)cc2)C1 ZINC000217555874 EE In-Stock Unstable COLA 25 44 COC(=O)CS[C@@H]1CCN(C(=O)COc2ccc(Cl)cc2)C1 ZINC000217555874 EE In-Stock Unstable GPR183 0 46 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NCC(C)C)cc1C(=O)O ZINC000217555913 EF In-Stock Unstable CASP3 0 40 Cc1cccc(CC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217555916 EG For-Sale Unstable NPY5R 26 40 COC(=O)CS[C@H]1CCN(C(=O)COc2ccc(Cl)cc2)C1 ZINC000217555974 EE In-Stock Unstable SLC6A1 29 42 COC(=O)CS[C@H]1CCN(C(=O)COc2ccc(Cl)cc2)C1 ZINC000217555974 EE In-Stock Unstable COLA 25 44 COC(=O)CS[C@H]1CCN(C(=O)COc2ccc(Cl)cc2)C1 ZINC000217555974 EE In-Stock Unstable GPR183 0 46 CCC[C@H](C)Nc1ccc(S(=O)(=O)NCC(C)C)cc1C(=O)O ZINC000217555989 EF In-Stock Unstable CASP3 0 40 Cc1cccc(CC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217555998 EG For-Sale Unstable NPY5R 26 40 Cc1ccc2nc(-c3ccc(NC(=O)NCCc4ccc(Br)cc4)cc3)sc2c1 ZINC000217556063 JK For-Sale Unstable LDHA 44 46 Cc1ccc2nc(-c3ccc(NC(=O)NCCc4ccc(Br)cc4)cc3)sc2c1 ZINC000217556063 JK For-Sale Unstable APP 27 53 Cc1ccc2nc(-c3ccc(NC(=O)NCCc4ccc(Br)cc4)cc3)sc2c1 ZINC000217556063 JK For-Sale Unstable PRMT3 63 35 COC(=O)CS[C@H]1CCN(C(=O)c2cc(Cl)ccc2OC)C1 ZINC000217556068 EE In-Stock Unstable RBP4 26 42 CCCCCNC(=O)[C@@H](C)N1CCC[C@@H](CN)C1 ZINC000217556092 CD On-Demand Unstable TPP2 42 44 COc1ccc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217556106 EF For-Sale Unstable GRM3 15 51 COc1ccc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217556106 EF For-Sale Unstable NPY5R 28 44 COC(=O)CS[C@@H]1CCN(C(=O)c2cc(Cl)ccc2OC)C1 ZINC000217556154 EE In-Stock Unstable RBP4 26 42 CCCCCNC(=O)[C@H](C)N1CCC[C@@H](CN)C1 ZINC000217556173 CD On-Demand Unstable TPP2 42 44 COc1ccc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217556175 EF For-Sale Unstable GRM3 15 51 COc1ccc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217556175 EF For-Sale Unstable NPY5R 28 44 COc1ccc(-c2ccc3nnc([C@@H]4CCCN4)n3n2)cc1 ZINC000217556219 CE In-Stock Unstable LRRK2 27 40 COC(=O)CS[C@@H]1CCN(C(=O)c2ccc(C(F)(F)F)cc2)C1 ZINC000217556250 EF In-Stock Unstable MCHR1 28 41 COC(=O)CS[C@@H]1CCN(C(=O)c2ccc(C(F)(F)F)cc2)C1 ZINC000217556250 EF In-Stock Unstable L3MBTL3 57 36 CCCCNC(=O)[C@@H](C)N1CCC[C@@H](CN)C1 ZINC000217556265 BC On-Demand Unstable TPP2 42 44 CCCNc1ccc(S(=O)(=O)N[C@@H](C)CC)cc1C(=O)O ZINC000217556281 DE In-Stock Unstable LEF 49 37 COc1ccc(-c2ccc3nnc([C@H]4CCCN4)n3n2)cc1 ZINC000217556283 CE In-Stock Unstable LRRK2 27 40 O=C1O[C@@]2(CCCN(C(=O)COc3ccccc3)C2)c2ccccc21 ZINC000217556288 EF In-Stock Unstable COLA 118 37 O=C1O[C@@]2(CCCN(C(=O)COc3ccccc3)C2)c2ccccc21 ZINC000217556288 EF In-Stock Unstable CPT1A 99 37 O=C1O[C@@]2(CCCN(C(=O)COc3ccccc3)C2)c2ccccc21 ZINC000217556288 EF In-Stock Unstable CPT2 48 37 O=C1O[C@@]2(CCCN(C(=O)COc3ccccc3)C2)c2ccccc21 ZINC000217556288 EF In-Stock Unstable NPY5R 37 44 O=C(NCCc1ccc(Br)cc1)Nc1ccc(I)cc1 ZINC000217556291 II For-Sale Unstable CA1 15 52 O=C(NCCc1ccc(Br)cc1)Nc1ccc(I)cc1 ZINC000217556291 II For-Sale Unstable CA12 15 52 O=C(NCCc1ccc(Br)cc1)Nc1ccc(I)cc1 ZINC000217556291 II For-Sale Unstable CA9 15 52 O=C(NCCc1ccc(Br)cc1)Nc1ccc(I)cc1 ZINC000217556291 II For-Sale Unstable NCE103 28 52 O=C(NCCc1ccc(Br)cc1)Nc1ccc(I)cc1 ZINC000217556291 II For-Sale Unstable LIG1 0 40 O=C(NCCc1ccc(Br)cc1)Nc1ccc(I)cc1 ZINC000217556291 II For-Sale Unstable P96878_MYCTU 15 41 O=C(/C=C\c1ccccc1F)N[C@@H]1CC[C@H](C(=O)O)C1 ZINC000217556293 CE For-Sale Unstable KCNQ2 41 38 COc1c([C@@H]2CCCNC2)ccc(F)c1Cl ZINC000217556298 BF For-Sale Unstable SLC6A2 19 40 Cc1cc(=O)c(O)c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)n1C ZINC000217556300 ED In-Stock Unstable CHRNA4 35 56 COC(=O)CS[C@H]1CCN(C(=O)c2ccc(C(F)(F)F)cc2)C1 ZINC000217556343 EF In-Stock Unstable MCHR1 28 41 COC(=O)CS[C@H]1CCN(C(=O)c2ccc(C(F)(F)F)cc2)C1 ZINC000217556343 EF In-Stock Unstable L3MBTL3 57 36 CCCCNC(=O)[C@H](C)N1CCC[C@@H](CN)C1 ZINC000217556347 BC On-Demand Unstable TPP2 42 44 CCCNc1ccc(S(=O)(=O)N[C@H](C)CC)cc1C(=O)O ZINC000217556367 DE In-Stock Unstable LEF 49 37 CNc1nc(C(=O)N2CCCC[C@@]2(C)C(=O)O)cs1 ZINC000217556374 CD In-Stock Unstable TRPC6 65 38 CNc1nc(C(=O)N2CCCC[C@@]2(C)C(=O)O)cs1 ZINC000217556374 CD In-Stock Unstable TRPC3 50 38 O=C1O[C@]2(CCCN(C(=O)COc3ccccc3)C2)c2ccccc21 ZINC000217556375 EF In-Stock Unstable COLA 118 37 O=C1O[C@]2(CCCN(C(=O)COc3ccccc3)C2)c2ccccc21 ZINC000217556375 EF In-Stock Unstable CPT1A 99 37 O=C1O[C@]2(CCCN(C(=O)COc3ccccc3)C2)c2ccccc21 ZINC000217556375 EF In-Stock Unstable CPT2 48 37 O=C1O[C@]2(CCCN(C(=O)COc3ccccc3)C2)c2ccccc21 ZINC000217556375 EF In-Stock Unstable NPY5R 37 44 COc1c([C@H]2CCCNC2)ccc(F)c1Cl ZINC000217556376 BF For-Sale Unstable SLC6A2 19 40 O=C(NCCc1ccc(Br)cc1)NCCc1c[nH]c2ccccc12 ZINC000217556388 GI On-Demand Unstable HTR1A 0 44 O=C(NCCc1ccc(Br)cc1)NCCc1c[nH]c2ccccc12 ZINC000217556388 GI On-Demand Unstable HTR1D 28 44 O=C(NCCc1ccc(Br)cc1)NCCc1c[nH]c2ccccc12 ZINC000217556388 GI On-Demand Unstable EDNRB 0 46 O=C(NCCc1ccc(Br)cc1)NCCc1c[nH]c2ccccc12 ZINC000217556388 GI On-Demand Unstable TACR1 15 46 O=C(NCCc1ccc(Br)cc1)NCCc1c[nH]c2ccccc12 ZINC000217556388 GI On-Demand Unstable MC4R 50 53 O=C(NCCc1ccc(Br)cc1)NCCc1c[nH]c2ccccc12 ZINC000217556388 GI On-Demand Unstable TRPV1 0 53 O=C(NCCc1ccc(Br)cc1)NCCc1c[nH]c2ccccc12 ZINC000217556388 GI On-Demand Unstable CCKAR 53 48 O=C(NCCc1ccc(Br)cc1)NCCc1c[nH]c2ccccc12 ZINC000217556388 GI On-Demand Unstable CTSL 0 42 O=C(NCCc1ccc(Br)cc1)NCCc1c[nH]c2ccccc12 ZINC000217556388 GI On-Demand Unstable BCHE 17 42 O=C(NCCc1ccc(Br)cc1)NCCc1c[nH]c2ccccc12 ZINC000217556388 GI On-Demand Unstable MPO 57 36 O=C(NCCc1ccc(Br)cc1)NCCc1c[nH]c2ccccc12 ZINC000217556388 GI On-Demand Unstable BRS3 51 54 O=C(NCCc1ccc(Br)cc1)NCCc1c[nH]c2ccccc12 ZINC000217556388 GI On-Demand Unstable NMBR 47 47 O=C(NCCc1ccc(Br)cc1)NCCc1c[nH]c2ccccc12 ZINC000217556388 GI On-Demand Unstable MC3R 50 38 O=C(NCCc1ccc(Br)cc1)NCCc1c[nH]c2ccccc12 ZINC000217556388 GI On-Demand Unstable MC5R 40 42 O=C(NCCc1ccc(Br)cc1)NCCc1c[nH]c2ccccc12 ZINC000217556388 GI On-Demand Unstable CA5B 17 40 O=C(NCCc1ccc(Br)cc1)NCCc1c[nH]c2ccccc12 ZINC000217556388 GI On-Demand Unstable CA5A 15 40 O=C(NCCc1ccc(Br)cc1)NCCc1c[nH]c2ccccc12 ZINC000217556388 GI On-Demand Unstable MTNR1A 15 53 O=C(NCCc1ccc(Br)cc1)NCCc1c[nH]c2ccccc12 ZINC000217556388 GI On-Demand Unstable MMP2 22 46 O=C(NCCc1ccc(Br)cc1)NCCc1c[nH]c2ccccc12 ZINC000217556388 GI On-Demand Unstable MMP8 30 46 O=C(NCCc1ccc(Br)cc1)NCCc1c[nH]c2ccccc12 ZINC000217556388 GI On-Demand Unstable MMP14 55 38 O=C(NCCc1ccc(Br)cc1)NCCc1c[nH]c2ccccc12 ZINC000217556388 GI On-Demand Unstable ECE1 37 48 O=C(NCCc1ccc(Br)cc1)NCCc1c[nH]c2ccccc12 ZINC000217556388 GI On-Demand Unstable MMP11 46 32 O=C(NCCc1ccc(Br)cc1)NCCc1c[nH]c2ccccc12 ZINC000217556388 GI On-Demand Unstable CCKBR 47 51 O=C(NCCc1ccc(Br)cc1)NCCc1c[nH]c2ccccc12 ZINC000217556388 GI On-Demand Unstable GHSR 53 43 O=C(NCCc1ccc(Br)cc1)NCCc1c[nH]c2ccccc12 ZINC000217556388 GI On-Demand Unstable ALOX15 18 47 O=C(NCCc1ccc(Br)cc1)NCCc1c[nH]c2ccccc12 ZINC000217556388 GI On-Demand Unstable MMP9 21 46 O=C(NCCc1ccc(Br)cc1)NCCc1c[nH]c2ccccc12 ZINC000217556388 GI On-Demand Unstable HDAC9 20 42 O=C(NCCc1ccc(Br)cc1)NCCc1c[nH]c2ccccc12 ZINC000217556388 GI On-Demand Unstable MC1R 57 39 O=C(NCCc1ccc(Br)cc1)NCCc1c[nH]c2ccccc12 ZINC000217556388 GI On-Demand Unstable HDAC7 21 42 O=C(NCCc1ccc(Br)cc1)NCCc1c[nH]c2ccccc12 ZINC000217556388 GI On-Demand Unstable SLC15A2 0 40 O=C(NCCc1ccc(Br)cc1)NCCc1c[nH]c2ccccc12 ZINC000217556388 GI On-Demand Unstable ABCG2 26 42 COc1ccc(-c2ccc3nnc([C@@H]4CCCN4)n3n2)cc1OC ZINC000217556405 EE In-Stock Unstable PDE4D 51 43 COc1ccc(-c2ccc3nnc([C@@H]4CCCN4)n3n2)cc1OC ZINC000217556405 EE In-Stock Unstable LRRK2 26 41 COC(=O)CS[C@@H]1CCN(C(=O)c2ccccc2C(F)(F)F)C1 ZINC000217556457 EF In-Stock Unstable P2RX7 41 35 COC(=O)CS[C@@H]1CCN(C(=O)c2ccccc2C(F)(F)F)C1 ZINC000217556457 EF In-Stock Unstable RBP4 78 39 COC(=O)CS[C@@H]1CCN(C(=O)c2ccccc2C(F)(F)F)C1 ZINC000217556457 EF In-Stock Unstable SCD1 24 41 COC(=O)CS[C@@H]1CCN(C(=O)c2ccccc2C(F)(F)F)C1 ZINC000217556457 EF In-Stock Unstable SFRP1 68 36 COC(=O)CS[C@@H]1CCN(C(=O)c2ccccc2C(F)(F)F)C1 ZINC000217556457 EF In-Stock Unstable SCD 29 41 COC(=O)CS[C@@H]1CCN(C(=O)c2ccccc2C(F)(F)F)C1 ZINC000217556457 EF In-Stock Unstable WNT3 47 32 CNc1nc(C(=O)N2CCCC[C@]2(C)C(=O)O)cs1 ZINC000217556461 CD In-Stock Unstable TRPC6 65 38 CNc1nc(C(=O)N2CCCC[C@]2(C)C(=O)O)cs1 ZINC000217556461 CD In-Stock Unstable TRPC3 50 38 CC[C@@H](C)NS(=O)(=O)c1ccc(NC(C)C)c(C(=O)O)c1 ZINC000217556477 DE In-Stock Unstable MMP12 47 37 CC[C@@H](C)NS(=O)(=O)c1ccc(NC(C)C)c(C(=O)O)c1 ZINC000217556477 DE In-Stock Unstable LEF 50 39 COc1ccc(-c2ccc3nnc([C@H]4CCCN4)n3n2)cc1OC ZINC000217556482 EE In-Stock Unstable PDE4D 51 43 COc1ccc(-c2ccc3nnc([C@H]4CCCN4)n3n2)cc1OC ZINC000217556482 EE In-Stock Unstable LRRK2 26 41 COc1c(C2CCNCC2)ccc(F)c1Cl ZINC000217556491 BF For-Sale Unstable SLC6A2 20 40 COc1ccccc1C(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217556492 EF For-Sale Unstable NPY5R 27 49 COC(=O)CS[C@H]1CCN(C(=O)c2ccccc2C(F)(F)F)C1 ZINC000217556545 EF In-Stock Unstable P2RX7 41 35 COC(=O)CS[C@H]1CCN(C(=O)c2ccccc2C(F)(F)F)C1 ZINC000217556545 EF In-Stock Unstable RBP4 78 39 COC(=O)CS[C@H]1CCN(C(=O)c2ccccc2C(F)(F)F)C1 ZINC000217556545 EF In-Stock Unstable SCD1 24 41 COC(=O)CS[C@H]1CCN(C(=O)c2ccccc2C(F)(F)F)C1 ZINC000217556545 EF In-Stock Unstable SFRP1 68 36 COC(=O)CS[C@H]1CCN(C(=O)c2ccccc2C(F)(F)F)C1 ZINC000217556545 EF In-Stock Unstable SCD 29 41 COC(=O)CS[C@H]1CCN(C(=O)c2ccccc2C(F)(F)F)C1 ZINC000217556545 EF In-Stock Unstable WNT3 47 32 CC[C@H](C)NS(=O)(=O)c1ccc(NC(C)C)c(C(=O)O)c1 ZINC000217556563 DE In-Stock Unstable MMP12 47 37 CC[C@H](C)NS(=O)(=O)c1ccc(NC(C)C)c(C(=O)O)c1 ZINC000217556563 DE In-Stock Unstable LEF 50 39 Cn1c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c(O)c1CN1CCC(Cc2ccccc2)CC1 ZINC000217556570 KG In-Stock Unstable CHRNA4 29 54 COc1ccccc1C(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217556573 EF For-Sale Unstable NPY5R 27 49 COc1ccc(OC)c(-c2ccc3nnc([C@@H]4CCCN4)n3n2)c1 ZINC000217556599 EE In-Stock Unstable LRRK2 24 42 C[C@H](C(N)=O)N1CCC[C@@H](CN)C1 ZINC000217556663 AB On-Demand Unstable XPNPEP1 53 30 C[C@H](C(N)=O)N1CCC[C@@H](CN)C1 ZINC000217556663 AB On-Demand Unstable XPNPEP2 53 30 CCCCNc1ccc(S(=O)(=O)N[C@@H](C)CC)cc1C(=O)O ZINC000217556678 EF In-Stock Unstable LEF 45 38 COc1nn(C)cc1C(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217556684 ED For-Sale Unstable NPY5R 26 41 COc1ccc(OC)c(-c2ccc3nnc([C@H]4CCCN4)n3n2)c1 ZINC000217556694 EE In-Stock Unstable LRRK2 24 42 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Cl)cc1C(F)(F)F ZINC000217556732 HK For-Sale Unstable TRPV1 15 49 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Cl)cc1C(F)(F)F ZINC000217556732 HK For-Sale Unstable RAF1 40 41 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Cl)cc1C(F)(F)F ZINC000217556732 HK For-Sale Unstable Q8MMZ8_EIMTE 29 41 C[C@@H](C(N)=O)N1CCC[C@@H](CN)C1 ZINC000217556747 AB On-Demand Unstable XPNPEP1 53 30 C[C@@H](C(N)=O)N1CCC[C@@H](CN)C1 ZINC000217556747 AB On-Demand Unstable XPNPEP2 53 30 CCCCNc1ccc(S(=O)(=O)N[C@H](C)CC)cc1C(=O)O ZINC000217556756 EF In-Stock Unstable LEF 45 38 COc1nn(C)cc1C(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217556774 ED For-Sale Unstable NPY5R 26 41 CCN(CC)C(=O)[C@@H](N[C@@H](c1ccccc1)C1CC1)c1ccccc1 ZINC000217556782 EI On-Demand Unstable NPY2R 45 39 COc1cccc(CNc2cnn([C@@]34C[C@@H]5C[C@@H](C[C@@H](C5)C3)[C@H]4C(=O)O)c(=O)c2Cl)c1 ZINC000217556835 IH In-Stock Unstable ROCK2 41 39 Cc1cc(C)c(NC(=O)NCCc2ccc(Br)cc2)c(Cl)c1 ZINC000217556854 GK On-Demand Unstable RAF1 24 41 Cc1cc(C)c(NC(=O)NCCc2ccc(Br)cc2)c(Cl)c1 ZINC000217556854 GK On-Demand Unstable Q8MMZ8_EIMTE 0 41 CCN(CC)C(=O)[C@H](N[C@@H](c1ccccc1)C1CC1)c1ccccc1 ZINC000217556878 EI On-Demand Unstable NPY2R 45 39 CC[C@@H](C)NS(=O)(=O)c1ccc(NCC(C)C)c(C(=O)O)c1 ZINC000217556888 EF In-Stock Unstable MTNN 61 33 CC[C@@H](C)NS(=O)(=O)c1ccc(NCC(C)C)c(C(=O)O)c1 ZINC000217556888 EF In-Stock Unstable LEF 45 37 CCOc1cccc(NC(=O)NC(=O)/C=C\C(=O)O)c1 ZINC000217556931 CD For-Sale Unstable PPIA 35 41 CCOc1cccc(NC(=O)NC(=O)/C=C\C(=O)O)c1 ZINC000217556931 CD For-Sale Unstable CCKAR 22 45 CCOc1cccc(NC(=O)NC(=O)/C=C\C(=O)O)c1 ZINC000217556931 CD For-Sale Unstable LPAR2 15 52 CCOc1cccc(NC(=O)NC(=O)/C=C\C(=O)O)c1 ZINC000217556931 CD For-Sale Unstable CCKBR 16 45 CCOc1cccc(NC(=O)NC(=O)/C=C\C(=O)O)c1 ZINC000217556931 CD For-Sale Unstable EPHX2 24 43 CCOc1cccc(NC(=O)NC(=O)/C=C\C(=O)O)c1 ZINC000217556931 CD For-Sale Unstable TAAR1 19 41 CCOc1cccc(NC(=O)NC(=O)/C=C\C(=O)O)c1 ZINC000217556931 CD For-Sale Unstable KCNK3 69 41 CCOc1cccc(NC(=O)NC(=O)/C=C\C(=O)O)c1 ZINC000217556931 CD For-Sale Unstable KCNK9 64 41 CCOc1cccc(NC(=O)NC(=O)/C=C\C(=O)O)c1 ZINC000217556931 CD For-Sale Unstable PDS 64 37 CCN(CC)C(=O)[C@@H](N[C@H](c1ccccc1)C1CC1)c1ccccc1 ZINC000217556952 EI On-Demand Unstable NPY2R 45 39 CC[C@H](C)NS(=O)(=O)c1ccc(NCC(C)C)c(C(=O)O)c1 ZINC000217556962 EF In-Stock Unstable MTNN 61 33 CC[C@H](C)NS(=O)(=O)c1ccc(NCC(C)C)c(C(=O)O)c1 ZINC000217556962 EF In-Stock Unstable LEF 45 37 COc1cc(NC(=O)NCCc2ccc(Br)cc2)c(OC)cc1Cl ZINC000217556967 HI On-Demand Unstable TRPV1 0 41 COc1cc(NC(=O)NCCc2ccc(Br)cc2)c(OC)cc1Cl ZINC000217556967 HI On-Demand Unstable RAF1 39 52 COc1cc(NC(=O)NCCc2ccc(Br)cc2)c(OC)cc1Cl ZINC000217556967 HI On-Demand Unstable Q8MMZ8_EIMTE 28 52 COc1cc(NC(=O)NCCc2ccc(Br)cc2)c(OC)cc1Cl ZINC000217556967 HI On-Demand Unstable NCE103 25 42 COc1cc(NC(=O)NCCc2ccc(Br)cc2)c(OC)cc1Cl ZINC000217556967 HI On-Demand Unstable CAN2 0 42 C[C@@H](CNCc1ccc2c(c1)NC(=O)CO2)N(C)C1CC1 ZINC000217557004 CD On-Demand Unstable NR3C2 26 41 CCN(CC)C(=O)[C@H](N[C@H](c1ccccc1)C1CC1)c1ccccc1 ZINC000217557019 EI On-Demand Unstable NPY2R 45 39 O=C(NCCc1ccc(Br)cc1)Nc1c(Cl)cccc1Cl ZINC000217557078 GK For-Sale Unstable NCE103 24 40 O=C(NCCc1ccc(Br)cc1)Nc1c(Cl)cccc1Cl ZINC000217557078 GK For-Sale Unstable LIG1 0 42 O=C(NCCc1ccc(Br)cc1)Nc1c(Cl)cccc1Cl ZINC000217557078 GK For-Sale Unstable ACAT 0 49 O=C(NCCc1ccc(Br)cc1)Nc1c(Cl)cccc1Cl ZINC000217557078 GK For-Sale Unstable CAN2 0 40 O=C1O[C@@]2(CCCN(C(=O)c3ccc(Cl)cc3)C2)c2ccccc21 ZINC000217557079 EH For-Sale Unstable NPY5R 28 48 C[C@H](CNCc1ccc2c(c1)NC(=O)CO2)N(C)C1CC1 ZINC000217557082 CD On-Demand Unstable NR3C2 26 41 CC[C@H](C)NS(=O)(=O)c1ccc(N[C@H](C)CC)c(C(=O)O)c1 ZINC000217557089 EF In-Stock Unstable MMP12 48 38 CC[C@H](C)NS(=O)(=O)c1ccc(N[C@H](C)CC)c(C(=O)O)c1 ZINC000217557089 EF In-Stock Unstable LEF 54 39 O=C([C@@H](N[C@@H](c1ccccc1)C1CC1)c1ccccc1)N1CCCCC1 ZINC000217557132 EI On-Demand Unstable MTTP 27 44 O=C([C@@H](N[C@@H](c1ccccc1)C1CC1)c1ccccc1)N1CCCCC1 ZINC000217557132 EI On-Demand Unstable DPP7 60 40 O=C1O[C@]2(CCCN(C(=O)c3ccc(Cl)cc3)C2)c2ccccc21 ZINC000217557166 EH For-Sale Unstable NPY5R 28 48 CC[C@H](C)Nc1ccc(S(=O)(=O)N[C@@H](C)CC)cc1C(=O)O ZINC000217557169 EF In-Stock Unstable MMP12 48 38 CC[C@H](C)Nc1ccc(S(=O)(=O)N[C@@H](C)CC)cc1C(=O)O ZINC000217557169 EF In-Stock Unstable LEF 54 39 Cc1cccc(N2CCN(C(=O)NCCc3ccc(Br)cc3)CC2)c1C ZINC000217557181 HI For-Sale Unstable HTR2A 23 41 Cc1cccc(N2CCN(C(=O)NCCc3ccc(Br)cc3)CC2)c1C ZINC000217557181 HI For-Sale Unstable HTR2C 28 41 O=C([C@H](N[C@@H](c1ccccc1)C1CC1)c1ccccc1)N1CCCCC1 ZINC000217557208 EI On-Demand Unstable MTTP 27 44 O=C([C@H](N[C@@H](c1ccccc1)C1CC1)c1ccccc1)N1CCCCC1 ZINC000217557208 EI On-Demand Unstable DPP7 60 40 CC[C@@H](C)Nc1ccc(S(=O)(=O)N[C@H](C)CC)cc1C(=O)O ZINC000217557260 EF In-Stock Unstable MMP12 48 38 CC[C@@H](C)Nc1ccc(S(=O)(=O)N[C@H](C)CC)cc1C(=O)O ZINC000217557260 EF In-Stock Unstable LEF 54 39 COC(=O)CS[C@@H]1CCN(C(=O)CCS(=O)(=O)c2ccccc2)C1 ZINC000217557265 FD In-Stock Unstable CCR8 42 34 O=C(/C=C\c1ccc(Cl)c(Cl)c1)N[C@@H]1CC[C@H](C(=O)O)C1 ZINC000217557270 EG For-Sale Unstable PYGL 28 50 O=C(/C=C\c1ccc(Cl)c(Cl)c1)N[C@@H]1CC[C@H](C(=O)O)C1 ZINC000217557270 EG For-Sale Unstable HK2 0 40 O=C(/C=C\c1ccc(Cl)c(Cl)c1)N[C@@H]1CC[C@H](C(=O)O)C1 ZINC000217557270 EG For-Sale Unstable CCR2 0 46 O=C1O[C@@]2(CCCN(C(=O)c3cc4ccccc4o3)C2)c2ccccc21 ZINC000217557271 EH For-Sale Unstable NPY5R 29 40 CCCC[C@@H](CC)CNC[C@@H](O)COCc1ccccc1 ZINC000217557278 CG For-Sale Unstable ADRB2 15 42 O=C(NCCc1ccc(Br)cc1)N1CCN(c2ccccc2)CC1 ZINC000217557292 GH On-Demand Unstable HTR1A 17 50 O=C(NCCc1ccc(Br)cc1)N1CCN(c2ccccc2)CC1 ZINC000217557292 GH On-Demand Unstable DRD3 15 43 O=C(NCCc1ccc(Br)cc1)N1CCN(c2ccccc2)CC1 ZINC000217557292 GH On-Demand Unstable ERBB2 0 41 O=C(NCCc1ccc(Br)cc1)N1CCN(c2ccccc2)CC1 ZINC000217557292 GH On-Demand Unstable AKR1C3 0 44 O=C(NCCc1ccc(Br)cc1)N1CCN(c2ccccc2)CC1 ZINC000217557292 GH On-Demand Unstable GPR183 0 41 O=C([C@@H](N[C@H](c1ccccc1)C1CC1)c1ccccc1)N1CCCCC1 ZINC000217557298 EI On-Demand Unstable MTTP 27 44 O=C([C@@H](N[C@H](c1ccccc1)C1CC1)c1ccccc1)N1CCCCC1 ZINC000217557298 EI On-Demand Unstable DPP7 60 40 COC(=O)CS[C@H]1CCN(C(=O)CCS(=O)(=O)c2ccccc2)C1 ZINC000217557348 FD In-Stock Unstable CCR8 42 34 CC[C@H](C)Nc1ccc(S(=O)(=O)N[C@H](C)CC)cc1C(=O)O ZINC000217557349 EF In-Stock Unstable MMP12 48 38 CC[C@H](C)Nc1ccc(S(=O)(=O)N[C@H](C)CC)cc1C(=O)O ZINC000217557349 EF In-Stock Unstable LEF 54 39 O=C1O[C@]2(CCCN(C(=O)c3cc4ccccc4o3)C2)c2ccccc21 ZINC000217557359 EH For-Sale Unstable NPY5R 29 40 CCCC[C@H](CC)CNC[C@@H](O)COCc1ccccc1 ZINC000217557371 CG For-Sale Unstable ADRB2 15 42 O=C([C@H](N[C@H](c1ccccc1)C1CC1)c1ccccc1)N1CCCCC1 ZINC000217557381 EI On-Demand Unstable MTTP 27 44 O=C([C@H](N[C@H](c1ccccc1)C1CC1)c1ccccc1)N1CCCCC1 ZINC000217557381 EI On-Demand Unstable DPP7 60 40 Cc1ccc(N2CCN(Cc3c(O)c(=O)cc(CN4C[C@@H]5C[C@H](C4)c4cccc(=O)n4C5)n3C)CC2)c(C)c1 ZINC000217557403 KF In-Stock Unstable CHRNA4 28 47 CCCC[C@@H](CC)CNC[C@H](O)COCc1ccccc1 ZINC000217557453 CG For-Sale Unstable ADRB2 15 42 CC[C@@H](C)NS(=O)(=O)c1ccc(NC(C)(C)C)c(C(=O)O)c1 ZINC000217557467 EF In-Stock Unstable ADAMTS4 40 32 CC[C@@H](C)NS(=O)(=O)c1ccc(NC(C)(C)C)c(C(=O)O)c1 ZINC000217557467 EF In-Stock Unstable LEF 45 37 COc1ccc([N+](=O)[O-])cc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217557516 GH On-Demand Unstable RAF1 17 44 COc1ccc([N+](=O)[O-])cc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217557516 GH On-Demand Unstable KCNMA1 21 50 COc1ccc([N+](=O)[O-])cc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217557516 GH On-Demand Unstable Q8MMZ8_EIMTE 0 44 CCCC[C@H](CC)CNC[C@H](O)COCc1ccccc1 ZINC000217557543 CG For-Sale Unstable ADRB2 15 42 CC[C@H](C)NS(=O)(=O)c1ccc(NC(C)(C)C)c(C(=O)O)c1 ZINC000217557556 EF In-Stock Unstable ADAMTS4 40 32 CC[C@H](C)NS(=O)(=O)c1ccc(NC(C)(C)C)c(C(=O)O)c1 ZINC000217557556 EF In-Stock Unstable LEF 45 37 COc1cc(Cl)c(C)cc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217557611 GJ For-Sale Unstable RAF1 24 63 COc1cc(Cl)c(C)cc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217557611 GJ For-Sale Unstable CAN2 0 41 O=C(CN1CCC[C@@H]2CCCC[C@H]21)c1ccc(Cl)cc1Cl ZINC000217557636 EJ For-Sale Unstable P2RX7 15 40 C=CCNc1ccc(S(=O)(=O)N[C@@H](C)CC)cc1C(=O)O ZINC000217557653 DE In-Stock Unstable ADAMTS4 41 33 Cc1cc(C)c(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c(C)c1 ZINC000217557674 EH For-Sale Unstable NPY5R 28 41 COC(=O)CS[C@@H]1CCN(C(=O)C2(c3ccc(Cl)cc3)CCCC2)C1 ZINC000217557675 GH In-Stock Unstable SLC6A1 0 40 O=C(CN1CCC[C@H]2CCCC[C@H]21)c1ccc(Cl)cc1Cl ZINC000217557714 EJ For-Sale Unstable P2RX7 15 40 C=CCNc1ccc(S(=O)(=O)N[C@H](C)CC)cc1C(=O)O ZINC000217557747 DE In-Stock Unstable ADAMTS4 41 33 Cc1cc(C)c(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c(C)c1 ZINC000217557762 EH For-Sale Unstable NPY5R 28 41 COC(=O)CS[C@H]1CCN(C(=O)C2(c3ccc(Cl)cc3)CCCC2)C1 ZINC000217557767 GH In-Stock Unstable SLC6A1 0 40 COC(=O)CS[C@H]1CCN(C(=O)C2(c3ccc(Cl)cc3)CCCC2)C1 ZINC000217557767 GH In-Stock Unstable CCR1 42 36 O=C(CN[C@@H](c1ccccc1)C1CC1)N1CCN(S(=O)(=O)c2c(F)cccc2F)CC1 ZINC000217557857 IF On-Demand Unstable PKM 26 49 CC[C@@H](C)NS(=O)(=O)c1ccc(NC2CC2)c(C(=O)O)c1 ZINC000217557858 DE In-Stock Unstable LEF 41 38 CC(C)CCNC(=O)NCCc1ccc(Br)cc1 ZINC000217557859 DG On-Demand Unstable ANPEP 22 43 CC(C)CCNC(=O)NCCc1ccc(Br)cc1 ZINC000217557859 DG On-Demand Unstable DNPEP 0 40 CC(C)CCNC(=O)NCCc1ccc(Br)cc1 ZINC000217557859 DG On-Demand Unstable AMP1_PLAFQ 23 43 CC(C)CCNC(=O)NCCc1ccc(Br)cc1 ZINC000217557859 DG On-Demand Unstable LIG1 0 41 CN(C)c1ccc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217557886 FG For-Sale Unstable NPY5R 25 40 O=C(CN1CC[C@@H](c2ccccc2)C1)NCc1nc(-c2cnccn2)n[nH]1 ZINC000217557921 FD In-Stock Unstable PRCP 26 41 O=C(CN1CC[C@@H](c2ccccc2)C1)NCc1nc(-c2cnccn2)n[nH]1 ZINC000217557921 FD In-Stock Unstable COLA 54 37 O=C(CN1CC[C@@H](c2ccccc2)C1)NCc1nc(-c2cnccn2)n[nH]1 ZINC000217557921 FD In-Stock Unstable CPT1A 45 37 O=C(CN[C@H](c1ccccc1)C1CC1)N1CCN(S(=O)(=O)c2c(F)cccc2F)CC1 ZINC000217557930 IF On-Demand Unstable PKM 26 49 CC[C@H](C)NS(=O)(=O)c1ccc(NC2CC2)c(C(=O)O)c1 ZINC000217557943 DE In-Stock Unstable LEF 41 38 CN(C)c1ccc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217557969 FG For-Sale Unstable NPY5R 25 40 O=C(CN1CC[C@H](c2ccccc2)C1)NCc1nc(-c2cnccn2)n[nH]1 ZINC000217558011 FD In-Stock Unstable PRCP 26 41 O=C(CN1CC[C@H](c2ccccc2)C1)NCc1nc(-c2cnccn2)n[nH]1 ZINC000217558011 FD In-Stock Unstable COLA 54 37 O=C(CN1CC[C@H](c2ccccc2)C1)NCc1nc(-c2cnccn2)n[nH]1 ZINC000217558011 FD In-Stock Unstable CPT1A 45 37 Cc1cccc(C)c1NC(=O)CN1CCN(C(=O)CN[C@@H](c2ccccc2)C2CC2)CC1 ZINC000217558044 IG On-Demand Unstable DRD4 19 50 CC[C@@H](C)NS(=O)(=O)c1ccc(NC2CCCC2)c(C(=O)O)c1 ZINC000217558047 EF In-Stock Unstable LEF 41 41 COC(=O)CS[C@H]1CCN(C(=O)c2ccc(S(=O)(=O)N(C)C)cc2)C1 ZINC000217558066 GD In-Stock Unstable L3MBTL3 45 35 CN(C)c1cccc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217558101 FG For-Sale Unstable NPY5R 26 40 CC[C@H](C)NS(=O)(=O)c1ccc(NC2CCCC2)c(C(=O)O)c1 ZINC000217558119 EF In-Stock Unstable LEF 41 41 Cc1cccc(C)c1NC(=O)CN1CCN(C(=O)CN[C@H](c2ccccc2)C2CC2)CC1 ZINC000217558121 IG On-Demand Unstable DRD4 19 50 COC(=O)CS[C@@H]1CCN(C(=O)c2ccc(S(=O)(=O)N(C)C)cc2)C1 ZINC000217558160 GD In-Stock Unstable L3MBTL3 45 35 Cn1c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c(O)c1CN1CCN(c2ccccn2)CC1 ZINC000217558177 KD In-Stock Unstable CHRNA4 29 49 O=C(NCCc1ccc(Br)cc1)N1CCN(c2ccccc2F)CC1 ZINC000217558195 HH On-Demand Unstable HTR1A 17 44 O=C(NCCc1ccc(Br)cc1)N1CCN(c2ccccc2F)CC1 ZINC000217558195 HH On-Demand Unstable DRD2 20 42 O=C(NCCc1ccc(Br)cc1)N1CCN(c2ccccc2F)CC1 ZINC000217558195 HH On-Demand Unstable DRD3 33 42 O=C(NCCc1ccc(Br)cc1)N1CCN(c2ccccc2F)CC1 ZINC000217558195 HH On-Demand Unstable CXCR3 16 42 CN(C)c1cccc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217558199 FG For-Sale Unstable NPY5R 26 40 COc1ccccc1/C=C\C(=O)N[C@@H]1CC[C@H](C(=O)O)C1 ZINC000217558213 CE On-Demand Unstable CYSP_PLAFA 40 34 CC[C@@H](C)NS(=O)(=O)c1ccc(NC2CCCCC2)c(C(=O)O)c1 ZINC000217558223 FG In-Stock Unstable MMP13 19 41 CC[C@@H](C)NS(=O)(=O)c1ccc(NC2CCCCC2)c(C(=O)O)c1 ZINC000217558223 FG In-Stock Unstable LEF 41 42 O=C(CN1CCC[C@@H]2CCCC[C@H]21)c1ccc(F)cc1 ZINC000217558240 CH For-Sale Unstable HTR2A 18 44 Cc1c(Cl)nc(C2CC2)nc1N1CCN(C)[C@@H](C)C1 ZINC000217558245 CE For-Sale Unstable CHRM3 19 47 O=C1[C@H]2[C@@H]3C=C[C@@H]([C@H]4C[C@@H]34)[C@H]2C(=O)N1c1cccc(C(F)(F)F)c1 ZINC000217558295 EG In-Stock Unstable ME1 0 43 O=C1[C@H]2[C@@H]3C=C[C@@H]([C@H]4C[C@@H]34)[C@H]2C(=O)N1c1cccc(C(F)(F)F)c1 ZINC000217558295 EG In-Stock Unstable GALR3 44 35 O=C1[C@H]2[C@@H]3C=C[C@@H]([C@H]4C[C@@H]34)[C@H]2C(=O)N1c1cccc(C(F)(F)F)c1 ZINC000217558295 EG In-Stock Unstable PDS 20 49 CC[C@H](C)NS(=O)(=O)c1ccc(NC2CCCCC2)c(C(=O)O)c1 ZINC000217558316 FG In-Stock Unstable MMP13 19 41 CC[C@H](C)NS(=O)(=O)c1ccc(NC2CCCCC2)c(C(=O)O)c1 ZINC000217558316 FG In-Stock Unstable LEF 41 42 O=C1O[C@@]2(CCCN(C(=O)c3ccc4c(c3)OCO4)C2)c2ccccc21 ZINC000217558328 FF For-Sale Unstable NPY5R 26 44 O=C(CN1CCC[C@H]2CCCC[C@H]21)c1ccc(F)cc1 ZINC000217558333 CH For-Sale Unstable HTR2A 18 44 O=C1O[C@]2(CCCN(C(=O)c3ccc4c(c3)OCO4)C2)c2ccccc21 ZINC000217558412 FF For-Sale Unstable NPY5R 26 44 Cc1ccc(NC(=O)NCCc2ccc(Br)cc2)c(Br)c1 ZINC000217558431 HJ For-Sale Unstable RAF1 31 40 COc1ccc(/C=C\C(=O)N[C@@H]2CC[C@H](C(=O)O)C2)cc1 ZINC000217558439 CE On-Demand Unstable MMP2 23 49 COc1ccc(/C=C\C(=O)N[C@@H]2CC[C@H](C(=O)O)C2)cc1 ZINC000217558439 CE On-Demand Unstable HDA106 0 41 COc1ccc(/C=C\C(=O)N[C@@H]2CC[C@H](C(=O)O)C2)cc1 ZINC000217558439 CE On-Demand Unstable HD1B 0 41 COc1ccc(/C=C\C(=O)N[C@@H]2CC[C@H](C(=O)O)C2)cc1 ZINC000217558439 CE On-Demand Unstable GPR183 0 41 COc1ccccc1-n1cc(CNC(=O)Cn2nc(C)c(Cl)c2C)cn1 ZINC000217558445 FF In-Stock Unstable P2RX7 24 45 COc1ccc(CC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217558529 FF For-Sale Unstable NPY5R 26 49 Cn1c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c(O)c1CN1CCN(c2cccc(Cl)c2)CC1 ZINC000217558556 KF In-Stock Unstable CHRNA4 28 47 COc1ccc(CC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217558621 FF For-Sale Unstable NPY5R 26 49 O=C(CN1CCC[C@@H]2CCCC[C@H]21)c1cccs1 ZINC000217558626 CH For-Sale Unstable NAMPT 40 34 CC[C@@H](C)NS(=O)(=O)c1ccc(NCCO)c(C(=O)O)c1 ZINC000217558644 DC In-Stock Unstable LEF 45 37 COC(=O)CS[C@@H]1CCN(C(=O)c2ccc(OC(F)(F)F)cc2)C1 ZINC000217558648 FF In-Stock Unstable GCGR 23 44 COC(=O)CS[C@@H]1CCN(C(=O)c2ccc(OC(F)(F)F)cc2)C1 ZINC000217558648 FF In-Stock Unstable EPHX2 49 45 COC(=O)CS[C@@H]1CCN(C(=O)c2ccc(OC(F)(F)F)cc2)C1 ZINC000217558648 FF In-Stock Unstable L3MBTL3 43 35 Cc1cc(NC(=O)NCCc2ccc(Br)cc2)ccc1Br ZINC000217558656 HJ For-Sale Unstable RAF1 30 44 Cc1cc(NC(=O)NCCc2ccc(Br)cc2)ccc1Br ZINC000217558656 HJ For-Sale Unstable CA12 15 42 Cc1cc(NC(=O)NCCc2ccc(Br)cc2)ccc1Br ZINC000217558656 HJ For-Sale Unstable Q8MMZ8_EIMTE 0 44 Cc1cc(NC(=O)NCCc2ccc(Br)cc2)ccc1Br ZINC000217558656 HJ For-Sale Unstable IDO1 16 42 O=C(CN1CCC[C@H]2CCCC[C@H]21)c1cccs1 ZINC000217558702 CH For-Sale Unstable NAMPT 40 34 CN(Cc1ccccc1)Cc1c(O)c(=O)cc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)n1C ZINC000217558724 JF In-Stock Unstable CHRNA4 31 56 COC(=O)CS[C@H]1CCN(C(=O)c2ccc(OC(F)(F)F)cc2)C1 ZINC000217558726 FF In-Stock Unstable GCGR 23 44 COC(=O)CS[C@H]1CCN(C(=O)c2ccc(OC(F)(F)F)cc2)C1 ZINC000217558726 FF In-Stock Unstable EPHX2 49 45 COC(=O)CS[C@H]1CCN(C(=O)c2ccc(OC(F)(F)F)cc2)C1 ZINC000217558726 FF In-Stock Unstable L3MBTL3 43 35 CC[C@H](C)NS(=O)(=O)c1ccc(NCCO)c(C(=O)O)c1 ZINC000217558729 DC In-Stock Unstable LEF 45 37 CCOc1ccccc1C(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217558736 FG For-Sale Unstable NPY5R 27 43 CCOc1ccccc1C(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217558736 FG For-Sale Unstable HCN1 62 39 CCOc1ccccc1C(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217558736 FG For-Sale Unstable HCN4 49 38 COc1ccc(-c2ccc3nnc([C@@H]4CCNC4)n3n2)cc1 ZINC000217558791 CD In-Stock Unstable LRRK2 26 45 O=C(CN1CCC[C@@H]2CCCC[C@H]21)c1ccc(Cl)c(Cl)c1 ZINC000217558794 EJ For-Sale Unstable OPRK1 17 43 O=C(CN1CCC[C@@H]2CCCC[C@H]21)c1ccc(Cl)c(Cl)c1 ZINC000217558794 EJ For-Sale Unstable KMO 0 42 CCOc1ccccc1C(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217558829 FG For-Sale Unstable NPY5R 27 43 CCOc1ccccc1C(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217558829 FG For-Sale Unstable HCN1 62 39 CCOc1ccccc1C(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217558829 FG For-Sale Unstable HCN4 49 38 CC[C@@H](C)NS(=O)(=O)c1ccc(NCCCO)c(C(=O)O)c1 ZINC000217558843 ED In-Stock Unstable LEF 44 35 COC(=O)CS[C@H]1CCN(C(=O)c2ccc(-c3cccc(OC)c3)cc2)C1 ZINC000217558845 GG In-Stock Unstable DRD4 41 33 COC(=O)CS[C@H]1CCN(C(=O)c2ccc(-c3cccc(OC)c3)cc2)C1 ZINC000217558845 GG In-Stock Unstable GRM3 15 40 COC(=O)CS[C@H]1CCN(C(=O)c2ccc(-c3cccc(OC)c3)cc2)C1 ZINC000217558845 GG In-Stock Unstable L3MBTL3 45 33 CN1C(=O)COc2ccc(C(=O)CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)cc21 ZINC000217558853 GD In-Stock Unstable CHRNA4 32 61 COc1ccc(-c2ccc3nnc([C@H]4CCNC4)n3n2)cc1 ZINC000217558871 CD In-Stock Unstable LRRK2 26 45 O=C(CN1CCC[C@H]2CCCC[C@H]21)c1ccc(Cl)c(Cl)c1 ZINC000217558886 EJ For-Sale Unstable OPRK1 17 43 O=C(CN1CCC[C@H]2CCCC[C@H]21)c1ccc(Cl)c(Cl)c1 ZINC000217558886 EJ For-Sale Unstable KMO 0 42 CC[C@H](C)NS(=O)(=O)c1ccc(NCCCO)c(C(=O)O)c1 ZINC000217558929 ED In-Stock Unstable LEF 44 35 COC(=O)CS[C@@H]1CCN(C(=O)c2ccc(-c3cccc(OC)c3)cc2)C1 ZINC000217558937 GG In-Stock Unstable DRD4 41 33 COC(=O)CS[C@@H]1CCN(C(=O)c2ccc(-c3cccc(OC)c3)cc2)C1 ZINC000217558937 GG In-Stock Unstable GRM3 15 40 CCOc1ccc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217558945 FG For-Sale Unstable AVPR1A 15 41 CCOc1ccc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217558945 FG For-Sale Unstable NPY5R 26 42 COc1ccc(-c2ccc3nnc([C@@H]4CCNC4)n3n2)cc1OC ZINC000217558984 ED In-Stock Unstable PDE4D 50 43 COc1ccc(-c2ccc3nnc([C@@H]4CCNC4)n3n2)cc1OC ZINC000217558984 ED In-Stock Unstable LRRK2 28 46 COc1ccc(CN2CCN(Cc3c(O)c(=O)cc(CN4C[C@@H]5C[C@H](C4)c4cccc(=O)n4C5)n3C)CC2)c(OC)c1OC ZINC000217559001 KE In-Stock Unstable CHRNA4 27 44 COc1ccc(CN2CCN(Cc3c(O)c(=O)cc(CN4C[C@@H]5C[C@H](C4)c4cccc(=O)n4C5)n3C)CC2)c(OC)c1OC ZINC000217559001 KE In-Stock Unstable SLC9A1 59 33 C[C@H](C(=O)N1CCCCC1)N1CCC[C@@H](CN)C1 ZINC000217559011 CD On-Demand Unstable DPP7 54 44 CCOc1ccc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217559030 FG For-Sale Unstable AVPR1A 15 41 CCOc1ccc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217559030 FG For-Sale Unstable NPY5R 26 42 COc1ccc(-c2ccc3nnc([C@H]4CCNC4)n3n2)cc1OC ZINC000217559056 ED In-Stock Unstable PDE4D 50 43 COc1ccc(-c2ccc3nnc([C@H]4CCNC4)n3n2)cc1OC ZINC000217559056 ED In-Stock Unstable LRRK2 28 46 CC[C@@H](C)NS(=O)(=O)c1ccc(NCCOC)c(C(=O)O)c1 ZINC000217559059 ED In-Stock Unstable LEF 40 37 C[C@@H](C(=O)N1CCCCC1)N1CCC[C@@H](CN)C1 ZINC000217559100 CD On-Demand Unstable DPP7 54 44 COc1cc2c(cc1OC)CN(Cc1c(O)c(=O)cc(CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)n1C)CC2 ZINC000217559108 KE In-Stock Unstable CHRNA4 35 45 COc1cc2c(cc1OC)CN(Cc1c(O)c(=O)cc(CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)n1C)CC2 ZINC000217559108 KE In-Stock Unstable ABCB1B 57 32 CC[C@@H](C)c1ccccc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217559127 GK For-Sale Unstable ANPEP 15 41 CC[C@@H](C)c1ccccc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217559127 GK For-Sale Unstable AMP1_PLAFQ 23 41 CC[C@@H](C)c1ccccc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217559127 GK For-Sale Unstable ACAT 0 51 CC[C@@H](C)c1ccccc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217559127 GK For-Sale Unstable AO-ACHE 0 40 COc1cccc(CC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217559131 FF For-Sale Unstable NPY5R 26 49 CC[C@H](C)NS(=O)(=O)c1ccc(NCCOC)c(C(=O)O)c1 ZINC000217559144 ED In-Stock Unstable LEF 40 37 COc1ccc(OC)c(-c2ccc3nnc([C@@H]4CCNC4)n3n2)c1 ZINC000217559153 ED In-Stock Unstable LRRK2 23 42 CC[C@H](C)c1ccccc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217559180 GK For-Sale Unstable ANPEP 15 41 CC[C@H](C)c1ccccc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217559180 GK For-Sale Unstable AMP1_PLAFQ 23 41 CC[C@H](C)c1ccccc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217559180 GK For-Sale Unstable ACAT 0 51 CC[C@H](C)c1ccccc1NC(=O)NCCc1ccc(Br)cc1 ZINC000217559180 GK For-Sale Unstable AO-ACHE 0 40 COc1cccc(CC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217559196 FF For-Sale Unstable NPY5R 26 49 Cc1ccc(-n2nc(C)cc2NC(=O)CN[C@@H](c2ccccc2)C2CC2)cc1 ZINC000217559213 FI On-Demand Unstable MAPK14 18 43 CC(=O)NCCOc1ccc(C(=O)N(C)C[C@@H]2COCCO2)cc1 ZINC000217559215 EC In-Stock Unstable OXTR 0 40 CC[C@@H](C)NS(=O)(=O)c1ccc(NCCCOC)c(C(=O)O)c1 ZINC000217559240 ED In-Stock Unstable BDKRB1 15 40 O=C(CN1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)c1ccc(Cl)cc1Cl ZINC000217559246 GG In-Stock Unstable CHRNA4 35 63 COc1ccc(OC)c(-c2ccc3nnc([C@H]4CCNC4)n3n2)c1 ZINC000217559248 ED In-Stock Unstable LRRK2 23 42 CC(=O)NCCOc1ccc(C(=O)N(C)C[C@H]2COCCO2)cc1 ZINC000217559286 EC In-Stock Unstable OXTR 0 40 Cc1ccc(-n2nc(C)cc2NC(=O)CN[C@H](c2ccccc2)C2CC2)cc1 ZINC000217559292 FI On-Demand Unstable MAPK14 18 43 CC[C@H](C)NS(=O)(=O)c1ccc(NCCCOC)c(C(=O)O)c1 ZINC000217559312 ED In-Stock Unstable BDKRB1 15 40 Cc1ccccc1OCC(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217559326 FG For-Sale Unstable NPY5R 25 43 Cn1c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c(O)c1CN1CCCC1 ZINC000217559343 HD In-Stock Unstable CHRNA4 32 52 C[C@H](C(=O)N1CCCCCC1)N1CCC[C@@H](CN)C1 ZINC000217559391 CD On-Demand Unstable DPP7 54 44 Cc1ccc(C(=O)CN2CCC[C@@H]3CCCC[C@H]32)cc1 ZINC000217559401 CH For-Sale Unstable HRH3 15 41 Cc1ccccc1OCC(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217559403 FG For-Sale Unstable NPY5R 25 43 CC[C@@H](C)NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217559414 FG In-Stock Unstable TRY2_BOVIN 56 33 CC[C@@H](C)NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217559414 FG In-Stock Unstable MMP12 47 40 CC[C@@H](C)NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217559414 FG In-Stock Unstable ADAMTS4 53 37 CC[C@@H](C)NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217559414 FG In-Stock Unstable ACPS 0 40 CC[C@@H](C)NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217559414 FG In-Stock Unstable PDS 40 32 COC(=O)CS[C@H]1CCN(C(=O)CCc2ccc(OC)c(OCc3ccccc3)c2)C1 ZINC000217559428 IH In-Stock Unstable GRIN2B 15 40 COC(=O)CS[C@H]1CCN(C(=O)CCc2ccc(OC)c(OCc3ccccc3)c2)C1 ZINC000217559428 IH In-Stock Unstable MTNR1B 20 43 O=C(NCCc1ccc(Br)cc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217559431 HH On-Demand Unstable CHRM2 24 48 O=C(NCCc1ccc(Br)cc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217559431 HH On-Demand Unstable CHRM1 18 47 O=C(NCCc1ccc(Br)cc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217559431 HH On-Demand Unstable DRD2 26 60 O=C(NCCc1ccc(Br)cc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217559431 HH On-Demand Unstable DRD4 60 60 O=C(NCCc1ccc(Br)cc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217559431 HH On-Demand Unstable ACHE 49 53 O=C(NCCc1ccc(Br)cc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217559431 HH On-Demand Unstable HRH2 26 46 O=C(NCCc1ccc(Br)cc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217559431 HH On-Demand Unstable DRD3 22 60 O=C(NCCc1ccc(Br)cc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217559431 HH On-Demand Unstable KCNH2 17 45 O=C(NCCc1ccc(Br)cc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217559431 HH On-Demand Unstable CHRM3 27 40 O=C(NCCc1ccc(Br)cc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217559431 HH On-Demand Unstable LTA4H 24 43 O=C(NCCc1ccc(Br)cc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217559431 HH On-Demand Unstable VACHT_TETCF 0 41 O=C(NCCc1ccc(Br)cc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217559431 HH On-Demand Unstable HRH3 15 47 O=C(NCCc1ccc(Br)cc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217559431 HH On-Demand Unstable SIGMAR1 72 71 O=C(NCCc1ccc(Br)cc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217559431 HH On-Demand Unstable SSTR5 52 38 O=C(NCCc1ccc(Br)cc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217559431 HH On-Demand Unstable BCHE 0 45 O=C(NCCc1ccc(Br)cc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217559431 HH On-Demand Unstable CCR3 56 48 O=C(NCCc1ccc(Br)cc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217559431 HH On-Demand Unstable NPFFR2 34 43 O=C(NCCc1ccc(Br)cc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217559431 HH On-Demand Unstable UTS2R 20 42 O=C(NCCc1ccc(Br)cc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217559431 HH On-Demand Unstable SLC6A5 33 48 O=C(NCCc1ccc(Br)cc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217559431 HH On-Demand Unstable EPHX2 29 60 O=C(NCCc1ccc(Br)cc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217559431 HH On-Demand Unstable TGM2 22 41 O=C(NCCc1ccc(Br)cc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217559431 HH On-Demand Unstable CXCR3 45 45 O=C(NCCc1ccc(Br)cc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217559431 HH On-Demand Unstable MCHR1 54 50 O=C(NCCc1ccc(Br)cc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217559431 HH On-Demand Unstable CACNA1G 35 44 O=C(NCCc1ccc(Br)cc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217559431 HH On-Demand Unstable CCR8 15 41 O=C(NCCc1ccc(Br)cc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217559431 HH On-Demand Unstable NPFFR1 56 43 O=C(NCCc1ccc(Br)cc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217559431 HH On-Demand Unstable ADIPOR1 0 46 O=C(NCCc1ccc(Br)cc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217559431 HH On-Demand Unstable ADIPOR2 0 46 Cn1c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c(O)c1CN1CCN(c2ccccc2)CC1 ZINC000217559458 KE In-Stock Unstable CHRNA4 38 52 C[C@@H](C(=O)N1CCCCCC1)N1CCC[C@@H](CN)C1 ZINC000217559481 CD On-Demand Unstable DPP7 69 44 Cc1ccc(C(=O)CN2CCC[C@H]3CCCC[C@H]32)cc1 ZINC000217559492 CH For-Sale Unstable HRH3 15 41 CC[C@H](C)NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217559493 FG In-Stock Unstable TRY2_BOVIN 56 33 CC[C@H](C)NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217559493 FG In-Stock Unstable MMP12 47 40 CC[C@H](C)NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217559493 FG In-Stock Unstable ADAMTS4 53 37 CC[C@H](C)NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217559493 FG In-Stock Unstable ACPS 0 40 CC[C@H](C)NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217559493 FG In-Stock Unstable PDS 40 32 COC(=O)CS[C@@H]1CCN(C(=O)CCc2ccc(OC)c(OCc3ccccc3)c2)C1 ZINC000217559512 IH In-Stock Unstable GRIN2B 15 40 COC(=O)CS[C@@H]1CCN(C(=O)CCc2ccc(OC)c(OCc3ccccc3)c2)C1 ZINC000217559512 IH In-Stock Unstable MTNR1B 20 43 Cc1cccc(OCC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217559515 FG For-Sale Unstable CPT2 41 35 Cc1cccc(OCC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217559515 FG For-Sale Unstable NPY5R 28 43 COc1ccc(-c2ccc3nnc(C4CCNCC4)n3n2)cc1 ZINC000217559587 DE In-Stock Unstable PDE4D 15 41 COc1ccc(-c2ccc3nnc(C4CCNCC4)n3n2)cc1 ZINC000217559587 DE In-Stock Unstable LRRK2 30 49 CC[C@@H](C)NS(=O)(=O)c1ccc(N[C@@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217559588 GH In-Stock Unstable BDKRB1 21 40 CC[C@@H](C)NS(=O)(=O)c1ccc(N[C@@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217559588 GH In-Stock Unstable MMP12 44 37 CC[C@@H](C)NS(=O)(=O)c1ccc(N[C@@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217559588 GH In-Stock Unstable ADAMTS4 41 32 CC[C@@H](C)NS(=O)(=O)c1ccc(N[C@@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217559588 GH In-Stock Unstable LEF 34 41 c1cncc(CN2CCN(C[C@@H]3[C@H]4CNC[C@H]43)CC2)c1 ZINC000217559589 CC In-Stock Unstable CHRNA7 20 40 c1cncc(CN2CCN(C[C@@H]3[C@H]4CNC[C@H]43)CC2)c1 ZINC000217559589 CC In-Stock Unstable CHRNA4 16 41 O=c1cc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)c2ccc(O)cc2o1 ZINC000217559598 FE In-Stock Unstable CHRNA4 33 55 O=c1cc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)c2ccc(O)cc2o1 ZINC000217559598 FE In-Stock Unstable HSD17B3 35 42 Cc1cccc(OCC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217559603 FG For-Sale Unstable CPT2 41 35 Cc1cccc(OCC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217559603 FG For-Sale Unstable NPY5R 28 43 C[C@@H]1CCCN(c2ccc(CBr)cc2)CC1 ZINC000217559622 CI For-Sale Unstable L3MBTL3 42 43 CC[C@H](C)NS(=O)(=O)c1ccc(N[C@@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217559668 GH In-Stock Unstable BDKRB1 21 40 CC[C@H](C)NS(=O)(=O)c1ccc(N[C@@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217559668 GH In-Stock Unstable MMP12 44 37 CC[C@H](C)NS(=O)(=O)c1ccc(N[C@@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217559668 GH In-Stock Unstable ADAMTS4 41 32 CC[C@H](C)NS(=O)(=O)c1ccc(N[C@@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217559668 GH In-Stock Unstable LEF 34 41 O=C(NCCc1ccc(Br)cc1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217559685 IG For-Sale Unstable BMP1 48 39 O=C(NCCc1ccc(Br)cc1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217559685 IG For-Sale Unstable NOS2 89 36 O=C(NCCc1ccc(Br)cc1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217559685 IG For-Sale Unstable SSTR3 44 30 O=C(NCCc1ccc(Br)cc1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217559685 IG For-Sale Unstable MCHR1 28 49 Cc1cccc(N2CCN(Cc3c(O)c(=O)cc(CN4C[C@@H]5C[C@H](C4)c4cccc(=O)n4C5)n3C)CC2)c1C ZINC000217559692 KF In-Stock Unstable CHRNA4 28 44 COc1ccc(-c2ccc3nnc(C4CCNCC4)n3n2)cc1OC ZINC000217559701 EE In-Stock Unstable PDE4D 53 45 COc1ccc(-c2ccc3nnc(C4CCNCC4)n3n2)cc1OC ZINC000217559701 EE In-Stock Unstable LRRK2 31 50 C[C@H]1CCCN(c2ccc(CBr)cc2)CC1 ZINC000217559708 CI For-Sale Unstable L3MBTL3 42 43 CSc1ccccc1C(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217559716 FH For-Sale Unstable NPY5R 26 43 O=C(CN1CCC[C@@H]2CCCC[C@H]21)c1cccc(Cl)c1 ZINC000217559743 CI For-Sale Unstable GRM5 19 41 CC[C@@H](C)NS(=O)(=O)c1ccc(N[C@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217559754 GH In-Stock Unstable BDKRB1 21 40 CC[C@@H](C)NS(=O)(=O)c1ccc(N[C@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217559754 GH In-Stock Unstable MMP12 44 37 CC[C@@H](C)NS(=O)(=O)c1ccc(N[C@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217559754 GH In-Stock Unstable ADAMTS4 41 32 CC[C@@H](C)NS(=O)(=O)c1ccc(N[C@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217559754 GH In-Stock Unstable LEF 34 41 CSc1ccccc1C(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217559790 FH For-Sale Unstable NPY5R 26 43 COc1ccc(OC)c(-c2ccc3nnc(C4CCNCC4)n3n2)c1 ZINC000217559796 EE In-Stock Unstable LRRK2 23 43 Cc1ccc(N)c(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217559811 EH For-Sale Unstable RAF1 28 41 COC(=O)CS[C@@H]1CCN(C(=O)CCc2cccc(Cl)c2)C1 ZINC000217559818 EF In-Stock Unstable FDFT1 40 32 O=C(CN1CCC[C@H]2CCCC[C@H]21)c1cccc(Cl)c1 ZINC000217559819 CI For-Sale Unstable GRM5 19 41 CC1(C)Cc2ccccc2-c2nc(CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)[nH]c(=O)c21 ZINC000217559843 IG In-Stock Unstable CHRNA4 31 51 CC[C@H](C)NS(=O)(=O)c1ccc(N[C@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217559844 GH In-Stock Unstable BDKRB1 21 40 CC[C@H](C)NS(=O)(=O)c1ccc(N[C@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217559844 GH In-Stock Unstable MMP12 44 37 CC[C@H](C)NS(=O)(=O)c1ccc(N[C@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217559844 GH In-Stock Unstable ADAMTS4 41 32 CC[C@H](C)NS(=O)(=O)c1ccc(N[C@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217559844 GH In-Stock Unstable LEF 34 41 CSc1ncccc1C(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217559901 FG For-Sale Unstable AVPR1A 17 42 CSc1ncccc1C(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217559901 FG For-Sale Unstable NPY5R 42 40 COC(=O)CS[C@H]1CCN(C(=O)CCc2cccc(Cl)c2)C1 ZINC000217559907 EF In-Stock Unstable FDFT1 40 32 COc1ccc(C(=O)CN2CCC[C@@H]3CCCC[C@H]32)cc1 ZINC000217559930 CH For-Sale Unstable HRH3 16 46 COc1ccc(C(=O)CN2CCC[C@@H]3CCCC[C@H]32)cc1 ZINC000217559930 CH For-Sale Unstable SIGMAR1 18 47 CC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217559937 GG In-Stock Unstable MMP13 33 42 CC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217559937 GG In-Stock Unstable TRY2_BOVIN 61 33 CC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217559937 GG In-Stock Unstable MMP2 32 42 CC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217559937 GG In-Stock Unstable MMP8 18 42 CC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217559937 GG In-Stock Unstable MMP12 42 35 CC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217559937 GG In-Stock Unstable ADAMTS4 50 34 Cc1nc2c(C(=O)N3CCCn4nc([C@@H](O)CO)cc4C3)cccc2[nH]1 ZINC000217559967 FD In-Stock Unstable PARP1 35 40 CSc1ncccc1C(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217559975 FG For-Sale Unstable AVPR1A 17 42 CSc1ncccc1C(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217559975 FG For-Sale Unstable NPY5R 42 40 Cn1c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c(O)c1CN1CCCCCC1 ZINC000217559985 IE In-Stock Unstable CHRNA4 31 51 COc1ccc(C(=O)CN2CCC[C@H]3CCCC[C@H]32)cc1 ZINC000217560018 CH For-Sale Unstable HRH3 16 46 COc1ccc(C(=O)CN2CCC[C@H]3CCCC[C@H]32)cc1 ZINC000217560018 CH For-Sale Unstable SIGMAR1 18 47 CC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217560020 GG In-Stock Unstable MMP13 33 42 CC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217560020 GG In-Stock Unstable TRY2_BOVIN 61 33 CC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217560020 GG In-Stock Unstable MMP2 32 42 CC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217560020 GG In-Stock Unstable MMP8 18 42 CC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217560020 GG In-Stock Unstable MMP12 42 35 CC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217560020 GG In-Stock Unstable ADAMTS4 50 34 COC(=O)CS[C@H]1CCN(C(=O)CCc2c(OC)ccc3ccccc23)C1 ZINC000217560027 GG In-Stock Unstable XIAP 55 38 Cc1nc2c(C(=O)N3CCCn4nc([C@H](O)CO)cc4C3)cccc2[nH]1 ZINC000217560039 FD In-Stock Unstable PARP1 35 40 NC[C@@H]1CCCN(C[C@@H](O)c2ccccc2)C1 ZINC000217560041 BD On-Demand Unstable SLC6A1 0 43 NC[C@@H]1CCCN(C[C@@H](O)c2ccccc2)C1 ZINC000217560041 BD On-Demand Unstable OPRK1 0 44 NC[C@@H]1CCCN(C[C@@H](O)c2ccccc2)C1 ZINC000217560041 BD On-Demand Unstable IGF1R 0 43 NC[C@@H]1CCCN(C[C@@H](O)c2ccccc2)C1 ZINC000217560041 BD On-Demand Unstable SLC18A3 27 42 O=C1O[C@@]2(CCCN(C(=O)COc3ccccc3F)C2)c2ccccc21 ZINC000217560092 FF For-Sale Unstable NPY5R 31 45 CC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217560120 HG In-Stock Unstable CA2 16 41 CC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217560120 HG In-Stock Unstable BMP1 90 40 CC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217560120 HG In-Stock Unstable CA1 16 43 CC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217560120 HG In-Stock Unstable MMP13 76 46 CC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217560120 HG In-Stock Unstable CA14 17 42 CC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217560120 HG In-Stock Unstable MMP2 48 42 CC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217560120 HG In-Stock Unstable MMP3 50 42 CC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217560120 HG In-Stock Unstable MMP8 35 42 CC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217560120 HG In-Stock Unstable MMP9 52 46 CC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217560120 HG In-Stock Unstable MMP12 52 39 CC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217560120 HG In-Stock Unstable PTGDR 30 42 CC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217560120 HG In-Stock Unstable MMP7 30 40 CC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217560120 HG In-Stock Unstable ADAMTS4 57 37 CC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217560120 HG In-Stock Unstable CA9 22 43 CC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217560120 HG In-Stock Unstable MMP1 52 40 CC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217560120 HG In-Stock Unstable AKR1C2 50 37 COC(=O)CS[C@@H]1CCN(C(=O)CCc2c(OC)ccc3ccccc23)C1 ZINC000217560121 GG In-Stock Unstable XIAP 55 38 O=C(CN1CCC[C@@H]2CCCC[C@H]21)c1ccccc1 ZINC000217560140 CH For-Sale Unstable SLC6A1 50 41 O=C(CN1CCC[C@@H]2CCCC[C@H]21)c1ccccc1 ZINC000217560140 CH For-Sale Unstable SLC18A3 40 38 O=C(CN1CCC[C@@H]2CCCC[C@H]21)c1ccccc1 ZINC000217560140 CH For-Sale Unstable PREP 47 43 O=C(CN1CCC[C@@H]2CCCC[C@H]21)c1ccccc1 ZINC000217560140 CH For-Sale Unstable CYP2J2 43 31 O=C1O[C@]2(CCCN(C(=O)COc3ccccc3F)C2)c2ccccc21 ZINC000217560168 FF For-Sale Unstable NPY5R 31 45 NC[C@@H]1CCCN([C@@H]2CCC[C@@H]2O)C1 ZINC000217560169 AC For-Sale Unstable SLC18A3 33 45 O=C(NCCc1ccc(Br)cc1)Nc1cc(F)ccc1F ZINC000217560196 FI On-Demand Unstable RAF1 31 42 CC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217560203 HG In-Stock Unstable CA2 16 41 CC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217560203 HG In-Stock Unstable BMP1 90 40 CC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217560203 HG In-Stock Unstable CA1 16 43 CC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217560203 HG In-Stock Unstable MMP13 76 46 CC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217560203 HG In-Stock Unstable CA14 17 42 CC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217560203 HG In-Stock Unstable MMP2 48 42 CC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217560203 HG In-Stock Unstable MMP3 50 42 CC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217560203 HG In-Stock Unstable MMP8 35 42 CC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217560203 HG In-Stock Unstable MMP9 52 46 CC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217560203 HG In-Stock Unstable MMP12 52 39 CC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217560203 HG In-Stock Unstable PTGDR 30 42 CC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217560203 HG In-Stock Unstable MMP7 30 40 CC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217560203 HG In-Stock Unstable ADAMTS4 57 37 CC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217560203 HG In-Stock Unstable CA9 22 43 CC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217560203 HG In-Stock Unstable MMP1 52 40 CC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217560203 HG In-Stock Unstable AKR1C2 50 37 COC(=O)CS[C@@H]1CCN(C(=O)CCc2ccc(S(C)(=O)=O)cc2)C1 ZINC000217560223 GD In-Stock Unstable GPR119 28 41 COc1ccc(-c2noc(CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)n2)cc1 ZINC000217560229 GF In-Stock Unstable CHRNA4 31 52 O=C(CN1CCC[C@H]2CCCC[C@H]21)c1ccccc1 ZINC000217560231 CH For-Sale Unstable SLC6A1 50 41 O=C(CN1CCC[C@H]2CCCC[C@H]21)c1ccccc1 ZINC000217560231 CH For-Sale Unstable SLC18A3 40 38 O=C(CN1CCC[C@H]2CCCC[C@H]21)c1ccccc1 ZINC000217560231 CH For-Sale Unstable PREP 47 43 O=C(CN1CCC[C@H]2CCCC[C@H]21)c1ccccc1 ZINC000217560231 CH For-Sale Unstable CYP2J2 43 31 O=C1O[C@@]2(CCCN(C(=O)COc3ccc(F)cc3)C2)c2ccccc21 ZINC000217560288 FF For-Sale Unstable CPT2 40 33 O=C1O[C@@]2(CCCN(C(=O)COc3ccc(F)cc3)C2)c2ccccc21 ZINC000217560288 FF For-Sale Unstable NPY5R 34 46 COC(=O)CS[C@H]1CCN(C(=O)CCc2ccc(S(C)(=O)=O)cc2)C1 ZINC000217560294 GD In-Stock Unstable GPR119 28 41 O=C(CN1CCC[C@@H]2CCCC[C@H]21)c1cccc(Br)c1 ZINC000217560309 EI For-Sale Unstable MBTD1 0 43 CC(C)(CO)NC(=O)NCCc1ccc(Br)cc1 ZINC000217560335 DE For-Sale Unstable LIG1 0 40 CC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217560339 IG In-Stock Unstable MMP12 46 34 CC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217560339 IG In-Stock Unstable IAP 0 42 CC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217560339 IG In-Stock Unstable ADAMTS4 51 33 CC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217560339 IG In-Stock Unstable SCMU_MYCTU 0 46 Cc1ccn2c(=O)cc(CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)nc2c1 ZINC000217560347 FD In-Stock Unstable CHRNA4 33 53 Cc1ccn2c(=O)cc(CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)nc2c1 ZINC000217560347 FD In-Stock Unstable PKM 15 50 O=C1O[C@]2(CCCN(C(=O)COc3ccc(F)cc3)C2)c2ccccc21 ZINC000217560384 FF For-Sale Unstable CPT2 40 33 O=C1O[C@]2(CCCN(C(=O)COc3ccc(F)cc3)C2)c2ccccc21 ZINC000217560384 FF For-Sale Unstable NPY5R 34 46 O=C(CN1CCC[C@H]2CCCC[C@H]21)c1cccc(Br)c1 ZINC000217560391 EI For-Sale Unstable MBTD1 0 43 COC(=O)CS[C@@H]1CCN(C(=O)CCc2ccc(C(F)(F)F)cc2)C1 ZINC000217560421 GG In-Stock Unstable EPHX2 15 43 COC(=O)CS[C@@H]1CCN(C(=O)CCc2ccc(C(F)(F)F)cc2)C1 ZINC000217560421 GG In-Stock Unstable LIPG 40 34 CC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217560422 IG In-Stock Unstable MMP12 46 34 CC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217560422 IG In-Stock Unstable IAP 0 42 CC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217560422 IG In-Stock Unstable ADAMTS4 51 33 CC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217560422 IG In-Stock Unstable SCMU_MYCTU 0 46 COC(=O)CCNC(=O)NCCc1ccc(Br)cc1 ZINC000217560436 ED For-Sale Unstable LIG1 0 43 COC(=O)CS[C@H]1CCN(C(=O)CCc2ccc(C(F)(F)F)cc2)C1 ZINC000217560501 GG In-Stock Unstable EPHX2 18 43 COC(=O)CS[C@H]1CCN(C(=O)CCc2ccc(C(F)(F)F)cc2)C1 ZINC000217560501 GG In-Stock Unstable MCHR1 23 40 COC(=O)CS[C@H]1CCN(C(=O)CCc2ccc(C(F)(F)F)cc2)C1 ZINC000217560501 GG In-Stock Unstable LIPG 40 34 O=C1O[C@@]2(CCCN(C(=O)Cc3ccc(Cl)cc3)C2)c2ccccc21 ZINC000217560507 FH For-Sale Unstable NPY5R 26 46 C[C@@H](N[C@@H](c1ccccc1)C1CC1)C(=O)NCc1ccccc1Cl ZINC000217560517 EI On-Demand Unstable P2RX7 40 43 C[C@@H](N[C@@H](c1ccccc1)C1CC1)C(=O)NCc1ccccc1Cl ZINC000217560517 EI On-Demand Unstable PSMB5 17 41 C[C@@H](N[C@@H](c1ccccc1)C1CC1)C(=O)NCc1ccccc1Cl ZINC000217560517 EI On-Demand Unstable BIRC8 53 31 O=C(CN1CCC[C@@H]2CCCC[C@H]21)c1ccccc1F ZINC000217560519 CH For-Sale Unstable SLC6A1 35 40 CCOC(=O)CCNC(=O)NCCc1ccc(Br)cc1 ZINC000217560550 EE For-Sale Unstable LIG1 0 43 C[C@H](N[C@@H](c1ccccc1)C1CC1)C(=O)NCc1ccccc1Cl ZINC000217560586 EI On-Demand Unstable P2RX7 40 43 C[C@H](N[C@@H](c1ccccc1)C1CC1)C(=O)NCc1ccccc1Cl ZINC000217560586 EI On-Demand Unstable PSMB5 17 41 C[C@H](N[C@@H](c1ccccc1)C1CC1)C(=O)NCc1ccccc1Cl ZINC000217560586 EI On-Demand Unstable BIRC8 53 31 O=C1O[C@]2(CCCN(C(=O)Cc3ccc(Cl)cc3)C2)c2ccccc21 ZINC000217560594 FH For-Sale Unstable NPY5R 26 46 O=C(CN1CCC[C@H]2CCCC[C@H]21)c1ccccc1F ZINC000217560602 CH For-Sale Unstable SLC6A1 35 40 Cn1c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c(O)c1CN1CCN(C2CCOCC2)CC1 ZINC000217560608 KD In-Stock Unstable CHRNA4 28 44 C[C@@H](N[C@H](c1ccccc1)C1CC1)C(=O)NCc1ccccc1Cl ZINC000217560667 EI On-Demand Unstable P2RX7 40 43 C[C@@H](N[C@H](c1ccccc1)C1CC1)C(=O)NCc1ccccc1Cl ZINC000217560667 EI On-Demand Unstable PSMB5 17 41 C[C@@H](N[C@H](c1ccccc1)C1CC1)C(=O)NCc1ccccc1Cl ZINC000217560667 EI On-Demand Unstable BIRC8 53 31 CCOC(=O)CNC(=O)NCCc1ccc(Br)cc1 ZINC000217560677 ED For-Sale Unstable LIG1 0 41 O=C1O[C@@]2(CCCN(C(=O)Cc3ccccc3Cl)C2)c2ccccc21 ZINC000217560724 FH For-Sale Unstable NPY5R 29 45 CC[C@@H](C)NS(=O)(=O)c1ccc(NC[C@@H]2CCCO2)c(C(=O)O)c1 ZINC000217560738 FE In-Stock Unstable BDKRB1 22 41 O=c1cc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)oc(CN2CCN(c3ccccc3)CC2)c1O ZINC000217560739 JE In-Stock Unstable CHRNA4 30 53 C[C@H](N[C@H](c1ccccc1)C1CC1)C(=O)NCc1ccccc1Cl ZINC000217560752 EI On-Demand Unstable P2RX7 40 43 C[C@H](N[C@H](c1ccccc1)C1CC1)C(=O)NCc1ccccc1Cl ZINC000217560752 EI On-Demand Unstable PSMB5 17 41 C[C@H](N[C@H](c1ccccc1)C1CC1)C(=O)NCc1ccccc1Cl ZINC000217560752 EI On-Demand Unstable BIRC8 53 31 Cc1ccc(/C=C\C(=O)N[C@@H]2CC[C@H](C(=O)O)C2)cc1 ZINC000217560767 CE On-Demand Unstable HDAC1 18 40 COC(=O)CNC(=O)NCCc1ccc(Br)cc1 ZINC000217560777 DD For-Sale Unstable LIG1 0 40 O=C1O[C@]2(CCCN(C(=O)Cc3ccccc3Cl)C2)c2ccccc21 ZINC000217560809 FH For-Sale Unstable NPY5R 29 45 CC[C@H](C)NS(=O)(=O)c1ccc(NC[C@@H]2CCCO2)c(C(=O)O)c1 ZINC000217560822 FE In-Stock Unstable BDKRB1 22 41 Cn1c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c(O)c1CN1CCN(Cc2ccccc2Cl)CC1 ZINC000217560843 KF In-Stock Unstable CHRNA4 29 50 Cc1ccc(C(=O)N2CCCC[C@@H]2CN2CCCC2)c(O)c1 ZINC000217560870 DF In-Stock Unstable OPRK1 22 50 O=C1CC[C@@H](C(=O)c2cccs2)N1 ZINC000217560872 AD For-Sale Unstable GLRA1 15 41 COC(=O)c1cccc(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217560879 GH On-Demand Unstable CCKAR 0 41 COC(=O)c1cccc(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217560879 GH On-Demand Unstable CCR3 36 40 COC(=O)c1cccc(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217560879 GH On-Demand Unstable RAF1 18 41 COC(=O)c1cccc(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217560879 GH On-Demand Unstable ROCK2 17 44 COC(=O)c1cccc(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217560879 GH On-Demand Unstable EPHX2 15 46 COC(=O)c1cccc(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217560879 GH On-Demand Unstable Q8MMZ8_EIMTE 0 41 COC(=O)c1cccc(NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217560879 GH On-Demand Unstable KCNK3 60 34 C[C@@H](N[C@@H](c1ccccc1)C1CC1)C(=O)Nc1ccc(Cl)cc1C(F)(F)F ZINC000217560883 GK On-Demand Unstable NR1H4 15 41 NC[C@@H]1CCCN([C@@H]2CCCC[C@@H]2O)C1 ZINC000217560889 BC For-Sale Unstable SLC18A3 39 49 C[C@H](C(=O)c1ccccc1)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217560905 CH For-Sale Unstable ACE 34 41 Fc1ccc(Cl)c(O[C@@H]2CCCNCC2)c1 ZINC000217560917 BG For-Sale Unstable SLC6A2 20 48 Fc1ccc(Cl)c(O[C@@H]2CCCNCC2)c1 ZINC000217560917 BG For-Sale Unstable SCD1 21 45 CC[C@@H](C)NS(=O)(=O)c1ccc(NC[C@H]2CCCO2)c(C(=O)O)c1 ZINC000217560918 FE In-Stock Unstable BDKRB1 22 41 CCCc1nnsc1C(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217560928 FF For-Sale Unstable NPY5R 26 40 O=c1cccc2n1C[C@H]1C[C@@H]2CN(Cc2cc(=O)n3ccsc3n2)C1 ZINC000217560947 FD In-Stock Unstable CHRNA4 34 54 Cc1ccc(C(=O)N2CCCC[C@H]2CN2CCCC2)c(O)c1 ZINC000217560957 DF In-Stock Unstable OPRK1 22 50 O=C1CC[C@H](C(=O)c2cccs2)N1 ZINC000217560964 AD For-Sale Unstable GLRA1 15 41 C[C@H](N[C@@H](c1ccccc1)C1CC1)C(=O)Nc1ccc(Cl)cc1C(F)(F)F ZINC000217560965 GK On-Demand Unstable NR1H4 15 41 Fc1ccc(Cl)c(O[C@H]2CCCNCC2)c1 ZINC000217561002 BG For-Sale Unstable SLC6A2 20 48 Fc1ccc(Cl)c(O[C@H]2CCCNCC2)c1 ZINC000217561002 BG For-Sale Unstable SCD1 21 45 C[C@@H](C(=O)c1ccccc1)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217561007 CH For-Sale Unstable ACE 34 41 CC[C@H](C)NS(=O)(=O)c1ccc(NC[C@H]2CCCO2)c(C(=O)O)c1 ZINC000217561009 FE In-Stock Unstable BDKRB1 22 41 CCCc1nnsc1C(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217561028 FF For-Sale Unstable NPY5R 26 40 C[C@@H](N[C@H](c1ccccc1)C1CC1)C(=O)Nc1ccc(Cl)cc1C(F)(F)F ZINC000217561046 GK On-Demand Unstable NR1H4 15 41 C[C@H](C(=O)c1cccc(Cl)c1)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217561105 DJ For-Sale Unstable GRM5 17 40 CC[C@@H](C)NS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217561110 EE In-Stock Unstable KCNQ2 71 39 CC[C@@H](C)NS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217561110 EE In-Stock Unstable TRY2_BOVIN 44 32 CC[C@@H](C)NS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217561110 EE In-Stock Unstable SLC6A9 24 43 C[C@H](N[C@H](c1ccccc1)C1CC1)C(=O)Nc1ccc(Cl)cc1C(F)(F)F ZINC000217561134 GK On-Demand Unstable NR1H4 15 41 O=c1cccc2n1C[C@H]1C[C@@H]2CN(Cc2cc(=O)n3ccccc3n2)C1 ZINC000217561139 ED In-Stock Unstable CHRNA4 34 59 O=c1cccc2n1C[C@H]1C[C@@H]2CN(Cc2cc(=O)n3ccccc3n2)C1 ZINC000217561139 ED In-Stock Unstable PKM 15 48 O=C1O[C@@]2(CCCN(C(=O)c3cnc4ccccc4n3)C2)c2ccccc21 ZINC000217561143 FF For-Sale Unstable NPY5R 42 45 C[C@@H](C(=O)c1cccc(Cl)c1)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217561183 DJ For-Sale Unstable GRM5 17 40 CC[C@H](C)NS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217561186 EE In-Stock Unstable KCNQ2 71 39 CC[C@H](C)NS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217561186 EE In-Stock Unstable TRY2_BOVIN 44 32 CC[C@H](C)NS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217561186 EE In-Stock Unstable SLC6A9 24 43 COC(=O)CS[C@@H]1CCN(C(=O)CCc2ccc(Cl)c(F)c2)C1 ZINC000217561216 FF In-Stock Unstable ENV 40 31 O=C(NCCc1ccc(Br)cc1)NCc1ccc(CO)cc1 ZINC000217561224 FF For-Sale Unstable LIG1 0 41 O=C1O[C@]2(CCCN(C(=O)c3cnc4ccccc4n3)C2)c2ccccc21 ZINC000217561235 FF For-Sale Unstable NPY5R 42 45 COc1ccc(NC(=O)[C@@H](N[C@@H](c2ccccc2)C2CC2)c2ccccc2)cc1 ZINC000217561255 GK On-Demand Unstable MMP13 20 40 COc1ccc(NC(=O)[C@@H](N[C@@H](c2ccccc2)C2CC2)c2ccccc2)cc1 ZINC000217561255 GK On-Demand Unstable CTSL 15 42 COc1ccc(NC(=O)[C@@H](N[C@@H](c2ccccc2)C2CC2)c2ccccc2)cc1 ZINC000217561255 GK On-Demand Unstable MTNR1B 15 40 COc1ccc(NC(=O)[C@@H](N[C@@H](c2ccccc2)C2CC2)c2ccccc2)cc1 ZINC000217561255 GK On-Demand Unstable MMP2 19 44 COc1ccc(NC(=O)[C@@H](N[C@@H](c2ccccc2)C2CC2)c2ccccc2)cc1 ZINC000217561255 GK On-Demand Unstable MMP9 15 44 Cn1c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c(O)c1CN1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217561268 KD In-Stock Unstable CHRNA4 28 47 C[C@H](C(=O)c1ccc(Cl)cc1)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217561278 DJ For-Sale Unstable SLC6A1 36 42 CC[C@@H](C)NS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217561294 EE In-Stock Unstable KCNQ2 65 38 CC[C@@H](C)NS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217561294 EE In-Stock Unstable TRY2_BOVIN 41 34 CC[C@@H](C)NS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217561294 EE In-Stock Unstable SLC6A9 24 45 COC(=O)CS[C@H]1CCN(C(=O)CCc2ccc(Cl)c(F)c2)C1 ZINC000217561304 FF In-Stock Unstable ENV 40 31 Cc1ccc(NC(=O)NCCc2ccc(Br)cc2)cn1 ZINC000217561335 EH On-Demand Unstable RAF1 28 41 Cc1ccc(NC(=O)NCCc2ccc(Br)cc2)cn1 ZINC000217561335 EH On-Demand Unstable Q8MMZ8_EIMTE 0 41 Cc1ccc(NC(=O)NCCc2ccc(Br)cc2)cn1 ZINC000217561335 EH On-Demand Unstable NAMPT 23 46 O=C1O[C@@]2(CCCN(C(=O)c3c(F)cccc3Cl)C2)c2ccccc21 ZINC000217561339 FH For-Sale Unstable NPY5R 33 46 Fc1ccc(Cl)cc1OC[C@@H]1CCCCN1 ZINC000217561341 BG For-Sale Unstable SSTR2 45 35 Fc1ccc(Cl)cc1OC[C@@H]1CCCCN1 ZINC000217561341 BG For-Sale Unstable LTA4H 17 60 Fc1ccc(Cl)cc1OC[C@@H]1CCCCN1 ZINC000217561341 BG For-Sale Unstable CHRNA2 29 44 Fc1ccc(Cl)cc1OC[C@@H]1CCCCN1 ZINC000217561341 BG For-Sale Unstable CHRNA3 18 45 Fc1ccc(Cl)cc1OC[C@@H]1CCCCN1 ZINC000217561341 BG For-Sale Unstable CHRNA10 63 58 COc1ccc(NC(=O)[C@H](N[C@@H](c2ccccc2)C2CC2)c2ccccc2)cc1 ZINC000217561348 GK On-Demand Unstable MMP13 20 40 COc1ccc(NC(=O)[C@H](N[C@@H](c2ccccc2)C2CC2)c2ccccc2)cc1 ZINC000217561348 GK On-Demand Unstable CTSL 15 42 COc1ccc(NC(=O)[C@H](N[C@@H](c2ccccc2)C2CC2)c2ccccc2)cc1 ZINC000217561348 GK On-Demand Unstable MTNR1B 15 40 COc1ccc(NC(=O)[C@H](N[C@@H](c2ccccc2)C2CC2)c2ccccc2)cc1 ZINC000217561348 GK On-Demand Unstable MMP2 19 44 COc1ccc(NC(=O)[C@H](N[C@@H](c2ccccc2)C2CC2)c2ccccc2)cc1 ZINC000217561348 GK On-Demand Unstable MMP9 15 44 C[C@@H](C(=O)c1ccc(Cl)cc1)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217561371 DJ For-Sale Unstable SLC6A1 36 42 CC[C@H](C)NS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217561380 EE In-Stock Unstable KCNQ2 65 38 CC[C@H](C)NS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217561380 EE In-Stock Unstable TRY2_BOVIN 41 34 CC[C@H](C)NS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217561380 EE In-Stock Unstable SLC6A9 24 45 O=C1O[C@]2(CCCN(C(=O)c3c(F)cccc3Cl)C2)c2ccccc21 ZINC000217561409 FH For-Sale Unstable NPY5R 33 46 Fc1ccc(Cl)cc1OC[C@H]1CCCCN1 ZINC000217561412 BG For-Sale Unstable SSTR2 45 35 Fc1ccc(Cl)cc1OC[C@H]1CCCCN1 ZINC000217561412 BG For-Sale Unstable LTA4H 17 60 Fc1ccc(Cl)cc1OC[C@H]1CCCCN1 ZINC000217561412 BG For-Sale Unstable CHRNA2 29 44 Fc1ccc(Cl)cc1OC[C@H]1CCCCN1 ZINC000217561412 BG For-Sale Unstable CHRNA3 18 45 Fc1ccc(Cl)cc1OC[C@H]1CCCCN1 ZINC000217561412 BG For-Sale Unstable CHRNA10 63 58 Cn1c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c(O)c1CN1CCO[C@H](c2ccccc2)C1 ZINC000217561427 KE In-Stock Unstable CHRNA4 36 48 COc1ccc(NC(=O)[C@@H](N[C@H](c2ccccc2)C2CC2)c2ccccc2)cc1 ZINC000217561437 GK On-Demand Unstable MMP13 20 40 COc1ccc(NC(=O)[C@@H](N[C@H](c2ccccc2)C2CC2)c2ccccc2)cc1 ZINC000217561437 GK On-Demand Unstable CTSL 15 42 COc1ccc(NC(=O)[C@@H](N[C@H](c2ccccc2)C2CC2)c2ccccc2)cc1 ZINC000217561437 GK On-Demand Unstable MTNR1B 15 40 COc1ccc(NC(=O)[C@@H](N[C@H](c2ccccc2)C2CC2)c2ccccc2)cc1 ZINC000217561437 GK On-Demand Unstable MMP2 19 44 COc1ccc(NC(=O)[C@@H](N[C@H](c2ccccc2)C2CC2)c2ccccc2)cc1 ZINC000217561437 GK On-Demand Unstable MMP9 15 44 O[C@H](c1ccccc1)c1cc2n(n1)CCN(c1ncnc3[nH]ccc13)C2 ZINC000217561468 EE In-Stock Unstable AKT2 42 42 O[C@H](c1ccccc1)c1cc2n(n1)CCN(c1ncnc3[nH]ccc13)C2 ZINC000217561468 EE In-Stock Unstable AKT3 35 46 O[C@H](c1ccccc1)c1cc2n(n1)CCN(c1ncnc3[nH]ccc13)C2 ZINC000217561468 EE In-Stock Unstable ROCK2 41 46 O[C@H](c1ccccc1)c1cc2n(n1)CCN(c1ncnc3[nH]ccc13)C2 ZINC000217561468 EE In-Stock Unstable AKT1 26 43 CC[C@@H](C)NS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1 ZINC000217561500 ED In-Stock Unstable MMP13 24 40 CC[C@@H](C)NS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1 ZINC000217561500 ED In-Stock Unstable SLC6A9 28 48 CC[C@@H](C)NS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1 ZINC000217561500 ED In-Stock Unstable MMP12 49 47 O=C(/C=C\c1cccnc1)N[C@@H]1CC[C@H](C(=O)O)C1 ZINC000217561523 CD On-Demand Unstable C3AR1 32 46 COc1ccc(-c2ccc3nnc([C@@H]4CCCNC4)n3n2)cc1 ZINC000217561531 DE In-Stock Unstable PDE4D 15 40 COc1ccc(-c2ccc3nnc([C@@H]4CCCNC4)n3n2)cc1 ZINC000217561531 DE In-Stock Unstable LRRK2 23 44 COc1ccc(NC(=O)[C@H](N[C@H](c2ccccc2)C2CC2)c2ccccc2)cc1 ZINC000217561536 GK On-Demand Unstable MMP13 20 40 COc1ccc(NC(=O)[C@H](N[C@H](c2ccccc2)C2CC2)c2ccccc2)cc1 ZINC000217561536 GK On-Demand Unstable CTSL 15 42 COc1ccc(NC(=O)[C@H](N[C@H](c2ccccc2)C2CC2)c2ccccc2)cc1 ZINC000217561536 GK On-Demand Unstable MTNR1B 15 40 COc1ccc(NC(=O)[C@H](N[C@H](c2ccccc2)C2CC2)c2ccccc2)cc1 ZINC000217561536 GK On-Demand Unstable MMP2 19 44 COc1ccc(NC(=O)[C@H](N[C@H](c2ccccc2)C2CC2)c2ccccc2)cc1 ZINC000217561536 GK On-Demand Unstable MMP9 15 44 Cn1c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c(O)c1CN1CCn2c(nnc2C(F)(F)F)C1 ZINC000217561543 KD In-Stock Unstable CHRNA4 27 44 O=C(NCCc1ccc(Br)cc1)Nc1ncc(Br)cn1 ZINC000217561558 HG For-Sale Unstable LIG1 0 40 O[C@@H](c1ccccc1)c1cc2n(n1)CCN(c1ncnc3[nH]ccc13)C2 ZINC000217561564 EE In-Stock Unstable AKT2 42 42 O[C@@H](c1ccccc1)c1cc2n(n1)CCN(c1ncnc3[nH]ccc13)C2 ZINC000217561564 EE In-Stock Unstable AKT3 35 46 O[C@@H](c1ccccc1)c1cc2n(n1)CCN(c1ncnc3[nH]ccc13)C2 ZINC000217561564 EE In-Stock Unstable ROCK2 41 46 O[C@@H](c1ccccc1)c1cc2n(n1)CCN(c1ncnc3[nH]ccc13)C2 ZINC000217561564 EE In-Stock Unstable AKT1 26 43 CC[C@H](C)NS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1 ZINC000217561578 ED In-Stock Unstable MMP13 24 40 CC[C@H](C)NS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1 ZINC000217561578 ED In-Stock Unstable SLC6A9 28 48 CC[C@H](C)NS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1 ZINC000217561578 ED In-Stock Unstable MMP12 49 47 COc1ccc(-c2ccc3nnc([C@H]4CCCNC4)n3n2)cc1 ZINC000217561634 DE In-Stock Unstable PDE4D 15 40 COc1ccc(-c2ccc3nnc([C@H]4CCCNC4)n3n2)cc1 ZINC000217561634 DE In-Stock Unstable LRRK2 23 44 Cn1c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c(O)c1CN1CC=C(c2ccc(F)cc2)CC1 ZINC000217561641 KG In-Stock Unstable CHRNA4 36 51 O=C(CN1CCC[C@@H]2CCCC[C@H]21)c1ccccc1Br ZINC000217561693 EI For-Sale Unstable SLC18A3 21 40 Fc1cc(Cl)ccc1OC[C@@H]1CCCCN1 ZINC000217561725 BG For-Sale Unstable SSTR2 55 35 Fc1cc(Cl)ccc1OC[C@@H]1CCCCN1 ZINC000217561725 BG For-Sale Unstable LTA4H 18 59 Fc1cc(Cl)ccc1OC[C@@H]1CCCCN1 ZINC000217561725 BG For-Sale Unstable CHRNA2 28 43 Fc1cc(Cl)ccc1OC[C@@H]1CCCCN1 ZINC000217561725 BG For-Sale Unstable CHRNA3 18 44 Fc1cc(Cl)ccc1OC[C@@H]1CCCCN1 ZINC000217561725 BG For-Sale Unstable CHRNA10 69 57 O=C1O[C@@]2(CCCN(C(=O)c3cc(-c4ccco4)on3)C2)c2ccccc21 ZINC000217561744 FG For-Sale Unstable NPY5R 29 45 COC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](N)C(C)C ZINC000217561748 DB On-Demand Unstable FOLH1 51 41 COC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](N)C(C)C ZINC000217561748 DB On-Demand Unstable ANPEP 40 36 COC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](N)C(C)C ZINC000217561748 DB On-Demand Unstable CTSK 16 40 COC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](N)C(C)C ZINC000217561748 DB On-Demand Unstable PGA 43 36 COC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](N)C(C)C ZINC000217561748 DB On-Demand Unstable HLA-A 54 52 COC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](N)C(C)C ZINC000217561748 DB On-Demand Unstable CTSS 15 40 COC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](N)C(C)C ZINC000217561748 DB On-Demand Unstable CAPN2 61 33 COC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](N)C(C)C ZINC000217561748 DB On-Demand Unstable NPR 47 46 COC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](N)C(C)C ZINC000217561748 DB On-Demand Unstable F2RL1 51 32 COc1ccc(-c2ccc3nnc([C@@H]4CCCNC4)n3n2)cc1OC ZINC000217561750 EE In-Stock Unstable PDE4D 49 42 COc1ccc(-c2ccc3nnc([C@@H]4CCCNC4)n3n2)cc1OC ZINC000217561750 EE In-Stock Unstable LRRK2 27 44 COc1ccccc1N1CCN(Cc2c(O)c(=O)cc(CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)n2C)CC1 ZINC000217561753 KE In-Stock Unstable HTR1A 88 44 COc1ccccc1N1CCN(Cc2c(O)c(=O)cc(CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)n2C)CC1 ZINC000217561753 KE In-Stock Unstable DRD2 61 44 COc1ccccc1N1CCN(Cc2c(O)c(=O)cc(CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)n2C)CC1 ZINC000217561753 KE In-Stock Unstable DRD1 32 40 COc1ccccc1N1CCN(Cc2c(O)c(=O)cc(CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)n2C)CC1 ZINC000217561753 KE In-Stock Unstable ADRA1D 54 41 COc1ccccc1N1CCN(Cc2c(O)c(=O)cc(CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)n2C)CC1 ZINC000217561753 KE In-Stock Unstable HTR2A 31 40 COc1ccccc1N1CCN(Cc2c(O)c(=O)cc(CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)n2C)CC1 ZINC000217561753 KE In-Stock Unstable ADRA1A 51 41 COc1ccccc1N1CCN(Cc2c(O)c(=O)cc(CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)n2C)CC1 ZINC000217561753 KE In-Stock Unstable ADRA1B 43 41 COc1ccccc1N1CCN(Cc2c(O)c(=O)cc(CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)n2C)CC1 ZINC000217561753 KE In-Stock Unstable DRD3 60 40 COc1ccccc1N1CCN(Cc2c(O)c(=O)cc(CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)n2C)CC1 ZINC000217561753 KE In-Stock Unstable HTR7 51 40 COc1ccccc1N1CCN(Cc2c(O)c(=O)cc(CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)n2C)CC1 ZINC000217561753 KE In-Stock Unstable CHRNA4 35 45 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Cl)cn1 ZINC000217561773 FH On-Demand Unstable KLKB1 30 40 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Cl)cn1 ZINC000217561773 FH On-Demand Unstable F10 46 30 O=C(NCCc1ccc(Br)cc1)Nc1ccc(Cl)cn1 ZINC000217561773 FH On-Demand Unstable POL 0 63 O=C(CN1CCC[C@H]2CCCC[C@H]21)c1ccccc1Br ZINC000217561775 EI For-Sale Unstable SLC18A3 21 40 Fc1cc(Cl)ccc1OC[C@H]1CCCCN1 ZINC000217561799 BG For-Sale Unstable SSTR2 55 35 Fc1cc(Cl)ccc1OC[C@H]1CCCCN1 ZINC000217561799 BG For-Sale Unstable LTA4H 18 59 Fc1cc(Cl)ccc1OC[C@H]1CCCCN1 ZINC000217561799 BG For-Sale Unstable CHRNA2 28 43 Fc1cc(Cl)ccc1OC[C@H]1CCCCN1 ZINC000217561799 BG For-Sale Unstable CHRNA3 18 44 Fc1cc(Cl)ccc1OC[C@H]1CCCCN1 ZINC000217561799 BG For-Sale Unstable CHRNA10 69 57 COC(=O)[C@@H](CC(C)C)NC(=O)CNC(=O)[C@H](N)C(C)C ZINC000217561813 DB On-Demand Unstable FOLH1 51 41 COC(=O)[C@@H](CC(C)C)NC(=O)CNC(=O)[C@H](N)C(C)C ZINC000217561813 DB On-Demand Unstable ANPEP 40 36 COC(=O)[C@@H](CC(C)C)NC(=O)CNC(=O)[C@H](N)C(C)C ZINC000217561813 DB On-Demand Unstable CTSK 16 40 COC(=O)[C@@H](CC(C)C)NC(=O)CNC(=O)[C@H](N)C(C)C ZINC000217561813 DB On-Demand Unstable PGA 43 36 COC(=O)[C@@H](CC(C)C)NC(=O)CNC(=O)[C@H](N)C(C)C ZINC000217561813 DB On-Demand Unstable HLA-A 54 52 COC(=O)[C@@H](CC(C)C)NC(=O)CNC(=O)[C@H](N)C(C)C ZINC000217561813 DB On-Demand Unstable CTSS 15 40 COC(=O)[C@@H](CC(C)C)NC(=O)CNC(=O)[C@H](N)C(C)C ZINC000217561813 DB On-Demand Unstable CAPN2 61 33 COC(=O)[C@@H](CC(C)C)NC(=O)CNC(=O)[C@H](N)C(C)C ZINC000217561813 DB On-Demand Unstable NPR 47 46 COC(=O)[C@@H](CC(C)C)NC(=O)CNC(=O)[C@H](N)C(C)C ZINC000217561813 DB On-Demand Unstable F2RL1 51 32 O=C1O[C@]2(CCCN(C(=O)c3cc(-c4ccco4)on3)C2)c2ccccc21 ZINC000217561826 FG For-Sale Unstable NPY5R 29 45 COc1ccc(-c2ccc3nnc([C@H]4CCCNC4)n3n2)cc1OC ZINC000217561832 EE In-Stock Unstable PDE4D 49 42 COc1ccc(-c2ccc3nnc([C@H]4CCCNC4)n3n2)cc1OC ZINC000217561832 EE In-Stock Unstable LRRK2 27 44 COc1ccccc1C(=O)CN1CCC[C@@H]2CCCC[C@H]21 ZINC000217561887 CH For-Sale Unstable HTR1A 39 42 COc1ccccc1C(=O)CN1CCC[C@@H]2CCCC[C@H]21 ZINC000217561887 CH For-Sale Unstable DRD2 43 36 COc1ccccc1C(=O)CN1CCC[C@@H]2CCCC[C@H]21 ZINC000217561887 CH For-Sale Unstable SLC6A1 26 41 COc1ccccc1C(=O)CN1CCC[C@@H]2CCCC[C@H]21 ZINC000217561887 CH For-Sale Unstable KCNA3 40 37 COc1ccccc1C(=O)CN1CCC[C@@H]2CCCC[C@H]21 ZINC000217561887 CH For-Sale Unstable HCN1 54 37 COc1ccccc1C(=O)CN1CCC[C@@H]2CCCC[C@H]21 ZINC000217561887 CH For-Sale Unstable HCN4 51 35 COc1ccccc1C(=O)CN1CCC[C@@H]2CCCC[C@H]21 ZINC000217561887 CH For-Sale Unstable ACKR3 61 31 O=C(c1ccc(F)cc1)[C@H]1[C@H]2C(=O)N(c3ccccc3)C(=O)[C@@H]2[C@H]2CCCN21 ZINC000217561903 GF In-Stock Unstable SLC18A3 25 40 CC(=O)N1CCc2cc(C(=O)CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)ccc21 ZINC000217561913 GE In-Stock Unstable CHRNA4 31 61 O=C1O[C@@]2(CCCN(C(=O)c3nc4ccccc4s3)C2)c2ccccc21 ZINC000217561919 FH In-Stock Unstable NPY5R 30 42 COc1cc2c(cc1OC)[C@@H]1C/C(=N/N=C3/C[C@@H]4c5cc(OC)c(OC)cc5CCN4C[C@@H]3CC(C)C)[C@@H](CC(C)C)CN1CC2 ZINC000217561946 KK In-Stock Unstable DRD1 24 52 COc1cc2c(cc1OC)[C@@H]1C/C(=N/N=C3/C[C@@H]4c5cc(OC)c(OC)cc5CCN4C[C@@H]3CC(C)C)[C@@H](CC(C)C)CN1CC2 ZINC000217561946 KK In-Stock Unstable SLC18A2 85 74 COc1cc2c(cc1OC)[C@@H]1C/C(=N/N=C3/C[C@@H]4c5cc(OC)c(OC)cc5CCN4C[C@@H]3CC(C)C)[C@@H](CC(C)C)CN1CC2 ZINC000217561946 KK In-Stock Unstable DPP4 28 47 COc1cc2c(cc1OC)[C@@H]1C/C(=N/N=C3/C[C@@H]4c5cc(OC)c(OC)cc5CCN4C[C@@H]3CC(C)C)[C@@H](CC(C)C)CN1CC2 ZINC000217561946 KK In-Stock Unstable F3 31 50 COc1cc2c(cc1OC)[C@@H]1C/C(=N/N=C3/C[C@@H]4c5cc(OC)c(OC)cc5CCN4C[C@@H]3CC(C)C)[C@@H](CC(C)C)CN1CC2 ZINC000217561946 KK In-Stock Unstable SLC2A1 16 45 COc1cc2c(cc1OC)[C@@H]1C/C(=N/N=C3/C[C@@H]4c5cc(OC)c(OC)cc5CCN4C[C@@H]3CC(C)C)[C@@H](CC(C)C)CN1CC2 ZINC000217561946 KK In-Stock Unstable RBBP9 0 45 COc1ccc(OC)c(-c2ccc3nnc([C@@H]4CCCNC4)n3n2)c1 ZINC000217561953 EE In-Stock Unstable LRRK2 36 54 CCCCCCCCCCNC[C@@H](C)N(C)C1CC1 ZINC000217561954 CI For-Sale Unstable Q8WS26_TRYCR 33 41 O=C(c1ccc(F)cc1)[C@@H]1[C@H]2C(=O)N(c3ccccc3)C(=O)[C@@H]2[C@H]2CCCN12 ZINC000217561975 GF In-Stock Unstable SLC18A3 25 40 COc1ccccc1C(=O)CN1CCC[C@H]2CCCC[C@H]21 ZINC000217561984 CH For-Sale Unstable HTR1A 39 42 COc1ccccc1C(=O)CN1CCC[C@H]2CCCC[C@H]21 ZINC000217561984 CH For-Sale Unstable DRD2 43 36 COc1ccccc1C(=O)CN1CCC[C@H]2CCCC[C@H]21 ZINC000217561984 CH For-Sale Unstable SLC6A1 26 41 COc1ccccc1C(=O)CN1CCC[C@H]2CCCC[C@H]21 ZINC000217561984 CH For-Sale Unstable KCNA3 40 37 COc1ccccc1C(=O)CN1CCC[C@H]2CCCC[C@H]21 ZINC000217561984 CH For-Sale Unstable HCN1 54 37 COc1ccccc1C(=O)CN1CCC[C@H]2CCCC[C@H]21 ZINC000217561984 CH For-Sale Unstable HCN4 51 35 COc1ccccc1C(=O)CN1CCC[C@H]2CCCC[C@H]21 ZINC000217561984 CH For-Sale Unstable ACKR3 61 31 O=C1O[C@]2(CCCN(C(=O)c3nc4ccccc4s3)C2)c2ccccc21 ZINC000217561999 FH In-Stock Unstable NPY5R 30 42 Cc1c(Cl)nc(C2CC2)nc1N[C@@H]1CC[C@@H](C)[C@@H](C)C1 ZINC000217562014 CJ For-Sale Unstable CHRM3 18 47 COc1ccc(OC)c(-c2ccc3nnc([C@H]4CCCNC4)n3n2)c1 ZINC000217562046 EE In-Stock Unstable LRRK2 36 54 CCCCCCCCCCNC[C@H](C)N(C)C1CC1 ZINC000217562056 CI For-Sale Unstable Q8WS26_TRYCR 33 41 COC(=O)CS[C@H]1CCN(C(=O)Cc2ccc(NC(C)=O)cc2)C1 ZINC000217562061 FD In-Stock Unstable MLNR 30 41 CCCCCNc1ccc(S(=O)(=O)N[C@@H](C)CC)cc1C(=O)O ZINC000217562062 EG In-Stock Unstable CASP3 0 41 CCCCCNc1ccc(S(=O)(=O)N[C@@H](C)CC)cc1C(=O)O ZINC000217562062 EG In-Stock Unstable LEF 44 37 Cc1cc(/C=C\C(=O)O)cc(C)c1OCCCCC#N ZINC000217562074 CG For-Sale Unstable PTGER2 0 40 CC1CCN(Cc2c(O)c(=O)cc(CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)n2C)CC1 ZINC000217562087 IE In-Stock Unstable CHRNA4 30 49 O=C(NCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562099 FH On-Demand Unstable HRH2 17 40 O=C(NCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562099 FH On-Demand Unstable SIGMAR1 15 42 O=C(NCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562099 FH On-Demand Unstable HDAC8 16 50 O=C(NCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562099 FH On-Demand Unstable CA5B 20 43 O=C(NCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562099 FH On-Demand Unstable CA5A 19 43 O=C(NCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562099 FH On-Demand Unstable MTNR1A 24 43 O=C(NCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562099 FH On-Demand Unstable MTNR1B 42 43 O=C(NCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562099 FH On-Demand Unstable MMP3 21 41 O=C(NCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562099 FH On-Demand Unstable FAAH 26 40 O=C(NCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562099 FH On-Demand Unstable SCN5A 0 42 O=C(NCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562099 FH On-Demand Unstable AMP1_PLAFQ 43 50 O=C(NCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562099 FH On-Demand Unstable NCE103 27 45 O=C(NCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562099 FH On-Demand Unstable CRTM 45 46 O=C(NCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562099 FH On-Demand Unstable P96878_MYCTU 15 43 COC(=O)c1ccc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217562107 FF For-Sale Unstable NPY5R 32 51 Cc1c(Cl)nc(C2CC2)nc1N[C@H]1CC[C@@H](C)[C@@H](C)C1 ZINC000217562114 CJ For-Sale Unstable CHRM3 18 47 COC(=O)CS[C@@H]1CCN(C(=O)Cc2ccc(NC(C)=O)cc2)C1 ZINC000217562131 FD In-Stock Unstable MLNR 30 41 CCCCCNc1ccc(S(=O)(=O)N[C@H](C)CC)cc1C(=O)O ZINC000217562152 EG In-Stock Unstable CASP3 0 41 CCCCCNc1ccc(S(=O)(=O)N[C@H](C)CC)cc1C(=O)O ZINC000217562152 EG In-Stock Unstable LEF 44 37 COc1ccc(OC)c(-c2ccc3nnc([C@@H]4CCCCN4)n3n2)c1 ZINC000217562161 EF In-Stock Unstable LRRK2 35 50 COC(=O)c1ccc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217562178 FF For-Sale Unstable NPY5R 32 51 Cc1c(Cl)nc(C2CC2)nc1N[C@@H]1CC[C@H](C)[C@@H](C)C1 ZINC000217562200 CJ For-Sale Unstable CHRM3 18 47 O=C(NCCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562216 GI For-Sale Unstable HRH2 15 41 O=C(NCCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562216 GI For-Sale Unstable SCNN1A 53 39 O=C(NCCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562216 GI For-Sale Unstable SDH1 0 47 O=C(NCCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562216 GI For-Sale Unstable CA1 15 49 O=C(NCCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562216 GI For-Sale Unstable SIGMAR1 18 47 O=C(NCCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562216 GI For-Sale Unstable SCN2A 22 42 O=C(NCCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562216 GI For-Sale Unstable HDAC8 15 49 O=C(NCCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562216 GI For-Sale Unstable CA5B 16 43 O=C(NCCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562216 GI For-Sale Unstable CA5A 15 49 O=C(NCCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562216 GI For-Sale Unstable MTNR1A 26 42 O=C(NCCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562216 GI For-Sale Unstable MTNR1B 27 42 O=C(NCCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562216 GI For-Sale Unstable MMP2 18 43 O=C(NCCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562216 GI For-Sale Unstable MMP3 25 42 O=C(NCCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562216 GI For-Sale Unstable HDAC1 15 45 O=C(NCCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562216 GI For-Sale Unstable FAAH 51 45 O=C(NCCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562216 GI For-Sale Unstable SCN5A 0 44 O=C(NCCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562216 GI For-Sale Unstable S1PR2 23 42 O=C(NCCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562216 GI For-Sale Unstable SLC6A5 29 47 O=C(NCCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562216 GI For-Sale Unstable CES1 58 39 O=C(NCCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562216 GI For-Sale Unstable HDAC9 20 41 O=C(NCCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562216 GI For-Sale Unstable AMP1_PLAFQ 39 51 O=C(NCCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562216 GI For-Sale Unstable HDA106 0 42 O=C(NCCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562216 GI For-Sale Unstable CRTM 30 42 O=C(NCCCCc1ccccc1)NCCc1ccc(Br)cc1 ZINC000217562216 GI For-Sale Unstable LIG1 0 43 COC(=O)CS[C@H]1CCN(C(=O)c2ccc(NC(C)=O)cc2)C1 ZINC000217562224 ED In-Stock Unstable AVPR1A 41 36 COC(=O)CS[C@H]1CCN(C(=O)c2ccc(NC(C)=O)cc2)C1 ZINC000217562224 ED In-Stock Unstable L3MBTL3 59 37 COc1ccc(C(=O)CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc1 ZINC000217562225 EE In-Stock Unstable CHRNA4 47 76 CC[C@@H](C)NS(=O)(=O)c1ccc(NCCC(C)C)c(C(=O)O)c1 ZINC000217562248 EF In-Stock Unstable LEF 49 36 COc1ccc(OC)c(-c2ccc3nnc([C@H]4CCCCN4)n3n2)c1 ZINC000217562249 EF In-Stock Unstable LRRK2 35 50 O=C(/C=C\c1cccc(Cl)c1)N[C@@H]1CC[C@H](C(=O)O)C1 ZINC000217562280 CF On-Demand Unstable TUBA4A 0 45 Cc1c(Cl)nc(C2CC2)nc1N[C@H]1CC[C@H](C)[C@@H](C)C1 ZINC000217562281 CJ For-Sale Unstable CHRM3 18 47 O=C1O[C@@]2(CCCN(C(=O)c3ccc4nsnc4c3)C2)c2ccccc21 ZINC000217562292 FF For-Sale Unstable NPY5R 30 42 COC(=O)CS[C@@H]1CCN(C(=O)c2ccc(NC(C)=O)cc2)C1 ZINC000217562316 ED In-Stock Unstable AVPR1A 41 36 COC(=O)CS[C@@H]1CCN(C(=O)c2ccc(NC(C)=O)cc2)C1 ZINC000217562316 ED In-Stock Unstable L3MBTL3 59 37 O=c1[nH]c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)nc2sc(-c3ccccc3)cc12 ZINC000217562324 IG In-Stock Unstable CHRNA4 31 55 CC[C@H](C)NS(=O)(=O)c1ccc(NCCC(C)C)c(C(=O)O)c1 ZINC000217562325 EF In-Stock Unstable LEF 49 36 COc1ccc(-c2ccc3nnc([C@@H]4CCCCN4)n3n2)cc1OC ZINC000217562375 EF In-Stock Unstable PDE4D 50 43 COc1ccc(-c2ccc3nnc([C@@H]4CCCCN4)n3n2)cc1OC ZINC000217562375 EF In-Stock Unstable LRRK2 27 41 O=C1O[C@]2(CCCN(C(=O)c3ccc4nsnc4c3)C2)c2ccccc21 ZINC000217562376 FF For-Sale Unstable NPY5R 30 42 CCC[C@@H](C)Nc1ccc(S(=O)(=O)N[C@@H](C)CC)cc1C(=O)O ZINC000217562429 EG In-Stock Unstable LEF 52 37 N#CCCNC(=O)NCCc1ccc(Br)cc1 ZINC000217562436 CE On-Demand Unstable LIG1 0 41 COc1ccc(-c2ccc3nnc([C@H]4CCCCN4)n3n2)cc1OC ZINC000217562443 EF In-Stock Unstable PDE4D 50 43 COc1ccc(-c2ccc3nnc([C@H]4CCCCN4)n3n2)cc1OC ZINC000217562443 EF In-Stock Unstable LRRK2 27 41 CC(C)(O)CN1CCC(COc2ccc(Cl)nc2)CC1 ZINC000217562472 CF On-Demand Unstable SIGMAR1 19 46 CC(C)(O)CN1CCC(COc2ccc(Cl)nc2)CC1 ZINC000217562472 CF On-Demand Unstable CHRNA4 29 47 COc1cccc(C(=O)CN2CCC[C@@H]3CCCC[C@H]32)c1 ZINC000217562473 CH For-Sale Unstable DRD2 17 44 COc1cccc(C(=O)CN2CCC[C@@H]3CCCC[C@H]32)c1 ZINC000217562473 CH For-Sale Unstable DRD4 49 37 COc1cccc(C(=O)CN2CCC[C@@H]3CCCC[C@H]32)c1 ZINC000217562473 CH For-Sale Unstable SIGMAR1 20 47 COc1cccc(C(=O)CN2CCC[C@@H]3CCCC[C@H]32)c1 ZINC000217562473 CH For-Sale Unstable MTNR1B 36 41 COc1cccc(C(=O)CN2CCC[C@@H]3CCCC[C@H]32)c1 ZINC000217562473 CH For-Sale Unstable CHRNA10 31 41 COc1cccc(C(=O)CN2CCC[C@@H]3CCCC[C@H]32)c1 ZINC000217562473 CH For-Sale Unstable ACKR3 51 31 CC(=O)Nc1cc(C(=O)NCc2ccccc2)ccc1N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217562478 JG In-Stock Unstable CHRNA4 28 48 CC(C)Oc1ccc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217562486 FH For-Sale Unstable CHRM5 24 48 CC(C)Oc1ccc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217562486 FH For-Sale Unstable NPY5R 25 41 CCC[C@H](C)Nc1ccc(S(=O)(=O)N[C@@H](C)CC)cc1C(=O)O ZINC000217562529 EG In-Stock Unstable LEF 52 37 C[C@@H](N)c1ccc(Br)cc1N1CC[C@@H](N2CCCC2)C1 ZINC000217562530 EG For-Sale Unstable L3MBTL3 72 38 C[C@@H](N)c1ccc(Br)cc1N1CC[C@@H](N2CCCC2)C1 ZINC000217562530 EG For-Sale Unstable MBTD1 0 43 O=C(NCCc1ccc(Br)cc1)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217562544 JF For-Sale Unstable CA1 15 40 O=C(NCCc1ccc(Br)cc1)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217562544 JF For-Sale Unstable CA5B 16 40 O=C(NCCc1ccc(Br)cc1)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217562544 JF For-Sale Unstable MMP3 19 50 O=C(NCCc1ccc(Br)cc1)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217562544 JF For-Sale Unstable TGM2 76 44 O=C(NCCc1ccc(Br)cc1)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217562544 JF For-Sale Unstable MMP7 17 50 O=C(NCCc1ccc(Br)cc1)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217562544 JF For-Sale Unstable F13A1 86 44 O=C(NCCc1ccc(Br)cc1)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217562544 JF For-Sale Unstable LIG1 0 43 O=C(NCCc1ccc(Br)cc1)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217562544 JF For-Sale Unstable NAMPT 43 40 O=C(NCCc1ccc(Br)cc1)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217562544 JF For-Sale Unstable HPN 32 41 COc1cccc(C(=O)CN2CCC[C@H]3CCCC[C@H]32)c1 ZINC000217562562 CH For-Sale Unstable DRD2 17 44 COc1cccc(C(=O)CN2CCC[C@H]3CCCC[C@H]32)c1 ZINC000217562562 CH For-Sale Unstable DRD4 49 37 COc1cccc(C(=O)CN2CCC[C@H]3CCCC[C@H]32)c1 ZINC000217562562 CH For-Sale Unstable SIGMAR1 20 47 COc1cccc(C(=O)CN2CCC[C@H]3CCCC[C@H]32)c1 ZINC000217562562 CH For-Sale Unstable MTNR1B 36 41 COc1cccc(C(=O)CN2CCC[C@H]3CCCC[C@H]32)c1 ZINC000217562562 CH For-Sale Unstable CHRNA10 31 41 COc1cccc(C(=O)CN2CCC[C@H]3CCCC[C@H]32)c1 ZINC000217562562 CH For-Sale Unstable ACKR3 51 31 COc1ccc(-c2ccc3nnc([C@@H]4CCCCN4)n3n2)cc1 ZINC000217562568 DF In-Stock Unstable PDE4D 15 43 COc1ccc(-c2ccc3nnc([C@@H]4CCCCN4)n3n2)cc1 ZINC000217562568 DF In-Stock Unstable LRRK2 25 40 CC(C)Oc1ccc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217562578 FH For-Sale Unstable CHRM5 24 48 CC(C)Oc1ccc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217562578 FH For-Sale Unstable NPY5R 25 41 COC(=O)CS[C@@H]1CCN(C(=O)c2cc(-c3ccccc3)n[nH]2)C1 ZINC000217562601 EE In-Stock Unstable TACR3 25 52 C[C@H](N)c1ccc(Br)cc1N1CC[C@@H](N2CCCC2)C1 ZINC000217562606 EG For-Sale Unstable L3MBTL3 72 38 C[C@H](N)c1ccc(Br)cc1N1CC[C@@H](N2CCCC2)C1 ZINC000217562606 EG For-Sale Unstable MBTD1 0 43 CCC[C@@H](C)Nc1ccc(S(=O)(=O)N[C@H](C)CC)cc1C(=O)O ZINC000217562610 EG In-Stock Unstable LEF 52 37 Cn1c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c(O)c1CN1CCOCC1 ZINC000217562614 IC In-Stock Unstable CHRNA4 30 49 Cn1c(=O)[nH]cc(CC(=O)NCc2nc3ccc(Cl)cc3[nH]2)c1=O ZINC000217562615 EC In-Stock Unstable NAMPT 0 40 CCOc1cc(/C=C\C(=O)O)ccc1OCCCCC#N ZINC000217562620 CG For-Sale Unstable APP 19 41 CCOc1cc(/C=C\C(=O)O)ccc1OCCCCC#N ZINC000217562620 CG For-Sale Unstable AKR1C3 36 55 COc1ccc(-c2ccc3nnc([C@H]4CCCCN4)n3n2)cc1 ZINC000217562638 DF In-Stock Unstable PDE4D 15 43 COc1ccc(-c2ccc3nnc([C@H]4CCCCN4)n3n2)cc1 ZINC000217562638 DF In-Stock Unstable LRRK2 25 40 Cc1ccc(S(=O)(=O)N2CCN(C(=O)NCCc3ccc(Br)cc3)CC2)cc1 ZINC000217562651 JG For-Sale Unstable CA1 16 43 Cc1ccc(S(=O)(=O)N2CCN(C(=O)NCCc3ccc(Br)cc3)CC2)cc1 ZINC000217562651 JG For-Sale Unstable MMP3 23 46 Cc1ccc(S(=O)(=O)N2CCN(C(=O)NCCc3ccc(Br)cc3)CC2)cc1 ZINC000217562651 JG For-Sale Unstable TGM2 68 40 Cc1ccc(S(=O)(=O)N2CCN(C(=O)NCCc3ccc(Br)cc3)CC2)cc1 ZINC000217562651 JG For-Sale Unstable MMP7 25 46 Cc1ccc(S(=O)(=O)N2CCN(C(=O)NCCc3ccc(Br)cc3)CC2)cc1 ZINC000217562651 JG For-Sale Unstable MMP1 19 46 Cc1ccc(S(=O)(=O)N2CCN(C(=O)NCCc3ccc(Br)cc3)CC2)cc1 ZINC000217562651 JG For-Sale Unstable F13A1 76 40 Cc1ccc(S(=O)(=O)N2CCN(C(=O)NCCc3ccc(Br)cc3)CC2)cc1 ZINC000217562651 JG For-Sale Unstable LIG1 0 44 Cc1ccc(S(=O)(=O)N2CCN(C(=O)NCCc3ccc(Br)cc3)CC2)cc1 ZINC000217562651 JG For-Sale Unstable NAMPT 44 43 Cc1ccc(S(=O)(=O)N2CCN(C(=O)NCCc3ccc(Br)cc3)CC2)cc1 ZINC000217562651 JG For-Sale Unstable HPN 23 45 O=C(/C=C\c1ccccc1)N[C@@H]1CC[C@H](C(=O)O)C1 ZINC000217562665 CE On-Demand Unstable HDAC8 47 40 O=C(/C=C\c1ccccc1)N[C@@H]1CC[C@H](C(=O)O)C1 ZINC000217562665 CE On-Demand Unstable F3 24 43 O=C(/C=C\c1ccccc1)N[C@@H]1CC[C@H](C(=O)O)C1 ZINC000217562665 CE On-Demand Unstable MMP2 21 54 O=C(/C=C\c1ccccc1)N[C@@H]1CC[C@H](C(=O)O)C1 ZINC000217562665 CE On-Demand Unstable HDAC6 31 51 O=C(/C=C\c1ccccc1)N[C@@H]1CC[C@H](C(=O)O)C1 ZINC000217562665 CE On-Demand Unstable FASN 39 40 O=C(/C=C\c1ccccc1)N[C@@H]1CC[C@H](C(=O)O)C1 ZINC000217562665 CE On-Demand Unstable MMP9 18 48 O=C(/C=C\c1ccccc1)N[C@@H]1CC[C@H](C(=O)O)C1 ZINC000217562665 CE On-Demand Unstable MMP1 18 45 O=C(CN1CCC[C@@H]2CCCC[C@H]21)c1ccccc1Cl ZINC000217562678 CI For-Sale Unstable SLC6A1 54 37 COC(=O)CS[C@H]1CCN(C(=O)c2cc(-c3ccccc3)n[nH]2)C1 ZINC000217562682 EE In-Stock Unstable TACR3 25 52 CN[C@@H](C)c1cc(Br)ccc1N1CC[C@@H](N2CCCC2)C1 ZINC000217562683 FG For-Sale Unstable MBTD1 0 42 CCC[C@H](C)Nc1ccc(S(=O)(=O)N[C@H](C)CC)cc1C(=O)O ZINC000217562686 EG In-Stock Unstable LEF 52 37 COc1ccc(CCC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217562693 FG For-Sale Unstable NPY5R 25 47 N#CCN(C(=O)c1cnn2ccccc12)C1CCCC1 ZINC000217562708 CE On-Demand Unstable JAK1 24 46 N#CCN(C(=O)c1cnn2ccccc12)C1CCCC1 ZINC000217562708 CE On-Demand Unstable TYK2 34 46 COc1ccc(S(=O)(=O)N2CCN(Cc3c(O)c(=O)cc(CN4C[C@@H]5C[C@H](C4)c4cccc(=O)n4C5)n3C)CC2)cc1 ZINC000217562730 KD In-Stock Unstable CHRNA4 27 43 CN[C@H](C)c1cc(Br)ccc1N1CC[C@@H](N2CCCC2)C1 ZINC000217562758 FG For-Sale Unstable MBTD1 0 42 O=C(CN1CCC[C@H]2CCCC[C@H]21)c1ccccc1Cl ZINC000217562765 CI For-Sale Unstable SLC6A1 54 37 COc1ccc(CCC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217562767 FG For-Sale Unstable NPY5R 25 47 CN[C@@H](C)c1ccc(Br)cc1N1CC[C@@H](N2CCCC2)C1 ZINC000217562835 FG For-Sale Unstable L3MBTL3 58 36 CN[C@@H](C)c1ccc(Br)cc1N1CC[C@@H](N2CCCC2)C1 ZINC000217562835 FG For-Sale Unstable MBTD1 0 42 O=C(Cn1cnc2ccccc2c1=O)NCCc1noc(C2CCCC2)n1 ZINC000217562862 FD In-Stock Unstable SMO 48 36 O=C(/C=C\c1ccccc1Cl)N[C@@H]1CC[C@H](C(=O)O)C1 ZINC000217562865 CF On-Demand Unstable KCNQ2 21 44 CCOc1ccc(CC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217562874 FG For-Sale Unstable NPY5R 24 41 O=C(CN1CCC[C@@H]2CCCC[C@H]21)c1cc(F)ccc1F ZINC000217562898 CH For-Sale Unstable SLC6A1 24 40 COc1cc(/C=C\C(=O)O)ccc1OCCCCC#N ZINC000217562911 CF For-Sale Unstable PTGER2 22 49 COc1cc(/C=C\C(=O)O)ccc1OCCCCC#N ZINC000217562911 CF For-Sale Unstable CYP1B1 23 40 COc1cc(/C=C\C(=O)O)ccc1OCCCCC#N ZINC000217562911 CF For-Sale Unstable LTB4R 43 36 COc1cc(/C=C\C(=O)O)ccc1OCCCCC#N ZINC000217562911 CF For-Sale Unstable APP 23 51 COc1cc(/C=C\C(=O)O)ccc1OCCCCC#N ZINC000217562911 CF For-Sale Unstable CYP1A1 24 40 COc1cc(/C=C\C(=O)O)ccc1OCCCCC#N ZINC000217562911 CF For-Sale Unstable TUBB1 55 39 COc1cc(/C=C\C(=O)O)ccc1OCCCCC#N ZINC000217562911 CF For-Sale Unstable AKR1C3 34 48 COc1cc(/C=C\C(=O)O)ccc1OCCCCC#N ZINC000217562911 CF For-Sale Unstable ABCG2 15 44 Cn1ccc(C(=O)N(CC#N)C2CCCC2)n1 ZINC000217562912 BD On-Demand Unstable ACE 42 37 CN[C@H](C)c1ccc(Br)cc1N1CC[C@@H](N2CCCC2)C1 ZINC000217562918 FG For-Sale Unstable L3MBTL3 58 36 CN[C@H](C)c1ccc(Br)cc1N1CC[C@@H](N2CCCC2)C1 ZINC000217562918 FG For-Sale Unstable MBTD1 0 42 COc1ccc(O)c(C(=O)O)c1Br ZINC000217562940 BD For-Sale Unstable APP 40 34 COc1ccc(O)c(C(=O)O)c1Br ZINC000217562940 BD For-Sale Unstable CA14 16 52 COc1ccc(O)c(C(=O)O)c1Br ZINC000217562940 BD For-Sale Unstable ALS 61 37 CCOc1ccc(CC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217562951 FG For-Sale Unstable NPY5R 24 41 Cn1c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c(O)c1CN1C[C@@]2(C)C[C@@H]1CC(C)(C)C2 ZINC000217562967 JG In-Stock Unstable CHRNA4 28 44 O=C(CN1CCC[C@H]2CCCC[C@H]21)c1cc(F)ccc1F ZINC000217562972 CH For-Sale Unstable SLC6A1 24 40 C[C@@H](N)c1cc(Br)ccc1N1CC[C@@H](N2CCCC2)C1 ZINC000217563003 EG For-Sale Unstable L3MBTL3 48 38 C[C@@H](N)c1cc(Br)ccc1N1CC[C@@H](N2CCCC2)C1 ZINC000217563003 EG For-Sale Unstable MBTD1 0 43 COc1ccc(/C=C\C(=O)O)cc1OCCCCC#N ZINC000217563009 CF For-Sale Unstable PTGER2 22 44 COc1ccc(/C=C\C(=O)O)cc1OCCCCC#N ZINC000217563009 CF For-Sale Unstable CYP1B1 21 40 COc1ccc(/C=C\C(=O)O)cc1OCCCCC#N ZINC000217563009 CF For-Sale Unstable APP 22 46 COc1ccc(/C=C\C(=O)O)cc1OCCCCC#N ZINC000217563009 CF For-Sale Unstable CYP1A1 21 40 COc1ccc(/C=C\C(=O)O)cc1OCCCCC#N ZINC000217563009 CF For-Sale Unstable TUBB1 55 39 COc1ccc(/C=C\C(=O)O)cc1OCCCCC#N ZINC000217563009 CF For-Sale Unstable AKR1C3 36 51 COc1ccc(/C=C\C(=O)O)cc1OCCCCC#N ZINC000217563009 CF For-Sale Unstable ABCG2 15 44 COc1c(C(=O)O)ccc(O)c1Br ZINC000217563049 BD For-Sale Unstable AKR1C2 46 38 O=C1O[C@@]2(CCCN(C(=O)C34CC5CC(CC(C5)C3)C4)C2)c2ccccc21 ZINC000217563058 FH For-Sale Unstable NPY5R 33 41 Cn1c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c(O)c1CN1CCN(S(C)(=O)=O)CC1 ZINC000217563076 KB In-Stock Unstable CHRNA4 39 51 C[C@H](N)c1cc(Br)ccc1N1CC[C@@H](N2CCCC2)C1 ZINC000217563078 EG For-Sale Unstable L3MBTL3 48 38 C[C@H](N)c1cc(Br)ccc1N1CC[C@@H](N2CCCC2)C1 ZINC000217563078 EG For-Sale Unstable MBTD1 0 43 N#CCCCCOc1ccc(/C=C\C(=O)O)cc1[N+](=O)[O-] ZINC000217563099 CF For-Sale Unstable AKR1C3 30 42 N#CCN(C(=O)c1cc(Cl)ccn1)C1CCCC1 ZINC000217563125 CF On-Demand Unstable ACE 49 40 O=C1O[C@]2(CCCN(C(=O)C34CC5CC(CC(C5)C3)C4)C2)c2ccccc21 ZINC000217563145 FH For-Sale Unstable NPY5R 33 41 C[C@@H](N)c1ccc(Br)cc1N1CC[C@@H](N2CCCCC2)C1 ZINC000217563151 FH For-Sale Unstable L3MBTL3 67 38 C[C@@H](N)c1ccc(Br)cc1N1CC[C@@H](N2CCCCC2)C1 ZINC000217563151 FH For-Sale Unstable MBTD1 0 43 Cc1cc(C(=O)O)c(O)c(Br)c1O ZINC000217563164 BD For-Sale Unstable AKR1C2 79 50 Cc1cc(C(=O)O)c(O)c(Br)c1O ZINC000217563164 BD For-Sale Unstable AKR1C1 78 50 COC(=O)CS[C@@H]1CCN(C(=O)c2ccc(-n3cccc3)cc2)C1 ZINC000217563170 EF In-Stock Unstable L3MBTL3 51 36 CCOc1cccc(/C=C\C(=O)O)c1OCCCCC#N ZINC000217563180 CG For-Sale Unstable PTGER2 45 43 CCOc1cccc(/C=C\C(=O)O)c1OCCCCC#N ZINC000217563180 CG For-Sale Unstable PTGER4 23 43 CCOc1cccc(/C=C\C(=O)O)c1OCCCCC#N ZINC000217563180 CG For-Sale Unstable PTGER3 20 41 CC(C)(C)OC(=O)N1CCN(C(=O)NCCc2ccc(Br)cc2)CC1 ZINC000217563222 HG On-Demand Unstable GPR119 41 41 CC(C)(C)OC(=O)N1CCN(C(=O)NCCc2ccc(Br)cc2)CC1 ZINC000217563222 HG On-Demand Unstable LIG1 0 40 O=c1cccc2n1C[C@H]1C[C@@H]2CN(Cc2cc(=O)n3cc(Cl)ccc3n2)C1 ZINC000217563226 GE In-Stock Unstable CHRNA4 33 56 C[C@H](N)c1ccc(Br)cc1N1CC[C@@H](N2CCCCC2)C1 ZINC000217563236 FH For-Sale Unstable L3MBTL3 67 38 C[C@H](N)c1ccc(Br)cc1N1CC[C@@H](N2CCCCC2)C1 ZINC000217563236 FH For-Sale Unstable MBTD1 0 43 N#CCN(C(=O)c1cc(Br)ccc1I)C1CCCC1 ZINC000217563249 IH On-Demand Unstable ACE 48 36 COC(=O)CS[C@H]1CCN(C(=O)c2ccc(-n3cccc3)cc2)C1 ZINC000217563252 EF In-Stock Unstable L3MBTL3 51 36 COc1cc(OC)cc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217563256 FG For-Sale Unstable NPY5R 28 46 COc1ccc(OCCCCC#N)c(/C=C\C(=O)O)c1 ZINC000217563265 CF For-Sale Unstable PTGER2 41 42 COc1ccc(OCCCCC#N)c(/C=C\C(=O)O)c1 ZINC000217563265 CF For-Sale Unstable PTGER4 23 42 COc1ccc(OCCCCC#N)c(/C=C\C(=O)O)c1 ZINC000217563265 CF For-Sale Unstable CYP1B1 38 45 COc1ccc(OCCCCC#N)c(/C=C\C(=O)O)c1 ZINC000217563265 CF For-Sale Unstable PTGER3 17 42 COc1ccc(OCCCCC#N)c(/C=C\C(=O)O)c1 ZINC000217563265 CF For-Sale Unstable LTB4R 48 43 COc1ccc(OCCCCC#N)c(/C=C\C(=O)O)c1 ZINC000217563265 CF For-Sale Unstable CYP1A1 36 45 COc1ccc(OCCCCC#N)c(/C=C\C(=O)O)c1 ZINC000217563265 CF For-Sale Unstable CYP1A2 15 45 COc1ccc(OCCCCC#N)c(/C=C\C(=O)O)c1 ZINC000217563265 CF For-Sale Unstable CYSP_PLAFA 40 44 Cn1c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c(O)c1CN1CCN(CCOc2ccccc2)CC1 ZINC000217563309 KE In-Stock Unstable CHRNA4 36 49 O=C(Nc1ccc([N+](=O)[O-])cc1C(=O)c1ccccc1)c1ccc2ncsc2c1 ZINC000217563321 HJ On-Demand Bother PYGL 27 40 CC(C)(C)OC(=O)N1CCC(NC(=O)NCCc2ccc(Br)cc2)CC1 ZINC000217563323 IH On-Demand Unstable EPHX2 40 46 CC(C)(C)OC(=O)N1CCC(NC(=O)NCCc2ccc(Br)cc2)CC1 ZINC000217563323 IH On-Demand Unstable GPR119 48 43 COc1cc(OC)cc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217563328 FG For-Sale Unstable NPY5R 28 46 C[C@@H](N)c1cc(Br)ccc1N1CC[C@@H](N2CCCCC2)C1 ZINC000217563330 FH For-Sale Unstable MBTD1 0 43 COc1cccc(/C=C\C(=O)O)c1OCCCCC#N ZINC000217563349 CF For-Sale Unstable PTGER2 50 51 COc1cccc(/C=C\C(=O)O)c1OCCCCC#N ZINC000217563349 CF For-Sale Unstable PTGER4 22 40 COc1cccc(/C=C\C(=O)O)c1OCCCCC#N ZINC000217563349 CF For-Sale Unstable PTGER3 22 51 Cc1nn(C)cc1C(=O)N(CC#N)C1CCCC1 ZINC000217563370 BD On-Demand Unstable ACE 41 34 C[C@H](N)c1cc(Br)ccc1N1CC[C@@H](N2CCCCC2)C1 ZINC000217563404 FH For-Sale Unstable MBTD1 0 43 COc1ccc2oc(=O)cc(CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)c2c1 ZINC000217563423 GF In-Stock Unstable CHRNA4 30 51 O=C(NCC1CCCC1)Nc1cccc(O)c1 ZINC000217563437 BF For-Sale Unstable CCR3 64 40 O=C(NCC1CCCC1)Nc1cccc(O)c1 ZINC000217563437 BF For-Sale Unstable LDLR 0 42 O=C(NCC1CCCC1)Nc1cccc(O)c1 ZINC000217563437 BF For-Sale Unstable EPHX2 37 71 O=C(NCC1CCCC1)Nc1cccc(O)c1 ZINC000217563437 BF For-Sale Unstable PRMT3 41 40 COc1cccc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1OC ZINC000217563458 FG For-Sale Unstable NPY5R 23 46 O=C(CN1CCC[C@@H]2CCCC[C@H]21)c1ccc(F)cc1F ZINC000217563468 CH For-Sale Unstable SLC6A1 23 40 CC(C)CNc1ccc(S(=O)(=O)NC(C)(C)C)cc1C(=O)O ZINC000217563491 EF In-Stock Unstable MTNN 61 33 COc1cccc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1OC ZINC000217563535 FG For-Sale Unstable NPY5R 23 46 O=c1[nH]c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)nc2ccsc12 ZINC000217563536 FD In-Stock Unstable CHRNA4 32 53 O=C(CN1CCC[C@H]2CCCC[C@H]21)c1ccc(F)cc1F ZINC000217563556 CH For-Sale Unstable SLC6A1 23 40 COc1cccc(OC)c1C(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217563638 FG For-Sale Unstable NPY5R 28 50 O=c1[nH]c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)nc2ccccc12 ZINC000217563645 ED In-Stock Unstable CHRNA4 34 62 O=c1[nH]c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)nc2ccccc12 ZINC000217563645 ED In-Stock Unstable PARP1 16 40 O=C(NCC1CCCC1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217563661 CE For-Sale Unstable CA2 29 49 O=C(NCC1CCCC1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217563661 CE For-Sale Unstable CA1 44 41 O=C(NCC1CCCC1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217563661 CE For-Sale Unstable CCR3 29 41 O=C(NCC1CCCC1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217563661 CE For-Sale Unstable EPHX2 48 61 O=C(NCC1CCCC1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217563661 CE For-Sale Unstable CA12 40 48 O=C(NCC1CCCC1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217563661 CE For-Sale Unstable CA9 37 48 O=C(NCC1CCCC1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217563661 CE For-Sale Unstable F13A1 70 42 O=C(NCC1CCCC1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217563661 CE For-Sale Unstable NCE103 39 41 O=C(NCC1CCCC1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217563661 CE For-Sale Unstable PRMT3 40 38 O=C(NCC1CCCC1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217563661 CE For-Sale Unstable MTCA1 46 48 O=C(NCC1CCCC1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217563661 CE For-Sale Unstable P96878_MYCTU 58 48 O=C(NCC1CCCC1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217563661 CE For-Sale Unstable NAMPT 50 45 COc1ccc(/C=C\C(=O)O)c(OCCCCC#N)c1 ZINC000217563680 CF For-Sale Unstable PTGER2 43 48 COc1ccc(/C=C\C(=O)O)c(OCCCCC#N)c1 ZINC000217563680 CF For-Sale Unstable PTGER4 23 48 COc1ccc(/C=C\C(=O)O)c(OCCCCC#N)c1 ZINC000217563680 CF For-Sale Unstable CYP1B1 43 44 COc1ccc(/C=C\C(=O)O)c(OCCCCC#N)c1 ZINC000217563680 CF For-Sale Unstable PTGER3 18 41 COc1ccc(/C=C\C(=O)O)c(OCCCCC#N)c1 ZINC000217563680 CF For-Sale Unstable LTB4R 44 42 COc1ccc(/C=C\C(=O)O)c(OCCCCC#N)c1 ZINC000217563680 CF For-Sale Unstable CYP1A1 43 44 COc1ccc(/C=C\C(=O)O)c(OCCCCC#N)c1 ZINC000217563680 CF For-Sale Unstable CYP1A2 18 44 COc1ccc(/C=C\C(=O)O)c(OCCCCC#N)c1 ZINC000217563680 CF For-Sale Unstable CYSP_PLAFA 36 41 CSc1ccccc1C(=O)Nc1ccc([N+](=O)[O-])cc1C(=O)c1ccccc1 ZINC000217563712 GJ On-Demand Unstable KCNMA1 33 49 CSc1ccccc1C(=O)Nc1ccc([N+](=O)[O-])cc1C(=O)c1ccccc1 ZINC000217563712 GJ On-Demand Unstable F2RL3 44 32 CSc1ccccc1C(=O)Nc1ccc([N+](=O)[O-])cc1C(=O)c1ccccc1 ZINC000217563712 GJ On-Demand Unstable AKR1C3 15 53 CSc1ccccc1C(=O)Nc1ccc([N+](=O)[O-])cc1C(=O)c1ccccc1 ZINC000217563712 GJ On-Demand Unstable WDR5 33 40 COc1cccc(OC)c1C(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217563720 FG For-Sale Unstable NPY5R 28 50 N#CCN(C(=O)c1ccc(C(F)(F)F)cn1)C1CCCC1 ZINC000217563723 CG On-Demand Unstable DHODH 0 41 N#CCN(C(=O)c1ccc(C(F)(F)F)cn1)C1CCCC1 ZINC000217563723 CG On-Demand Unstable HSD11B1 15 40 COC(=O)CS[C@@H]1CCN(C(=O)/C=C/c2ccccc2Cl)C1 ZINC000217563727 EF In-Stock Unstable ITGAL 49 42 C[C@@H]1CN(C[C@@H](O)CO)C[C@@H](C)O1 ZINC000217563745 AB On-Demand Unstable ERG2 19 40 C[C@@H]1CN(C[C@@H](O)CO)C[C@@H](C)O1 ZINC000217563745 AB On-Demand Unstable ZM.86993 0 40 C[C@@H]1CN(C[C@@H](O)CO)C[C@@H](C)O1 ZINC000217563745 AB On-Demand Unstable Q2TU57_MAIZE 21 40 COc1cc2nc(CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)[nH]c(=O)c2cc1OC ZINC000217563764 HD In-Stock Unstable CHRNA4 31 51 CC(C)(C)Nc1ccc(S(=O)(=O)NC(C)(C)C)cc1C(=O)O ZINC000217563774 EF In-Stock Unstable PRTN3 45 35 O=C(NCC1CCCC1)Nc1cccc(S(=O)(=O)O)c1 ZINC000217563783 CE For-Sale Unstable LPL 41 32 O=C(NCC1CCCC1)Nc1cccc(S(=O)(=O)O)c1 ZINC000217563783 CE For-Sale Unstable CCR3 70 45 O=C(NCC1CCCC1)Nc1cccc(S(=O)(=O)O)c1 ZINC000217563783 CE For-Sale Unstable EPHX2 39 69 O=C(NCC1CCCC1)Nc1cccc(S(=O)(=O)O)c1 ZINC000217563783 CE For-Sale Unstable ST14 42 35 O=C(NCC1CCCC1)Nc1cccc(S(=O)(=O)O)c1 ZINC000217563783 CE For-Sale Unstable NAMPT 32 40 Cc1noc(C)c1COc1ccc(CC(=O)Nc2ccc([N+](=O)[O-])cc2C(=O)c2ccccc2)cc1 ZINC000217563807 JK On-Demand Unstable RORC 19 46 COC(=O)CS[C@H]1CCN(C(=O)/C=C/c2ccccc2Cl)C1 ZINC000217563808 EF In-Stock Unstable ITGAL 49 42 COc1ccc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1OC ZINC000217563834 FG For-Sale Unstable NPY5R 27 47 C[C@@H]1[C@H](c2ccccc2)[C@H](CO)N1C ZINC000217563858 AD For-Sale Unstable HSD17B2 42 33 O=C(NCc1ccccc1)c1ccc(N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)c(NC(=O)c2ccco2)c1 ZINC000217563872 KI In-Stock Unstable CHRNA4 26 44 CC[C@@H]1CCCCN1C[C@@H](O)CO ZINC000217563915 AC On-Demand Unstable SLC18A2 53 39 COc1ccc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1OC ZINC000217563925 FG For-Sale Unstable NPY5R 27 47 C[C@H]1[C@H](c2ccccc2)[C@H](CO)N1C ZINC000217563941 AD For-Sale Unstable HSD17B2 42 33 C/C=C/S[C@H](NC(=O)CC[C@H](N)C(=O)O)C(=O)O ZINC000217563945 CB Annotated Unstable GLO1 42 38 C/C=C/S[C@H](NC(=O)CC[C@H](N)C(=O)O)C(=O)O ZINC000217563945 CB Annotated Unstable GRM8 24 42 C/C=C/S[C@H](NC(=O)CC[C@H](N)C(=O)O)C(=O)O ZINC000217563945 CB Annotated Unstable GRIK3 35 42 C/C=C/S[C@H](NC(=O)CC[C@H](N)C(=O)O)C(=O)O ZINC000217563945 CB Annotated Unstable GRIK1 32 42 C/C=C/S[C@H](NC(=O)CC[C@H](N)C(=O)O)C(=O)O ZINC000217563945 CB Annotated Unstable BHMT 56 39 C/C=C/S[C@H](NC(=O)CC[C@H](N)C(=O)O)C(=O)O ZINC000217563945 CB Annotated Unstable NOD1 100 48 COc1ccc(C(=O)N(CC#N)C2CCCC2)c(F)c1 ZINC000217563953 CF On-Demand Unstable ACE 52 36 CC(C)(C)NS(=O)(=O)c1ccc(NC2CC2)c(C(=O)O)c1 ZINC000217563980 DE In-Stock Unstable SFRP1 70 33 CC[C@H]1CCCCN1C[C@@H](O)CO ZINC000217563995 AC On-Demand Unstable SLC18A2 53 39 COc1ccc(CNC(=O)[C@@H]2CC[C@@H](CNC(=O)[C@@H]3Cc4ccccc4CN3)CC2)cc1 ZINC000217564004 IF In-Stock Unstable MC4R 35 41 COc1ccc(CNC(=O)[C@@H]2CC[C@@H](CNC(=O)[C@@H]3Cc4ccccc4CN3)CC2)cc1 ZINC000217564004 IF In-Stock Unstable NPY2R 34 43 COc1ccc(CNC(=O)[C@@H]2CC[C@@H](CNC(=O)[C@@H]3Cc4ccccc4CN3)CC2)cc1 ZINC000217564004 IF In-Stock Unstable MTNR1A 34 45 COc1ccc(CNC(=O)[C@@H]2CC[C@@H](CNC(=O)[C@@H]3Cc4ccccc4CN3)CC2)cc1 ZINC000217564004 IF In-Stock Unstable MTNR1B 31 45 C[C@@H]1[C@@H](c2ccccc2)[C@H](CO)N1C ZINC000217564016 AD For-Sale Unstable HSD17B2 42 33 COc1ccccc1OCC(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217564024 FF For-Sale Unstable NPY5R 26 49 O=C(NCC1CCCC1)Nc1ccc(O)cc1 ZINC000217564037 BF For-Sale Unstable LDLR 0 43 O=C(NCC1CCCC1)Nc1ccc(O)cc1 ZINC000217564037 BF For-Sale Unstable EPHX2 43 68 O=C(NCC1CCCC1)Nc1ccc(O)cc1 ZINC000217564037 BF For-Sale Unstable CYP2B1 0 40 O=C(NCC1CCCC1)Nc1ccc(O)cc1 ZINC000217564037 BF For-Sale Unstable PRMT3 34 41 C[C@@H]1CCC[C@@]([C@@H](N)Cc2cc(F)ccc2F)(N(C)C)C1 ZINC000217564044 CG For-Sale Unstable DPP4 28 44 COC(=O)CS[C@@H]1CCN(C(=O)c2cccc(F)c2)C1 ZINC000217564097 CD In-Stock Unstable CCR3 41 42 CC(C)(C)NS(=O)(=O)c1ccc(NC2CCCC2)c(C(=O)O)c1 ZINC000217564099 EF In-Stock Unstable SFRP1 64 32 CC(C)(C)NS(=O)(=O)c1ccc(NC2CCCC2)c(C(=O)O)c1 ZINC000217564099 EF In-Stock Unstable WNT3 47 31 COc1ccccc1OCC(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217564106 FF For-Sale Unstable NPY5R 26 49 Cn1c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c(O)c1CN1CCN(Cc2cccc(Cl)c2)CC1 ZINC000217564128 KF In-Stock Unstable CHRNA4 30 55 CCCCc1ccc(NC(=O)NCC2CCCC2)cc1 ZINC000217564139 CI For-Sale Unstable CCR3 54 41 CCCCc1ccc(NC(=O)NCC2CCCC2)cc1 ZINC000217564139 CI For-Sale Unstable SCN2A 15 50 CCCCc1ccc(NC(=O)NCC2CCCC2)cc1 ZINC000217564139 CI For-Sale Unstable S1PR4 28 40 CCCCc1ccc(NC(=O)NCC2CCCC2)cc1 ZINC000217564139 CI For-Sale Unstable S1PR3 21 40 CCCCc1ccc(NC(=O)NCC2CCCC2)cc1 ZINC000217564139 CI For-Sale Unstable CFTR 47 38 CCCCc1ccc(NC(=O)NCC2CCCC2)cc1 ZINC000217564139 CI For-Sale Unstable EPHX2 31 61 CCCCc1ccc(NC(=O)NCC2CCCC2)cc1 ZINC000217564139 CI For-Sale Unstable SPHK1 39 44 CCCCc1ccc(NC(=O)NCC2CCCC2)cc1 ZINC000217564139 CI For-Sale Unstable S1PR5 27 40 CCCCc1ccc(NC(=O)NCC2CCCC2)cc1 ZINC000217564139 CI For-Sale Unstable PLM2_PLAFA 34 40 CCCCc1ccc(NC(=O)NCC2CCCC2)cc1 ZINC000217564139 CI For-Sale Unstable ACAT 0 49 Cc1nc2ccccc2cc1C(=O)N1CCc2sccc2[C@@H]1c1cccs1 ZINC000217564162 GK On-Demand Unstable TRPM8 19 45 COC(=O)CS[C@H]1CCN(C(=O)c2cccc(F)c2)C1 ZINC000217564181 CD In-Stock Unstable CCR3 41 42 CC(C)(C)NS(=O)(=O)c1ccc(NC2CCCCC2)c(C(=O)O)c1 ZINC000217564214 FG In-Stock Unstable SFRP1 60 31 CC(C)(C)NS(=O)(=O)c1ccc(NC2CCCCC2)c(C(=O)O)c1 ZINC000217564214 FG In-Stock Unstable WNT3 47 31 COc1cccc(OCC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217564219 FF For-Sale Unstable COLA 40 34 COc1cccc(OCC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217564219 FF For-Sale Unstable CPT2 40 34 COc1cccc(OCC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217564219 FF For-Sale Unstable NPY5R 30 51 C[C@@H]1CCC[C@]([C@@H](N)Cc2cc(F)ccc2F)(N(C)C)C1 ZINC000217564222 CG For-Sale Unstable DPP4 28 44 CC(=O)Nc1ccc(C(=O)CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc1 ZINC000217564225 FE In-Stock Unstable CHRNA4 37 74 Cc1nc2ccccc2cc1C(=O)N1CCc2sccc2[C@H]1c1cccs1 ZINC000217564246 GK On-Demand Unstable TRPM8 19 45 CC(C)[C@@H](N)c1nnc2ccc(-c3ccccc3)nn12 ZINC000217564262 CE In-Stock Unstable MET 15 40 COc1cccc(OCC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217564295 FF For-Sale Unstable COLA 40 34 COc1cccc(OCC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217564295 FF For-Sale Unstable CPT2 40 34 COc1cccc(OCC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217564295 FF For-Sale Unstable NPY5R 30 51 O=C(CN1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)c1ccc2c(c1)OCCCO2 ZINC000217564307 GE In-Stock Unstable CHRNA4 33 66 CN(C(=O)[C@@H]1C[C@@H]1c1ccccc1C(F)(F)F)C1CCCCCC1 ZINC000217564346 EJ On-Demand Unstable RBP4 85 40 CC(C)[C@H](N)c1nnc2ccc(-c3ccccc3)nn12 ZINC000217564347 CE In-Stock Unstable MET 15 40 O=C(NCC1CCCC1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217564382 GI For-Sale Unstable F2 15 46 O=C(NCC1CCCC1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217564382 GI For-Sale Unstable CNR1 16 68 O=C(NCC1CCCC1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217564382 GI For-Sale Unstable OPRM1 0 46 O=C(NCC1CCCC1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217564382 GI For-Sale Unstable OPRD1 29 44 O=C(NCC1CCCC1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217564382 GI For-Sale Unstable OPRK1 26 44 O=C(NCC1CCCC1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217564382 GI For-Sale Unstable OPRL1 23 44 O=C(NCC1CCCC1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217564382 GI For-Sale Unstable SLC6A3 15 44 O=C(NCC1CCCC1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217564382 GI For-Sale Unstable NPY2R 24 41 O=C(NCC1CCCC1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217564382 GI For-Sale Unstable SMO 15 43 O=C(NCC1CCCC1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217564382 GI For-Sale Unstable NMUR2 0 61 O=C(NCC1CCCC1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217564382 GI For-Sale Unstable NMUR1 0 61 O=C1O[C@@]2(CCCN(C(=O)CSCc3ccccc3)C2)c2ccccc21 ZINC000217564409 FH For-Sale Unstable NPY5R 26 41 COc1ccc2c(c1)cc(CN1C[C@@H]3C[C@H](C1)c1cccc(=O)n1C3)c(=O)n2C ZINC000217564411 GE In-Stock Unstable CHRNA4 31 51 CN(C(=O)[C@H]1C[C@@H]1c1ccccc1C(F)(F)F)C1CCCCCC1 ZINC000217564425 EJ On-Demand Unstable RBP4 85 40 O=C(/C=C\c1cc(Cl)ccc1Cl)N[C@@H]1CC[C@H](C(=O)O)C1 ZINC000217564469 EG For-Sale Unstable BOTA 22 43 O=C1O[C@]2(CCCN(C(=O)CSCc3ccccc3)C2)c2ccccc21 ZINC000217564490 FH For-Sale Unstable NPY5R 26 41 O=C(NCC1CCCC1)N1CCCc2ccccc21 ZINC000217564491 CG For-Sale Unstable AVPR2 48 45 O=C(NCC1CCCC1)N1CCCc2ccccc21 ZINC000217564491 CG For-Sale Unstable AVPR1A 26 43 O=C(NCC1CCCC1)N1CCCc2ccccc21 ZINC000217564491 CG For-Sale Unstable CACNA1I 48 33 CN(C(=O)[C@@H]1C[C@H]1c1ccccc1C(F)(F)F)C1CCCCCC1 ZINC000217564511 EJ On-Demand Unstable RBP4 85 40 CCCOC(=O)/C=C\c1ccccc1OC ZINC000217564527 BF For-Sale Unstable PTGER2 40 43 CCCOC(=O)/C=C\c1ccccc1OC ZINC000217564527 BF For-Sale Unstable PTGER4 22 43 CCCOC(=O)/C=C\c1ccccc1OC ZINC000217564527 BF For-Sale Unstable CYP1B1 22 42 CCCOC(=O)/C=C\c1ccccc1OC ZINC000217564527 BF For-Sale Unstable PTGER3 18 40 CCCOC(=O)/C=C\c1ccccc1OC ZINC000217564527 BF For-Sale Unstable HCAR2 0 45 CCCOC(=O)/C=C\c1ccccc1OC ZINC000217564527 BF For-Sale Unstable AKR1B10 50 55 CCCOC(=O)/C=C\c1ccccc1OC ZINC000217564527 BF For-Sale Unstable CYSP_PLAFA 43 34 O=C(CN1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)c1ccc2ccccc2c1 ZINC000217564569 FG In-Stock Unstable CHRNA4 48 78 CN(C(=O)[C@H]1C[C@H]1c1ccccc1C(F)(F)F)C1CCCCCC1 ZINC000217564581 EJ On-Demand Unstable RBP4 85 40 CCSc1ccccc1C(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217564604 FI For-Sale Unstable NPY5R 23 41 O=C(NCC1CCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217564609 DH On-Demand Unstable F2 19 43 O=C(NCC1CCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217564609 DH On-Demand Unstable PRSS1 15 43 O=C(NCC1CCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217564609 DH On-Demand Unstable CHRM2 24 41 O=C(NCC1CCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217564609 DH On-Demand Unstable FKBP1A 42 39 O=C(NCC1CCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217564609 DH On-Demand Unstable DRD4 15 42 O=C(NCC1CCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217564609 DH On-Demand Unstable ACHE 19 43 O=C(NCC1CCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217564609 DH On-Demand Unstable GRIN1 0 41 O=C(NCC1CCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217564609 DH On-Demand Unstable HTR4 42 41 O=C(NCC1CCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217564609 DH On-Demand Unstable GRIN2B 88 48 O=C(NCC1CCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217564609 DH On-Demand Unstable SIGMAR1 41 45 O=C(NCC1CCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217564609 DH On-Demand Unstable CCR3 69 49 O=C(NCC1CCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217564609 DH On-Demand Unstable CCR5 15 41 O=C(NCC1CCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217564609 DH On-Demand Unstable C3AR1 40 37 O=C(NCC1CCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217564609 DH On-Demand Unstable REN 40 35 O=C(NCC1CCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217564609 DH On-Demand Unstable CAPN1 38 43 O=C(NCC1CCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217564609 DH On-Demand Unstable CAPN2 39 43 O=C(NCC1CCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217564609 DH On-Demand Unstable EPHX2 33 42 O=C(NCC1CCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217564609 DH On-Demand Unstable GRIN2C 18 41 O=C(NCC1CCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217564609 DH On-Demand Unstable GRIN3A 0 42 O=C(NCC1CCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217564609 DH On-Demand Unstable AMP1_PLAFQ 23 52 O=C(NCC1CCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217564609 DH On-Demand Unstable CACNA1I 54 37 O=C(NCC1CCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217564609 DH On-Demand Unstable SMO 25 44 COC(=O)CS[C@@H]1CCN(C(=O)c2cccc(Br)c2)C1 ZINC000217564648 FF In-Stock Unstable L3MBTL1 0 50 COC(=O)CS[C@@H]1CCN(C(=O)c2cccc(Br)c2)C1 ZINC000217564648 FF In-Stock Unstable MBTD1 0 46 COCCNc1ccc(S(=O)(=O)NC(C)(C)C)cc1C(=O)O ZINC000217564660 ED In-Stock Unstable PRTN3 44 31 O=C([C@@H]1CC(=O)N(c2n[nH]c3ccccc23)C1)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217564677 HD In-Stock Unstable CHRNA4 26 40 COc1cc(C(C)C)c(Cl)cc1[C@H](O)CN ZINC000217564679 BE For-Sale Unstable P2RX2 77 38 COc1cc(C(C)C)c(Cl)cc1[C@H](O)CN ZINC000217564679 BE For-Sale Unstable P2RX3 56 33 CCSc1ccccc1C(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217564681 FI For-Sale Unstable NPY5R 23 41 Cc1ccc(NC(=O)c2cc3ccccc3nc2C)cc1C(F)(F)F ZINC000217564696 EK On-Demand Unstable ABL1 45 35 Cc1ccc(NC(=O)c2cc3ccccc3nc2C)cc1C(F)(F)F ZINC000217564696 EK On-Demand Unstable JUN 20 40 Cc1ccc(NC(=O)c2cc3ccccc3nc2C)cc1C(F)(F)F ZINC000217564696 EK On-Demand Unstable LCK 45 45 Cc1ccc(NC(=O)c2cc3ccccc3nc2C)cc1C(F)(F)F ZINC000217564696 EK On-Demand Unstable MAPK14 15 45 Cc1ccc(NC(=O)c2cc3ccccc3nc2C)cc1C(F)(F)F ZINC000217564696 EK On-Demand Unstable TRPV1 23 44 Cc1ccc(NC(=O)c2cc3ccccc3nc2C)cc1C(F)(F)F ZINC000217564696 EK On-Demand Unstable FLT1 23 42 Cc1ccc(NC(=O)c2cc3ccccc3nc2C)cc1C(F)(F)F ZINC000217564696 EK On-Demand Unstable KDR 26 45 Cc1ccc(NC(=O)c2cc3ccccc3nc2C)cc1C(F)(F)F ZINC000217564696 EK On-Demand Unstable GRM4 25 44 Cc1ccc(NC(=O)c2cc3ccccc3nc2C)cc1C(F)(F)F ZINC000217564696 EK On-Demand Unstable MTTP 59 38 Cc1ccc(NC(=O)c2cc3ccccc3nc2C)cc1C(F)(F)F ZINC000217564696 EK On-Demand Unstable S1PR1 16 43 Cc1ccc(NC(=O)c2cc3ccccc3nc2C)cc1C(F)(F)F ZINC000217564696 EK On-Demand Unstable LYN 47 35 Cc1ccc(NC(=O)c2cc3ccccc3nc2C)cc1C(F)(F)F ZINC000217564696 EK On-Demand Unstable CSF1R 15 42 Cc1ccc(NC(=O)c2cc3ccccc3nc2C)cc1C(F)(F)F ZINC000217564696 EK On-Demand Unstable TEK 27 42 Cc1ccc(NC(=O)c2cc3ccccc3nc2C)cc1C(F)(F)F ZINC000217564696 EK On-Demand Unstable BTK 28 40 Cc1ccc(NC(=O)c2cc3ccccc3nc2C)cc1C(F)(F)F ZINC000217564696 EK On-Demand Unstable NR2E3 56 38 Cc1ccc(NC(=O)c2cc3ccccc3nc2C)cc1C(F)(F)F ZINC000217564696 EK On-Demand Unstable SHH 55 48 Cc1ccc(NC(=O)c2cc3ccccc3nc2C)cc1C(F)(F)F ZINC000217564696 EK On-Demand Unstable KCNK3 78 44 Cc1ccc(NC(=O)c2cc3ccccc3nc2C)cc1C(F)(F)F ZINC000217564696 EK On-Demand Unstable KCNK9 66 40 Cc1ccc(NC(=O)c2cc3ccccc3nc2C)cc1C(F)(F)F ZINC000217564696 EK On-Demand Unstable TMPRSS4 0 40 COC(=O)CS[C@H]1CCN(C(=O)c2cccc(Br)c2)C1 ZINC000217564728 FF In-Stock Unstable L3MBTL1 0 50 COC(=O)CS[C@H]1CCN(C(=O)c2cccc(Br)c2)C1 ZINC000217564728 FF In-Stock Unstable MBTD1 0 46 COc1cc(C(C)C)c(Cl)cc1[C@@H](O)CN ZINC000217564757 BE For-Sale Unstable P2RX2 77 38 COc1cc(C(C)C)c(Cl)cc1[C@@H](O)CN ZINC000217564757 BE For-Sale Unstable P2RX3 56 33 O=C([C@H]1CC(=O)N(c2n[nH]c3ccccc23)C1)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217564773 HD In-Stock Unstable CHRNA4 26 40 CC(C)[C@@H](N)c1nnc2ccc(-c3ccc(F)cc3)nn12 ZINC000217564775 CF In-Stock Unstable PDE1A 21 40 CC(C)[C@@H](N)c1nnc2ccc(-c3ccc(F)cc3)nn12 ZINC000217564775 CF In-Stock Unstable MET 16 40 O=C1O[C@@]2(CCCN(C(=O)CCSc3ccccc3)C2)c2ccccc21 ZINC000217564790 FH In-Stock Unstable NPY5R 24 40 Cc1cc(NC(=O)[C@@H]2C[C@@H]2c2ccccc2Cl)n(-c2ccc(F)cc2)n1 ZINC000217564821 FJ On-Demand Unstable PRCP 47 38 CC(C)[C@H](N)c1nnc2ccc(-c3ccc(F)cc3)nn12 ZINC000217564856 CF In-Stock Unstable PDE1A 21 40 CC(C)[C@H](N)c1nnc2ccc(-c3ccc(F)cc3)nn12 ZINC000217564856 CF In-Stock Unstable MET 16 40 O=C(NCC1CCCC1)NC(c1ccccc1)c1ccccc1 ZINC000217564868 DI On-Demand Unstable AMY2 44 31 O=C(NCC1CCCC1)NC(c1ccccc1)c1ccccc1 ZINC000217564868 DI On-Demand Unstable XIAP 49 37 O=C(NCC1CCCC1)NC(c1ccccc1)c1ccccc1 ZINC000217564868 DI On-Demand Unstable BIRC8 53 35 COc1cc(C(C)C)c(Cl)cc1[C@H](N)CO ZINC000217564870 BE For-Sale Unstable P2RX2 75 38 COc1cc(C(C)C)c(Cl)cc1[C@H](N)CO ZINC000217564870 BE For-Sale Unstable P2RX3 60 38 O=C1O[C@]2(CCCN(C(=O)CCSc3ccccc3)C2)c2ccccc21 ZINC000217564873 FH In-Stock Unstable NPY5R 24 40 Cc1cc(NC(=O)[C@H]2C[C@@H]2c2ccccc2Cl)n(-c2ccc(F)cc2)n1 ZINC000217564889 FJ On-Demand Unstable PRCP 47 38 Cc1noc(C)c1C(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217564891 DD In-Stock Unstable CHRNA4 38 50 CC(C)(C)NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217564922 FG In-Stock Unstable PRTN3 45 33 COc1cc(C(C)C)c(Cl)cc1[C@@H](N)CO ZINC000217564951 BE For-Sale Unstable P2RX2 75 38 COc1cc(C(C)C)c(Cl)cc1[C@@H](N)CO ZINC000217564951 BE For-Sale Unstable P2RX3 60 38 CC(C)[C@@H](N)c1nnc2ccc(-c3ccc(Cl)cc3)nn12 ZINC000217564962 DG In-Stock Unstable PDE1A 21 40 Cc1cc(NC(=O)[C@@H]2C[C@H]2c2ccccc2Cl)n(-c2ccc(F)cc2)n1 ZINC000217564967 FJ On-Demand Unstable PRCP 47 38 NS(=O)(=O)c1ccc(NC(=O)NCC2CCCC2)cc1 ZINC000217564978 CD On-Demand Unstable CA2 141 52 NS(=O)(=O)c1ccc(NC(=O)NCC2CCCC2)cc1 ZINC000217564978 CD On-Demand Unstable CA1 117 56 NS(=O)(=O)c1ccc(NC(=O)NCC2CCCC2)cc1 ZINC000217564978 CD On-Demand Unstable CA7 88 46 NS(=O)(=O)c1ccc(NC(=O)NCC2CCCC2)cc1 ZINC000217564978 CD On-Demand Unstable CA5B 65 46 NS(=O)(=O)c1ccc(NC(=O)NCC2CCCC2)cc1 ZINC000217564978 CD On-Demand Unstable CA4 109 54 NS(=O)(=O)c1ccc(NC(=O)NCC2CCCC2)cc1 ZINC000217564978 CD On-Demand Unstable CA5A 69 46 NS(=O)(=O)c1ccc(NC(=O)NCC2CCCC2)cc1 ZINC000217564978 CD On-Demand Unstable CA14 85 45 NS(=O)(=O)c1ccc(NC(=O)NCC2CCCC2)cc1 ZINC000217564978 CD On-Demand Unstable CDK1 0 43 NS(=O)(=O)c1ccc(NC(=O)NCC2CCCC2)cc1 ZINC000217564978 CD On-Demand Unstable CA12 124 64 NS(=O)(=O)c1ccc(NC(=O)NCC2CCCC2)cc1 ZINC000217564978 CD On-Demand Unstable CA9 124 64 NS(=O)(=O)c1ccc(NC(=O)NCC2CCCC2)cc1 ZINC000217564978 CD On-Demand Unstable CAH_METTE 23 40 NS(=O)(=O)c1ccc(NC(=O)NCC2CCCC2)cc1 ZINC000217564978 CD On-Demand Unstable F13A1 55 41 NS(=O)(=O)c1ccc(NC(=O)NCC2CCCC2)cc1 ZINC000217564978 CD On-Demand Unstable CYNT 48 42 NS(=O)(=O)c1ccc(NC(=O)NCC2CCCC2)cc1 ZINC000217564978 CD On-Demand Unstable NCE103 70 53 NS(=O)(=O)c1ccc(NC(=O)NCC2CCCC2)cc1 ZINC000217564978 CD On-Demand Unstable MTCA1 52 64 NS(=O)(=O)c1ccc(NC(=O)NCC2CCCC2)cc1 ZINC000217564978 CD On-Demand Unstable P96878_MYCTU 71 52 NS(=O)(=O)c1ccc(NC(=O)NCC2CCCC2)cc1 ZINC000217564978 CD On-Demand Unstable NAMPT 42 38 O=C1O[C@@]2(CCCN(C(=O)CSc3ccc(F)cc3)C2)c2ccccc21 ZINC000217564979 FH In-Stock Unstable NPY5R 29 45 CC(C)(C)[C@@H]1CC[C@@](CC(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)(n2cccc2)CC1 ZINC000217565005 IJ In-Stock Unstable CHRNA4 27 44 COc1cc(C(C)=O)cc(F)c1Br ZINC000217565019 BF For-Sale Unstable TUBB1 22 40 COC(=O)CS[C@@H]1CCN(C(=O)Cc2c[nH]c3ccccc23)C1 ZINC000217565027 EE In-Stock Unstable SSTR2 65 36 COC(=O)CS[C@@H]1CCN(C(=O)Cc2c[nH]c3ccccc23)C1 ZINC000217565027 EE In-Stock Unstable EDNRA 22 41 COC(=O)CS[C@@H]1CCN(C(=O)Cc2c[nH]c3ccccc23)C1 ZINC000217565027 EE In-Stock Unstable MC4R 44 35 COC(=O)CS[C@@H]1CCN(C(=O)Cc2c[nH]c3ccccc23)C1 ZINC000217565027 EE In-Stock Unstable TACR2 39 42 COC(=O)CS[C@@H]1CCN(C(=O)Cc2c[nH]c3ccccc23)C1 ZINC000217565027 EE In-Stock Unstable CCKAR 48 39 COC(=O)CS[C@@H]1CCN(C(=O)Cc2c[nH]c3ccccc23)C1 ZINC000217565027 EE In-Stock Unstable CCKBR 50 39 COC(=O)CS[C@@H]1CCN(C(=O)Cc2c[nH]c3ccccc23)C1 ZINC000217565027 EE In-Stock Unstable GHSR 53 37 COC(=O)CS[C@@H]1CCN(C(=O)Cc2c[nH]c3ccccc23)C1 ZINC000217565027 EE In-Stock Unstable CCR2 54 35 CC(C)[C@H](N)c1nnc2ccc(-c3ccc(Cl)cc3)nn12 ZINC000217565039 DG In-Stock Unstable PDE1A 21 40 Cc1cc(NC(=O)[C@H]2C[C@H]2c2ccccc2Cl)n(-c2ccc(F)cc2)n1 ZINC000217565048 FJ On-Demand Unstable PRCP 47 38 O=C1O[C@]2(CCCN(C(=O)CSc3ccc(F)cc3)C2)c2ccccc21 ZINC000217565068 FH In-Stock Unstable NPY5R 29 45 C[C@@H](NC(=O)NCC1CCCC1)C12CC3CC(CC(C3)C1)C2 ZINC000217565087 DI For-Sale Unstable EPHX2 38 64 COC(=O)CS[C@H]1CCN(C(=O)Cc2c[nH]c3ccccc23)C1 ZINC000217565100 EE In-Stock Unstable SSTR2 65 36 COC(=O)CS[C@H]1CCN(C(=O)Cc2c[nH]c3ccccc23)C1 ZINC000217565100 EE In-Stock Unstable EDNRA 22 41 COC(=O)CS[C@H]1CCN(C(=O)Cc2c[nH]c3ccccc23)C1 ZINC000217565100 EE In-Stock Unstable MC4R 44 35 COC(=O)CS[C@H]1CCN(C(=O)Cc2c[nH]c3ccccc23)C1 ZINC000217565100 EE In-Stock Unstable TACR2 39 42 COC(=O)CS[C@H]1CCN(C(=O)Cc2c[nH]c3ccccc23)C1 ZINC000217565100 EE In-Stock Unstable CCKAR 48 39 COC(=O)CS[C@H]1CCN(C(=O)Cc2c[nH]c3ccccc23)C1 ZINC000217565100 EE In-Stock Unstable CCKBR 50 39 COC(=O)CS[C@H]1CCN(C(=O)Cc2c[nH]c3ccccc23)C1 ZINC000217565100 EE In-Stock Unstable GHSR 53 37 COC(=O)CS[C@H]1CCN(C(=O)Cc2c[nH]c3ccccc23)C1 ZINC000217565100 EE In-Stock Unstable CCR2 54 35 Cn1c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c(O)c1CN1CC[C@H](c2ccccc2)C1 ZINC000217565113 JF In-Stock Unstable CHRNA4 30 52 CC(C)[C@@H](N)c1nnc2ccc(-c3ccc(Cl)cc3Cl)nn12 ZINC000217565169 EH In-Stock Unstable DPP4 0 42 CC(C)[C@@H](N)c1nnc2ccc(-c3ccc(Cl)cc3Cl)nn12 ZINC000217565169 EH In-Stock Unstable DPP8 24 42 CC(C)[C@@H](N)c1nnc2ccc(-c3ccc(Cl)cc3Cl)nn12 ZINC000217565169 EH In-Stock Unstable DPP9 31 41 Cc1cc(NC(=O)CCc2c(C)nc3c4ccccc4nn3c2C)n(-c2ccc(F)cc2)n1 ZINC000217565171 IJ On-Demand Unstable PANK1 0 52 Cc1cc(NC(=O)CCc2c(C)nc3c4ccccc4nn3c2C)n(-c2ccc(F)cc2)n1 ZINC000217565171 IJ On-Demand Unstable PANK2 0 47 Cc1cc(NC(=O)CCc2c(C)nc3c4ccccc4nn3c2C)n(-c2ccc(F)cc2)n1 ZINC000217565171 IJ On-Demand Unstable PANK3 0 52 C[C@H](NC(=O)NCC1CCCC1)C12CC3CC(CC(C3)C1)C2 ZINC000217565174 DI For-Sale Unstable EPHX2 38 64 O=C1O[C@@]2(CCCN(C(=O)COc3ccc(Cl)cc3)C2)c2ccccc21 ZINC000217565180 FG For-Sale Unstable CPT2 41 38 O=C1O[C@@]2(CCCN(C(=O)COc3ccc(Cl)cc3)C2)c2ccccc21 ZINC000217565180 FG For-Sale Unstable NPY5R 27 46 CC(C)(C)NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217565240 GG In-Stock Unstable PRTN3 45 32 CC(C)(C)NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217565240 GG In-Stock Unstable AKR1C3 21 48 CC(C)[C@H](N)c1nnc2ccc(-c3ccc(Cl)cc3Cl)nn12 ZINC000217565257 EH In-Stock Unstable DPP4 0 42 CC(C)[C@H](N)c1nnc2ccc(-c3ccc(Cl)cc3Cl)nn12 ZINC000217565257 EH In-Stock Unstable DPP8 24 42 CC(C)[C@H](N)c1nnc2ccc(-c3ccc(Cl)cc3Cl)nn12 ZINC000217565257 EH In-Stock Unstable DPP9 31 41 O=C1O[C@]2(CCCN(C(=O)COc3ccc(Cl)cc3)C2)c2ccccc21 ZINC000217565274 FG For-Sale Unstable CPT2 41 38 O=C1O[C@]2(CCCN(C(=O)COc3ccc(Cl)cc3)C2)c2ccccc21 ZINC000217565274 FG For-Sale Unstable NPY5R 27 46 O=C(NCC1CCCC1)Nc1cccc2c(O)cccc12 ZINC000217565288 CH For-Sale Unstable TRPV1 39 40 Cn1c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c(O)c1CN1CCCCC1 ZINC000217565349 HD In-Stock Unstable CHRNA4 31 51 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)(C)C)cc2C(=O)O)cc1 ZINC000217565354 HG In-Stock Unstable CA2 19 41 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)(C)C)cc2C(=O)O)cc1 ZINC000217565354 HG In-Stock Unstable BMP1 89 38 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)(C)C)cc2C(=O)O)cc1 ZINC000217565354 HG In-Stock Unstable CA1 20 44 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)(C)C)cc2C(=O)O)cc1 ZINC000217565354 HG In-Stock Unstable MMP13 59 43 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)(C)C)cc2C(=O)O)cc1 ZINC000217565354 HG In-Stock Unstable MMP3 46 39 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)(C)C)cc2C(=O)O)cc1 ZINC000217565354 HG In-Stock Unstable PRTN3 45 32 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)(C)C)cc2C(=O)O)cc1 ZINC000217565354 HG In-Stock Unstable MMP9 49 40 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)(C)C)cc2C(=O)O)cc1 ZINC000217565354 HG In-Stock Unstable PTGDR 26 43 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)(C)C)cc2C(=O)O)cc1 ZINC000217565354 HG In-Stock Unstable IAP 0 41 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)(C)C)cc2C(=O)O)cc1 ZINC000217565354 HG In-Stock Unstable CA9 25 44 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)(C)C)cc2C(=O)O)cc1 ZINC000217565354 HG In-Stock Unstable MMP1 52 40 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)(C)C)cc2C(=O)O)cc1 ZINC000217565354 HG In-Stock Unstable AKR1C3 30 43 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)(C)C)cc2C(=O)O)cc1 ZINC000217565354 HG In-Stock Unstable AKR1C2 52 38 COc1ccc(-c2ccc3nnc([C@@H](N)C(C)C)n3n2)cc1 ZINC000217565375 CE In-Stock Unstable MET 15 41 CN(C)c1ccccc1C(=O)N1CCC[C@@](C)(O)CC1 ZINC000217565387 CE In-Stock Unstable L3MBTL1 0 40 CN(C)c1ccccc1C(=O)N1CCC[C@@](C)(O)CC1 ZINC000217565387 CE In-Stock Unstable TP53BP1 0 40 COc1ccc(Cl)cc1C(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217565389 FH In-Stock Unstable AVPR1A 0 51 COc1ccc(Cl)cc1C(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217565389 FH In-Stock Unstable CHRM5 38 42 COc1ccc(Cl)cc1C(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217565389 FH In-Stock Unstable NPY5R 26 44 Cc1cc(O)ccc1NC(=O)NCC1CCCC1 ZINC000217565398 BG For-Sale Unstable THRB 16 42 Cc1cc(O)ccc1NC(=O)NCC1CCCC1 ZINC000217565398 BG For-Sale Unstable LDLR 0 47 COC(=O)CS[C@@H]1CCN(C(=O)c2ccc3ccccc3n2)C1 ZINC000217565414 EE In-Stock Unstable SMO 54 38 CCc1ccc(-c2nc(CC(=O)NCc3ccc(F)c(C)c3)cs2)cc1 ZINC000217565437 FJ On-Demand Unstable P2RX7 30 40 CCc1ccc(-c2nc(CC(=O)NCc3ccc(F)c(C)c3)cs2)cc1 ZINC000217565437 FJ On-Demand Unstable SUCNR1 51 37 Cc1cccc2nc(CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)cc(=O)n12 ZINC000217565456 FD In-Stock Unstable CHRNA4 33 55 CN(C)c1ccccc1C(=O)N1CCC[C@](C)(O)CC1 ZINC000217565462 CE In-Stock Unstable L3MBTL1 0 40 CN(C)c1ccccc1C(=O)N1CCC[C@](C)(O)CC1 ZINC000217565462 CE In-Stock Unstable TP53BP1 0 40 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)(C)C)cc2C(=O)O)cc1OC ZINC000217565463 IG In-Stock Unstable PTGDR 20 42 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)(C)C)cc2C(=O)O)cc1OC ZINC000217565463 IG In-Stock Unstable IAP 0 42 COc1ccc(CCNc2ccc(S(=O)(=O)NC(C)(C)C)cc2C(=O)O)cc1OC ZINC000217565463 IG In-Stock Unstable SCMU_MYCTU 0 49 COc1ccc(-c2ccc3nnc([C@H](N)C(C)C)n3n2)cc1 ZINC000217565466 CE In-Stock Unstable MET 15 41 COc1ccc(Cl)cc1C(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217565471 FH In-Stock Unstable AVPR1A 0 51 COc1ccc(Cl)cc1C(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217565471 FH In-Stock Unstable CHRM5 38 42 COc1ccc(Cl)cc1C(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217565471 FH In-Stock Unstable NPY5R 26 44 COC(=O)CS[C@H]1CCN(C(=O)c2ccc3ccccc3n2)C1 ZINC000217565482 EE In-Stock Unstable SMO 54 38 O=C1O[C@@]2(CCCN(C(=O)c3cc(-c4ccccc4)on3)C2)c2ccccc21 ZINC000217565557 FH For-Sale Unstable NPY5R 44 46 COc1ccc(-c2ccc3nnc([C@@H](N)C(C)C)n3n2)cc1OC ZINC000217565577 EE In-Stock Unstable PRKDC 0 40 COc1ccc(-c2ccc3nnc([C@@H](N)C(C)C)n3n2)cc1OC ZINC000217565577 EE In-Stock Unstable PDE4D 51 45 COc1ccc(-c2ccc3nnc([C@@H](N)C(C)C)n3n2)cc1OC ZINC000217565577 EE In-Stock Unstable MET 15 48 Cn1c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c(O)c1CN1CCN(C/C=C/c2ccccc2)CC1 ZINC000217565579 KF In-Stock Unstable CHRNA4 28 48 COc1ccc([C@@H](C)NC(=O)NCC2CCCC2)cc1 ZINC000217565612 CG On-Demand Unstable SDH1 0 40 COc1ccc([C@@H](C)NC(=O)NCC2CCCC2)cc1 ZINC000217565612 CG On-Demand Unstable MTR1B_CHICK 0 40 COc1ccc([C@@H](C)NC(=O)NCC2CCCC2)cc1 ZINC000217565612 CG On-Demand Unstable ACACB 35 40 O=C1O[C@]2(CCCN(C(=O)c3cc(-c4ccccc4)on3)C2)c2ccccc21 ZINC000217565648 FH For-Sale Unstable NPY5R 44 46 COc1ccc(-c2ccc3nnc([C@H](N)C(C)C)n3n2)cc1OC ZINC000217565656 EE In-Stock Unstable PRKDC 0 40 COc1ccc(-c2ccc3nnc([C@H](N)C(C)C)n3n2)cc1OC ZINC000217565656 EE In-Stock Unstable PDE4D 51 45 COc1ccc(-c2ccc3nnc([C@H](N)C(C)C)n3n2)cc1OC ZINC000217565656 EE In-Stock Unstable MET 15 48 COc1ccc2c(CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)cc(=O)oc2c1 ZINC000217565676 GF In-Stock Unstable CYP19A1 20 47 COc1ccc2c(CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)cc(=O)oc2c1 ZINC000217565676 GF In-Stock Unstable CYP11B1 19 43 COc1ccc2c(CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)cc(=O)oc2c1 ZINC000217565676 GF In-Stock Unstable CHRNA4 31 52 COc1ccc2c(CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)cc(=O)oc2c1 ZINC000217565676 GF In-Stock Unstable CYP11B2 0 43 COc1ccc([C@H](C)NC(=O)NCC2CCCC2)cc1 ZINC000217565694 CG On-Demand Unstable SDH1 0 40 COc1ccc([C@H](C)NC(=O)NCC2CCCC2)cc1 ZINC000217565694 CG On-Demand Unstable MTR1B_CHICK 0 40 COc1ccc([C@H](C)NC(=O)NCC2CCCC2)cc1 ZINC000217565694 CG On-Demand Unstable ACACB 35 40 CC(C)(C)NS(=O)(=O)c1ccc(NC[C@@H]2CCCO2)c(C(=O)O)c1 ZINC000217565698 FE In-Stock Unstable BDKRB1 22 42 CC(C)(C)NS(=O)(=O)c1ccc(NC[C@@H]2CCCO2)c(C(=O)O)c1 ZINC000217565698 FE In-Stock Unstable TNK2 42 38 CCOC(=O)[C@@H](C)NC(=O)[C@@H]1CC[C@@H](C)O1 ZINC000217565726 BC For-Sale Unstable METAP2 23 42 O=C1O[C@@]2(CCCN(C(=O)c3cccc(C(F)(F)F)c3)C2)c2ccccc21 ZINC000217565761 GI For-Sale Unstable CHRM5 40 48 O=C1O[C@@]2(CCCN(C(=O)c3cccc(C(F)(F)F)c3)C2)c2ccccc21 ZINC000217565761 GI For-Sale Unstable NPY5R 27 44 COc1ccc(OC)c(-c2ccc3nnc([C@@H](N)C(C)C)n3n2)c1 ZINC000217565769 EE In-Stock Unstable LRRK2 26 43 CC(C)(C)NS(=O)(=O)c1ccc(NC[C@H]2CCCO2)c(C(=O)O)c1 ZINC000217565785 FE In-Stock Unstable BDKRB1 22 42 CC(C)(C)NS(=O)(=O)c1ccc(NC[C@H]2CCCO2)c(C(=O)O)c1 ZINC000217565785 FE In-Stock Unstable TNK2 42 38 COC(=O)CS[C@H]1CCN(C(=O)c2ccc(C(C)(C)C)cc2)C1 ZINC000217565789 EG In-Stock Unstable L3MBTL3 63 38 CCOC(=O)[C@H](C)NC(=O)[C@@H]1CC[C@@H](C)O1 ZINC000217565806 BC On-Demand Unstable METAP2 23 42 O=c1[nH]c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)nc2cc(Cl)ccc12 ZINC000217565809 GE In-Stock Unstable CHRNA4 40 55 O=C(/C=C\c1ccc(O)cc1)N[C@@H]1CC[C@H](C(=O)O)C1 ZINC000217565816 CD For-Sale Unstable F3 27 44 O=C(/C=C\c1ccc(O)cc1)N[C@@H]1CC[C@H](C(=O)O)C1 ZINC000217565816 CD For-Sale Unstable MMP2 20 48 O=C(/C=C\c1ccc(O)cc1)N[C@@H]1CC[C@H](C(=O)O)C1 ZINC000217565816 CD For-Sale Unstable MMP9 19 48 O=C(/C=C\c1ccc(O)cc1)N[C@@H]1CC[C@H](C(=O)O)C1 ZINC000217565816 CD For-Sale Unstable MMP1 23 48 O=C(/C=C\c1ccc(O)cc1)N[C@@H]1CC[C@H](C(=O)O)C1 ZINC000217565816 CD For-Sale Unstable SSSIM 15 45 O=C1O[C@]2(CCCN(C(=O)c3cccc(C(F)(F)F)c3)C2)c2ccccc21 ZINC000217565851 GI For-Sale Unstable CHRM5 40 48 O=C1O[C@]2(CCCN(C(=O)c3cccc(C(F)(F)F)c3)C2)c2ccccc21 ZINC000217565851 GI For-Sale Unstable NPY5R 27 44 O=C(CN1CCC[C@@H]2CCCC[C@H]21)c1cccc(F)c1 ZINC000217565861 CH For-Sale Unstable GRM5 0 43 COc1ccc(OC)c(-c2ccc3nnc([C@H](N)C(C)C)n3n2)c1 ZINC000217565863 EE In-Stock Unstable LRRK2 26 43 COC(=O)CS[C@@H]1CCN(C(=O)c2ccc(C(C)(C)C)cc2)C1 ZINC000217565874 EG In-Stock Unstable L3MBTL3 63 38 CCOC(=O)[C@@H](C)NC(=O)[C@H]1CC[C@@H](C)O1 ZINC000217565883 BC For-Sale Unstable METAP2 23 42 O=C(CC1(n2cccc2)CCCCC1)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217565902 GG In-Stock Unstable CHRNA4 30 47 CC(C)(C)NS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217565904 EE In-Stock Unstable SLC6A9 20 45 CC(C)(C)NS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217565904 EE In-Stock Unstable SFRP1 88 34 CC(C)(C)NS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217565904 EE In-Stock Unstable WNT3 72 34 O=C(CN1CCC[C@H]2CCCC[C@H]21)c1cccc(F)c1 ZINC000217565951 CH For-Sale Unstable GRM5 0 43 CCOC(=O)[C@H](C)NC(=O)[C@H]1CC[C@@H](C)O1 ZINC000217565966 BC On-Demand Unstable METAP2 23 42 O=C1O[C@@]2(CCCN(C(=O)c3ccc(C(F)(F)F)cc3)C2)c2ccccc21 ZINC000217565969 GI For-Sale Unstable CHRM5 24 45 O=C1O[C@@]2(CCCN(C(=O)c3ccc(C(F)(F)F)cc3)C2)c2ccccc21 ZINC000217565969 GI For-Sale Unstable NPY5R 26 51 O=C1O[C@@]2(CCCN(C(=O)c3ccc(C(F)(F)F)cc3)C2)c2ccccc21 ZINC000217565969 GI For-Sale Unstable MLYCD 18 40 CC(C)(C)NS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217566014 EE In-Stock Unstable SLC6A9 20 46 CC(C)(C)NS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217566014 EE In-Stock Unstable SFRP1 81 33 CC(C)(C)NS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217566014 EE In-Stock Unstable WNT3 66 33 CC[C@@H](NC(=O)NCC1CCCC1)c1ccc2c(c1)CCCC2 ZINC000217566016 DJ For-Sale Unstable MTR1B_CHICK 0 41 COc1cc(C(C)C)c([C@H](O)CN)cc1Cl ZINC000217566022 BE For-Sale Unstable P2RX2 78 44 COc1cc(C(C)C)c([C@H](O)CN)cc1Cl ZINC000217566022 BE For-Sale Unstable P2RX3 56 33 O=C1O[C@]2(CCCN(C(=O)c3ccc(C(F)(F)F)cc3)C2)c2ccccc21 ZINC000217566052 GI For-Sale Unstable CHRM5 24 45 O=C1O[C@]2(CCCN(C(=O)c3ccc(C(F)(F)F)cc3)C2)c2ccccc21 ZINC000217566052 GI For-Sale Unstable NPY5R 26 51 O=C1O[C@]2(CCCN(C(=O)c3ccc(C(F)(F)F)cc3)C2)c2ccccc21 ZINC000217566052 GI For-Sale Unstable MLYCD 18 40 O=c1cccc2n1C[C@H]1C[C@@H]2CN(Cc2nc(-c3ccco3)no2)C1 ZINC000217566065 EE In-Stock Unstable CHRNA4 33 54 COc1cc(C(C)C)c([C@@H](O)CN)cc1Cl ZINC000217566097 BE For-Sale Unstable P2RX2 78 44 COc1cc(C(C)C)c([C@@H](O)CN)cc1Cl ZINC000217566097 BE For-Sale Unstable P2RX3 56 33 CC[C@H](NC(=O)NCC1CCCC1)c1ccc2c(c1)CCCC2 ZINC000217566101 DJ For-Sale Unstable MTR1B_CHICK 0 41 CC(C)(C)NS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1 ZINC000217566120 ED In-Stock Unstable SLC6A9 23 49 CC[C@@H](C(=O)N[C@@H](c1ccccc1)C1CC1)c1ccccc1 ZINC000217566140 CI On-Demand Unstable KCNQ2 53 46 CC[C@@H](C(=O)N[C@@H](c1ccccc1)C1CC1)c1ccccc1 ZINC000217566140 CI On-Demand Unstable TACR3 37 42 CC[C@@H](C(=O)N[C@@H](c1ccccc1)C1CC1)c1ccccc1 ZINC000217566140 CI On-Demand Unstable XIAP 45 34 COC(=O)[C@@H]1CCCN1C[C@@H](C)CN ZINC000217566146 BC For-Sale Unstable HSD11B1 26 41 O=c1cccc2n1C[C@H]1C[C@@H]2CN(Cc2nnnn2-c2ccccc2)C1 ZINC000217566163 ED In-Stock Unstable CHRNA4 34 63 CC(C)[C@@H](N)c1nnc2ccc(-c3cccc(Br)c3)nn12 ZINC000217566172 EG In-Stock Unstable PDE1A 23 40 CC(C)[C@@H](N)c1nnc2ccc(-c3cccc(Br)c3)nn12 ZINC000217566172 EG In-Stock Unstable MET 15 43 COC(=O)CS[C@@H]1CCN(S(=O)(=O)c2ccccc2F)C1 ZINC000217566191 ED In-Stock Unstable EPHX2 19 47 COc1cc(C(C)C)c([C@H](N)CO)cc1Cl ZINC000217566202 BE For-Sale Unstable P2RX2 75 43 COc1cc(C(C)C)c([C@H](N)CO)cc1Cl ZINC000217566202 BE For-Sale Unstable P2RX3 59 38 N#Cc1ccc(C(=O)CN2CCC[C@@H]3CCCC[C@H]32)cc1 ZINC000217566211 CG For-Sale Unstable NR3C2 22 47 O=C(/C=C\c1cccc(F)c1)N[C@@H]1CC[C@H](C(=O)O)C1 ZINC000217566215 CE On-Demand Unstable MMP2 15 45 CC[C@H](C(=O)N[C@@H](c1ccccc1)C1CC1)c1ccccc1 ZINC000217566218 CI On-Demand Unstable KCNQ2 53 46 CC[C@H](C(=O)N[C@@H](c1ccccc1)C1CC1)c1ccccc1 ZINC000217566218 CI On-Demand Unstable TACR3 37 42 CC[C@H](C(=O)N[C@@H](c1ccccc1)C1CC1)c1ccccc1 ZINC000217566218 CI On-Demand Unstable XIAP 49 37 C[C@@H](NC(=O)NCC1CCCC1)c1ccc2c(c1)CCCC2 ZINC000217566223 DI For-Sale Unstable MTR1B_CHICK 0 40 COC(=O)[C@@H]1CCCN1C[C@@H](O)c1ccc(CN)cc1 ZINC000217566225 CC For-Sale Unstable FKBP1A 46 34 COC(=O)[C@@H]1CCCN1C[C@@H](O)c1ccc(CN)cc1 ZINC000217566225 CC For-Sale Unstable SLC6A3 20 42 COC(=O)[C@@H]1CCCN1C[C@@H](O)c1ccc(CN)cc1 ZINC000217566225 CC For-Sale Unstable LGMN 50 33 COc1ccc(N2CCN(Cc3c(O)c(=O)cc(CN4C[C@@H]5C[C@H](C4)c4cccc(=O)n4C5)n3C)CC2)cc1 ZINC000217566249 KE In-Stock Unstable CHRNA4 27 44 CC(C)[C@H](N)c1nnc2ccc(-c3cccc(Br)c3)nn12 ZINC000217566256 EG In-Stock Unstable PDE1A 23 40 CC(C)[C@H](N)c1nnc2ccc(-c3cccc(Br)c3)nn12 ZINC000217566256 EG In-Stock Unstable MET 15 43 COC(=O)CS[C@H]1CCN(S(=O)(=O)c2ccccc2F)C1 ZINC000217566273 ED In-Stock Unstable EPHX2 19 47 COc1cc(C(C)C)c([C@@H](N)CO)cc1Cl ZINC000217566280 BE For-Sale Unstable P2RX2 75 43 COc1cc(C(C)C)c([C@@H](N)CO)cc1Cl ZINC000217566280 BE For-Sale Unstable P2RX3 59 38 C[C@H](NC(=O)NCC1CCCC1)c1ccc2c(c1)CCCC2 ZINC000217566297 DI For-Sale Unstable MTR1B_CHICK 0 40 N#Cc1ccc(C(=O)CN2CCC[C@H]3CCCC[C@H]32)cc1 ZINC000217566298 CG For-Sale Unstable NR3C2 22 47 CC[C@@H](C(=O)N[C@H](c1ccccc1)C1CC1)c1ccccc1 ZINC000217566304 CI On-Demand Unstable KCNQ2 53 46 CC[C@@H](C(=O)N[C@H](c1ccccc1)C1CC1)c1ccccc1 ZINC000217566304 CI On-Demand Unstable TACR3 37 42 CC[C@@H](C(=O)N[C@H](c1ccccc1)C1CC1)c1ccccc1 ZINC000217566304 CI On-Demand Unstable XIAP 49 37 COC(=O)[C@H]1CCCN1C[C@@H](O)c1ccc(CN)cc1 ZINC000217566319 CC For-Sale Unstable FKBP1A 46 34 COC(=O)[C@H]1CCCN1C[C@@H](O)c1ccc(CN)cc1 ZINC000217566319 CC For-Sale Unstable SLC6A3 20 42 COC(=O)[C@H]1CCCN1C[C@@H](O)c1ccc(CN)cc1 ZINC000217566319 CC For-Sale Unstable LGMN 50 33 Cn1c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c(O)c1CN1CCC(c2ccccc2)CC1 ZINC000217566340 KG In-Stock Unstable CHRNA4 30 52 NCCc1nnc2ccc(-c3cccc(Br)c3)nn12 ZINC000217566353 DE In-Stock Unstable MET 20 43 O=C1O[C@@]2(CCCN(C(=O)c3cc4ccccc4oc3=O)C2)c2ccccc21 ZINC000217566363 GG For-Sale Unstable NPY5R 29 41 CC[C@H](C(=O)N[C@H](c1ccccc1)C1CC1)c1ccccc1 ZINC000217566378 CI On-Demand Unstable KCNQ2 53 46 CC[C@H](C(=O)N[C@H](c1ccccc1)C1CC1)c1ccccc1 ZINC000217566378 CI On-Demand Unstable TACR3 37 42 CC[C@H](C(=O)N[C@H](c1ccccc1)C1CC1)c1ccccc1 ZINC000217566378 CI On-Demand Unstable XIAP 49 37 CCc1ccc(C(=O)CN2CCC[C@@H]3CCCC[C@H]32)cc1 ZINC000217566388 CI For-Sale Unstable HRH3 18 40 COc1cc([N+](=O)[O-])ccc1NC(=O)NCC1CCCC1 ZINC000217566409 CF On-Demand Unstable EPHX1 0 56 COc1cc([N+](=O)[O-])ccc1NC(=O)NCC1CCCC1 ZINC000217566409 CF On-Demand Unstable CACNA1C 42 37 COc1cc([N+](=O)[O-])ccc1NC(=O)NCC1CCCC1 ZINC000217566409 CF On-Demand Unstable TBXA2R 26 43 COc1cc([N+](=O)[O-])ccc1NC(=O)NCC1CCCC1 ZINC000217566409 CF On-Demand Unstable CACNA1D 69 37 COc1cc([N+](=O)[O-])ccc1NC(=O)NCC1CCCC1 ZINC000217566409 CF On-Demand Unstable KCNMA1 25 54 COc1cc([N+](=O)[O-])ccc1NC(=O)NCC1CCCC1 ZINC000217566409 CF On-Demand Unstable SLC27A4 44 34 O=c1[nH]c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)nc2ccc(F)cc12 ZINC000217566429 FD In-Stock Unstable CHRNA4 34 62 COCCN1CCC(Nc2ncc(C#C[Si](C)(C)C)cn2)CC1 ZINC000217566435 EE For-Sale Unstable EHMT2 48 30 O=C1O[C@]2(CCCN(C(=O)c3cc4ccccc4oc3=O)C2)c2ccccc21 ZINC000217566437 GG For-Sale Unstable NPY5R 29 41 CCc1ccc(C(=O)CN2CCC[C@H]3CCCC[C@H]32)cc1 ZINC000217566484 CI For-Sale Unstable HRH3 18 40 NCCc1nnc2ccc(-c3ccc(Br)cc3)nn12 ZINC000217566487 DE In-Stock Unstable MET 18 40 COc1ccc(C(=O)CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc1OC ZINC000217566523 FE In-Stock Unstable CHRNA4 34 68 COc1ccc(C(=O)N[C@@H](c2ccccc2)C2CC2)c(O)c1 ZINC000217566546 CG On-Demand Unstable SOAT1 0 42 COc1ccc(C(=O)N[C@@H](c2ccccc2)C2CC2)c(O)c1 ZINC000217566546 CG On-Demand Unstable AKR1C2 51 35 COC(=O)[C@@H]1CCCN1[C@@H](C)CCN ZINC000217566595 BC For-Sale Unstable ACE 25 42 O=C(CN1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)c1ccc2c(c1)OCCO2 ZINC000217566597 FD In-Stock Unstable CHRNA4 34 68 NCCc1nnc2ccc(-c3ccc(Cl)cc3Cl)nn12 ZINC000217566608 DF In-Stock Unstable DPP4 27 42 NCCc1nnc2ccc(-c3ccc(Cl)cc3Cl)nn12 ZINC000217566608 DF In-Stock Unstable DPP8 41 32 COc1ccc(C(=O)N[C@H](c2ccccc2)C2CC2)c(O)c1 ZINC000217566632 CG On-Demand Unstable SOAT1 0 42 COc1ccc(C(=O)N[C@H](c2ccccc2)C2CC2)c(O)c1 ZINC000217566632 CG On-Demand Unstable AKR1C2 51 35 COc1ccc(-c2ccc3nnc(CCN)n3n2)cc1 ZINC000217566700 CD In-Stock Unstable MET 23 49 COC(=O)[C@@H]1CCCN1[C@@H](C)CN ZINC000217566716 AB For-Sale Unstable XPNPEP1 59 36 COC(=O)[C@@H]1CCCN1[C@@H](C)CN ZINC000217566716 AB For-Sale Unstable XPNPEP2 67 36 C[C@@H]1CSCCN1C(=O)c1cc(Br)ccc1O ZINC000217566737 DF For-Sale Unstable PYK 56 32 CCCCOc1ccc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217566742 GI For-Sale Unstable AVPR1A 18 43 CCCCOc1ccc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217566742 GI For-Sale Unstable PLA2G4B 51 35 CCCCOc1ccc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217566742 GI For-Sale Unstable NPY5R 23 41 COc1ccc(Cn2nc(-c3ccncc3)nc2C2(C(N)=O)CC2)cc1 ZINC000217566756 ED In-Stock Unstable PROKR1 43 31 O=C1COc2ccc(C(=O)CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)cc2N1 ZINC000217566781 GD In-Stock Unstable CHRNA4 32 64 CCc1ccc(S(=O)(=O)N2CC[C@H](SCC(=O)OC)C2)cc1 ZINC000217566786 ED In-Stock Unstable MMP13 47 41 CCc1ccc(S(=O)(=O)N2CC[C@H](SCC(=O)OC)C2)cc1 ZINC000217566786 ED In-Stock Unstable MMP2 29 41 CCc1ccc(S(=O)(=O)N2CC[C@H](SCC(=O)OC)C2)cc1 ZINC000217566786 ED In-Stock Unstable MMP3 45 41 CCc1ccc(S(=O)(=O)N2CC[C@H](SCC(=O)OC)C2)cc1 ZINC000217566786 ED In-Stock Unstable MMP8 17 41 CCc1ccc(S(=O)(=O)N2CC[C@H](SCC(=O)OC)C2)cc1 ZINC000217566786 ED In-Stock Unstable MMP9 30 42 CCc1ccc(S(=O)(=O)N2CC[C@H](SCC(=O)OC)C2)cc1 ZINC000217566786 ED In-Stock Unstable TGM2 49 36 CCc1ccc(S(=O)(=O)N2CC[C@H](SCC(=O)OC)C2)cc1 ZINC000217566786 ED In-Stock Unstable MMP7 60 41 CCc1ccc(S(=O)(=O)N2CC[C@H](SCC(=O)OC)C2)cc1 ZINC000217566786 ED In-Stock Unstable MMP1 44 37 CCc1ccc(S(=O)(=O)N2CC[C@H](SCC(=O)OC)C2)cc1 ZINC000217566786 ED In-Stock Unstable F13A1 50 36 COc1ccc(-c2ccc3nnc(CCN)n3n2)cc1OC ZINC000217566807 CD In-Stock Unstable PDE4D 42 42 COc1ccc(-c2ccc3nnc(CCN)n3n2)cc1OC ZINC000217566807 CD In-Stock Unstable MET 23 47 CCCCOc1ccc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217566818 GI For-Sale Unstable AVPR1A 18 43 CCCCOc1ccc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217566818 GI For-Sale Unstable PLA2G4B 51 35 CCCCOc1ccc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217566818 GI For-Sale Unstable NPY5R 23 41 C[C@H]1CSCCN1C(=O)c1cc(Br)ccc1O ZINC000217566823 DF For-Sale Unstable PYK 56 32 COc1ccc(O)c(C(=O)N[C@@H](c2ccccc2)C2CC2)c1 ZINC000217566834 CG On-Demand Unstable TACR3 15 41 COc1ccc(O)c(C(=O)N[C@@H](c2ccccc2)C2CC2)c1 ZINC000217566834 CG On-Demand Unstable AKR1C2 40 34 CCc1ccc(S(=O)(=O)N2CC[C@@H](SCC(=O)OC)C2)cc1 ZINC000217566877 ED In-Stock Unstable MMP13 47 41 CCc1ccc(S(=O)(=O)N2CC[C@@H](SCC(=O)OC)C2)cc1 ZINC000217566877 ED In-Stock Unstable MMP2 29 41 CCc1ccc(S(=O)(=O)N2CC[C@@H](SCC(=O)OC)C2)cc1 ZINC000217566877 ED In-Stock Unstable MMP3 45 41 CCc1ccc(S(=O)(=O)N2CC[C@@H](SCC(=O)OC)C2)cc1 ZINC000217566877 ED In-Stock Unstable MMP8 17 41 CCc1ccc(S(=O)(=O)N2CC[C@@H](SCC(=O)OC)C2)cc1 ZINC000217566877 ED In-Stock Unstable MMP9 30 42 CCc1ccc(S(=O)(=O)N2CC[C@@H](SCC(=O)OC)C2)cc1 ZINC000217566877 ED In-Stock Unstable TGM2 49 36 CCc1ccc(S(=O)(=O)N2CC[C@@H](SCC(=O)OC)C2)cc1 ZINC000217566877 ED In-Stock Unstable MMP7 60 41 CCc1ccc(S(=O)(=O)N2CC[C@@H](SCC(=O)OC)C2)cc1 ZINC000217566877 ED In-Stock Unstable MMP1 44 37 CCc1ccc(S(=O)(=O)N2CC[C@@H](SCC(=O)OC)C2)cc1 ZINC000217566877 ED In-Stock Unstable F13A1 50 36 CCNC(=O)c1ccc(N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)c(NC(C)=O)c1 ZINC000217566879 GE In-Stock Unstable CHRNA4 28 49 O=C(O)c1ccccc1C(=O)N1CC2CCC(CC2)C1 ZINC000217566893 CF In-Stock Unstable SLC6A1 40 33 O=C(O)c1ccccc1C(=O)N1CC2CCC(CC2)C1 ZINC000217566893 CF In-Stock Unstable VACHT_TETCF 0 42 O=C(O)c1ccccc1C(=O)N1CC2CCC(CC2)C1 ZINC000217566893 CF In-Stock Unstable HSD11B1 0 41 O=C(O)c1ccccc1C(=O)N1CC2CCC(CC2)C1 ZINC000217566893 CF In-Stock Unstable L3MBTL1 0 54 O=C(O)c1ccccc1C(=O)N1CC2CCC(CC2)C1 ZINC000217566893 CF In-Stock Unstable L3MBTL3 57 43 O=C(O)c1ccccc1C(=O)N1CC2CCC(CC2)C1 ZINC000217566893 CF In-Stock Unstable MBTD1 0 43 O=C(O)c1ccccc1C(=O)N1CC2CCC(CC2)C1 ZINC000217566893 CF In-Stock Unstable TP53BP1 0 54 COc1ccc(O)c(C(=O)N[C@H](c2ccccc2)C2CC2)c1 ZINC000217566895 CG On-Demand Unstable TACR3 15 41 COc1ccc(O)c(C(=O)N[C@H](c2ccccc2)C2CC2)c1 ZINC000217566895 CG On-Demand Unstable AKR1C2 40 34 N[C@@H]1CC[C@@H](c2ccccc2)C[C@@H]1N1CCCOCC1 ZINC000217566907 CE For-Sale Unstable SLC18A3 50 40 COc1ccc(OC)c(-c2ccc3nnc(CCN)n3n2)c1 ZINC000217566910 CD In-Stock Unstable MET 17 45 COc1ccc(OC)c(-c2ccc3nnc(CCN)n3n2)c1 ZINC000217566910 CD In-Stock Unstable LRRK2 29 43 CCCCOC(=O)c1ccccc1NC(=O)NCC1CCCC1 ZINC000217566942 DH For-Sale Unstable AMY2 45 31 CC(C)c1ccc(OCC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217566943 GH For-Sale Unstable NPY5R 23 41 O=C(CCCC[C@@H]1CCSS1)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217566958 GH In-Stock Unstable CHRNA4 30 52 N[C@H]1CC[C@@H](c2ccccc2)C[C@@H]1N1CCCOCC1 ZINC000217566996 CE For-Sale Unstable SLC18A3 50 40 C=CCNS(=O)(=O)c1ccc(NCCC)c(C(=O)O)c1 ZINC000217567006 CD In-Stock Unstable CASP3 0 40 COC(=O)CS[C@H]1CCN(S(=O)(=O)c2cc(C)ccc2C)C1 ZINC000217567007 ED In-Stock Unstable EPHX2 34 43 O=C(CCCC[C@H]1CCSS1)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217567041 GH In-Stock Unstable CHRNA4 30 52 CC(C)c1ccc(OCC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217567049 GH For-Sale Unstable NPY5R 23 41 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N[C@@H](c2ccccc2)C2CC2)[C@@H](C)O)cc1 ZINC000217567070 HE On-Demand Unstable MMP13 47 48 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N[C@@H](c2ccccc2)C2CC2)[C@@H](C)O)cc1 ZINC000217567070 HE On-Demand Unstable CAPNS1 25 40 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N[C@@H](c2ccccc2)C2CC2)[C@@H](C)O)cc1 ZINC000217567070 HE On-Demand Unstable MMP2 39 48 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N[C@@H](c2ccccc2)C2CC2)[C@@H](C)O)cc1 ZINC000217567070 HE On-Demand Unstable MMP3 21 48 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N[C@@H](c2ccccc2)C2CC2)[C@@H](C)O)cc1 ZINC000217567070 HE On-Demand Unstable MMP8 16 44 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N[C@@H](c2ccccc2)C2CC2)[C@@H](C)O)cc1 ZINC000217567070 HE On-Demand Unstable MMP14 16 41 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N[C@@H](c2ccccc2)C2CC2)[C@@H](C)O)cc1 ZINC000217567070 HE On-Demand Unstable CAPN1 21 40 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N[C@@H](c2ccccc2)C2CC2)[C@@H](C)O)cc1 ZINC000217567070 HE On-Demand Unstable MMP9 19 41 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N[C@@H](c2ccccc2)C2CC2)[C@@H](C)O)cc1 ZINC000217567070 HE On-Demand Unstable MMP12 50 44 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N[C@@H](c2ccccc2)C2CC2)[C@@H](C)O)cc1 ZINC000217567070 HE On-Demand Unstable MMP7 16 44 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N[C@@H](c2ccccc2)C2CC2)[C@@H](C)O)cc1 ZINC000217567070 HE On-Demand Unstable ADAMTS4 61 35 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N[C@@H](c2ccccc2)C2CC2)[C@@H](C)O)cc1 ZINC000217567070 HE On-Demand Unstable LEF 24 41 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N[C@@H](c2ccccc2)C2CC2)[C@@H](C)O)cc1 ZINC000217567070 HE On-Demand Unstable BIRC8 44 31 CN1CCC[C@@H](CN[C@H](c2ccc(Cl)cc2)C2CC2)C1 ZINC000217567071 CH On-Demand Unstable SLC6A1 40 37 COC(=O)CS[C@@H]1CCN(S(=O)(=O)c2cc(C)ccc2C)C1 ZINC000217567077 ED In-Stock Unstable EPHX2 34 43 N[C@@H]1CC[C@H](c2ccccc2)C[C@@H]1N1CCCOCC1 ZINC000217567087 CE For-Sale Unstable SLC18A3 50 40 O=c1cccc2n1C[C@H]1C[C@@H]2CN(Cc2nc(-c3ccccc3)no2)C1 ZINC000217567116 EF In-Stock Unstable CHRNA4 34 62 O=c1cccc2n1C[C@H]1C[C@@H]2CN(Cc2nc(-c3ccccc3)no2)C1 ZINC000217567116 EF In-Stock Unstable GRM5 15 40 Cc1ccc(/C=C\C(=O)N[C@@H]2CC[C@H](C(=O)O)C2)cc1Cl ZINC000217567143 DG For-Sale Unstable PYGL 24 42 COc1ccc(CC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1OC ZINC000217567158 GF In-Stock Unstable NPY5R 24 43 CN1CCC[C@H](CN[C@H](c2ccc(Cl)cc2)C2CC2)C1 ZINC000217567160 CH On-Demand Unstable SLC6A1 40 37 Nc1ccc(NC(=O)NCC2CCCC2)c(Cl)c1 ZINC000217567164 CG For-Sale Unstable CACNA1I 45 36 N[C@H]1CC[C@H](c2ccccc2)C[C@@H]1N1CCCOCC1 ZINC000217567168 CE For-Sale Unstable SLC18A3 50 40 COC(=O)CS[C@H]1CCN(S(=O)(=O)c2ccc(F)c(C)c2)C1 ZINC000217567173 ED In-Stock Unstable LEF 70 39 C=CCNS(=O)(=O)c1ccc(NCCCC)c(C(=O)O)c1 ZINC000217567211 DE In-Stock Unstable CASP3 0 41 C=CCNS(=O)(=O)c1ccc(NCCCC)c(C(=O)O)c1 ZINC000217567211 DE In-Stock Unstable BDKRB1 0 40 Cc1c(O)ccc(/C=C/C(=O)O)c1C ZINC000217567212 AE For-Sale Unstable PTGER2 38 40 Cn1c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c(O)c1CN1CCSCC1 ZINC000217567222 ID In-Stock Unstable CHRNA4 30 49 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N[C@H](c2ccccc2)C2CC2)[C@@H](C)O)cc1 ZINC000217567229 HE On-Demand Unstable MMP13 47 48 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N[C@H](c2ccccc2)C2CC2)[C@@H](C)O)cc1 ZINC000217567229 HE On-Demand Unstable CAPNS1 25 40 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N[C@H](c2ccccc2)C2CC2)[C@@H](C)O)cc1 ZINC000217567229 HE On-Demand Unstable MMP2 39 48 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N[C@H](c2ccccc2)C2CC2)[C@@H](C)O)cc1 ZINC000217567229 HE On-Demand Unstable MMP3 21 48 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N[C@H](c2ccccc2)C2CC2)[C@@H](C)O)cc1 ZINC000217567229 HE On-Demand Unstable MMP8 16 44 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N[C@H](c2ccccc2)C2CC2)[C@@H](C)O)cc1 ZINC000217567229 HE On-Demand Unstable MMP14 16 41 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N[C@H](c2ccccc2)C2CC2)[C@@H](C)O)cc1 ZINC000217567229 HE On-Demand Unstable CAPN1 21 40 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N[C@H](c2ccccc2)C2CC2)[C@@H](C)O)cc1 ZINC000217567229 HE On-Demand Unstable MMP9 19 41 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N[C@H](c2ccccc2)C2CC2)[C@@H](C)O)cc1 ZINC000217567229 HE On-Demand Unstable MMP12 50 44 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N[C@H](c2ccccc2)C2CC2)[C@@H](C)O)cc1 ZINC000217567229 HE On-Demand Unstable MMP7 16 44 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N[C@H](c2ccccc2)C2CC2)[C@@H](C)O)cc1 ZINC000217567229 HE On-Demand Unstable ADAMTS4 61 35 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N[C@H](c2ccccc2)C2CC2)[C@@H](C)O)cc1 ZINC000217567229 HE On-Demand Unstable LEF 24 41 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N[C@H](c2ccccc2)C2CC2)[C@@H](C)O)cc1 ZINC000217567229 HE On-Demand Unstable BIRC8 44 31 COc1ccc(CC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1OC ZINC000217567241 GF In-Stock Unstable NPY5R 24 43 COC(=O)CS[C@@H]1CCN(S(=O)(=O)c2ccc(F)c(C)c2)C1 ZINC000217567259 ED In-Stock Unstable LEF 70 39 Nc1ccc(NC(=O)NCC2CCCC2)cc1Cl ZINC000217567263 CG For-Sale Unstable HTR4 30 42 Nc1ccc(NC(=O)NCC2CCCC2)cc1Cl ZINC000217567263 CG For-Sale Unstable EPHX2 20 63 Nc1ccc(NC(=O)NCC2CCCC2)cc1Cl ZINC000217567263 CG For-Sale Unstable CACNA1I 41 34 Nc1ccc(NC(=O)NCC2CCCC2)cc1Cl ZINC000217567263 CG For-Sale Unstable PRMT3 34 41 C=CCNS(=O)(=O)c1ccc(NCC(C)C)c(C(=O)O)c1 ZINC000217567311 DD In-Stock Unstable BDKRB1 0 43 C=CCNS(=O)(=O)c1ccc(NCC(C)C)c(C(=O)O)c1 ZINC000217567311 DD In-Stock Unstable F3 46 35 C=CCNS(=O)(=O)c1ccc(NCC(C)C)c(C(=O)O)c1 ZINC000217567311 DD In-Stock Unstable MTNN 40 33 CCNC(=O)c1ccc(N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)c(NC(=O)C(=O)OCC)c1 ZINC000217567325 JD In-Stock Unstable CHRNA4 26 42 CCOc1ccc(OCC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217567343 GG For-Sale Unstable COLA 26 41 CCOc1ccc(OCC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217567343 GG For-Sale Unstable CPT1A 24 41 CCOc1ccc(OCC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217567343 GG For-Sale Unstable CPT2 35 41 CCOc1ccc(OCC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217567343 GG For-Sale Unstable NPY5R 27 42 C=CCN(CC=C)C(=O)NCC1CCCC1 ZINC000217567362 BF On-Demand Unstable ADH4 0 40 O=C(N[C@@H](c1ccccc1)C1CC1)c1cc(N2CCCC2)ccn1 ZINC000217567390 DH On-Demand Unstable AKT1 0 42 O=C(N[C@@H](c1ccccc1)C1CC1)c1cc(N2CCCC2)ccn1 ZINC000217567390 DH On-Demand Unstable TTK 36 41 COc1ccc(-c2ncccc2CO)cc1 ZINC000217567403 BE For-Sale Unstable PTGS1 15 40 COc1ccc(-c2ncccc2CO)cc1 ZINC000217567403 BE For-Sale Unstable CYP11B2 23 50 Cn1c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c(O)c1CN1CCN(CCOc2ccc(F)cc2)CC1 ZINC000217567410 KE In-Stock Unstable CHRNA4 36 51 CCOc1ccc(OCC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217567414 GG For-Sale Unstable COLA 26 41 CCOc1ccc(OCC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217567414 GG For-Sale Unstable CPT1A 24 41 CCOc1ccc(OCC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217567414 GG For-Sale Unstable CPT2 35 41 CCOc1ccc(OCC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217567414 GG For-Sale Unstable NPY5R 27 42 O=C(N[C@H](c1ccccc1)C1CC1)c1cc(N2CCCC2)ccn1 ZINC000217567462 DH On-Demand Unstable AKT1 0 42 O=C(N[C@H](c1ccccc1)C1CC1)c1cc(N2CCCC2)ccn1 ZINC000217567462 DH On-Demand Unstable TTK 36 41 CN1CCN(C(=O)NCC2CCCC2)CC1 ZINC000217567465 BD On-Demand Unstable CACNA1I 47 33 Cc1cccc(NC(=O)[C@@H]2CC[C@@H](CNC(=O)[C@@H]3Cc4ccccc4CN3)CC2)c1 ZINC000217567471 HH In-Stock Unstable CCKAR 23 40 Cc1cccc(NC(=O)[C@@H]2CC[C@@H](CNC(=O)[C@@H]3Cc4ccccc4CN3)CC2)c1 ZINC000217567471 HH In-Stock Unstable CCKBR 25 40 O=c1cccc2n1C[C@H]1C[C@@H]2CN(Cc2nnnn2-c2ccc(F)cc2)C1 ZINC000217567506 FD In-Stock Unstable CHRNA4 35 65 Cc1cccc(/C=C\C(=O)N[C@@H]2CC[C@H](C(=O)O)C2)c1 ZINC000217567526 CE On-Demand Unstable HDAC8 53 38 O=C(NCC1CCCC1)NC1CCCCCCCCCCC1 ZINC000217567551 DK For-Sale Unstable ADH1B 0 41 O=C(NCC1CCCC1)NC1CCCCCCCCCCC1 ZINC000217567551 DK For-Sale Unstable ADH1C 0 41 O=C(NCC1CCCC1)NC1CCCCCCCCCCC1 ZINC000217567551 DK For-Sale Unstable ADH4 0 41 O=C(NCC1CCCC1)NC1CCCCCCCCCCC1 ZINC000217567551 DK For-Sale Unstable EPHX2 31 56 O=C(NCC1CCCC1)NC1CCCCCCCCCCC1 ZINC000217567551 DK For-Sale Unstable P95276_MYCTO 0 43 COC(=O)CS[C@@H]1CCN(S(=O)(=O)c2cccc(Cl)c2)C1 ZINC000217567563 EE In-Stock Unstable FBP1 0 42 COC(=O)CS[C@@H]1CCN(S(=O)(=O)c2cccc(Cl)c2)C1 ZINC000217567563 EE In-Stock Unstable AKR1C3 43 37 CCCC[C@@H](N)C(=O)N[C@@]1(C(=O)O)CCC[C@@H](C)C1 ZINC000217567619 CD For-Sale Unstable DPP7 15 40 CCCC[C@@H](N)C(=O)N[C@@]1(C(=O)O)CCC[C@@H](C)C1 ZINC000217567619 CD For-Sale Unstable NOD1 40 32 COC(=O)CS[C@H]1CCN(S(=O)(=O)c2cccc(Cl)c2)C1 ZINC000217567636 EE In-Stock Unstable FBP1 0 42 COC(=O)CS[C@H]1CCN(S(=O)(=O)c2cccc(Cl)c2)C1 ZINC000217567636 EE In-Stock Unstable AKR1C3 43 37 COc1ccc(C(=O)Nc2cc(C(=O)NCc3ccccc3)ccc2N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc1 ZINC000217567643 KJ In-Stock Unstable CYSLTR2 42 33 COc1ccc(C(=O)Nc2cc(C(=O)NCc3ccccc3)ccc2N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc1 ZINC000217567643 KJ In-Stock Unstable CHRNA4 25 43 O=C1O[C@@]2(CCCN(C(=O)C3(c4ccccc4)CCOCC3)C2)c2ccccc21 ZINC000217567707 GG For-Sale Unstable NPY5R 28 41 CCCC[C@H](N)C(=O)N[C@@]1(C(=O)O)CCC[C@@H](C)C1 ZINC000217567710 CD For-Sale Unstable DPP7 15 40 CCCC[C@H](N)C(=O)N[C@@]1(C(=O)O)CCC[C@@H](C)C1 ZINC000217567710 CD For-Sale Unstable NOD1 40 32 COC(=O)CS[C@@H]1CCN(S(=O)(=O)c2ccccc2Cl)C1 ZINC000217567734 EE In-Stock Unstable CCR1 15 41 COC(=O)CS[C@@H]1CCN(S(=O)(=O)c2ccccc2Cl)C1 ZINC000217567734 EE In-Stock Unstable EPHX2 36 40 Cn1c(N)c(C(=O)CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)c(=O)n(C)c1=O ZINC000217567758 GB In-Stock Unstable CHRNA4 44 62 O=C(NCCN1CCNCC1)NCC1CCCC1 ZINC000217567766 CC On-Demand Unstable CACNA1H 15 40 O=C1O[C@]2(CCCN(C(=O)C3(c4ccccc4)CCOCC3)C2)c2ccccc21 ZINC000217567788 GG For-Sale Unstable NPY5R 28 41 CCCC[C@@H](N)C(=O)N[C@]1(C(=O)O)CCC[C@@H](C)C1 ZINC000217567789 CD For-Sale Unstable DPP7 15 40 CCCC[C@@H](N)C(=O)N[C@]1(C(=O)O)CCC[C@@H](C)C1 ZINC000217567789 CD For-Sale Unstable NOD1 40 32 COC(=O)CS[C@H]1CCN(S(=O)(=O)c2ccccc2Cl)C1 ZINC000217567827 EE In-Stock Unstable CCR1 15 41 COC(=O)CS[C@H]1CCN(S(=O)(=O)c2ccccc2Cl)C1 ZINC000217567827 EE In-Stock Unstable EPHX2 36 40 Cn1c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c(O)c1CN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217567850 KF In-Stock Unstable CHRNA4 27 46 CCN(C(=O)NCC1CCCC1)c1ccccc1 ZINC000217567868 BG For-Sale Unstable CHRM2 24 40 CCN(C(=O)NCC1CCCC1)c1ccccc1 ZINC000217567868 BG For-Sale Unstable CHRM1 27 40 CCN(C(=O)NCC1CCCC1)c1ccccc1 ZINC000217567868 BG For-Sale Unstable ACE 40 34 CCN(C(=O)NCC1CCCC1)c1ccccc1 ZINC000217567868 BG For-Sale Unstable CHRM3 29 40 CCN(C(=O)NCC1CCCC1)c1ccccc1 ZINC000217567868 BG For-Sale Unstable AMY2 61 38 CCN(C(=O)NCC1CCCC1)c1ccccc1 ZINC000217567868 BG For-Sale Unstable GPR88 0 41 CCCC[C@H](N)C(=O)N[C@]1(C(=O)O)CCC[C@@H](C)C1 ZINC000217567873 CD For-Sale Unstable DPP7 15 40 CCCC[C@H](N)C(=O)N[C@]1(C(=O)O)CCC[C@@H](C)C1 ZINC000217567873 CD For-Sale Unstable NOD1 40 32 CN1CC[C@@H](NC(=O)c2cc([N+](=O)[O-])ccc2F)C1=O ZINC000217567886 CC On-Demand Unstable WDR5 35 41 C=CCNS(=O)(=O)c1ccc(NC2CCCC2)c(C(=O)O)c1 ZINC000217567900 DE In-Stock Unstable CASP3 0 41 C=CCNS(=O)(=O)c1ccc(NC2CCCC2)c(C(=O)O)c1 ZINC000217567900 DE In-Stock Unstable F13A1 40 35 CS(=O)(=O)N1CCC(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)CC1 ZINC000217567903 GD For-Sale Unstable NPY5R 50 39 CCOC(=O)[C@@H]1CCCN1[C@@H]1C[C@@H](C)CC[C@@H]1CN ZINC000217567938 CD For-Sale Unstable FKBP12.6 0 43 CS(=O)(=O)N1CCC(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)CC1 ZINC000217567971 GD For-Sale Unstable NPY5R 50 39 CN1CC[C@H](NC(=O)c2cc([N+](=O)[O-])ccc2F)C1=O ZINC000217567972 CC On-Demand Unstable WDR5 35 41 NCc1cccc(CNC(=O)NCC2CCCC2)c1 ZINC000217567978 CE For-Sale Unstable TPSAB1 53 40 C=Cc1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217567984 AF For-Sale Unstable KDM4B 0 49 Cn1c(=O)c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc2ccccc21 ZINC000217567988 FE In-Stock Unstable CHRNA4 35 60 CCOC(=O)[C@H]1CCCN1[C@@H]1C[C@@H](C)CC[C@@H]1CN ZINC000217568017 CD For-Sale Unstable FKBP12.6 0 43 Cc1ccn2cc(-c3ccc(NC(=O)c4ccc5ncsc5c4)cc3)nc2c1 ZINC000217568028 GK For-Sale Unstable MAP3K5 48 33 O=C(NCC1CCCC1)Nc1cc(Cl)ccc1O ZINC000217568092 CG For-Sale Unstable EPHX2 15 61 O=C(NCC1CCCC1)Nc1cc(Cl)ccc1O ZINC000217568092 CG For-Sale Unstable KCNMA1 28 48 O=C(NCC1CCCC1)Nc1cc(Cl)ccc1O ZINC000217568092 CG For-Sale Unstable CACNA1I 51 36 CO[C@@H](C)C(=O)N[C@@H]1CCN(C)C1=O ZINC000217568116 BB On-Demand Unstable ACE 16 40 CO[C@@H](C)C(=O)N[C@@H]1CCN(C)C1=O ZINC000217568116 BB On-Demand Unstable BIRC2 40 33 Cn1c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c(O)c1CN1CCN(c2ccc(Cl)cc2)CC1 ZINC000217568118 KF In-Stock Unstable CHRNA4 28 47 COC(=O)CS[C@H]1CCN(S(=O)(=O)c2cc(Cl)ccc2OC)C1 ZINC000217568144 GE In-Stock Unstable AVPR1B 46 33 COC(=O)CS[C@H]1CCN(S(=O)(=O)c2cc(Cl)ccc2OC)C1 ZINC000217568144 GE In-Stock Unstable F10 15 49 COC(=O)CS[C@H]1CCN(S(=O)(=O)c2cc(Cl)ccc2OC)C1 ZINC000217568144 GE In-Stock Unstable COLA 105 45 COC(=O)CS[C@H]1CCN(S(=O)(=O)c2cc(Cl)ccc2OC)C1 ZINC000217568144 GE In-Stock Unstable CPT1A 98 45 COC(=O)CS[C@H]1CCN(S(=O)(=O)c2cc(Cl)ccc2OC)C1 ZINC000217568144 GE In-Stock Unstable CPT2 57 45 COC(=O)CS[C@H]1CCN(S(=O)(=O)c2cc(Cl)ccc2OC)C1 ZINC000217568144 GE In-Stock Unstable EPHX2 18 40 COC(=O)CS[C@H]1CCN(S(=O)(=O)c2cc(Cl)ccc2OC)C1 ZINC000217568144 GE In-Stock Unstable CPT1B 94 43 CO[C@H](C)C(=O)N[C@@H]1CCN(C)C1=O ZINC000217568195 BB On-Demand Unstable ACE 16 40 CO[C@H](C)C(=O)N[C@@H]1CCN(C)C1=O ZINC000217568195 BB On-Demand Unstable BIRC2 40 33 O=C(NCC1CCCC1)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217568206 HF For-Sale Unstable LPL 48 41 O=C(NCC1CCCC1)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217568206 HF For-Sale Unstable CNR2 0 41 O=C(NCC1CCCC1)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217568206 HF For-Sale Unstable CASP3 0 42 O=C(NCC1CCCC1)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217568206 HF For-Sale Unstable EPHX2 24 43 O=C(NCC1CCCC1)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217568206 HF For-Sale Unstable MURF 0 41 O=C(NCC1CCCC1)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217568206 HF For-Sale Unstable CACNA1I 59 36 O=C(NCC1CCCC1)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217568206 HF For-Sale Unstable F13A1 51 38 O=C(NCC1CCCC1)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217568206 HF For-Sale Unstable LIPG 20 41 O=C(NCC1CCCC1)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217568206 HF For-Sale Unstable NAMPT 39 43 COC(=O)CS[C@@H]1CCN(S(=O)(=O)c2cc(Cl)ccc2OC)C1 ZINC000217568221 GE In-Stock Unstable AVPR1B 46 33 COC(=O)CS[C@@H]1CCN(S(=O)(=O)c2cc(Cl)ccc2OC)C1 ZINC000217568221 GE In-Stock Unstable F10 15 49 COC(=O)CS[C@@H]1CCN(S(=O)(=O)c2cc(Cl)ccc2OC)C1 ZINC000217568221 GE In-Stock Unstable COLA 105 45 COC(=O)CS[C@@H]1CCN(S(=O)(=O)c2cc(Cl)ccc2OC)C1 ZINC000217568221 GE In-Stock Unstable CPT1A 98 45 COC(=O)CS[C@@H]1CCN(S(=O)(=O)c2cc(Cl)ccc2OC)C1 ZINC000217568221 GE In-Stock Unstable CPT2 57 45 COC(=O)CS[C@@H]1CCN(S(=O)(=O)c2cc(Cl)ccc2OC)C1 ZINC000217568221 GE In-Stock Unstable EPHX2 18 40 COC(=O)CS[C@@H]1CCN(S(=O)(=O)c2cc(Cl)ccc2OC)C1 ZINC000217568221 GE In-Stock Unstable CPT1B 94 43 CC(C)c1ccc2oc(=O)cc(CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)c2c1 ZINC000217568230 GH In-Stock Unstable CHRNA4 38 51 COc1cccc(/C=C\C(=O)N[C@@H]2CC[C@H](C(=O)O)C2)c1 ZINC000217568249 CE On-Demand Unstable MTNR1A 22 42 COc1cccc(/C=C\C(=O)N[C@@H]2CC[C@H](C(=O)O)C2)c1 ZINC000217568249 CE On-Demand Unstable MTNR1B 28 40 COc1cccc(/C=C\C(=O)N[C@@H]2CC[C@H](C(=O)O)C2)c1 ZINC000217568249 CE On-Demand Unstable HDA106 0 41 COc1cccc(/C=C\C(=O)N[C@@H]2CC[C@H](C(=O)O)C2)c1 ZINC000217568249 CE On-Demand Unstable HD1B 0 41 CC(C)(Oc1ccc(Cl)cc1)C(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217568250 GI For-Sale Unstable NPY5R 25 44 CO[C@@H](C)C(=O)N[C@H]1CCN(C)C1=O ZINC000217568265 BB On-Demand Unstable ACE 16 40 CO[C@@H](C)C(=O)N[C@H]1CCN(C)C1=O ZINC000217568265 BB On-Demand Unstable BIRC2 40 33 COC(=O)CS[C@@H]1CCN(S(=O)(=O)c2cccc(C(F)(F)F)c2)C1 ZINC000217568323 GE In-Stock Unstable CACNA1B 66 42 COC(=O)CS[C@@H]1CCN(S(=O)(=O)c2cccc(C(F)(F)F)c2)C1 ZINC000217568323 GE In-Stock Unstable BDKRB1 27 42 COC(=O)CS[C@@H]1CCN(S(=O)(=O)c2cccc(C(F)(F)F)c2)C1 ZINC000217568323 GE In-Stock Unstable CCR2 54 38 COC(=O)CS[C@@H]1CCN(S(=O)(=O)c2cccc(C(F)(F)F)c2)C1 ZINC000217568323 GE In-Stock Unstable AKR1C3 50 34 COC(=O)CS[C@@H]1CCN(S(=O)(=O)c2cccc(C(F)(F)F)c2)C1 ZINC000217568323 GE In-Stock Unstable SFRP1 45 35 COC(=O)CS[C@@H]1CCN(S(=O)(=O)c2cccc(C(F)(F)F)c2)C1 ZINC000217568323 GE In-Stock Unstable RHOA 0 41 CC(C)(Oc1ccc(Cl)cc1)C(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217568328 GI For-Sale Unstable NPY5R 25 44 Cn1c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)c(Br)c(=O)n(C)c1=O ZINC000217568332 HC In-Stock Unstable CHRNA4 36 60 CO[C@H](C)C(=O)N[C@H]1CCN(C)C1=O ZINC000217568354 BB On-Demand Unstable ACE 16 40 CO[C@H](C)C(=O)N[C@H]1CCN(C)C1=O ZINC000217568354 BB On-Demand Unstable BIRC2 40 33 COC(=O)CS[C@H]1CCN(S(=O)(=O)c2cccc(C(F)(F)F)c2)C1 ZINC000217568395 GE In-Stock Unstable CACNA1B 66 42 COC(=O)CS[C@H]1CCN(S(=O)(=O)c2cccc(C(F)(F)F)c2)C1 ZINC000217568395 GE In-Stock Unstable BDKRB1 27 42 COC(=O)CS[C@H]1CCN(S(=O)(=O)c2cccc(C(F)(F)F)c2)C1 ZINC000217568395 GE In-Stock Unstable CCR2 72 38 COC(=O)CS[C@H]1CCN(S(=O)(=O)c2cccc(C(F)(F)F)c2)C1 ZINC000217568395 GE In-Stock Unstable AKR1C3 50 34 COC(=O)CS[C@H]1CCN(S(=O)(=O)c2cccc(C(F)(F)F)c2)C1 ZINC000217568395 GE In-Stock Unstable SFRP1 50 37 COC(=O)CS[C@H]1CCN(S(=O)(=O)c2cccc(C(F)(F)F)c2)C1 ZINC000217568395 GE In-Stock Unstable RHOA 0 41 C=CCNS(=O)(=O)c1ccc(NCCOC)c(C(=O)O)c1 ZINC000217568431 DC In-Stock Unstable BDKRB1 0 42 COC(=O)CS[C@@H]1CCN(S(=O)(=O)c2ccccc2Br)C1 ZINC000217568497 GE In-Stock Unstable EPHX2 15 44 C[C@@H](CO)S(=O)(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217568524 CD For-Sale Unstable KIF11 0 53 C=CCNS(=O)(=O)c1ccc(NCCCOC)c(C(=O)O)c1 ZINC000217568545 ED In-Stock Unstable BDKRB1 17 42 COC(=O)CS[C@H]1CCN(S(=O)(=O)c2ccccc2Br)C1 ZINC000217568579 GE In-Stock Unstable EPHX2 15 44 C[C@H](CO)S(=O)(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217568603 CD For-Sale Unstable KIF11 0 53 O=C1O[C@@]2(CCCN(C(=O)C3c4ccccc4Oc4ccccc43)C2)c2ccccc21 ZINC000217568630 HJ For-Sale Unstable NPY5R 33 40 O=C1O[C@]2(CCCN(C(=O)C3c4ccccc4Oc4ccccc43)C2)c2ccccc21 ZINC000217568709 HJ For-Sale Unstable NPY5R 33 40 C=CCNS(=O)(=O)c1ccc(N[C@@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217568750 FG In-Stock Unstable BDKRB1 0 41 Cc1nc2ccc(F)cc2c(=O)n1CC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217568760 HD In-Stock Unstable CHRNA4 28 49 Cc1nc2ccc(F)cc2c(=O)n1CC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217568760 HD In-Stock Unstable Q8MHZ5_SHEEP 40 38 C=CCNS(=O)(=O)c1ccc(N[C@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217568830 FG In-Stock Unstable BDKRB1 0 41 COC(=O)CS[C@@H]1CCN(S(=O)(=O)Cc2ccccc2)C1 ZINC000217568860 ED In-Stock Unstable SIGMAR1 18 49 Cn1c(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c(O)c1CN1CCc2ccccc2C1 ZINC000217568903 JE In-Stock Unstable CHRNA4 30 49 C=CCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217568930 FF In-Stock Unstable BDKRB1 0 40 COC(=O)CS[C@H]1CCN(S(=O)(=O)Cc2ccccc2)C1 ZINC000217568935 ED In-Stock Unstable SIGMAR1 18 49 Cc1ccc(O)c(NC(=O)NCC2CCCC2)c1 ZINC000217568960 BG For-Sale Unstable THRA 20 44 Cc1ccc(O)c(NC(=O)NCC2CCCC2)c1 ZINC000217568960 BG For-Sale Unstable THRB 27 44 Cc1ccc(O)c(NC(=O)NCC2CCCC2)c1 ZINC000217568960 BG For-Sale Unstable KCNMA1 17 42 COc1ccc(Br)c(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217569004 HH For-Sale Unstable NPY5R 24 46 COc1ccc(Br)c(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217569004 HH For-Sale Unstable SCN5A 15 40 CC(C)C(=O)N[C@@H]1CCN(C)C1=O ZINC000217569008 AB On-Demand Unstable BIRC2 48 34 C=CCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217569051 GF In-Stock Unstable TBXA2R 32 40 C=CCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217569051 GF In-Stock Unstable BMP1 48 37 C=CCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217569051 GF In-Stock Unstable PTGDR 26 41 C=CCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217569051 GF In-Stock Unstable IAP 0 44 C=CCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217569051 GF In-Stock Unstable CA9 22 41 C=CCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217569051 GF In-Stock Unstable AKR1C3 27 42 C=CCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217569051 GF In-Stock Unstable FFAR4 15 40 C=CCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217569051 GF In-Stock Unstable AKR1C2 45 36 O=C(c1ccc2cc[nH]c2c1)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217569081 EF In-Stock Unstable CHRNA4 38 52 O=C(c1ccc2cc[nH]c2c1)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217569081 EF In-Stock Unstable GHSR 0 46 COc1ccc(Br)c(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217569083 HH For-Sale Unstable NPY5R 24 46 COc1ccc(Br)c(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217569083 HH For-Sale Unstable SCN5A 15 40 CC(C)C(=O)N[C@H]1CCN(C)C1=O ZINC000217569105 AB On-Demand Unstable BIRC2 48 34 C=CCNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217569160 HF In-Stock Unstable IAP 0 45 C=CCNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217569160 HF In-Stock Unstable SCMU_MYCTU 0 44 CCN(Cc1ccccc1)C(=O)NCC1CCCC1 ZINC000217569186 CG On-Demand Unstable OPRD1 22 42 CCN(Cc1ccccc1)C(=O)NCC1CCCC1 ZINC000217569186 CG On-Demand Unstable TSPO 31 40 CCN(Cc1ccccc1)C(=O)NCC1CCCC1 ZINC000217569186 CG On-Demand Unstable AMY2 47 34 CCN(Cc1ccccc1)C(=O)NCC1CCCC1 ZINC000217569186 CG On-Demand Unstable GHSR 0 40 CCN(Cc1ccccc1)C(=O)NCC1CCCC1 ZINC000217569186 CG On-Demand Unstable TRPM8 27 40 CCN(Cc1ccccc1)C(=O)NCC1CCCC1 ZINC000217569186 CG On-Demand Unstable PTGES 25 58 CCN(Cc1ccccc1)C(=O)NCC1CCCC1 ZINC000217569186 CG On-Demand Unstable LIMK2 42 36 COc1cc2c(cc1OC)CC(=O)N(CC(=O)N1C[C@@H]3C[C@H](C1)c1cccc(=O)n1C3)C=C2 ZINC000217569196 ID In-Stock Unstable CHRNA4 26 44 Cc1onc(-c2ccccc2Cl)c1C(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217569197 HJ For-Sale Unstable NPY5R 26 47 Cc1onc(-c2ccccc2Cl)c1C(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217569197 HJ For-Sale Unstable GPBAR1 30 43 CCCC(=O)N[C@@H]1CCN(C)C1=O ZINC000217569201 AC On-Demand Unstable LUXR 54 42 CCCC(=O)N[C@@H]1CCN(C)C1=O ZINC000217569201 AC On-Demand Unstable TRAR 24 41 CCCC(=O)N[C@@H]1CCN(C)C1=O ZINC000217569201 AC On-Demand Unstable LASR 32 41 CCCC(=O)N[C@@H]1CCN(C)C1=O ZINC000217569201 AC On-Demand Unstable PHZR 0 41 Cc1onc(-c2ccccc2Cl)c1C(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217569273 HJ For-Sale Unstable NPY5R 26 47 Cc1onc(-c2ccccc2Cl)c1C(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217569273 HJ For-Sale Unstable GPBAR1 30 43 CCCC(=O)N[C@H]1CCN(C)C1=O ZINC000217569276 AC On-Demand Unstable LUXR 54 42 CCCC(=O)N[C@H]1CCN(C)C1=O ZINC000217569276 AC On-Demand Unstable TRAR 24 41 CCCC(=O)N[C@H]1CCN(C)C1=O ZINC000217569276 AC On-Demand Unstable LASR 32 41 CCCC(=O)N[C@H]1CCN(C)C1=O ZINC000217569276 AC On-Demand Unstable PHZR 0 41 C=CCNS(=O)(=O)c1ccc(NC[C@@H]2CCCO2)c(C(=O)O)c1 ZINC000217569374 ED In-Stock Unstable BDKRB1 22 42 COC(=O)CS[C@@H]1CCN(S(=O)(=O)c2ccc(Oc3ccccc3Cl)cc2)C1 ZINC000217569435 IH In-Stock Unstable MMP13 58 42 COC(=O)CS[C@@H]1CCN(S(=O)(=O)c2ccc(Oc3ccccc3Cl)cc2)C1 ZINC000217569435 IH In-Stock Unstable MMP3 49 39 COC(=O)CS[C@@H]1CCN(S(=O)(=O)c2ccc(Oc3ccccc3Cl)cc2)C1 ZINC000217569435 IH In-Stock Unstable MMP9 43 39 COC(=O)CS[C@@H]1CCN(S(=O)(=O)c2ccc(Oc3ccccc3Cl)cc2)C1 ZINC000217569435 IH In-Stock Unstable EPHX2 16 41 COC(=O)CS[C@@H]1CCN(S(=O)(=O)c2ccc(Oc3ccccc3Cl)cc2)C1 ZINC000217569435 IH In-Stock Unstable TGM2 45 37 COC(=O)CS[C@@H]1CCN(S(=O)(=O)c2ccc(Oc3ccccc3Cl)cc2)C1 ZINC000217569435 IH In-Stock Unstable MMP7 55 39 COC(=O)CS[C@@H]1CCN(S(=O)(=O)c2ccc(Oc3ccccc3Cl)cc2)C1 ZINC000217569435 IH In-Stock Unstable MMP1 53 39 COC(=O)CS[C@@H]1CCN(S(=O)(=O)c2ccc(Oc3ccccc3Cl)cc2)C1 ZINC000217569435 IH In-Stock Unstable F13A1 49 36 Cc1ccn2cc(-c3ccc(NC(=O)c4cnn(-c5ccccc5)c4C(F)(F)F)cc3)nc2c1 ZINC000217569440 JK On-Demand Unstable MST1R 47 45 Cc1ccn2cc(-c3ccc(NC(=O)c4cnn(-c5ccccc5)c4C(F)(F)F)cc3)nc2c1 ZINC000217569440 JK On-Demand Unstable PDE10A 17 45 C=CCNS(=O)(=O)c1ccc(NC[C@H]2CCCO2)c(C(=O)O)c1 ZINC000217569463 ED In-Stock Unstable BDKRB1 22 42 COC(=O)CS[C@H]1CCN(S(=O)(=O)c2ccc(Oc3ccccc3Cl)cc2)C1 ZINC000217569518 IH In-Stock Unstable MMP13 58 42 COC(=O)CS[C@H]1CCN(S(=O)(=O)c2ccc(Oc3ccccc3Cl)cc2)C1 ZINC000217569518 IH In-Stock Unstable MMP3 49 39 COC(=O)CS[C@H]1CCN(S(=O)(=O)c2ccc(Oc3ccccc3Cl)cc2)C1 ZINC000217569518 IH In-Stock Unstable MMP9 43 39 COC(=O)CS[C@H]1CCN(S(=O)(=O)c2ccc(Oc3ccccc3Cl)cc2)C1 ZINC000217569518 IH In-Stock Unstable EPHX2 16 41 COC(=O)CS[C@H]1CCN(S(=O)(=O)c2ccc(Oc3ccccc3Cl)cc2)C1 ZINC000217569518 IH In-Stock Unstable TGM2 45 37 COC(=O)CS[C@H]1CCN(S(=O)(=O)c2ccc(Oc3ccccc3Cl)cc2)C1 ZINC000217569518 IH In-Stock Unstable MMP7 55 39 COC(=O)CS[C@H]1CCN(S(=O)(=O)c2ccc(Oc3ccccc3Cl)cc2)C1 ZINC000217569518 IH In-Stock Unstable MMP1 53 39 COC(=O)CS[C@H]1CCN(S(=O)(=O)c2ccc(Oc3ccccc3Cl)cc2)C1 ZINC000217569518 IH In-Stock Unstable F13A1 49 36 Cc1nc2ccccc2c(-c2ccccc2)c1CC(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000217569543 JK On-Demand Unstable DRD4 17 40 Cc1nc2ccccc2c(-c2ccccc2)c1CC(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000217569543 JK On-Demand Unstable TACR2 22 41 Cc1nc2ccccc2c(-c2ccccc2)c1CC(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000217569543 JK On-Demand Unstable SSTR5 35 40 Cc1nc2ccccc2c(-c2ccccc2)c1CC(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000217569543 JK On-Demand Unstable ADAM17 55 40 Cc1nc2ccccc2c(-c2ccccc2)c1CC(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000217569543 JK On-Demand Unstable TACR3 43 39 Cc1nc2ccccc2c(-c2ccccc2)c1CC(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000217569543 JK On-Demand Unstable MCHR1 15 41 Cc1nc2ccccc2c(-c2ccccc2)c1CC(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000217569543 JK On-Demand Unstable CCR8 71 39 COC(=O)[C@@H](C)CN(C)C[C@@H](O)c1ccc(CN)cc1 ZINC000217569556 CC For-Sale Unstable AOC3 24 42 C=CCNS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217569574 DD In-Stock Unstable SFRP1 50 32 COC(=O)[C@H](C)CN(C)C[C@@H](O)c1ccc(CN)cc1 ZINC000217569640 CC For-Sale Unstable AOC3 24 42 COC(=O)CS[C@@H]1CCN(S(=O)(=O)Cc2cccc(C(F)(F)F)c2)C1 ZINC000217569643 GF In-Stock Unstable CACNA1B 57 38 COC(=O)CS[C@@H]1CCN(S(=O)(=O)Cc2cccc(C(F)(F)F)c2)C1 ZINC000217569643 GF In-Stock Unstable CCR2 52 38 COC(=O)CS[C@@H]1CCN(S(=O)(=O)Cc2cccc(C(F)(F)F)c2)C1 ZINC000217569643 GF In-Stock Unstable LIPG 42 32 CCNC(=O)c1ccc(N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)c(NC(=O)/C=C/c2ccc(OC)c(OC)c2)c1 ZINC000217569667 KH In-Stock Unstable CHRNA4 23 40 C=CCNS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217569687 DD In-Stock Unstable SFRP1 46 32 COC(=O)CS[C@H]1CCN(S(=O)(=O)Cc2cccc(C(F)(F)F)c2)C1 ZINC000217569734 GF In-Stock Unstable CACNA1B 57 38 COC(=O)CS[C@H]1CCN(S(=O)(=O)Cc2cccc(C(F)(F)F)c2)C1 ZINC000217569734 GF In-Stock Unstable CCR2 72 38 COC(=O)CS[C@H]1CCN(S(=O)(=O)Cc2cccc(C(F)(F)F)c2)C1 ZINC000217569734 GF In-Stock Unstable LIPG 42 32 COc1cccc(NC(=O)[C@@H]2CC[C@@H](CNC(=O)[C@@H]3Cc4ccccc4CN3)CC2)c1 ZINC000217569758 HG In-Stock Unstable NPY2R 38 41 COc1cccc(NC(=O)[C@@H]2CC[C@@H](CNC(=O)[C@@H]3Cc4ccccc4CN3)CC2)c1 ZINC000217569758 HG In-Stock Unstable MTNR1A 42 52 COc1cccc(NC(=O)[C@@H]2CC[C@@H](CNC(=O)[C@@H]3Cc4ccccc4CN3)CC2)c1 ZINC000217569758 HG In-Stock Unstable MTNR1B 44 52 COc1cccc(NC(=O)[C@@H]2CC[C@@H](CNC(=O)[C@@H]3Cc4ccccc4CN3)CC2)c1 ZINC000217569758 HG In-Stock Unstable ROCK2 18 44 COc1cccc(NC(=O)[C@@H]2CC[C@@H](CNC(=O)[C@@H]3Cc4ccccc4CN3)CC2)c1 ZINC000217569758 HG In-Stock Unstable NPY5R 17 41 COc1cccc(NC(=O)[C@@H]2CC[C@@H](CNC(=O)[C@@H]3Cc4ccccc4CN3)CC2)c1 ZINC000217569758 HG In-Stock Unstable LIMK2 19 43 COc1ccc(CCNC(=O)OC(C)(C)C)nn1 ZINC000217569760 CD In-Stock Unstable PAPA1_CARPA 43 34 O=C1O[C@@]2(CCCN(C(=O)[C@H]3CC=CCC3)C2)c2ccccc21 ZINC000217569766 DG For-Sale Unstable NPY5R 46 41 C=CCNS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1 ZINC000217569786 EC In-Stock Unstable SLC6A9 15 45 CCNC(=O)c1ccc(N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)c(NC(=O)/C=C/c2ccc3c(c2)OCO3)c1 ZINC000217569835 KH In-Stock Unstable CHRNA4 23 40 CCNC(=O)c1ccc(N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)c(NC(=O)/C=C/c2ccc3c(c2)OCO3)c1 ZINC000217569835 KH In-Stock Unstable DYRK2 44 32 O=C1O[C@]2(CCCN(C(=O)[C@H]3CC=CCC3)C2)c2ccccc21 ZINC000217569841 DG For-Sale Unstable NPY5R 46 41 O=C1O[C@@]2(CCCN(C(=O)[C@@H]3CC=CCC3)C2)c2ccccc21 ZINC000217569917 DG For-Sale Unstable NPY5R 46 41 CC(C)CCN(CCC(C)C)C[C@@H](O)c1ccccc1 ZINC000217569930 CI For-Sale Unstable AOC3 32 61 CO[C@@H]1CC[C@@H](NC(=O)c2ccc(N(C)CCO)cc2)CC1 ZINC000217569965 DD In-Stock Unstable MAPK14 19 41 O=C1O[C@]2(CCCN(C(=O)[C@@H]3CC=CCC3)C2)c2ccccc21 ZINC000217570000 DG For-Sale Unstable NPY5R 46 41 CCNC(=O)c1ccc(N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)c(NC(=O)c2cncc(Br)c2)c1 ZINC000217570002 KH In-Stock Unstable CHRNA4 25 41 CC(C)CCN(CCC(C)C)C[C@H](O)c1ccccc1 ZINC000217570014 CI For-Sale Unstable AOC3 32 61 CN(C)CCN(C)c1ccc(CBr)cc1[N+](=O)[O-] ZINC000217570019 DE For-Sale Unstable MDAA 0 40 Cc1oncc1C(=O)NCC1(c2ccsc2)CCCC1 ZINC000217570060 CG In-Stock Unstable ACAT 0 50 c1cc(-c2ccc3c(c2)OCCO3)ccn1 ZINC000217570102 BF In-Stock Unstable CYP11B2 18 64 c1cc(-c2ccc3c(c2)OCCO3)ccn1 ZINC000217570102 BF In-Stock Unstable GSK3A 23 40 c1cc(-c2ccc3c(c2)OCCO3)ccn1 ZINC000217570102 BF In-Stock Unstable DYRK1A 38 40 c1cc(-c2ccc3c(c2)OCCO3)ccn1 ZINC000217570102 BF In-Stock Unstable CLK1 33 40 c1cc(-c2ccc3c(c2)OCCO3)ccn1 ZINC000217570102 BF In-Stock Unstable CLK4 65 40 O=C1O[C@@]2(CCCN(C(=O)c3ccc(OC(F)(F)F)cc3)C2)c2ccccc21 ZINC000217570113 GH For-Sale Unstable CHRM5 26 48 CC[C@@H](CSC)Nc1ccnc(N)n1 ZINC000217570119 BD For-Sale Unstable HRH4 0 47 C=CCNS(=O)(=O)c1ccc(NCCCCC)c(C(=O)O)c1 ZINC000217570121 EE In-Stock Unstable CASP3 0 42 C=CCNS(=O)(=O)c1ccc(NCCCCC)c(C(=O)O)c1 ZINC000217570121 EE In-Stock Unstable BDKRB1 0 40 Nc1cnn(CC(=O)N2CCC[C@@H](OCc3cccnc3)C2)c1 ZINC000217570145 DD In-Stock Unstable C3AR1 42 38 O=C(CSC1CCCC1)NCC1(c2ccsc2)CCCC1 ZINC000217570171 DI In-Stock Unstable ACAT 0 49 O=C1O[C@]2(CCCN(C(=O)c3ccc(OC(F)(F)F)cc3)C2)c2ccccc21 ZINC000217570191 GH For-Sale Unstable CHRM5 26 48 CN1CC[C@@H](NC(=O)c2cc(Cl)nc(Cl)c2)C1=O ZINC000217570199 CD On-Demand Unstable CACNA1I 44 32 CC[C@H](CSC)Nc1ccnc(N)n1 ZINC000217570205 BD For-Sale Unstable HRH4 0 47 c1cc2c(cc1-c1cn[nH]c1)OCCO2 ZINC000217570216 BD In-Stock Unstable ROCK2 48 37 c1cc2c(cc1-c1cn[nH]c1)OCCO2 ZINC000217570216 BD In-Stock Unstable HSP82 0 43 Nc1cnn(CC(=O)N2CCC[C@H](OCc3cccnc3)C2)c1 ZINC000217570229 DD In-Stock Unstable C3AR1 42 38 C=CCNS(=O)(=O)c1ccc(NCCC(C)C)c(C(=O)O)c1 ZINC000217570244 EE In-Stock Unstable BDKRB1 15 40 CN1CC[C@H](NC(=O)c2cc(Cl)nc(Cl)c2)C1=O ZINC000217570285 CD On-Demand Unstable CACNA1I 44 32 Cn1nc(-c2ccc(F)cc2)cc1C(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217570288 HH For-Sale Unstable NPY5R 39 46 C=CCNS(=O)(=O)c1ccc(N[C@@H](C)CCC)c(C(=O)O)c1 ZINC000217570354 EE In-Stock Unstable CASP3 0 40 Cn1nc(-c2ccc(F)cc2)cc1C(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217570366 HH For-Sale Unstable NPY5R 39 46 CC(C)(C)OC(=O)N1CCC([C@@H]2C[C@H](O)CCO2)CC1 ZINC000217570374 CE For-Sale Unstable GPR119 33 48 O=C(c1ccccc1F)N1C[C@H]2CNC[C@@H](C2)C1 ZINC000217570389 BD For-Sale Unstable CHRNA7 29 58 C=CCNS(=O)(=O)c1ccc(N[C@H](C)CCC)c(C(=O)O)c1 ZINC000217570426 EE In-Stock Unstable CASP3 0 40 COC[C@](C)(O)CNC(=O)Cc1c(F)cccc1Cl ZINC000217570433 CD In-Stock Unstable P2RX7 37 47 COc1ccc(OC)c(-c2cc(C(=O)N3CCC[C@]4(C3)OC(=O)c3ccccc34)n(C)n2)c1 ZINC000217570464 IG For-Sale Unstable NPY5R 22 43 CC(C)(C)OC(=O)N1CCC([C@H]2C[C@H](O)CCO2)CC1 ZINC000217570465 CE For-Sale Unstable GPR119 33 48 Nc1ccc(N(C(=O)NCC2CCCC2)c2ccccc2)cc1 ZINC000217570494 DI For-Sale Unstable AMY2 46 32 C[C@H]1c2ccsc2CCN1[C@H](C)C(=O)c1ccccc1 ZINC000217570510 CH For-Sale Unstable TRPM8 18 44 COC[C@@](C)(O)CNC(=O)Cc1c(F)cccc1Cl ZINC000217570516 CD In-Stock Unstable P2RX7 37 47 COc1ccc(OC)c(-c2cc(C(=O)N3CCC[C@@]4(C3)OC(=O)c3ccccc34)n(C)n2)c1 ZINC000217570534 IG For-Sale Unstable NPY5R 22 43 CC(C)(C)OC(=O)N1CCC([C@@H]2C[C@@H](O)CCO2)CC1 ZINC000217570558 CE For-Sale Unstable GPR119 33 48 CN(c1ccccc1)S(=O)(=O)c1ccccc1C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000217570570 JI On-Demand Unstable PPARA 18 45 CN(c1ccccc1)S(=O)(=O)c1ccccc1C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000217570570 JI On-Demand Unstable GRIN2B 0 44 CN(c1ccccc1)S(=O)(=O)c1ccccc1C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000217570570 JI On-Demand Unstable SCN9A 0 45 COc1cccc(C(=O)NCCC(=O)NC[C@@H]2COCCO2)c1 ZINC000217570577 DC In-Stock Unstable DRD4 56 43 COc1cccc(C(=O)NCCC(=O)NC[C@@H]2COCCO2)c1 ZINC000217570577 DC In-Stock Unstable MTNR1A 46 34 COc1cccc(C(=O)NCCC(=O)NC[C@@H]2COCCO2)c1 ZINC000217570577 DC In-Stock Unstable MTNR1B 41 36 COc1cccc(C(=O)NCCC(=O)NC[C@@H]2COCCO2)c1 ZINC000217570577 DC In-Stock Unstable BRPF1 0 40 O=C(NCC1CCCC1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217570611 DJ For-Sale Unstable ADRB1 16 41 O=C(NCC1CCCC1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217570611 DJ For-Sale Unstable LTA4H 17 40 O=C(NCC1CCCC1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217570611 DJ For-Sale Unstable CCR3 46 44 O=C(NCC1CCCC1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217570611 DJ For-Sale Unstable EPHX2 49 63 O=C(NCC1CCCC1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217570611 DJ For-Sale Unstable DGAT1 17 42 O=C(NCC1CCCC1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217570611 DJ For-Sale Unstable ACAT 0 47 O=C(NCC1CCCC1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217570611 DJ For-Sale Unstable UPPS 0 40 O=C(NCC1CCCC1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217570611 DJ For-Sale Unstable NAMPT 33 43 O=C(NCC1CCCC1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217570611 DJ For-Sale Unstable P95276_MYCTO 0 46 CC(C)(C)OC(=O)N1CCC([C@H]2C[C@@H](O)CCO2)CC1 ZINC000217570644 CE For-Sale Unstable GPR119 33 48 O=C(c1ccc(F)cc1)N1C[C@H]2CNC[C@@H](C2)C1 ZINC000217570649 BD For-Sale Unstable CHRNA7 36 68 O=C(c1ccc(F)cc1)N1C[C@H]2CNC[C@@H](C2)C1 ZINC000217570649 BD For-Sale Unstable L3MBTL3 50 39 O=C(O)c1ccc(-c2cccc3c2OCCO3)o1 ZINC000217570653 BE In-Stock Unstable MAP 0 57 COCC(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217570661 CD For-Sale Unstable NPY5R 29 43 COc1cccc(C(=O)NCCC(=O)NC[C@H]2COCCO2)c1 ZINC000217570668 DC In-Stock Unstable DRD4 56 43 COc1cccc(C(=O)NCCC(=O)NC[C@H]2COCCO2)c1 ZINC000217570668 DC In-Stock Unstable MTNR1A 46 34 COc1cccc(C(=O)NCCC(=O)NC[C@H]2COCCO2)c1 ZINC000217570668 DC In-Stock Unstable MTNR1B 41 36 COc1cccc(C(=O)NCCC(=O)NC[C@H]2COCCO2)c1 ZINC000217570668 DC In-Stock Unstable BRPF1 0 40 C[C@H]1c2ccsc2CCN1[C@H](C)C(=O)c1ccc(Cl)cc1 ZINC000217570692 DJ For-Sale Unstable TRPM8 16 41 Cc1cccc(NC(=O)NCC2CCCC2)n1 ZINC000217570713 BF On-Demand Unstable GRM5 19 48 Cc1cccc(NC(=O)NCC2CCCC2)n1 ZINC000217570713 BF On-Demand Unstable SORT1 17 43 CCCNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217570720 CD In-Stock Unstable CCR8 81 36 CCCNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217570720 CD In-Stock Unstable SFRP1 98 37 CCCNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217570720 CD In-Stock Unstable WNT3 77 36 COCC(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217570740 CD For-Sale Unstable NPY5R 29 43 O=C(CCCc1c[nH]c2ccccc12)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217570784 GG In-Stock Unstable MC4R 39 41 O=C(CCCc1c[nH]c2ccccc12)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217570784 GG In-Stock Unstable TACR2 0 45 O=C(CCCc1c[nH]c2ccccc12)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217570784 GG In-Stock Unstable CHRNA4 30 50 O=C(CCCc1c[nH]c2ccccc12)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217570784 GG In-Stock Unstable MC5R 33 40 O=C(CCCc1c[nH]c2ccccc12)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217570784 GG In-Stock Unstable CCKBR 53 34 O=C(CCCc1c[nH]c2ccccc12)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217570784 GG In-Stock Unstable MC1R 15 40 CCS(=O)(=O)N1CCC(C(=O)NCc2ccc(OC(F)(F)F)cc2)(c2ccccc2)CC1 ZINC000217570788 JH On-Demand Unstable P2RY1 45 35 CCS(=O)(=O)N1CCC(C(=O)NCc2ccc(OC(F)(F)F)cc2)(c2ccccc2)CC1 ZINC000217570788 JH On-Demand Unstable SLC6A9 30 44 CCS(=O)(=O)N1CCC(C(=O)NCc2ccc(OC(F)(F)F)cc2)(c2ccccc2)CC1 ZINC000217570788 JH On-Demand Unstable EPHX2 42 46 CCS(=O)(=O)N1CCC(C(=O)NCc2ccc(OC(F)(F)F)cc2)(c2ccccc2)CC1 ZINC000217570788 JH On-Demand Unstable SCN10A 20 43 CCS(=O)(=O)N1CCC(C(=O)NCc2ccc(OC(F)(F)F)cc2)(c2ccccc2)CC1 ZINC000217570788 JH On-Demand Unstable PDS 50 35 CC(C)Nc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217570825 CD In-Stock Unstable CCR8 73 35 CC(C)Nc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217570825 CD In-Stock Unstable SFRP1 94 35 CC(C)Nc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217570825 CD In-Stock Unstable WNT3 77 35 O=C(NCCCCCO)NCC1CCCC1 ZINC000217570838 BD On-Demand Unstable EPHX2 49 46 Cc1ccc(C)c(S(=O)(=O)NCC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217570860 IE For-Sale Unstable NPY5R 24 41 O=[S@@](C[C@@H]1CCCN1)c1ccccc1Cl ZINC000217570918 BE For-Sale Unstable CHRNA10 30 41 CCCCNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217570937 DE In-Stock Unstable CCR8 79 35 CCCCNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217570937 DE In-Stock Unstable SFRP1 93 35 CCCCNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217570937 DE In-Stock Unstable WNT3 73 35 Cc1ccc(C)c(S(=O)(=O)NCC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217570946 IE For-Sale Unstable NPY5R 24 41 CC(C)(C)CC(C)(C)NC(=O)NCC1CCCC1 ZINC000217570959 CH For-Sale Unstable CACNA1I 42 34 O=[S@](C[C@@H]1CCCN1)c1ccccc1Cl ZINC000217570995 BE For-Sale Unstable CHRNA10 30 41 COC[C@](C)(O)CNC(=O)c1ccc(OC)c(F)c1 ZINC000217571021 CC In-Stock Unstable PPARD 18 42 COC[C@](C)(O)CNC(=O)c1ccc(OC)c(F)c1 ZINC000217571021 CC In-Stock Unstable MT-ND1 24 40 CC(C)CNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217571034 DD In-Stock Unstable MTNN 45 32 CC(C)CNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217571034 DD In-Stock Unstable CCR8 79 34 CC(C)CNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217571034 DD In-Stock Unstable SFRP1 98 37 CC(C)CNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217571034 DD In-Stock Unstable WNT3 78 38 O=C1O[C@@]2(CCCN(C(=O)c3ccc(NS(=O)(=O)c4cccc(F)c4)cc3)C2)c2ccccc21 ZINC000217571044 JH For-Sale Unstable NPY5R 25 44 O=[S@@](C[C@H]1CCCN1)c1ccccc1Cl ZINC000217571078 BE For-Sale Unstable CHRNA10 30 41 COC[C@@](C)(O)CNC(=O)c1ccc(OC)c(F)c1 ZINC000217571098 CC In-Stock Unstable PPARD 18 42 COC[C@@](C)(O)CNC(=O)c1ccc(OC)c(F)c1 ZINC000217571098 CC In-Stock Unstable MT-ND1 24 40 O=C1O[C@]2(CCCN(C(=O)c3ccc(NS(=O)(=O)c4cccc(F)c4)cc3)C2)c2ccccc21 ZINC000217571119 JH For-Sale Unstable NPY5R 25 44 CC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217571139 DE In-Stock Unstable CCR8 73 36 CC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217571139 DE In-Stock Unstable SFRP1 82 35 CC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217571139 DE In-Stock Unstable WNT3 60 35 O=[S@](C[C@H]1CCCN1)c1ccccc1Cl ZINC000217571158 BE For-Sale Unstable CHRNA10 30 41 CC[C@H](C)Nc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217571201 DE In-Stock Unstable CCR8 73 36 CC[C@H](C)Nc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217571201 DE In-Stock Unstable SFRP1 82 35 CC[C@H](C)Nc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217571201 DE In-Stock Unstable WNT3 60 35 O=C1O[C@@]2(CCCN(C(=O)CNS(=O)(=O)c3cccc(Cl)c3)C2)c2ccccc21 ZINC000217571225 IE For-Sale Unstable NPY5R 25 47 Cc1cc(=O)[nH]c(NCCNC(=O)c2n[nH]c3ccccc23)n1 ZINC000217571243 DC In-Stock Unstable ITK 28 40 COc1ccc(Cl)cc1N1C(=O)[C@@H]2[C@@H](C(=O)c3ccccc3)N3CCC[C@@H]3[C@@H]2C1=O ZINC000217571254 HG In-Stock Unstable COLA 48 38 COc1ccc(Cl)cc1N1C(=O)[C@@H]2[C@@H](C(=O)c3ccccc3)N3CCC[C@@H]3[C@@H]2C1=O ZINC000217571254 HG In-Stock Unstable CPT1A 48 38 OC[C@@H]1CCCCN1C[C@@H](O)COCc1ccccc1 ZINC000217571265 CD On-Demand Unstable SLC18A2 68 42 O=C1O[C@]2(CCCN(C(=O)CNS(=O)(=O)c3cccc(Cl)c3)C2)c2ccccc21 ZINC000217571298 IE For-Sale Unstable NPY5R 25 47 CC(C)(C)Nc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217571324 DE In-Stock Unstable CCR8 78 35 CC(C)(C)Nc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217571324 DE In-Stock Unstable SFRP1 108 38 CC(C)(C)Nc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217571324 DE In-Stock Unstable WNT3 83 37 COc1ccc(Cl)cc1N1C(=O)[C@H]2[C@H](C1=O)[C@H]1CCCN1[C@@H]2C(=O)c1ccccc1 ZINC000217571338 HG In-Stock Unstable COLA 48 38 COc1ccc(Cl)cc1N1C(=O)[C@H]2[C@H](C1=O)[C@H]1CCCN1[C@@H]2C(=O)c1ccccc1 ZINC000217571338 HG In-Stock Unstable CPT1A 48 38 COc1ccc2nc(CCNC(=O)[C@@H](C)Sc3ccccn3)[nH]c2c1 ZINC000217571354 FF In-Stock Unstable MTNR1B 45 38 COc1ccc2nc(CCNC(=O)[C@@H](C)Sc3ccccn3)[nH]c2c1 ZINC000217571354 FF In-Stock Unstable CYP2C19 26 40 COc1ccc2nc(CCNC(=O)[C@@H](C)Sc3ccccn3)[nH]c2c1 ZINC000217571354 FF In-Stock Unstable FABK 0 41 COc1ccc2c(c1)CCC[C@@H]2NC[C@@H]1CCCN(C)C1 ZINC000217571398 CG On-Demand Unstable NPY2R 47 44 COc1ccc2c(c1)CCC[C@@H]2NC[C@@H]1CCCN(C)C1 ZINC000217571398 CG On-Demand Unstable EBP 33 47 O=C1O[C@@]2(CCCN(C(=O)CNS(=O)(=O)c3cccc(F)c3)C2)c2ccccc21 ZINC000217571415 HD For-Sale Unstable NPY5R 28 45 COc1ccc2nc(CCNC(=O)[C@H](C)Sc3ccccn3)[nH]c2c1 ZINC000217571431 FF In-Stock Unstable MTNR1B 45 38 COc1ccc2nc(CCNC(=O)[C@H](C)Sc3ccccn3)[nH]c2c1 ZINC000217571431 FF In-Stock Unstable CYP2C19 26 40 COc1ccc2nc(CCNC(=O)[C@H](C)Sc3ccccn3)[nH]c2c1 ZINC000217571431 FF In-Stock Unstable FABK 0 41 C=CCNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217571443 CD In-Stock Unstable F13A1 22 40 C=CCNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217571443 CD In-Stock Unstable CCR8 43 34 C=CCNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217571443 CD In-Stock Unstable SFRP1 95 36 C=CCNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217571443 CD In-Stock Unstable WNT3 48 30 COc1ccc2c(c1)CCC[C@@H]2NC[C@H]1CCCN(C)C1 ZINC000217571482 CG On-Demand Unstable NPY2R 47 44 COc1ccc2c(c1)CCC[C@@H]2NC[C@H]1CCCN(C)C1 ZINC000217571482 CG On-Demand Unstable EBP 33 47 O=C1O[C@]2(CCCN(C(=O)CNS(=O)(=O)c3cccc(F)c3)C2)c2ccccc21 ZINC000217571485 HD For-Sale Unstable NPY5R 28 45 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NC1CC1 ZINC000217571554 CD In-Stock Unstable CCR8 66 35 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NC1CC1 ZINC000217571554 CD In-Stock Unstable SFRP1 97 36 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NC1CC1 ZINC000217571554 CD In-Stock Unstable WNT3 73 34 Cc1cc(C)c(C)c(S(=O)(=O)NCC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1C ZINC000217571593 JF For-Sale Unstable NPY5R 24 42 C[C@@H]1CN(C[C@@H](O)COc2ccccc2C#N)CCCO1 ZINC000217571603 CD On-Demand Unstable ADRB2 41 50 C[C@@H]1CN(C[C@@H](O)COc2ccccc2C#N)CCCO1 ZINC000217571603 CD On-Demand Unstable ADRB1 60 36 C[C@@H]1CN(C[C@@H](O)COc2ccccc2C#N)CCCO1 ZINC000217571603 CD On-Demand Unstable ADRB3 42 45 C[C@@H]1CN(C[C@@H](O)COc2ccccc2C#N)CCCO1 ZINC000217571603 CD On-Demand Unstable CASR 38 41 C[C@@H]1CN(C[C@@H](O)COc2ccccc2C#N)CCCO1 ZINC000217571603 CD On-Demand Unstable CYP2D6 15 41 C[C@@H]1CN(C[C@@H](O)COc2ccccc2C#N)CCCO1 ZINC000217571603 CD On-Demand Unstable ABCB1 62 42 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NC1CCCC1 ZINC000217571654 DE In-Stock Unstable CCR8 53 40 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NC1CCCC1 ZINC000217571654 DE In-Stock Unstable SFRP1 96 34 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NC1CCCC1 ZINC000217571654 DE In-Stock Unstable WNT3 76 34 Cc1cc(C)c(C)c(S(=O)(=O)NCC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1C ZINC000217571681 JF For-Sale Unstable NPY5R 24 42 C[C@H]1CN(C[C@@H](O)COc2ccccc2C#N)CCCO1 ZINC000217571688 CD On-Demand Unstable ADRB2 41 50 C[C@H]1CN(C[C@@H](O)COc2ccccc2C#N)CCCO1 ZINC000217571688 CD On-Demand Unstable ADRB1 60 36 C[C@H]1CN(C[C@@H](O)COc2ccccc2C#N)CCCO1 ZINC000217571688 CD On-Demand Unstable ADRB3 42 45 C[C@H]1CN(C[C@@H](O)COc2ccccc2C#N)CCCO1 ZINC000217571688 CD On-Demand Unstable CASR 38 41 C[C@H]1CN(C[C@@H](O)COc2ccccc2C#N)CCCO1 ZINC000217571688 CD On-Demand Unstable CYP2D6 15 41 C[C@H]1CN(C[C@@H](O)COc2ccccc2C#N)CCCO1 ZINC000217571688 CD On-Demand Unstable ABCB1 62 42 O=C(C[C@@H](Cn1cnnn1)c1ccc(Cl)cc1)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217571725 IE In-Stock Unstable CHRNA4 26 42 O=[S@@](C[C@@H]1CCCN1)c1cccc(Cl)c1 ZINC000217571750 BE For-Sale Unstable GHSR 26 42 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NC1CCCCC1 ZINC000217571767 EF In-Stock Unstable CCR8 48 42 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NC1CCCCC1 ZINC000217571767 EF In-Stock Unstable SFRP1 93 34 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NC1CCCCC1 ZINC000217571767 EF In-Stock Unstable WNT3 75 34 COC[C@](C)(O)CNS(=O)(=O)c1cccc2cccnc12 ZINC000217571772 DC In-Stock Unstable C0L093_TOBAC 46 31 O=C(C[C@H](Cn1cnnn1)c1ccc(Cl)cc1)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217571816 IE In-Stock Unstable CHRNA4 26 42 O=[S@](C[C@@H]1CCCN1)c1cccc(Cl)c1 ZINC000217571830 BE For-Sale Unstable GHSR 26 42 COC[C@@](C)(O)CNS(=O)(=O)c1cccc2cccnc12 ZINC000217571848 DC In-Stock Unstable C0L093_TOBAC 46 31 O=C(NCC1CCCC1)Nc1ccccc1N1CCOCC1 ZINC000217571855 DF For-Sale Unstable DRD2 15 41 O=C(NCC1CCCC1)Nc1ccccc1N1CCOCC1 ZINC000217571855 DF For-Sale Unstable KCNQ2 92 44 O=C(NCC1CCCC1)Nc1ccccc1N1CCOCC1 ZINC000217571855 DF For-Sale Unstable MTOR 47 37 O=C(NCC1CCCC1)Nc1ccccc1N1CCOCC1 ZINC000217571855 DF For-Sale Unstable EPHX2 16 44 O=C(NCC1CCCC1)Nc1ccccc1N1CCOCC1 ZINC000217571855 DF For-Sale Unstable CSF1R 28 48 O=C(NCC1CCCC1)Nc1ccccc1N1CCOCC1 ZINC000217571855 DF For-Sale Unstable AKR1C3 22 42 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NCCC1=CCCCC1 ZINC000217571895 FG In-Stock Unstable SFRP1 68 32 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NCCC1=CCCCC1 ZINC000217571895 FG In-Stock Unstable WNT3 52 32 O=[S@@](C[C@H]1CCCN1)c1cccc(Cl)c1 ZINC000217571914 BE For-Sale Unstable GHSR 26 42 O=C1O[C@@]2(CCCN(C(=O)c3ccc(NS(=O)(=O)c4ccccc4F)cc3)C2)c2ccccc21 ZINC000217571979 JH For-Sale Unstable NPY5R 24 41 O=[S@](C[C@H]1CCCN1)c1cccc(Cl)c1 ZINC000217571980 BE For-Sale Unstable GHSR 26 42 O=C(NCC1CCCC1)Nc1ccc(N2CCCCC2)cc1 ZINC000217571992 DH On-Demand Unstable CCR3 39 40 O=C(NCC1CCCC1)Nc1ccc(N2CCCCC2)cc1 ZINC000217571992 DH On-Demand Unstable MTOR 43 39 O=C(NCC1CCCC1)Nc1ccc(N2CCCCC2)cc1 ZINC000217571992 DH On-Demand Unstable EPHX2 48 62 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NCCO ZINC000217571997 DC In-Stock Unstable CCR8 76 35 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NCCO ZINC000217571997 DC In-Stock Unstable SFRP1 97 37 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NCCO ZINC000217571997 DC In-Stock Unstable WNT3 74 35 CN(CCO)c1ccc(C(=O)NC2(c3ccccc3)CC2)cc1 ZINC000217572037 DF In-Stock Unstable TACR3 54 32 O=C1O[C@]2(CCCN(C(=O)c3ccc(NS(=O)(=O)c4ccccc4F)cc3)C2)c2ccccc21 ZINC000217572066 JH For-Sale Unstable NPY5R 24 41 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NCCCO ZINC000217572092 DC In-Stock Unstable CCR8 74 34 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NCCCO ZINC000217572092 DC In-Stock Unstable SFRP1 95 36 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NCCCO ZINC000217572092 DC In-Stock Unstable WNT3 72 34 CS(=O)(=O)c1ccc([C@H](N)C(=O)O)c(F)c1 ZINC000217572176 BC For-Sale Unstable PTGS2 30 44 O=C1O[C@@]2(CCCN(C(=O)CNS(=O)(=O)c3ccccc3F)C2)c2ccccc21 ZINC000217572177 HD For-Sale Unstable NPY5R 26 43 Nc1ncc([C@@H](N)C(=O)O)s1 ZINC000217572180 AB For-Sale Unstable CACNA2D1 0 44 O=C(O)[C@@H]1CC[C@@H](CNC(=O)[C@@H]2Cc3ccccc3CN2)CC1 ZINC000217572181 DD In-Stock Unstable VCP 38 41 CN1CC[C@@H](NC(=O)c2ccc(C(=O)O)nc2)C1=O ZINC000217572196 CB On-Demand Unstable P4HTM 0 49 CN1CC[C@@H](NC(=O)c2ccc(C(=O)O)nc2)C1=O ZINC000217572196 CB On-Demand Unstable P4HA1 0 45 COCCNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217572218 DC In-Stock Unstable CCR8 81 36 COCCNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217572218 DC In-Stock Unstable SFRP1 87 35 COCCNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217572218 DC In-Stock Unstable WNT3 67 35 COC[C@@](C)(O)CNS(=O)(=O)C[C@@]12CC[C@@H](CC1=O)C2(C)C ZINC000217572220 EC In-Stock Unstable CA5B 29 51 COC[C@@](C)(O)CNS(=O)(=O)C[C@@]12CC[C@@H](CC1=O)C2(C)C ZINC000217572220 EC In-Stock Unstable CA5A 32 51 O=C(C[C@@H](Cn1cccc1)c1ccc(Cl)cc1)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217572239 II In-Stock Unstable CHRNA4 28 45 CS(=O)(=O)c1ccc([C@@H](N)C(=O)O)c(F)c1 ZINC000217572261 BC For-Sale Unstable PTGS2 30 44 CN1CC[C@H](NC(=O)c2ccc(C(=O)O)nc2)C1=O ZINC000217572273 CB On-Demand Unstable P4HTM 0 49 CN1CC[C@H](NC(=O)c2ccc(C(=O)O)nc2)C1=O ZINC000217572273 CB On-Demand Unstable P4HA1 0 45 O=C1O[C@]2(CCCN(C(=O)CNS(=O)(=O)c3ccccc3F)C2)c2ccccc21 ZINC000217572280 HD For-Sale Unstable NPY5R 26 43 O=C(NCC1CCCC1)N(Cc1ccccc1)c1ccccc1 ZINC000217572318 DJ For-Sale Unstable CHRM2 29 46 O=C(NCC1CCCC1)N(Cc1ccccc1)c1ccccc1 ZINC000217572318 DJ For-Sale Unstable CHRM1 26 48 O=C(NCC1CCCC1)N(Cc1ccccc1)c1ccccc1 ZINC000217572318 DJ For-Sale Unstable CHRM3 29 48 O=C(NCC1CCCC1)N(Cc1ccccc1)c1ccccc1 ZINC000217572318 DJ For-Sale Unstable AMY2 44 30 O=C(NCC1CCCC1)N(Cc1ccccc1)c1ccccc1 ZINC000217572318 DJ For-Sale Unstable PTGES 0 50 O=C(C[C@H](Cn1cccc1)c1ccc(Cl)cc1)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217572327 II In-Stock Unstable CHRNA4 28 45 COCCCNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217572334 ED In-Stock Unstable CCR8 79 35 COCCCNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217572334 ED In-Stock Unstable SFRP1 83 34 COCCCNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217572334 ED In-Stock Unstable WNT3 63 34 CS(=O)(=O)c1ccc([C@H](N)C(=O)O)cc1F ZINC000217572368 BC For-Sale Unstable GRM8 15 46 O=C1O[C@@]2(CCCN(C(=O)CNS(=O)(=O)c3c(Cl)cccc3Cl)C2)c2ccccc21 ZINC000217572414 JF For-Sale Unstable NPY5R 28 48 O=C(NCC1CCCC1)Nc1ccc2ccccc2c1 ZINC000217572416 CI On-Demand Unstable F2 15 41 O=C(NCC1CCCC1)Nc1ccc2ccccc2c1 ZINC000217572416 CI On-Demand Unstable CMA1 23 40 O=C(NCC1CCCC1)Nc1ccc2ccccc2c1 ZINC000217572416 CI On-Demand Unstable CA1 31 48 O=C(NCC1CCCC1)Nc1ccc2ccccc2c1 ZINC000217572416 CI On-Demand Unstable CCR3 52 39 O=C(NCC1CCCC1)Nc1ccc2ccccc2c1 ZINC000217572416 CI On-Demand Unstable EPHX2 36 62 O=C(NCC1CCCC1)Nc1ccc2ccccc2c1 ZINC000217572416 CI On-Demand Unstable PLAU 15 46 O=C(NCC1CCCC1)Nc1ccc2ccccc2c1 ZINC000217572416 CI On-Demand Unstable MCHR1 17 40 O=C(NCC1CCCC1)Nc1ccc2ccccc2c1 ZINC000217572416 CI On-Demand Unstable PRMT3 44 42 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NCc1ccccc1 ZINC000217572430 EE In-Stock Unstable TGM2 19 42 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NCc1ccccc1 ZINC000217572430 EE In-Stock Unstable F13A1 21 42 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NCc1ccccc1 ZINC000217572430 EE In-Stock Unstable CCR8 82 38 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NCc1ccccc1 ZINC000217572430 EE In-Stock Unstable SFRP1 109 39 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NCc1ccccc1 ZINC000217572430 EE In-Stock Unstable WNT3 83 38 CS(=O)(=O)c1ccc([C@@H](N)C(=O)O)cc1F ZINC000217572442 BC For-Sale Unstable GRM8 15 46 O=C1O[C@]2(CCCN(C(=O)CNS(=O)(=O)c3c(Cl)cccc3Cl)C2)c2ccccc21 ZINC000217572503 JF For-Sale Unstable NPY5R 28 48 C[C@@H]1CCCC[C@@]1(NC(=O)/C=C\c1ccccc1)C(=O)O ZINC000217572532 CF For-Sale Unstable MMP2 17 41 C[C@@H]1CCCC[C@@]1(NC(=O)/C=C\c1ccccc1)C(=O)O ZINC000217572532 CF For-Sale Unstable HDAC6 26 44 c1csc(-c2ccccc2N[C@H]2C[C@@H]3CC[C@H]2C3)c1 ZINC000217572534 CK For-Sale Unstable BRS3 24 41 C[C@@H](Nc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O)c1ccccc1 ZINC000217572540 FF In-Stock Unstable CCR8 43 33 O=C1O[C@@]2(CCCN(C(=O)CCNS(=O)(=O)c3c(Cl)cccc3Cl)C2)c2ccccc21 ZINC000217572596 JG For-Sale Unstable NPY5R 23 45 C[C@H](Nc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O)c1ccccc1 ZINC000217572624 FF In-Stock Unstable CCR8 43 33 C[C@H]1CCCC[C@@]1(NC(=O)/C=C\c1ccccc1)C(=O)O ZINC000217572631 CF For-Sale Unstable MMP2 17 41 C[C@H]1CCCC[C@@]1(NC(=O)/C=C\c1ccccc1)C(=O)O ZINC000217572631 CF For-Sale Unstable HDAC6 26 44 c1csc(-c2ccccc2N[C@H]2C[C@H]3CC[C@H]2C3)c1 ZINC000217572635 CK For-Sale Unstable BRS3 24 41 O=C1O[C@]2(CCCN(C(=O)CCNS(=O)(=O)c3c(Cl)cccc3Cl)C2)c2ccccc21 ZINC000217572698 JG For-Sale Unstable NPY5R 23 45 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NCCc1ccccc1 ZINC000217572730 FE In-Stock Unstable PTGDR 28 40 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NCCc1ccccc1 ZINC000217572730 FE In-Stock Unstable CCR8 80 37 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NCCc1ccccc1 ZINC000217572730 FE In-Stock Unstable SFRP1 107 38 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NCCc1ccccc1 ZINC000217572730 FE In-Stock Unstable WNT3 82 37 COc1ccc(OC)c2[nH]c(C(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)cc12 ZINC000217572754 GF In-Stock Unstable CHRNA4 27 45 O=[S@@](C[C@@H]1CCNC1)c1ccc(Cl)cc1 ZINC000217572797 BE For-Sale Unstable SLC6A1 0 42 CCC(=O)N[C@@H]1CCN(C)C1=O ZINC000217572799 AB On-Demand Unstable LASR 44 34 CCC(=O)N[C@@H]1CCN(C)C1=O ZINC000217572799 AB On-Demand Unstable PHZR 41 34 O=C1O[C@@]2(CCCN(C(=O)CCNS(=O)(=O)c3cccc(Cl)c3)C2)c2ccccc21 ZINC000217572818 IF For-Sale Unstable NPY5R 22 44 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CC3)cc2C(=O)O)cc1 ZINC000217572829 GE In-Stock Unstable BMP1 74 36 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CC3)cc2C(=O)O)cc1 ZINC000217572829 GE In-Stock Unstable MMP13 66 41 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CC3)cc2C(=O)O)cc1 ZINC000217572829 GE In-Stock Unstable MMP2 40 41 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CC3)cc2C(=O)O)cc1 ZINC000217572829 GE In-Stock Unstable MMP3 58 41 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CC3)cc2C(=O)O)cc1 ZINC000217572829 GE In-Stock Unstable MMP9 52 39 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CC3)cc2C(=O)O)cc1 ZINC000217572829 GE In-Stock Unstable PTGDR 34 41 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CC3)cc2C(=O)O)cc1 ZINC000217572829 GE In-Stock Unstable MMP7 47 39 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CC3)cc2C(=O)O)cc1 ZINC000217572829 GE In-Stock Unstable CA9 22 42 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CC3)cc2C(=O)O)cc1 ZINC000217572829 GE In-Stock Unstable MMP1 59 40 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CC3)cc2C(=O)O)cc1 ZINC000217572829 GE In-Stock Unstable CCR8 69 44 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CC3)cc2C(=O)O)cc1 ZINC000217572829 GE In-Stock Unstable SFRP1 83 32 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CC3)cc2C(=O)O)cc1 ZINC000217572829 GE In-Stock Unstable AKR1C2 49 37 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CC3)cc2C(=O)O)cc1 ZINC000217572829 GE In-Stock Unstable WNT3 50 32 N[C@H](C(=O)O)c1ccccc1SCC(F)F ZINC000217572843 BE For-Sale Unstable CACNA2D1 38 53 COc1ccc2cc(C(=O)NC[C@H](O)Cc3ccccc3)[nH]c2c1 ZINC000217572873 DF In-Stock Unstable ADRB3 17 40 COc1ccc2cc(C(=O)NC[C@H](O)Cc3ccccc3)[nH]c2c1 ZINC000217572873 DF In-Stock Unstable NQO2 15 40 COc1ccc2cc(C(=O)NC[C@H](O)Cc3ccccc3)[nH]c2c1 ZINC000217572873 DF In-Stock Unstable PYGL 43 45 COc1ccc2cc(C(=O)NC[C@H](O)Cc3ccccc3)[nH]c2c1 ZINC000217572873 DF In-Stock Unstable ROCK1 24 49 COc1ccc2cc(C(=O)NC[C@H](O)Cc3ccccc3)[nH]c2c1 ZINC000217572873 DF In-Stock Unstable MTNR1A 54 40 COc1ccc2cc(C(=O)NC[C@H](O)Cc3ccccc3)[nH]c2c1 ZINC000217572873 DF In-Stock Unstable MTNR1B 51 36 COc1ccc2cc(C(=O)NC[C@H](O)Cc3ccccc3)[nH]c2c1 ZINC000217572873 DF In-Stock Unstable ROCK2 17 49 COc1ccc2cc(C(=O)NC[C@H](O)Cc3ccccc3)[nH]c2c1 ZINC000217572873 DF In-Stock Unstable TUBB2B 39 44 COc1ccc2cc(C(=O)NC[C@H](O)Cc3ccccc3)[nH]c2c1 ZINC000217572873 DF In-Stock Unstable PLCG2 0 40 COc1ccc2cc(C(=O)NC[C@H](O)Cc3ccccc3)[nH]c2c1 ZINC000217572873 DF In-Stock Unstable POL 0 44 COc1ccc2cc(C(=O)NC[C@H](O)Cc3ccccc3)[nH]c2c1 ZINC000217572873 DF In-Stock Unstable BLA1_STEMA 17 40 CCC(=O)N[C@H]1CCN(C)C1=O ZINC000217572883 AB On-Demand Unstable LASR 44 34 CCC(=O)N[C@H]1CCN(C)C1=O ZINC000217572883 AB On-Demand Unstable PHZR 41 34 O=[S@](C[C@@H]1CCNC1)c1ccc(Cl)cc1 ZINC000217572884 BE For-Sale Unstable SLC6A1 0 42 O=C1O[C@]2(CCCN(C(=O)CCNS(=O)(=O)c3cccc(Cl)c3)C2)c2ccccc21 ZINC000217572897 IF For-Sale Unstable NPY5R 22 44 N[C@@H](C(=O)O)c1ccccc1SCC(F)F ZINC000217572932 BE For-Sale Unstable CACNA2D1 38 53 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CC3)cc2C(=O)O)cc1OC ZINC000217572939 HE In-Stock Unstable ADRA1D 26 45 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CC3)cc2C(=O)O)cc1OC ZINC000217572939 HE In-Stock Unstable ADRA1A 18 45 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CC3)cc2C(=O)O)cc1OC ZINC000217572939 HE In-Stock Unstable ADRA1B 32 45 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CC3)cc2C(=O)O)cc1OC ZINC000217572939 HE In-Stock Unstable IAP 0 41 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CC3)cc2C(=O)O)cc1OC ZINC000217572939 HE In-Stock Unstable CCR8 54 41 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CC3)cc2C(=O)O)cc1OC ZINC000217572939 HE In-Stock Unstable SFRP1 54 33 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CC3)cc2C(=O)O)cc1OC ZINC000217572939 HE In-Stock Unstable SCMU_MYCTU 0 44 O=CNCCCNC(=O)NCC1CCCC1 ZINC000217572951 BC For-Sale Unstable ADH1B 0 50 O=CNCCCNC(=O)NCC1CCCC1 ZINC000217572951 BC For-Sale Unstable ADH4 0 50 COc1ccc2cc(C(=O)NC[C@@H](O)Cc3ccccc3)[nH]c2c1 ZINC000217572956 DF In-Stock Unstable ADRB3 17 40 COc1ccc2cc(C(=O)NC[C@@H](O)Cc3ccccc3)[nH]c2c1 ZINC000217572956 DF In-Stock Unstable NQO2 15 40 COc1ccc2cc(C(=O)NC[C@@H](O)Cc3ccccc3)[nH]c2c1 ZINC000217572956 DF In-Stock Unstable CCKAR 0 43 COc1ccc2cc(C(=O)NC[C@@H](O)Cc3ccccc3)[nH]c2c1 ZINC000217572956 DF In-Stock Unstable PYGL 43 45 COc1ccc2cc(C(=O)NC[C@@H](O)Cc3ccccc3)[nH]c2c1 ZINC000217572956 DF In-Stock Unstable ROCK1 24 49 COc1ccc2cc(C(=O)NC[C@@H](O)Cc3ccccc3)[nH]c2c1 ZINC000217572956 DF In-Stock Unstable MTNR1A 54 40 COc1ccc2cc(C(=O)NC[C@@H](O)Cc3ccccc3)[nH]c2c1 ZINC000217572956 DF In-Stock Unstable MTNR1B 51 36 COc1ccc2cc(C(=O)NC[C@@H](O)Cc3ccccc3)[nH]c2c1 ZINC000217572956 DF In-Stock Unstable ROCK2 17 49 COc1ccc2cc(C(=O)NC[C@@H](O)Cc3ccccc3)[nH]c2c1 ZINC000217572956 DF In-Stock Unstable TUBB2B 39 44 COc1ccc2cc(C(=O)NC[C@@H](O)Cc3ccccc3)[nH]c2c1 ZINC000217572956 DF In-Stock Unstable PLCG2 0 40 COc1ccc2cc(C(=O)NC[C@@H](O)Cc3ccccc3)[nH]c2c1 ZINC000217572956 DF In-Stock Unstable POL 0 44 COc1ccc2cc(C(=O)NC[C@@H](O)Cc3ccccc3)[nH]c2c1 ZINC000217572956 DF In-Stock Unstable BLA1_STEMA 17 40 CN1CCC[C@@H](CNC[C@@H](O)c2ccccc2)C1 ZINC000217572968 BD For-Sale Unstable SLC6A1 0 43 CN1CCC[C@@H](CNC[C@@H](O)c2ccccc2)C1 ZINC000217572968 BD For-Sale Unstable SLC6A3 22 40 O=[S@@](C[C@H]1CCNC1)c1ccc(Cl)cc1 ZINC000217572969 BE For-Sale Unstable SLC6A1 0 42 C[C@@H]1CN(C[C@@H](O)COc2ccc(C#N)cc2)CCCO1 ZINC000217572992 CD On-Demand Unstable ABCB1 33 40 CC(=O)NCC1CCN(C(=O)c2ccc(Br)c(Cl)c2)CC1 ZINC000217573041 FG On-Demand Unstable CCR3 23 42 CC(=O)NCC1CCN(C(=O)c2ccc(Br)c(Cl)c2)CC1 ZINC000217573041 FG On-Demand Unstable CACNA1I 55 44 CC(=O)NCC1CCN(C(=O)c2ccc(Br)c(Cl)c2)CC1 ZINC000217573041 FG On-Demand Unstable L3MBTL1 0 40 CC(=O)NCC1CCN(C(=O)c2ccc(Br)c(Cl)c2)CC1 ZINC000217573041 FG On-Demand Unstable L3MBTL3 64 38 CC(=O)NCC1CCN(C(=O)c2ccc(Br)c(Cl)c2)CC1 ZINC000217573041 FG On-Demand Unstable MBTD1 0 40 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NCc1ccco1 ZINC000217573048 EE In-Stock Unstable CCR8 68 33 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NCc1ccco1 ZINC000217573048 EE In-Stock Unstable SFRP1 93 36 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NCc1ccco1 ZINC000217573048 EE In-Stock Unstable WNT3 76 33 CN1CCC[C@H](CNC[C@@H](O)c2ccccc2)C1 ZINC000217573053 BD For-Sale Unstable SLC6A1 0 43 CN1CCC[C@H](CNC[C@@H](O)c2ccccc2)C1 ZINC000217573053 BD For-Sale Unstable SLC6A3 22 40 N[C@H](C(=O)O)c1ccc(SCC(F)F)cc1 ZINC000217573056 BE For-Sale Unstable CACNA2D1 27 50 O=[S@](C[C@H]1CCNC1)c1ccc(Cl)cc1 ZINC000217573069 BE For-Sale Unstable SLC6A1 0 42 C[C@H]1CN(C[C@@H](O)COc2ccc(C#N)cc2)CCCO1 ZINC000217573084 CD On-Demand Unstable ABCB1 33 40 O=S(=O)(NC1CCCCCCC1)c1ccccc1CO ZINC000217573127 CF For-Sale Unstable CCR8 95 50 O=S(=O)(NC1CCCCCCC1)c1ccccc1CO ZINC000217573127 CF For-Sale Unstable SFRP1 107 34 O=S(=O)(NC1CCCCCCC1)c1ccccc1CO ZINC000217573127 CF For-Sale Unstable WNT3 73 34 N[C@@H](C(=O)O)c1ccc(SCC(F)F)cc1 ZINC000217573136 BE For-Sale Unstable CACNA2D1 27 50 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NC[C@@H]1CCCO1 ZINC000217573153 ED In-Stock Unstable CCR8 71 35 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NC[C@@H]1CCCO1 ZINC000217573153 ED In-Stock Unstable SFRP1 90 33 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NC[C@@H]1CCCO1 ZINC000217573153 ED In-Stock Unstable WNT3 74 33 CC(=O)NCC1CCN(C(=O)c2cc(C)ccc2Br)CC1 ZINC000217573157 FF On-Demand Unstable CACNA1I 42 33 C[C@@H]1CN(C[C@@H](O)COc2cccc(C#N)c2)CCCO1 ZINC000217573175 CD For-Sale Unstable ACOX1 62 32 C[C@@H]1CN(C[C@@H](O)COc2cccc(C#N)c2)CCCO1 ZINC000217573175 CD For-Sale Unstable ABCB1 38 43 C[C@@H]1CN(C[C@@H](O)COc2cccc(C#N)c2)CCCO1 ZINC000217573175 CD For-Sale Unstable CHRNA10 25 44 Cc1cccc(S(=O)(=O)NCC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217573192 HD For-Sale Unstable NPY5R 23 40 CCOC(=O)C(F)(F)Sc1nc2ccccc2[nH]1 ZINC000217573214 CF In-Stock Unstable CACNA1G 0 45 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NC[C@H]1CCCO1 ZINC000217573238 ED In-Stock Unstable CCR8 71 35 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NC[C@H]1CCCO1 ZINC000217573238 ED In-Stock Unstable SFRP1 90 33 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1NC[C@H]1CCCO1 ZINC000217573238 ED In-Stock Unstable WNT3 74 33 C[C@H]1CN(C[C@@H](O)COc2cccc(C#N)c2)CCCO1 ZINC000217573252 CD For-Sale Unstable ACOX1 62 32 C[C@H]1CN(C[C@@H](O)COc2cccc(C#N)c2)CCCO1 ZINC000217573252 CD For-Sale Unstable ABCB1 38 43 C[C@H]1CN(C[C@@H](O)COc2cccc(C#N)c2)CCCO1 ZINC000217573252 CD For-Sale Unstable CHRNA10 25 44 Cc1cccc(S(=O)(=O)NCC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217573268 HD For-Sale Unstable NPY5R 23 40 CN1CC[C@@H](NC(=O)c2ccc(F)c([N+](=O)[O-])c2)C1=O ZINC000217573301 CC For-Sale Unstable TAAR1 17 44 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1N1CCCC1 ZINC000217573335 DD In-Stock Unstable SLC6A9 16 43 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1N1CCCC1 ZINC000217573335 DD In-Stock Unstable CCR8 46 32 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1N1CCCC1 ZINC000217573335 DD In-Stock Unstable LIPG 46 34 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1N1CCCC1 ZINC000217573335 DD In-Stock Unstable SFRP1 113 39 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1N1CCCC1 ZINC000217573335 DD In-Stock Unstable WNT3 87 40 CN1CC[C@H](NC(=O)c2ccc(F)c([N+](=O)[O-])c2)C1=O ZINC000217573357 CC For-Sale Unstable TAAR1 17 44 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1N1CCCCC1 ZINC000217573428 DD In-Stock Unstable SLC6A9 15 45 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1N1CCCCC1 ZINC000217573428 DD In-Stock Unstable LIPG 40 34 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1N1CCCCC1 ZINC000217573428 DD In-Stock Unstable SFRP1 112 39 O=C(O)c1cc(S(=O)(=O)NC2CC2)ccc1N1CCCCC1 ZINC000217573428 DD In-Stock Unstable WNT3 86 39 CN(C)c1cccc(NC(=O)NCC2CCCC2)c1 ZINC000217573442 CG For-Sale Unstable CCR3 63 39 CN(C)c1cccc(NC(=O)NCC2CCCC2)c1 ZINC000217573442 CG For-Sale Unstable EPHX2 25 65 CN(C)c1cccc(NC(=O)NCC2CCCC2)c1 ZINC000217573442 CG For-Sale Unstable ACAT 0 43 O=C(CCc1cccc(Cl)c1)NC[C@@H](O)Cc1ccccc1 ZINC000217573473 DF In-Stock Unstable CMA1 18 61 O=C(CCc1cccc(Cl)c1)NC[C@@H](O)Cc1ccccc1 ZINC000217573473 DF In-Stock Unstable PAM 0 44 O=C(CCc1cccc(Cl)c1)NC[C@@H](O)Cc1ccccc1 ZINC000217573473 DF In-Stock Unstable CTSV 38 41 O=C(CCc1cccc(Cl)c1)NC[C@@H](O)Cc1ccccc1 ZINC000217573473 DF In-Stock Unstable PDS 56 39 O=C(CCc1cccc(Cl)c1)NC[C@@H](O)Cc1ccccc1 ZINC000217573473 DF In-Stock Unstable LMGT2 0 45 CCOCCCNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217573529 ED In-Stock Unstable CCR8 76 36 CCOCCCNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217573529 ED In-Stock Unstable SFRP1 82 33 CCOCCCNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217573529 ED In-Stock Unstable WNT3 59 33 O=C(NCC1CCCC1)Nc1ccc2nc[nH]c2c1 ZINC000217573549 CF For-Sale Unstable QPCT 19 41 O=C(NCC1CCCC1)Nc1ccc2nc[nH]c2c1 ZINC000217573549 CF For-Sale Unstable PRMT3 70 45 O=C(CCc1cccc(Cl)c1)NC[C@H](O)Cc1ccccc1 ZINC000217573558 DF In-Stock Unstable CMA1 18 61 O=C(CCc1cccc(Cl)c1)NC[C@H](O)Cc1ccccc1 ZINC000217573558 DF In-Stock Unstable PAM 0 44 O=C(CCc1cccc(Cl)c1)NC[C@H](O)Cc1ccccc1 ZINC000217573558 DF In-Stock Unstable CTSV 38 41 O=C(CCc1cccc(Cl)c1)NC[C@H](O)Cc1ccccc1 ZINC000217573558 DF In-Stock Unstable PDS 56 39 O=C(CCc1cccc(Cl)c1)NC[C@H](O)Cc1ccccc1 ZINC000217573558 DF In-Stock Unstable LMGT2 0 45 CC(C)OCCCNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217573638 FE In-Stock Unstable SFRP1 87 34 CC(C)OCCCNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217573638 FE In-Stock Unstable WNT3 49 31 COc1ccc(C(=O)NC[C@H](O)Cc2ccccc2)cc1F ZINC000217573660 DE In-Stock Unstable PPARG 17 42 COc1ccc(C(=O)NC[C@H](O)Cc2ccccc2)cc1F ZINC000217573660 DE In-Stock Unstable PPARA 22 41 COc1ccc(C(=O)NC[C@H](O)Cc2ccccc2)cc1F ZINC000217573660 DE In-Stock Unstable MME 26 44 COc1ccc(C(=O)NC[C@H](O)Cc2ccccc2)cc1F ZINC000217573660 DE In-Stock Unstable TRPV1 0 40 COc1ccc(C(=O)NC[C@H](O)Cc2ccccc2)cc1F ZINC000217573660 DE In-Stock Unstable CPT1A 45 31 COc1ccc(C(=O)NC[C@H](O)Cc2ccccc2)cc1F ZINC000217573660 DE In-Stock Unstable PPARD 23 44 COc1ccc(C(=O)NC[C@H](O)Cc2ccccc2)cc1F ZINC000217573660 DE In-Stock Unstable POL 0 42 COc1ccc(C(=O)NC[C@H](O)Cc2ccccc2)cc1F ZINC000217573660 DE In-Stock Unstable PDS 47 34 O=C(CCn1c(=O)[nH]c2ccccc21)NCCc1nc(C(=O)O)cs1 ZINC000217573671 FD In-Stock Unstable PLD1 51 34 O=C(CCn1c(=O)[nH]c2ccccc21)NCCc1nc(C(=O)O)cs1 ZINC000217573671 FD In-Stock Unstable PLD2 45 36 O=C1O[C@@]2(CCCN(C(=O)CNS(=O)(=O)c3ccc(F)c(Cl)c3)C2)c2ccccc21 ZINC000217573729 JE For-Sale Unstable NPY5R 25 44 CC(C)(C)OC(=O)N1Cc2ccccc2C[C@H]1C(=O)NC[C@@H]1CC[C@@H](C(=O)NCc2ccco2)CC1 ZINC000217573731 JI In-Stock Unstable OPRM1 0 40 CC(C)(C)OC(=O)N1Cc2ccccc2C[C@H]1C(=O)NC[C@@H]1CC[C@@H](C(=O)NCc2ccco2)CC1 ZINC000217573731 JI In-Stock Unstable OPRD1 49 35 CC(C)(C)OC(=O)N1Cc2ccccc2C[C@H]1C(=O)NC[C@@H]1CC[C@@H](C(=O)NCc2ccco2)CC1 ZINC000217573731 JI In-Stock Unstable HDAC8 0 41 CC(C)(C)OC(=O)N1Cc2ccccc2C[C@H]1C(=O)NC[C@@H]1CC[C@@H](C(=O)NCc2ccco2)CC1 ZINC000217573731 JI In-Stock Unstable PREP 18 42 CC(C)(C)OC(=O)N1Cc2ccccc2C[C@H]1C(=O)NC[C@@H]1CC[C@@H](C(=O)NCc2ccco2)CC1 ZINC000217573731 JI In-Stock Unstable CFTR 51 31 CCCCCNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217573734 EE In-Stock Unstable TBXA2R 15 40 CCCCCNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217573734 EE In-Stock Unstable CCR8 78 35 CCCCCNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217573734 EE In-Stock Unstable SFRP1 87 35 CCCCCNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217573734 EE In-Stock Unstable WNT3 66 35 CC(C)CNC[C@H](O)CO[C@@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217573737 CG For-Sale Unstable TRPM8 0 40 COc1ccc(C(=O)NC[C@@H](O)Cc2ccccc2)cc1F ZINC000217573739 DE In-Stock Unstable PPARG 17 42 COc1ccc(C(=O)NC[C@@H](O)Cc2ccccc2)cc1F ZINC000217573739 DE In-Stock Unstable PPARA 22 41 COc1ccc(C(=O)NC[C@@H](O)Cc2ccccc2)cc1F ZINC000217573739 DE In-Stock Unstable MME 26 44 COc1ccc(C(=O)NC[C@@H](O)Cc2ccccc2)cc1F ZINC000217573739 DE In-Stock Unstable TRPV1 0 40 COc1ccc(C(=O)NC[C@@H](O)Cc2ccccc2)cc1F ZINC000217573739 DE In-Stock Unstable CPT1A 45 31 COc1ccc(C(=O)NC[C@@H](O)Cc2ccccc2)cc1F ZINC000217573739 DE In-Stock Unstable PPARD 23 44 COc1ccc(C(=O)NC[C@@H](O)Cc2ccccc2)cc1F ZINC000217573739 DE In-Stock Unstable POL 0 42 COc1ccc(C(=O)NC[C@@H](O)Cc2ccccc2)cc1F ZINC000217573739 DE In-Stock Unstable PDS 47 34 O=C1O[C@]2(CCCN(C(=O)CNS(=O)(=O)c3ccc(F)c(Cl)c3)C2)c2ccccc21 ZINC000217573832 JE For-Sale Unstable NPY5R 25 44 CC(C)CCNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217573854 EE In-Stock Unstable CCR8 76 33 CC(C)CCNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217573854 EE In-Stock Unstable SFRP1 87 35 CC(C)CCNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217573854 EE In-Stock Unstable WNT3 67 36 CCO[C@@H]1C[C@@H](NC(=O)c2ccc(F)nc2)C1(C)C ZINC000217573904 CE For-Sale Unstable SSTR5 25 40 COc1cc(CN[C@@]23C[C@@H]4C[C@@](C)(C[C@@](C)(C4)C2)C3)ccc1OCC(N)=O ZINC000217573929 FG In-Stock Unstable DRTS_TRYCR 44 30 O=C1O[C@@]2(CCCN(C(=O)CCNS(=O)(=O)c3ccc(F)c(Cl)c3)C2)c2ccccc21 ZINC000217573945 JF For-Sale Unstable NPY5R 22 41 O=C(c1cc2c(Cl)cccc2[nH]1)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217573966 FG In-Stock Unstable CHRNA4 36 48 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217573970 EE In-Stock Unstable CCR8 63 34 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217573970 EE In-Stock Unstable SFRP1 71 34 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217573970 EE In-Stock Unstable WNT3 47 34 N#C[C@@H]1CC[C@@H](c2ccccc2)C[C@@H]1N1CCCOCC1 ZINC000217573976 CG For-Sale Unstable SLC18A3 43 38 CCO[C@H]1C[C@@H](NC(=O)c2ccc(F)nc2)C1(C)C ZINC000217573978 CE For-Sale Unstable SSTR5 25 40 CN1CCC[C@@H](CNC[C@@H](O)COc2ccc(F)cc2)C1 ZINC000217573990 CD For-Sale Unstable ADRB2 52 40 CN1CCC[C@@H](CNC[C@@H](O)COc2ccc(F)cc2)C1 ZINC000217573990 CD For-Sale Unstable ADRB1 67 45 CN1CCC[C@@H](CNC[C@@H](O)COc2ccc(F)cc2)C1 ZINC000217573990 CD For-Sale Unstable GRIN1 23 43 CN1CCC[C@@H](CNC[C@@H](O)COc2ccc(F)cc2)C1 ZINC000217573990 CD For-Sale Unstable ADRB3 45 44 CN1CCC[C@@H](CNC[C@@H](O)COc2ccc(F)cc2)C1 ZINC000217573990 CD For-Sale Unstable ABCB1 22 41 CN1CCC[C@@H](CNC[C@@H](O)COc2ccc(F)cc2)C1 ZINC000217573990 CD For-Sale Unstable CHRNA10 50 34 CC(C)(C)OC(=O)N1CCC([C@@H]2CC(=O)CCO2)CC1 ZINC000217574001 CE For-Sale Unstable GPR119 36 47 CCN1CCN(C(=O)NCC2CCCC2)CC1 ZINC000217574010 BD On-Demand Unstable CACNA1I 46 35 O=C1O[C@]2(CCCN(C(=O)CCNS(=O)(=O)c3ccc(F)c(Cl)c3)C2)c2ccccc21 ZINC000217574041 JF For-Sale Unstable NPY5R 22 41 CCO[C@@H]1C[C@H](NC(=O)c2ccc(F)nc2)C1(C)C ZINC000217574067 CE For-Sale Unstable SSTR5 25 40 CCC[C@H](C)Nc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217574069 EE In-Stock Unstable CCR8 63 34 CCC[C@H](C)Nc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217574069 EE In-Stock Unstable SFRP1 71 34 CCC[C@H](C)Nc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217574069 EE In-Stock Unstable WNT3 47 34 N#C[C@H]1CC[C@@H](c2ccccc2)C[C@@H]1N1CCCOCC1 ZINC000217574074 CG For-Sale Unstable SLC18A3 43 38 CN1CCC[C@H](CNC[C@@H](O)COc2ccc(F)cc2)C1 ZINC000217574076 CD For-Sale Unstable ADRB2 52 40 CN1CCC[C@H](CNC[C@@H](O)COc2ccc(F)cc2)C1 ZINC000217574076 CD For-Sale Unstable ADRB1 67 45 CN1CCC[C@H](CNC[C@@H](O)COc2ccc(F)cc2)C1 ZINC000217574076 CD For-Sale Unstable GRIN1 23 43 CN1CCC[C@H](CNC[C@@H](O)COc2ccc(F)cc2)C1 ZINC000217574076 CD For-Sale Unstable ADRB3 45 45 CN1CCC[C@H](CNC[C@@H](O)COc2ccc(F)cc2)C1 ZINC000217574076 CD For-Sale Unstable ABCB1 22 41 CN1CCC[C@H](CNC[C@@H](O)COc2ccc(F)cc2)C1 ZINC000217574076 CD For-Sale Unstable CHRNA10 50 34 CC(C)(C)OC(=O)N1CCC([C@H]2CC(=O)CCO2)CC1 ZINC000217574103 CE For-Sale Unstable GPR119 36 47 N#C[C@@H]1CC[C@H](c2ccccc2)C[C@@H]1N1CCCOCC1 ZINC000217574144 CG For-Sale Unstable SLC18A3 43 38 CCO[C@H]1C[C@H](NC(=O)c2ccc(F)nc2)C1(C)C ZINC000217574156 CE For-Sale Unstable SSTR5 25 40 C=C(CC)COc1c(/C=C\C(=O)O)cccc1OC ZINC000217574160 CG For-Sale Unstable PTGER2 54 50 C=C(CC)COc1c(/C=C\C(=O)O)cccc1OC ZINC000217574160 CG For-Sale Unstable PTGER4 26 43 C=C(CC)COc1c(/C=C\C(=O)O)cccc1OC ZINC000217574160 CG For-Sale Unstable PTGER3 22 50 O=C1O[C@@]2(CCCN(C(=O)CCNS(=O)(=O)c3cccc(F)c3)C2)c2ccccc21 ZINC000217574165 IE For-Sale Unstable NPY5R 25 44 COC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217574167 ED In-Stock Unstable CCR8 55 31 COC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217574167 ED In-Stock Unstable SFRP1 73 33 COC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217574167 ED In-Stock Unstable WNT3 52 33 O=C(NC[C@@H]1C[C@@H]1c1ccsc1)OCc1ccccc1 ZINC000217574191 CH For-Sale Unstable PAPA1_CARPA 42 33 O=C(NC[C@@H]1C[C@@H]1c1ccsc1)OCc1ccccc1 ZINC000217574191 CH For-Sale Unstable CAPNS1 58 33 O=C(NC[C@@H]1C[C@@H]1c1ccsc1)OCc1ccccc1 ZINC000217574191 CH For-Sale Unstable CAPN1 55 38 O=C(NC[C@@H]1C[C@@H]1c1ccsc1)OCc1ccccc1 ZINC000217574191 CH For-Sale Unstable CAPN2 92 38 O=C(NC[C@@H]1C[C@@H]1c1ccsc1)OCc1ccccc1 ZINC000217574191 CH For-Sale Unstable NPR 61 36 O=C(NC[C@@H]1C[C@@H]1c1ccsc1)OCc1ccccc1 ZINC000217574191 CH For-Sale Unstable KDM1A 24 49 N#C[C@H]1CC[C@H](c2ccccc2)C[C@@H]1N1CCCOCC1 ZINC000217574222 CG For-Sale Unstable SLC18A3 43 38 O=C1O[C@]2(CCCN(C(=O)CCNS(=O)(=O)c3cccc(F)c3)C2)c2ccccc21 ZINC000217574228 IE For-Sale Unstable NPY5R 25 44 O=S(=O)(NC[C@@H](O)Cc1ccccc1)c1cccc2cccnc12 ZINC000217574235 EE In-Stock Unstable NFKBIA 0 42 O=S(=O)(NC[C@@H](O)Cc1ccccc1)c1cccc2cccnc12 ZINC000217574235 EE In-Stock Unstable C0L093_TOBAC 46 31 COC[C@H](C)Nc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217574249 ED In-Stock Unstable CCR8 55 31 COC[C@H](C)Nc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217574249 ED In-Stock Unstable SFRP1 73 33 COC[C@H](C)Nc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217574249 ED In-Stock Unstable WNT3 52 33 C=C(CC)COc1cc(OCCC)ccc1/C=C\C(=O)O ZINC000217574265 CH For-Sale Unstable PLA2G4B 62 35 O=C(NC[C@H]1C[C@@H]1c1ccsc1)OCc1ccccc1 ZINC000217574295 CH For-Sale Unstable PAPA1_CARPA 42 33 O=C(NC[C@H]1C[C@@H]1c1ccsc1)OCc1ccccc1 ZINC000217574295 CH For-Sale Unstable CAPNS1 58 33 O=C(NC[C@H]1C[C@@H]1c1ccsc1)OCc1ccccc1 ZINC000217574295 CH For-Sale Unstable CAPN1 55 38 O=C(NC[C@H]1C[C@@H]1c1ccsc1)OCc1ccccc1 ZINC000217574295 CH For-Sale Unstable CAPN2 92 38 O=C(NC[C@H]1C[C@@H]1c1ccsc1)OCc1ccccc1 ZINC000217574295 CH For-Sale Unstable NPR 61 36 O=C(NC[C@H]1C[C@@H]1c1ccsc1)OCc1ccccc1 ZINC000217574295 CH For-Sale Unstable KDM1A 24 49 O=S(=O)(NC[C@H](O)Cc1ccccc1)c1cccc2cccnc12 ZINC000217574308 EE In-Stock Unstable NFKBIA 0 42 O=S(=O)(NC[C@H](O)Cc1ccccc1)c1cccc2cccnc12 ZINC000217574308 EE In-Stock Unstable C0L093_TOBAC 46 31 O=C1O[C@@]2(CCCN(C(=O)CNS(=O)(=O)c3c(F)cccc3F)C2)c2ccccc21 ZINC000217574348 ID For-Sale Unstable NPY5R 26 43 O=C(NCC1CCCC1)Nc1ccc2cn[nH]c2c1 ZINC000217574354 CF For-Sale Unstable CCR3 20 43 O=C(NCC1CCCC1)Nc1ccc2cn[nH]c2c1 ZINC000217574354 CF For-Sale Unstable ROCK1 15 47 O=C(NCC1CCCC1)Nc1ccc2cn[nH]c2c1 ZINC000217574354 CF For-Sale Unstable ROCK2 22 57 O=C(NCC1CCCC1)Nc1ccc2cn[nH]c2c1 ZINC000217574354 CF For-Sale Unstable PRMT3 41 40 CCCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217574372 EE In-Stock Unstable CCR8 81 39 CCCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217574372 EE In-Stock Unstable SFRP1 98 36 CCCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217574372 EE In-Stock Unstable WNT3 79 35 O=C(NC[C@@H]1C[C@H]1c1ccsc1)OCc1ccccc1 ZINC000217574389 CH For-Sale Unstable PAPA1_CARPA 42 33 O=C(NC[C@@H]1C[C@H]1c1ccsc1)OCc1ccccc1 ZINC000217574389 CH For-Sale Unstable CAPNS1 58 33 O=C(NC[C@@H]1C[C@H]1c1ccsc1)OCc1ccccc1 ZINC000217574389 CH For-Sale Unstable CAPN1 55 38 O=C(NC[C@@H]1C[C@H]1c1ccsc1)OCc1ccccc1 ZINC000217574389 CH For-Sale Unstable CAPN2 92 38 O=C(NC[C@@H]1C[C@H]1c1ccsc1)OCc1ccccc1 ZINC000217574389 CH For-Sale Unstable NPR 61 36 O=C(NC[C@@H]1C[C@H]1c1ccsc1)OCc1ccccc1 ZINC000217574389 CH For-Sale Unstable KDM1A 24 49 O=C1COc2c(Br)cc(O)cc2N1 ZINC000217574411 BD For-Sale Unstable ADRB2 15 45 O=C1COc2c(Br)cc(O)cc2N1 ZINC000217574411 BD For-Sale Unstable ADRB1 15 45 O=C1O[C@]2(CCCN(C(=O)CNS(=O)(=O)c3c(F)cccc3F)C2)c2ccccc21 ZINC000217574429 ID For-Sale Unstable NPY5R 26 43 Cn1cc([C@H](O)CNC(=O)c2ccc3ncsc3c2)c2ccccc21 ZINC000217574432 FG In-Stock Unstable UL54 43 33 O=C(NCC1CCCC1)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217574467 FK For-Sale Unstable CCR3 18 40 O=C(NCC1CCCC1)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217574467 FK For-Sale Unstable EPHX2 31 53 O=C(NCC1CCCC1)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217574467 FK For-Sale Unstable CACNA1I 39 46 O=C(NCC1CCCC1)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217574467 FK For-Sale Unstable PTPA 0 44 O=C(NC[C@H]1C[C@H]1c1ccsc1)OCc1ccccc1 ZINC000217574474 CH For-Sale Unstable PAPA1_CARPA 42 33 O=C(NC[C@H]1C[C@H]1c1ccsc1)OCc1ccccc1 ZINC000217574474 CH For-Sale Unstable CAPNS1 58 33 O=C(NC[C@H]1C[C@H]1c1ccsc1)OCc1ccccc1 ZINC000217574474 CH For-Sale Unstable CAPN1 55 38 O=C(NC[C@H]1C[C@H]1c1ccsc1)OCc1ccccc1 ZINC000217574474 CH For-Sale Unstable CAPN2 92 38 O=C(NC[C@H]1C[C@H]1c1ccsc1)OCc1ccccc1 ZINC000217574474 CH For-Sale Unstable NPR 61 36 O=C(NC[C@H]1C[C@H]1c1ccsc1)OCc1ccccc1 ZINC000217574474 CH For-Sale Unstable KDM1A 24 49 CC(C)Nc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217574477 EE In-Stock Unstable CCR8 73 39 CC(C)Nc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217574477 EE In-Stock Unstable SFRP1 91 34 CC(C)Nc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217574477 EE In-Stock Unstable WNT3 74 34 Cn1cc([C@@H](O)CNC(=O)c2ccc3ncsc3c2)c2ccccc21 ZINC000217574511 FG In-Stock Unstable UL54 43 33 O=C1O[C@@]2(CCCN(C(=O)CCNS(=O)(=O)c3c(F)cccc3F)C2)c2ccccc21 ZINC000217574548 JE For-Sale Unstable NPY5R 23 42 Nc1ccc(C(=O)NC(=O)NCC2CCCC2)cc1 ZINC000217574563 CD For-Sale Unstable LDLR 0 41 Nc1ccc(C(=O)NC(=O)NCC2CCCC2)cc1 ZINC000217574563 CD For-Sale Unstable CACNA1I 41 34 CCCCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217574596 EF In-Stock Unstable CCR8 80 38 CCCCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217574596 EF In-Stock Unstable SFRP1 93 35 CCCCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217574596 EF In-Stock Unstable WNT3 77 34 Fc1cc(CN[C@@H]2C[C@@H]3C[C@@H]2[C@@H]2CCC[C@@H]32)ccc1Cl ZINC000217574608 CI For-Sale Unstable SSTR3 22 44 O=C1O[C@]2(CCCN(C(=O)CCNS(=O)(=O)c3c(F)cccc3F)C2)c2ccccc21 ZINC000217574614 JE For-Sale Unstable NPY5R 23 42 CCN(CC)c1ccc(NC(=O)NCC2CCCC2)cc1 ZINC000217574664 CH For-Sale Unstable GHSR 0 46 CCN(CC)c1ccc(NC(=O)NCC2CCCC2)cc1 ZINC000217574664 CH For-Sale Unstable EPHX2 32 64 Fc1cc(CN[C@H]2C[C@@H]3C[C@@H]2[C@@H]2CCC[C@@H]32)ccc1Cl ZINC000217574674 CI For-Sale Unstable SSTR3 22 44 CC(C)CNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217574694 EF In-Stock Unstable MTNN 71 33 CC(C)CNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217574694 EF In-Stock Unstable CCR8 79 39 CC(C)CNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217574694 EF In-Stock Unstable SFRP1 99 36 CC(C)CNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217574694 EF In-Stock Unstable WNT3 79 37 Fc1cc(CN[C@@H]2C[C@H]3C[C@@H]2[C@@H]2CCC[C@@H]32)ccc1Cl ZINC000217574775 CI For-Sale Unstable SSTR3 22 44 CC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217574827 EF In-Stock Unstable CCR8 70 37 CC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217574827 EF In-Stock Unstable SFRP1 80 34 CC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217574827 EF In-Stock Unstable WNT3 64 34 Fc1cc(CN[C@H]2C[C@H]3C[C@@H]2[C@@H]2CCC[C@@H]32)ccc1Cl ZINC000217574843 CI For-Sale Unstable SSTR3 22 44 O=C(NC1CCCCC1)[C@@H]1CC[C@@H](CNC(=O)[C@@H]2Cc3ccccc3CN2)CC1 ZINC000217574887 GG In-Stock Unstable NPY2R 0 40 O=C(NC1CCCCC1)[C@@H]1CC[C@@H](CNC(=O)[C@@H]2Cc3ccccc3CN2)CC1 ZINC000217574887 GG In-Stock Unstable EPHX2 33 42 CC[C@H](C)Nc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217574911 EF In-Stock Unstable CCR8 70 37 CC[C@H](C)Nc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217574911 EF In-Stock Unstable SFRP1 80 34 CC[C@H](C)Nc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217574911 EF In-Stock Unstable WNT3 64 34 O=C(Nc1nc(=O)n([C@@H]2O[C@H](COC(=O)c3ccccc3)[C@@H](OC(=O)c3ccccc3)[C@@H]2OC(=O)c2ccccc2)cc1F)c1ccccc1 ZINC000217574917 KJ In-Stock Unstable TYMS 23 43 O=C(Nc1nc(=O)n([C@@H]2O[C@H](COC(=O)c3ccccc3)[C@@H](OC(=O)c3ccccc3)[C@@H]2OC(=O)c2ccccc2)cc1F)c1ccccc1 ZINC000217574917 KJ In-Stock Unstable P2RY4 41 31 O=C(Nc1nc(=O)n([C@@H]2O[C@H](COC(=O)c3ccccc3)[C@@H](OC(=O)c3ccccc3)[C@@H]2OC(=O)c2ccccc2)cc1F)c1ccccc1 ZINC000217574917 KJ In-Stock Unstable P2RY2 40 36 O=S(=O)(NC1CCCCCCC1)c1ccc(CO)cc1 ZINC000217574930 CF For-Sale Unstable TBXA2R 15 43 O=S(=O)(NC1CCCCCCC1)c1ccc(CO)cc1 ZINC000217574930 CF For-Sale Unstable CHUK 32 40 CN1CCC[C@@H](CNC[C@@H](O)COc2ccccc2Cl)C1 ZINC000217574980 DE For-Sale Unstable ADRB2 37 48 CN1CCC[C@@H](CNC[C@@H](O)COc2ccccc2Cl)C1 ZINC000217574980 DE For-Sale Unstable ADRB1 51 47 CN1CCC[C@@H](CNC[C@@H](O)COc2ccccc2Cl)C1 ZINC000217574980 DE For-Sale Unstable ADRB3 27 49 CN1CCC[C@@H](CNC[C@@H](O)COc2ccccc2Cl)C1 ZINC000217574980 DE For-Sale Unstable CYP2D26 0 40 CN1CCC[C@@H](CNC[C@@H](O)COc2ccccc2Cl)C1 ZINC000217574980 DE For-Sale Unstable ABCB1 45 38 COC(=O)[C@@H](C)CN1CCc2sccc2[C@@H]1C ZINC000217574992 CE For-Sale Unstable TRPM8 16 40 CC(C)(C)Nc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217575020 EF In-Stock Unstable CCR8 78 41 CC(C)(C)Nc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217575020 EF In-Stock Unstable SFRP1 108 37 CC(C)(C)Nc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217575020 EF In-Stock Unstable WNT3 84 38 CN1CCC[C@H](CNC[C@@H](O)COc2ccccc2Cl)C1 ZINC000217575072 DE For-Sale Unstable ADRB2 37 48 CN1CCC[C@H](CNC[C@@H](O)COc2ccccc2Cl)C1 ZINC000217575072 DE For-Sale Unstable ADRB1 51 47 CN1CCC[C@H](CNC[C@@H](O)COc2ccccc2Cl)C1 ZINC000217575072 DE For-Sale Unstable ADRB3 27 49 CN1CCC[C@H](CNC[C@@H](O)COc2ccccc2Cl)C1 ZINC000217575072 DE For-Sale Unstable CYP2D26 0 40 CN1CCC[C@H](CNC[C@@H](O)COc2ccccc2Cl)C1 ZINC000217575072 DE For-Sale Unstable ABCB1 45 38 C=CCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217575122 DE In-Stock Unstable F13A1 29 41 C=CCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217575122 DE In-Stock Unstable CCR8 43 33 C=CCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217575122 DE In-Stock Unstable SFRP1 93 35 C=CCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217575122 DE In-Stock Unstable WNT3 74 34 O=C(NCC1CCCC1)Nc1cc(Cl)cc(Cl)c1 ZINC000217575133 CI For-Sale Unstable CCR3 17 46 O=C(NCC1CCCC1)Nc1cc(Cl)cc(Cl)c1 ZINC000217575133 CI For-Sale Unstable EPHX2 16 73 O=C(NCC1CCCC1)Nc1cc(Cl)cc(Cl)c1 ZINC000217575133 CI For-Sale Unstable CACNA1I 82 45 Cn1cc([C@H](O)CNC(=O)CCc2cccc(Cl)c2)c2ccccc21 ZINC000217575159 FH In-Stock Unstable UL54 54 36 CN1CCC[C@@H](CNC[C@@H](O)COc2ccc(Cl)cc2)C1 ZINC000217575181 DE For-Sale Unstable ADRB2 49 40 CN1CCC[C@@H](CNC[C@@H](O)COc2ccc(Cl)cc2)C1 ZINC000217575181 DE For-Sale Unstable ADRB1 63 44 CN1CCC[C@@H](CNC[C@@H](O)COc2ccc(Cl)cc2)C1 ZINC000217575181 DE For-Sale Unstable GRIN1 25 43 CN1CCC[C@@H](CNC[C@@H](O)COc2ccc(Cl)cc2)C1 ZINC000217575181 DE For-Sale Unstable ADRB3 43 42 CN1CCC[C@@H](CNC[C@@H](O)COc2ccc(Cl)cc2)C1 ZINC000217575181 DE For-Sale Unstable EBP 19 42 CN1CCC[C@@H](CNC[C@@H](O)COc2ccc(Cl)cc2)C1 ZINC000217575181 DE For-Sale Unstable CHRNA10 33 46 O=C(c1ccc(Cl)cc1)[C@H]1[C@H]2C(=O)N(c3cccc(C(F)(F)F)c3)C(=O)[C@@H]2[C@H]2CCCN21 ZINC000217575189 JI In-Stock Unstable CCR2 18 40 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NC1CC1 ZINC000217575201 DE In-Stock Unstable CCR8 53 40 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NC1CC1 ZINC000217575201 DE In-Stock Unstable SFRP1 96 34 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NC1CC1 ZINC000217575201 DE In-Stock Unstable WNT3 76 34 C[C@@H]1CCCC[C@@]1(NC(=O)/C=C\c1cccnc1)C(=O)O ZINC000217575234 CE For-Sale Unstable C3AR1 25 44 Cn1cc([C@@H](O)CNC(=O)CCc2cccc(Cl)c2)c2ccccc21 ZINC000217575256 FH In-Stock Unstable UL54 54 36 CN1CCC[C@H](CNC[C@@H](O)COc2ccc(Cl)cc2)C1 ZINC000217575267 DE For-Sale Unstable ADRB2 49 40 CN1CCC[C@H](CNC[C@@H](O)COc2ccc(Cl)cc2)C1 ZINC000217575267 DE For-Sale Unstable ADRB1 63 44 CN1CCC[C@H](CNC[C@@H](O)COc2ccc(Cl)cc2)C1 ZINC000217575267 DE For-Sale Unstable GRIN1 25 43 CN1CCC[C@H](CNC[C@@H](O)COc2ccc(Cl)cc2)C1 ZINC000217575267 DE For-Sale Unstable ADRB3 43 42 CN1CCC[C@H](CNC[C@@H](O)COc2ccc(Cl)cc2)C1 ZINC000217575267 DE For-Sale Unstable EBP 19 42 CN1CCC[C@H](CNC[C@@H](O)COc2ccc(Cl)cc2)C1 ZINC000217575267 DE For-Sale Unstable CHRNA10 33 46 O=C(c1ccc(Cl)cc1)[C@@H]1[C@H]2C(=O)N(c3cccc(C(F)(F)F)c3)C(=O)[C@@H]2[C@H]2CCCN12 ZINC000217575268 JI In-Stock Unstable CCR2 18 40 O=C1O[C@@]2(CCCN(C(=O)c3cccc(NS(=O)(=O)c4cccc(F)c4)c3)C2)c2ccccc21 ZINC000217575309 JH For-Sale Unstable NPY5R 23 43 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NC1CCCC1 ZINC000217575313 FF In-Stock Unstable CCR8 41 31 C[C@H]1CCCC[C@@]1(NC(=O)/C=C\c1cccnc1)C(=O)O ZINC000217575319 CE For-Sale Unstable C3AR1 25 44 OC1CCC(NC[C@H](O)c2ccccc2)CC1 ZINC000217575344 BD On-Demand Unstable SLC6A3 15 63 OC1CCC(NC[C@H](O)c2ccccc2)CC1 ZINC000217575344 BD On-Demand Unstable AOC3 19 49 CCNC(=O)c1ccc(N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)c(NC(=O)c2ccc(C)n(C)c2=O)c1 ZINC000217575364 KE In-Stock Unstable CHRNA4 26 43 COc1ccc(C(=O)NC[C@@H](O)c2cn(C)c3ccccc23)cc1F ZINC000217575371 EF In-Stock Unstable CYSLTR1 23 40 COc1ccc(C(=O)NC[C@@H](O)c2cn(C)c3ccccc23)cc1F ZINC000217575371 EF In-Stock Unstable CPT1A 49 34 O=C1O[C@]2(CCCN(C(=O)c3cccc(NS(=O)(=O)c4cccc(F)c4)c3)C2)c2ccccc21 ZINC000217575386 JH For-Sale Unstable NPY5R 23 43 CN1CCC[C@@H](CNC[C@@H](O)COc2cccc(Cl)c2)C1 ZINC000217575405 DE For-Sale Unstable ADRB2 40 50 CN1CCC[C@@H](CNC[C@@H](O)COc2cccc(Cl)c2)C1 ZINC000217575405 DE For-Sale Unstable ADRB1 59 41 CN1CCC[C@@H](CNC[C@@H](O)COc2cccc(Cl)c2)C1 ZINC000217575405 DE For-Sale Unstable PTGFR 20 40 CN1CCC[C@@H](CNC[C@@H](O)COc2cccc(Cl)c2)C1 ZINC000217575405 DE For-Sale Unstable GRIN1 0 40 CN1CCC[C@@H](CNC[C@@H](O)COc2cccc(Cl)c2)C1 ZINC000217575405 DE For-Sale Unstable ADRB3 46 44 CN1CCC[C@@H](CNC[C@@H](O)COc2cccc(Cl)c2)C1 ZINC000217575405 DE For-Sale Unstable CHRNA10 61 51 CCOC1CCN(c2ccccc2)CC1 ZINC000217575425 BF For-Sale Unstable HTR1A 18 44 CCOC1CCN(c2ccccc2)CC1 ZINC000217575425 BF For-Sale Unstable DRD2 15 47 CCOC1CCN(c2ccccc2)CC1 ZINC000217575425 BF For-Sale Unstable TIMP3 57 33 OC1CCC(NC[C@@H](O)c2ccccc2)CC1 ZINC000217575431 BD On-Demand Unstable SLC6A3 15 63 OC1CCC(NC[C@@H](O)c2ccccc2)CC1 ZINC000217575431 BD On-Demand Unstable AOC3 19 49 C=CCOc1cnc(C(=O)Nc2ccc(F)c([C@@]3(C(F)F)N=C(N)O[C@@H]4C[C@@H]43)c2)cn1 ZINC000217575433 IF Annotated Unstable BACE2 46 48 C=CCOc1cnc(C(=O)Nc2ccc(F)c([C@@]3(C(F)F)N=C(N)O[C@@H]4C[C@@H]43)c2)cn1 ZINC000217575433 IF Annotated Unstable BACE1 30 49 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NC1CCCCC1 ZINC000217575435 FG In-Stock Unstable CCR8 54 43 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NC1CCCCC1 ZINC000217575435 FG In-Stock Unstable SFRP1 96 35 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NC1CCCCC1 ZINC000217575435 FG In-Stock Unstable WNT3 76 35 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NC1CCCCC1 ZINC000217575435 FG In-Stock Unstable BRD4 0 40 CCN1CCN(Cc2nc(C(C)C)nn2Cc2ccc3c(c2)OCO3)CC1 ZINC000217575448 FE In-Stock Unstable SSTR3 47 30 COc1ccc(C(=O)NC[C@H](O)c2cn(C)c3ccccc23)cc1F ZINC000217575464 EF In-Stock Unstable CYSLTR1 23 40 COc1ccc(C(=O)NC[C@H](O)c2cn(C)c3ccccc23)cc1F ZINC000217575464 EF In-Stock Unstable CPT1A 49 34 C[C@@H]1Cc2ccccc2N1C(=O)NCC1CCCC1 ZINC000217575496 CG On-Demand Unstable DRD4 31 46 C[C@@H]1Cc2ccccc2N1C(=O)NCC1CCCC1 ZINC000217575496 CG On-Demand Unstable TPP2 56 38 CN1CCC[C@H](CNC[C@@H](O)COc2cccc(Cl)c2)C1 ZINC000217575502 DE For-Sale Unstable ADRB2 40 50 CN1CCC[C@H](CNC[C@@H](O)COc2cccc(Cl)c2)C1 ZINC000217575502 DE For-Sale Unstable ADRB1 59 41 CN1CCC[C@H](CNC[C@@H](O)COc2cccc(Cl)c2)C1 ZINC000217575502 DE For-Sale Unstable PTGFR 20 40 CN1CCC[C@H](CNC[C@@H](O)COc2cccc(Cl)c2)C1 ZINC000217575502 DE For-Sale Unstable GRIN1 0 40 CN1CCC[C@H](CNC[C@@H](O)COc2cccc(Cl)c2)C1 ZINC000217575502 DE For-Sale Unstable ADRB3 46 44 CN1CCC[C@H](CNC[C@@H](O)COc2cccc(Cl)c2)C1 ZINC000217575502 DE For-Sale Unstable CHRNA10 61 51 COc1ccc(Br)cc1CCC(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217575512 II For-Sale Unstable NPY5R 20 41 O=C(NCc1ccco1)[C@@H]1CC[C@@H](CNC(=O)[C@@H]2Cc3ccccc3CN2)CC1 ZINC000217575521 GF In-Stock Unstable MC4R 21 42 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NCCC1=CCCCC1 ZINC000217575529 GH In-Stock Unstable SFRP1 61 32 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NCCC1=CCCCC1 ZINC000217575529 GH In-Stock Unstable WNT3 49 31 Cn1cc([C@H](O)CNC(=O)N2CCNC2=O)c2ccccc21 ZINC000217575570 DC In-Stock Unstable PRKCG 44 35 NC/C=C\COc1ccc(Cl)cc1Cl ZINC000217575580 BF For-Sale Unstable S1PR4 27 48 C[C@H]1Cc2ccccc2N1C(=O)NCC1CCCC1 ZINC000217575584 CG On-Demand Unstable DRD4 31 46 C[C@H]1Cc2ccccc2N1C(=O)NCC1CCCC1 ZINC000217575584 CG On-Demand Unstable TPP2 56 38 COc1ccc(Br)cc1CCC(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217575600 II For-Sale Unstable NPY5R 20 41 C[C@]1(C(=O)O)C[C@@H]1CN ZINC000217575616 AC For-Sale Unstable GRM1 0 42 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NCCO ZINC000217575636 ED In-Stock Unstable CCR8 76 40 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NCCO ZINC000217575636 ED In-Stock Unstable SFRP1 97 36 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NCCO ZINC000217575636 ED In-Stock Unstable WNT3 78 35 Cn1cc([C@@H](O)CNC(=O)N2CCNC2=O)c2ccccc21 ZINC000217575652 DC In-Stock Unstable PRKCG 44 35 Cc1cccc(N2CCN(C(=O)NCC3CCCC3)CC2)c1 ZINC000217575695 DG On-Demand Unstable GYRB 0 43 Cc1cccc(N2CCN(C(=O)NCC3CCCC3)CC2)c1 ZINC000217575695 DG On-Demand Unstable HTR1A 23 48 Cc1cccc(N2CCN(C(=O)NCC3CCCC3)CC2)c1 ZINC000217575695 DG On-Demand Unstable CCR1 0 42 Cc1cccc(N2CCN(C(=O)NCC3CCCC3)CC2)c1 ZINC000217575695 DG On-Demand Unstable CACNA1I 51 33 C[C@]1(C(=O)O)C[C@H]1CN ZINC000217575710 AC For-Sale Unstable GRM1 0 42 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NCCCO ZINC000217575750 ED In-Stock Unstable CCR8 72 39 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NCCCO ZINC000217575750 ED In-Stock Unstable SFRP1 92 35 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NCCCO ZINC000217575750 ED In-Stock Unstable WNT3 73 34 O=C(O)/C=C\c1ccc(CNC(=O)Cn2cncn2)cc1 ZINC000217575800 CC For-Sale Unstable HIS3 47 35 C[C@@]1(C(=O)O)C[C@H]1CN ZINC000217575802 AC For-Sale Unstable GRM1 0 42 NC/C=C\COc1cccc(F)c1 ZINC000217575809 AD For-Sale Unstable CHRNA10 30 43 O=C(NCC1CCCC1)N1CCN(c2cccc(Cl)c2)CC1 ZINC000217575810 DG On-Demand Unstable GYRB 0 42 O=C(NCC1CCCC1)N1CCN(c2cccc(Cl)c2)CC1 ZINC000217575810 DG On-Demand Unstable HTR1A 31 49 O=C(NCC1CCCC1)N1CCN(c2cccc(Cl)c2)CC1 ZINC000217575810 DG On-Demand Unstable DRD4 41 35 O=C(NCC1CCCC1)N1CCN(c2cccc(Cl)c2)CC1 ZINC000217575810 DG On-Demand Unstable HTR2A 24 49 O=C(NCC1CCCC1)N1CCN(c2cccc(Cl)c2)CC1 ZINC000217575810 DG On-Demand Unstable ERBB2 0 40 O=C(NCC1CCCC1)N1CCN(c2cccc(Cl)c2)CC1 ZINC000217575810 DG On-Demand Unstable HTR7 24 45 O=C(NCC1CCCC1)N1CCN(c2cccc(Cl)c2)CC1 ZINC000217575810 DG On-Demand Unstable MAPK1 0 46 O=C(NCC1CCCC1)N1CCN(c2cccc(Cl)c2)CC1 ZINC000217575810 DG On-Demand Unstable CACNA1I 55 43 O=C(NCC1CCCC1)N1CCN(c2cccc(Cl)c2)CC1 ZINC000217575810 DG On-Demand Unstable ADAM10 28 42 COCCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217575868 ED In-Stock Unstable CCR8 81 40 COCCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217575868 ED In-Stock Unstable SFRP1 92 34 COCCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217575868 ED In-Stock Unstable WNT3 76 34 COCCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217575868 ED In-Stock Unstable BRD4 21 40 Cc1ccc2nc(-c3ccc(NC(=O)NCC4CCCC4)cc3)sc2c1 ZINC000217575918 FK For-Sale Unstable PPARA 0 41 Cc1ccc2nc(-c3ccc(NC(=O)NCC4CCCC4)cc3)sc2c1 ZINC000217575918 FK For-Sale Unstable CSNK1D 30 40 Cc1ccc2nc(-c3ccc(NC(=O)NCC4CCCC4)cc3)sc2c1 ZINC000217575918 FK For-Sale Unstable NMT1 32 40 Cc1ccc2nc(-c3ccc(NC(=O)NCC4CCCC4)cc3)sc2c1 ZINC000217575918 FK For-Sale Unstable APP 27 54 Cc1ccc2nc(-c3ccc(NC(=O)NCC4CCCC4)cc3)sc2c1 ZINC000217575918 FK For-Sale Unstable EPHX2 15 48 Cc1ccc2nc(-c3ccc(NC(=O)NCC4CCCC4)cc3)sc2c1 ZINC000217575918 FK For-Sale Unstable PRMT3 67 44 Cc1ccc2nc(-c3ccc(NC(=O)NCC4CCCC4)cc3)sc2c1 ZINC000217575918 FK For-Sale Unstable ETHR 18 41 NC/C=C\COc1cccc2ccccc12 ZINC000217575926 BF For-Sale Unstable CYP2D26 0 41 CCOC(=O)C(F)(F)S(=O)(=O)c1nc2ccccc2[nH]1 ZINC000217575949 DD In-Stock Unstable CACNA1G 0 42 COCCCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217575979 FE In-Stock Unstable CCR8 43 35 COCCCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217575979 FE In-Stock Unstable SFRP1 89 33 COCCCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217575979 FE In-Stock Unstable WNT3 51 31 CC(C)(C)CC(=O)NCc1ccc(/C=C\C(=O)O)cc1 ZINC000217576017 CF For-Sale Unstable HDAC1 15 40 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NCc1ccccc1 ZINC000217576079 FG In-Stock Unstable TGM2 21 43 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NCc1ccccc1 ZINC000217576079 FG In-Stock Unstable F13A1 25 43 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NCc1ccccc1 ZINC000217576079 FG In-Stock Unstable CCR8 82 43 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NCc1ccccc1 ZINC000217576079 FG In-Stock Unstable SFRP1 109 39 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NCc1ccccc1 ZINC000217576079 FG In-Stock Unstable WNT3 85 39 O=C1O[C@@]2(CCCN(C(=O)CCc3cccc(Cl)c3)C2)c2ccccc21 ZINC000217576086 FH For-Sale Unstable NPY5R 24 45 O=C(O)/C=C\c1ccc(CNC(=O)Cc2cccs2)cc1 ZINC000217576099 DF For-Sale Unstable CA5B 40 59 O=C(O)/C=C\c1ccc(CNC(=O)Cc2cccs2)cc1 ZINC000217576099 DF For-Sale Unstable CA5A 40 59 Cc1ccc(NC(=O)NCC2CCCC2)c(O)c1 ZINC000217576148 BG For-Sale Unstable THRB 16 42 Cc1ccc(NC(=O)NCC2CCCC2)c(O)c1 ZINC000217576148 BG For-Sale Unstable LDLR 0 40 O=C1O[C@]2(CCCN(C(=O)CCc3cccc(Cl)c3)C2)c2ccccc21 ZINC000217576167 FH For-Sale Unstable NPY5R 24 45 O=C(O)C(F)(F)[S@@](=O)c1nc2ccccc2[nH]1 ZINC000217576171 CD In-Stock Anodyne STK33 44 35 O=C(O)C(F)(F)[S@@](=O)c1nc2ccccc2[nH]1 ZINC000217576171 CD In-Stock Anodyne IDO2 0 44 C[C@@H](Nc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O)c1ccccc1 ZINC000217576187 GH In-Stock Unstable CCR8 85 40 C[C@@H](Nc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O)c1ccccc1 ZINC000217576187 GH In-Stock Unstable SFRP1 124 35 C[C@@H](Nc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O)c1ccccc1 ZINC000217576187 GH In-Stock Unstable WNT3 86 35 CNC[C@H](O)c1ccc(S(C)(=O)=O)cc1F ZINC000217576188 BC For-Sale Unstable PTGS2 18 42 O=C(O)C(F)(F)[S@](=O)c1nc2ccccc2[nH]1 ZINC000217576248 CD In-Stock Anodyne STK33 44 35 O=C(O)C(F)(F)[S@](=O)c1nc2ccccc2[nH]1 ZINC000217576248 CD In-Stock Anodyne IDO2 0 44 O=C(NCC1CCCC1)Nc1c(Cl)cccc1Cl ZINC000217576255 CI For-Sale Unstable CXCL8 40 31 O=C(NCC1CCCC1)Nc1c(Cl)cccc1Cl ZINC000217576255 CI For-Sale Unstable P2RX7 15 43 O=C(NCC1CCCC1)Nc1c(Cl)cccc1Cl ZINC000217576255 CI For-Sale Unstable EPHX2 15 63 O=C(NCC1CCCC1)Nc1c(Cl)cccc1Cl ZINC000217576255 CI For-Sale Unstable CACNA1I 52 36 O=C(NCC1CCCC1)Nc1c(Cl)cccc1Cl ZINC000217576255 CI For-Sale Unstable ACAT 0 52 C[C@H](Nc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O)c1ccccc1 ZINC000217576262 GH In-Stock Unstable CCR8 78 40 C[C@H](Nc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O)c1ccccc1 ZINC000217576262 GH In-Stock Unstable SFRP1 99 35 C[C@H](Nc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O)c1ccccc1 ZINC000217576262 GH In-Stock Unstable WNT3 79 35 O=C(O)/C=C\c1cccc(CNC(=O)c2ccoc2)c1 ZINC000217576268 CE For-Sale Unstable HDAC6 15 42 O=C1O[C@@]2(CCCN(C(=O)CCc3c(F)cccc3Cl)C2)c2ccccc21 ZINC000217576272 GI For-Sale Unstable NPY5R 31 42 CNC[C@@H](O)c1ccc(S(C)(=O)=O)cc1F ZINC000217576273 BC For-Sale Unstable PTGS2 18 42 CCNC(=O)c1ccc(N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)c(NC(=O)c2cccnc2Cl)c1 ZINC000217576303 JH In-Stock Unstable CHRNA4 25 42 CCNC(=O)c1ccc(N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)c(NC(=O)c2cccnc2Cl)c1 ZINC000217576303 JH In-Stock Unstable G2YM83_BOTF4 79 43 O=C1O[C@]2(CCCN(C(=O)CCc3c(F)cccc3Cl)C2)c2ccccc21 ZINC000217576353 GI For-Sale Unstable NPY5R 31 42 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NCCc1ccccc1 ZINC000217576367 GG In-Stock Unstable TGM2 25 40 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NCCc1ccccc1 ZINC000217576367 GG In-Stock Unstable F13A1 21 40 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NCCc1ccccc1 ZINC000217576367 GG In-Stock Unstable CCR8 95 49 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NCCc1ccccc1 ZINC000217576367 GG In-Stock Unstable SFRP1 134 38 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NCCc1ccccc1 ZINC000217576367 GG In-Stock Unstable WNT3 89 38 C[C@@H](Cc1ccncc1Br)C(=O)O ZINC000217576373 BE For-Sale Unstable TBXAS1 15 48 Cc1cccc(N2CCN(C(=O)NCC3CCCC3)CC2)c1C ZINC000217576381 DG On-Demand Unstable HTR1A 26 42 Cc1cccc(N2CCN(C(=O)NCC3CCCC3)CC2)c1C ZINC000217576381 DG On-Demand Unstable DRD2 23 44 Cc1cccc(N2CCN(C(=O)NCC3CCCC3)CC2)c1C ZINC000217576381 DG On-Demand Unstable HTR2A 24 43 Cc1cccc(N2CCN(C(=O)NCC3CCCC3)CC2)c1C ZINC000217576381 DG On-Demand Unstable HTR2C 30 46 Cc1cccc(N2CCN(C(=O)NCC3CCCC3)CC2)c1C ZINC000217576381 DG On-Demand Unstable ABCB1 0 42 CNC[C@H](O)c1ccc(S(C)(=O)=O)c(F)c1 ZINC000217576387 BC For-Sale Unstable ADRB1 15 50 CNC[C@H](O)c1ccc(S(C)(=O)=O)c(F)c1 ZINC000217576387 BC For-Sale Unstable ADRB3 19 50 O=C(O)/C=C\c1cccc(CNC(=O)CC(F)(F)F)c1 ZINC000217576437 CE For-Sale Unstable PTGER2 19 42 O=C1O[C@@]2(CCCN(C(=O)CCc3ccc(Cl)cc3Cl)C2)c2ccccc21 ZINC000217576444 HJ For-Sale Unstable NPY5R 26 43 C[C@H](Cc1ccncc1Br)C(=O)O ZINC000217576454 BE For-Sale Unstable TBXAS1 15 48 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCC3)cc2C(=O)O)cc1 ZINC000217576470 HG In-Stock Unstable BMP1 59 38 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCC3)cc2C(=O)O)cc1 ZINC000217576470 HG In-Stock Unstable MMP13 68 42 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCC3)cc2C(=O)O)cc1 ZINC000217576470 HG In-Stock Unstable ADAM17 35 40 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCC3)cc2C(=O)O)cc1 ZINC000217576470 HG In-Stock Unstable MMP2 41 43 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCC3)cc2C(=O)O)cc1 ZINC000217576470 HG In-Stock Unstable MMP3 57 40 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCC3)cc2C(=O)O)cc1 ZINC000217576470 HG In-Stock Unstable MMP8 34 40 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCC3)cc2C(=O)O)cc1 ZINC000217576470 HG In-Stock Unstable MMP9 51 40 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCC3)cc2C(=O)O)cc1 ZINC000217576470 HG In-Stock Unstable MMP12 23 40 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCC3)cc2C(=O)O)cc1 ZINC000217576470 HG In-Stock Unstable PTGDR 32 40 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCC3)cc2C(=O)O)cc1 ZINC000217576470 HG In-Stock Unstable MMP7 47 39 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCC3)cc2C(=O)O)cc1 ZINC000217576470 HG In-Stock Unstable CA9 19 41 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCC3)cc2C(=O)O)cc1 ZINC000217576470 HG In-Stock Unstable MMP1 62 40 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCC3)cc2C(=O)O)cc1 ZINC000217576470 HG In-Stock Unstable CCR8 63 43 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCC3)cc2C(=O)O)cc1 ZINC000217576470 HG In-Stock Unstable TYRO3 15 41 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCC3)cc2C(=O)O)cc1 ZINC000217576470 HG In-Stock Unstable SFRP1 75 32 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCC3)cc2C(=O)O)cc1 ZINC000217576470 HG In-Stock Unstable AKR1C2 45 35 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCC3)cc2C(=O)O)cc1 ZINC000217576470 HG In-Stock Unstable WNT3 54 31 CNC[C@@H](O)c1ccc(S(C)(=O)=O)c(F)c1 ZINC000217576472 BC For-Sale Unstable ADRB1 15 50 CNC[C@@H](O)c1ccc(S(C)(=O)=O)c(F)c1 ZINC000217576472 BC For-Sale Unstable ADRB3 19 50 O=C1O[C@]2(CCCN(C(=O)CCc3ccc(Cl)cc3Cl)C2)c2ccccc21 ZINC000217576510 HJ For-Sale Unstable NPY5R 26 43 CC[S@@](=O)CCNc1nc(Cl)nc(NC)n1 ZINC000217576540 CC For-Sale Unstable AT1 0 40 CC[S@@](=O)CCNc1nc(Cl)nc(NC)n1 ZINC000217576540 CC For-Sale Unstable PPX1 0 46 Cn1c(SC(F)(F)C(=O)O)nc2ccccc21 ZINC000217576547 CE In-Stock Unstable PTGDR2 17 42 CS(=O)(=O)c1ccc([C@H](N)CCO)c(F)c1 ZINC000217576567 BC For-Sale Unstable PTGS2 22 43 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCC3)cc2C(=O)O)cc1OC ZINC000217576585 IG In-Stock Unstable FKBP1A 41 42 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCC3)cc2C(=O)O)cc1OC ZINC000217576585 IG In-Stock Unstable ADRA1D 21 42 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCC3)cc2C(=O)O)cc1OC ZINC000217576585 IG In-Stock Unstable ADRA1A 15 42 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCC3)cc2C(=O)O)cc1OC ZINC000217576585 IG In-Stock Unstable ADRA1B 26 42 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCC3)cc2C(=O)O)cc1OC ZINC000217576585 IG In-Stock Unstable ABCC8 19 43 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCC3)cc2C(=O)O)cc1OC ZINC000217576585 IG In-Stock Unstable PTGDR 26 40 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCC3)cc2C(=O)O)cc1OC ZINC000217576585 IG In-Stock Unstable IAP 0 40 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCC3)cc2C(=O)O)cc1OC ZINC000217576585 IG In-Stock Unstable CCR8 48 40 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCC3)cc2C(=O)O)cc1OC ZINC000217576585 IG In-Stock Unstable SFRP1 57 33 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCC3)cc2C(=O)O)cc1OC ZINC000217576585 IG In-Stock Unstable WNT3 45 31 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCC3)cc2C(=O)O)cc1OC ZINC000217576585 IG In-Stock Unstable SCMU_MYCTU 0 43 COc1ccc([N+](=O)[O-])cc1NC(=O)NCC1CCCC1 ZINC000217576606 CF On-Demand Unstable CACNA1C 40 37 COc1ccc([N+](=O)[O-])cc1NC(=O)NCC1CCCC1 ZINC000217576606 CF On-Demand Unstable CACNA1D 68 37 COc1ccc([N+](=O)[O-])cc1NC(=O)NCC1CCCC1 ZINC000217576606 CF On-Demand Unstable KCNMA1 23 53 COc1ccc([N+](=O)[O-])cc1NC(=O)NCC1CCCC1 ZINC000217576606 CF On-Demand Unstable SLC27A4 43 33 COc1ccc([N+](=O)[O-])cc1NC(=O)NCC1CCCC1 ZINC000217576606 CF On-Demand Unstable WDR5 32 41 O=C1O[C@@]2(CCCN(C(=O)CCc3c(Cl)cccc3Cl)C2)c2ccccc21 ZINC000217576610 HJ For-Sale Unstable NPY5R 33 46 CC[S@](=O)CCNc1nc(Cl)nc(NC)n1 ZINC000217576620 CC For-Sale Unstable AT1 0 40 CC[S@](=O)CCNc1nc(Cl)nc(NC)n1 ZINC000217576620 CC For-Sale Unstable PPX1 0 46 CS(=O)(=O)c1ccc([C@@H](N)CCO)c(F)c1 ZINC000217576645 BC For-Sale Unstable PTGS2 22 43 Cc1cc(N[C@@H](C)c2ccccc2)nc(NCCc2ccc(Cl)cc2)n1 ZINC000217576668 FK For-Sale Unstable HTR7 24 60 Cc1cc(N[C@@H](C)c2ccccc2)nc(NCCc2ccc(Cl)cc2)n1 ZINC000217576668 FK For-Sale Unstable METAP1 40 37 Cc1cc(N[C@@H](C)c2ccccc2)nc(NCCc2ccc(Cl)cc2)n1 ZINC000217576668 FK For-Sale Unstable PLK1 15 40 Cc1cc(N[C@@H](C)c2ccccc2)nc(NCCc2ccc(Cl)cc2)n1 ZINC000217576668 FK For-Sale Unstable MRGPRX1 35 41 O=C1O[C@]2(CCCN(C(=O)CCc3c(Cl)cccc3Cl)C2)c2ccccc21 ZINC000217576676 HJ For-Sale Unstable NPY5R 33 46 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NCc1ccco1 ZINC000217576695 FF In-Stock Unstable CCR8 40 31 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NCc1ccco1 ZINC000217576695 FF In-Stock Unstable WNT3 42 32 CCN(C(=O)NCC1CCCC1)c1cccc(C)c1 ZINC000217576717 CH For-Sale Unstable AMY2 45 32 CC[S@@](=O)CCNc1nc(N)nc(Cl)n1 ZINC000217576727 BC For-Sale Unstable PPX1 0 41 O=C(NC[C@](O)(c1ccccc1)C1CC1)c1cc2ccccc2[nH]1 ZINC000217576731 DG In-Stock Unstable CCKAR 33 54 O=C(NC[C@](O)(c1ccccc1)C1CC1)c1cc2ccccc2[nH]1 ZINC000217576731 DG In-Stock Unstable CYP51A1 22 44 O=C(NC[C@](O)(c1ccccc1)C1CC1)c1cc2ccccc2[nH]1 ZINC000217576731 DG In-Stock Unstable PYGL 86 41 O=C(NC[C@](O)(c1ccccc1)C1CC1)c1cc2ccccc2[nH]1 ZINC000217576731 DG In-Stock Unstable PLD1 41 45 O=C(NC[C@](O)(c1ccccc1)C1CC1)c1cc2ccccc2[nH]1 ZINC000217576731 DG In-Stock Unstable PLD2 36 48 O=C(NC[C@](O)(c1ccccc1)C1CC1)c1cc2ccccc2[nH]1 ZINC000217576731 DG In-Stock Unstable AKR1C3 18 43 COc1cccc(Br)c1C(=O)CN ZINC000217576746 BD For-Sale Unstable ALS 49 44 O=C1O[C@@]2(CCCN(C(=O)CCc3ccc(Cl)c(Cl)c3)C2)c2ccccc21 ZINC000217576794 HJ For-Sale Unstable NPY5R 28 44 O=C(NC[C@@](O)(c1ccccc1)C1CC1)c1cc2ccccc2[nH]1 ZINC000217576802 DG In-Stock Unstable CCKAR 33 54 O=C(NC[C@@](O)(c1ccccc1)C1CC1)c1cc2ccccc2[nH]1 ZINC000217576802 DG In-Stock Unstable CYP51A1 22 44 O=C(NC[C@@](O)(c1ccccc1)C1CC1)c1cc2ccccc2[nH]1 ZINC000217576802 DG In-Stock Unstable PYGL 86 41 O=C(NC[C@@](O)(c1ccccc1)C1CC1)c1cc2ccccc2[nH]1 ZINC000217576802 DG In-Stock Unstable PLD1 41 45 O=C(NC[C@@](O)(c1ccccc1)C1CC1)c1cc2ccccc2[nH]1 ZINC000217576802 DG In-Stock Unstable PLD2 36 48 O=C(NC[C@@](O)(c1ccccc1)C1CC1)c1cc2ccccc2[nH]1 ZINC000217576802 DG In-Stock Unstable AKR1C3 18 43 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NC[C@@H]1CCCO1 ZINC000217576803 FE In-Stock Unstable CCR8 41 31 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NC[C@@H]1CCCO1 ZINC000217576803 FE In-Stock Unstable SFRP1 89 32 CC[S@](=O)CCNc1nc(N)nc(Cl)n1 ZINC000217576807 BC For-Sale Unstable PPX1 0 41 CN1CCC[C@@H](CNC[C@@H](O)c2ccc(F)cc2)C1 ZINC000217576834 CD For-Sale Unstable SLC6A4 15 42 CN1CCC[C@@H](CNC[C@@H](O)c2ccc(F)cc2)C1 ZINC000217576834 CD For-Sale Unstable SLC6A3 33 42 CN1CCC[C@@H](CNC[C@@H](O)c2ccc(F)cc2)C1 ZINC000217576834 CD For-Sale Unstable CCR3 46 33 Cc1ccnc(NC(=O)NCC2CCCC2)c1 ZINC000217576835 BF On-Demand Unstable TYK2 44 34 O=C1O[C@]2(CCCN(C(=O)CCc3ccc(Cl)c(Cl)c3)C2)c2ccccc21 ZINC000217576867 HJ For-Sale Unstable NPY5R 28 44 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NC[C@H]1CCCO1 ZINC000217576880 FE In-Stock Unstable TNK2 43 38 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NC[C@H]1CCCO1 ZINC000217576880 FE In-Stock Unstable CCR8 76 38 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NC[C@H]1CCCO1 ZINC000217576880 FE In-Stock Unstable SFRP1 109 33 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1NC[C@H]1CCCO1 ZINC000217576880 FE In-Stock Unstable WNT3 77 33 CN1CCC[C@H](CNC[C@@H](O)c2ccc(F)cc2)C1 ZINC000217576924 CD For-Sale Unstable SLC6A4 15 42 CN1CCC[C@H](CNC[C@@H](O)c2ccc(F)cc2)C1 ZINC000217576924 CD For-Sale Unstable SLC6A3 33 42 CN1CCC[C@H](CNC[C@@H](O)c2ccc(F)cc2)C1 ZINC000217576924 CD For-Sale Unstable CCR3 46 33 CS(=O)(=O)c1ccc([C@H](O)CCN)c(F)c1 ZINC000217576928 BC For-Sale Unstable PTGS2 23 43 CC[C@@H](C)c1ccccc1NC(=O)NCC1CCCC1 ZINC000217576939 CJ For-Sale Unstable KCNQ2 44 36 CC[C@@H](C)c1ccccc1NC(=O)NCC1CCCC1 ZINC000217576939 CJ For-Sale Unstable NMBR 17 41 CC[C@@H](C)c1ccccc1NC(=O)NCC1CCCC1 ZINC000217576939 CJ For-Sale Unstable SOAT1 24 42 CC[C@@H](C)c1ccccc1NC(=O)NCC1CCCC1 ZINC000217576939 CJ For-Sale Unstable ACAT 0 45 CC[C@@H](C)c1ccccc1NC(=O)NCC1CCCC1 ZINC000217576939 CJ For-Sale Unstable AO-ACHE 0 44 CCOC(=O)C(F)(F)Sc1nc2ccccc2n1C ZINC000217576959 CF In-Stock Unstable PTGDR2 15 41 O=C(C[C@@H]1NC(=O)N(CCc2ccccc2)C1=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217576965 ID In-Stock Unstable CHRNA4 30 50 CCOc1ccccc1CCC(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217576973 GH For-Sale Unstable NPY5R 27 43 CCOc1ccccc1CCC(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217576973 GH For-Sale Unstable HCN1 43 32 CCOc1ccccc1CCC(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217576973 GH For-Sale Unstable HCN4 40 31 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1N1CCCC1 ZINC000217576983 EE In-Stock Unstable SLC6A9 15 42 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1N1CCCC1 ZINC000217576983 EE In-Stock Unstable LIPG 46 34 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1N1CCCC1 ZINC000217576983 EE In-Stock Unstable SFRP1 112 38 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1N1CCCC1 ZINC000217576983 EE In-Stock Unstable WNT3 86 39 CS(=O)(=O)c1ccc([C@@H](O)CCN)c(F)c1 ZINC000217577000 BC For-Sale Unstable PTGS2 23 43 NC(=O)[C@@H](Nc1cncc(B(O)O)c1)c1ccccc1 ZINC000217577008 CB For-Sale Unstable CSNK1G1 20 46 CC[C@H](C)c1ccccc1NC(=O)NCC1CCCC1 ZINC000217577021 CJ For-Sale Unstable KCNQ2 44 36 CC[C@H](C)c1ccccc1NC(=O)NCC1CCCC1 ZINC000217577021 CJ For-Sale Unstable NMBR 17 41 CC[C@H](C)c1ccccc1NC(=O)NCC1CCCC1 ZINC000217577021 CJ For-Sale Unstable SOAT1 24 42 CC[C@H](C)c1ccccc1NC(=O)NCC1CCCC1 ZINC000217577021 CJ For-Sale Unstable ACAT 0 45 CC[C@H](C)c1ccccc1NC(=O)NCC1CCCC1 ZINC000217577021 CJ For-Sale Unstable AO-ACHE 0 44 CN1CCC[C@@H](CNC[C@@H](O)c2cccc(Br)c2)C1 ZINC000217577029 EE For-Sale Unstable PHES 0 46 CCOc1ccccc1CCC(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217577062 GH For-Sale Unstable NPY5R 27 43 CCOc1ccccc1CCC(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217577062 GH For-Sale Unstable HCN1 43 32 CCOc1ccccc1CCC(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217577062 GH For-Sale Unstable HCN4 40 31 O=C(O)C(F)(F)S(=O)(=O)c1nc2ccccc2s1 ZINC000217577080 CD In-Stock Anodyne CA2 34 45 O=C(O)C(F)(F)S(=O)(=O)c1nc2ccccc2s1 ZINC000217577080 CD In-Stock Anodyne CA1 30 58 O=C(O)C(F)(F)S(=O)(=O)c1nc2ccccc2s1 ZINC000217577080 CD In-Stock Anodyne CA4 38 45 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1N1CCCCC1 ZINC000217577084 FF In-Stock Unstable SLC6A9 15 44 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1N1CCCCC1 ZINC000217577084 FF In-Stock Unstable EPHX2 29 41 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1N1CCCCC1 ZINC000217577084 FF In-Stock Unstable LIPG 43 33 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1N1CCCCC1 ZINC000217577084 FF In-Stock Unstable SFRP1 111 38 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1N1CCCCC1 ZINC000217577084 FF In-Stock Unstable WNT3 86 39 NC(=O)[C@H](Nc1cncc(B(O)O)c1)c1ccccc1 ZINC000217577094 CB For-Sale Unstable CSNK1G1 20 46 CN1CCC[C@H](CNC[C@@H](O)c2cccc(Br)c2)C1 ZINC000217577110 EE For-Sale Unstable PHES 0 46 O=C1O[C@@]2(CCCN(C(=O)CCc3ccccc3F)C2)c2ccccc21 ZINC000217577160 FG For-Sale Unstable NPY5R 26 43 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1N1CCOCC1 ZINC000217577185 FD In-Stock Unstable SLC6A9 21 46 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1N1CCOCC1 ZINC000217577185 FD In-Stock Unstable SFRP1 99 41 O=C(O)c1cc(S(=O)(=O)NC2CCCC2)ccc1N1CCOCC1 ZINC000217577185 FD In-Stock Unstable WNT3 80 41 O=C1O[C@]2(CCCN(C(=O)CCc3ccccc3F)C2)c2ccccc21 ZINC000217577234 FG For-Sale Unstable NPY5R 26 43 C[C@H](N)[C@H](O)c1ccc(S(C)(=O)=O)cc1F ZINC000217577266 BC For-Sale Unstable PTGS2 25 44 CCOCCCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217577287 FE In-Stock Unstable CCR8 42 36 CCOCCCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217577287 FE In-Stock Unstable SFRP1 83 32 CCOCCCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217577287 FE In-Stock Unstable WNT3 51 32 C[C@@H](N)[C@H](O)c1ccc(S(C)(=O)=O)cc1F ZINC000217577330 BC For-Sale Unstable PTGS2 25 44 COc1ccc2ccccc2c1CCC(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217577342 HI For-Sale Unstable NPY5R 24 43 O=C(O)C(F)(F)[S@@](=O)c1nc2ccccc2s1 ZINC000217577366 CE In-Stock Anodyne BCL2L1 40 33 CN1CCC[C@@H](CNC[C@@H](O)c2ccc(Cl)cc2)C1 ZINC000217577391 CE For-Sale Unstable SLC6A1 62 42 C[C@H]1CN(C/C=C\CN)C[C@@H](C)O1 ZINC000217577396 AC For-Sale Unstable ERG2 17 40 C[C@H]1CN(C/C=C\CN)C[C@@H](C)O1 ZINC000217577396 AC For-Sale Unstable ZM.86993 0 40 C[C@H]1CN(C/C=C\CN)C[C@@H](C)O1 ZINC000217577396 AC For-Sale Unstable Q2TU57_MAIZE 19 40 CC(C)OCCCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217577403 GF In-Stock Unstable CCR8 74 38 CC(C)OCCCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217577403 GF In-Stock Unstable SFRP1 100 33 CC(C)OCCCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217577403 GF In-Stock Unstable WNT3 67 33 CC[S@@](=O)CCNc1ccnc(N)n1 ZINC000217577411 BC For-Sale Unstable HRH4 30 63 COc1ccc2ccccc2c1CCC(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217577419 HI For-Sale Unstable NPY5R 24 43 C[C@H](N)[C@@H](O)c1ccc(S(C)(=O)=O)cc1F ZINC000217577423 BC For-Sale Unstable PTGS2 25 44 O=C(O)C(F)(F)[S@](=O)c1nc2ccccc2s1 ZINC000217577440 CE In-Stock Anodyne BCL2L1 40 33 COc1ccc(N2CCC[C@H](C(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)C2)nn1 ZINC000217577461 HD In-Stock Unstable CHRNA4 25 41 CN1CCC[C@H](CNC[C@@H](O)c2ccc(Cl)cc2)C1 ZINC000217577477 CE For-Sale Unstable SLC6A1 62 42 Cc1noc(C)c1CC(=O)NC[C@@](O)(c1ccccc1)C1CC1 ZINC000217577481 DE In-Stock Unstable P2RX7 22 54 CC(C)(CO)NC(=O)NCC1CCCC1 ZINC000217577493 BD For-Sale Unstable CACNA1I 41 32 CC[S@](=O)CCNc1ccnc(N)n1 ZINC000217577495 BC For-Sale Unstable HRH4 30 63 C[C@@H](N)[C@@H](O)c1ccc(S(C)(=O)=O)cc1F ZINC000217577502 BC For-Sale Unstable PTGS2 25 44 CCCCCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217577510 FG In-Stock Unstable TBXA2R 15 45 CCCCCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217577510 FG In-Stock Unstable CCR8 79 38 CCCCCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217577510 FG In-Stock Unstable SFRP1 92 34 CCCCCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217577510 FG In-Stock Unstable WNT3 76 34 COc1ccc(N2CCC[C@@H](C(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)C2)nn1 ZINC000217577546 HD In-Stock Unstable CHRNA4 25 41 Cc1noc(C)c1CC(=O)NC[C@](O)(c1ccccc1)C1CC1 ZINC000217577565 DE In-Stock Unstable P2RX7 22 54 CC(C)CCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217577638 FG In-Stock Unstable CCR8 76 38 CC(C)CCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217577638 FG In-Stock Unstable SFRP1 92 34 CC(C)CCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217577638 FG In-Stock Unstable WNT3 76 35 O=C(NCc1ccc(CO)cc1)NCC1CCCC1 ZINC000217577721 CE On-Demand Unstable TPSAB1 17 42 O=C(NCc1ccc(CO)cc1)NCC1CCCC1 ZINC000217577721 CE On-Demand Unstable PROC 43 32 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217577744 FG In-Stock Unstable CCR8 58 35 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217577744 FG In-Stock Unstable SFRP1 67 33 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217577744 FG In-Stock Unstable WNT3 56 33 O=C(O)/C=C\c1cccc(CNC(=O)[C@@H]2CCC(=O)N2)c1 ZINC000217577795 CC For-Sale Unstable PLG 60 35 O=C(O)/C=C\c1cccc(CNC(=O)[C@@H]2CCC(=O)N2)c1 ZINC000217577795 CC For-Sale Unstable KLKB1 37 41 O=C(O)/C=C\c1cccc(CNC(=O)[C@@H]2CCC(=O)N2)c1 ZINC000217577795 CC For-Sale Unstable TRYP_PIG 49 34 O=C(O)/C=C\c1cccc(CNC(=O)[C@@H]2CCC(=O)N2)c1 ZINC000217577795 CC For-Sale Unstable HDAC2 17 41 O=C(O)/C=C\c1cccc(CNC(=O)[C@@H]2CCC(=O)N2)c1 ZINC000217577795 CC For-Sale Unstable LNPEP 48 36 O=C(O)/C=C\c1cccc(CNC(=O)[C@@H]2CCC(=O)N2)c1 ZINC000217577795 CC For-Sale Unstable PROC 32 41 O=S(=O)(c1ccc(N2CCOCC2)c(NCc2ccccc2Cl)c1)N1CCCCC1 ZINC000217577815 JH On-Demand Unstable LPL 40 37 O=S(=O)(c1ccc(N2CCOCC2)c(NCc2ccccc2Cl)c1)N1CCCCC1 ZINC000217577815 JH On-Demand Unstable KCNQ2 30 42 O=S(=O)(c1ccc(N2CCOCC2)c(NCc2ccccc2Cl)c1)N1CCCCC1 ZINC000217577815 JH On-Demand Unstable NAMPT 22 40 CCC[C@H](C)Nc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217577834 FG In-Stock Unstable CCR8 58 35 CCC[C@H](C)Nc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217577834 FG In-Stock Unstable SFRP1 67 33 CCC[C@H](C)Nc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217577834 FG In-Stock Unstable WNT3 56 33 O=C(O)/C=C\c1cccc(CNC(=O)[C@H]2CCC(=O)N2)c1 ZINC000217577891 CC For-Sale Unstable PLG 60 35 O=C(O)/C=C\c1cccc(CNC(=O)[C@H]2CCC(=O)N2)c1 ZINC000217577891 CC For-Sale Unstable KLKB1 37 41 O=C(O)/C=C\c1cccc(CNC(=O)[C@H]2CCC(=O)N2)c1 ZINC000217577891 CC For-Sale Unstable TRYP_PIG 49 34 O=C(O)/C=C\c1cccc(CNC(=O)[C@H]2CCC(=O)N2)c1 ZINC000217577891 CC For-Sale Unstable HDAC2 17 41 O=C(O)/C=C\c1cccc(CNC(=O)[C@H]2CCC(=O)N2)c1 ZINC000217577891 CC For-Sale Unstable LNPEP 48 36 O=C(O)/C=C\c1cccc(CNC(=O)[C@H]2CCC(=O)N2)c1 ZINC000217577891 CC For-Sale Unstable PROC 32 41 CN1CCC[C@@H](CNC[C@@H](O)c2ccccc2Cl)C1 ZINC000217577950 CE For-Sale Unstable OPRL1 42 39 O=C(NCc1ccc(Br)cc1)NCC1CCCC1 ZINC000217577952 DG On-Demand Unstable TPSAB1 17 41 O=C(NCc1ccc(Br)cc1)NCC1CCCC1 ZINC000217577952 DG On-Demand Unstable PROC 42 32 COC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217577958 FE In-Stock Unstable SFRP1 55 32 COC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217577958 FE In-Stock Unstable WNT3 40 31 CCC(CC)C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217577976 CF For-Sale Unstable PTGER2 25 42 CCC(CC)C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217577976 CF For-Sale Unstable ANPEP 21 40 CCC(CC)C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217577976 CF For-Sale Unstable HDAC1 15 41 CCC(CC)C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217577976 CF For-Sale Unstable AMP1_PLAFQ 46 37 CCC(CC)C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217577976 CF For-Sale Unstable AKR1C3 41 42 CCC(CC)C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217577976 CF For-Sale Unstable PDS 52 37 O=C1CCCNC[C@H]1C(=O)OCc1ccccc1 ZINC000217577989 BD For-Sale Unstable SLC12A5 46 39 CCNc1nccc(NCC[S@@](=O)CC)n1 ZINC000217578001 BD For-Sale Unstable HRH4 0 43 CC(C)CNC(=O)[C@@H](C)NCC1(c2ccccc2)CCCC1 ZINC000217578022 DG On-Demand Unstable KCNA3 46 38 COC[C@H](C)Nc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217578043 FE In-Stock Unstable SFRP1 55 32 COC[C@H](C)Nc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217578043 FE In-Stock Unstable WNT3 40 31 CN1CCC[C@H](CNC[C@@H](O)c2ccccc2Cl)C1 ZINC000217578044 CE For-Sale Unstable OPRL1 42 39 O=C(Cc1c[nH]c2ccccc12)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217578055 EF In-Stock Unstable CHRNA4 30 47 O=C(Cc1c[nH]c2ccccc12)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217578055 EF In-Stock Unstable CCKBR 43 36 CCNc1nccc(NCC[S@](=O)CC)n1 ZINC000217578060 BD For-Sale Unstable HRH4 0 43 Cc1ncsc1C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217578064 DE For-Sale Unstable PTGER2 0 40 O=C1CCCNC[C@@H]1C(=O)OCc1ccccc1 ZINC000217578075 BD For-Sale Unstable SLC12A5 46 39 CS(=O)(=O)c1ccc(CCC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217578099 HF For-Sale Unstable NPY5R 21 42 CC(C)CNC(=O)[C@H](C)NCC1(c2ccccc2)CCCC1 ZINC000217578115 DG On-Demand Unstable KCNA3 46 38 CN1CCC[C@@H](CNC[C@@H](O)c2cc(Cl)ccc2Cl)C1 ZINC000217578143 DF For-Sale Unstable CACNA1I 42 35 CCCNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217578151 EF In-Stock Unstable CCR8 81 41 CCCNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217578151 EF In-Stock Unstable SFRP1 95 35 CCCNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217578151 EF In-Stock Unstable WNT3 78 35 COc1ccc(Cl)cc1CN[C@@H]1C[C@@H]2C[C@@H]1[C@@H]1CCC[C@@H]21 ZINC000217578159 DI For-Sale Unstable TACR1 23 41 CC[S@@](=O)CCNc1ccnc(NC)n1 ZINC000217578164 BC For-Sale Unstable HRH4 15 40 CS(=O)(=O)c1ccc(CCC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217578175 HF For-Sale Unstable NPY5R 21 42 CCCCC(=O)N[C@@H](C)c1ccc(/C=C\C(=O)O)cc1 ZINC000217578202 CG For-Sale Unstable ACACA 42 43 CCCCC(=O)N[C@@H](C)c1ccc(/C=C\C(=O)O)cc1 ZINC000217578202 CG For-Sale Unstable AKR1C3 25 40 CCCCC(=O)N[C@@H](C)c1ccc(/C=C\C(=O)O)cc1 ZINC000217578202 CG For-Sale Unstable NOD1 75 37 CCCCC(=O)N[C@@H](C)c1ccc(/C=C\C(=O)O)cc1 ZINC000217578202 CG For-Sale Unstable ACER2 0 44 CC(C)(C)OC(=O)NCC1CCN(CC#N)CC1 ZINC000217578231 CD On-Demand Unstable PAPA1_CARPA 44 39 CC(C)(C)OC(=O)NCC1CCN(CC#N)CC1 ZINC000217578231 CD On-Demand Unstable CACNA1I 59 39 CN1CCC[C@H](CNC[C@@H](O)c2cc(Cl)ccc2Cl)C1 ZINC000217578237 DF For-Sale Unstable CACNA1I 42 35 COc1ccc(Cl)cc1CN[C@H]1C[C@@H]2C[C@@H]1[C@@H]1CCC[C@@H]21 ZINC000217578249 DI For-Sale Unstable TACR1 23 41 CC[S@](=O)CCNc1ccnc(NC)n1 ZINC000217578252 BC For-Sale Unstable HRH4 15 40 CC(C)Nc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217578264 EF In-Stock Unstable CCR8 62 41 CC(C)Nc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217578264 EF In-Stock Unstable SFRP1 90 34 CC(C)Nc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217578264 EF In-Stock Unstable WNT3 73 34 CCCCC(=O)N[C@H](C)c1ccc(/C=C\C(=O)O)cc1 ZINC000217578284 CG For-Sale Unstable ACACA 42 43 CCCCC(=O)N[C@H](C)c1ccc(/C=C\C(=O)O)cc1 ZINC000217578284 CG For-Sale Unstable AKR1C3 25 40 CCCCC(=O)N[C@H](C)c1ccc(/C=C\C(=O)O)cc1 ZINC000217578284 CG For-Sale Unstable NOD1 75 37 CCCCC(=O)N[C@H](C)c1ccc(/C=C\C(=O)O)cc1 ZINC000217578284 CG For-Sale Unstable ACER2 0 44 Cc1cc(C(=O)CN)cc(Br)c1O ZINC000217578296 BD For-Sale Unstable SLC22A12 55 33 Cc1ccc(CCNC(=O)NCC2CCCC2)cc1 ZINC000217578308 CG On-Demand Unstable MMP2 64 41 Cc1ccc(CCNC(=O)NCC2CCCC2)cc1 ZINC000217578308 CG On-Demand Unstable GPBAR1 22 44 COc1ccc(Cl)cc1CN[C@@H]1C[C@H]2C[C@@H]1[C@@H]1CCC[C@@H]21 ZINC000217578320 DI For-Sale Unstable TACR1 23 41 Cn1cccc1C(=O)NCc1ccc(/C=C\C(=O)O)cc1 ZINC000217578360 CE For-Sale Unstable HDAC6 25 65 CCCCNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217578368 FG In-Stock Unstable CCR8 79 40 CCCCNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217578368 FG In-Stock Unstable SFRP1 92 34 CCCCNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217578368 FG In-Stock Unstable WNT3 76 34 O=C(NCCc1ccc(Br)cc1)NCC1CCCC1 ZINC000217578403 EG On-Demand Unstable MMP2 46 33 COc1ccc(Cl)cc1CN[C@H]1C[C@H]2C[C@@H]1[C@@H]1CCC[C@@H]21 ZINC000217578406 DI For-Sale Unstable TACR1 23 41 N#Cc1ccc(OC[C@@H](O)CN2CCC[C@@H](O)C2)cc1 ZINC000217578452 CC In-Stock Unstable ABCB1 37 40 N#Cc1ccc(OC[C@@H](O)CN2CCC[C@@H](O)C2)cc1 ZINC000217578452 CC In-Stock Unstable MEN1 45 39 CC(C)CNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217578477 FG In-Stock Unstable MTNN 70 32 CC(C)CNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217578477 FG In-Stock Unstable CCR8 79 41 CC(C)CNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217578477 FG In-Stock Unstable SFRP1 95 35 CC(C)CNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217578477 FG In-Stock Unstable WNT3 78 36 COc1ccc(C(=O)NC[C@@](O)(c2ccccc2)C2CC2)cc1F ZINC000217578484 EF In-Stock Unstable CPT1A 44 30 COc1ccc(C(=O)NC[C@@](O)(c2ccccc2)C2CC2)cc1F ZINC000217578484 EF In-Stock Unstable ACKR3 64 33 O=C(CCc1nc(-c2ccncc2)no1)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217578499 GD In-Stock Unstable CHRNA4 28 48 Cc1ccc(NC(=O)NCC2CCCC2)cn1 ZINC000217578512 BF On-Demand Unstable EPHX2 16 59 Cc1ccc(NC(=O)NCC2CCCC2)cn1 ZINC000217578512 BF On-Demand Unstable NAMPT 27 43 N#Cc1ccc(OC[C@H](O)CN2CCC[C@@H](O)C2)cc1 ZINC000217578539 CC In-Stock Unstable ABCB1 37 40 N#Cc1ccc(OC[C@H](O)CN2CCC[C@@H](O)C2)cc1 ZINC000217578539 CC In-Stock Unstable MEN1 45 39 COc1ccc(C(=O)NC[C@](O)(c2ccccc2)C2CC2)cc1F ZINC000217578552 EF In-Stock Unstable CPT1A 44 30 COc1ccc(C(=O)NC[C@](O)(c2ccccc2)C2CC2)cc1F ZINC000217578552 EF In-Stock Unstable ACKR3 64 33 CC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217578590 FG In-Stock Unstable CCR8 65 38 CC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217578590 FG In-Stock Unstable SFRP1 79 34 CC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217578590 FG In-Stock Unstable WNT3 58 34 Cc1ccc(NC(=O)NCC2CCCC2)nc1 ZINC000217578624 BF On-Demand Unstable GYRB 0 40 Cc1ccc(NC(=O)NCC2CCCC2)nc1 ZINC000217578624 BF On-Demand Unstable GCK 34 48 Cc1ccc(NC(=O)NCC2CCCC2)nc1 ZINC000217578624 BF On-Demand Unstable LUCI_LUCLA 23 44 O=C1O[C@@]2(CCCN(C(=O)CCc3ccc(C(F)(F)F)cc3)C2)c2ccccc21 ZINC000217578639 HI For-Sale Unstable NPY5R 22 47 O[C@@H]1CCCN(C[C@@H](O)COCc2ccccc2)C1 ZINC000217578660 CD In-Stock Unstable ABCB1 46 43 CC[C@H](C)Nc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217578662 FG In-Stock Unstable CCR8 65 38 CC[C@H](C)Nc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217578662 FG In-Stock Unstable SFRP1 79 34 CC[C@H](C)Nc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217578662 FG In-Stock Unstable WNT3 58 34 CCCCCCOC(=O)CCC(C)([N+](=O)[O-])[N+](=O)[O-] ZINC000217578665 CE For-Sale Unstable PLA2G4B 50 37 O=C1NCCN1C(=O)NC[C@](O)(c1ccccc1)C1CC1 ZINC000217578668 CD In-Stock Unstable CYP2J2 43 30 O=C(c1cc2ccccc2[nH]1)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217578707 EF In-Stock Unstable HRH4 21 47 O=C(c1cc2ccccc2[nH]1)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217578707 EF In-Stock Unstable CHRNA4 29 47 O=C(c1cc2ccccc2[nH]1)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217578707 EF In-Stock Unstable AKR1C3 19 44 O=C1O[C@]2(CCCN(C(=O)CCc3ccc(C(F)(F)F)cc3)C2)c2ccccc21 ZINC000217578712 HI For-Sale Unstable NPY5R 22 47 N#Cc1c(-n2cnnn2)sc2c1CCCC2 ZINC000217578725 BD In-Stock Unstable MAPK10 0 40 CCCCCCCOC(=O)CCC(C)([N+](=O)[O-])[N+](=O)[O-] ZINC000217578744 CF For-Sale Unstable PLA2G4B 50 37 CN1CCC[C@@H](CNC[C@@H](O)c2cccc(F)c2)C1 ZINC000217578746 CD For-Sale Unstable SLC6A2 15 42 CN1CCC[C@@H](CNC[C@@H](O)c2cccc(F)c2)C1 ZINC000217578746 CD For-Sale Unstable CHRNA10 45 42 O=C1NCCN1C(=O)NC[C@@](O)(c1ccccc1)C1CC1 ZINC000217578752 CD In-Stock Unstable CYP2J2 43 30 CC(C)(C)Nc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217578766 FG In-Stock Unstable CCR8 78 42 CC(C)(C)Nc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217578766 FG In-Stock Unstable SFRP1 107 36 CC(C)(C)Nc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217578766 FG In-Stock Unstable WNT3 83 37 CN1CCC[C@H](CNC[C@@H](O)c2cccc(F)c2)C1 ZINC000217578815 CD For-Sale Unstable SLC6A2 15 42 CN1CCC[C@H](CNC[C@@H](O)c2cccc(F)c2)C1 ZINC000217578815 CD For-Sale Unstable CHRNA10 45 42 O=C(O)/C=C\c1cccc(CNC(=O)Cn2cncn2)c1 ZINC000217578816 CC For-Sale Unstable HIS3 43 38 COc1ccc(CCC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c(OC)c1OC ZINC000217578828 IG For-Sale Unstable NPY5R 19 42 Cc1ccc(-c2c(C)nnn2-c2ccc([N+](=O)[O-])cc2)cc1 ZINC000217578832 CG In-Stock Unstable NPY5R 22 45 C=CCNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217578870 EF In-Stock Unstable F13A1 30 41 C=CCNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217578870 EF In-Stock Unstable CCR8 42 32 C=CCNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217578870 EF In-Stock Unstable SFRP1 92 35 C=CCNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217578870 EF In-Stock Unstable WNT3 73 35 C[C@H]1CCCC[C@]1(N)C(=O)O[C@H](C)c1ccccc1 ZINC000217578899 CG For-Sale Unstable AMY2 44 30 Cc1ccc(C(=O)NCc2cccc(/C=C\C(=O)O)c2)s1 ZINC000217578903 DG For-Sale Unstable PTGER2 27 42 Cc1ccc(C(=O)NCc2cccc(/C=C\C(=O)O)c2)s1 ZINC000217578903 DG For-Sale Unstable HDAC1 16 43 Cc1ccc(C(=O)NCc2cccc(/C=C\C(=O)O)c2)s1 ZINC000217578903 DG For-Sale Unstable HDAC6 16 43 COc1ccc(CCC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c(OC)c1OC ZINC000217578908 IG For-Sale Unstable NPY5R 19 42 O=C(NCC1CCCC1)Nc1ccc(Cl)cn1 ZINC000217578935 CG On-Demand Unstable GCK 23 44 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NC1CC1 ZINC000217578950 EF In-Stock Unstable CCR8 48 42 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NC1CC1 ZINC000217578950 EF In-Stock Unstable SFRP1 93 34 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NC1CC1 ZINC000217578950 EF In-Stock Unstable WNT3 75 34 CC(C)c1ccc(C(=O)O)c(Br)n1 ZINC000217578966 BF For-Sale Unstable PRS 44 32 C[C@H]1CCCC[C@@]1(N)C(=O)O[C@H](C)c1ccccc1 ZINC000217578985 CG For-Sale Unstable AMY2 44 30 Cc1ccsc1C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217578988 DG For-Sale Unstable PTGER2 0 41 O=C(CCc1c[nH]c2ccccc12)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217578994 FF In-Stock Unstable TACR2 20 50 O=C(CCc1c[nH]c2ccccc12)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217578994 FF In-Stock Unstable CHRNA4 38 48 O=C(CCc1c[nH]c2ccccc12)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217578994 FF In-Stock Unstable MC5R 34 45 O=C(CCc1c[nH]c2ccccc12)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217578994 FF In-Stock Unstable CCKBR 42 34 COc1cc(OC)c(CCC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c(OC)c1 ZINC000217579023 IG For-Sale Unstable NPY5R 25 45 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NC1CCCC1 ZINC000217579029 FG In-Stock Unstable CCR8 54 43 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NC1CCCC1 ZINC000217579029 FG In-Stock Unstable SFRP1 96 35 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NC1CCCC1 ZINC000217579029 FG In-Stock Unstable WNT3 76 35 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NC1CCCC1 ZINC000217579029 FG In-Stock Unstable BRD4 0 40 O=C(CCc1ccc(C(F)(F)F)cc1)NC[C@](O)(c1ccccc1)C1CC1 ZINC000217579063 GI In-Stock Unstable MCHR1 15 43 O=C(CCc1ccc(C(F)(F)F)cc1)NC[C@](O)(c1ccccc1)C1CC1 ZINC000217579063 GI In-Stock Unstable MLYCD 19 43 O=C(CCc1ccc(C(F)(F)F)cc1)NC[C@](O)(c1ccccc1)C1CC1 ZINC000217579063 GI In-Stock Unstable LUXR 23 40 O=C(CCc1ccc(C(F)(F)F)cc1)NC[C@](O)(c1ccccc1)C1CC1 ZINC000217579063 GI In-Stock Unstable TRAR 19 47 O=C(NCC1CCCC1)Nc1cc(Cl)ccn1 ZINC000217579068 CG For-Sale Unstable EPHX2 15 61 O=C(NCC1CCCC1)Nc1cc(Cl)ccn1 ZINC000217579068 CG For-Sale Unstable TYK2 66 38 O=C(NCC1CCCC1)Nc1cc(Cl)ccn1 ZINC000217579068 CG For-Sale Unstable CACNA1I 52 36 CC(C)(C)CC(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217579081 CF For-Sale Unstable PTGER2 22 45 CC(C)(C)CC(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217579081 CF For-Sale Unstable HDAC8 44 38 CC(C)(C)CC(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217579081 CF For-Sale Unstable HDAC1 26 41 CC(C)(C)CC(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217579081 CF For-Sale Unstable HDAC2 15 41 COc1cc(OC)c(CCC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c(OC)c1 ZINC000217579106 IG For-Sale Unstable NPY5R 25 45 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NC1CCCCC1 ZINC000217579109 GH In-Stock Unstable CCR8 54 43 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NC1CCCCC1 ZINC000217579109 GH In-Stock Unstable SFRP1 96 35 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NC1CCCCC1 ZINC000217579109 GH In-Stock Unstable WNT3 76 35 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NC1CCCCC1 ZINC000217579109 GH In-Stock Unstable BRD4 0 40 O=C(CCc1ccc(C(F)(F)F)cc1)NC[C@@](O)(c1ccccc1)C1CC1 ZINC000217579146 GI In-Stock Unstable MLYCD 19 43 O=C(CCc1ccc(C(F)(F)F)cc1)NC[C@@](O)(c1ccccc1)C1CC1 ZINC000217579146 GI In-Stock Unstable LUXR 23 40 O=C(CCc1ccc(C(F)(F)F)cc1)NC[C@@](O)(c1ccccc1)C1CC1 ZINC000217579146 GI In-Stock Unstable TRAR 19 47 C[C@H](NC(=O)c1ccco1)c1ccc(/C=C\C(=O)O)cc1 ZINC000217579151 CF For-Sale Unstable ADAM12 24 41 O=C(NCC1CCCC1)Nc1cc(Br)ccn1 ZINC000217579174 CG For-Sale Unstable TYK2 45 34 Cc1ccnc2ccc(C(=O)N3CCC[C@]4(C3)OC(=O)c3ccccc34)cc12 ZINC000217579205 FH For-Sale Unstable NPY5R 29 41 Cc1ccc(C(=O)O)cc1N[C@@H]1C[C@@H]2CC[C@@]1(C)C2(C)C ZINC000217579208 CI For-Sale Unstable RARA 40 31 Cc1ccc(C(=O)O)cc1N[C@@H]1C[C@@H]2CC[C@@]1(C)C2(C)C ZINC000217579208 CI For-Sale Unstable RARG 42 35 Cc1ccc(C(=O)O)cc1N[C@@H]1C[C@@H]2CC[C@@]1(C)C2(C)C ZINC000217579208 CI For-Sale Unstable RXRG 48 35 Cc1ccc(C(=O)O)cc1N[C@@H]1C[C@@H]2CC[C@@]1(C)C2(C)C ZINC000217579208 CI For-Sale Unstable RXRB 47 35 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NCCC1=CCCCC1 ZINC000217579223 HI In-Stock Unstable SFRP1 53 32 C[C@@H](NC(=O)c1ccco1)c1ccc(/C=C\C(=O)O)cc1 ZINC000217579236 CF For-Sale Unstable ADAM12 24 41 O=C(NCCCCc1ccccc1)NCC1CCCC1 ZINC000217579274 CG On-Demand Unstable FKBP1A 44 50 O=C(NCCCCc1ccccc1)NCC1CCCC1 ZINC000217579274 CG On-Demand Unstable GRIN2B 34 43 O=C(NCCCCc1ccccc1)NCC1CCCC1 ZINC000217579274 CG On-Demand Unstable SIGMAR1 24 43 O=C(NCCCCc1ccccc1)NCC1CCCC1 ZINC000217579274 CG On-Demand Unstable CCR3 25 46 O=C(NCCCCc1ccccc1)NCC1CCCC1 ZINC000217579274 CG On-Demand Unstable SCN2A 18 41 O=C(NCCCCc1ccccc1)NCC1CCCC1 ZINC000217579274 CG On-Demand Unstable S1PR3 16 40 O=C(NCCCCc1ccccc1)NCC1CCCC1 ZINC000217579274 CG On-Demand Unstable PREP 56 38 O=C(NCCCCc1ccccc1)NCC1CCCC1 ZINC000217579274 CG On-Demand Unstable MTNR1A 31 42 O=C(NCCCCc1ccccc1)NCC1CCCC1 ZINC000217579274 CG On-Demand Unstable MTNR1B 42 42 O=C(NCCCCc1ccccc1)NCC1CCCC1 ZINC000217579274 CG On-Demand Unstable MMP2 43 41 O=C(NCCCCc1ccccc1)NCC1CCCC1 ZINC000217579274 CG On-Demand Unstable MMP3 23 44 O=C(NCCCCc1ccccc1)NCC1CCCC1 ZINC000217579274 CG On-Demand Unstable FAAH 58 45 O=C(NCCCCc1ccccc1)NCC1CCCC1 ZINC000217579274 CG On-Demand Unstable SCN5A 0 42 O=C(NCCCCc1ccccc1)NCC1CCCC1 ZINC000217579274 CG On-Demand Unstable CES1 56 36 O=C(NCCCCc1ccccc1)NCC1CCCC1 ZINC000217579274 CG On-Demand Unstable EPHX2 23 53 O=C(NCCCCc1ccccc1)NCC1CCCC1 ZINC000217579274 CG On-Demand Unstable AMP1_PLAFQ 28 40 O=C(NCCCCc1ccccc1)NCC1CCCC1 ZINC000217579274 CG On-Demand Unstable CRTM 42 38 Cc1ccnc2ccc(C(=O)N3CCC[C@@]4(C3)OC(=O)c3ccccc34)cc12 ZINC000217579289 FH For-Sale Unstable NPY5R 29 41 Cc1ccc(C(=O)O)cc1N[C@H]1C[C@@H]2CC[C@@]1(C)C2(C)C ZINC000217579291 CI For-Sale Unstable RARA 40 31 Cc1ccc(C(=O)O)cc1N[C@H]1C[C@@H]2CC[C@@]1(C)C2(C)C ZINC000217579291 CI For-Sale Unstable RARG 42 35 Cc1ccc(C(=O)O)cc1N[C@H]1C[C@@H]2CC[C@@]1(C)C2(C)C ZINC000217579291 CI For-Sale Unstable RXRG 48 35 Cc1ccc(C(=O)O)cc1N[C@H]1C[C@@H]2CC[C@@]1(C)C2(C)C ZINC000217579291 CI For-Sale Unstable RXRB 47 35 CN(C)c1ccc(C(=O)O)c(Br)c1 ZINC000217579306 BE For-Sale Unstable SLC16A3 0 48 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NCCO ZINC000217579341 ED In-Stock Unstable CCR8 76 42 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NCCO ZINC000217579341 ED In-Stock Unstable SFRP1 97 36 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NCCO ZINC000217579341 ED In-Stock Unstable WNT3 77 35 Cc1ccc(C(=O)O)cc1N[C@@H]1C[C@H]2CC[C@@]1(C)C2(C)C ZINC000217579371 CI For-Sale Unstable RARA 40 31 Cc1ccc(C(=O)O)cc1N[C@@H]1C[C@H]2CC[C@@]1(C)C2(C)C ZINC000217579371 CI For-Sale Unstable RARG 42 35 Cc1ccc(C(=O)O)cc1N[C@@H]1C[C@H]2CC[C@@]1(C)C2(C)C ZINC000217579371 CI For-Sale Unstable RXRG 48 35 Cc1ccc(C(=O)O)cc1N[C@@H]1C[C@H]2CC[C@@]1(C)C2(C)C ZINC000217579371 CI For-Sale Unstable RXRB 47 35 O=C1O[C@@]2(CCCN(C(=O)CCc3ccc(F)c(Cl)c3)C2)c2ccccc21 ZINC000217579393 GI For-Sale Unstable NPY5R 24 42 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NCCCO ZINC000217579440 FD In-Stock Unstable CCR8 69 40 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NCCCO ZINC000217579440 FD In-Stock Unstable SFRP1 92 35 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NCCCO ZINC000217579440 FD In-Stock Unstable WNT3 73 34 Cc1ccc(C(=O)O)cc1N[C@H]1C[C@H]2CC[C@@]1(C)C2(C)C ZINC000217579446 CI For-Sale Unstable RARA 40 31 Cc1ccc(C(=O)O)cc1N[C@H]1C[C@H]2CC[C@@]1(C)C2(C)C ZINC000217579446 CI For-Sale Unstable RARG 42 35 Cc1ccc(C(=O)O)cc1N[C@H]1C[C@H]2CC[C@@]1(C)C2(C)C ZINC000217579446 CI For-Sale Unstable RXRG 48 35 Cc1ccc(C(=O)O)cc1N[C@H]1C[C@H]2CC[C@@]1(C)C2(C)C ZINC000217579446 CI For-Sale Unstable RXRB 47 35 O=C1O[C@]2(CCCN(C(=O)CCc3ccc(F)c(Cl)c3)C2)c2ccccc21 ZINC000217579469 GI For-Sale Unstable NPY5R 24 42 CN1CCC[C@@H](CNC[C@@H](O)c2ccc3c(c2)OCO3)C1 ZINC000217579496 CD For-Sale Unstable NOS2 45 34 COCCNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217579544 FE In-Stock Unstable CCR8 93 41 COCCNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217579544 FE In-Stock Unstable SFRP1 113 34 COCCNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217579544 FE In-Stock Unstable WNT3 80 34 CN1CCC[C@H](CNC[C@@H](O)c2ccc3c(c2)OCO3)C1 ZINC000217579565 CD For-Sale Unstable NOS2 45 34 O=C(c1cccc2[nH]ccc12)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217579579 EF In-Stock Unstable CHRNA4 30 48 COC(=O)Nc1ccc(S(=O)(=O)NC[C@@](O)(c2ccccc2)C2CC2)cc1 ZINC000217579623 GE In-Stock Unstable NPY2R 31 48 COC(=O)Nc1ccc(S(=O)(=O)NC[C@@](O)(c2ccccc2)C2CC2)cc1 ZINC000217579623 GE In-Stock Unstable MMP2 15 41 OCc1cc2n(n1)CCN(C1CCN(CCc3ccccc3)CC1)C2 ZINC000217579645 ED In-Stock Unstable L3MBTL3 40 37 COCCCNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217579652 FE In-Stock Unstable CCR8 43 34 COCCCNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217579652 FE In-Stock Unstable SFRP1 83 33 COCCCNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217579652 FE In-Stock Unstable WNT3 50 31 O=C(c1ccc2[nH]ccc2c1)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217579682 EF In-Stock Unstable CHRNA4 30 51 C[C@@H](NC(=O)[C@@H]1CC[C@@H](CNC(=O)[C@@H]2Cc3ccccc3CN2)CC1)c1ccccc1 ZINC000217579698 HH In-Stock Unstable F11 46 38 COC(=O)Nc1ccc(S(=O)(=O)NC[C@](O)(c2ccccc2)C2CC2)cc1 ZINC000217579701 GE In-Stock Unstable NPY2R 31 48 COC(=O)Nc1ccc(S(=O)(=O)NC[C@](O)(c2ccccc2)C2CC2)cc1 ZINC000217579701 GE In-Stock Unstable MMP2 15 41 CCOC(=O)CN1CC(Br)=C(Br)C1=O ZINC000217579714 ED In-Stock Unstable PIN4 0 40 Cc1cccc(NS(=O)(=O)c2cc(NC(=O)c3cc4ccccc4nc3C)ccc2C)c1 ZINC000217579757 IK On-Demand Unstable PLA2G7 15 42 Cc1cccc(NS(=O)(=O)c2cc(NC(=O)c3cc4ccccc4nc3C)ccc2C)c1 ZINC000217579757 IK On-Demand Unstable KCNK3 86 43 Cc1cccc(NS(=O)(=O)c2cc(NC(=O)c3cc4ccccc4nc3C)ccc2C)c1 ZINC000217579757 IK On-Demand Unstable KCNK9 72 43 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NCc1ccccc1 ZINC000217579768 GH In-Stock Unstable TGM2 22 43 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NCc1ccccc1 ZINC000217579768 GH In-Stock Unstable F13A1 25 43 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NCc1ccccc1 ZINC000217579768 GH In-Stock Unstable CCR8 82 45 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NCc1ccccc1 ZINC000217579768 GH In-Stock Unstable SFRP1 108 39 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NCc1ccccc1 ZINC000217579768 GH In-Stock Unstable WNT3 84 38 Nc1cc(Br)cc(CCC(=O)O)c1 ZINC000217579777 BE For-Sale Unstable THRB 21 50 Nc1cc(Br)cc(CCC(=O)O)c1 ZINC000217579777 BE For-Sale Unstable FFAR1 50 43 C[C@H](NC(=O)[C@@H]1CC[C@@H](CNC(=O)[C@@H]2Cc3ccccc3CN2)CC1)c1ccccc1 ZINC000217579783 HH In-Stock Unstable F11 46 38 O=C1C(Br)=C(Br)CN1c1ccccc1 ZINC000217579805 DG In-Stock Unstable CMA1 15 40 O=C1C(Br)=C(Br)CN1c1ccccc1 ZINC000217579805 DG In-Stock Unstable CTSG 27 40 C[C@@H](Nc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O)c1ccccc1 ZINC000217579866 HI In-Stock Unstable CCR8 82 41 C[C@@H](Nc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O)c1ccccc1 ZINC000217579866 HI In-Stock Unstable SFRP1 123 35 C[C@@H](Nc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O)c1ccccc1 ZINC000217579866 HI In-Stock Unstable WNT3 85 35 C[C@@H](NC(=O)c1cc(-c2ccco2)nn1-c1ccccc1)c1ccc(S(N)(=O)=O)cc1 ZINC000217579868 IG On-Demand Unstable CA2 29 40 C[C@@H](NC(=O)c1cc(-c2ccco2)nn1-c1ccccc1)c1ccc(S(N)(=O)=O)cc1 ZINC000217579868 IG On-Demand Unstable CARM1 15 41 Nc1ccc(Br)cc1CCC(=O)O ZINC000217579887 BE For-Sale Unstable FFAR1 23 40 CN1CCC[C@@H](CNC[C@@H](O)COc2ccccc2)C1 ZINC000217579923 CD For-Sale Unstable ADRB2 68 53 CN1CCC[C@@H](CNC[C@@H](O)COc2ccccc2)C1 ZINC000217579923 CD For-Sale Unstable ADRB1 90 46 CN1CCC[C@@H](CNC[C@@H](O)COc2ccccc2)C1 ZINC000217579923 CD For-Sale Unstable ADRB3 72 46 CN1CCC[C@@H](CNC[C@@H](O)COc2ccccc2)C1 ZINC000217579923 CD For-Sale Unstable CASR 17 43 CN1CCC[C@@H](CNC[C@@H](O)COc2ccccc2)C1 ZINC000217579923 CD For-Sale Unstable CYP2D6 0 40 CN1CCC[C@@H](CNC[C@@H](O)COc2ccccc2)C1 ZINC000217579923 CD For-Sale Unstable ABCB1 42 45 CN1CCC[C@@H](CNC[C@@H](O)COc2ccccc2)C1 ZINC000217579923 CD For-Sale Unstable CHRNA10 70 45 CC(C)(C)OC(=O)N1CCN(C(=O)NCC2CCCC2)CC1 ZINC000217579924 DE On-Demand Unstable CACNA1I 50 34 C[C@H](NC(=O)c1cc(-c2ccco2)nn1-c1ccccc1)c1ccc(S(N)(=O)=O)cc1 ZINC000217579957 IG On-Demand Unstable CA2 29 40 C[C@H](NC(=O)c1cc(-c2ccco2)nn1-c1ccccc1)c1ccc(S(N)(=O)=O)cc1 ZINC000217579957 IG On-Demand Unstable CARM1 15 41 C[C@H](Nc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O)c1ccccc1 ZINC000217579974 HI In-Stock Unstable CCR8 82 41 C[C@H](Nc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O)c1ccccc1 ZINC000217579974 HI In-Stock Unstable SFRP1 123 35 C[C@H](Nc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O)c1ccccc1 ZINC000217579974 HI In-Stock Unstable WNT3 85 35 CN1CCC[C@H](CNC[C@@H](O)COc2ccccc2)C1 ZINC000217580015 CD For-Sale Unstable ADRB2 68 53 CN1CCC[C@H](CNC[C@@H](O)COc2ccccc2)C1 ZINC000217580015 CD For-Sale Unstable ADRB1 90 46 CN1CCC[C@H](CNC[C@@H](O)COc2ccccc2)C1 ZINC000217580015 CD For-Sale Unstable ADRB3 72 46 CN1CCC[C@H](CNC[C@@H](O)COc2ccccc2)C1 ZINC000217580015 CD For-Sale Unstable CYP2D6 0 40 CN1CCC[C@H](CNC[C@@H](O)COc2ccccc2)C1 ZINC000217580015 CD For-Sale Unstable ABCB1 42 45 CN1CCC[C@H](CNC[C@@H](O)COc2ccccc2)C1 ZINC000217580015 CD For-Sale Unstable CHRNA10 70 45 CC1(C)[C@H]2CC[C@@]1(CS(=O)(=O)NC[C@@](O)(c1ccccc1)C1CC1)C(=O)C2 ZINC000217580056 GF In-Stock Unstable CA5B 31 53 CC1(C)[C@H]2CC[C@@]1(CS(=O)(=O)NC[C@@](O)(c1ccccc1)C1CC1)C(=O)C2 ZINC000217580056 GF In-Stock Unstable CA5A 33 53 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NCCc1ccccc1 ZINC000217580077 HH In-Stock Unstable EPHX2 20 40 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NCCc1ccccc1 ZINC000217580077 HH In-Stock Unstable CCR8 93 49 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NCCc1ccccc1 ZINC000217580077 HH In-Stock Unstable SFRP1 131 38 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NCCc1ccccc1 ZINC000217580077 HH In-Stock Unstable WNT3 88 37 Cc1cc(CCC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)ccc1Cl ZINC000217580123 GI In-Stock Unstable NPY5R 24 43 CN1CCC[C@@H](CNC[C@@H](O)COc2ccccc2F)C1 ZINC000217580130 CD For-Sale Unstable ADRB2 37 47 CN1CCC[C@@H](CNC[C@@H](O)COc2ccccc2F)C1 ZINC000217580130 CD For-Sale Unstable ADRB1 63 37 CN1CCC[C@@H](CNC[C@@H](O)COc2ccccc2F)C1 ZINC000217580130 CD For-Sale Unstable HTR1A 0 54 CN1CCC[C@@H](CNC[C@@H](O)COc2ccccc2F)C1 ZINC000217580130 CD For-Sale Unstable ADRB3 27 49 CN1CCC[C@@H](CNC[C@@H](O)COc2ccccc2F)C1 ZINC000217580130 CD For-Sale Unstable ABCB1 43 38 CN1CCC[C@@H](CNC[C@@H](O)COc2ccccc2F)C1 ZINC000217580130 CD For-Sale Unstable CHRNA10 27 48 O=C(Nc1ccc(S(=O)(=O)O)cc1)NC1CCCC1 ZINC000217580152 CD For-Sale Unstable CA2 26 76 O=C(Nc1ccc(S(=O)(=O)O)cc1)NC1CCCC1 ZINC000217580152 CD For-Sale Unstable CA1 33 65 O=C(Nc1ccc(S(=O)(=O)O)cc1)NC1CCCC1 ZINC000217580152 CD For-Sale Unstable EPHX2 85 62 O=C(Nc1ccc(S(=O)(=O)O)cc1)NC1CCCC1 ZINC000217580152 CD For-Sale Unstable CA12 36 76 O=C(Nc1ccc(S(=O)(=O)O)cc1)NC1CCCC1 ZINC000217580152 CD For-Sale Unstable CA9 33 76 O=C(Nc1ccc(S(=O)(=O)O)cc1)NC1CCCC1 ZINC000217580152 CD For-Sale Unstable F13A1 65 39 O=C(Nc1ccc(S(=O)(=O)O)cc1)NC1CCCC1 ZINC000217580152 CD For-Sale Unstable NCE103 34 65 O=C(Nc1ccc(S(=O)(=O)O)cc1)NC1CCCC1 ZINC000217580152 CD For-Sale Unstable MTCA1 50 76 O=C(Nc1ccc(S(=O)(=O)O)cc1)NC1CCCC1 ZINC000217580152 CD For-Sale Unstable P96878_MYCTU 61 76 O=C(Nc1ccc(S(=O)(=O)O)cc1)NC1CCCC1 ZINC000217580152 CD For-Sale Unstable NAMPT 40 38 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCC3)cc2C(=O)O)cc1 ZINC000217580188 IH In-Stock Unstable BMP1 53 39 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCC3)cc2C(=O)O)cc1 ZINC000217580188 IH In-Stock Unstable MMP13 65 44 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCC3)cc2C(=O)O)cc1 ZINC000217580188 IH In-Stock Unstable ADAM17 32 41 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCC3)cc2C(=O)O)cc1 ZINC000217580188 IH In-Stock Unstable MMP2 42 44 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCC3)cc2C(=O)O)cc1 ZINC000217580188 IH In-Stock Unstable MMP3 56 42 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCC3)cc2C(=O)O)cc1 ZINC000217580188 IH In-Stock Unstable MMP9 48 41 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCC3)cc2C(=O)O)cc1 ZINC000217580188 IH In-Stock Unstable PTGDR 29 40 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCC3)cc2C(=O)O)cc1 ZINC000217580188 IH In-Stock Unstable MMP7 47 40 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCC3)cc2C(=O)O)cc1 ZINC000217580188 IH In-Stock Unstable CA9 19 40 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCC3)cc2C(=O)O)cc1 ZINC000217580188 IH In-Stock Unstable MMP1 57 41 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCC3)cc2C(=O)O)cc1 ZINC000217580188 IH In-Stock Unstable CCR8 56 43 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCC3)cc2C(=O)O)cc1 ZINC000217580188 IH In-Stock Unstable TYRO3 15 41 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCC3)cc2C(=O)O)cc1 ZINC000217580188 IH In-Stock Unstable SFRP1 65 31 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCC3)cc2C(=O)O)cc1 ZINC000217580188 IH In-Stock Unstable AKR1C2 44 35 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCC3)cc2C(=O)O)cc1 ZINC000217580188 IH In-Stock Unstable WNT3 51 31 O=C(Cn1cnc2c(cnn2-c2ccccc2)c1=O)N1CCN(Cc2cccc(Cl)c2)CC1 ZINC000217580189 JF On-Demand Unstable HTR1A 15 45 O=C(Cn1cnc2c(cnn2-c2ccccc2)c1=O)N1CCN(Cc2cccc(Cl)c2)CC1 ZINC000217580189 JF On-Demand Unstable HTR7 17 45 O=C(Cn1cnc2c(cnn2-c2ccccc2)c1=O)N1CCN(Cc2cccc(Cl)c2)CC1 ZINC000217580189 JF On-Demand Unstable FAAH 25 48 Nc1ccc(Br)c(CCC(=O)O)c1 ZINC000217580201 BE For-Sale Unstable THRB 20 46 Nc1ccc(Br)c(CCC(=O)O)c1 ZINC000217580201 BE For-Sale Unstable FFAR1 30 41 CN1CCC[C@H](CNC[C@@H](O)COc2ccccc2F)C1 ZINC000217580212 CD For-Sale Unstable ADRB2 37 47 CN1CCC[C@H](CNC[C@@H](O)COc2ccccc2F)C1 ZINC000217580212 CD For-Sale Unstable ADRB1 63 37 CN1CCC[C@H](CNC[C@@H](O)COc2ccccc2F)C1 ZINC000217580212 CD For-Sale Unstable HTR1A 0 54 CN1CCC[C@H](CNC[C@@H](O)COc2ccccc2F)C1 ZINC000217580212 CD For-Sale Unstable ADRB3 27 49 CN1CCC[C@H](CNC[C@@H](O)COc2ccccc2F)C1 ZINC000217580212 CD For-Sale Unstable CYP2D26 0 40 CN1CCC[C@H](CNC[C@@H](O)COc2ccccc2F)C1 ZINC000217580212 CD For-Sale Unstable ABCB1 43 38 CN1CCC[C@H](CNC[C@@H](O)COc2ccccc2F)C1 ZINC000217580212 CD For-Sale Unstable CHRNA10 27 48 CC(C)CCCCCCNC[C@@H](O)c1ccccc1 ZINC000217580224 CH For-Sale Unstable ADRB2 51 48 CC(C)CCCCCCNC[C@@H](O)c1ccccc1 ZINC000217580224 CH For-Sale Unstable ADRB1 59 43 CC(C)CCCCCCNC[C@@H](O)c1ccccc1 ZINC000217580224 CH For-Sale Unstable ADRB3 72 46 CC(C)CCCCCCNC[C@@H](O)c1ccccc1 ZINC000217580224 CH For-Sale Unstable AOC3 16 46 Cc1cc(CCC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)ccc1Cl ZINC000217580228 GI In-Stock Unstable NPY5R 23 43 CC(C)CCC(=O)NCc1ccc(/C=C\C(=O)O)cc1 ZINC000217580246 CF For-Sale Unstable TPSAB1 17 44 CC(C)(C)OC(=O)N1CCC(N2CC(Br)=C(Br)C2=O)CC1 ZINC000217580252 HG In-Stock Unstable GPR119 35 42 O=C(Nc1cccc(S(=O)(=O)O)c1)NC1CCCC1 ZINC000217580273 CD For-Sale Unstable FAAH 0 41 O=C(Nc1cccc(S(=O)(=O)O)c1)NC1CCCC1 ZINC000217580273 CD For-Sale Unstable EPHX2 83 67 O=C(Nc1cccc(S(=O)(=O)O)c1)NC1CCCC1 ZINC000217580273 CD For-Sale Unstable ST14 41 44 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCC3)cc2C(=O)O)cc1OC ZINC000217580297 JH In-Stock Unstable FKBP1A 41 42 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCC3)cc2C(=O)O)cc1OC ZINC000217580297 JH In-Stock Unstable ADRA1D 19 41 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCC3)cc2C(=O)O)cc1OC ZINC000217580297 JH In-Stock Unstable ADRA1B 23 41 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCC3)cc2C(=O)O)cc1OC ZINC000217580297 JH In-Stock Unstable ABCC8 19 44 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCC3)cc2C(=O)O)cc1OC ZINC000217580297 JH In-Stock Unstable PTGDR 24 40 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCC3)cc2C(=O)O)cc1OC ZINC000217580297 JH In-Stock Unstable CCR8 42 40 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCC3)cc2C(=O)O)cc1OC ZINC000217580297 JH In-Stock Unstable SFRP1 48 32 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCC3)cc2C(=O)O)cc1OC ZINC000217580297 JH In-Stock Unstable WNT3 43 30 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCC3)cc2C(=O)O)cc1OC ZINC000217580297 JH In-Stock Unstable SCMU_MYCTU 0 43 CC(C)CCCCCCNC[C@H](O)c1ccccc1 ZINC000217580304 CH For-Sale Unstable ADRB2 51 48 CC(C)CCCCCCNC[C@H](O)c1ccccc1 ZINC000217580304 CH For-Sale Unstable ADRB1 59 43 CC(C)CCCCCCNC[C@H](O)c1ccccc1 ZINC000217580304 CH For-Sale Unstable ADRB3 72 46 CC(C)CCCCCCNC[C@H](O)c1ccccc1 ZINC000217580304 CH For-Sale Unstable AOC3 16 46 COc1c2ccc(C(=O)N3CCC[C@]4(C3)OC(=O)c3ccccc34)cc2nn1C ZINC000217580336 GF For-Sale Unstable NPY5R 25 43 NC/C=C\CN1C(=O)c2ccccc2S1(=O)=O ZINC000217580341 CC For-Sale Unstable ELANE 0 57 NC/C=C\CN1C(=O)c2ccccc2S1(=O)=O ZINC000217580341 CC For-Sale Unstable CA12 0 70 Cc1ccc(Br)cc1N[C@H]1C[C@H](C)CC[C@H]1C(C)C ZINC000217580369 DK For-Sale Unstable TRPM8 15 42 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NCc1ccco1 ZINC000217580371 GG In-Stock Unstable CCR8 70 39 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NCc1ccco1 ZINC000217580371 GG In-Stock Unstable SFRP1 116 35 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NCc1ccco1 ZINC000217580371 GG In-Stock Unstable WNT3 81 35 O=C(Nc1cccc2c(O)cccc12)NC1CCCC1 ZINC000217580380 CH For-Sale Unstable TRPV1 30 46 O=C(Nc1cccc2c(O)cccc12)NC1CCCC1 ZINC000217580380 CH For-Sale Unstable EPHX2 45 54 COc1c2ccc(C(=O)N3CCC[C@@]4(C3)OC(=O)c3ccccc34)cc2nn1C ZINC000217580402 GF For-Sale Unstable NPY5R 25 43 O=C1C(Br)=C(Br)CN1CCc1ccccc1 ZINC000217580450 EG In-Stock Unstable SIGMAR1 21 40 O=C1C(Br)=C(Br)CN1CCc1ccccc1 ZINC000217580450 EG In-Stock Unstable ALDH1A1 33 41 Cc1ccc(Br)cc1N[C@H]1C[C@@H](C)CC[C@H]1C(C)C ZINC000217580458 DK For-Sale Unstable TRPM8 15 42 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NC[C@@H]1CCCO1 ZINC000217580477 GF In-Stock Unstable TNK2 42 37 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NC[C@@H]1CCCO1 ZINC000217580477 GF In-Stock Unstable CCR8 71 40 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NC[C@@H]1CCCO1 ZINC000217580477 GF In-Stock Unstable SFRP1 95 33 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NC[C@@H]1CCCO1 ZINC000217580477 GF In-Stock Unstable WNT3 57 33 O=C(Cn1c(COc2ccccc2)nc2ccccc21)Nc1ccc(CN2CCOCC2)cc1 ZINC000217580500 JI On-Demand Unstable LTA4H 38 47 O=C(Cn1c(COc2ccccc2)nc2ccccc21)Nc1ccc(CN2CCOCC2)cc1 ZINC000217580500 JI On-Demand Unstable PDE6D 54 33 O=C(Cn1c(COc2ccccc2)nc2ccccc21)Nc1ccc(CN2CCOCC2)cc1 ZINC000217580500 JI On-Demand Unstable FAAH 18 41 O=C(Cn1c(COc2ccccc2)nc2ccccc21)Nc1ccc(CN2CCOCC2)cc1 ZINC000217580500 JI On-Demand Unstable EPHX2 16 46 O=C(Cn1c(COc2ccccc2)nc2ccccc21)Nc1ccc(CN2CCOCC2)cc1 ZINC000217580500 JI On-Demand Unstable MCHR1 24 41 O=C(Cn1c(COc2ccccc2)nc2ccccc21)Nc1ccc(CN2CCOCC2)cc1 ZINC000217580500 JI On-Demand Unstable IMDH_CRYPV 40 46 O=C(Cn1c(COc2ccccc2)nc2ccccc21)Nc1ccc(CN2CCOCC2)cc1 ZINC000217580500 JI On-Demand Unstable NOD1 25 40 CCOc1ccc(C)cc1[C@@H](C)NC(=O)NC1CCCC1 ZINC000217580501 CH For-Sale Unstable EPHX2 30 40 Cn1nc2cc(Br)ccc2c1C(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217580513 IH For-Sale Unstable NPY5R 27 44 Cc1nnsc1C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217580516 DD For-Sale Unstable HDAC8 34 40 Cc1nnsc1C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217580516 DD For-Sale Unstable HDAC6 25 40 COc1ccc2cc(C(=O)NC[C@@](C)(O)c3cccs3)[nH]c2c1 ZINC000217580527 EF In-Stock Unstable ROCK1 16 43 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NC[C@H]1CCCO1 ZINC000217580547 GF In-Stock Unstable CCR8 66 40 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NC[C@H]1CCCO1 ZINC000217580547 GF In-Stock Unstable SFRP1 77 32 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1NC[C@H]1CCCO1 ZINC000217580547 GF In-Stock Unstable WNT3 57 33 C=C(CC)COc1ccc2ccccc2c1/C=C\C(=O)O ZINC000217580558 CI For-Sale Unstable AKR1C3 22 43 CCOc1ccc(C)cc1[C@H](C)NC(=O)NC1CCCC1 ZINC000217580582 CH For-Sale Unstable EPHX2 30 40 Cn1nc2cc(Br)ccc2c1C(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217580594 IH For-Sale Unstable NPY5R 27 44 Cc1nn(-c2ccccc2)c(C)c1CNC(=O)Cn1cnc2c(cnn2-c2ccccc2)c1=O ZINC000217580604 JF On-Demand Unstable P2RX7 24 52 COc1ccc2cc(C(=O)NC[C@](C)(O)c3cccs3)[nH]c2c1 ZINC000217580613 EF In-Stock Unstable ROCK1 16 43 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1N1CCCC1 ZINC000217580627 FF In-Stock Unstable SLC6A9 15 44 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1N1CCCC1 ZINC000217580627 FF In-Stock Unstable EPHX2 29 41 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1N1CCCC1 ZINC000217580627 FF In-Stock Unstable LIPG 43 33 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1N1CCCC1 ZINC000217580627 FF In-Stock Unstable SFRP1 111 38 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1N1CCCC1 ZINC000217580627 FF In-Stock Unstable WNT3 86 39 CC[C@@H](NC(=O)NC1CCCC1)c1ccc2c(c1)CCCC2 ZINC000217580685 DI For-Sale Unstable EPHX2 22 42 O=C(O)/C=C\c1cccc(CNC(=O)Cc2cccs2)c1 ZINC000217580686 DF For-Sale Unstable CA5B 38 51 O=C(O)/C=C\c1cccc(CNC(=O)Cc2cccs2)c1 ZINC000217580686 DF For-Sale Unstable CA5A 38 51 O=C(O)/C=C\c1cccc(CNC(=O)Cc2cccs2)c1 ZINC000217580686 DF For-Sale Unstable HCAR2 0 40 O=C(Cn1ccc2c([N+](=O)[O-])cccc21)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217580697 GE In-Stock Unstable CHRNA4 28 45 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1N1CCCCC1 ZINC000217580710 FF In-Stock Unstable SLC6A9 15 44 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1N1CCCCC1 ZINC000217580710 FF In-Stock Unstable EPHX2 29 41 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1N1CCCCC1 ZINC000217580710 FF In-Stock Unstable LIPG 43 33 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1N1CCCCC1 ZINC000217580710 FF In-Stock Unstable SFRP1 111 38 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1N1CCCCC1 ZINC000217580710 FF In-Stock Unstable WNT3 86 39 CN1CCC[C@@H](CNC[C@@H](O)COc2ccc(Br)cc2)C1 ZINC000217580724 FE For-Sale Unstable ADRB2 48 40 CN1CCC[C@@H](CNC[C@@H](O)COc2ccc(Br)cc2)C1 ZINC000217580724 FE For-Sale Unstable ADRB1 59 44 CN1CCC[C@@H](CNC[C@@H](O)COc2ccc(Br)cc2)C1 ZINC000217580724 FE For-Sale Unstable ADRB3 40 41 O=C(c1ccccc1)[C@H]1[C@H]2C(=O)N(c3ccc(Cl)c(Cl)c3)C(=O)[C@H]2[C@H]2CCCN12 ZINC000217580757 IH In-Stock Unstable BCL2A1 50 34 CC[C@H](NC(=O)NC1CCCC1)c1ccc2c(c1)CCCC2 ZINC000217580770 DI For-Sale Unstable EPHX2 22 42 O=C(CC[C@@H]1NC(=O)N(CCc2ccccc2)C1=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217580780 ID In-Stock Unstable CHRNA4 31 51 CC(=O)NCC(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217580782 CC For-Sale Unstable PTGER2 23 43 C=C(CC)COc1c(OC)cc(/C=C\C(=O)O)cc1OC ZINC000217580800 CG For-Sale Unstable TNFRSF1A 30 44 C=C(CC)COc1c(OC)cc(/C=C\C(=O)O)cc1OC ZINC000217580800 CG For-Sale Unstable TUBB1 43 38 C=C(CC)COc1c(OC)cc(/C=C\C(=O)O)cc1OC ZINC000217580800 CG For-Sale Unstable NFE2L2 0 42 CN1CCC[C@H](CNC[C@@H](O)COc2ccc(Br)cc2)C1 ZINC000217580802 FE For-Sale Unstable ADRB2 48 40 CN1CCC[C@H](CNC[C@@H](O)COc2ccc(Br)cc2)C1 ZINC000217580802 FE For-Sale Unstable ADRB1 59 44 CN1CCC[C@H](CNC[C@@H](O)COc2ccc(Br)cc2)C1 ZINC000217580802 FE For-Sale Unstable ADRB3 40 41 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1N1CCOCC1 ZINC000217580824 FD In-Stock Unstable SLC6A9 20 45 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1N1CCOCC1 ZINC000217580824 FD In-Stock Unstable SFRP1 99 40 O=C(O)c1cc(S(=O)(=O)NC2CCCCC2)ccc1N1CCOCC1 ZINC000217580824 FD In-Stock Unstable WNT3 79 40 O=S(=O)(NC1CCCCCCC1)c1cccc(CO)c1 ZINC000217580867 CF For-Sale Unstable FAAH 17 48 O=S(=O)(NC1CCCCCCC1)c1cccc(CO)c1 ZINC000217580867 CF For-Sale Unstable SFRP1 88 33 O=S(=O)(NC1CCCCCCC1)c1cccc(CO)c1 ZINC000217580867 CF For-Sale Unstable WNT3 57 34 O=C(NCCCCl)NC1CCCC1 ZINC000217580899 BD For-Sale Unstable EPHX2 27 63 CCOCCCNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217580909 GF In-Stock Unstable CCR8 85 41 CCOCCCNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217580909 GF In-Stock Unstable SFRP1 96 34 CCOCCCNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217580909 GF In-Stock Unstable WNT3 65 34 CN1CCC[C@@H](CNC[C@@H](O)COc2cccc(Br)c2)C1 ZINC000217580945 FE For-Sale Unstable ADRB2 35 41 CN1CCC[C@@H](CNC[C@@H](O)COc2cccc(Br)c2)C1 ZINC000217580945 FE For-Sale Unstable ADRB1 47 41 CN1CCC[C@@H](CNC[C@@H](O)COc2cccc(Br)c2)C1 ZINC000217580945 FE For-Sale Unstable ADRB3 33 42 CN1CCC[C@@H](CNC[C@@H](O)COc2cccc(Br)c2)C1 ZINC000217580945 FE For-Sale Unstable CHRNA10 58 37 Cc1nc(-c2cccs2)ccc1C(=O)NCCCOCC(C)C ZINC000217580948 EH On-Demand Unstable GPR142 40 31 COc1ccc2c(c1)cc(C(=O)N1C[C@@H]3C[C@H](C1)c1cccc(=O)n1C3)n2C ZINC000217580997 GF In-Stock Unstable CHRNA4 27 45 CCCCOC(=O)c1ccccc1NC(=O)NC1CCCC1 ZINC000217581004 DH For-Sale Unstable CNR2 24 43 CCCCOC(=O)c1ccccc1NC(=O)NC1CCCC1 ZINC000217581004 DH For-Sale Unstable AMY2 46 32 CCCCOC(=O)c1ccccc1NC(=O)NC1CCCC1 ZINC000217581004 DH For-Sale Unstable EPHX2 43 46 CCCCOC(=O)c1ccccc1NC(=O)NC1CCCC1 ZINC000217581004 DH For-Sale Unstable NAAA 43 34 CC(C)OCCCNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217581009 GG In-Stock Unstable CCR8 71 37 CC(C)OCCCNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217581009 GG In-Stock Unstable SFRP1 96 33 CC(C)OCCCNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217581009 GG In-Stock Unstable WNT3 67 33 CN1CCC[C@H](CNC[C@@H](O)COc2cccc(Br)c2)C1 ZINC000217581037 FE For-Sale Unstable ADRB2 35 41 CN1CCC[C@H](CNC[C@@H](O)COc2cccc(Br)c2)C1 ZINC000217581037 FE For-Sale Unstable ADRB1 47 41 CN1CCC[C@H](CNC[C@@H](O)COc2cccc(Br)c2)C1 ZINC000217581037 FE For-Sale Unstable ADRB3 33 42 CN1CCC[C@H](CNC[C@@H](O)COc2cccc(Br)c2)C1 ZINC000217581037 FE For-Sale Unstable CHRNA10 58 37 C[C@H](NC(=O)C1CCCC1)c1ccc(/C=C\C(=O)O)cc1 ZINC000217581076 CG For-Sale Unstable SDH1 0 59 C[C@H](C(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)n1cnc2ccccc2c1=O ZINC000217581102 GD In-Stock Unstable CHRNA4 27 43 O=C(Nc1ccccc1Sc1ccccc1)NC1CCCC1 ZINC000217581106 DJ For-Sale Unstable EPHX2 34 56 CCCCCNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217581111 FH In-Stock Unstable TBXA2R 15 46 CCCCCNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217581111 FH In-Stock Unstable CCR8 78 39 CCCCCNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217581111 FH In-Stock Unstable SFRP1 89 34 CCCCCNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217581111 FH In-Stock Unstable WNT3 72 33 CN1CCC[C@@H](CNC[C@@H](O)COCc2ccccc2)C1 ZINC000217581124 CD For-Sale Unstable ADRB1 21 41 CN1CCC[C@@H](CNC[C@@H](O)COCc2ccccc2)C1 ZINC000217581124 CD For-Sale Unstable ADRB3 16 40 C[C@@H](NC(=O)C1CCCC1)c1ccc(/C=C\C(=O)O)cc1 ZINC000217581151 CG For-Sale Unstable SDH1 0 59 O=C(NC1CCCCCCCCCCC1)NC1CCCC1 ZINC000217581196 CJ For-Sale Unstable MMP2 0 56 O=C(NC1CCCCCCCCCCC1)NC1CCCC1 ZINC000217581196 CJ For-Sale Unstable ADH1B 0 42 O=C(NC1CCCCCCCCCCC1)NC1CCCC1 ZINC000217581196 CJ For-Sale Unstable P95276_MYCTO 0 55 CN1CCC[C@H](CNC[C@@H](O)COCc2ccccc2)C1 ZINC000217581219 CD For-Sale Unstable ADRB1 21 41 CN1CCC[C@H](CNC[C@@H](O)COCc2ccccc2)C1 ZINC000217581219 CD For-Sale Unstable ADRB3 16 40 CC(C)CCNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217581234 FG In-Stock Unstable CCR8 76 39 CC(C)CCNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217581234 FG In-Stock Unstable SFRP1 89 34 CC(C)CCNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217581234 FG In-Stock Unstable WNT3 73 35 COc1ccc2nnc(CCCC(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)n2n1 ZINC000217581259 HD In-Stock Unstable CHRNA4 27 48 O=C(Nc1cc(Cl)ccc1O)NC1CCCC1 ZINC000217581316 CG For-Sale Unstable CNR1 18 40 O=C(Nc1cc(Cl)ccc1O)NC1CCCC1 ZINC000217581316 CG For-Sale Unstable EPHX2 38 58 O=C(Nc1cc(Cl)ccc1O)NC1CCCC1 ZINC000217581316 CG For-Sale Unstable KCNMA1 29 51 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217581355 FH In-Stock Unstable CCR8 56 36 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217581355 FH In-Stock Unstable SFRP1 56 33 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217581355 FH In-Stock Unstable WNT3 45 33 CCOc1cc(C(=O)Nc2ccccc2Oc2ccccc2)cc(Cl)c1O ZINC000217581396 GK On-Demand Unstable TSPO 45 44 CCOc1cc(C(=O)Nc2ccccc2Oc2ccccc2)cc(Cl)c1O ZINC000217581396 GK On-Demand Unstable PYGM 30 42 CCc1ccc(NC(=O)[C@@H]2CC[C@@H](CNC(=O)[C@@H]3Cc4ccccc4CN3)CC2)cc1 ZINC000217581409 HH In-Stock Unstable CFTR 44 33 O=C(Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl)NC1CCCC1 ZINC000217581426 GE For-Sale Unstable LPL 47 41 O=C(Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl)NC1CCCC1 ZINC000217581426 GE For-Sale Unstable CNR2 16 46 O=C(Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl)NC1CCCC1 ZINC000217581426 GE For-Sale Unstable EPHX2 50 48 O=C(Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl)NC1CCCC1 ZINC000217581426 GE For-Sale Unstable TGM2 48 39 O=C(Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl)NC1CCCC1 ZINC000217581426 GE For-Sale Unstable MURF 0 43 O=C(Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl)NC1CCCC1 ZINC000217581426 GE For-Sale Unstable F13A1 40 36 O=C(Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl)NC1CCCC1 ZINC000217581426 GE For-Sale Unstable MERTK 31 42 O=C(Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl)NC1CCCC1 ZINC000217581426 GE For-Sale Unstable LIPG 19 41 CCC[C@H](C)Nc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217581437 FH In-Stock Unstable CCR8 56 36 CCC[C@H](C)Nc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217581437 FH In-Stock Unstable SFRP1 56 33 CCC[C@H](C)Nc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217581437 FH In-Stock Unstable WNT3 45 33 CC[C@@H](C)NCC(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217581488 CF For-Sale Unstable ACE 18 41 CC[C@@H](C)NCC(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217581488 CF For-Sale Unstable DPP4 23 48 CC[C@@H](C)NCC(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217581488 CF For-Sale Unstable PREP 22 41 CC[C@@H](C)NCC(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217581488 CF For-Sale Unstable DPP7 27 40 O=C1O[C@@]2(CCCN(C(=O)CCc3ccc([N+](=O)[O-])cc3)C2)c2ccccc21 ZINC000217581496 GG For-Sale Unstable NPY5R 20 42 CC(=O)N[C@@H](CC(=O)Nc1ccccc1Oc1ccccc1)c1ccc(Br)cc1 ZINC000217581504 JK On-Demand Unstable ACACA 16 41 CC(=O)N[C@@H](CC(=O)Nc1ccccc1Oc1ccccc1)c1ccc(Br)cc1 ZINC000217581504 JK On-Demand Unstable ACACB 15 41 CCCCN(CCC)C(=O)NC1CCCC1 ZINC000217581526 BG For-Sale Unstable USP1 0 41 COC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217581552 FE In-Stock Unstable CCR8 54 36 COC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217581552 FE In-Stock Unstable SFRP1 63 33 COC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217581552 FE In-Stock Unstable WNT3 51 33 CC[C@H](C)NCC(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217581578 CF For-Sale Unstable ACE 18 41 CC[C@H](C)NCC(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217581578 CF For-Sale Unstable DPP4 23 48 CC[C@H](C)NCC(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217581578 CF For-Sale Unstable PREP 22 41 CC[C@H](C)NCC(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217581578 CF For-Sale Unstable DPP7 27 40 O=C1O[C@]2(CCCN(C(=O)CCc3ccc([N+](=O)[O-])cc3)C2)c2ccccc21 ZINC000217581593 GG For-Sale Unstable NPY5R 20 42 CC(=O)N[C@H](CC(=O)Nc1ccccc1Oc1ccccc1)c1ccc(Br)cc1 ZINC000217581595 JK On-Demand Unstable ACACA 16 41 CC(=O)N[C@H](CC(=O)Nc1ccccc1Oc1ccccc1)c1ccc(Br)cc1 ZINC000217581595 JK On-Demand Unstable ACACB 15 41 CC(C)n1nnc(-c2ccc(C(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)cc2)n1 ZINC000217581598 HE In-Stock Unstable CHRNA4 27 43 COC[C@H](C)Nc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217581640 FE In-Stock Unstable SFRP1 50 33 CC[C@@H](C)NCC(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217581661 CF For-Sale Unstable ACE 18 41 CC[C@@H](C)NCC(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217581661 CF For-Sale Unstable DPP4 23 48 CC[C@@H](C)NCC(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217581661 CF For-Sale Unstable PREP 22 41 CC[C@@H](C)NCC(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217581661 CF For-Sale Unstable DPP7 27 40 N#Cc1ccc(CCC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217581699 FG For-Sale Unstable NPY5R 20 41 CCCNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217581703 FG In-Stock Unstable CCR8 81 41 CCCNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217581703 FG In-Stock Unstable SFRP1 95 35 CCCNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217581703 FG In-Stock Unstable WNT3 78 35 Cc1ccc(O)c(NC(=O)NC2CCCC2)c1 ZINC000217581755 BF For-Sale Unstable FAAH 0 45 Cc1ccc(O)c(NC(=O)NC2CCCC2)c1 ZINC000217581755 BF For-Sale Unstable EPHX2 49 50 Cc1ccc(O)c(NC(=O)NC2CCCC2)c1 ZINC000217581755 BF For-Sale Unstable KCNMA1 17 41 CC[C@H](C)NCC(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217581762 CF For-Sale Unstable ACE 18 41 CC[C@H](C)NCC(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217581762 CF For-Sale Unstable DPP4 23 48 CC[C@H](C)NCC(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217581762 CF For-Sale Unstable PREP 22 41 CC[C@H](C)NCC(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217581762 CF For-Sale Unstable DPP7 27 40 N#Cc1ccc(CCC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217581774 FG For-Sale Unstable NPY5R 20 41 Cc1ccccc1CN1CCN(CC2CC2)C[C@@H](C(=O)O)C1 ZINC000217581780 DE In-Stock Unstable SLC6A1 145 47 Cc1ccccc1CN1CCN(CC2CC2)C[C@@H](C(=O)O)C1 ZINC000217581780 DE In-Stock Unstable VACHT_TETCF 0 46 Cc1ccccc1CN1CCN(CC2CC2)C[C@@H](C(=O)O)C1 ZINC000217581780 DE In-Stock Unstable S1PR3 23 40 CC(C)Nc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217581786 FG In-Stock Unstable CCR8 62 41 CC(C)Nc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217581786 FG In-Stock Unstable SFRP1 90 34 CC(C)Nc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217581786 FG In-Stock Unstable WNT3 73 34 COc1ccccc1CN1C(=O)N[C@@H](CC(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)C1=O ZINC000217581794 JD In-Stock Unstable CHRNA4 27 42 CCCCNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217581869 FH In-Stock Unstable CCR8 79 40 CCCCNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217581869 FH In-Stock Unstable SFRP1 92 34 CCCCNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217581869 FH In-Stock Unstable WNT3 76 34 O=C(NC1CCCC1)N(Cc1ccccc1)Cc1ccccc1 ZINC000217581870 DI On-Demand Unstable SIGMAR1 22 43 O=C(NC1CCCC1)N(Cc1ccccc1)Cc1ccccc1 ZINC000217581870 DI On-Demand Unstable PREP 47 34 O=C(NC1CCCC1)N(Cc1ccccc1)Cc1ccccc1 ZINC000217581870 DI On-Demand Unstable FAAH 21 45 O=C(NC1CCCC1)N(Cc1ccccc1)Cc1ccccc1 ZINC000217581870 DI On-Demand Unstable EPHX2 30 56 O=C(NC1CCCC1)N(Cc1ccccc1)Cc1ccccc1 ZINC000217581870 DI On-Demand Unstable PTGES 28 70 O=C(NC1CCCC1)N(Cc1ccccc1)Cc1ccccc1 ZINC000217581870 DI On-Demand Unstable UPPS 0 45 O=C(NC1CCCC1)N(Cc1ccccc1)Cc1ccccc1 ZINC000217581870 DI On-Demand Unstable USP1 0 40 O=C(NC1CCCC1)N(Cc1ccccc1)Cc1ccccc1 ZINC000217581870 DI On-Demand Unstable LUXN 0 40 O=C1O[C@@]2(CCCN(C(=O)c3cc4cc(F)ccc4s3)C2)c2ccccc21 ZINC000217581901 GI For-Sale Unstable NPY5R 30 44 CC(C)CNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217581952 FG In-Stock Unstable MTNN 70 32 CC(C)CNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217581952 FG In-Stock Unstable CCR8 79 41 CC(C)CNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217581952 FG In-Stock Unstable SFRP1 95 35 CC(C)CNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217581952 FG In-Stock Unstable WNT3 78 36 Cc1ccc2nc(SC/C=C\CN)[nH]c2c1 ZINC000217581978 BE For-Sale Unstable CYP2C8 27 42 Cc1ccc2nc(SC/C=C\CN)[nH]c2c1 ZINC000217581978 BE For-Sale Unstable CYP2C19 36 44 Nc1ccc(N(C(=O)NC2CCCC2)c2ccccc2)cc1 ZINC000217581979 CI For-Sale Unstable EPHX2 20 48 CCC[C@@H](C)C(=O)NCc1ccc(/C=C\C(=O)O)cc1 ZINC000217581984 CF For-Sale Unstable AMP1_PLAFQ 40 39 COc1ccccc1CN1C(=O)N[C@@H](CCC(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)C1=O ZINC000217581985 JD In-Stock Unstable CHRNA4 27 44 O=C1O[C@]2(CCCN(C(=O)c3cc4cc(F)ccc4s3)C2)c2ccccc21 ZINC000217581997 GI For-Sale Unstable NPY5R 30 44 CC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217582019 FH In-Stock Unstable CCR8 65 38 CC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217582019 FH In-Stock Unstable SFRP1 79 34 CC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217582019 FH In-Stock Unstable WNT3 58 34 O=C(NC1CCCC1)[C@@H]1CC[C@@H](CNC(=O)[C@@H]2Cc3ccccc3CN2)CC1 ZINC000217582059 GF In-Stock Unstable NPY2R 23 40 O=C(NC1CCCC1)[C@@H]1CC[C@@H](CNC(=O)[C@@H]2Cc3ccccc3CN2)CC1 ZINC000217582059 GF In-Stock Unstable EPHX2 29 40 CC[C@H](C)[C@@H](NC(=O)CN[C@H](C)CC)C(=O)OC ZINC000217582064 CD For-Sale Unstable LASB 0 41 C[C@H](F)[C@@H]1Cc2cc(Br)ccc2N1 ZINC000217582067 BG For-Sale Unstable PNMT 21 50 CCC[C@H](C)C(=O)NCc1ccc(/C=C\C(=O)O)cc1 ZINC000217582073 CF For-Sale Unstable AMP1_PLAFQ 40 39 CC(=O)N(C(=O)NC1CCCC1)c1cccc(N)c1 ZINC000217582077 CE For-Sale Unstable FAAH 19 46 COc1ccc(OC/C=C\CN)cc1 ZINC000217582078 AD For-Sale Unstable AOC3 21 50 CC[C@H](C)Nc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217582101 FH In-Stock Unstable CCR8 65 38 CC[C@H](C)Nc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217582101 FH In-Stock Unstable SFRP1 79 34 CC[C@H](C)Nc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217582101 FH In-Stock Unstable WNT3 58 34 CC(=O)Nc1ccc(CC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217582104 GF In-Stock Unstable NPY5R 33 42 O=C(N[C@@H]1CCN2CCCC[C@@H]12)c1ccnc(F)c1 ZINC000217582113 CD On-Demand Unstable L3MBTL3 49 33 C[C@@H](F)[C@@H]1Cc2cc(Br)ccc2N1 ZINC000217582153 BG For-Sale Unstable PNMT 21 50 Cn1nccc1C(=O)NCc1ccc(/C=C\C(=O)O)cc1 ZINC000217582175 CD For-Sale Unstable HDAC6 25 43 CC(=O)Nc1ccc(CC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217582187 GF In-Stock Unstable NPY5R 31 46 CC(C)(C)Nc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217582196 FH In-Stock Unstable CCR8 78 42 CC(C)(C)Nc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217582196 FH In-Stock Unstable SFRP1 107 36 CC(C)(C)Nc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217582196 FH In-Stock Unstable WNT3 83 37 NC/C=C\COc1ccc(Oc2ccccc2)cc1 ZINC000217582199 CG For-Sale Unstable TAAR1 26 55 O=C(N[C@H]1CCN2CCCC[C@@H]12)c1ccnc(F)c1 ZINC000217582214 CD On-Demand Unstable L3MBTL3 49 33 C[C@H](F)[C@H]1Cc2cc(Br)ccc2N1 ZINC000217582228 BG For-Sale Unstable PNMT 21 50 C=CCNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217582271 FF In-Stock Unstable TGM2 17 41 C=CCNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217582271 FF In-Stock Unstable F13A1 30 41 C=CCNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217582271 FF In-Stock Unstable CCR8 77 40 C=CCNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217582271 FF In-Stock Unstable SFRP1 92 35 C=CCNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217582271 FF In-Stock Unstable WNT3 73 35 O=C(NCC1(c2ccsc2)CCCC1)c1cc2ccccc2[nH]1 ZINC000217582280 DI In-Stock Unstable CCKAR 29 45 O=C(NCC1(c2ccsc2)CCCC1)c1cc2ccccc2[nH]1 ZINC000217582280 DI In-Stock Unstable PYGL 67 41 O=C(NCC1(c2ccsc2)CCCC1)c1cc2ccccc2[nH]1 ZINC000217582280 DI In-Stock Unstable PYGM 32 41 O=C(NCC1(c2ccsc2)CCCC1)c1cc2ccccc2[nH]1 ZINC000217582280 DI In-Stock Unstable ACAT 0 48 CCc1nc2ccc(C(=O)N3CCC[C@]4(C3)OC(=O)c3ccccc34)cc2s1 ZINC000217582288 GI For-Sale Unstable NPY5R 29 42 C[C@@H](F)[C@H]1Cc2cc(Br)ccc2N1 ZINC000217582314 BG For-Sale Unstable PNMT 21 50 Cc1cc(Cl)cc(=O)n1C[C@@H]1CCCO1 ZINC000217582346 BD In-Stock Unstable PDE8B 51 36 Cn1nnc(-c2ccc(OCC(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)cc2)n1 ZINC000217582353 HD In-Stock Unstable CHRNA4 28 44 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NC1CC1 ZINC000217582360 FF In-Stock Unstable SFRP1 93 34 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NC1CC1 ZINC000217582360 FF In-Stock Unstable WNT3 40 30 CCc1nc2ccc(C(=O)N3CCC[C@@]4(C3)OC(=O)c3ccccc34)cc2s1 ZINC000217582365 GI For-Sale Unstable NPY5R 29 42 N#CSc1ccc(NC(=O)NC2CCCC2)cc1 ZINC000217582370 CG For-Sale Unstable DHODH 52 38 N#CSc1ccc(NC(=O)NC2CCCC2)cc1 ZINC000217582370 CG For-Sale Unstable EPHX2 53 51 Cc1noc(C)c1CCC(=O)NCC1(c2ccsc2)CCCC1 ZINC000217582394 EH In-Stock Unstable ACAT 0 46 NC/C=C\COc1ccc2ccccc2c1 ZINC000217582404 BF For-Sale Unstable CYP2A5 0 42 Cc1cc(Cl)cc(=O)n1C[C@H]1CCCO1 ZINC000217582405 BD In-Stock Unstable PDE8B 51 36 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1ccc(I)cc1Cl ZINC000217582413 GK For-Sale Unstable TRPM8 16 46 Cc1ccc(C(=O)C2C(=O)CCCC2=O)cc1 ZINC000217582421 BE For-Sale Unstable HPD 19 47 Cn1cccc1C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217582432 CE For-Sale Unstable HDAC8 42 40 Cn1cccc1C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217582432 CE For-Sale Unstable HDAC1 16 41 Cn1cccc1C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217582432 CE For-Sale Unstable HDAC6 37 53 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NC1CCCC1 ZINC000217582437 GH In-Stock Unstable CCR8 59 43 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NC1CCCC1 ZINC000217582437 GH In-Stock Unstable SFRP1 119 35 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NC1CCCC1 ZINC000217582437 GH In-Stock Unstable WNT3 80 35 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NC1CCCC1 ZINC000217582437 GH In-Stock Unstable BRD4 0 40 C[C@H](F)[C@@H]1Cc2ccc(Br)cc2N1 ZINC000217582439 BG For-Sale Unstable PNMT 29 44 Cc1ccc(F)cc1C(=O)N1c2ccccc2CC[C@@H]1C ZINC000217582462 CI On-Demand Unstable DRD4 17 40 Cc1ccc(F)cc1C(=O)N1c2ccccc2CC[C@@H]1C ZINC000217582462 CI On-Demand Unstable AVPR2 48 40 Cc1ccc(F)cc1C(=O)N1c2ccccc2CC[C@@H]1C ZINC000217582462 CI On-Demand Unstable AVPR1A 24 40 CC(=O)Nc1ccc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217582468 FF For-Sale Unstable NPY5R 38 45 CC(=O)Nc1ccc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217582468 FF For-Sale Unstable EPHX2 17 40 O=C(NC1CCCC1)N(Cc1ccccc1)c1ccccc1 ZINC000217582482 CI For-Sale Unstable CHRM2 22 45 O=C(NC1CCCC1)N(Cc1ccccc1)c1ccccc1 ZINC000217582482 CI For-Sale Unstable CHRM1 25 45 O=C(NC1CCCC1)N(Cc1ccccc1)c1ccccc1 ZINC000217582482 CI For-Sale Unstable DRD4 15 41 O=C(NC1CCCC1)N(Cc1ccccc1)c1ccccc1 ZINC000217582482 CI For-Sale Unstable CHRM3 27 45 O=C(NC1CCCC1)N(Cc1ccccc1)c1ccccc1 ZINC000217582482 CI For-Sale Unstable SIGMAR1 22 48 O=C(NC1CCCC1)N(Cc1ccccc1)c1ccccc1 ZINC000217582482 CI For-Sale Unstable FAAH 18 41 O=C(NC1CCCC1)N(Cc1ccccc1)c1ccccc1 ZINC000217582482 CI For-Sale Unstable EPHX2 22 52 O=C(NC1CCCC1)N(Cc1ccccc1)c1ccccc1 ZINC000217582482 CI For-Sale Unstable PTGES 18 52 O=C(NC1CCCC1)N(Cc1ccccc1)c1ccccc1 ZINC000217582482 CI For-Sale Unstable UPPS 0 43 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1ccc(I)cc1Cl ZINC000217582492 GK For-Sale Unstable TRPM8 16 46 C[C@@H](F)[C@@H]1Cc2ccc(Br)cc2N1 ZINC000217582510 BG For-Sale Unstable PNMT 29 44 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NC1CCCCC1 ZINC000217582513 GI In-Stock Unstable CCR8 59 43 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NC1CCCCC1 ZINC000217582513 GI In-Stock Unstable SFRP1 119 35 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NC1CCCCC1 ZINC000217582513 GI In-Stock Unstable WNT3 80 35 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NC1CCCCC1 ZINC000217582513 GI In-Stock Unstable BRD4 0 40 Cc1ccc(F)cc1C(=O)N1c2ccccc2CC[C@H]1C ZINC000217582550 CI On-Demand Unstable DRD4 17 40 Cc1ccc(F)cc1C(=O)N1c2ccccc2CC[C@H]1C ZINC000217582550 CI On-Demand Unstable AVPR2 48 40 Cc1ccc(F)cc1C(=O)N1c2ccccc2CC[C@H]1C ZINC000217582550 CI On-Demand Unstable AVPR1A 24 40 CC(=O)Nc1ccc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217582551 FF For-Sale Unstable NPY5R 38 45 CC(=O)Nc1ccc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217582551 FF For-Sale Unstable EPHX2 17 40 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1ccc(I)cc1Cl ZINC000217582556 GK For-Sale Unstable TRPM8 16 46 COc1ccc2[nH]c(C(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)cc2c1 ZINC000217582564 FF In-Stock Unstable CHRNA4 26 43 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NCCC1=CCCCC1 ZINC000217582610 HJ In-Stock Unstable SFRP1 53 32 O=C(Cc1c(F)cccc1Cl)NCC1(c2ccsc2)CCCC1 ZINC000217582613 FJ In-Stock Unstable ACAT 0 50 C[C@H](F)[C@H]1Cc2ccc(Br)cc2N1 ZINC000217582614 BG For-Sale Unstable PNMT 29 44 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1ccc(I)cc1Cl ZINC000217582644 GK For-Sale Unstable TRPM8 16 46 COCCOc1ccc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217582667 GG For-Sale Unstable NPY5R 23 43 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NCCO ZINC000217582684 FD In-Stock Unstable CCR8 76 42 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NCCO ZINC000217582684 FD In-Stock Unstable SFRP1 97 36 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NCCO ZINC000217582684 FD In-Stock Unstable WNT3 77 35 C[C@@H](F)[C@H]1Cc2ccc(Br)cc2N1 ZINC000217582696 BG For-Sale Unstable PNMT 29 44 O=CNCCCNC(=O)NC1CCCC1 ZINC000217582698 BC For-Sale Unstable EPHX2 24 62 Cn1cc(C(=O)NCC2(c3ccsc3)CCCC2)nn1 ZINC000217582706 CE In-Stock Unstable ACAT 0 55 COCCOc1ccc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217582746 GG For-Sale Unstable NPY5R 23 43 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NCCCO ZINC000217582775 FE In-Stock Unstable CCR8 73 40 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NCCCO ZINC000217582775 FE In-Stock Unstable SFRP1 112 40 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NCCCO ZINC000217582775 FE In-Stock Unstable WNT3 76 34 COc1ccc(C(=O)NCC2(c3ccsc3)CCCC2)cc1F ZINC000217582792 EI In-Stock Unstable ACAT 0 47 CCO[C@@H]1C[C@@H](NC(=O)c2ccc(C#N)cc2)C1(C)C ZINC000217582821 CE For-Sale Unstable ABCC9 38 40 CCO[C@@H]1C[C@@H](NC(=O)c2ccc(C#N)cc2)C1(C)C ZINC000217582821 CE For-Sale Unstable CTRB_BOVIN 46 33 O=C1O[C@@]2(CCCN(C(=O)CCCCCN3C(=O)c4ccccc4C3=O)C2)c2ccccc21 ZINC000217582843 IH For-Sale Unstable NPY5R 28 40 CC1(C)C[C@H]2C[C@@](C)(CN2C(=O)NC2CCCC2)C1 ZINC000217582849 CH On-Demand Unstable AVPR2 15 41 CC1(C)C[C@H]2C[C@@](C)(CN2C(=O)NC2CCCC2)C1 ZINC000217582849 CH On-Demand Unstable AVPR1A 34 41 COCCNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217582858 FE In-Stock Unstable CCR8 44 35 COCCNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217582858 FE In-Stock Unstable SFRP1 90 34 COCCNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217582858 FE In-Stock Unstable WNT3 51 32 Cc1cncnc1C1CCN(C(=O)CCC(F)(F)F)CC1 ZINC000217582864 DF In-Stock Unstable ETHR 77 46 CCO[C@H]1C[C@@H](NC(=O)c2ccc(C#N)cc2)C1(C)C ZINC000217582891 CE For-Sale Unstable ABCC9 38 40 CCO[C@H]1C[C@@H](NC(=O)c2ccc(C#N)cc2)C1(C)C ZINC000217582891 CE For-Sale Unstable CTRB_BOVIN 46 33 O=C1NCCN1C(=O)NCC1(c2ccsc2)CCCC1 ZINC000217582900 CE In-Stock Unstable ACAT 0 48 N#C[C@H](c1ccccc1)N1CCN(C(=O)[C@@H]2C[C@@H]2c2ccc(C(F)(F)F)cc2)CC1 ZINC000217582912 HI On-Demand Unstable PTAFR 50 48 O=C1O[C@]2(CCCN(C(=O)CCCCCN3C(=O)c4ccccc4C3=O)C2)c2ccccc21 ZINC000217582923 IH For-Sale Unstable NPY5R 28 40 COCCCNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217582930 GF In-Stock Unstable CCR8 91 40 COCCCNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217582930 GF In-Stock Unstable SFRP1 101 33 COCCCNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217582930 GF In-Stock Unstable WNT3 68 33 Nc1ccccc1C(=O)NC(=O)NC1CCCC1 ZINC000217582962 BD For-Sale Unstable EPHX2 28 49 CCO[C@@H]1C[C@H](NC(=O)c2ccc(C#N)cc2)C1(C)C ZINC000217582970 CE For-Sale Unstable ABCC9 38 40 CCO[C@@H]1C[C@H](NC(=O)c2ccc(C#N)cc2)C1(C)C ZINC000217582970 CE For-Sale Unstable CTRB_BOVIN 46 33 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NCc1ccccc1 ZINC000217583001 HH In-Stock Unstable TGM2 22 43 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NCc1ccccc1 ZINC000217583001 HH In-Stock Unstable F13A1 25 43 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NCc1ccccc1 ZINC000217583001 HH In-Stock Unstable CCR8 97 47 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NCc1ccccc1 ZINC000217583001 HH In-Stock Unstable SFRP1 135 39 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NCc1ccccc1 ZINC000217583001 HH In-Stock Unstable WNT3 90 38 O=C(CCc1ccccc1F)NCC1(c2ccsc2)CCCC1 ZINC000217583003 EI In-Stock Unstable ACAT 0 49 CCO[C@H]1C[C@H](NC(=O)c2ccc(C#N)cc2)C1(C)C ZINC000217583039 CE For-Sale Unstable ABCC9 38 40 CCO[C@H]1C[C@H](NC(=O)c2ccc(C#N)cc2)C1(C)C ZINC000217583039 CE For-Sale Unstable CTRB_BOVIN 46 33 N#C[C@H](c1ccccc1)N1CCN(C(=O)[C@H]2C[C@@H]2c2ccc(C(F)(F)F)cc2)CC1 ZINC000217583070 HI On-Demand Unstable PTAFR 50 48 C[C@@H](Nc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O)c1ccccc1 ZINC000217583074 HJ In-Stock Unstable CCR8 82 41 C[C@@H](Nc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O)c1ccccc1 ZINC000217583074 HJ In-Stock Unstable SFRP1 123 35 C[C@@H](Nc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O)c1ccccc1 ZINC000217583074 HJ In-Stock Unstable WNT3 85 35 O=C(Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1)NC1CCCC1 ZINC000217583087 EJ For-Sale Unstable JUN 24 44 O=C(Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1)NC1CCCC1 ZINC000217583087 EJ For-Sale Unstable ATF1 31 40 O=C(Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1)NC1CCCC1 ZINC000217583087 EJ For-Sale Unstable NFKB1 29 40 O=C(Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1)NC1CCCC1 ZINC000217583087 EJ For-Sale Unstable EPHX2 63 55 O=C(Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1)NC1CCCC1 ZINC000217583087 EJ For-Sale Unstable CXCR3 22 58 O=C(Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1)NC1CCCC1 ZINC000217583087 EJ For-Sale Unstable PTPA 0 47 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](CCSC)C(=O)NC[C@@H]3C[C@H]4C=C[C@@H]3C4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217583107 KJ In-Stock Unstable TUBA1A 16 57 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](CCSC)C(=O)NC[C@@H]3C[C@H]4C=C[C@@H]3C4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217583107 KJ In-Stock Unstable TPPP 0 56 O=C(/C=C/c1ccoc1)NCC1(c2ccsc2)CCCC1 ZINC000217583111 DH In-Stock Unstable ACAT 0 46 C[C@H](Nc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O)c1ccccc1 ZINC000217583149 HJ In-Stock Unstable CCR8 82 41 C[C@H](Nc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O)c1ccccc1 ZINC000217583149 HJ In-Stock Unstable SFRP1 123 35 C[C@H](Nc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O)c1ccccc1 ZINC000217583149 HJ In-Stock Unstable WNT3 85 35 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](CCSC)C(=O)NC[C@@H]3C[C@@H]4C=C[C@@H]3C4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217583174 KJ In-Stock Unstable TUBA1A 16 57 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](CCSC)C(=O)NC[C@@H]3C[C@@H]4C=C[C@@H]3C4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217583174 KJ In-Stock Unstable TPPP 0 56 Nc1ccc(C(=O)NC(=O)NC2CCCC2)cc1 ZINC000217583201 BD For-Sale Unstable EPHX2 45 43 COc1cccc(C(=O)NCC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217583217 GE For-Sale Unstable DRD4 52 40 COc1cccc(C(=O)NCC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217583217 GE For-Sale Unstable NPY5R 26 48 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NCCc1ccccc1 ZINC000217583237 HI In-Stock Unstable EPHX2 20 40 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NCCc1ccccc1 ZINC000217583237 HI In-Stock Unstable CCR8 93 49 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NCCc1ccccc1 ZINC000217583237 HI In-Stock Unstable SFRP1 131 38 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NCCc1ccccc1 ZINC000217583237 HI In-Stock Unstable WNT3 88 37 N#C[C@H](c1ccccc1)N1CCN(C(=O)[C@@H]2C[C@@H]2c2ccccc2C(F)(F)F)CC1 ZINC000217583283 HI On-Demand Unstable PTAFR 49 45 N#C[C@H](c1ccccc1)N1CCN(C(=O)[C@@H]2C[C@@H]2c2ccccc2C(F)(F)F)CC1 ZINC000217583283 HI On-Demand Unstable RBP4 91 42 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Oc1ncc(CO)cc1Cl ZINC000217583291 CI For-Sale Unstable TRPM8 0 40 COc1cccc(C(=O)NCC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217583296 GE For-Sale Unstable DRD4 52 40 COc1cccc(C(=O)NCC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217583296 GE For-Sale Unstable NPY5R 26 48 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCCC3)cc2C(=O)O)cc1 ZINC000217583302 II In-Stock Unstable BMP1 53 39 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCCC3)cc2C(=O)O)cc1 ZINC000217583302 II In-Stock Unstable MMP13 65 44 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCCC3)cc2C(=O)O)cc1 ZINC000217583302 II In-Stock Unstable ADAM17 32 41 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCCC3)cc2C(=O)O)cc1 ZINC000217583302 II In-Stock Unstable MMP2 42 44 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCCC3)cc2C(=O)O)cc1 ZINC000217583302 II In-Stock Unstable MMP3 56 42 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCCC3)cc2C(=O)O)cc1 ZINC000217583302 II In-Stock Unstable MMP9 48 41 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCCC3)cc2C(=O)O)cc1 ZINC000217583302 II In-Stock Unstable PTGDR 29 40 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCCC3)cc2C(=O)O)cc1 ZINC000217583302 II In-Stock Unstable MMP7 47 40 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCCC3)cc2C(=O)O)cc1 ZINC000217583302 II In-Stock Unstable CA9 19 40 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCCC3)cc2C(=O)O)cc1 ZINC000217583302 II In-Stock Unstable MMP1 57 41 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCCC3)cc2C(=O)O)cc1 ZINC000217583302 II In-Stock Unstable CCR8 56 43 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCCC3)cc2C(=O)O)cc1 ZINC000217583302 II In-Stock Unstable TYRO3 15 41 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCCC3)cc2C(=O)O)cc1 ZINC000217583302 II In-Stock Unstable SFRP1 65 31 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCCC3)cc2C(=O)O)cc1 ZINC000217583302 II In-Stock Unstable AKR1C2 44 35 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCCC3)cc2C(=O)O)cc1 ZINC000217583302 II In-Stock Unstable WNT3 51 31 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Oc1ncc(CO)cc1Cl ZINC000217583364 CI For-Sale Unstable TRPM8 0 40 Cn1cc(C(=O)NCc2ccc(/C=C\C(=O)O)cc2)cn1 ZINC000217583381 CD For-Sale Unstable HDAC8 35 45 Cn1cc(C(=O)NCc2ccc(/C=C\C(=O)O)cc2)cn1 ZINC000217583381 CD For-Sale Unstable HDAC1 35 45 Cn1cc(C(=O)NCc2ccc(/C=C\C(=O)O)cc2)cn1 ZINC000217583381 CD For-Sale Unstable HDAC2 0 45 Cn1cc(C(=O)NCc2ccc(/C=C\C(=O)O)cc2)cn1 ZINC000217583381 CD For-Sale Unstable HDAC4 0 45 Cn1cc(C(=O)NCc2ccc(/C=C\C(=O)O)cc2)cn1 ZINC000217583381 CD For-Sale Unstable HDAC9 15 45 Cn1cc(C(=O)NCc2ccc(/C=C\C(=O)O)cc2)cn1 ZINC000217583381 CD For-Sale Unstable NAMPT 49 39 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCCC3)cc2C(=O)O)cc1OC ZINC000217583386 JI In-Stock Unstable FKBP1A 41 42 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCCC3)cc2C(=O)O)cc1OC ZINC000217583386 JI In-Stock Unstable ADRA1D 19 41 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCCC3)cc2C(=O)O)cc1OC ZINC000217583386 JI In-Stock Unstable ADRA1B 23 41 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCCC3)cc2C(=O)O)cc1OC ZINC000217583386 JI In-Stock Unstable ABCC8 19 44 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCCC3)cc2C(=O)O)cc1OC ZINC000217583386 JI In-Stock Unstable PTGDR 24 40 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCCC3)cc2C(=O)O)cc1OC ZINC000217583386 JI In-Stock Unstable CCR8 42 40 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCCC3)cc2C(=O)O)cc1OC ZINC000217583386 JI In-Stock Unstable SFRP1 48 32 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCCC3)cc2C(=O)O)cc1OC ZINC000217583386 JI In-Stock Unstable WNT3 43 30 COc1ccc(CCNc2ccc(S(=O)(=O)NC3CCCCCC3)cc2C(=O)O)cc1OC ZINC000217583386 JI In-Stock Unstable SCMU_MYCTU 0 43 CN1CCC(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)CC1 ZINC000217583401 EE For-Sale Unstable NPY5R 48 41 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Oc1ncc(CO)cc1Cl ZINC000217583443 CI For-Sale Unstable TRPM8 0 40 N#C[C@H](c1ccccc1)N1CCN(C(=O)[C@H]2C[C@@H]2c2ccccc2C(F)(F)F)CC1 ZINC000217583446 HI On-Demand Unstable PTAFR 49 45 N#C[C@H](c1ccccc1)N1CCN(C(=O)[C@H]2C[C@@H]2c2ccccc2C(F)(F)F)CC1 ZINC000217583446 HI On-Demand Unstable RBP4 91 42 CCCCCC(=O)NCc1ccc(/C=C\C(=O)O)cc1 ZINC000217583469 CF For-Sale Unstable CNR1 0 55 CCCCCC(=O)NCc1ccc(/C=C\C(=O)O)cc1 ZINC000217583469 CF For-Sale Unstable TRPV1 0 50 CCCCCC(=O)NCc1ccc(/C=C\C(=O)O)cc1 ZINC000217583469 CF For-Sale Unstable HDAC8 26 42 CCCCCC(=O)NCc1ccc(/C=C\C(=O)O)cc1 ZINC000217583469 CF For-Sale Unstable S1PR2 27 40 CCCCCC(=O)NCc1ccc(/C=C\C(=O)O)cc1 ZINC000217583469 CF For-Sale Unstable AKR1C3 33 41 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NCc1ccco1 ZINC000217583476 GH In-Stock Unstable CCR8 70 39 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NCc1ccco1 ZINC000217583476 GH In-Stock Unstable SFRP1 116 35 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NCc1ccco1 ZINC000217583476 GH In-Stock Unstable WNT3 81 35 CN1CCC(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)CC1 ZINC000217583485 EE For-Sale Unstable NPY5R 48 41 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Oc1ncc(CO)cc1Cl ZINC000217583519 CI For-Sale Unstable TRPM8 0 40 O=C(NC[C@H](O)c1ccc2c(c1)CCO2)c1cc2ccccc2[nH]1 ZINC000217583536 DF In-Stock Unstable ADRB2 27 41 O=C(NC[C@H](O)c1ccc2c(c1)CCO2)c1cc2ccccc2[nH]1 ZINC000217583536 DF In-Stock Unstable PYGL 72 41 O=C(NC[C@H](O)c1ccc2c(c1)CCO2)c1cc2ccccc2[nH]1 ZINC000217583536 DF In-Stock Unstable AKR1C3 0 44 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NC[C@@H]1CCCO1 ZINC000217583547 GF In-Stock Unstable BDKRB1 0 42 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NC[C@@H]1CCCO1 ZINC000217583547 GF In-Stock Unstable TNK2 42 37 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NC[C@@H]1CCCO1 ZINC000217583547 GF In-Stock Unstable CCR8 71 40 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NC[C@@H]1CCCO1 ZINC000217583547 GF In-Stock Unstable SFRP1 95 33 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NC[C@@H]1CCCO1 ZINC000217583547 GF In-Stock Unstable WNT3 57 33 CC(C)C(=O)NCc1ccc(/C=C\C(=O)O)cc1 ZINC000217583591 BE For-Sale Unstable PTGER2 0 40 CC(C)C(=O)NCc1ccc(/C=C\C(=O)O)cc1 ZINC000217583591 BE For-Sale Unstable ANPEP 21 43 CC(C)C(=O)NCc1ccc(/C=C\C(=O)O)cc1 ZINC000217583591 BE For-Sale Unstable AMP1_PLAFQ 52 43 O=C1O[C@@]2(CCCN(C(=O)Cn3cc(-c4ccc(F)cc4)cn3)C2)c2ccccc21 ZINC000217583601 HG For-Sale Unstable NPY5R 36 50 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NC[C@H]1CCCO1 ZINC000217583627 GF In-Stock Unstable TNK2 42 37 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NC[C@H]1CCCO1 ZINC000217583627 GF In-Stock Unstable CCR8 71 40 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NC[C@H]1CCCO1 ZINC000217583627 GF In-Stock Unstable SFRP1 95 33 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1NC[C@H]1CCCO1 ZINC000217583627 GF In-Stock Unstable WNT3 57 33 O=C(NC[C@@H](O)c1ccc2c(c1)CCO2)c1cc2ccccc2[nH]1 ZINC000217583629 DF In-Stock Unstable ADRB2 27 41 O=C(NC[C@@H](O)c1ccc2c(c1)CCO2)c1cc2ccccc2[nH]1 ZINC000217583629 DF In-Stock Unstable PYGL 72 41 O=C(NC[C@@H](O)c1ccc2c(c1)CCO2)c1cc2ccccc2[nH]1 ZINC000217583629 DF In-Stock Unstable AKR1C3 0 44 Cc1ccc2nc(-c3ccc(NC(=O)NC4CCCC4)cc3)sc2c1 ZINC000217583632 FK For-Sale Unstable KIT 23 41 Cc1ccc2nc(-c3ccc(NC(=O)NC4CCCC4)cc3)sc2c1 ZINC000217583632 FK For-Sale Unstable LCK 17 48 Cc1ccc2nc(-c3ccc(NC(=O)NC4CCCC4)cc3)sc2c1 ZINC000217583632 FK For-Sale Unstable NMT1 30 42 Cc1ccc2nc(-c3ccc(NC(=O)NC4CCCC4)cc3)sc2c1 ZINC000217583632 FK For-Sale Unstable APP 28 57 Cc1ccc2nc(-c3ccc(NC(=O)NC4CCCC4)cc3)sc2c1 ZINC000217583632 FK For-Sale Unstable KDR 20 45 Cc1ccc2nc(-c3ccc(NC(=O)NC4CCCC4)cc3)sc2c1 ZINC000217583632 FK For-Sale Unstable FAAH 23 59 Cc1ccc2nc(-c3ccc(NC(=O)NC4CCCC4)cc3)sc2c1 ZINC000217583632 FK For-Sale Unstable EPHX2 49 49 COc1cc2c(c(OC)c1OC)-c1ccc(NCCCCCC(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217583641 KJ In-Stock Unstable TUBA1A 15 56 COc1cc2c(c(OC)c1OC)-c1ccc(NCCCCCC(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217583641 KJ In-Stock Unstable TPPP 0 54 O=C1O[C@]2(CCCN(C(=O)Cn3cc(-c4ccc(F)cc4)cn3)C2)c2ccccc21 ZINC000217583691 HG For-Sale Unstable NPY5R 36 50 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1N1CCCC1 ZINC000217583693 FF In-Stock Unstable SLC6A9 15 44 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1N1CCCC1 ZINC000217583693 FF In-Stock Unstable EPHX2 29 41 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1N1CCCC1 ZINC000217583693 FF In-Stock Unstable LIPG 43 33 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1N1CCCC1 ZINC000217583693 FF In-Stock Unstable SFRP1 111 38 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1N1CCCC1 ZINC000217583693 FF In-Stock Unstable WNT3 86 39 O=C(NC(=O)C1CCNCC1)NC1CCCC1 ZINC000217583737 BC For-Sale Unstable EPHX2 32 41 O=C(O)/C=C\c1cccc(CNC(=O)c2cc(Cl)c[nH]2)c1 ZINC000217583761 DF For-Sale Unstable MAPK1 24 48 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1N1CCCCC1 ZINC000217583763 GG In-Stock Unstable SLC6A9 15 44 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1N1CCCCC1 ZINC000217583763 GG In-Stock Unstable EPHX2 29 41 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1N1CCCCC1 ZINC000217583763 GG In-Stock Unstable LIPG 43 33 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1N1CCCCC1 ZINC000217583763 GG In-Stock Unstable SFRP1 111 38 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1N1CCCCC1 ZINC000217583763 GG In-Stock Unstable WNT3 86 39 O=C1O[C@@]2(CCCN(C(=O)c3n[nH]c4cc(F)ccc34)C2)c2ccccc21 ZINC000217583792 FG For-Sale Unstable NPY5R 34 45 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1N1CCOCC1 ZINC000217583838 GE In-Stock Unstable SLC6A9 20 45 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1N1CCOCC1 ZINC000217583838 GE In-Stock Unstable SFRP1 99 40 O=C(O)c1cc(S(=O)(=O)NC2CCCCCC2)ccc1N1CCOCC1 ZINC000217583838 GE In-Stock Unstable WNT3 79 40 Cc1cc(C)c(NC(=O)NC2CCCC2)c(Cl)c1 ZINC000217583845 CI On-Demand Unstable EPHX2 40 58 CC(C)CCC(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217583846 CF For-Sale Unstable PTGER2 0 42 CC(C)CCC(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217583846 CF For-Sale Unstable ANPEP 16 42 CC(C)CCC(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217583846 CF For-Sale Unstable AKR1C3 42 47 O=C1O[C@]2(CCCN(C(=O)c3n[nH]c4cc(F)ccc34)C2)c2ccccc21 ZINC000217583865 FG For-Sale Unstable NPY5R 34 45 O=C(Cn1c(COc2ccccc2)nc2ccccc21)N1CCN(c2cccc(O)c2)CC1 ZINC000217583894 IH On-Demand Unstable CPT1A 29 41 O=C(CC[C@@H]1NC(=O)N(Cc2cccc(F)c2)C1=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217583923 JD In-Stock Unstable CHRNA4 29 51 CCOCCCNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217583926 GG In-Stock Unstable CCR8 85 41 CCOCCCNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217583926 GG In-Stock Unstable SFRP1 96 34 CCOCCCNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217583926 GG In-Stock Unstable WNT3 65 34 CCN(CC)c1ccc(NC(=O)NC2CCCC2)c(C)c1 ZINC000217583955 CH For-Sale Unstable EPHX2 42 50 O=C(O)CNC(=O)c1ccnc(F)c1 ZINC000217583959 AC On-Demand Unstable EGLN1 0 47 O=C(O)CNC(=O)c1ccnc(F)c1 ZINC000217583959 AC On-Demand Unstable KDM4E 35 45 O=C(O)CNC(=O)c1ccnc(F)c1 ZINC000217583959 AC On-Demand Unstable FTO 40 36 O=C1O[C@@]2(CCCN(C(=O)CC34CC5CC(CC(C5)C3)C4)C2)c2ccccc21 ZINC000217583987 GI For-Sale Unstable NPY5R 27 40 CC(C)OCCCNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217584003 HH In-Stock Unstable CCR8 71 37 CC(C)OCCCNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217584003 HH In-Stock Unstable SFRP1 96 33 CC(C)OCCCNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217584003 HH In-Stock Unstable WNT3 67 33 O=C1O[C@]2(CCCN(C(=O)CC34CC5CC(CC(C5)C3)C4)C2)c2ccccc21 ZINC000217584069 GI For-Sale Unstable NPY5R 27 40 Cc1nc(O)nc(C)c1CCC(=O)NCCc1noc(-c2ccccc2)n1 ZINC000217584073 FE In-Stock Unstable KCNQ1 0 40 Cc1ccnc(NC(=O)NC2CCCC2)c1 ZINC000217584075 BE On-Demand Unstable EPHX2 37 49 Cc1ccnc(NC(=O)NC2CCCC2)c1 ZINC000217584075 BE On-Demand Unstable TYK2 54 35 CCCCCNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217584090 GH In-Stock Unstable TBXA2R 15 46 CCCCCNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217584090 GH In-Stock Unstable CCR8 78 39 CCCCCNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217584090 GH In-Stock Unstable SFRP1 89 34 CCCCCNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217584090 GH In-Stock Unstable WNT3 72 33 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@H](C(=O)NC[C@@H]3C[C@H]4C=C[C@@H]3C4)C(C)C)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217584107 KJ In-Stock Unstable TUBA1A 17 60 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@H](C(=O)NC[C@@H]3C[C@H]4C=C[C@@H]3C4)C(C)C)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217584107 KJ In-Stock Unstable TPPP 0 59 CC(C)CCNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217584157 GH In-Stock Unstable CCR8 76 39 CC(C)CCNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217584157 GH In-Stock Unstable SFRP1 89 34 CC(C)CCNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217584157 GH In-Stock Unstable WNT3 73 35 CC/C(=N/O)c1cccc(Br)c1 ZINC000217584160 BG For-Sale Unstable CYSP_TRYCR 0 59 O=C1O[C@@]2(CCCN(C(=O)c3ccc(-c4cccs4)cc3)C2)c2ccccc21 ZINC000217584182 GJ For-Sale Unstable NPY5R 30 42 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@H](C(=O)NC[C@@H]3C[C@@H]4C=C[C@@H]3C4)C(C)C)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217584184 KJ In-Stock Unstable TUBA1A 17 60 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@H](C(=O)NC[C@@H]3C[C@@H]4C=C[C@@H]3C4)C(C)C)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217584184 KJ In-Stock Unstable TPPP 0 59 CC[C@@H](C)c1ccccc1NC(=O)NC1CCCC1 ZINC000217584195 CI For-Sale Unstable KCNQ2 47 37 CC[C@@H](C)c1ccccc1NC(=O)NC1CCCC1 ZINC000217584195 CI For-Sale Unstable EPHX2 48 50 CC[C@@H](C)c1ccccc1NC(=O)NC1CCCC1 ZINC000217584195 CI For-Sale Unstable ACAT 0 44 CC[C@@H](C)c1ccccc1NC(=O)NC1CCCC1 ZINC000217584195 CI For-Sale Unstable AO-ACHE 0 43 O=C(Cn1c(COc2ccccc2)nc2ccccc21)N1CC=C(c2ccc(O)cc2)CC1 ZINC000217584206 IJ On-Demand Unstable PTGDR2 15 41 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217584235 GH In-Stock Unstable CCR8 56 36 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217584235 GH In-Stock Unstable SFRP1 56 33 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217584235 GH In-Stock Unstable WNT3 45 33 O=C1O[C@]2(CCCN(C(=O)c3ccc(-c4cccs4)cc3)C2)c2ccccc21 ZINC000217584258 GJ For-Sale Unstable NPY5R 30 42 CC[C@H](C)c1ccccc1NC(=O)NC1CCCC1 ZINC000217584274 CI For-Sale Unstable KCNQ2 47 37 CC[C@H](C)c1ccccc1NC(=O)NC1CCCC1 ZINC000217584274 CI For-Sale Unstable EPHX2 48 50 CC[C@H](C)c1ccccc1NC(=O)NC1CCCC1 ZINC000217584274 CI For-Sale Unstable ACAT 0 44 CC[C@H](C)c1ccccc1NC(=O)NC1CCCC1 ZINC000217584274 CI For-Sale Unstable AO-ACHE 0 43 CCC[C@H](C)Nc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217584310 GH In-Stock Unstable CCR8 70 36 CCC[C@H](C)Nc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217584310 GH In-Stock Unstable SFRP1 69 33 CCC[C@H](C)Nc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217584310 GH In-Stock Unstable WNT3 52 33 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cccc(C[S@@](C)=O)c3)CC2)cc1 ZINC000217584318 IF On-Demand Unstable DRD4 24 46 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cccc(C[S@@](C)=O)c3)CC2)cc1 ZINC000217584318 IF On-Demand Unstable AVPR1A 19 43 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cccc(C[S@@](C)=O)c3)CC2)cc1 ZINC000217584318 IF On-Demand Unstable SIGMAR1 15 43 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cccc(C[S@@](C)=O)c3)CC2)cc1 ZINC000217584318 IF On-Demand Unstable SSTR5 53 42 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cccc(C[S@@](C)=O)c3)CC2)cc1 ZINC000217584318 IF On-Demand Unstable CCR3 19 41 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cccc(C[S@@](C)=O)c3)CC2)cc1 ZINC000217584318 IF On-Demand Unstable UTS2R 21 44 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cccc(C[S@@](C)=O)c3)CC2)cc1 ZINC000217584318 IF On-Demand Unstable SLC6A5 38 44 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cccc(C[S@@](C)=O)c3)CC2)cc1 ZINC000217584318 IF On-Demand Unstable PLAU 23 44 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cccc(C[S@@](C)=O)c3)CC2)cc1 ZINC000217584318 IF On-Demand Unstable MCHR1 22 46 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cccc(C[S@@](C)=O)c3)CC2)cc1 ZINC000217584318 IF On-Demand Unstable L3MBTL3 42 33 CSc1nc2cc(O)ccc2o1 ZINC000217584348 AE For-Sale Unstable ESR1 19 51 CSc1nc2cc(O)ccc2o1 ZINC000217584348 AE For-Sale Unstable ESR2 19 53 COCCC(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217584349 CD For-Sale Unstable NPY5R 26 41 CCn1cc(CNC(=O)CN(C)Cc2cccnc2)cn1 ZINC000217584379 CD In-Stock Unstable NAMPT 46 38 O=C(NCc1ccc(CO)cc1)NC1CCCC1 ZINC000217584387 BD On-Demand Unstable EPHX2 33 56 COC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217584391 GF In-Stock Unstable CCR8 51 36 COC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217584391 GF In-Stock Unstable SFRP1 50 33 COC[C@@H](C)Nc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217584391 GF In-Stock Unstable WNT3 45 33 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cccc(C[S@](C)=O)c3)CC2)cc1 ZINC000217584400 IF On-Demand Unstable DRD4 24 46 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cccc(C[S@](C)=O)c3)CC2)cc1 ZINC000217584400 IF On-Demand Unstable AVPR1A 19 43 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cccc(C[S@](C)=O)c3)CC2)cc1 ZINC000217584400 IF On-Demand Unstable SIGMAR1 15 43 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cccc(C[S@](C)=O)c3)CC2)cc1 ZINC000217584400 IF On-Demand Unstable SSTR5 53 42 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cccc(C[S@](C)=O)c3)CC2)cc1 ZINC000217584400 IF On-Demand Unstable CCR3 19 41 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cccc(C[S@](C)=O)c3)CC2)cc1 ZINC000217584400 IF On-Demand Unstable UTS2R 21 44 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cccc(C[S@](C)=O)c3)CC2)cc1 ZINC000217584400 IF On-Demand Unstable SLC6A5 38 44 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cccc(C[S@](C)=O)c3)CC2)cc1 ZINC000217584400 IF On-Demand Unstable PLAU 23 44 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cccc(C[S@](C)=O)c3)CC2)cc1 ZINC000217584400 IF On-Demand Unstable MCHR1 22 46 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cccc(C[S@](C)=O)c3)CC2)cc1 ZINC000217584400 IF On-Demand Unstable L3MBTL3 42 33 COc1ccccc1CNC(=O)[C@@H]1CC[C@@H](CNC(=O)[C@@H]2Cc3ccccc3CN2)CC1 ZINC000217584406 IF In-Stock Unstable MC4R 27 41 COc1ccccc1CNC(=O)[C@@H]1CC[C@@H](CNC(=O)[C@@H]2Cc3ccccc3CN2)CC1 ZINC000217584406 IF In-Stock Unstable MTNR1A 27 40 COc1ccccc1CNC(=O)[C@@H]1CC[C@@H](CNC(=O)[C@@H]2Cc3ccccc3CN2)CC1 ZINC000217584406 IF In-Stock Unstable MTNR1B 22 45 COCCC(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217584427 CD For-Sale Unstable NPY5R 26 41 COC[C@H](C)Nc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217584460 GF In-Stock Unstable CCR8 54 36 COC[C@H](C)Nc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217584460 GF In-Stock Unstable SFRP1 63 33 COC[C@H](C)Nc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217584460 GF In-Stock Unstable WNT3 51 33 CN1CCc2ccc(F)c(Br)c2C1 ZINC000217584498 BF For-Sale Unstable DRD1 15 40 Cc1ccc(NC(=O)NC2CCCC2)nc1 ZINC000217584501 BE On-Demand Unstable EPHX2 43 47 Cc1ccc(NC(=O)NC2CCCC2)nc1 ZINC000217584501 BE On-Demand Unstable GCK 21 46 Cc1ccc(NC(=O)NC2CCCC2)nc1 ZINC000217584501 BE On-Demand Unstable LUCI_LUCLA 30 45 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cc(-c4ccco4)nn3-c3ccccc3)CC2)cc1 ZINC000217584509 JJ On-Demand Unstable AVPR1A 19 41 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cc(-c4ccco4)nn3-c3ccccc3)CC2)cc1 ZINC000217584509 JJ On-Demand Unstable INHA 64 33 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cc(-c4ccco4)nn3-c3ccccc3)CC2)cc1 ZINC000217584509 JJ On-Demand Unstable CNR2 15 41 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cc(-c4ccco4)nn3-c3ccccc3)CC2)cc1 ZINC000217584509 JJ On-Demand Unstable SSTR5 45 37 Cn1nc(-c2ccccc2)cc1C(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217584532 GG For-Sale Unstable NPY5R 43 49 CC[C@@H](C)C(=O)N[C@@H](C)c1ccc(/C=C\C(=O)O)cc1 ZINC000217584553 CG For-Sale Unstable ACE2 45 34 CN1CCC[C@@H](CNC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217584596 CE For-Sale Unstable F2 28 42 CN1CCC[C@@H](CNC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217584596 CE For-Sale Unstable SLC6A1 109 41 CN1CCC[C@@H](CNC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217584596 CE For-Sale Unstable OPRK1 19 42 CN1CCC[C@@H](CNC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217584596 CE For-Sale Unstable CCR3 22 41 CN1CCC[C@@H](CNC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217584596 CE For-Sale Unstable CCR5 34 40 CN1CCC[C@@H](CNC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217584596 CE For-Sale Unstable CACNA1I 68 36 CCCCc1nc(C)sc1C(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217584602 FG In-Stock Unstable CHRNA4 29 46 O=C(Nc1ncc(Br)cn1)NC1CCCC1 ZINC000217584605 CE For-Sale Unstable EPHX2 30 49 CN1CCc2ccc(Br)c(F)c2C1 ZINC000217584625 BF For-Sale Unstable DRD1 17 40 Cn1nc(-c2ccccc2)cc1C(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217584630 GG For-Sale Unstable NPY5R 43 49 CC[C@H](C)C(=O)N[C@@H](C)c1ccc(/C=C\C(=O)O)cc1 ZINC000217584635 CG For-Sale Unstable ACE2 45 34 CN1CCC[C@H](CNC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217584668 CE For-Sale Unstable F2 28 42 CN1CCC[C@H](CNC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217584668 CE For-Sale Unstable SLC6A1 109 41 CN1CCC[C@H](CNC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217584668 CE For-Sale Unstable OPRK1 19 42 CN1CCC[C@H](CNC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217584668 CE For-Sale Unstable CCR3 22 41 CN1CCC[C@H](CNC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217584668 CE For-Sale Unstable CCR5 34 40 CN1CCC[C@H](CNC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217584668 CE For-Sale Unstable CACNA1I 68 36 CC(C)Nc1ccc(S(=O)(=O)NCCC2=CCCCC2)cc1C(=O)O ZINC000217584681 FG In-Stock Unstable TBXA2R 41 34 O=C(Nc1ccc(Cl)cn1)NC1CCCC1 ZINC000217584710 BF On-Demand Unstable CNR1 18 44 O=C(Nc1ccc(Cl)cn1)NC1CCCC1 ZINC000217584710 BF On-Demand Unstable F10 48 32 O=C(Nc1ccc(Cl)cn1)NC1CCCC1 ZINC000217584710 BF On-Demand Unstable CETP 0 42 O=C(Nc1ccc(Cl)cn1)NC1CCCC1 ZINC000217584710 BF On-Demand Unstable EPHX2 36 50 O=C(Nc1ccc(Cl)cn1)NC1CCCC1 ZINC000217584710 BF On-Demand Unstable LUCI_LUCLA 30 40 COc1ccc(CCN2C(=O)N[C@@H](CC(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)C2=O)cc1 ZINC000217584722 JD In-Stock Unstable CHRNA4 28 49 CCOc1cc(C(=O)Nc2ccc(C)c(C(F)(F)F)c2)cc(Cl)c1O ZINC000217584765 FK On-Demand Unstable ABL1 47 36 CCOc1cc(C(=O)Nc2ccc(C)c(C(F)(F)F)c2)cc(Cl)c1O ZINC000217584765 FK On-Demand Unstable LCK 29 43 CCOc1cc(C(=O)Nc2ccc(C)c(C(F)(F)F)c2)cc(Cl)c1O ZINC000217584765 FK On-Demand Unstable MAPK14 15 43 CCOc1cc(C(=O)Nc2ccc(C)c(C(F)(F)F)c2)cc(Cl)c1O ZINC000217584765 FK On-Demand Unstable TRPV1 15 42 CCOc1cc(C(=O)Nc2ccc(C)c(C(F)(F)F)c2)cc(Cl)c1O ZINC000217584765 FK On-Demand Unstable ATF1 44 35 CCOc1cc(C(=O)Nc2ccc(C)c(C(F)(F)F)c2)cc(Cl)c1O ZINC000217584765 FK On-Demand Unstable KDR 18 43 CCOc1cc(C(=O)Nc2ccc(C)c(C(F)(F)F)c2)cc(Cl)c1O ZINC000217584765 FK On-Demand Unstable NFKB1 41 35 CCOc1cc(C(=O)Nc2ccc(C)c(C(F)(F)F)c2)cc(Cl)c1O ZINC000217584765 FK On-Demand Unstable BRAF 22 42 CCOc1cc(C(=O)Nc2ccc(C)c(C(F)(F)F)c2)cc(Cl)c1O ZINC000217584765 FK On-Demand Unstable TAAR1 28 41 CCOc1cc(C(=O)Nc2ccc(C)c(C(F)(F)F)c2)cc(Cl)c1O ZINC000217584765 FK On-Demand Unstable SHH 35 41 CCOc1cc(C(=O)Nc2ccc(C)c(C(F)(F)F)c2)cc(Cl)c1O ZINC000217584765 FK On-Demand Unstable KCNK3 65 47 CCOc1cc(C(=O)Nc2ccc(C)c(C(F)(F)F)c2)cc(Cl)c1O ZINC000217584765 FK On-Demand Unstable KCNK9 60 47 O=C(Nc1cc(Cl)ccn1)NC1CCCC1 ZINC000217584805 BF On-Demand Unstable GRM5 15 40 O=C(Nc1cc(Cl)ccn1)NC1CCCC1 ZINC000217584805 BF On-Demand Unstable EPHX2 29 49 O=C(Nc1cc(Cl)ccn1)NC1CCCC1 ZINC000217584805 BF On-Demand Unstable TYK2 73 40 O=C(C[C@@H]1NC(=O)N(Cc2ccccc2Cl)C1=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217584857 JD In-Stock Unstable CHRNA4 27 46 CC(C)CNc1ccc(S(=O)(=O)NCCC2=CCCCC2)cc1C(=O)O ZINC000217584898 GH In-Stock Unstable BDKRB1 17 42 CCCC(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217584910 CE For-Sale Unstable NPY5R 30 41 O=C(Nc1cc(Br)ccn1)NC1CCCC1 ZINC000217584921 CF On-Demand Unstable TYK2 57 36 CCCC(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217584995 CE For-Sale Unstable NPY5R 30 41 CCc1nc(C)sc1C(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217585080 EE In-Stock Unstable CHRNA4 29 47 NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217585092 CC On-Demand Unstable CA2 195 70 NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217585092 CC On-Demand Unstable CA6 35 44 NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217585092 CC On-Demand Unstable CA1 174 59 NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217585092 CC On-Demand Unstable CA7 96 64 NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217585092 CC On-Demand Unstable CA13 39 44 NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217585092 CC On-Demand Unstable CA5B 69 51 NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217585092 CC On-Demand Unstable CA4 146 61 NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217585092 CC On-Demand Unstable CA5A 75 51 NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217585092 CC On-Demand Unstable CA14 71 66 NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217585092 CC On-Demand Unstable CA12 130 65 NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217585092 CC On-Demand Unstable CA9 134 56 NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217585092 CC On-Demand Unstable CAH_METTE 49 50 NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217585092 CC On-Demand Unstable UREA_CANEN 30 44 NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217585092 CC On-Demand Unstable IDO1 30 40 NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217585092 CC On-Demand Unstable CYNT 57 50 NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217585092 CC On-Demand Unstable NCE103 70 45 NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217585092 CC On-Demand Unstable MTCA1 74 65 NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217585092 CC On-Demand Unstable P96878_MYCTU 91 65 NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217585092 CC On-Demand Unstable CA 0 44 NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217585092 CC On-Demand Unstable Q5TU56_ANOGA 0 44 CC(=O)N[C@@H](CC(=O)NCc1ccc(F)c(C)c1)c1ccc(Br)cc1 ZINC000217585096 HH On-Demand Unstable LEF 65 39 O=C1O[C@@]2(CCCN(C(=O)c3cc(-c4ccccc4)n[nH]3)C2)c2ccccc21 ZINC000217585103 FG For-Sale Unstable TACR3 20 42 O=C1O[C@@]2(CCCN(C(=O)c3cc(-c4ccccc4)n[nH]3)C2)c2ccccc21 ZINC000217585103 FG For-Sale Unstable NPY5R 45 60 O=C(O)/C=C\c1cccc(CNC(=O)Cc2ccsc2)c1 ZINC000217585148 DF For-Sale Unstable PTGER2 24 43 CCOC(=O)NCCNC(=O)NC1CCCC1 ZINC000217585159 BC For-Sale Unstable EPHX2 27 56 O=C1O[C@]2(CCCN(C(=O)c3cc(-c4ccccc4)n[nH]3)C2)c2ccccc21 ZINC000217585186 FG For-Sale Unstable TACR3 20 42 O=C1O[C@]2(CCCN(C(=O)c3cc(-c4ccccc4)n[nH]3)C2)c2ccccc21 ZINC000217585186 FG For-Sale Unstable NPY5R 45 60 CC(=O)N[C@H](CC(=O)NCc1ccc(F)c(C)c1)c1ccc(Br)cc1 ZINC000217585187 HH On-Demand Unstable LEF 65 39 CC(C)(C)OC(=O)N1Cc2ccccc2C[C@H]1C(=O)NC[C@@H]1CC[C@@H](C(=O)NC2CCCC2)CC1 ZINC000217585193 JI In-Stock Unstable OPRM1 24 43 CC(C)(C)OC(=O)N1Cc2ccccc2C[C@H]1C(=O)NC[C@@H]1CC[C@@H](C(=O)NC2CCCC2)CC1 ZINC000217585193 JI In-Stock Unstable OPRD1 53 37 CC(C)(C)OC(=O)N1Cc2ccccc2C[C@H]1C(=O)NC[C@@H]1CC[C@@H](C(=O)NC2CCCC2)CC1 ZINC000217585193 JI In-Stock Unstable HDAC8 20 42 CC(C)(C)OC(=O)N1Cc2ccccc2C[C@H]1C(=O)NC[C@@H]1CC[C@@H](C(=O)NC2CCCC2)CC1 ZINC000217585193 JI In-Stock Unstable PREP 25 46 CC(C)(C)OC(=O)N1Cc2ccccc2C[C@H]1C(=O)NC[C@@H]1CC[C@@H](C(=O)NC2CCCC2)CC1 ZINC000217585193 JI In-Stock Unstable CFTR 63 35 CC(C)(C)OC(=O)N1Cc2ccccc2C[C@H]1C(=O)NC[C@@H]1CC[C@@H](C(=O)NC2CCCC2)CC1 ZINC000217585193 JI In-Stock Unstable ADAM9 59 33 Cc1noc(C)c1CC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217585202 ED In-Stock Unstable CHRNA4 29 48 Cc1ccc(C(=O)NCc2cccc(/C=C\C(=O)O)c2)o1 ZINC000217585229 CF For-Sale Unstable PTGER2 22 40 Cc1ccc(C(=O)NCc2cccc(/C=C\C(=O)O)c2)o1 ZINC000217585229 CF For-Sale Unstable MMP13 17 44 COc1ccc([N+](=O)[O-])cc1NC(=O)C(F)F ZINC000217585237 BD On-Demand Unstable KCNMA1 31 60 COc1ccc([N+](=O)[O-])cc1NC(=O)C(F)F ZINC000217585237 BD On-Demand Unstable WDR5 33 43 O=C(CCc1ccc(C(F)(F)F)cc1)NC[C@H](O)c1ccc2c(c1)CCO2 ZINC000217585277 GG In-Stock Unstable TRAR 18 44 CCOc1cc(C(=O)N2CCC(NC(=O)c3ccccc3)CC2)cc(Cl)c1O ZINC000217585286 HG On-Demand Unstable DRD2 19 48 CCOc1cc(C(=O)N2CCC(NC(=O)c3ccccc3)CC2)cc(Cl)c1O ZINC000217585286 HG On-Demand Unstable CNR1 17 40 CCOc1cc(C(=O)N2CCC(NC(=O)c3ccccc3)CC2)cc(Cl)c1O ZINC000217585286 HG On-Demand Unstable DRD4 32 44 CCOc1cc(C(=O)N2CCC(NC(=O)c3ccccc3)CC2)cc(Cl)c1O ZINC000217585286 HG On-Demand Unstable DRD3 16 43 CCOc1cc(C(=O)N2CCC(NC(=O)c3ccccc3)CC2)cc(Cl)c1O ZINC000217585286 HG On-Demand Unstable HTR4 31 43 CCOc1cc(C(=O)N2CCC(NC(=O)c3ccccc3)CC2)cc(Cl)c1O ZINC000217585286 HG On-Demand Unstable P2RY12 27 41 CCOc1cc(C(=O)N2CCC(NC(=O)c3ccccc3)CC2)cc(Cl)c1O ZINC000217585286 HG On-Demand Unstable TACR1 17 42 CCOc1cc(C(=O)N2CCC(NC(=O)c3ccccc3)CC2)cc(Cl)c1O ZINC000217585286 HG On-Demand Unstable SIGMAR1 17 44 CCOc1cc(C(=O)N2CCC(NC(=O)c3ccccc3)CC2)cc(Cl)c1O ZINC000217585286 HG On-Demand Unstable SSTR5 67 49 CCOc1cc(C(=O)N2CCC(NC(=O)c3ccccc3)CC2)cc(Cl)c1O ZINC000217585286 HG On-Demand Unstable UTS2R 26 44 CCOc1cc(C(=O)N2CCC(NC(=O)c3ccccc3)CC2)cc(Cl)c1O ZINC000217585286 HG On-Demand Unstable SLC6A5 35 40 CCOc1cc(C(=O)N2CCC(NC(=O)c3ccccc3)CC2)cc(Cl)c1O ZINC000217585286 HG On-Demand Unstable EPHX2 39 41 CCOc1cc(C(=O)N2CCC(NC(=O)c3ccccc3)CC2)cc(Cl)c1O ZINC000217585286 HG On-Demand Unstable MCHR1 25 45 CCOc1cc(C(=O)N2CCC(NC(=O)c3ccccc3)CC2)cc(Cl)c1O ZINC000217585286 HG On-Demand Unstable CCR8 50 37 CCOc1cc(C(=O)N2CCC(NC(=O)c3ccccc3)CC2)cc(Cl)c1O ZINC000217585286 HG On-Demand Unstable SHH 23 43 CCOc1cc(C(=O)N2CCC(NC(=O)c3ccccc3)CC2)cc(Cl)c1O ZINC000217585286 HG On-Demand Unstable HCN1 49 33 CCOc1cc(C(=O)N2CCC(NC(=O)c3ccccc3)CC2)cc(Cl)c1O ZINC000217585286 HG On-Demand Unstable HCN4 42 33 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable ACE 48 45 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable OPRM1 28 42 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable OPRD1 35 42 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable MME 131 45 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable ANPEP 73 38 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable EDNRB 18 40 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable EDNRA 18 45 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable CTSD 20 41 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable PGC 21 46 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable CTRA_BOVIN 15 45 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable FCER2 67 36 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable CASP3 33 52 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable TACR2 23 42 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable CASP8 26 47 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable KLK3 65 41 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable CTSB 77 72 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable PAPA1_CARPA 76 52 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable CTSK 20 48 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable CTSL 51 52 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable CPA1 53 41 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable PGA 43 40 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable CTRB1 32 41 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable CAPNS1 84 49 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable MMP2 17 40 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable HLA-DRB1 74 43 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable LNPEP 18 41 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable PCSK5 44 37 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable CTSH 33 48 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable CAPN1 162 72 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable CASP1 73 67 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable CAPN2 84 58 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable ACE2 84 40 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable CASP6 32 40 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable CASP9 45 40 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable BACE1 21 40 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable FPR1 56 38 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable AMP1_PLAFQ 47 37 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable GAG-PRO 49 35 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable PSMB2 45 42 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable PSMB5 24 42 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable POLG_WNV 64 33 CC(=O)N[C@@H](C(=O)N[C@H](C=O)Cc1ccccc1)C(C)C ZINC000217585304 CD For-Sale Unstable BRCA1 64 38 Cc1noc(C)c1CCC(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217585318 FF For-Sale Unstable NPY5R 28 43 CCCCCC(=O)N(C)Cc1ccc(/C=C\C(=O)O)cc1 ZINC000217585321 CG For-Sale Unstable AKR1C3 25 41 CCCCCC(=O)N(C)Cc1ccc(/C=C\C(=O)O)cc1 ZINC000217585321 CG For-Sale Unstable TRPM2 0 41 O=C(CCc1ccc(C(F)(F)F)cc1)NC[C@@H](O)c1ccc2c(c1)CCO2 ZINC000217585350 GG In-Stock Unstable TRAR 18 44 O=C(C[C@@H]1NC(=O)N(Cc2ccccc2)C1=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217585360 HD In-Stock Unstable CHRNA4 30 57 COc1ccc(NC(=O)NCC2CCCCC2)cc1OC ZINC000217585368 CG On-Demand Unstable PDE4A 30 45 COc1ccc(NC(=O)NCC2CCCCC2)cc1OC ZINC000217585368 CG On-Demand Unstable EPHX2 23 41 COc1ccc(NC(=O)NCC2CCCCC2)cc1OC ZINC000217585368 CG On-Demand Unstable PDGFRA 43 49 COc1ccc(NC(=O)NCC2CCCCC2)cc1OC ZINC000217585368 CG On-Demand Unstable STK17B 45 40 COc1ccc(NC(=O)NCC2CCCCC2)cc1OC ZINC000217585368 CG On-Demand Unstable QRFPR 50 41 COc1ccc(NC(=O)NCC2CCCCC2)cc1OC ZINC000217585368 CG On-Demand Unstable PRMT3 60 46 COc1ccc(NC(=O)NCC2CCCCC2)cc1OC ZINC000217585368 CG On-Demand Unstable ENPP1 64 37 COc1ccc(NC(=O)NCC2CCCCC2)cc1OC ZINC000217585368 CG On-Demand Unstable METAP2 0 45 COc1ccc(NC(=O)NCC2CCCCC2)cc1OC ZINC000217585368 CG On-Demand Unstable PDEC 0 40 Cc1noc(C)c1CCC(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217585384 FF For-Sale Unstable NPY5R 28 43 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable ACE 48 45 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable OPRM1 28 42 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable OPRD1 35 42 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable MME 131 45 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable ANPEP 73 38 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable EDNRB 18 40 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable EDNRA 18 45 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable CTSD 20 41 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable PGC 21 46 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable CTRA_BOVIN 15 45 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable FCER2 67 36 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable CASP3 33 52 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable TACR2 23 42 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable CASP8 26 47 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable KLK3 65 41 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable CTSB 77 72 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable PAPA1_CARPA 76 52 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable CTSK 20 48 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable CTSL 51 52 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable CPA1 53 41 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable PGA 43 40 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable CTRB1 32 41 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable CAPNS1 84 49 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable MMP2 17 40 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable HLA-DRB1 74 43 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable LNPEP 18 41 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable PCSK5 44 37 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable CTSH 33 48 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable CAPN1 162 72 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable CASP1 73 67 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable CAPN2 84 58 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable ACE2 84 40 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable CASP6 32 40 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable CASP9 45 40 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable BACE1 21 40 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable FPR1 56 38 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable AMP1_PLAFQ 47 37 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable GAG-PRO 49 35 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable PSMB2 45 42 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable PSMB5 24 42 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable POLG_WNV 64 33 CC(=O)N[C@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585388 CD For-Sale Unstable BRCA1 64 38 CC(=O)N[C@@H](CC(=O)N1CCC(NC(=O)c2ccccc2)CC1)c1ccc(Br)cc1 ZINC000217585395 JG On-Demand Unstable EPHX2 21 44 O=C(Nc1cc(C(F)(F)F)ccc1Cl)C(F)F ZINC000217585401 CH On-Demand Anodyne TEK 19 42 Cc1ccc2c(c1)nc([C@H](C)Cl)n2C[C@@H]1CCCN(C)C1 ZINC000217585430 DH For-Sale Unstable Q8MHZ5_SHEEP 73 38 O=C(NCCCN1CCCC1=O)NCC1CCCCC1 ZINC000217585465 CD On-Demand Unstable TYRO3 27 43 COc1cc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc(OC)c1OC ZINC000217585466 GG For-Sale Unstable HRH1 24 40 COc1cc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc(OC)c1OC ZINC000217585466 GG For-Sale Unstable TACR1 35 41 COc1cc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc(OC)c1OC ZINC000217585466 GG For-Sale Unstable TACR2 17 41 COc1cc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc(OC)c1OC ZINC000217585466 GG For-Sale Unstable NPY5R 27 47 CC(=O)N[C@H](CC(=O)N1CCC(NC(=O)c2ccccc2)CC1)c1ccc(Br)cc1 ZINC000217585468 JG On-Demand Unstable EPHX2 21 44 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable ACE 48 45 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable OPRM1 28 42 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable OPRD1 35 42 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable MME 131 45 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable ANPEP 73 38 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable EDNRB 18 40 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable EDNRA 18 45 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable CTSD 20 41 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable PGC 21 46 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable CTRA_BOVIN 15 45 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable FCER2 67 36 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable CASP3 33 52 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable TACR2 23 42 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable CASP8 26 47 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable KLK3 65 41 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable CTSB 77 72 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable PAPA1_CARPA 76 52 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable CTSK 20 48 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable CTSL 51 52 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable CPA1 53 41 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable PGA 43 40 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable CTRB1 32 41 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable CAPNS1 84 49 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable MMP2 17 40 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable HLA-DRB1 74 43 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable LNPEP 18 41 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable PCSK5 44 37 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable CTSH 33 48 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable CAPN1 162 72 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable CASP1 73 67 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable CAPN2 84 58 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable ACE2 84 40 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable CASP6 32 40 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable CASP9 45 40 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable BACE1 21 40 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable FPR1 56 38 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable AMP1_PLAFQ 47 37 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable GAG-PRO 49 35 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable PSMB2 45 42 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable PSMB5 24 42 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable POLG_WNV 64 33 CC(=O)N[C@@H](C(=O)N[C@@H](C=O)Cc1ccccc1)C(C)C ZINC000217585473 CD For-Sale Unstable BRCA1 64 38 FC(F)(F)c1cc(Cl)nc2[nH]ncc12 ZINC000217585476 BF For-Sale Anodyne TRPA1 26 41 Cc1ccc2c(c1)nc([C@H](C)Cl)n2C[C@H]1CCCN(C)C1 ZINC000217585510 DH For-Sale Unstable Q8MHZ5_SHEEP 73 38 O=C(NC12CC3CC(CC(C3)C1)C2)C(F)F ZINC000217585518 BE On-Demand Unstable EPHX2 90 59 O=C(NC12CC3CC(CC(C3)C1)C2)C(F)F ZINC000217585518 BE On-Demand Unstable P95276_MYCTO 0 44 COc1cc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc(OC)c1OC ZINC000217585546 GG For-Sale Unstable HRH1 24 40 COc1cc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc(OC)c1OC ZINC000217585546 GG For-Sale Unstable TACR1 35 41 COc1cc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc(OC)c1OC ZINC000217585546 GG For-Sale Unstable TACR2 17 41 COc1cc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc(OC)c1OC ZINC000217585546 GG For-Sale Unstable NPY5R 27 47 O=C(NCC1CCCCC1)Nc1ccccc1[N+](=O)[O-] ZINC000217585555 CG For-Sale Unstable COLA 77 32 CCOc1cc(C(=O)N2CCC(CCc3ccccc3)CC2)cc(Cl)c1O ZINC000217585567 GJ On-Demand Unstable ACHE 43 43 CCOc1cc(C(=O)N2CCC(CCc3ccccc3)CC2)cc(Cl)c1O ZINC000217585567 GJ On-Demand Unstable GRIN2B 58 47 CCOc1cc(C(=O)N2CCC(CCc3ccccc3)CC2)cc(Cl)c1O ZINC000217585567 GJ On-Demand Unstable SIGMAR1 22 41 CCOc1cc(C(=O)N2CCC(CCc3ccccc3)CC2)cc(Cl)c1O ZINC000217585567 GJ On-Demand Unstable CACNA1I 45 34 CC(C)Cc1ccc(-c2cc(C(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)[nH]n2)cc1 ZINC000217585613 HH In-Stock Unstable CHRNA4 36 46 O=C1O[C@@]2(CCCN(C(=O)c3ccccc3Cl)C2)c2ccccc21 ZINC000217585635 EH For-Sale Unstable AVPR1A 15 49 O=C1O[C@@]2(CCCN(C(=O)c3ccccc3Cl)C2)c2ccccc21 ZINC000217585635 EH For-Sale Unstable NPY5R 33 48 O=C(NCC1CCCCC1)Nc1cccc(O)c1 ZINC000217585679 BG For-Sale Unstable CCR3 60 39 O=C(NCC1CCCCC1)Nc1cccc(O)c1 ZINC000217585679 BG For-Sale Unstable LDLR 0 43 O=C(NCC1CCCCC1)Nc1cccc(O)c1 ZINC000217585679 BG For-Sale Unstable EPHX2 35 74 O=C(NCC1CCCCC1)Nc1cccc(O)c1 ZINC000217585679 BG For-Sale Unstable PRMT3 43 42 O=C(NCC1CCCCC1)Nc1cccc(O)c1 ZINC000217585679 BG For-Sale Unstable ACAT 0 41 CC(=O)N[C@@H](CC(=O)N1CCC(CCc2ccccc2)CC1)c1ccc(Br)cc1 ZINC000217585686 JJ On-Demand Unstable PTAFR 17 42 O=C1O[C@]2(CCCN(C(=O)c3ccccc3Cl)C2)c2ccccc21 ZINC000217585716 EH For-Sale Unstable AVPR1A 15 49 O=C1O[C@]2(CCCN(C(=O)c3ccccc3Cl)C2)c2ccccc21 ZINC000217585716 EH For-Sale Unstable NPY5R 33 48 CC(=O)N[C@H](CC(=O)N1CCC(CCc2ccccc2)CC1)c1ccc(Br)cc1 ZINC000217585751 JJ On-Demand Unstable PTAFR 17 42 CN1CC=CC[C@H](NC(=O)OC(C)(C)C)C1=O ZINC000217585756 BD For-Sale Unstable NAAA 15 49 O=C(O)c1cc(S(=O)(=O)NCCC2=CCCCC2)ccc1NCCC1=CCCCC1 ZINC000217585764 IJ In-Stock Unstable TBXA2R 42 33 Cc1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217585787 BH On-Demand Unstable CCR3 21 46 Cc1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217585787 BH On-Demand Unstable EPHX2 39 46 Cc1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217585787 BH On-Demand Unstable CA12 15 44 Cc1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217585787 BH On-Demand Unstable CA9 15 44 Cc1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217585787 BH On-Demand Unstable NCE103 24 40 Cc1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217585787 BH On-Demand Unstable PRMT3 35 42 Fc1ccc(Br)c(C[C@@H]2CCN2)c1 ZINC000217585794 BE For-Sale Unstable CHRNA10 24 42 CC(=O)NCC(=O)N[C@@H](C)c1ccc(/C=C\C(=O)O)cc1 ZINC000217585815 CD For-Sale Unstable ACACA 45 37 O=C1O[C@@]2(CCCN(C(=O)COc3ccc4ccccc4c3)C2)c2ccccc21 ZINC000217585833 GH For-Sale Unstable NPY5R 29 42 CCOc1nc(C)c(NC(=O)COc2ccccc2)c(C)n1 ZINC000217585838 DF In-Stock Unstable ADORA2A 15 50 CCOc1cc(C(=O)NCc2ccc(OC(F)(F)F)cc2)cc(Cl)c1O ZINC000217585852 GI On-Demand Unstable GCGR 52 45 CCOc1cc(C(=O)NCc2ccc(OC(F)(F)F)cc2)cc(Cl)c1O ZINC000217585852 GI On-Demand Unstable PPARA 30 46 CCOc1cc(C(=O)NCc2ccc(OC(F)(F)F)cc2)cc(Cl)c1O ZINC000217585852 GI On-Demand Unstable GRIN2B 19 43 CCOc1cc(C(=O)NCc2ccc(OC(F)(F)F)cc2)cc(Cl)c1O ZINC000217585852 GI On-Demand Unstable PPARD 29 46 CCOc1cc(C(=O)NCc2ccc(OC(F)(F)F)cc2)cc(Cl)c1O ZINC000217585852 GI On-Demand Unstable ADCYAP1R1 42 31 CCOc1cc(C(=O)NCc2ccc(OC(F)(F)F)cc2)cc(Cl)c1O ZINC000217585852 GI On-Demand Unstable AKR1C2 15 43 CCOc1cc(C(=O)NCc2ccc(OC(F)(F)F)cc2)cc(Cl)c1O ZINC000217585852 GI On-Demand Unstable PDS 55 37 Fc1ccc(Br)c(C[C@H]2CCN2)c1 ZINC000217585870 BE For-Sale Unstable CHRNA10 24 42 CC(=O)NCC(=O)N[C@H](C)c1ccc(/C=C\C(=O)O)cc1 ZINC000217585883 CD For-Sale Unstable ACACA 45 37 CC(=O)N(C(=O)NCC1CCCCC1)c1ccc(N)cc1 ZINC000217585898 CF For-Sale Unstable AMY2 43 30 O=C1O[C@]2(CCCN(C(=O)COc3ccc4ccccc4c3)C2)c2ccccc21 ZINC000217585931 GH For-Sale Unstable NPY5R 29 42 CC[C@@H](C)[C@H](Nc1ccc2c(cc1=O)[C@@H](NC(C)=O)CCc1cc(OC)c(OC)c(OC)c1-2)C(=O)NC[C@@H]1C[C@H]2C=C[C@@H]1C2 ZINC000217585941 KK In-Stock Unstable TUBA1A 17 60 CCOc1nc(C)c(NC(=O)CCCc2ccccc2)c(C)n1 ZINC000217585943 DG In-Stock Unstable FAAH 57 37 CCOc1nc(C)c(NC(=O)CCCc2ccccc2)c(C)n1 ZINC000217585943 DG In-Stock Unstable CES1 50 35 CCOc1nc(C)c(NC(=O)CCCc2ccccc2)c(C)n1 ZINC000217585943 DG In-Stock Unstable CES1D 54 32 O=C(NCC1CCCCC1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217585993 DF For-Sale Unstable CA2 25 51 O=C(NCC1CCCCC1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217585993 DF For-Sale Unstable CA1 38 43 O=C(NCC1CCCCC1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217585993 DF For-Sale Unstable CCR3 28 40 O=C(NCC1CCCCC1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217585993 DF For-Sale Unstable EPHX2 45 64 O=C(NCC1CCCCC1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217585993 DF For-Sale Unstable CA12 36 47 O=C(NCC1CCCCC1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217585993 DF For-Sale Unstable CA9 32 47 O=C(NCC1CCCCC1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217585993 DF For-Sale Unstable F13A1 64 41 O=C(NCC1CCCCC1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217585993 DF For-Sale Unstable NCE103 36 43 O=C(NCC1CCCCC1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217585993 DF For-Sale Unstable PRMT3 41 40 O=C(NCC1CCCCC1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217585993 DF For-Sale Unstable MTCA1 45 47 O=C(NCC1CCCCC1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217585993 DF For-Sale Unstable P96878_MYCTU 56 47 O=C(NCC1CCCCC1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217585993 DF For-Sale Unstable NAMPT 52 45 CC[C@@H](C)[C@H](Nc1ccc2c(cc1=O)[C@@H](NC(C)=O)CCc1cc(OC)c(OC)c(OC)c1-2)C(=O)NC[C@@H]1C[C@@H]2C=C[C@@H]1C2 ZINC000217586009 KK In-Stock Unstable TUBA1A 17 60 O=C1O[C@@]2(CCCN(C(=O)c3cnn(-c4ccccc4)n3)C2)c2ccccc21 ZINC000217586033 FF For-Sale Unstable NPY5R 34 46 COc1ccccc1C(=O)N1CCN(c2cnnc(N(C)C)c2)CC1 ZINC000217586047 ED In-Stock Unstable TACR3 24 42 O=C(NCC1CCCCC1)Nc1cccc(S(=O)(=O)O)c1 ZINC000217586102 DF For-Sale Unstable NPY2R 17 44 O=C(NCC1CCCCC1)Nc1cccc(S(=O)(=O)O)c1 ZINC000217586102 DF For-Sale Unstable CCR3 67 44 O=C(NCC1CCCCC1)Nc1cccc(S(=O)(=O)O)c1 ZINC000217586102 DF For-Sale Unstable EPHX2 38 71 O=C(NCC1CCCCC1)Nc1cccc(S(=O)(=O)O)c1 ZINC000217586102 DF For-Sale Unstable ST14 44 37 O=C(NCC1CCCCC1)Nc1cccc(S(=O)(=O)O)c1 ZINC000217586102 DF For-Sale Unstable PRMT3 41 39 O=C1O[C@]2(CCCN(C(=O)c3cnn(-c4ccccc4)n3)C2)c2ccccc21 ZINC000217586103 FF For-Sale Unstable NPY5R 34 46 CCCCC/C=C\C=C/C=C\C(N)=O ZINC000217586106 AF For-Sale Unstable CNR1 26 53 CCCCC/C=C\C=C/C=C\C(N)=O ZINC000217586106 AF For-Sale Unstable FABP4 17 44 CCCCC/C=C\C=C/C=C\C(N)=O ZINC000217586106 AF For-Sale Unstable FAAH 30 49 CCCCC/C=C\C=C/C=C\C(N)=O ZINC000217586106 AF For-Sale Unstable FABP3 34 44 CCCCC/C=C\C=C/C=C\C(N)=O ZINC000217586106 AF For-Sale Unstable OXER1 22 46 CCc1ccc(C(=O)N2CCN(c3cnnc(N(C)C)c3)CC2)cc1 ZINC000217586157 EE In-Stock Unstable LSS 16 41 CCc1ccc(C(=O)N2CCN(c3cnnc(N(C)C)c3)CC2)cc1 ZINC000217586157 EE In-Stock Unstable SLC6A7 0 51 O=C(O)/C=C\c1ccc(CNC(=O)c2ccccc2)cc1 ZINC000217586189 CF For-Sale Unstable PTGER2 36 42 O=C(O)/C=C\c1ccc(CNC(=O)c2ccccc2)cc1 ZINC000217586189 CF For-Sale Unstable PTGER4 0 42 O=C(O)/C=C\c1ccc(CNC(=O)c2ccccc2)cc1 ZINC000217586189 CF For-Sale Unstable PTGER3 15 42 O=C(O)/C=C\c1ccc(CNC(=O)c2ccccc2)cc1 ZINC000217586189 CF For-Sale Unstable HDAC8 31 54 O=C(O)/C=C\c1ccc(CNC(=O)c2ccccc2)cc1 ZINC000217586189 CF For-Sale Unstable CTRB1 19 40 O=C(O)/C=C\c1ccc(CNC(=O)c2ccccc2)cc1 ZINC000217586189 CF For-Sale Unstable F3 24 41 O=C(O)/C=C\c1ccc(CNC(=O)c2ccccc2)cc1 ZINC000217586189 CF For-Sale Unstable HDAC1 40 47 O=C(O)/C=C\c1ccc(CNC(=O)c2ccccc2)cc1 ZINC000217586189 CF For-Sale Unstable HDAC2 28 58 O=C(O)/C=C\c1ccc(CNC(=O)c2ccccc2)cc1 ZINC000217586189 CF For-Sale Unstable HDAC3 16 42 O=C(O)/C=C\c1ccc(CNC(=O)c2ccccc2)cc1 ZINC000217586189 CF For-Sale Unstable HDAC6 28 58 O=C(O)/C=C\c1ccc(CNC(=O)c2ccccc2)cc1 ZINC000217586189 CF For-Sale Unstable AMP1_PLAFQ 33 40 COCCCNc1ccc(S(=O)(=O)NCCC2=CCCCC2)cc1C(=O)O ZINC000217586196 GG In-Stock Unstable BDKRB1 16 40 Cc1ccc(NC(=O)NCC2CCCCC2)cc1Cl ZINC000217586222 CI For-Sale Unstable DHODH 15 46 Cc1ccc(NC(=O)NCC2CCCCC2)cc1Cl ZINC000217586222 CI For-Sale Unstable NPY2R 43 39 Cc1ccc(NC(=O)NCC2CCCCC2)cc1Cl ZINC000217586222 CI For-Sale Unstable CCR3 64 40 Cc1ccc(NC(=O)NCC2CCCCC2)cc1Cl ZINC000217586222 CI For-Sale Unstable RAF1 25 44 Cc1ccc(NC(=O)NCC2CCCCC2)cc1Cl ZINC000217586222 CI For-Sale Unstable LDLR 0 42 Cc1ccc(NC(=O)NCC2CCCCC2)cc1Cl ZINC000217586222 CI For-Sale Unstable EPHX2 57 67 Cc1ccc(NC(=O)NCC2CCCCC2)cc1Cl ZINC000217586222 CI For-Sale Unstable MCHR1 26 41 Cc1ccc(NC(=O)NCC2CCCCC2)cc1Cl ZINC000217586222 CI For-Sale Unstable Q8MMZ8_EIMTE 31 44 Cc1ccc(NC(=O)NCC2CCCCC2)cc1Cl ZINC000217586222 CI For-Sale Unstable CACNA1I 68 38 Cc1ccc(NC(=O)NCC2CCCCC2)cc1Cl ZINC000217586222 CI For-Sale Unstable PRMT3 37 45 Cc1ccc(NC(=O)NCC2CCCCC2)cc1Cl ZINC000217586222 CI For-Sale Unstable HSPB1 0 41 Cc1c(CCC(=O)O)ccc(OCc2c(-c3ccc(Cl)cc3)nsc2C(F)(F)F)c1C ZINC000217586256 JK Annotated Unstable PPARD 38 40 CCC[C@@H](C)C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217586265 CF For-Sale Unstable PTGER2 22 40 CCC[C@@H](C)C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217586265 CF For-Sale Unstable ANPEP 15 43 CCC[C@@H](C)C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217586265 CF For-Sale Unstable FURIN 44 33 CCC[C@@H](C)C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217586265 CF For-Sale Unstable CAPN2 40 37 CCC[C@@H](C)C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217586265 CF For-Sale Unstable AKR1C3 39 43 CCC[C@@H](C)C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217586265 CF For-Sale Unstable CARM1 42 36 CCC[C@@H](C)C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217586265 CF For-Sale Unstable PDS 51 33 O=C(O)c1cc(S(=O)(=O)NCCC2=CCCCC2)ccc1NCc1ccccc1 ZINC000217586297 HI In-Stock Unstable TBXA2R 48 38 Cc1c(Cl)cccc1NC(=O)NCC1CCCCC1 ZINC000217586340 CI On-Demand Unstable CXCL8 53 34 Cc1c(Cl)cccc1NC(=O)NCC1CCCCC1 ZINC000217586340 CI On-Demand Unstable P2RX7 16 40 Cc1c(Cl)cccc1NC(=O)NCC1CCCCC1 ZINC000217586340 CI On-Demand Unstable EPHX2 15 58 Cc1c(Cl)cccc1NC(=O)NCC1CCCCC1 ZINC000217586340 CI On-Demand Unstable CACNA1I 40 33 Cc1c(Cl)cccc1NC(=O)NCC1CCCCC1 ZINC000217586340 CI On-Demand Unstable ACAT 0 45 CCC[C@H](C)C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217586350 CF For-Sale Unstable PTGER2 22 40 CCC[C@H](C)C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217586350 CF For-Sale Unstable ANPEP 15 43 CCC[C@H](C)C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217586350 CF For-Sale Unstable FURIN 44 33 CCC[C@H](C)C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217586350 CF For-Sale Unstable CAPN2 40 37 CCC[C@H](C)C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217586350 CF For-Sale Unstable AKR1C3 39 43 CCC[C@H](C)C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217586350 CF For-Sale Unstable CARM1 42 36 CCC[C@H](C)C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217586350 CF For-Sale Unstable PDS 51 33 CCCCC/C=C/C=C/C=C\C(N)=O ZINC000217586354 AF For-Sale Unstable CNR1 26 53 CCCCC/C=C/C=C/C=C\C(N)=O ZINC000217586354 AF For-Sale Unstable FABP4 17 44 CCCCC/C=C/C=C/C=C\C(N)=O ZINC000217586354 AF For-Sale Unstable FAAH 30 49 CCCCC/C=C/C=C/C=C\C(N)=O ZINC000217586354 AF For-Sale Unstable FABP3 34 44 CCCCC/C=C/C=C/C=C\C(N)=O ZINC000217586354 AF For-Sale Unstable OXER1 22 46 O=C(NCCCn1ccnc1)c1nccc(N2CCCCC2)n1 ZINC000217586368 DD In-Stock Unstable TBXAS1 52 51 O=C(NCCCn1ccnc1)c1nccc(N2CCCCC2)n1 ZINC000217586368 DD In-Stock Unstable QPCT 40 42 O=C(NCCCn1ccnc1)c1nccc(N2CCCCC2)n1 ZINC000217586368 DD In-Stock Unstable NAMPT 24 41 O=C(C(F)F)N1CCCCCC1 ZINC000217586376 AD On-Demand Unstable DPP7 51 43 O=C1O[C@@]2(CCCN(C(=O)c3cc4ccccc4[nH]3)C2)c2ccccc21 ZINC000217586411 EG In-Stock Unstable HRH4 21 49 O=C1O[C@@]2(CCCN(C(=O)c3cc4ccccc4[nH]3)C2)c2ccccc21 ZINC000217586411 EG In-Stock Unstable NPY5R 32 43 O=C1O[C@@]2(CCCN(C(=O)c3cc4ccccc4[nH]3)C2)c2ccccc21 ZINC000217586411 EG In-Stock Unstable AKR1C3 18 44 C[C@@H](Nc1ccc(S(=O)(=O)NCCC2=CCCCC2)cc1C(=O)O)c1ccccc1 ZINC000217586413 IJ In-Stock Unstable BDKRB1 16 40 Cn1nccc1C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217586427 CD For-Sale Unstable HDAC8 49 41 Cn1nccc1C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217586427 CD For-Sale Unstable HDAC1 22 41 Cn1nccc1C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217586427 CD For-Sale Unstable HDAC6 41 41 C=C(CC)COc1c(Br)cc(/C=C\C(=O)O)cc1OCC ZINC000217586432 FI For-Sale Unstable AKR1C3 18 40 COC(=O)CCNC(=O)N1[C@H](C(=O)O)C[C@@H]2CCCC[C@@H]21 ZINC000217586435 CC For-Sale Unstable ACE 18 57 CCOC(=O)c1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217586448 DH On-Demand Unstable CHRM2 0 41 CCOC(=O)c1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217586448 DH On-Demand Unstable CHRM1 17 43 CCOC(=O)c1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217586448 DH On-Demand Unstable CHRM3 20 43 CCOC(=O)c1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217586448 DH On-Demand Unstable CA1 20 41 CCOC(=O)c1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217586448 DH On-Demand Unstable EPHX2 30 63 CCOC(=O)c1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217586448 DH On-Demand Unstable ACR 59 38 CC1CCN(C(=O)c2nccc(N3CCCCC3)n2)CC1 ZINC000217586462 CE In-Stock Unstable SORD 74 38 CC1CCN(C(=O)c2nccc(N3CCCCC3)n2)CC1 ZINC000217586462 CE In-Stock Unstable L3MBTL3 58 37 CC1CCN(C(=O)c2nccc(N3CCCCC3)n2)CC1 ZINC000217586462 CE In-Stock Unstable TRPC6 43 37 COc1ccc2nnc(CCC(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)n2n1 ZINC000217586479 GC In-Stock Unstable CHRNA4 26 44 O=C1O[C@]2(CCCN(C(=O)c3cc4ccccc4[nH]3)C2)c2ccccc21 ZINC000217586480 EG In-Stock Unstable HRH4 21 49 O=C1O[C@]2(CCCN(C(=O)c3cc4ccccc4[nH]3)C2)c2ccccc21 ZINC000217586480 EG In-Stock Unstable NPY5R 32 43 O=C1O[C@]2(CCCN(C(=O)c3cc4ccccc4[nH]3)C2)c2ccccc21 ZINC000217586480 EG In-Stock Unstable AKR1C3 18 44 FC(F)(F)c1ncnc(NC2CC2)c1I ZINC000217586488 EF In-Stock Unstable CD38 34 41 C[C@H](Nc1ccc(S(=O)(=O)NCCC2=CCCCC2)cc1C(=O)O)c1ccccc1 ZINC000217586492 IJ In-Stock Unstable BDKRB1 16 40 Cn1cc(C(=O)NCc2cccc(/C=C\C(=O)O)c2)cn1 ZINC000217586507 CD For-Sale Unstable MMP13 19 41 Cn1cc(C(=O)NCc2cccc(/C=C\C(=O)O)c2)cn1 ZINC000217586507 CD For-Sale Unstable HDAC8 58 42 Cn1cc(C(=O)NCc2cccc(/C=C\C(=O)O)c2)cn1 ZINC000217586507 CD For-Sale Unstable HDAC1 36 49 Cn1cc(C(=O)NCc2cccc(/C=C\C(=O)O)c2)cn1 ZINC000217586507 CD For-Sale Unstable HDAC2 0 49 Cn1cc(C(=O)NCc2cccc(/C=C\C(=O)O)c2)cn1 ZINC000217586507 CD For-Sale Unstable HDAC6 50 42 Cn1cc(C(=O)NCc2cccc(/C=C\C(=O)O)c2)cn1 ZINC000217586507 CD For-Sale Unstable HDAC9 15 49 Cn1cc(C(=O)NCc2cccc(/C=C\C(=O)O)c2)cn1 ZINC000217586507 CD For-Sale Unstable NAMPT 40 36 COC(=O)CCNC(=O)N1[C@H](C(=O)O)C[C@H]2CCCC[C@@H]21 ZINC000217586515 CC For-Sale Unstable ACE 18 57 C=C(CC)COc1cc(OC)ccc1/C=C\C(=O)O ZINC000217586545 CG For-Sale Unstable PTGER2 43 45 C=C(CC)COc1cc(OC)ccc1/C=C\C(=O)O ZINC000217586545 CG For-Sale Unstable PTGER4 24 45 C=C(CC)COc1cc(OC)ccc1/C=C\C(=O)O ZINC000217586545 CG For-Sale Unstable CYP1B1 41 43 C=C(CC)COc1cc(OC)ccc1/C=C\C(=O)O ZINC000217586545 CG For-Sale Unstable PTGER3 17 44 C=C(CC)COc1cc(OC)ccc1/C=C\C(=O)O ZINC000217586545 CG For-Sale Unstable CYP1A1 41 43 C=C(CC)COc1cc(OC)ccc1/C=C\C(=O)O ZINC000217586545 CG For-Sale Unstable CYSP_PLAFA 41 42 O=C(NCC1CCCCC1)Nc1ccccc1Cl ZINC000217586562 CI On-Demand Unstable LPL 32 44 O=C(NCC1CCCCC1)Nc1ccccc1Cl ZINC000217586562 CI On-Demand Unstable CXCL8 57 41 O=C(NCC1CCCCC1)Nc1ccccc1Cl ZINC000217586562 CI On-Demand Unstable KCNQ2 42 39 O=C(NCC1CCCCC1)Nc1ccccc1Cl ZINC000217586562 CI On-Demand Unstable EPHX2 15 60 O=C(NCC1CCCCC1)Nc1ccccc1Cl ZINC000217586562 CI On-Demand Unstable EPHB3 46 33 O=C(NCC1CCCCC1)Nc1ccccc1Cl ZINC000217586562 CI On-Demand Unstable LIPG 15 44 O=C1O[C@@]2(CCCN(C(=O)c3ccc4nc[nH]c4c3)C2)c2ccccc21 ZINC000217586590 EF For-Sale Unstable ACACA 18 40 O=C1O[C@@]2(CCCN(C(=O)c3ccc4nc[nH]c4c3)C2)c2ccccc21 ZINC000217586590 EF For-Sale Unstable ACACB 18 41 O=C1O[C@@]2(CCCN(C(=O)c3ccc4nc[nH]c4c3)C2)c2ccccc21 ZINC000217586590 EF For-Sale Unstable NPY5R 32 43 O=C(O)c1cc(S(=O)(=O)NCCC2=CCCCC2)ccc1NCCc1ccccc1 ZINC000217586603 II In-Stock Unstable TBXA2R 50 40 O=C1O[C@]2(CCCN(C(=O)c3ccc4nc[nH]c4c3)C2)c2ccccc21 ZINC000217586665 EF For-Sale Unstable ACACA 18 40 O=C1O[C@]2(CCCN(C(=O)c3ccc4nc[nH]c4c3)C2)c2ccccc21 ZINC000217586665 EF For-Sale Unstable ACACB 18 41 O=C1O[C@]2(CCCN(C(=O)c3ccc4nc[nH]c4c3)C2)c2ccccc21 ZINC000217586665 EF For-Sale Unstable NPY5R 32 43 CC(C)c1ccccc1NC(=O)NCC1CCCCC1 ZINC000217586676 CJ On-Demand Unstable HTR4 32 42 CC(C)c1ccccc1NC(=O)NCC1CCCCC1 ZINC000217586676 CJ On-Demand Unstable DEF 0 41 CC(C)c1ccccc1NC(=O)NCC1CCCCC1 ZINC000217586676 CJ On-Demand Unstable KCNQ2 42 35 CC(C)c1ccccc1NC(=O)NCC1CCCCC1 ZINC000217586676 CJ On-Demand Unstable NMBR 37 49 CC(C)c1ccccc1NC(=O)NCC1CCCCC1 ZINC000217586676 CJ On-Demand Unstable AMY2 42 29 CC(C)c1ccccc1NC(=O)NCC1CCCCC1 ZINC000217586676 CJ On-Demand Unstable SOAT1 45 48 CC(C)c1ccccc1NC(=O)NCC1CCCCC1 ZINC000217586676 CJ On-Demand Unstable ACAT 0 58 COc1ccc(CCNc2ccc(S(=O)(=O)NCCC3=CCCCC3)cc2C(=O)O)cc1 ZINC000217586715 JI In-Stock Unstable TBXA2R 44 42 COc1ccc(CCNc2ccc(S(=O)(=O)NCCC3=CCCCC3)cc2C(=O)O)cc1 ZINC000217586715 JI In-Stock Unstable TBXAS1 15 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCCC3=CCCCC3)cc2C(=O)O)cc1 ZINC000217586715 JI In-Stock Unstable IAP 0 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCCC3=CCCCC3)cc2C(=O)O)cc1 ZINC000217586715 JI In-Stock Unstable AKR1C3 19 45 O=C(CC[C@@H]1NC(=O)N(Cc2ccccc2)C1=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217586717 ID In-Stock Unstable CHRNA4 31 58 O=C1O[C@@]2(CCCN(C(=O)Cn3cccn3)C2)c2ccccc21 ZINC000217586779 DD For-Sale Unstable NPY5R 39 43 O=C(NCC1CCCCC1)Nc1cccc(Cl)c1Cl ZINC000217586781 DJ On-Demand Unstable CXCL8 52 33 O=C(NCC1CCCCC1)Nc1cccc(Cl)c1Cl ZINC000217586781 DJ On-Demand Unstable P2RX7 16 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCCC3=CCCCC3)cc2C(=O)O)cc1OC ZINC000217586850 JI In-Stock Unstable TBXA2R 43 39 COc1ccc(CCNc2ccc(S(=O)(=O)NCCC3=CCCCC3)cc2C(=O)O)cc1OC ZINC000217586850 JI In-Stock Unstable IAP 0 42 COc1ccc(CCNc2ccc(S(=O)(=O)NCCC3=CCCCC3)cc2C(=O)O)cc1OC ZINC000217586850 JI In-Stock Unstable SCMU_MYCTU 0 41 O=C1O[C@]2(CCCN(C(=O)Cn3cccn3)C2)c2ccccc21 ZINC000217586858 DD For-Sale Unstable NPY5R 39 43 O=C(NCC1CCCCC1)Nc1cc(Cl)ccc1Cl ZINC000217586874 DJ For-Sale Unstable CNR1 15 49 O=C(NCC1CCCCC1)Nc1cc(Cl)ccc1Cl ZINC000217586874 DJ For-Sale Unstable P2RX7 25 43 O=C(NCC1CCCCC1)Nc1cc(Cl)ccc1Cl ZINC000217586874 DJ For-Sale Unstable EPHX2 23 64 O=C(NCC1CCCCC1)Nc1cc(Cl)ccc1Cl ZINC000217586874 DJ For-Sale Unstable CACNA1I 55 37 O=C(CC[C@@H]1NC(=O)N(Cc2ccco2)C1=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217586948 HD In-Stock Unstable CHRNA4 28 44 O=C1O[C@@]2(CCCN(C(=O)/C=C/c3ccc(Cl)cc3)C2)c2ccccc21 ZINC000217586953 FI For-Sale Unstable NPY5R 27 47 COc1ccc(NC(=O)NCC2CCCCC2)cc1Cl ZINC000217586995 CI On-Demand Unstable HTR4 41 44 COc1ccc(NC(=O)NCC2CCCCC2)cc1Cl ZINC000217586995 CI On-Demand Unstable PDE4A 24 42 COc1ccc(NC(=O)NCC2CCCCC2)cc1Cl ZINC000217586995 CI On-Demand Unstable CYSP_TRYCR 0 43 COc1ccc(NC(=O)NCC2CCCCC2)cc1Cl ZINC000217586995 CI On-Demand Unstable CCR3 28 42 COc1ccc(NC(=O)NCC2CCCCC2)cc1Cl ZINC000217586995 CI On-Demand Unstable GRM4 20 47 COc1ccc(NC(=O)NCC2CCCCC2)cc1Cl ZINC000217586995 CI On-Demand Unstable EPHX2 28 63 COc1ccc(NC(=O)NCC2CCCCC2)cc1Cl ZINC000217586995 CI On-Demand Unstable PDGFRA 31 45 COc1ccc(NC(=O)NCC2CCCCC2)cc1Cl ZINC000217586995 CI On-Demand Unstable MCHR1 16 41 COc1ccc(NC(=O)NCC2CCCCC2)cc1Cl ZINC000217586995 CI On-Demand Unstable CACNA1I 52 34 COc1ccc(NC(=O)NCC2CCCCC2)cc1Cl ZINC000217586995 CI On-Demand Unstable QRFPR 49 43 COc1ccc(NC(=O)NCC2CCCCC2)cc1Cl ZINC000217586995 CI On-Demand Unstable PRMT3 35 41 COc1ccc(NC(=O)NCC2CCCCC2)cc1Cl ZINC000217586995 CI On-Demand Unstable ENPP1 54 32 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217587012 JE In-Stock Unstable CHRNA4 34 44 O=C1O[C@]2(CCCN(C(=O)/C=C/c3ccc(Cl)cc3)C2)c2ccccc21 ZINC000217587033 FI For-Sale Unstable NPY5R 27 47 COc1ccc(F)cc1-c1ncnc2[nH]c(I)cc12 ZINC000217587076 FG For-Sale Unstable KIT 18 44 CCOC(=O)c1ccccc1NC(=O)NCC1CCCCC1 ZINC000217587112 DH For-Sale Unstable HCN1 40 31 CCOC(=O)c1ccccc1NC(=O)NCC1CCCCC1 ZINC000217587112 DH For-Sale Unstable HCN4 41 33 C[C@@H]1CCC[C@@]([C@@H](N)CCCc2ccccc2)(N(C)C)C1 ZINC000217587122 CH For-Sale Unstable GHRHR 40 32 O=C(O)/C=C\c1ccc(CNC(=O)c2ccccn2)cc1 ZINC000217587126 CE For-Sale Unstable GRM4 49 37 O=C(O)/C=C\c1ccc(CNC(=O)c2ccccn2)cc1 ZINC000217587126 CE For-Sale Unstable HDAC1 27 47 O=C(O)/C=C\c1ccc(CNC(=O)c2ccccn2)cc1 ZINC000217587126 CE For-Sale Unstable HDAC6 15 40 O=C(O)/C=C\c1ccc(CNC(=O)c2ccccn2)cc1 ZINC000217587126 CE For-Sale Unstable NAMPT 27 40 COc1ncccc1C(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217587127 EE In-Stock Unstable NPY5R 35 44 COc1cccc(CC(=O)NCc2nn(C3CCCC3)c3c2COCC3)c1 ZINC000217587130 FF In-Stock Unstable DRD4 42 32 O=C(O)/C=C\c1ccc(CNC(=O)c2ccncc2)cc1 ZINC000217587202 CE For-Sale Unstable NAMPT 52 40 O=C(NCC1CCCCC1)Nc1ccc(O)cc1 ZINC000217587211 BG For-Sale Unstable LDLR 0 45 O=C(NCC1CCCCC1)Nc1ccc(O)cc1 ZINC000217587211 BG For-Sale Unstable EPHX2 41 70 O=C(NCC1CCCCC1)Nc1ccc(O)cc1 ZINC000217587211 BG For-Sale Unstable NCE103 24 40 O=C(NCC1CCCCC1)Nc1ccc(O)cc1 ZINC000217587211 BG For-Sale Unstable PRMT3 36 43 COc1ncccc1C(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217587213 EE In-Stock Unstable NPY5R 35 44 O=C(O)c1cc(S(=O)(=O)NCCC2=CCCCC2)ccc1N1CCCC1 ZINC000217587236 GG In-Stock Unstable TBXA2R 45 32 Cc1noc(-c2ccc(-c3ccccc3)cc2)n1 ZINC000217587238 BH On-Demand Unstable LUCI_PHOPY 17 53 Cc1noc(-c2ccc(-c3ccccc3)cc2)n1 ZINC000217587238 BH On-Demand Unstable LUCI_PHOPE 42 53 Cc1noc(-c2ccc(-c3ccccc3)cc2)n1 ZINC000217587238 BH On-Demand Unstable SCARB1 48 32 COc1cc2c(c(OC)c1OC)-c1ccc(NCCCC(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217587287 KH In-Stock Unstable TUBA1A 15 58 COc1cc2c(c(OC)c1OC)-c1ccc(NCCCC(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217587287 KH In-Stock Unstable TPPP 0 55 O=C(O)/C=C\c1ccc(CNC(=O)c2cccnc2)cc1 ZINC000217587288 CE For-Sale Unstable TBXAS1 63 61 O=C(O)/C=C\c1ccc(CNC(=O)c2cccnc2)cc1 ZINC000217587288 CE For-Sale Unstable HDAC1 20 41 O=C(O)/C=C\c1ccc(CNC(=O)c2cccnc2)cc1 ZINC000217587288 CE For-Sale Unstable NAMPT 102 42 C[C@@H]1CCC[C@]([C@@H](N)CCCc2ccccc2)(N(C)C)C1 ZINC000217587295 CH For-Sale Unstable GHRHR 40 32 O=C1O[C@@]2(CCCN(C(=O)c3ccc4[nH]ccc4c3)C2)c2ccccc21 ZINC000217587320 EG For-Sale Unstable NPY5R 30 44 O=C(Cl)c1cnc(Cl)nc1C(F)F ZINC000217587332 BE In-Stock Reactive ATF1 41 36 O=C(O)c1cc(S(=O)(=O)NCCC2=CCCCC2)ccc1N1CCCCC1 ZINC000217587336 GH In-Stock Unstable TBXA2R 42 34 COc1ccc(Cl)cc1NC(=O)NCC1CCCCC1 ZINC000217587337 CI On-Demand Unstable HTR4 19 53 COc1ccc(Cl)cc1NC(=O)NCC1CCCCC1 ZINC000217587337 CI On-Demand Unstable CYSP_TRYCR 0 43 COc1ccc(Cl)cc1NC(=O)NCC1CCCCC1 ZINC000217587337 CI On-Demand Unstable COLA 40 34 COc1ccc(Cl)cc1NC(=O)NCC1CCCCC1 ZINC000217587337 CI On-Demand Unstable PYGL 31 44 COc1ccc(Cl)cc1NC(=O)NCC1CCCCC1 ZINC000217587337 CI On-Demand Unstable RBP4 27 47 COc1ccc(Cl)cc1NC(=O)NCC1CCCCC1 ZINC000217587337 CI On-Demand Unstable STK17B 40 36 COc1ccc(Cl)cc1NC(=O)NCC1CCCCC1 ZINC000217587337 CI On-Demand Unstable CACNA1I 47 34 COc1ccc(Cl)cc1NC(=O)NCC1CCCCC1 ZINC000217587337 CI On-Demand Unstable QRFPR 50 40 COc1ccc(Cl)cc1NC(=O)NCC1CCCCC1 ZINC000217587337 CI On-Demand Unstable METAP2 0 44 CCCCCC(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217587370 CF For-Sale Unstable CNR1 24 55 CCCCCC(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217587370 CF For-Sale Unstable PTGER2 0 42 CCCCCC(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217587370 CF For-Sale Unstable TRPV1 0 50 CCCCCC(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217587370 CF For-Sale Unstable HDAC1 22 41 CCCCCC(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217587370 CF For-Sale Unstable HDAC4 15 41 CCCCCC(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217587370 CF For-Sale Unstable HDAC6 22 41 CCCCCC(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217587370 CF For-Sale Unstable HDAC9 20 41 CCCCCC(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217587370 CF For-Sale Unstable HDAC7 27 41 CCCCCC(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217587370 CF For-Sale Unstable AKR1C3 40 46 O=C1O[C@]2(CCCN(C(=O)c3ccc4[nH]ccc4c3)C2)c2ccccc21 ZINC000217587390 EG For-Sale Unstable NPY5R 30 44 CC[S@@](=O)CCNc1ccnc(NN)n1 ZINC000217587401 BB For-Sale Unstable HRH4 21 42 CC(C)C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217587444 BE For-Sale Unstable PTGER2 35 46 CC(C)C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217587444 BE For-Sale Unstable ANPEP 27 44 CC(C)C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217587444 BE For-Sale Unstable PTGER4 0 40 CC(C)C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217587444 BE For-Sale Unstable NR1H4 29 40 CC(C)C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217587444 BE For-Sale Unstable HDAC1 16 40 CC(C)C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217587444 BE For-Sale Unstable FURIN 41 33 CC(C)C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217587444 BE For-Sale Unstable AMP1_PLAFQ 58 41 CC(C)C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217587444 BE For-Sale Unstable AKR1C3 42 44 CC(C)C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217587444 BE For-Sale Unstable CARM1 45 37 CC(C)C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217587444 BE For-Sale Unstable PDS 48 34 CCCCc1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217587454 CJ For-Sale Unstable CCR3 52 40 CCCCc1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217587454 CJ For-Sale Unstable SCN2A 15 49 CCCCc1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217587454 CJ For-Sale Unstable MMP2 52 33 CCCCc1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217587454 CJ For-Sale Unstable CFTR 46 39 CCCCc1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217587454 CJ For-Sale Unstable EPHX2 32 63 CCCCc1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217587454 CJ For-Sale Unstable SPHK1 33 46 CCCCc1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217587454 CJ For-Sale Unstable PRMT3 41 40 CCCCc1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217587454 CJ For-Sale Unstable ACAT 0 48 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](C)C(=O)NC[C@@H]3C[C@H]4C=C[C@@H]3C4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217587467 KH In-Stock Unstable TUBA1A 17 62 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](C)C(=O)NC[C@@H]3C[C@H]4C=C[C@@H]3C4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217587467 KH In-Stock Unstable TPPP 0 58 CC[S@](=O)CCNc1ccnc(NN)n1 ZINC000217587490 BB For-Sale Unstable HRH4 21 42 O=C1O[C@@]2(CCCN(C(=O)c3ccc4cc[nH]c4c3)C2)c2ccccc21 ZINC000217587504 EG For-Sale Unstable NPY5R 31 44 FC(F)(F)c1cnn(-c2ncccc2Cl)c1 ZINC000217587533 BF For-Sale Anodyne TRPV1 16 43 CC(C)(C)C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217587538 CE For-Sale Unstable HDAC6 28 43 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](C)C(=O)NC[C@@H]3C[C@@H]4C=C[C@@H]3C4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217587546 KH In-Stock Unstable TUBA1A 17 62 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](C)C(=O)NC[C@@H]3C[C@@H]4C=C[C@@H]3C4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217587546 KH In-Stock Unstable TPPP 0 58 O=C(NCc1nn(C2CCCC2)c2c1COCC2)c1cccc(C(F)(F)F)c1 ZINC000217587549 GI In-Stock Unstable CCR2 85 45 O=C1O[C@]2(CCCN(C(=O)c3ccc4cc[nH]c4c3)C2)c2ccccc21 ZINC000217587580 EG For-Sale Unstable NPY5R 31 44 CC(C)N(Cc1ccccc1)C(=O)NCC1CCCCC1 ZINC000217587589 CI On-Demand Unstable F2 28 43 CC(C)N(Cc1ccccc1)C(=O)NCC1CCCCC1 ZINC000217587589 CI On-Demand Unstable ACE 47 39 CC(C)N(Cc1ccccc1)C(=O)NCC1CCCCC1 ZINC000217587589 CI On-Demand Unstable FKBP1A 42 38 CC(C)N(Cc1ccccc1)C(=O)NCC1CCCCC1 ZINC000217587589 CI On-Demand Unstable PGC 36 40 CC(C)N(Cc1ccccc1)C(=O)NCC1CCCCC1 ZINC000217587589 CI On-Demand Unstable CTSB 34 40 CC(C)N(Cc1ccccc1)C(=O)NCC1CCCCC1 ZINC000217587589 CI On-Demand Unstable CTSL 23 40 CC(C)N(Cc1ccccc1)C(=O)NCC1CCCCC1 ZINC000217587589 CI On-Demand Unstable CACNA1B 47 37 CC(C)N(Cc1ccccc1)C(=O)NCC1CCCCC1 ZINC000217587589 CI On-Demand Unstable PGA 23 40 CC(C)N(Cc1ccccc1)C(=O)NCC1CCCCC1 ZINC000217587589 CI On-Demand Unstable AMY2 48 33 CC(C)N(Cc1ccccc1)C(=O)NCC1CCCCC1 ZINC000217587589 CI On-Demand Unstable MMP3 23 44 CC(C)N(Cc1ccccc1)C(=O)NCC1CCCCC1 ZINC000217587589 CI On-Demand Unstable REN 76 38 CC(C)N(Cc1ccccc1)C(=O)NCC1CCCCC1 ZINC000217587589 CI On-Demand Unstable CAPN1 35 44 CC(C)N(Cc1ccccc1)C(=O)NCC1CCCCC1 ZINC000217587589 CI On-Demand Unstable CAPN2 45 44 CC(C)N(Cc1ccccc1)C(=O)NCC1CCCCC1 ZINC000217587589 CI On-Demand Unstable POL 0 44 CC(C)N(Cc1ccccc1)C(=O)NCC1CCCCC1 ZINC000217587589 CI On-Demand Unstable NPR 45 33 CC(C)N(Cc1ccccc1)C(=O)NCC1CCCCC1 ZINC000217587589 CI On-Demand Unstable PTGES 23 47 CC(C)N(Cc1ccccc1)C(=O)NCC1CCCCC1 ZINC000217587589 CI On-Demand Unstable LIMK2 41 35 CC(C)N(Cc1ccccc1)C(=O)NCC1CCCCC1 ZINC000217587589 CI On-Demand Unstable METAP2 22 40 CCCCC(=O)N(C)Cc1ccc(/C=C\C(=O)O)cc1 ZINC000217587622 CF For-Sale Unstable AKR1C3 34 41 COc1cc2c(c(OC)c1OC)-c1ccc(NCCCC(=O)NC[C@@H]3C[C@H]4C=C[C@@H]3C4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217587639 KI In-Stock Unstable TUBA1A 16 61 CN(C(=O)NCC1CCCCC1)C1CCCCC1 ZINC000217587668 CH On-Demand Unstable ADH4 0 41 O=C1O[C@@]2(CCCN(C(=O)CCCc3ccccc3)C2)c2ccccc21 ZINC000217587676 EH For-Sale Unstable GHRHR 43 35 O=C1O[C@@]2(CCCN(C(=O)CCCc3ccccc3)C2)c2ccccc21 ZINC000217587676 EH For-Sale Unstable PREP 48 43 O=C1O[C@@]2(CCCN(C(=O)CCCc3ccccc3)C2)c2ccccc21 ZINC000217587676 EH For-Sale Unstable NPY5R 27 43 C[C@@H]1Oc2ccccc2N(CC(=O)N2CCN([C@@H](C#N)c3ccccc3)CC2)C1=O ZINC000217587683 HE On-Demand Unstable PTAFR 54 49 CN(Cc1ccc(/C=C\C(=O)O)cc1)C(=O)c1ccco1 ZINC000217587713 CF For-Sale Unstable NR1H4 18 48 COc1cc2c(c(OC)c1OC)-c1ccc(NCCCC(=O)NC[C@@H]3C[C@@H]4C=C[C@@H]3C4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217587719 KI In-Stock Unstable TUBA1A 16 61 O=C1O[C@]2(CCCN(C(=O)CCCc3ccccc3)C2)c2ccccc21 ZINC000217587742 EH For-Sale Unstable GHRHR 43 35 O=C1O[C@]2(CCCN(C(=O)CCCc3ccccc3)C2)c2ccccc21 ZINC000217587742 EH For-Sale Unstable PREP 48 43 O=C1O[C@]2(CCCN(C(=O)CCCc3ccccc3)C2)c2ccccc21 ZINC000217587742 EH For-Sale Unstable NPY5R 27 43 O=c1cc(C(F)F)[nH]c(=O)[nH]1 ZINC000217587755 AC In-Stock Anodyne TOPB 48 36 C[C@H]1Oc2ccccc2N(CC(=O)N2CCN([C@@H](C#N)c3ccccc3)CC2)C1=O ZINC000217587771 HE On-Demand Unstable PTAFR 54 49 O=C(NCC1CCCCC1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217587799 GJ For-Sale Unstable CHRM1 15 43 O=C(NCC1CCCCC1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217587799 GJ For-Sale Unstable CNR1 17 70 O=C(NCC1CCCCC1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217587799 GJ For-Sale Unstable OPRL1 23 46 O=C(NCC1CCCCC1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217587799 GJ For-Sale Unstable NPY2R 23 41 O=C(NCC1CCCCC1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217587799 GJ For-Sale Unstable AMY2 42 29 O=C(NCC1CCCCC1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217587799 GJ For-Sale Unstable EPHX2 22 41 O=C(NCC1CCCCC1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217587799 GJ For-Sale Unstable SMO 16 42 O=C(NCC1CCCCC1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217587799 GJ For-Sale Unstable NMUR2 0 63 O=C(NCC1CCCCC1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217587799 GJ For-Sale Unstable NMUR1 0 63 C[C@@H]1Oc2ccccc2N(CC(=O)N2CCN([C@H](C#N)c3ccccc3)CC2)C1=O ZINC000217587848 HE On-Demand Unstable PTAFR 54 49 COc1cc2c(c(OC)c1OC)-c1ccc(NCCCCCC(=O)NC[C@@H]3C[C@H]4C=C[C@@H]3C4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217587857 KK In-Stock Unstable TUBA1A 16 59 O=c1[nH]c(C(F)F)c(Br)c(=O)[nH]1 ZINC000217587864 BC In-Stock Anodyne DEOA 15 46 COc1ccc(OCC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217587870 FF For-Sale Unstable COLA 55 37 COc1ccc(OCC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217587870 FF For-Sale Unstable CPT1A 47 37 COc1ccc(OCC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217587870 FF For-Sale Unstable NPY5R 28 45 C[C@H]1Oc2ccccc2N(CC(=O)N2CCN([C@H](C#N)c3ccccc3)CC2)C1=O ZINC000217587932 HE On-Demand Unstable PTAFR 54 49 COc1cc2c(c(OC)c1OC)-c1ccc(NCCCCCC(=O)NC[C@@H]3C[C@@H]4C=C[C@@H]3C4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217587933 KK In-Stock Unstable TUBA1A 16 59 CN1CCC[C@@H](CNC(=O)C[C@@H](N)c2ccccc2)C1 ZINC000217587937 CD On-Demand Unstable F2 32 43 CN1CCC[C@@H](CNC(=O)C[C@@H](N)c2ccccc2)C1 ZINC000217587937 CD On-Demand Unstable SLC6A3 24 42 CN1CCC[C@@H](CNC(=O)C[C@@H](N)c2ccccc2)C1 ZINC000217587937 CD On-Demand Unstable DPP4 22 41 CN1CCC[C@@H](CNC(=O)C[C@@H](N)c2ccccc2)C1 ZINC000217587937 CD On-Demand Unstable CACNA1I 41 34 COc1ccc(OCC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217587946 FF For-Sale Unstable COLA 55 37 COc1ccc(OCC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217587946 FF For-Sale Unstable CPT1A 47 37 COc1ccc(OCC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217587946 FF For-Sale Unstable NPY5R 28 45 O=C(NCC1CCCCC1)N1CCCc2ccccc21 ZINC000217587988 CH For-Sale Unstable AVPR2 46 45 O=C(NCC1CCCCC1)N1CCCc2ccccc21 ZINC000217587988 CH For-Sale Unstable AVPR1A 23 42 CN1CCC[C@H](CNC(=O)C[C@@H](N)c2ccccc2)C1 ZINC000217588021 CD On-Demand Unstable F2 32 43 CN1CCC[C@H](CNC(=O)C[C@@H](N)c2ccccc2)C1 ZINC000217588021 CD On-Demand Unstable SLC6A3 24 42 CN1CCC[C@H](CNC(=O)C[C@@H](N)c2ccccc2)C1 ZINC000217588021 CD On-Demand Unstable DPP4 22 41 CN1CCC[C@H](CNC(=O)C[C@@H](N)c2ccccc2)C1 ZINC000217588021 CD On-Demand Unstable CACNA1I 41 34 O=C1O[C@@]2(CCCN(C(=O)Cc3ccc(Br)cc3)C2)c2ccccc21 ZINC000217588048 HH For-Sale Unstable NPY5R 25 40 CCn1cc(C(=O)O)c(=O)c2cc(F)c(N3CCN(C(=S)N[C@@H]4C[C@@H]5C=C[C@@H]4C5)CC3)cc21 ZINC000217588053 JF In-Stock Unstable POLC 26 45 CCn1cc(C(=O)O)c(=O)c2cc(F)c(N3CCN(C(=S)N[C@@H]4C[C@@H]5C=C[C@@H]4C5)CC3)cc21 ZINC000217588053 JF In-Stock Unstable G 0 46 CCn1cc(C(=O)O)c(=O)c2cc(F)c(N3CCN(C(=S)N[C@@H]4C[C@@H]5C=C[C@@H]4C5)CC3)cc21 ZINC000217588053 JF In-Stock Unstable ATP6V1B2 0 40 CCn1cc(C(=O)O)c(=O)c2cc(F)c(N3CCN(C(=S)N[C@@H]4C[C@@H]5C=C[C@@H]4C5)CC3)cc21 ZINC000217588053 JF In-Stock Unstable ICL 0 56 O=C(CC[C@@H]1NC(=O)N(Cc2ccccc2Cl)C1=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217588069 JE In-Stock Unstable CHRNA4 28 47 O=C(NCc1ccccc1Cl)NCC1CCCCC1 ZINC000217588109 CH On-Demand Unstable GRIN2B 15 40 O=C(NCc1ccccc1Cl)NCC1CCCCC1 ZINC000217588109 CH On-Demand Unstable P2RX7 47 39 O=C(NCc1ccccc1Cl)NCC1CCCCC1 ZINC000217588109 CH On-Demand Unstable EPHX2 24 40 O=C(NCc1ccccc1Cl)NCC1CCCCC1 ZINC000217588109 CH On-Demand Unstable Q2TU57_MAIZE 15 57 CCn1cc(C(=O)O)c(=O)c2cc(F)c(N3CCN(C(=S)N[C@H]4C[C@@H]5C=C[C@@H]4C5)CC3)cc21 ZINC000217588141 JF In-Stock Unstable POLC 26 45 CCn1cc(C(=O)O)c(=O)c2cc(F)c(N3CCN(C(=S)N[C@H]4C[C@@H]5C=C[C@@H]4C5)CC3)cc21 ZINC000217588141 JF In-Stock Unstable G 0 46 CCn1cc(C(=O)O)c(=O)c2cc(F)c(N3CCN(C(=S)N[C@H]4C[C@@H]5C=C[C@@H]4C5)CC3)cc21 ZINC000217588141 JF In-Stock Unstable ATP6V1B2 0 40 CCn1cc(C(=O)O)c(=O)c2cc(F)c(N3CCN(C(=S)N[C@H]4C[C@@H]5C=C[C@@H]4C5)CC3)cc21 ZINC000217588141 JF In-Stock Unstable ICL 0 56 O=C1O[C@]2(CCCN(C(=O)Cc3ccc(Br)cc3)C2)c2ccccc21 ZINC000217588146 HH For-Sale Unstable NPY5R 25 40 CO[C@@H]1[C@H]2CC[C@@H]1CN(C(=O)c1ccc3c(c1)nc(C)n3-c1ccccc1)C2 ZINC000217588158 GH In-Stock Unstable HPD 45 36 CO[C@@H]1[C@H]2CC[C@@H]1CN(C(=O)c1ccc3c(c1)nc(C)n3-c1ccccc1)C2 ZINC000217588158 GH In-Stock Unstable HPGD 48 40 O=C(CC[C@@H]1NC(=O)N(CCc2cccc(F)c2)C1=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217588221 JD In-Stock Unstable CHRNA4 30 49 CCn1cc(C(=O)O)c(=O)c2cc(F)c(N3CCN(C(=S)N[C@@H]4C[C@H]5C=C[C@@H]4C5)CC3)cc21 ZINC000217588227 JF In-Stock Unstable POLC 26 45 CCn1cc(C(=O)O)c(=O)c2cc(F)c(N3CCN(C(=S)N[C@@H]4C[C@H]5C=C[C@@H]4C5)CC3)cc21 ZINC000217588227 JF In-Stock Unstable G 0 46 CCn1cc(C(=O)O)c(=O)c2cc(F)c(N3CCN(C(=S)N[C@@H]4C[C@H]5C=C[C@@H]4C5)CC3)cc21 ZINC000217588227 JF In-Stock Unstable ATP6V1B2 0 40 CCn1cc(C(=O)O)c(=O)c2cc(F)c(N3CCN(C(=S)N[C@@H]4C[C@H]5C=C[C@@H]4C5)CC3)cc21 ZINC000217588227 JF In-Stock Unstable ICL 0 56 CCCCOCCCNC(=O)NCC1CCCCC1 ZINC000217588229 CG On-Demand Unstable EPHX2 0 48 CC[C@@H](C)c1ccccc1OC/C=C\CN ZINC000217588244 BG For-Sale Unstable AO-ACHE 0 44 Cn1cc(CC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c2ccccc21 ZINC000217588254 FG For-Sale Unstable PRKCG 41 34 Cn1cc(CC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c2ccccc21 ZINC000217588254 FG For-Sale Unstable NPY5R 23 40 CC(C)N(C)S(=O)(=O)c1ccc(C(=O)N2CCN([C@@H](C#N)c3ccccc3)CC2)cc1 ZINC000217588257 IF On-Demand Unstable PTAFR 53 48 CCn1cc(C(=O)O)c(=O)c2cc(F)c(N3CCN(C(=S)N[C@H]4C[C@H]5C=C[C@@H]4C5)CC3)cc21 ZINC000217588305 JF In-Stock Unstable POLC 26 45 CCn1cc(C(=O)O)c(=O)c2cc(F)c(N3CCN(C(=S)N[C@H]4C[C@H]5C=C[C@@H]4C5)CC3)cc21 ZINC000217588305 JF In-Stock Unstable G 0 46 CCn1cc(C(=O)O)c(=O)c2cc(F)c(N3CCN(C(=S)N[C@H]4C[C@H]5C=C[C@@H]4C5)CC3)cc21 ZINC000217588305 JF In-Stock Unstable ATP6V1B2 0 40 CCn1cc(C(=O)O)c(=O)c2cc(F)c(N3CCN(C(=S)N[C@H]4C[C@H]5C=C[C@@H]4C5)CC3)cc21 ZINC000217588305 JF In-Stock Unstable ICL 0 56 C[C@@H](C(=O)NCc1cc(COc2ccccc2)cs1)n1cncn1 ZINC000217588312 EF In-Stock Unstable CARM1 58 38 Cn1cc(CC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c2ccccc21 ZINC000217588332 FG For-Sale Unstable PRKCG 41 34 Cn1cc(CC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c2ccccc21 ZINC000217588332 FG For-Sale Unstable NPY5R 23 40 CC[C@H](C)c1ccccc1OC/C=C\CN ZINC000217588335 BG For-Sale Unstable AO-ACHE 0 44 CC(C)N(C)S(=O)(=O)c1ccc(C(=O)N2CCN([C@H](C#N)c3ccccc3)CC2)cc1 ZINC000217588340 IF On-Demand Unstable PTAFR 53 48 O=C(NCC1CCCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217588345 DI For-Sale Unstable F2 20 43 O=C(NCC1CCCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217588345 DI For-Sale Unstable CHRM2 27 41 O=C(NCC1CCCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217588345 DI For-Sale Unstable FKBP1A 41 38 O=C(NCC1CCCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217588345 DI For-Sale Unstable ACHE 25 42 O=C(NCC1CCCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217588345 DI For-Sale Unstable GRIN1 0 40 O=C(NCC1CCCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217588345 DI For-Sale Unstable HTR4 44 41 O=C(NCC1CCCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217588345 DI For-Sale Unstable GRIN2B 110 47 O=C(NCC1CCCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217588345 DI For-Sale Unstable SIGMAR1 43 47 O=C(NCC1CCCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217588345 DI For-Sale Unstable CCR3 69 48 O=C(NCC1CCCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217588345 DI For-Sale Unstable CCR5 17 42 O=C(NCC1CCCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217588345 DI For-Sale Unstable F2R 0 41 O=C(NCC1CCCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217588345 DI For-Sale Unstable C3AR1 44 38 O=C(NCC1CCCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217588345 DI For-Sale Unstable PREP 46 38 O=C(NCC1CCCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217588345 DI For-Sale Unstable REN 64 39 O=C(NCC1CCCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217588345 DI For-Sale Unstable CTSS 39 41 O=C(NCC1CCCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217588345 DI For-Sale Unstable CAPN1 28 44 O=C(NCC1CCCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217588345 DI For-Sale Unstable CAPN2 28 44 O=C(NCC1CCCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217588345 DI For-Sale Unstable EPHX2 44 42 O=C(NCC1CCCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217588345 DI For-Sale Unstable GRIN2C 20 40 O=C(NCC1CCCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217588345 DI For-Sale Unstable GRIN3A 0 42 O=C(NCC1CCCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217588345 DI For-Sale Unstable AMP1_PLAFQ 22 51 O=C(NCC1CCCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217588345 DI For-Sale Unstable CACNA1I 57 36 O=C(NCC1CCCCC1)N1CCC(Cc2ccccc2)CC1 ZINC000217588345 DI For-Sale Unstable SMO 23 44 COc1ccc(CN2C(=O)N[C@@H](CC(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)C2=O)cc1 ZINC000217588374 JD In-Stock Unstable CHRNA4 28 47 CCCNc1ccc(S(=O)(=O)NCCO)cc1C(=O)O ZINC000217588382 DC In-Stock Unstable CASP3 15 42 CCCNc1ccc(S(=O)(=O)NCCO)cc1C(=O)O ZINC000217588382 DC In-Stock Unstable BDKRB1 0 41 C[C@H](C(=O)NCc1cc(COc2ccccc2)cs1)n1cncn1 ZINC000217588384 EF In-Stock Unstable CARM1 58 38 O=C1O[C@@]2(CCCN(C(=O)Cn3cccc3)C2)c2ccccc21 ZINC000217588440 DE For-Sale Unstable NPY5R 27 41 CC(C)Nc1ccc(S(=O)(=O)NCCO)cc1C(=O)O ZINC000217588485 DC In-Stock Unstable CASP3 23 40 CC(C)Nc1ccc(S(=O)(=O)NCCO)cc1C(=O)O ZINC000217588485 DC In-Stock Unstable CHUK 17 41 COc1cc2c(cc1OC)CN(C(=O)c1ccc(NC(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)cc1)CC2 ZINC000217588510 KH In-Stock Unstable CHRNA4 31 41 O=C1O[C@]2(CCCN(C(=O)Cn3cccc3)C2)c2ccccc21 ZINC000217588535 DE For-Sale Unstable NPY5R 27 41 COc1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217588538 CG On-Demand Unstable BMP1 24 40 COc1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217588538 CG On-Demand Unstable MTR1B_CHICK 0 41 COc1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217588538 CG On-Demand Unstable CCR3 26 41 COc1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217588538 CG On-Demand Unstable MTNR1A 44 36 COc1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217588538 CG On-Demand Unstable MTNR1B 64 38 COc1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217588538 CG On-Demand Unstable MMP2 48 34 COc1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217588538 CG On-Demand Unstable MMP3 25 41 COc1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217588538 CG On-Demand Unstable MMP1 32 42 COc1ccc(O[C@@H]2C(=O)N(C[C@H]3CCCO3)[C@@H]2c2ccc3c(c2)OCO3)cc1 ZINC000217588549 GF In-Stock Unstable EDNRB 60 40 COc1ccc(O[C@@H]2C(=O)N(C[C@H]3CCCO3)[C@@H]2c2ccc3c(c2)OCO3)cc1 ZINC000217588549 GF In-Stock Unstable EDNRA 61 39 COc1ccc(O[C@@H]2C(=O)N(C[C@H]3CCCO3)[C@@H]2c2ccc3c(c2)OCO3)cc1 ZINC000217588549 GF In-Stock Unstable SCN9A 0 50 COc1cc2c(cc1OC)CN(C(=O)c1ccc(NC(=O)N3C[C@H]4C[C@H](C3)c3cccc(=O)n3C4)cc1)CC2 ZINC000217588593 KH In-Stock Unstable CHRNA4 31 41 CCCCNc1ccc(S(=O)(=O)NCCO)cc1C(=O)O ZINC000217588594 DC In-Stock Unstable CASP3 16 43 CCCCNc1ccc(S(=O)(=O)NCCO)cc1C(=O)O ZINC000217588594 DC In-Stock Unstable BDKRB1 0 42 CN(CCO)CC(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217588603 CD On-Demand Unstable FAP 0 40 O=C(NCc1ccc(Cl)cc1)NCC1CCCCC1 ZINC000217588652 CH On-Demand Unstable SLC6A1 39 44 O=C(NCc1ccc(Cl)cc1)NCC1CCCCC1 ZINC000217588652 CH On-Demand Unstable P2RX7 17 43 O=C(NCc1ccc(Cl)cc1)NCC1CCCCC1 ZINC000217588652 CH On-Demand Unstable CCR1 15 45 O=C(NCc1ccc(Cl)cc1)NCC1CCCCC1 ZINC000217588652 CH On-Demand Unstable EPHX2 17 42 O=C(NCc1ccc(Cl)cc1)NCC1CCCCC1 ZINC000217588652 CH On-Demand Unstable TPSAB1 16 40 O=C(NCc1ccc(Cl)cc1)NCC1CCCCC1 ZINC000217588652 CH On-Demand Unstable PROC 44 33 O=C(NCc1ccc(Cl)cc1)NCC1CCCCC1 ZINC000217588652 CH On-Demand Unstable CACNA1I 49 35 O=C1O[C@@]2(CCCN(C(=O)c3cncc(Br)c3)C2)c2ccccc21 ZINC000217588659 GG In-Stock Unstable NPY5R 38 42 CC(C)CNc1ccc(S(=O)(=O)NCCO)cc1C(=O)O ZINC000217588701 DC In-Stock Unstable CASP3 18 42 CC(C)CNc1ccc(S(=O)(=O)NCCO)cc1C(=O)O ZINC000217588701 DC In-Stock Unstable BDKRB1 0 46 CC(C)CNc1ccc(S(=O)(=O)NCCO)cc1C(=O)O ZINC000217588701 DC In-Stock Unstable MTNN 51 32 COc1ccc(CN2C(=O)N[C@@H](CC(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)C2=O)cc1OC ZINC000217588704 JD In-Stock Unstable CHRNA4 26 43 CN(CCO)CC(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217588705 CD On-Demand Unstable FAP 0 40 O=C1O[C@]2(CCCN(C(=O)c3cncc(Br)c3)C2)c2ccccc21 ZINC000217588729 GG In-Stock Unstable NPY5R 38 42 CN1CCC[C@@H](CNC(=O)[C@@H]2NCCc3ccccc32)C1 ZINC000217588734 CD On-Demand Unstable PRCP 41 33 C[C@@H](NC(=O)NCC1CCCCC1)c1ccccc1 ZINC000217588756 CH On-Demand Unstable CTSB 29 42 C[C@@H](NC(=O)NCC1CCCCC1)c1ccccc1 ZINC000217588756 CH On-Demand Unstable CTSK 53 37 C[C@@H](NC(=O)NCC1CCCCC1)c1ccccc1 ZINC000217588756 CH On-Demand Unstable NMBR 18 40 C[C@@H](NC(=O)NCC1CCCCC1)c1ccccc1 ZINC000217588756 CH On-Demand Unstable AMY2 48 33 C[C@@H](NC(=O)NCC1CCCCC1)c1ccccc1 ZINC000217588756 CH On-Demand Unstable REN 46 36 C[C@@H](NC(=O)NCC1CCCCC1)c1ccccc1 ZINC000217588756 CH On-Demand Unstable CTSS 24 42 C[C@@H](NC(=O)NCC1CCCCC1)c1ccccc1 ZINC000217588756 CH On-Demand Unstable CAPN1 37 46 C[C@@H](NC(=O)NCC1CCCCC1)c1ccccc1 ZINC000217588756 CH On-Demand Unstable CAPN2 53 46 C[C@@H](NC(=O)NCC1CCCCC1)c1ccccc1 ZINC000217588756 CH On-Demand Unstable PROTEASE 0 41 C[C@@H](NC(=O)NCC1CCCCC1)c1ccccc1 ZINC000217588756 CH On-Demand Unstable XIAP 44 36 C[C@@H](NC(=O)NCC1CCCCC1)c1ccccc1 ZINC000217588756 CH On-Demand Unstable BIRC8 42 34 O=C(O)/C=C\c1cccc(CNC(=O)c2ccccc2)c1 ZINC000217588795 CF For-Sale Unstable PTGER2 34 43 O=C(O)/C=C\c1cccc(CNC(=O)c2ccccc2)c1 ZINC000217588795 CF For-Sale Unstable GRIN2B 0 48 O=C(O)/C=C\c1cccc(CNC(=O)c2ccccc2)c1 ZINC000217588795 CF For-Sale Unstable PTGER4 0 43 O=C(O)/C=C\c1cccc(CNC(=O)c2ccccc2)c1 ZINC000217588795 CF For-Sale Unstable HDAC8 40 45 O=C(O)/C=C\c1cccc(CNC(=O)c2ccccc2)c1 ZINC000217588795 CF For-Sale Unstable HDAC1 30 48 O=C(O)/C=C\c1cccc(CNC(=O)c2ccccc2)c1 ZINC000217588795 CF For-Sale Unstable HDAC2 18 51 O=C(O)/C=C\c1cccc(CNC(=O)c2ccccc2)c1 ZINC000217588795 CF For-Sale Unstable HDAC6 32 55 O=C(O)/C=C\c1cccc(CNC(=O)c2ccccc2)c1 ZINC000217588795 CF For-Sale Unstable AKR1C3 39 40 O=C(O)/C=C\c1cccc(CNC(=O)c2ccccc2)c1 ZINC000217588795 CF For-Sale Unstable KCNK3 48 36 O=C(O)/C=C\c1cccc(CNC(=O)c2ccccc2)c1 ZINC000217588795 CF For-Sale Unstable PDS 41 32 O=C(C(F)F)N1CCc2ccccc2C1 ZINC000217588809 BD On-Demand Unstable CHRNA6 0 43 O=C(C(F)F)N1CCc2ccccc2C1 ZINC000217588809 BD On-Demand Unstable DPP8 35 56 CN1CCC[C@H](CNC(=O)[C@@H]2NCCc3ccccc32)C1 ZINC000217588816 CD On-Demand Unstable PRCP 41 33 CC[C@@H](C)Nc1ccc(S(=O)(=O)NCCO)cc1C(=O)O ZINC000217588817 DC In-Stock Unstable CASP3 0 41 O=C1O[C@@]2(CCCN(C(=O)Cn3cnnn3)C2)c2ccccc21 ZINC000217588832 DC For-Sale Unstable NPY5R 26 40 C[C@H](NC(=O)NCC1CCCCC1)c1ccccc1 ZINC000217588835 CH On-Demand Unstable CTSB 29 42 C[C@H](NC(=O)NCC1CCCCC1)c1ccccc1 ZINC000217588835 CH On-Demand Unstable CTSK 53 37 C[C@H](NC(=O)NCC1CCCCC1)c1ccccc1 ZINC000217588835 CH On-Demand Unstable NMBR 18 40 C[C@H](NC(=O)NCC1CCCCC1)c1ccccc1 ZINC000217588835 CH On-Demand Unstable AMY2 48 33 C[C@H](NC(=O)NCC1CCCCC1)c1ccccc1 ZINC000217588835 CH On-Demand Unstable REN 46 36 C[C@H](NC(=O)NCC1CCCCC1)c1ccccc1 ZINC000217588835 CH On-Demand Unstable CTSS 24 42 C[C@H](NC(=O)NCC1CCCCC1)c1ccccc1 ZINC000217588835 CH On-Demand Unstable CAPN1 37 46 C[C@H](NC(=O)NCC1CCCCC1)c1ccccc1 ZINC000217588835 CH On-Demand Unstable CAPN2 53 46 C[C@H](NC(=O)NCC1CCCCC1)c1ccccc1 ZINC000217588835 CH On-Demand Unstable PROTEASE 0 41 C[C@H](NC(=O)NCC1CCCCC1)c1ccccc1 ZINC000217588835 CH On-Demand Unstable XIAP 44 36 C[C@H](NC(=O)NCC1CCCCC1)c1ccccc1 ZINC000217588835 CH On-Demand Unstable BIRC8 42 34 O=C(NCC(=O)N1CCN(CCOc2ccccc2Cl)CC1)c1ccc(Br)cc1 ZINC000217588848 JG On-Demand Unstable HTR1A 21 40 O=C(NCC(=O)N1CCN(CCOc2ccccc2Cl)CC1)c1ccc(Br)cc1 ZINC000217588848 JG On-Demand Unstable DRD2 29 40 O=C(NCC(=O)N1CCN(CCOc2ccccc2Cl)CC1)c1ccc(Br)cc1 ZINC000217588848 JG On-Demand Unstable DRD3 52 40 O=C(NCC(=O)N1CCN(CCOc2ccccc2Cl)CC1)c1ccc(Br)cc1 ZINC000217588848 JG On-Demand Unstable SCD 18 41 CC[C@H](C)Nc1ccc(S(=O)(=O)NCCO)cc1C(=O)O ZINC000217588895 DC In-Stock Unstable CASP3 0 41 O=C1O[C@]2(CCCN(C(=O)Cn3cnnn3)C2)c2ccccc21 ZINC000217588904 DC For-Sale Unstable NPY5R 26 40 CNCCc1c(Br)cccc1OC ZINC000217588927 BE For-Sale Unstable TAAR1 18 49 O=C(NCC1CCCCC1)NC(c1ccccc1)c1ccccc1 ZINC000217588932 DJ For-Sale Unstable CHRM1 16 42 O=C(NCC1CCCCC1)NC(c1ccccc1)c1ccccc1 ZINC000217588932 DJ For-Sale Unstable CHRM3 15 42 O=C(NCC1CCCCC1)NC(c1ccccc1)c1ccccc1 ZINC000217588932 DJ For-Sale Unstable AMY2 47 32 O=C(NCC1CCCCC1)NC(c1ccccc1)c1ccccc1 ZINC000217588932 DJ For-Sale Unstable CTSS 22 41 O=C(NCC1CCCCC1)NC(c1ccccc1)c1ccccc1 ZINC000217588932 DJ For-Sale Unstable EPHX2 15 52 O=C(NCC1CCCCC1)NC(c1ccccc1)c1ccccc1 ZINC000217588932 DJ For-Sale Unstable XIAP 50 37 O=C(NCC1CCCCC1)NC(c1ccccc1)c1ccccc1 ZINC000217588932 DJ For-Sale Unstable BIRC8 56 35 O=C(NCC1CCCCC1)NC(c1ccccc1)c1ccccc1 ZINC000217588932 DJ For-Sale Unstable METAP2 24 44 CN(Cc1ccc(/C=C\C(=O)O)cc1)C(=O)C1CCC1 ZINC000217588976 CF For-Sale Unstable NR1H4 36 45 O=C(NCC(=O)N1CCN(CCOc2ccccc2Cl)CC1)c1cccc(F)c1 ZINC000217588982 HE On-Demand Unstable HTR1A 34 42 O=C(NCC(=O)N1CCN(CCOc2ccccc2Cl)CC1)c1cccc(F)c1 ZINC000217588982 HE On-Demand Unstable DRD2 45 44 O=C(NCC(=O)N1CCN(CCOc2ccccc2Cl)CC1)c1cccc(F)c1 ZINC000217588982 HE On-Demand Unstable DRD1 19 41 O=C(NCC(=O)N1CCN(CCOc2ccccc2Cl)CC1)c1cccc(F)c1 ZINC000217588982 HE On-Demand Unstable DRD4 51 42 O=C(NCC(=O)N1CCN(CCOc2ccccc2Cl)CC1)c1cccc(F)c1 ZINC000217588982 HE On-Demand Unstable HTR2A 36 51 O=C(NCC(=O)N1CCN(CCOc2ccccc2Cl)CC1)c1cccc(F)c1 ZINC000217588982 HE On-Demand Unstable SLC6A4 20 45 O=C(NCC(=O)N1CCN(CCOc2ccccc2Cl)CC1)c1cccc(F)c1 ZINC000217588982 HE On-Demand Unstable DRD3 60 44 O=C(NCC(=O)N1CCN(CCOc2ccccc2Cl)CC1)c1cccc(F)c1 ZINC000217588982 HE On-Demand Unstable HTR7 34 60 O=C(NCC(=O)N1CCN(CCOc2ccccc2Cl)CC1)c1cccc(F)c1 ZINC000217588982 HE On-Demand Unstable ECR 15 41 O=C(NCC(=O)N1CCN(CCOc2ccccc2Cl)CC1)c1cccc(F)c1 ZINC000217588982 HE On-Demand Unstable CCR2 25 41 O=C(NCC(=O)N1CCN(CCOc2ccccc2Cl)CC1)c1cccc(F)c1 ZINC000217588982 HE On-Demand Unstable PLD2 47 35 O=C(NCC(=O)N1CCN(CCOc2ccccc2Cl)CC1)c1cccc(F)c1 ZINC000217588982 HE On-Demand Unstable SCD1 16 41 CC1(C)CCC(=O)/C(=N\Nc2ccc(C(=O)O)cc2)C1 ZINC000217588984 CF For-Sale Unstable RARA 44 38 CC1(C)CCC(=O)/C(=N\Nc2ccc(C(=O)O)cc2)C1 ZINC000217588984 CF For-Sale Unstable RARG 42 32 CC1(C)CCC(=O)/C(=N\Nc2ccc(C(=O)O)cc2)C1 ZINC000217588984 CF For-Sale Unstable RXRG 57 35 CC1(C)CCC(=O)/C(=N\Nc2ccc(C(=O)O)cc2)C1 ZINC000217588984 CF For-Sale Unstable RXRB 55 36 CC(C)(C)Nc1ccc(S(=O)(=O)NCCO)cc1C(=O)O ZINC000217588994 DC In-Stock Unstable CHUK 16 41 CC(C)(C)Nc1ccc(S(=O)(=O)NCCO)cc1C(=O)O ZINC000217588994 DC In-Stock Unstable PRTN3 46 37 CC(C)(C)Nc1ccc(S(=O)(=O)NCCO)cc1C(=O)O ZINC000217588994 DC In-Stock Unstable AKR1C3 20 40 O=C1O[C@@]2(CCCN(C(=O)c3cc(Br)ccc3Cl)C2)c2ccccc21 ZINC000217589015 HI In-Stock Unstable NPY5R 28 45 CN(Cc1ccc(/C=C\C(=O)O)cc1)C(=O)C1CCCC1 ZINC000217589054 CF For-Sale Unstable NR1H4 37 47 CC(=O)N1CCN(C(=O)NCC2CCCCC2)CC1 ZINC000217589069 CD For-Sale Unstable DPP7 18 40 CC(=O)N1CCN(C(=O)NCC2CCCCC2)CC1 ZINC000217589069 CD For-Sale Unstable CACNA1I 40 32 O=C1O[C@]2(CCCN(C(=O)c3cc(Br)ccc3Cl)C2)c2ccccc21 ZINC000217589090 HI In-Stock Unstable NPY5R 28 45 C=CCNc1ccc(S(=O)(=O)NCCO)cc1C(=O)O ZINC000217589093 DC In-Stock Unstable BDKRB1 0 40 CSc1ccccc1C(=O)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000217589109 GH On-Demand Unstable HTR1A 20 42 CSc1ccccc1C(=O)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000217589109 GH On-Demand Unstable DRD2 20 42 CSc1ccccc1C(=O)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000217589109 GH On-Demand Unstable THRB 27 41 CSc1ccccc1C(=O)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000217589109 GH On-Demand Unstable HTR7 23 45 O=C(O)/C=C\c1cnc(NC(=O)CCn2ccnc2)s1 ZINC000217589143 CD For-Sale Unstable TBXAS1 49 47 C[C@@H](NC(=O)NCC1CCCCC1)C12CC3CC(CC(C3)C1)C2 ZINC000217589185 DI For-Sale Unstable EPHX2 37 63 O=C(O)c1cc(S(=O)(=O)NCCO)ccc1NC1CC1 ZINC000217589197 DC In-Stock Unstable CASP3 0 41 O=C1O[C@@]2(CCCN(C(=O)c3ccc(-n4cccc4)cc3)C2)c2ccccc21 ZINC000217589198 FH In-Stock Unstable NPY5R 25 43 CCOc1cc(C(=O)N2CCN(CCOc3ccccc3Cl)CC2)cc(Cl)c1O ZINC000217589219 IH On-Demand Unstable HTR1A 21 43 CCOc1cc(C(=O)N2CCN(CCOc3ccccc3Cl)CC2)cc(Cl)c1O ZINC000217589219 IH On-Demand Unstable DRD2 20 43 CCOc1cc(C(=O)N2CCN(CCOc3ccccc3Cl)CC2)cc(Cl)c1O ZINC000217589219 IH On-Demand Unstable HTR4 28 43 C[C@H](NC(=O)NCC1CCCCC1)C12CC3CC(CC(C3)C1)C2 ZINC000217589262 DI For-Sale Unstable EPHX2 37 63 O=C1O[C@]2(CCCN(C(=O)c3ccc(-n4cccc4)cc3)C2)c2ccccc21 ZINC000217589277 FH In-Stock Unstable NPY5R 25 43 Cc1ncnc(NCC2CC2)c1I ZINC000217589280 CE In-Stock Unstable PRKCQ 43 34 O=C(O)c1cc(S(=O)(=O)NCCO)ccc1NC1CCCC1 ZINC000217589306 ED In-Stock Unstable CASP3 0 44 Cc1c(N)nc(C2CC2)nc1N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217589326 CE For-Sale Unstable CHRM3 22 46 Cc1noc(C)c1COc1ccc(CC(=O)N2CCN(CCOc3ccccc3Cl)CC2)cc1 ZINC000217589328 JI On-Demand Unstable LTA4H 40 36 Cc1noc(C)c1COc1ccc(CC(=O)N2CCN(CCOc3ccccc3Cl)CC2)cc1 ZINC000217589328 JI On-Demand Unstable NR1H4 62 37 Cc1noc(C)c1COc1ccc(CC(=O)N2CCN(CCOc3ccccc3Cl)CC2)cc1 ZINC000217589328 JI On-Demand Unstable KCNJ1 45 34 Cc1noc(C)c1COc1ccc(CC(=O)N2CCN(CCOc3ccccc3Cl)CC2)cc1 ZINC000217589328 JI On-Demand Unstable GPR183 0 41 O=C(NCC1CCCCC1)Nc1cccc2c(O)cccc12 ZINC000217589355 CI For-Sale Unstable TRPV1 35 40 O=C(NCC1CCCCC1)Nc1cccc2c(O)cccc12 ZINC000217589355 CI For-Sale Unstable NMBR 22 41 Cc1ccc(NC(=O)[C@@H]2CC[C@@H](CNC(=O)[C@@H]3Cc4ccccc4CN3)CC2)c(C)c1 ZINC000217589360 HH In-Stock Unstable EPHX2 15 40 O=C1O[C@@]2(CCCN(C(=O)CCCCc3ccccc3)C2)c2ccccc21 ZINC000217589390 FI For-Sale Unstable GHRHR 43 34 O=C1O[C@@]2(CCCN(C(=O)CCCCc3ccccc3)C2)c2ccccc21 ZINC000217589390 FI For-Sale Unstable PREP 44 42 O=C1O[C@@]2(CCCN(C(=O)CCCCc3ccccc3)C2)c2ccccc21 ZINC000217589390 FI For-Sale Unstable FAAH 42 39 O=C1O[C@@]2(CCCN(C(=O)CCCCc3ccccc3)C2)c2ccccc21 ZINC000217589390 FI For-Sale Unstable NPY5R 26 43 O=C1O[C@@]2(CCCN(C(=O)CCCCc3ccccc3)C2)c2ccccc21 ZINC000217589390 FI For-Sale Unstable CES1 51 34 NC/C=C\CN1CCN(Cc2ccccc2)CC1 ZINC000217589396 BD For-Sale Unstable DRD2 0 51 NC/C=C\CN1CCN(Cc2ccccc2)CC1 ZINC000217589396 BD For-Sale Unstable DRD4 36 40 NC/C=C\CN1CCN(Cc2ccccc2)CC1 ZINC000217589396 BD For-Sale Unstable DRD3 27 42 NC/C=C\CN1CCN(Cc2ccccc2)CC1 ZINC000217589396 BD For-Sale Unstable SIGMAR1 70 62 Cc1ncnc(NC2CC2)c1I ZINC000217589404 CD In-Stock Unstable IRAK4 16 41 O=C(O)c1cc(S(=O)(=O)NCCO)ccc1NC1CCCCC1 ZINC000217589417 ED In-Stock Unstable CASP3 0 44 O=C(O)c1cc(S(=O)(=O)NCCO)ccc1NC1CCCCC1 ZINC000217589417 ED In-Stock Unstable CHUK 17 40 Cc1c(N)nc(C2CC2)nc1N[C@H]1CCN2CCCC[C@@H]12 ZINC000217589421 CE For-Sale Unstable CHRM3 22 46 O=C(NCc1ccc(Cl)cc1)C(F)F ZINC000217589434 BE On-Demand Unstable AVPR1A 24 41 O=C(NCc1ccc(Cl)cc1)C(F)F ZINC000217589434 BE On-Demand Unstable SLC6A11 0 40 O=C(NCc1ccc(Cl)cc1)C(F)F ZINC000217589434 BE On-Demand Unstable SLC6A12 0 42 O=C(NCc1ccc(Cl)cc1)C(F)F ZINC000217589434 BE On-Demand Unstable U38 0 41 O=C(NCc1ccc(Cl)cc1)C(F)F ZINC000217589434 BE On-Demand Unstable Q76353_9HIV1 0 41 O=C(c1cc(N2CCOCC2)ccn1)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000217589459 IE On-Demand Unstable HTR2C 18 40 O=C(c1cc(N2CCOCC2)ccn1)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000217589459 IE On-Demand Unstable PRKDC 16 43 O=C1O[C@]2(CCCN(C(=O)CCCCc3ccccc3)C2)c2ccccc21 ZINC000217589478 FI For-Sale Unstable GHRHR 43 34 O=C1O[C@]2(CCCN(C(=O)CCCCc3ccccc3)C2)c2ccccc21 ZINC000217589478 FI For-Sale Unstable PREP 44 42 O=C1O[C@]2(CCCN(C(=O)CCCCc3ccccc3)C2)c2ccccc21 ZINC000217589478 FI For-Sale Unstable FAAH 42 39 O=C1O[C@]2(CCCN(C(=O)CCCCc3ccccc3)C2)c2ccccc21 ZINC000217589478 FI For-Sale Unstable NPY5R 26 43 O=C1O[C@]2(CCCN(C(=O)CCCCc3ccccc3)C2)c2ccccc21 ZINC000217589478 FI For-Sale Unstable CES1 51 34 Cc1cccc(N2CCN(C/C=C\CN)CC2)c1 ZINC000217589501 BD For-Sale Unstable HTR1A 18 59 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](CC(C)C)C(=O)NC[C@@H]3C[C@H]4C=C[C@@H]3C4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217589537 KK In-Stock Unstable TUBA1A 17 61 COc1ccc(/C=C/C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1OC ZINC000217589564 GG For-Sale Unstable NPY5R 25 44 COc1ccc([C@@H](C)NC(=O)NCC2CCCCC2)cc1OC ZINC000217589575 DH On-Demand Unstable PDE4A 31 40 COc1ccc([C@@H](C)NC(=O)NCC2CCCCC2)cc1OC ZINC000217589575 DH On-Demand Unstable STK17B 41 35 COc1ccc([C@@H](C)NC(=O)NCC2CCCCC2)cc1OC ZINC000217589575 DH On-Demand Unstable METAP2 0 42 CC[C@@H](C)[C@@H](N)C(=O)N1CCCO[C@@H](C)C1 ZINC000217589579 BC For-Sale Unstable DPP9 16 40 O=C(c1cc(N2CCCC2)ccn1)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000217589581 HG On-Demand Unstable HTR1A 47 39 O=C(c1cc(N2CCCC2)ccn1)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000217589581 HG On-Demand Unstable HTR2A 41 39 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](CC(C)C)C(=O)NC[C@@H]3C[C@@H]4C=C[C@@H]3C4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217589610 KK In-Stock Unstable TUBA1A 17 61 O=C(O)c1cc(S(=O)(=O)NCCO)ccc1NCCO ZINC000217589614 DB In-Stock Unstable CASP3 0 41 O=C(O)c1cc(S(=O)(=O)NCCO)ccc1NCCO ZINC000217589614 DB In-Stock Unstable BDKRB1 0 42 O=C(O)c1cc(S(=O)(=O)NCCO)ccc1NCCO ZINC000217589614 DB In-Stock Unstable AKR1C3 15 40 COc1ccc(/C=C/C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1OC ZINC000217589647 GG For-Sale Unstable NPY5R 25 44 CC[C@H](C)[C@@H](N)C(=O)N1CCCO[C@@H](C)C1 ZINC000217589658 BC On-Demand Unstable DPP9 0 40 COc1ccc([C@H](C)NC(=O)NCC2CCCCC2)cc1OC ZINC000217589664 DH On-Demand Unstable PDE4A 32 42 COc1ccc([C@H](C)NC(=O)NCC2CCCCC2)cc1OC ZINC000217589664 DH On-Demand Unstable STK17B 41 35 COc1ccc([C@H](C)NC(=O)NCC2CCCCC2)cc1OC ZINC000217589664 DH On-Demand Unstable METAP2 0 42 Cc1ncnc(NC2CCCCC2)c1I ZINC000217589700 DG In-Stock Unstable CD38 39 43 O=C(O)c1cc(S(=O)(=O)NCCO)ccc1NCCCO ZINC000217589722 DB In-Stock Unstable CASP3 16 40 O=C(O)c1cc(S(=O)(=O)NCCO)ccc1NCCCO ZINC000217589722 DB In-Stock Unstable BDKRB1 0 42 O=C1O[C@@]2(CCCN(C(=O)c3ccc4n[nH]nc4c3)C2)c2ccccc21 ZINC000217589742 EE For-Sale Unstable NPY5R 33 44 CSc1ccc(C(=O)Nc2ccc(Sc3nccn3C)cc2)cc1[N+](=O)[O-] ZINC000217589744 HI On-Demand Unstable GSTM2 65 36 CSc1ccc(C(=O)Nc2ccc(Sc3nccn3C)cc2)cc1[N+](=O)[O-] ZINC000217589744 HI On-Demand Unstable GCK 16 42 O=C(O)/C=C\c1ccc(CNC(=O)C2CCCCC2)cc1 ZINC000217589778 CF For-Sale Unstable NR1H4 20 41 O=C(O)/C=C\c1ccc(CNC(=O)C2CCCCC2)cc1 ZINC000217589778 CF For-Sale Unstable PROC 43 33 NC[C@@H]1CCCCN1[C@@H]1CCCCc2ccccc21 ZINC000217589779 CG For-Sale Unstable HTR3B 0 40 COc1ccc([C@@H](C)NC(=O)NCC2CCCCC2)cc1 ZINC000217589780 CH On-Demand Unstable BMP1 15 41 COc1ccc([C@@H](C)NC(=O)NCC2CCCCC2)cc1 ZINC000217589780 CH On-Demand Unstable ACACA 69 39 COc1ccc([C@@H](C)NC(=O)NCC2CCCCC2)cc1 ZINC000217589780 CH On-Demand Unstable CTSL 15 41 COc1ccc([C@@H](C)NC(=O)NCC2CCCCC2)cc1 ZINC000217589780 CH On-Demand Unstable CACNA1B 20 45 COc1ccc([C@@H](C)NC(=O)NCC2CCCCC2)cc1 ZINC000217589780 CH On-Demand Unstable MMP3 15 44 COc1ccc([C@@H](C)NC(=O)NCC2CCCCC2)cc1 ZINC000217589780 CH On-Demand Unstable CTSS 20 40 COc1ccc([C@@H](C)NC(=O)NCC2CCCCC2)cc1 ZINC000217589780 CH On-Demand Unstable F7 15 43 COc1ccc([C@@H](C)NC(=O)NCC2CCCCC2)cc1 ZINC000217589780 CH On-Demand Unstable MMP1 15 44 COc1ccc([C@@H](C)NC(=O)NCC2CCCCC2)cc1 ZINC000217589780 CH On-Demand Unstable METAP2 18 44 CC(C)(C)OC(=O)N1Cc2ccccc2C[C@H]1C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217589793 HG In-Stock Unstable OPRM1 31 45 CC(C)(C)OC(=O)N1Cc2ccccc2C[C@H]1C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217589793 HG In-Stock Unstable OPRD1 66 39 CC(C)(C)OC(=O)N1Cc2ccccc2C[C@H]1C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217589793 HG In-Stock Unstable AGTR2 51 38 CC(C)(C)OC(=O)N1Cc2ccccc2C[C@H]1C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217589793 HG In-Stock Unstable NPY2R 0 41 CC(C)(C)OC(=O)N1Cc2ccccc2C[C@H]1C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217589793 HG In-Stock Unstable HDAC8 23 46 CC(C)(C)OC(=O)N1Cc2ccccc2C[C@H]1C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217589793 HG In-Stock Unstable PREP 24 47 CC(C)(C)OC(=O)N1Cc2ccccc2C[C@H]1C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217589793 HG In-Stock Unstable CFTR 66 36 CC(C)(C)OC(=O)N1Cc2ccccc2C[C@H]1C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217589793 HG In-Stock Unstable ADAM9 63 37 Cc1ncnc(N2CCN(C)CC2)c1I ZINC000217589804 DD In-Stock Unstable HRH4 31 44 O=C1O[C@]2(CCCN(C(=O)c3ccc4n[nH]nc4c3)C2)c2ccccc21 ZINC000217589811 EE For-Sale Unstable NPY5R 33 44 COCCNc1ccc(S(=O)(=O)NCCO)cc1C(=O)O ZINC000217589843 DB In-Stock Unstable BDKRB1 0 43 COc1ccc([C@H](C)NC(=O)NCC2CCCCC2)cc1 ZINC000217589861 CH On-Demand Unstable BMP1 15 41 COc1ccc([C@H](C)NC(=O)NCC2CCCCC2)cc1 ZINC000217589861 CH On-Demand Unstable ACACA 69 39 COc1ccc([C@H](C)NC(=O)NCC2CCCCC2)cc1 ZINC000217589861 CH On-Demand Unstable CTSL 15 41 COc1ccc([C@H](C)NC(=O)NCC2CCCCC2)cc1 ZINC000217589861 CH On-Demand Unstable CACNA1B 20 45 COc1ccc([C@H](C)NC(=O)NCC2CCCCC2)cc1 ZINC000217589861 CH On-Demand Unstable MMP3 15 44 COc1ccc([C@H](C)NC(=O)NCC2CCCCC2)cc1 ZINC000217589861 CH On-Demand Unstable CTSS 20 40 COc1ccc([C@H](C)NC(=O)NCC2CCCCC2)cc1 ZINC000217589861 CH On-Demand Unstable F7 15 43 COc1ccc([C@H](C)NC(=O)NCC2CCCCC2)cc1 ZINC000217589861 CH On-Demand Unstable MMP1 15 44 COc1ccc([C@H](C)NC(=O)NCC2CCCCC2)cc1 ZINC000217589861 CH On-Demand Unstable METAP2 18 44 O=C1O[C@@]2(CCCN(C(=O)Cn3ccc4ccccc43)C2)c2ccccc21 ZINC000217589907 FG In-Stock Unstable NPY5R 27 41 O=C(O)/C=C\c1cccc(CNC(=O)c2ccccn2)c1 ZINC000217589947 CE For-Sale Unstable MMP13 16 50 O=C(O)/C=C\c1cccc(CNC(=O)c2ccccn2)c1 ZINC000217589947 CE For-Sale Unstable GRM4 57 41 O=C(O)/C=C\c1cccc(CNC(=O)c2ccccn2)c1 ZINC000217589947 CE For-Sale Unstable HDAC1 19 43 COCCCNc1ccc(S(=O)(=O)NCCO)cc1C(=O)O ZINC000217589948 EC In-Stock Unstable BDKRB1 0 44 COC(=O)c1ccccc1N(C)C(=O)c1ccc(-c2ccccc2)cc1 ZINC000217589965 EI On-Demand Unstable E1 0 41 Cc1cc(C(=O)O)ccc1N[C@@H]1C[C@@H]2CC[C@@]1(C)C2(C)C ZINC000217589966 CI For-Sale Unstable RARA 40 31 Cc1cc(C(=O)O)ccc1N[C@@H]1C[C@@H]2CC[C@@]1(C)C2(C)C ZINC000217589966 CI For-Sale Unstable RARG 41 33 Cc1cc(C(=O)O)ccc1N[C@@H]1C[C@@H]2CC[C@@]1(C)C2(C)C ZINC000217589966 CI For-Sale Unstable RXRG 48 35 Cc1cc(C(=O)O)ccc1N[C@@H]1C[C@@H]2CC[C@@]1(C)C2(C)C ZINC000217589966 CI For-Sale Unstable RXRB 47 35 O=C1O[C@]2(CCCN(C(=O)Cn3ccc4ccccc43)C2)c2ccccc21 ZINC000217589985 FG In-Stock Unstable NPY5R 27 41 CN(Cc1ccc(/C=C\C(=O)O)cc1)C(=O)c1cccs1 ZINC000217590014 DG For-Sale Unstable HSD17B2 29 46 CN1CCN(c2ncnc(C(F)(F)F)c2I)CC1 ZINC000217590017 FD In-Stock Unstable HRH4 18 41 COc1ccccc1CCN1C(=O)N[C@@H](CCC(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)C1=O ZINC000217590021 JD In-Stock Unstable CHRNA4 28 45 CC(C)(C)OC(=O)N1Cc2ccccc2C[C@H]1C(=O)NC[C@@H]1CC[C@@H](C(=O)NC2CCCCC2)CC1 ZINC000217590042 JJ In-Stock Unstable OPRM1 23 42 CC(C)(C)OC(=O)N1Cc2ccccc2C[C@H]1C(=O)NC[C@@H]1CC[C@@H](C(=O)NC2CCCCC2)CC1 ZINC000217590042 JJ In-Stock Unstable OPRD1 49 36 CC(C)(C)OC(=O)N1Cc2ccccc2C[C@H]1C(=O)NC[C@@H]1CC[C@@H](C(=O)NC2CCCCC2)CC1 ZINC000217590042 JJ In-Stock Unstable HDAC8 19 41 CC(C)(C)OC(=O)N1Cc2ccccc2C[C@H]1C(=O)NC[C@@H]1CC[C@@H](C(=O)NC2CCCCC2)CC1 ZINC000217590042 JJ In-Stock Unstable PREP 23 46 CC(C)(C)OC(=O)N1Cc2ccccc2C[C@H]1C(=O)NC[C@@H]1CC[C@@H](C(=O)NC2CCCCC2)CC1 ZINC000217590042 JJ In-Stock Unstable CFTR 62 36 CC(C)(C)OC(=O)N1Cc2ccccc2C[C@H]1C(=O)NC[C@@H]1CC[C@@H](C(=O)NC2CCCCC2)CC1 ZINC000217590042 JJ In-Stock Unstable ADAM9 59 32 Cc1cc(C(=O)O)ccc1N[C@H]1C[C@@H]2CC[C@@]1(C)C2(C)C ZINC000217590061 CI For-Sale Unstable RARA 40 31 Cc1cc(C(=O)O)ccc1N[C@H]1C[C@@H]2CC[C@@]1(C)C2(C)C ZINC000217590061 CI For-Sale Unstable RARG 41 33 Cc1cc(C(=O)O)ccc1N[C@H]1C[C@@H]2CC[C@@]1(C)C2(C)C ZINC000217590061 CI For-Sale Unstable RXRG 48 35 Cc1cc(C(=O)O)ccc1N[C@H]1C[C@@H]2CC[C@@]1(C)C2(C)C ZINC000217590061 CI For-Sale Unstable RXRB 47 35 O=C(O)c1cc(S(=O)(=O)NCCO)ccc1NCc1ccccc1 ZINC000217590067 FD In-Stock Unstable CA7 16 40 O=C(O)c1cc(S(=O)(=O)NCCO)ccc1NCc1ccccc1 ZINC000217590067 FD In-Stock Unstable BDKRB1 0 42 O=C(O)c1cc(S(=O)(=O)NCCO)ccc1NCc1ccccc1 ZINC000217590067 FD In-Stock Unstable CA5B 34 40 O=C(O)c1cc(S(=O)(=O)NCCO)ccc1NCc1ccccc1 ZINC000217590067 FD In-Stock Unstable CA5A 39 40 Cc1noc(C)c1CC(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217590094 EF For-Sale Unstable NPY5R 25 41 Cc1cc(C(=O)O)ccc1N[C@@H]1C[C@H]2CC[C@@]1(C)C2(C)C ZINC000217590132 CI For-Sale Unstable RARA 40 31 Cc1cc(C(=O)O)ccc1N[C@@H]1C[C@H]2CC[C@@]1(C)C2(C)C ZINC000217590132 CI For-Sale Unstable RARG 41 33 Cc1cc(C(=O)O)ccc1N[C@@H]1C[C@H]2CC[C@@]1(C)C2(C)C ZINC000217590132 CI For-Sale Unstable RXRG 48 35 Cc1cc(C(=O)O)ccc1N[C@@H]1C[C@H]2CC[C@@]1(C)C2(C)C ZINC000217590132 CI For-Sale Unstable RXRB 47 35 CC[C@@H](NC(=O)NCC1CCCCC1)c1ccc2c(c1)CCCC2 ZINC000217590160 EJ For-Sale Unstable MTR1B_CHICK 0 40 C[C@@H](Nc1ccc(S(=O)(=O)NCCO)cc1C(=O)O)c1ccccc1 ZINC000217590166 FD In-Stock Unstable CASP3 21 40 C[C@@H](Nc1ccc(S(=O)(=O)NCCO)cc1C(=O)O)c1ccccc1 ZINC000217590166 FD In-Stock Unstable BDKRB1 0 44 Cc1noc(C)c1CC(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217590167 EF For-Sale Unstable NPY5R 25 41 O=C(c1ccc(O)cn1)N1CC[C@@](O)(c2ccccc2)[C@H]2CCCC[C@@H]21 ZINC000217590195 FG In-Stock Unstable CNR2 0 74 Cc1cc(C(=O)O)ccc1N[C@H]1C[C@H]2CC[C@@]1(C)C2(C)C ZINC000217590210 CI For-Sale Unstable RARA 40 31 Cc1cc(C(=O)O)ccc1N[C@H]1C[C@H]2CC[C@@]1(C)C2(C)C ZINC000217590210 CI For-Sale Unstable RARG 41 33 Cc1cc(C(=O)O)ccc1N[C@H]1C[C@H]2CC[C@@]1(C)C2(C)C ZINC000217590210 CI For-Sale Unstable RXRG 48 35 Cc1cc(C(=O)O)ccc1N[C@H]1C[C@H]2CC[C@@]1(C)C2(C)C ZINC000217590210 CI For-Sale Unstable RXRB 47 35 Cn1cc(C(=O)O)cc(I)c1=O ZINC000217590229 CC In-Stock Unstable TPMT 0 47 CC[C@H](NC(=O)NCC1CCCCC1)c1ccc2c(c1)CCCC2 ZINC000217590233 EJ For-Sale Unstable MTR1B_CHICK 0 40 C[C@H](Nc1ccc(S(=O)(=O)NCCO)cc1C(=O)O)c1ccccc1 ZINC000217590263 FD In-Stock Unstable CASP3 21 40 C[C@H](Nc1ccc(S(=O)(=O)NCCO)cc1C(=O)O)c1ccccc1 ZINC000217590263 FD In-Stock Unstable BDKRB1 0 44 Cc1noc(C)c1C(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217590274 EF In-Stock Unstable NPY5R 27 41 CCc1ccc([C@@H](C)NC(=O)NCC2CCCCC2)cc1 ZINC000217590343 CI For-Sale Unstable ACACA 53 38 COc1ccc2cc(C(=O)N3[C@H]4CC[C@H]3CC(SC)C4)[nH]c2c1 ZINC000217590346 EH In-Stock Unstable GRIN2B 15 46 CNc1nc(C2CC2)nc(N[C@@H]2CCN3CCC[C@@H]23)c1C ZINC000217590347 CE For-Sale Unstable CHRM3 20 44 Cc1noc(C)c1C(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217590353 EF In-Stock Unstable NPY5R 27 41 O=C(O)c1cc(S(=O)(=O)NCCO)ccc1NCCc1ccccc1 ZINC000217590373 FD In-Stock Unstable CA2 20 43 O=C(O)c1cc(S(=O)(=O)NCCO)ccc1NCCc1ccccc1 ZINC000217590373 FD In-Stock Unstable TBXA2R 52 42 O=C(O)c1cc(S(=O)(=O)NCCO)ccc1NCCc1ccccc1 ZINC000217590373 FD In-Stock Unstable CA1 15 43 O=C(O)c1cc(S(=O)(=O)NCCO)ccc1NCCc1ccccc1 ZINC000217590373 FD In-Stock Unstable BDKRB1 0 41 COc1ccc(CCN2C(=O)N[C@@H](CCC(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)C2=O)cc1 ZINC000217590417 JD In-Stock Unstable CHRNA4 29 49 CCc1ccc([C@H](C)NC(=O)NCC2CCCCC2)cc1 ZINC000217590424 CI For-Sale Unstable ACACA 53 38 CNc1nc(C2CC2)nc(N[C@H]2CCN3CCC[C@@H]23)c1C ZINC000217590430 CE For-Sale Unstable CHRM3 20 44 CC(=O)N1CCC(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)CC1 ZINC000217590463 FD For-Sale Unstable NPY5R 49 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCCO)cc2C(=O)O)cc1 ZINC000217590479 GD In-Stock Unstable CA2 19 44 COc1ccc(CCNc2ccc(S(=O)(=O)NCCO)cc2C(=O)O)cc1 ZINC000217590479 GD In-Stock Unstable TBXA2R 50 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCCO)cc2C(=O)O)cc1 ZINC000217590479 GD In-Stock Unstable TBXAS1 23 44 COc1ccc(CCNc2ccc(S(=O)(=O)NCCO)cc2C(=O)O)cc1 ZINC000217590479 GD In-Stock Unstable BMP1 57 37 COc1ccc(CCNc2ccc(S(=O)(=O)NCCO)cc2C(=O)O)cc1 ZINC000217590479 GD In-Stock Unstable CA1 19 44 COc1ccc(CCNc2ccc(S(=O)(=O)NCCO)cc2C(=O)O)cc1 ZINC000217590479 GD In-Stock Unstable MMP13 56 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCCO)cc2C(=O)O)cc1 ZINC000217590479 GD In-Stock Unstable ADAM17 43 37 COc1ccc(CCNc2ccc(S(=O)(=O)NCCO)cc2C(=O)O)cc1 ZINC000217590479 GD In-Stock Unstable MMP2 31 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCCO)cc2C(=O)O)cc1 ZINC000217590479 GD In-Stock Unstable MMP8 23 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCCO)cc2C(=O)O)cc1 ZINC000217590479 GD In-Stock Unstable MMP14 18 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCCO)cc2C(=O)O)cc1 ZINC000217590479 GD In-Stock Unstable MMP9 50 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCCO)cc2C(=O)O)cc1 ZINC000217590479 GD In-Stock Unstable MMP12 27 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCCO)cc2C(=O)O)cc1 ZINC000217590479 GD In-Stock Unstable PTGDR 23 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCCO)cc2C(=O)O)cc1 ZINC000217590479 GD In-Stock Unstable IAP 0 46 COc1ccc(CCNc2ccc(S(=O)(=O)NCCO)cc2C(=O)O)cc1 ZINC000217590479 GD In-Stock Unstable CA9 23 44 COc1ccc(CCNc2ccc(S(=O)(=O)NCCO)cc2C(=O)O)cc1 ZINC000217590479 GD In-Stock Unstable MMP1 53 37 COc1ccc(CCNc2ccc(S(=O)(=O)NCCO)cc2C(=O)O)cc1 ZINC000217590479 GD In-Stock Unstable AKR1C3 30 47 COc1ccc(CCNc2ccc(S(=O)(=O)NCCO)cc2C(=O)O)cc1 ZINC000217590479 GD In-Stock Unstable AKR1C2 51 38 CC(C)C[C@@H](C(=O)N1CCN(Cc2cccnc2)CC1)N1C(=O)c2ccccc2C1=O ZINC000217590499 HE On-Demand Unstable PTAFR 15 52 O=C(Cc1c[nH]cn1)NC[C@@H](c1ccccc1)N1CCCCC1 ZINC000217590506 DE In-Stock Unstable HRH2 45 43 O=C(Cc1c[nH]cn1)NC[C@@H](c1ccccc1)N1CCCCC1 ZINC000217590506 DE In-Stock Unstable HRH1 21 43 O=C(Cc1c[nH]cn1)NC[C@@H](c1ccccc1)N1CCCCC1 ZINC000217590506 DE In-Stock Unstable PGC 41 34 O=C(Cc1c[nH]cn1)NC[C@@H](c1ccccc1)N1CCCCC1 ZINC000217590506 DE In-Stock Unstable HRAS 50 35 O=C(Cc1c[nH]cn1)NC[C@@H](c1ccccc1)N1CCCCC1 ZINC000217590506 DE In-Stock Unstable HRH3 57 45 O=C(Cc1c[nH]cn1)NC[C@@H](c1ccccc1)N1CCCCC1 ZINC000217590506 DE In-Stock Unstable HDH 0 40 O=C(Cc1c[nH]cn1)NC[C@@H](c1ccccc1)N1CCCCC1 ZINC000217590506 DE In-Stock Unstable HISD 0 40 O=C(c1ccc(F)cc1)[C@H]1[C@H]2C(=O)N(c3ccccc3Cl)C(=O)[C@@H]2[C@H]2CCCN21 ZINC000217590526 HG In-Stock Unstable SLC18A3 23 41 CC(=O)N1CCC(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)CC1 ZINC000217590545 FD For-Sale Unstable NPY5R 49 41 CC[S@@](=O)CCNc1nc(NN)nc(N(C)C)n1 ZINC000217590551 CB For-Sale Unstable AT1 0 41 CC(C)C[C@H](C(=O)N1CCN(Cc2cccnc2)CC1)N1C(=O)c2ccccc2C1=O ZINC000217590571 HE On-Demand Unstable PTAFR 15 52 COc1ccc(CCNc2ccc(S(=O)(=O)NCCO)cc2C(=O)O)cc1OC ZINC000217590583 HD In-Stock Unstable TBXA2R 44 40 COc1ccc(CCNc2ccc(S(=O)(=O)NCCO)cc2C(=O)O)cc1OC ZINC000217590583 HD In-Stock Unstable TBXAS1 20 45 COc1ccc(CCNc2ccc(S(=O)(=O)NCCO)cc2C(=O)O)cc1OC ZINC000217590583 HD In-Stock Unstable IAP 0 47 COc1ccc(CCNc2ccc(S(=O)(=O)NCCO)cc2C(=O)O)cc1OC ZINC000217590583 HD In-Stock Unstable AKR1C3 15 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCCO)cc2C(=O)O)cc1OC ZINC000217590583 HD In-Stock Unstable SCMU_MYCTU 0 46 O=C(Cc1c[nH]cn1)NC[C@H](c1ccccc1)N1CCCCC1 ZINC000217590596 DE In-Stock Unstable HRH2 45 43 O=C(Cc1c[nH]cn1)NC[C@H](c1ccccc1)N1CCCCC1 ZINC000217590596 DE In-Stock Unstable HRH1 21 43 O=C(Cc1c[nH]cn1)NC[C@H](c1ccccc1)N1CCCCC1 ZINC000217590596 DE In-Stock Unstable PGC 41 34 O=C(Cc1c[nH]cn1)NC[C@H](c1ccccc1)N1CCCCC1 ZINC000217590596 DE In-Stock Unstable HRAS 50 35 O=C(Cc1c[nH]cn1)NC[C@H](c1ccccc1)N1CCCCC1 ZINC000217590596 DE In-Stock Unstable HRH3 57 45 O=C(Cc1c[nH]cn1)NC[C@H](c1ccccc1)N1CCCCC1 ZINC000217590596 DE In-Stock Unstable HDH 0 40 O=C(Cc1c[nH]cn1)NC[C@H](c1ccccc1)N1CCCCC1 ZINC000217590596 DE In-Stock Unstable HISD 0 40 O=C(c1ccc(F)cc1)[C@@H]1[C@H]2C(=O)N(c3ccccc3Cl)C(=O)[C@@H]2[C@H]2CCCN12 ZINC000217590618 HG In-Stock Unstable SLC18A3 23 41 CC[S@](=O)CCNc1nc(NN)nc(N(C)C)n1 ZINC000217590623 CB For-Sale Unstable AT1 0 41 O=C1O[C@@]2(CCCN(C(=O)CCn3cnc4ccccc4c3=O)C2)c2ccccc21 ZINC000217590651 HE For-Sale Unstable NPY5R 25 40 O=C(NCC1CCCCC1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217590709 DK For-Sale Unstable ADRB1 22 41 O=C(NCC1CCCCC1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217590709 DK For-Sale Unstable PDGFRB 23 41 O=C(NCC1CCCCC1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217590709 DK For-Sale Unstable GRIN2B 20 40 O=C(NCC1CCCCC1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217590709 DK For-Sale Unstable LTA4H 65 44 O=C(NCC1CCCCC1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217590709 DK For-Sale Unstable CA1 56 49 O=C(NCC1CCCCC1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217590709 DK For-Sale Unstable RAF1 34 42 O=C(NCC1CCCCC1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217590709 DK For-Sale Unstable MMP2 26 42 O=C(NCC1CCCCC1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217590709 DK For-Sale Unstable FAAH 22 50 O=C(NCC1CCCCC1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217590709 DK For-Sale Unstable NPY5R 21 40 O=C(NCC1CCCCC1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217590709 DK For-Sale Unstable MMP9 26 40 O=C(NCC1CCCCC1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217590709 DK For-Sale Unstable EPHX2 46 62 O=C(NCC1CCCCC1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217590709 DK For-Sale Unstable PLAU 16 47 O=C(NCC1CCCCC1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217590709 DK For-Sale Unstable TGM2 15 44 O=C(NCC1CCCCC1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217590709 DK For-Sale Unstable CA12 24 49 O=C(NCC1CCCCC1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217590709 DK For-Sale Unstable PDGFRA 29 45 O=C(NCC1CCCCC1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217590709 DK For-Sale Unstable CA9 24 49 O=C(NCC1CCCCC1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217590709 DK For-Sale Unstable Q8MMZ8_EIMTE 47 42 O=C(NCC1CCCCC1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217590709 DK For-Sale Unstable F13A1 26 44 O=C(NCC1CCCCC1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217590709 DK For-Sale Unstable NCE103 35 42 O=C(NCC1CCCCC1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217590709 DK For-Sale Unstable PRMT3 40 39 O=C(NCC1CCCCC1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217590709 DK For-Sale Unstable P96878_MYCTU 15 49 O=C(NCC1CCCCC1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217590709 DK For-Sale Unstable ACAT 0 47 O=C(NCC1CCCCC1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217590709 DK For-Sale Unstable METAP2 0 42 O=C(NCC1CCCCC1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217590709 DK For-Sale Unstable UPPS 0 42 O=C(NCC1CCCCC1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217590709 DK For-Sale Unstable NAMPT 37 52 O=C(NCC1CCCCC1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217590709 DK For-Sale Unstable PFKFB3 43 34 O=C1O[C@]2(CCCN(C(=O)CCn3cnc4ccccc4c3=O)C2)c2ccccc21 ZINC000217590730 HE For-Sale Unstable NPY5R 25 40 COc1ccc(O)c(C(=O)NCCCn2ccc3ccccc32)c1 ZINC000217590737 DG On-Demand Unstable DRD2 17 43 COc1ccc(O)c(C(=O)NCCCn2ccc3ccccc32)c1 ZINC000217590737 DG On-Demand Unstable DRD4 43 34 COc1ccc(O)c(C(=O)NCCCn2ccc3ccccc32)c1 ZINC000217590737 DG On-Demand Unstable DRD3 41 43 COc1ccc(O)c(C(=O)NCCCn2ccc3ccccc32)c1 ZINC000217590737 DG On-Demand Unstable THRB 16 42 COc1ccc(O)c(C(=O)NCCCn2ccc3ccccc32)c1 ZINC000217590737 DG On-Demand Unstable NQO2 20 42 COc1ccc(O)c(C(=O)NCCCn2ccc3ccccc32)c1 ZINC000217590737 DG On-Demand Unstable MTNR1A 68 44 COc1ccc(O)c(C(=O)NCCCn2ccc3ccccc32)c1 ZINC000217590737 DG On-Demand Unstable MTNR1B 61 44 COc1ccc(O)c(C(=O)NCCCn2ccc3ccccc32)c1 ZINC000217590737 DG On-Demand Unstable POLR1A 48 34 O=C(Nc1nc2ccccc2s1)c1nc2ccccc2s1 ZINC000217590740 DI In-Stock Anodyne LCK 30 40 O=C(Nc1nc2ccccc2s1)c1nc2ccccc2s1 ZINC000217590740 DI In-Stock Anodyne CSNK1D 46 60 O=C(Nc1nc2ccccc2s1)c1nc2ccccc2s1 ZINC000217590740 DI In-Stock Anodyne PIK3CA 21 43 O=C(Nc1nc2ccccc2s1)c1nc2ccccc2s1 ZINC000217590740 DI In-Stock Anodyne HSD17B1 16 52 O=C(Nc1nc2ccccc2s1)c1nc2ccccc2s1 ZINC000217590740 DI In-Stock Anodyne ST14 48 36 O=C(Nc1nc2ccccc2s1)c1nc2ccccc2s1 ZINC000217590740 DI In-Stock Anodyne BCL2L1 32 43 O=C(Nc1nc2ccccc2s1)c1nc2ccccc2s1 ZINC000217590740 DI In-Stock Anodyne FABK 0 49 O=C(Nc1nc2ccccc2s1)c1nc2ccccc2s1 ZINC000217590740 DI In-Stock Anodyne MCA2 0 40 O=C(Nc1nc2ccccc2s1)c1nc2ccccc2s1 ZINC000217590740 DI In-Stock Anodyne PORCN 0 45 O=C(Nc1nc2ccccc2s1)c1nc2ccccc2s1 ZINC000217590740 DI In-Stock Anodyne TMPRSS6 71 36 O=C(Nc1nc2ccccc2s1)c1nc2ccccc2s1 ZINC000217590740 DI In-Stock Anodyne ISPD 0 42 O=C(O)c1cc(S(=O)(=O)NCCO)ccc1NC[C@@H]1CCCO1 ZINC000217590800 EC In-Stock Unstable BDKRB1 0 42 COc1ccc(CN2C(=O)N[C@@H](CCC(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)C2=O)cc1 ZINC000217590812 JD In-Stock Unstable CHRNA4 28 48 Cc1ccc(Cl)cc1NC(=O)NCC1CCCCC1 ZINC000217590819 CI On-Demand Unstable CNR1 18 47 Cc1ccc(Cl)cc1NC(=O)NCC1CCCCC1 ZINC000217590819 CI On-Demand Unstable LDLR 0 46 Cc1ccc(Cl)cc1NC(=O)NCC1CCCCC1 ZINC000217590819 CI On-Demand Unstable EPHX2 22 62 Cc1ccc(Cl)cc1NC(=O)NCC1CCCCC1 ZINC000217590819 CI On-Demand Unstable CACNA1I 63 37 Cc1ccc(Cl)cc1NC(=O)NCC1CCCCC1 ZINC000217590819 CI On-Demand Unstable ACAT 0 43 Cc1ccc(Cl)cc1NC(=O)NCC1CCCCC1 ZINC000217590819 CI On-Demand Unstable METAP2 22 46 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1cc(Br)ccc1Br ZINC000217590838 GK For-Sale Unstable TRPM8 16 42 O=C1O[C@@]2(CCCN(C(=O)Cn3cncn3)C2)c2ccccc21 ZINC000217590843 DC For-Sale Unstable NPY5R 29 41 O=C(c1ccsc1)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217590853 GI In-Stock Unstable CHRM2 33 41 O=C(c1ccsc1)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217590853 GI In-Stock Unstable HRH1 18 43 O=C(c1ccsc1)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217590853 GI In-Stock Unstable CCR3 25 43 O=C(c1ccsc1)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217590853 GI In-Stock Unstable L3MBTL1 0 42 O=C(c1ccsc1)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217590853 GI In-Stock Unstable L3MBTL3 91 42 O=C(c1ccsc1)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217590853 GI In-Stock Unstable MBTD1 0 42 O=C(c1ccsc1)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217590853 GI In-Stock Unstable TP53BP1 0 40 O=C(O)c1cc(S(=O)(=O)NCCO)ccc1NC[C@H]1CCCO1 ZINC000217590880 EC In-Stock Unstable BDKRB1 0 42 O=C1O[C@]2(CCCN(C(=O)Cn3cncn3)C2)c2ccccc21 ZINC000217590920 DC For-Sale Unstable NPY5R 29 41 COc1ccc(OC)c(NC(=O)NCC2CCCCC2)c1 ZINC000217590929 CG On-Demand Unstable MTR1B_CHICK 0 42 COc1ccc(OC)c(NC(=O)NCC2CCCCC2)c1 ZINC000217590929 CG On-Demand Unstable MTNR1B 49 45 COc1ccc(OC)c(NC(=O)NCC2CCCCC2)c1 ZINC000217590929 CG On-Demand Unstable STK17B 41 37 COc1ccc(OC)c(NC(=O)NCC2CCCCC2)c1 ZINC000217590929 CG On-Demand Unstable AKR1C2 48 34 COc1ccc(OC)c(NC(=O)NCC2CCCCC2)c1 ZINC000217590929 CG On-Demand Unstable QRFPR 41 33 COc1ccc(OC)c(NC(=O)NCC2CCCCC2)c1 ZINC000217590929 CG On-Demand Unstable ACAT 0 44 COc1ccc(OC)c(NC(=O)NCC2CCCCC2)c1 ZINC000217590929 CG On-Demand Unstable METAP2 0 43 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1cc(Br)ccc1Br ZINC000217590932 GK For-Sale Unstable TRPM8 16 42 O=C(CC1CCCC1)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217590961 GI In-Stock Unstable CHRM2 40 39 O=C(CC1CCCC1)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217590961 GI In-Stock Unstable HRH3 30 45 O=C(CC1CCCC1)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217590961 GI In-Stock Unstable CCR3 27 44 O=C(CC1CCCC1)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217590961 GI In-Stock Unstable L3MBTL3 74 39 O=C(c1n[nH]c2c1COc1ccccc1-2)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217590965 GE In-Stock Unstable CHRNA4 26 42 O=C(O)c1cc(S(=O)(=O)NCCO)ccc1N1CCCC1 ZINC000217590994 DC In-Stock Unstable SFRP1 59 33 O=C(O)c1cc(S(=O)(=O)NCCO)ccc1N1CCCC1 ZINC000217590994 DC In-Stock Unstable WNT3 42 33 Cc1c(N)nc(C2CC2)nc1N[C@@H]1CCN2CCC[C@@H]12 ZINC000217591009 CD For-Sale Unstable CHRM3 20 44 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1cc(Br)ccc1Br ZINC000217591013 GK For-Sale Unstable TRPM8 16 42 O=C(O)/C=C\c1cccc(CNC(=O)c2ccncc2)c1 ZINC000217591017 CE For-Sale Unstable MMP13 15 43 O=C(O)/C=C\c1cccc(CNC(=O)c2ccncc2)c1 ZINC000217591017 CE For-Sale Unstable HDAC1 15 45 O=C(O)/C=C\c1cccc(CNC(=O)c2ccncc2)c1 ZINC000217591017 CE For-Sale Unstable HDAC6 21 44 O=C(O)/C=C\c1cccc(CNC(=O)c2ccncc2)c1 ZINC000217591017 CE For-Sale Unstable NAMPT 46 38 O=C(O)/C=C\c1cccc(CNC(=O)c2ccncc2)c1 ZINC000217591017 CE For-Sale Unstable KCNK3 17 43 O=C1O[C@@]2(CCCN(C(=O)CCCN3C(=O)c4ccccc4C3=O)C2)c2ccccc21 ZINC000217591022 HF For-Sale Unstable NPY5R 25 41 Cc1cc(C)c(NC(=O)NCC2CCCCC2)c(C)c1 ZINC000217591045 CI On-Demand Unstable CACNA1I 40 31 Cc1cc(C)c(NC(=O)NCC2CCCCC2)c(C)c1 ZINC000217591045 CI On-Demand Unstable ACAT 0 49 COc1ccccc1CCN1C(=O)N[C@@H](CC(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)C1=O ZINC000217591063 JD In-Stock Unstable CHRNA4 27 42 O=C(CCCCN1C/C=C/COCc2cccc(c2)-c2ccnc(n2)Nc2cccc(c2)C1)NO ZINC000217591064 JI Annotated Unstable JAK1 21 55 O=C(CCCCN1C/C=C/COCc2cccc(c2)-c2ccnc(n2)Nc2cccc(c2)C1)NO ZINC000217591064 JI Annotated Unstable FLT3 48 74 O=C(CCCCN1C/C=C/COCc2cccc(c2)-c2ccnc(n2)Nc2cccc(c2)C1)NO ZINC000217591064 JI Annotated Unstable TYK2 55 59 CCCCCCCCCC(=O)N(CCCN)CCCN ZINC000217591068 CF Annotated Unstable FABP5 15 43 CCCCCCCCCC(=O)N(CCCN)CCCN ZINC000217591068 CF Annotated Unstable CQSS 63 40 Cc1nnsc1C(=O)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217591070 HG In-Stock Unstable CHRM2 41 38 Cc1nnsc1C(=O)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217591070 HG In-Stock Unstable HRH1 18 41 Cc1nnsc1C(=O)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217591070 HG In-Stock Unstable CCR3 26 41 Cc1nnsc1C(=O)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217591070 HG In-Stock Unstable SCD1 46 35 Cc1nnsc1C(=O)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217591070 HG In-Stock Unstable L3MBTL3 72 37 Cc1c(N)nc(C2CC2)nc1N[C@H]1CCN2CCC[C@@H]12 ZINC000217591095 CD For-Sale Unstable CHRM3 20 44 O=C(O)/C=C\c1cccc(CNC(=O)c2cccnc2)c1 ZINC000217591098 CE For-Sale Unstable TBXAS1 73 52 O=C(O)/C=C\c1cccc(CNC(=O)c2cccnc2)c1 ZINC000217591098 CE For-Sale Unstable HDAC1 17 43 O=C(O)/C=C\c1cccc(CNC(=O)c2cccnc2)c1 ZINC000217591098 CE For-Sale Unstable HDAC6 17 45 O=C(O)/C=C\c1cccc(CNC(=O)c2cccnc2)c1 ZINC000217591098 CE For-Sale Unstable NAMPT 86 42 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1cc(Br)ccc1Br ZINC000217591101 GK For-Sale Unstable TRPM8 16 42 C[C@@H]1CN(C[C@@H](O)c2ccccc2)CCCO1 ZINC000217591102 BD On-Demand Unstable OPRK1 0 46 O=C1O[C@]2(CCCN(C(=O)CCCN3C(=O)c4ccccc4C3=O)C2)c2ccccc21 ZINC000217591103 HF For-Sale Unstable NPY5R 25 41 O=C(O)c1cc(S(=O)(=O)NCCO)ccc1N1CCCCC1 ZINC000217591116 EC In-Stock Unstable SFRP1 51 33 O=C1CCc2ccc(OCC(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)cc2N1 ZINC000217591144 GD In-Stock Unstable CHRNA4 26 42 O=C(CCCCCN1C/C=C/COCc2cccc(c2)-c2ccnc(n2)Nc2cccc(c2)C1)NO ZINC000217591149 JJ Annotated Unstable JAK3 18 54 O=C(CCCCCN1C/C=C/COCc2cccc(c2)-c2ccnc(n2)Nc2cccc(c2)C1)NO ZINC000217591149 JJ Annotated Unstable JAK1 42 59 O=C(CCCCCN1C/C=C/COCc2cccc(c2)-c2ccnc(n2)Nc2cccc(c2)C1)NO ZINC000217591149 JJ Annotated Unstable FLT3 47 75 O=C(CCCCCN1C/C=C/COCc2cccc(c2)-c2ccnc(n2)Nc2cccc(c2)C1)NO ZINC000217591149 JJ Annotated Unstable TYK2 54 59 COC(=O)c1ccccc1NC(=O)NCC1CCCCC1 ZINC000217591150 CG For-Sale Unstable CCR3 24 40 COC(=O)c1ccccc1NC(=O)NCC1CCCCC1 ZINC000217591150 CG For-Sale Unstable ACAT 0 48 COC(=O)c1ccccc1NC(=O)NCC1CCCCC1 ZINC000217591150 CG For-Sale Unstable FAS 23 46 O=C(c1cc2ccccc2o1)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217591176 HJ In-Stock Unstable CHRM2 42 44 O=C(c1cc2ccccc2o1)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217591176 HJ In-Stock Unstable HRH1 22 45 O=C(c1cc2ccccc2o1)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217591176 HJ In-Stock Unstable GRIN2B 19 40 O=C(c1cc2ccccc2o1)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217591176 HJ In-Stock Unstable HRH3 31 42 O=C(c1cc2ccccc2o1)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217591176 HJ In-Stock Unstable CCR3 31 45 O=C(c1cc2ccccc2o1)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217591176 HJ In-Stock Unstable L3MBTL1 0 43 O=C(c1cc2ccccc2o1)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217591176 HJ In-Stock Unstable L3MBTL3 80 43 O=C(O)/C=C\c1cccc(CNC(=O)c2ccco2)c1 ZINC000217591182 CE For-Sale Unstable ADAM12 26 44 Cc1nc2c(OCc3c(F)cccc3F)cccn2c1C(=O)O ZINC000217591186 DG In-Stock Unstable PTGER1 17 43 Cc1nc2c(OCc3c(F)cccc3F)cccn2c1C(=O)O ZINC000217591186 DG In-Stock Unstable BDKRB2 41 54 C[C@H]1CN(C[C@@H](O)c2ccccc2)CCCO1 ZINC000217591197 BD On-Demand Unstable OPRK1 0 46 O=C(O)c1cc(S(=O)(=O)NCCO)ccc1N1CCOCC1 ZINC000217591229 EB In-Stock Unstable SLC6A9 17 46 COc1cc([N+](=O)[O-])ccc1NC(=O)NCC1CCCCC1 ZINC000217591255 DG On-Demand Unstable EPHX1 0 55 COc1cc([N+](=O)[O-])ccc1NC(=O)NCC1CCCCC1 ZINC000217591255 DG On-Demand Unstable CACNA1C 40 37 COc1cc([N+](=O)[O-])ccc1NC(=O)NCC1CCCCC1 ZINC000217591255 DG On-Demand Unstable TBXA2R 26 44 COc1cc([N+](=O)[O-])ccc1NC(=O)NCC1CCCCC1 ZINC000217591255 DG On-Demand Unstable CACNA1D 68 37 COc1cc([N+](=O)[O-])ccc1NC(=O)NCC1CCCCC1 ZINC000217591255 DG On-Demand Unstable KCNMA1 24 53 COc1cc([N+](=O)[O-])ccc1NC(=O)NCC1CCCCC1 ZINC000217591255 DG On-Demand Unstable SLC27A4 43 35 CN(Cc1ccc(/C=C\C(=O)O)cc1)C(=O)c1ccsc1 ZINC000217591258 DG For-Sale Unstable HSD17B2 24 43 O=C(CSCc1ccccc1)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217591275 IJ In-Stock Unstable HRH1 23 43 O=C(CSCc1ccccc1)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217591275 IJ In-Stock Unstable HRH3 15 41 O=C(CSCc1ccccc1)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217591275 IJ In-Stock Unstable CCR3 29 43 O=C(CSCc1ccccc1)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217591275 IJ In-Stock Unstable SCD1 24 41 O=C(CSCc1ccccc1)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217591275 IJ In-Stock Unstable SCD 28 41 O=C(CSCc1ccccc1)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217591275 IJ In-Stock Unstable L3MBTL3 51 39 Cn1c(CCNC(=O)c2cc(N3CCCCC3)ccc2Cl)nc2ccccc21 ZINC000217591299 GI In-Stock Unstable DRD4 43 33 Cn1c(CCNC(=O)c2cc(N3CCCCC3)ccc2Cl)nc2ccccc21 ZINC000217591299 GI In-Stock Unstable HTR2A 32 42 Cn1c(CCNC(=O)c2cc(N3CCCCC3)ccc2Cl)nc2ccccc21 ZINC000217591299 GI In-Stock Unstable HTR2C 29 42 Cn1c(CCNC(=O)c2cc(N3CCCCC3)ccc2Cl)nc2ccccc21 ZINC000217591299 GI In-Stock Unstable GRM2 0 46 CCOCCCNc1ccc(S(=O)(=O)NCCO)cc1C(=O)O ZINC000217591331 EC In-Stock Unstable CASP3 0 40 CCOCCCNc1ccc(S(=O)(=O)NCCO)cc1C(=O)O ZINC000217591331 EC In-Stock Unstable BDKRB1 0 41 O=C(NC1CCCCC1)C(F)F ZINC000217591371 AD On-Demand Unstable EPHX2 25 40 O=C(NC1CCCCC1)C(F)F ZINC000217591371 AD On-Demand Unstable P95276_MYCTO 0 40 O=C1O[C@@]2(CCCN(C(=O)C3CCCC3)C2)c2ccccc21 ZINC000217591376 CF For-Sale Unstable NPY5R 52 44 O=C(c1cc(-c2ccco2)[nH]n1)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217591378 IH In-Stock Unstable HRH1 17 40 O=C(c1cc(-c2ccco2)[nH]n1)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217591378 IH In-Stock Unstable CCR3 31 40 O=C(c1cc(-c2ccco2)[nH]n1)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217591378 IH In-Stock Unstable L3MBTL3 57 34 COc1ccc(CN2C(=O)N[C@@H](CCC(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)C2=O)cc1OC ZINC000217591407 JD In-Stock Unstable CHRNA4 27 44 CC(=O)c1cc(F)ccc1OCc1csc(COc2ccc(C)cc2)n1 ZINC000217591414 FJ On-Demand Unstable PPARD 27 41 CC(C)OCCCNc1ccc(S(=O)(=O)NCCO)cc1C(=O)O ZINC000217591433 FC In-Stock Unstable BDKRB1 0 41 O=C1O[C@]2(CCCN(C(=O)C3CCCC3)C2)c2ccccc21 ZINC000217591450 CF For-Sale Unstable NPY5R 52 44 C[C@@H]1CN(C[C@@](C)(O)c2ccccc2)CCCO1 ZINC000217591455 BE On-Demand Unstable CYP2J2 46 35 C[C@H]1CN(C[C@@](C)(O)c2ccccc2)CCCO1 ZINC000217591528 BE On-Demand Unstable CYP2J2 46 35 CCCCCNc1ccc(S(=O)(=O)NCCO)cc1C(=O)O ZINC000217591541 ED In-Stock Unstable CASP3 16 44 CCCCCNc1ccc(S(=O)(=O)NCCO)cc1C(=O)O ZINC000217591541 ED In-Stock Unstable BDKRB1 0 41 O=C1O[C@@]2(CCCN(C(=O)/C=C/c3ccccc3Cl)C2)c2ccccc21 ZINC000217591559 FI For-Sale Unstable NPY5R 31 46 O=S(=O)(c1cccs1)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217591585 HH In-Stock Unstable HRH1 17 40 O=S(=O)(c1cccs1)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217591585 HH In-Stock Unstable CCR3 29 40 O=S(=O)(c1cccs1)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217591585 HH In-Stock Unstable FAAH 0 40 O=C1O[C@]2(CCCN(C(=O)/C=C/c3ccccc3Cl)C2)c2ccccc21 ZINC000217591636 FI For-Sale Unstable NPY5R 31 46 CC(C)CCNc1ccc(S(=O)(=O)NCCO)cc1C(=O)O ZINC000217591659 ED In-Stock Unstable CASP3 17 43 O=S(=O)(c1ccccc1F)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217591687 IH In-Stock Unstable ADRA1D 19 45 O=S(=O)(c1ccccc1F)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217591687 IH In-Stock Unstable ADRA1A 15 45 O=S(=O)(c1ccccc1F)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217591687 IH In-Stock Unstable HRH1 18 43 O=S(=O)(c1ccccc1F)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217591687 IH In-Stock Unstable ADRA1B 21 45 O=S(=O)(c1ccccc1F)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217591687 IH In-Stock Unstable HRH3 16 41 O=S(=O)(c1ccccc1F)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217591687 IH In-Stock Unstable CCR1 16 44 O=S(=O)(c1ccccc1F)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217591687 IH In-Stock Unstable CCR3 31 43 O=C(NCC1CCCCC1)Nc1ccccc1O ZINC000217591704 BG For-Sale Unstable ACAT 0 40 O=C1O[C@@]2(CCCN(C(=O)Cc3c(F)cccc3Cl)C2)c2ccccc21 ZINC000217591745 FH For-Sale Unstable NPY5R 27 42 Clc1ncnc(NC2CCCCC2)c1I ZINC000217591746 EG In-Stock Unstable CD38 36 43 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NCCO)cc1C(=O)O ZINC000217591758 ED In-Stock Unstable CASP3 15 43 O=S(=O)(/C=C/c1ccccc1)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217591793 II In-Stock Unstable CCR3 25 40 CCOc1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217591803 CH On-Demand Unstable ADRB1 23 42 CCOc1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217591803 CH On-Demand Unstable KCNQ1 0 40 CCOc1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217591803 CH On-Demand Unstable EPHX2 48 46 CCOc1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217591803 CH On-Demand Unstable CA12 20 40 CCOc1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217591803 CH On-Demand Unstable PDGFRA 18 45 CCOc1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217591803 CH On-Demand Unstable CA9 21 40 CCOc1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217591803 CH On-Demand Unstable NCE103 27 40 O=C1O[C@]2(CCCN(C(=O)Cc3c(F)cccc3Cl)C2)c2ccccc21 ZINC000217591811 FH For-Sale Unstable NPY5R 27 42 CCC[C@H](C)Nc1ccc(S(=O)(=O)NCCO)cc1C(=O)O ZINC000217591832 ED In-Stock Unstable CASP3 15 43 Clc1ncnc(NC2CCCC2)c1I ZINC000217591845 DG In-Stock Unstable CD38 39 42 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591859 FE For-Sale Unstable ADORA1 72 52 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591859 FE For-Sale Unstable SLC29A1 64 41 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591859 FE For-Sale Unstable ADORA2A 49 52 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591859 FE For-Sale Unstable ADORA2B 20 46 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591859 FE For-Sale Unstable ADK 24 52 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591859 FE For-Sale Unstable AHCY 103 47 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591859 FE For-Sale Unstable P2RX4 43 42 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591859 FE For-Sale Unstable P2RX1 45 40 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591859 FE For-Sale Unstable P2RY1 110 61 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591859 FE For-Sale Unstable ADCY5 44 38 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591859 FE For-Sale Unstable AMD1 36 45 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591859 FE For-Sale Unstable GAPDH 19 40 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591859 FE For-Sale Unstable ITPR1 60 45 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591859 FE For-Sale Unstable P2RY2 20 43 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591859 FE For-Sale Unstable PRKACA 40 31 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591859 FE For-Sale Unstable NS5B 33 49 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591859 FE For-Sale Unstable ADORA3 36 52 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591859 FE For-Sale Unstable OXGR1 132 43 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591859 FE For-Sale Unstable IMPDH2 42 36 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591859 FE For-Sale Unstable RNASE1 49 39 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591859 FE For-Sale Unstable PANC 42 44 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591859 FE For-Sale Unstable Q4VQ11_PIG 40 38 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591859 FE For-Sale Unstable DOT1L 75 38 O=C1O[C@@]2(CCCN(C(=O)c3c(F)cccc3F)C2)c2ccccc21 ZINC000217591902 EG For-Sale Unstable NPY5R 31 43 CCCCOC(=O)c1ccccc1NC(=O)NCC1CCCCC1 ZINC000217591907 EI For-Sale Unstable AMY2 47 33 CCCCOC(=O)c1ccccc1NC(=O)NCC1CCCCC1 ZINC000217591907 EI For-Sale Unstable ACAT 0 50 CCCNC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217591908 ED In-Stock Unstable EDNRA 30 41 CCCNC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217591908 ED In-Stock Unstable TACR1 21 41 CCCNC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217591908 ED In-Stock Unstable MC4R 42 40 CCCNC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217591908 ED In-Stock Unstable BRS3 22 41 Cc1ccc(S(=O)(=O)N2CCC(N3CCC(Oc4ccccc4F)CC3)CC2)cc1C ZINC000217591910 II In-Stock Unstable CHRM2 36 41 Cc1ccc(S(=O)(=O)N2CCC(N3CCC(Oc4ccccc4F)CC3)CC2)cc1C ZINC000217591910 II In-Stock Unstable ADRA1D 31 42 Cc1ccc(S(=O)(=O)N2CCC(N3CCC(Oc4ccccc4F)CC3)CC2)cc1C ZINC000217591910 II In-Stock Unstable ADRA1A 22 42 Cc1ccc(S(=O)(=O)N2CCC(N3CCC(Oc4ccccc4F)CC3)CC2)cc1C ZINC000217591910 II In-Stock Unstable HRH1 20 43 Cc1ccc(S(=O)(=O)N2CCC(N3CCC(Oc4ccccc4F)CC3)CC2)cc1C ZINC000217591910 II In-Stock Unstable ADRA1B 35 42 Cc1ccc(S(=O)(=O)N2CCC(N3CCC(Oc4ccccc4F)CC3)CC2)cc1C ZINC000217591910 II In-Stock Unstable CCR3 31 43 Cc1ccc(S(=O)(=O)N2CCC(N3CCC(Oc4ccccc4F)CC3)CC2)cc1C ZINC000217591910 II In-Stock Unstable PKM 35 40 O=C1O[C@]2(CCCN(C(=O)c3c(F)cccc3F)C2)c2ccccc21 ZINC000217591986 EG For-Sale Unstable NPY5R 31 43 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591993 FE For-Sale Unstable ADORA1 72 52 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591993 FE For-Sale Unstable SLC29A1 64 41 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591993 FE For-Sale Unstable ADORA2A 49 52 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591993 FE For-Sale Unstable ADORA2B 20 46 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591993 FE For-Sale Unstable ADK 24 52 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591993 FE For-Sale Unstable AHCY 103 47 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591993 FE For-Sale Unstable P2RX4 43 42 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591993 FE For-Sale Unstable P2RX1 45 40 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591993 FE For-Sale Unstable P2RY1 110 61 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591993 FE For-Sale Unstable ADCY5 44 38 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591993 FE For-Sale Unstable AMD1 36 45 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591993 FE For-Sale Unstable GAPDH 19 40 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591993 FE For-Sale Unstable ITPR1 60 45 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591993 FE For-Sale Unstable P2RY2 20 43 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591993 FE For-Sale Unstable PRKACA 40 31 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591993 FE For-Sale Unstable NS5B 33 49 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591993 FE For-Sale Unstable ADORA3 36 52 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591993 FE For-Sale Unstable OXGR1 132 43 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591993 FE For-Sale Unstable IMPDH2 42 36 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591993 FE For-Sale Unstable RNASE1 49 39 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591993 FE For-Sale Unstable PANC 42 44 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591993 FE For-Sale Unstable Q4VQ11_PIG 40 38 CC(C)(C)[Si](C)(C)O[C@@H]1C[C@@H](CO)O[C@@H]1n1cnc2c(N)ncnc21 ZINC000217591993 FE For-Sale Unstable DOT1L 75 38 COc1ccc(/C=C2\Oc3c(ccc4c3[C@H](c3ccccc3)CC(=O)O4)C2=O)cc1 ZINC000217592008 GJ In-Stock Unstable TRPM8 0 44 N#Cc1ccccc1S(=O)(=O)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217592042 IG In-Stock Unstable HRH1 16 41 N#Cc1ccccc1S(=O)(=O)N1CCC(N2CCC(Oc3ccccc3F)CC2)CC1 ZINC000217592042 IG In-Stock Unstable CCR3 28 41 COc1ccc(/C=C2\Oc3c(ccc4c3[C@@H](c3ccccc3)CC(=O)O4)C2=O)cc1 ZINC000217592080 GJ In-Stock Unstable TRPM8 0 44 Cc1cccc(NC(=O)NCC2CCCCC2)c1C ZINC000217592089 CI On-Demand Unstable CCR3 15 40 Cc1cccc(NC(=O)NCC2CCCCC2)c1C ZINC000217592089 CI On-Demand Unstable ACAT 0 44 CCO[C@@H]1C[C@@H](NC(=O)c2cccnc2Cl)C1(C)C ZINC000217592091 CF For-Sale Unstable G2YM83_BOTF4 87 43 CCCNc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O ZINC000217592125 DC In-Stock Unstable CASP3 17 47 CCCNc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O ZINC000217592125 DC In-Stock Unstable BDKRB1 0 42 O=C(c1ccsc1)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217592145 GG In-Stock Unstable HRH1 17 41 O=C(c1ccsc1)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217592145 GG In-Stock Unstable CCR3 42 43 O=C(c1ccsc1)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217592145 GG In-Stock Unstable L3MBTL1 0 47 O=C(c1ccsc1)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217592145 GG In-Stock Unstable L3MBTL3 102 47 O=C(c1ccsc1)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217592145 GG In-Stock Unstable L3MBTL4 0 42 O=C(c1ccsc1)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217592145 GG In-Stock Unstable MBTD1 0 46 O=C(c1ccsc1)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217592145 GG In-Stock Unstable TP53BP1 0 42 CCO[C@H]1C[C@@H](NC(=O)c2cccnc2Cl)C1(C)C ZINC000217592180 CF For-Sale Unstable G2YM83_BOTF4 87 43 NC[C@@H]1CCCCN1[C@@H]1CCCc2ccccc21 ZINC000217592181 BF For-Sale Unstable HTR3B 0 42 Cc1ccc(NC(=O)NCC2CCCCC2)c(C)c1 ZINC000217592197 CI On-Demand Unstable LDLR 0 42 Cc1ccc(NC(=O)NCC2CCCCC2)c(C)c1 ZINC000217592197 CI On-Demand Unstable EPHX2 19 45 CC(C)Nc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O ZINC000217592245 DC In-Stock Unstable CASP3 22 44 CC(C)Nc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O ZINC000217592245 DC In-Stock Unstable BDKRB1 0 40 CCO[C@@H]1C[C@H](NC(=O)c2cccnc2Cl)C1(C)C ZINC000217592247 CF For-Sale Unstable G2YM83_BOTF4 87 43 O=C(c1ccc(F)cc1Cl)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217592254 HI In-Stock Unstable CHRM2 27 40 O=C(c1ccc(F)cc1Cl)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217592254 HI In-Stock Unstable HRH1 22 49 O=C(c1ccc(F)cc1Cl)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217592254 HI In-Stock Unstable HRH3 19 41 O=C(c1ccc(F)cc1Cl)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217592254 HI In-Stock Unstable P2RX7 17 40 O=C(c1ccc(F)cc1Cl)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217592254 HI In-Stock Unstable CCR3 33 44 O=C(c1ccc(F)cc1Cl)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217592254 HI In-Stock Unstable L3MBTL1 0 42 O=C(c1ccc(F)cc1Cl)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217592254 HI In-Stock Unstable L3MBTL3 88 42 O=C(c1ccc(F)cc1Cl)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217592254 HI In-Stock Unstable MBTD1 0 42 O=C(c1ccc(F)cc1Cl)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217592254 HI In-Stock Unstable TP53BP1 0 42 CC(C)CC(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217592265 CE For-Sale Unstable ANPEP 27 43 CC(C)CC(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217592265 CE For-Sale Unstable AKR1C3 30 45 CC(C)CC(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217592265 CE For-Sale Unstable PDS 44 33 COc1ccc(C)cc1NC(=O)NCC1CCCCC1 ZINC000217592298 CH On-Demand Unstable STK17B 41 37 COc1ccc(C)cc1NC(=O)NCC1CCCCC1 ZINC000217592298 CH On-Demand Unstable QRFPR 42 37 O=C1O[C@@]2(CCCN(C(=O)c3ccc4noc(-c5ccccc5)c4c3)C2)c2ccccc21 ZINC000217592300 HJ For-Sale Unstable NPY5R 35 43 CCO[C@H]1C[C@H](NC(=O)c2cccnc2Cl)C1(C)C ZINC000217592312 CF For-Sale Unstable G2YM83_BOTF4 87 43 CCCCNc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O ZINC000217592334 ED In-Stock Unstable CASP3 16 46 COC(=O)C[C@@H](C1=C(O)C(=O)c2ccccc2C1=O)c1cc(OC)c(O)c(OC)c1 ZINC000217592350 HF In-Stock Unstable TNF 21 41 O=C(O)/C=C\c1cccc(CNC(=O)C2CCCCC2)c1 ZINC000217592359 CF For-Sale Unstable NR1H4 28 43 O=C(O)/C=C\c1cccc(CNC(=O)C2CCCCC2)c1 ZINC000217592359 CF For-Sale Unstable HDAC6 24 48 NC[C@@H]1CCCCN1[C@@H]1CCN(Cc2ccccc2)C1 ZINC000217592364 CE For-Sale Unstable DRD4 32 45 NC[C@@H]1CCCCN1[C@@H]1CCN(Cc2ccccc2)C1 ZINC000217592364 CE For-Sale Unstable ACHE 25 44 NC[C@@H]1CCCCN1[C@@H]1CCN(Cc2ccccc2)C1 ZINC000217592364 CE For-Sale Unstable SIGMAR1 64 45 NC[C@@H]1CCCCN1[C@@H]1CCN(Cc2ccccc2)C1 ZINC000217592364 CE For-Sale Unstable SLC18A3 25 40 O=C1O[C@]2(CCCN(C(=O)c3ccc4noc(-c5ccccc5)c4c3)C2)c2ccccc21 ZINC000217592370 HJ For-Sale Unstable NPY5R 35 43 COC(=O)c1ccc(C(=O)N2CCC(N3CCC(Oc4nccs4)CC3)CC2)cc1 ZINC000217592372 IG In-Stock Unstable CHRM2 38 41 COC(=O)c1ccc(C(=O)N2CCC(N3CCC(Oc4nccs4)CC3)CC2)cc1 ZINC000217592372 IG In-Stock Unstable HRH1 18 41 COC(=O)c1ccc(C(=O)N2CCC(N3CCC(Oc4nccs4)CC3)CC2)cc1 ZINC000217592372 IG In-Stock Unstable HRH3 26 40 COC(=O)c1ccc(C(=O)N2CCC(N3CCC(Oc4nccs4)CC3)CC2)cc1 ZINC000217592372 IG In-Stock Unstable CCR3 24 41 COC(=O)c1ccc(C(=O)N2CCC(N3CCC(Oc4nccs4)CC3)CC2)cc1 ZINC000217592372 IG In-Stock Unstable L3MBTL1 0 51 COC(=O)c1ccc(C(=O)N2CCC(N3CCC(Oc4nccs4)CC3)CC2)cc1 ZINC000217592372 IG In-Stock Unstable L3MBTL3 110 51 COC(=O)c1ccc(C(=O)N2CCC(N3CCC(Oc4nccs4)CC3)CC2)cc1 ZINC000217592372 IG In-Stock Unstable L3MBTL4 0 46 COC(=O)c1ccc(C(=O)N2CCC(N3CCC(Oc4nccs4)CC3)CC2)cc1 ZINC000217592372 IG In-Stock Unstable MBTD1 0 50 COC(=O)c1ccc(C(=O)N2CCC(N3CCC(Oc4nccs4)CC3)CC2)cc1 ZINC000217592372 IG In-Stock Unstable TP53BP1 0 46 Cc1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217592384 BH On-Demand Unstable LPL 47 33 Cc1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217592384 BH On-Demand Unstable CCKAR 39 51 Cc1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217592384 BH On-Demand Unstable CCR3 49 44 Cc1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217592384 BH On-Demand Unstable KDR 17 42 Cc1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217592384 BH On-Demand Unstable CCKBR 47 44 Cc1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217592384 BH On-Demand Unstable EPHX2 30 72 Cc1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217592384 BH On-Demand Unstable PRMT3 35 41 Cc1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217592384 BH On-Demand Unstable ACAT 0 57 Cc1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217592384 BH On-Demand Unstable PSBA 0 45 Cc1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217592384 BH On-Demand Unstable KCNK3 62 42 Cc1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217592384 BH On-Demand Unstable KCNK9 60 42 COC(=O)C[C@H](C1=C(O)C(=O)c2ccccc2C1=O)c1cc(OC)c(O)c(OC)c1 ZINC000217592420 HF In-Stock Unstable TNF 21 41 CC[C@@H](C)C(=O)N(C)Cc1ccc(/C=C\C(=O)O)cc1 ZINC000217592435 CF For-Sale Unstable NR1H4 24 40 CC(C)CNc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O ZINC000217592440 ED In-Stock Unstable CASP3 17 45 CC(C)CNc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O ZINC000217592440 ED In-Stock Unstable MTNN 40 32 COc1cccc2cc(C(=O)N3CCC(N4CCC(Oc5nccs5)CC4)CC3)oc12 ZINC000217592450 II In-Stock Unstable CHRM2 44 41 COc1cccc2cc(C(=O)N3CCC(N4CCC(Oc5nccs5)CC4)CC3)oc12 ZINC000217592450 II In-Stock Unstable L3MBTL1 0 41 COc1cccc2cc(C(=O)N3CCC(N4CCC(Oc5nccs5)CC4)CC3)oc12 ZINC000217592450 II In-Stock Unstable L3MBTL3 76 41 O=C1O[C@@]2(CCCN(C(=O)Cn3cnc4ccccc43)C2)c2ccccc21 ZINC000217592466 FF For-Sale Unstable NPY5R 30 41 NC[C@@H]1CCCCN1[C@@H]1CCCN(Cc2ccccc2)C1 ZINC000217592485 CE For-Sale Unstable SLC6A1 45 33 NC[C@@H]1CCCCN1[C@@H]1CCCN(Cc2ccccc2)C1 ZINC000217592485 CE For-Sale Unstable SIGMAR1 59 46 O=C(NCC1CCCCC1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217592491 EK For-Sale Unstable DHODH 0 40 O=C(NCC1CCCCC1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217592491 EK For-Sale Unstable P2RX7 17 40 O=C(NCC1CCCCC1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217592491 EK For-Sale Unstable GUAB 0 44 O=C(NCC1CCCCC1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217592491 EK For-Sale Unstable RAF1 44 48 O=C(NCC1CCCCC1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217592491 EK For-Sale Unstable EPHX2 49 63 O=C(NCC1CCCCC1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217592491 EK For-Sale Unstable Q8MMZ8_EIMTE 67 51 O=C(NCC1CCCCC1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217592491 EK For-Sale Unstable CACNA1I 57 37 O=C(NCC1CCCCC1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217592491 EK For-Sale Unstable BRAF 17 48 O=C(NCC1CCCCC1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217592491 EK For-Sale Unstable PTPA 0 45 O=C(NCC1CCCCC1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217592491 EK For-Sale Unstable RIPK1 15 42 O=C(NCC1CCCCC1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217592491 EK For-Sale Unstable PRMT3 36 43 O=C(NCC1CCCCC1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217592491 EK For-Sale Unstable IMDH_CRYPV 23 46 O=C(NCC1CCCCC1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217592491 EK For-Sale Unstable BLM 0 46 O=C1O[C@]2(CCCN(C(=O)Cn3cnc4ccccc43)C2)c2ccccc21 ZINC000217592509 FF For-Sale Unstable NPY5R 30 41 CC[C@H](C)C(=O)N(C)Cc1ccc(/C=C\C(=O)O)cc1 ZINC000217592519 CF For-Sale Unstable NR1H4 24 40 O=C([C@H]1CC=CCC1)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217592530 GG In-Stock Unstable L3MBTL3 63 37 CC[C@@H](C)Nc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O ZINC000217592544 ED In-Stock Unstable CASP3 17 43 Nc1ccc(NC(=O)NCC2CCCCC2)c(Cl)c1 ZINC000217592569 CH For-Sale Unstable HTR4 16 40 Nc1ccc(NC(=O)NCC2CCCCC2)c(Cl)c1 ZINC000217592569 CH For-Sale Unstable CACNA1I 42 35 CCS(=O)(=O)Nc1ccc(C(=O)NCCc2nc3ccccc3n2C)cc1 ZINC000217592581 GE In-Stock Unstable PYGM 44 43 CCS(=O)(=O)Nc1ccc(C(=O)NCCc2nc3ccccc3n2C)cc1 ZINC000217592581 GE In-Stock Unstable NOD1 17 44 C=C(CC)COc1c(Br)cccc1/C=C\C(=O)O ZINC000217592583 DH For-Sale Unstable PTGER2 44 39 O=C([C@@H]1CC=CCC1)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217592606 GG In-Stock Unstable L3MBTL3 63 37 CC[C@H](C)Nc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O ZINC000217592628 ED In-Stock Unstable CASP3 17 43 COC(=O)c1ccccc1C(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217592643 FF For-Sale Unstable NPY5R 32 46 Nc1ccc(NC(=O)NCC2CCCCC2)cc1Cl ZINC000217592656 CH For-Sale Unstable HTR4 28 44 Nc1ccc(NC(=O)NCC2CCCCC2)cc1Cl ZINC000217592656 CH For-Sale Unstable EPHX2 18 65 Nc1ccc(NC(=O)NCC2CCCCC2)cc1Cl ZINC000217592656 CH For-Sale Unstable PRMT3 36 42 COC(=O)c1ccccc1C(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217592723 FF For-Sale Unstable NPY5R 32 46 CC(C)(C)Nc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O ZINC000217592727 ED In-Stock Unstable CASP3 16 43 Cc1cc(I)ccc1NC(=O)NCC1CCCCC1 ZINC000217592731 FI For-Sale Unstable LDLR 0 43 Cc1cc(I)ccc1NC(=O)NCC1CCCCC1 ZINC000217592731 FI For-Sale Unstable MAP2K1 21 44 O=C(O)/C=C\c1cnc(NC(=O)CCn2cncn2)s1 ZINC000217592744 CC For-Sale Unstable HIS3 44 30 CSc1ccc(CCC(=O)N2CCC(N3CCC(Oc4nccs4)CC3)CC2)cc1 ZINC000217592745 II In-Stock Unstable L3MBTL3 65 35 CCO[C@@H]1C[C@@H](NC(=O)c2ccc(Cl)nc2)C1(C)C ZINC000217592765 CF For-Sale Unstable SSTR5 24 42 C=C(CC)COc1ccc(/C=C\C(=O)O)cc1Cl ZINC000217592780 CH For-Sale Unstable AKR1C3 31 47 C=C(CC)COc1ccc(/C=C\C(=O)O)cc1Cl ZINC000217592780 CH For-Sale Unstable NR0B2 0 42 O=C(Nc1ccccc1Br)C(F)F ZINC000217592799 CF On-Demand Anodyne CXCR2 15 48 CCO[C@H]1C[C@@H](NC(=O)c2ccc(Cl)nc2)C1(C)C ZINC000217592821 CF For-Sale Unstable SSTR5 24 42 C=CCN(CC=C)C(=O)NCC1CCCCC1 ZINC000217592828 BF On-Demand Unstable ADH4 0 43 C=CCNc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O ZINC000217592835 DC In-Stock Unstable CASP3 0 42 C=CCNc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O ZINC000217592835 DC In-Stock Unstable BDKRB1 0 41 O=C1O[C@@]2(CCCN(C(=O)c3cccc(F)c3)C2)c2ccccc21 ZINC000217592836 EG For-Sale Unstable NPY5R 36 49 Clc1ccc2c(c1)[C@H](Cl)CCO2 ZINC000217592845 BG For-Sale Unstable AKR1B1 15 59 Cc1ccc2cccc(C(=O)N3CCC(N4CCC(Oc5nccs5)CC4)CC3)c2n1 ZINC000217592850 II In-Stock Unstable CHRM2 41 42 Cc1ccc2cccc(C(=O)N3CCC(N4CCC(Oc5nccs5)CC4)CC3)c2n1 ZINC000217592850 II In-Stock Unstable HRH1 17 44 Cc1ccc2cccc(C(=O)N3CCC(N4CCC(Oc5nccs5)CC4)CC3)c2n1 ZINC000217592850 II In-Stock Unstable CCR3 22 44 Cc1ccc2cccc(C(=O)N3CCC(N4CCC(Oc5nccs5)CC4)CC3)c2n1 ZINC000217592850 II In-Stock Unstable L3MBTL1 0 43 Cc1ccc2cccc(C(=O)N3CCC(N4CCC(Oc5nccs5)CC4)CC3)c2n1 ZINC000217592850 II In-Stock Unstable L3MBTL3 83 43 Cc1ccc2cccc(C(=O)N3CCC(N4CCC(Oc5nccs5)CC4)CC3)c2n1 ZINC000217592850 II In-Stock Unstable MBTD1 0 40 Cc1ccc2cccc(C(=O)N3CCC(N4CCC(Oc5nccs5)CC4)CC3)c2n1 ZINC000217592850 II In-Stock Unstable TP53BP1 0 43 NC(=O)c1ccc(NC(=O)CC[C@@H]2NC(=O)N(Cc3ccccc3)C2=O)cc1 ZINC000217592851 GD In-Stock Unstable ACHE 16 40 NC(=O)c1ccc(NC(=O)CC[C@@H]2NC(=O)N(Cc3ccccc3)C2=O)cc1 ZINC000217592851 GD In-Stock Unstable PROTEASE 0 40 O=C(c1ccccc1)N(OCc1ccccc1)N(OCc1ccccc1)C(=O)c1ccccc1 ZINC000217592884 JK For-Sale Unstable SRD5A2 18 41 O=C(c1ccccc1)N(OCc1ccccc1)N(OCc1ccccc1)C(=O)c1ccccc1 ZINC000217592884 JK For-Sale Unstable CAPN2 43 30 O=C(c1ccccc1)N(OCc1ccccc1)N(OCc1ccccc1)C(=O)c1ccccc1 ZINC000217592884 JK For-Sale Unstable NPR 43 33 O=C(c1ccccc1)N(OCc1ccccc1)N(OCc1ccccc1)C(=O)c1ccccc1 ZINC000217592884 JK For-Sale Unstable MLYCD 15 40 CCO[C@@H]1C[C@H](NC(=O)c2ccc(Cl)nc2)C1(C)C ZINC000217592898 CF For-Sale Unstable SSTR5 24 42 Brc1cc(CN2CCNCC2)c[nH]1 ZINC000217592910 BD For-Sale Unstable CXCR4 24 47 O=C(NCC1CCCCC1)N1CCN(Cc2ccccc2)CC1 ZINC000217592911 DG On-Demand Unstable CHRM2 28 41 O=C(NCC1CCCCC1)N1CCN(Cc2ccccc2)CC1 ZINC000217592911 DG On-Demand Unstable HTR1A 22 43 O=C(NCC1CCCCC1)N1CCN(Cc2ccccc2)CC1 ZINC000217592911 DG On-Demand Unstable DRD2 38 48 O=C(NCC1CCCCC1)N1CCN(Cc2ccccc2)CC1 ZINC000217592911 DG On-Demand Unstable DRD4 60 41 O=C(NCC1CCCCC1)N1CCN(Cc2ccccc2)CC1 ZINC000217592911 DG On-Demand Unstable ACHE 45 45 O=C(NCC1CCCCC1)N1CCN(Cc2ccccc2)CC1 ZINC000217592911 DG On-Demand Unstable SLC6A1 0 41 O=C(NCC1CCCCC1)N1CCN(Cc2ccccc2)CC1 ZINC000217592911 DG On-Demand Unstable DRD3 32 44 O=C(NCC1CCCCC1)N1CCN(Cc2ccccc2)CC1 ZINC000217592911 DG On-Demand Unstable HTR4 39 46 O=C(NCC1CCCCC1)N1CCN(Cc2ccccc2)CC1 ZINC000217592911 DG On-Demand Unstable CHRM3 31 44 O=C(NCC1CCCCC1)N1CCN(Cc2ccccc2)CC1 ZINC000217592911 DG On-Demand Unstable GRIN2B 43 38 O=C(NCC1CCCCC1)N1CCN(Cc2ccccc2)CC1 ZINC000217592911 DG On-Demand Unstable LTA4H 31 44 O=C(NCC1CCCCC1)N1CCN(Cc2ccccc2)CC1 ZINC000217592911 DG On-Demand Unstable VACHT_TETCF 0 46 O=C(NCC1CCCCC1)N1CCN(Cc2ccccc2)CC1 ZINC000217592911 DG On-Demand Unstable HRH3 27 47 O=C(NCC1CCCCC1)N1CCN(Cc2ccccc2)CC1 ZINC000217592911 DG On-Demand Unstable SIGMAR1 86 49 O=C(NCC1CCCCC1)N1CCN(Cc2ccccc2)CC1 ZINC000217592911 DG On-Demand Unstable CACNA1B 26 42 O=C(NCC1CCCCC1)N1CCN(Cc2ccccc2)CC1 ZINC000217592911 DG On-Demand Unstable BCHE 23 44 O=C(NCC1CCCCC1)N1CCN(Cc2ccccc2)CC1 ZINC000217592911 DG On-Demand Unstable CCR3 49 48 O=C(NCC1CCCCC1)N1CCN(Cc2ccccc2)CC1 ZINC000217592911 DG On-Demand Unstable CCR5 23 43 O=C(NCC1CCCCC1)N1CCN(Cc2ccccc2)CC1 ZINC000217592911 DG On-Demand Unstable FAAH 35 47 O=C(NCC1CCCCC1)N1CCN(Cc2ccccc2)CC1 ZINC000217592911 DG On-Demand Unstable MCHR1 29 41 O=C(NCC1CCCCC1)N1CCN(Cc2ccccc2)CC1 ZINC000217592911 DG On-Demand Unstable CACNA1G 34 44 O=C(NCC1CCCCC1)N1CCN(Cc2ccccc2)CC1 ZINC000217592911 DG On-Demand Unstable CACNA1I 49 41 O=C(NCC1CCCCC1)N1CCN(Cc2ccccc2)CC1 ZINC000217592911 DG On-Demand Unstable MGLL 0 46 O=C(NCC1CCCCC1)N1CCN(Cc2ccccc2)CC1 ZINC000217592911 DG On-Demand Unstable BIRC2 30 41 O=C(NCC1CCCCC1)N1CCN(Cc2ccccc2)CC1 ZINC000217592911 DG On-Demand Unstable ABHD6 0 43 O=C(NCC1CCCCC1)N1CCN(Cc2ccccc2)CC1 ZINC000217592911 DG On-Demand Unstable NPFFR1 53 37 O=C(NCC1CCCCC1)N1CCN(Cc2ccccc2)CC1 ZINC000217592911 DG On-Demand Unstable SLC12A5 26 42 O=C(NCC1CCCCC1)N1CCN(Cc2ccccc2)CC1 ZINC000217592911 DG On-Demand Unstable ADIPOR1 0 40 O=C(NCC1CCCCC1)N1CCN(Cc2ccccc2)CC1 ZINC000217592911 DG On-Demand Unstable ADIPOR2 0 40 O=C1O[C@]2(CCCN(C(=O)c3cccc(F)c3)C2)c2ccccc21 ZINC000217592919 EG For-Sale Unstable NPY5R 36 49 Clc1ccc2c(c1)[C@@H](Cl)CCO2 ZINC000217592926 BG For-Sale Unstable AKR1B1 15 59 O=C(c1cc(-c2ccccc2)n[nH]1)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217592957 IH In-Stock Unstable HRH1 17 43 O=C(c1cc(-c2ccccc2)n[nH]1)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217592957 IH In-Stock Unstable CCR3 32 43 O=C(c1cc(-c2ccccc2)n[nH]1)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217592957 IH In-Stock Unstable TACR3 19 45 O=C(c1cc(-c2ccccc2)n[nH]1)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217592957 IH In-Stock Unstable L3MBTL1 0 41 O=C(c1cc(-c2ccccc2)n[nH]1)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217592957 IH In-Stock Unstable L3MBTL3 85 41 O=C(c1cc(-c2ccccc2)n[nH]1)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217592957 IH In-Stock Unstable MBTD1 0 41 O=C(O)c1cc(S(=O)(=O)NCCCO)ccc1NC1CC1 ZINC000217592969 DC In-Stock Unstable TBXA2R 15 40 O=C(O)c1cc(S(=O)(=O)NCCCO)ccc1NC1CC1 ZINC000217592969 DC In-Stock Unstable CASP3 0 44 CCO[C@H]1C[C@H](NC(=O)c2ccc(Cl)nc2)C1(C)C ZINC000217592972 CF For-Sale Unstable SSTR5 24 42 COc1ccc2ccc(OC)c(C(=O)c3ccc([N+](=O)[O-])cc3)c2c1C(=O)c1ccc([N+](=O)[O-])cc1 ZINC000217592979 JK For-Sale Unstable KCNMA1 19 41 CCc1cccc(OCCOc2cc(C)ccc2C(N)=O)c1 ZINC000217592987 CG On-Demand Unstable MAOB 19 40 CCc1cccc(OCCOc2cc(C)ccc2C(N)=O)c1 ZINC000217592987 CG On-Demand Unstable PLA2G2A 42 39 O=C(Nc1ccc(Br)cc1)C(F)F ZINC000217592995 CF On-Demand Anodyne IDO1 20 40 O=C1O[C@@]2(CCCN(C(=O)CN3C(=O)c4ccccc4C3=O)C2)c2ccccc21 ZINC000217593033 GD For-Sale Unstable NPY5R 28 40 CN1CCN(C(=O)NCC2CCCCC2)CC1 ZINC000217593036 BD On-Demand Unstable DPP7 15 40 CN1CCN(C(=O)NCC2CCCCC2)CC1 ZINC000217593036 BD On-Demand Unstable CACNA1I 47 34 O=C(O)c1cc(S(=O)(=O)NCCCO)ccc1NC1CCCC1 ZINC000217593066 ED In-Stock Unstable CASP3 0 47 O=C(Cc1c(F)cccc1Cl)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217593072 II In-Stock Unstable HRH1 19 41 O=C(Cc1c(F)cccc1Cl)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217593072 II In-Stock Unstable CCR3 30 43 O=C(Cc1c(F)cccc1Cl)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217593072 II In-Stock Unstable SCD 20 43 O=C(Cc1c(F)cccc1Cl)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217593072 II In-Stock Unstable L3MBTL3 50 34 Cc1ccc(C(N)=O)c(OCCOc2cc(Cl)ccc2Cl)c1 ZINC000217593084 EH On-Demand Unstable S1PR4 39 47 O=C1O[C@]2(CCCN(C(=O)CN3C(=O)c4ccccc4C3=O)C2)c2ccccc21 ZINC000217593095 GD For-Sale Unstable NPY5R 28 40 O=C(NCC1CCCCC1)NC1CCCCCCCCCCC1 ZINC000217593108 DK For-Sale Unstable ADH1B 0 41 O=C(NCC1CCCCC1)NC1CCCCCCCCCCC1 ZINC000217593108 DK For-Sale Unstable ADH1C 0 41 O=C(NCC1CCCCC1)NC1CCCCCCCCCCC1 ZINC000217593108 DK For-Sale Unstable ADH4 0 41 O=C(NCC1CCCCC1)NC1CCCCCCCCCCC1 ZINC000217593108 DK For-Sale Unstable EPHX2 31 56 O=C(NCC1CCCCC1)NC1CCCCCCCCCCC1 ZINC000217593108 DK For-Sale Unstable P95276_MYCTO 0 43 O=C(O)c1cc(S(=O)(=O)NCCCO)ccc1NC1CCCCC1 ZINC000217593155 FD In-Stock Unstable CASP3 0 46 Cc1cccc(NC(=O)C(F)F)c1 ZINC000217593182 AE On-Demand Unstable CCKAR 24 44 Cc1cccc(NC(=O)C(F)F)c1 ZINC000217593182 AE On-Demand Unstable F12 0 43 Cc1cccc(NC(=O)C(F)F)c1 ZINC000217593182 AE On-Demand Unstable TAAR1 18 40 Cc1cccc(NC(=O)C(F)F)c1 ZINC000217593182 AE On-Demand Unstable AKR1C3 18 44 Cc1cccc(NC(=O)C(F)F)c1 ZINC000217593182 AE On-Demand Unstable PARP14 42 35 Cc1cccc(NC(=O)C(F)F)c1 ZINC000217593182 AE On-Demand Unstable PARP15 47 35 Cc1cccc(NC(=O)C(F)F)c1 ZINC000217593182 AE On-Demand Unstable PSBA 0 57 Cc1cccc(NC(=O)C(F)F)c1 ZINC000217593182 AE On-Demand Unstable KCNK3 101 53 Cc1cccc(NC(=O)C(F)F)c1 ZINC000217593182 AE On-Demand Unstable KCNK9 94 53 Cc1cccc(NC(=O)C(F)F)c1 ZINC000217593182 AE On-Demand Unstable PARP10 63 38 O=C(c1ccc(Br)o1)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217593195 IH In-Stock Unstable CHRM2 20 41 O=C(c1ccc(Br)o1)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217593195 IH In-Stock Unstable L3MBTL1 0 54 O=C(c1ccc(Br)o1)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217593195 IH In-Stock Unstable L3MBTL3 91 54 O=C(c1ccc(Br)o1)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217593195 IH In-Stock Unstable MBTD1 0 41 O=C1O[C@@]2(CCCN(C(=O)Cc3noc4ccccc34)C2)c2ccccc21 ZINC000217593200 FG For-Sale Unstable NPY5R 24 41 CN1CCC(c2cc(Br)n[nH]2)CC1 ZINC000217593205 BD For-Sale Unstable PKNB 29 40 O=C1O[C@]2(CCCN(C(=O)Cc3noc4ccccc34)C2)c2ccccc21 ZINC000217593260 FG For-Sale Unstable NPY5R 24 41 O=C(c1ccccc1)[C@H]1[C@H]2C(=O)N(c3cccc(C(F)(F)F)c3)C(=O)[C@H]2[C@H]2CCCN12 ZINC000217593262 IH In-Stock Unstable ME1 0 42 O=C(c1ccccc1)[C@H]1[C@H]2C(=O)N(c3cccc(C(F)(F)F)c3)C(=O)[C@H]2[C@H]2CCCN12 ZINC000217593262 IH In-Stock Unstable PDS 18 40 Cc1cc(C)n(-c2ccc(C(=O)NO)cc2)n1 ZINC000217593279 BD In-Stock Unstable HDAC8 22 42 Cc1cc(C)n(-c2ccc(C(=O)NO)cc2)n1 ZINC000217593279 BD In-Stock Unstable HDAC6 26 44 Cn1cc(-c2ccc(Oc3nccnc3-c3ccncc3)cc2)c2ncccc21 ZINC000217593306 GJ Annotated Unstable BRAF 21 41 O=C(Cc1cccc2ccccc12)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217593318 II In-Stock Unstable CHRM2 33 44 O=C(Cc1cccc2ccccc12)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217593318 II In-Stock Unstable CCR3 27 42 O=C(Cc1cccc2ccccc12)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217593318 II In-Stock Unstable L3MBTL3 68 39 O=C(Cc1cccc2ccccc12)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217593318 II In-Stock Unstable ETHR 42 36 Cc1ccccc1NC(=O)C(F)F ZINC000217593321 AE On-Demand Unstable CXCL8 44 38 Cc1ccccc1NC(=O)C(F)F ZINC000217593321 AE On-Demand Unstable KCNQ2 47 38 Cc1ccccc1NC(=O)C(F)F ZINC000217593321 AE On-Demand Unstable DDX3X 0 48 O=C(O)c1cc(S(=O)(=O)NCCCO)ccc1NCCO ZINC000217593365 DB In-Stock Unstable CASP3 17 42 O=C(O)c1cc(S(=O)(=O)NCCCO)ccc1NCCO ZINC000217593365 DB In-Stock Unstable BDKRB1 0 42 O=C(NCC(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12)c1ccccc1 ZINC000217593379 FE For-Sale Unstable NPY5R 30 43 O=C(O)/C=C\c1cccc(CNC(=O)C2CCCC2)c1 ZINC000217593393 CF For-Sale Unstable NR1H4 27 42 O=C(O)/C=C\c1cccc(CNC(=O)C2CCCC2)c1 ZINC000217593393 CF For-Sale Unstable HDAC6 25 46 Cc1ccc(CNC(=O)NCC2CCCCC2)cc1 ZINC000217593397 CG On-Demand Unstable MMP2 40 33 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)NCC(C)C)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217593409 JG In-Stock Unstable TUBA1A 19 71 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)NCC(C)C)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217593409 JG In-Stock Unstable TPPP 0 67 CC(C)(C)c1ccc(C(=O)N2CCC(N3CCC(Oc4nccs4)CC3)CC2)cc1 ZINC000217593445 IJ In-Stock Unstable CHRM2 26 41 CC(C)(C)c1ccc(C(=O)N2CCC(N3CCC(Oc4nccs4)CC3)CC2)cc1 ZINC000217593445 IJ In-Stock Unstable HRH1 17 41 CC(C)(C)c1ccc(C(=O)N2CCC(N3CCC(Oc4nccs4)CC3)CC2)cc1 ZINC000217593445 IJ In-Stock Unstable HRH3 23 40 CC(C)(C)c1ccc(C(=O)N2CCC(N3CCC(Oc4nccs4)CC3)CC2)cc1 ZINC000217593445 IJ In-Stock Unstable CCR3 22 41 CC(C)(C)c1ccc(C(=O)N2CCC(N3CCC(Oc4nccs4)CC3)CC2)cc1 ZINC000217593445 IJ In-Stock Unstable L3MBTL1 0 51 CC(C)(C)c1ccc(C(=O)N2CCC(N3CCC(Oc4nccs4)CC3)CC2)cc1 ZINC000217593445 IJ In-Stock Unstable L3MBTL3 110 51 CC(C)(C)c1ccc(C(=O)N2CCC(N3CCC(Oc4nccs4)CC3)CC2)cc1 ZINC000217593445 IJ In-Stock Unstable L3MBTL4 0 46 CC(C)(C)c1ccc(C(=O)N2CCC(N3CCC(Oc4nccs4)CC3)CC2)cc1 ZINC000217593445 IJ In-Stock Unstable MBTD1 0 50 CC(C)(C)c1ccc(C(=O)N2CCC(N3CCC(Oc4nccs4)CC3)CC2)cc1 ZINC000217593445 IJ In-Stock Unstable TP53BP1 0 46 O=C(NCC(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12)c1ccccc1 ZINC000217593446 FE For-Sale Unstable NPY5R 30 43 CC[C@@H](C)[C@@H](C(=O)N1CCC[C@@H](Cl)C1)c1ccccc1 ZINC000217593464 CI For-Sale Unstable CHRM1 16 41 CC[C@@H](C)[C@@H](C(=O)N1CCC[C@@H](Cl)C1)c1ccccc1 ZINC000217593464 CI For-Sale Unstable ACE 46 44 CC[C@@H](C)[C@@H](C(=O)N1CCC[C@@H](Cl)C1)c1ccccc1 ZINC000217593464 CI For-Sale Unstable CHRM4 16 40 CC[C@@H](C)[C@@H](C(=O)N1CCC[C@@H](Cl)C1)c1ccccc1 ZINC000217593464 CI For-Sale Unstable MME 19 44 CC[C@@H](C)[C@@H](C(=O)N1CCC[C@@H](Cl)C1)c1ccccc1 ZINC000217593464 CI For-Sale Unstable CCR1 27 41 CC[C@@H](C)[C@@H](C(=O)N1CCC[C@@H](Cl)C1)c1ccccc1 ZINC000217593464 CI For-Sale Unstable DPP7 54 36 CC[C@@H](C)[C@@H](C(=O)N1CCC[C@@H](Cl)C1)c1ccccc1 ZINC000217593464 CI For-Sale Unstable XIAP 36 40 CC[C@@H](C)[C@@H](C(=O)N1CCC[C@@H](Cl)C1)c1ccccc1 ZINC000217593464 CI For-Sale Unstable RHODESAIN 0 40 O=C(O)c1cc(S(=O)(=O)NCCCO)ccc1NCCCO ZINC000217593469 EB In-Stock Unstable CASP3 17 43 COc1cccc(NC(=O)C(F)F)c1 ZINC000217593477 BD On-Demand Unstable CCR3 22 44 COc1cccc(NC(=O)C(F)F)c1 ZINC000217593477 BD On-Demand Unstable MTNR1A 38 55 COc1cccc(NC(=O)C(F)F)c1 ZINC000217593477 BD On-Demand Unstable MTNR1B 35 55 COc1cccc(NC(=O)C(F)F)c1 ZINC000217593477 BD On-Demand Unstable ACR 24 41 COc1cccc(NC(=O)C(F)F)c1 ZINC000217593477 BD On-Demand Unstable PDGFRA 22 41 COc1cccc(NC(=O)C(F)F)c1 ZINC000217593477 BD On-Demand Unstable ALS 51 31 COc1cccc(NC(=O)C(F)F)c1 ZINC000217593477 BD On-Demand Unstable TAAR1 40 53 COc1cccc(NC(=O)C(F)F)c1 ZINC000217593477 BD On-Demand Unstable AKR1C3 25 48 COc1cccc(NC(=O)C(F)F)c1 ZINC000217593477 BD On-Demand Unstable AKR1C2 52 39 COc1cccc(NC(=O)C(F)F)c1 ZINC000217593477 BD On-Demand Unstable PSBA 0 61 COc1cccc(NC(=O)C(F)F)c1 ZINC000217593477 BD On-Demand Unstable KCNK3 83 52 COc1cccc(NC(=O)C(F)F)c1 ZINC000217593477 BD On-Demand Unstable KCNK9 81 45 COc1cccc(NC(=O)C(F)F)c1 ZINC000217593477 BD On-Demand Unstable PARP10 0 41 COc1cccc(NC(=O)C(F)F)c1 ZINC000217593477 BD On-Demand Unstable BRPF1 0 42 COc1ccc(N2CCN(C(=O)CC/C(C)=C/Cc3c(O)c4c(c(C)c3OC)COC4=O)CC2)cc1 ZINC000217593502 JI In-Stock Unstable IMPDH1 0 64 COc1ccc(N2CCN(C(=O)CC/C(C)=C/Cc3c(O)c4c(c(C)c3OC)COC4=O)CC2)cc1 ZINC000217593502 JI In-Stock Unstable IMPDH2 0 64 CCN(C(=O)NCC1CCCCC1)c1ccccc1 ZINC000217593522 CH For-Sale Unstable AMY2 55 39 O=C(c1cc(-c2ccco2)[nH]n1)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217593540 IG In-Stock Unstable L3MBTL3 77 37 CC[C@H](C)[C@@H](C(=O)N1CCC[C@@H](Cl)C1)c1ccccc1 ZINC000217593553 CI For-Sale Unstable CHRM1 16 41 CC[C@H](C)[C@@H](C(=O)N1CCC[C@@H](Cl)C1)c1ccccc1 ZINC000217593553 CI For-Sale Unstable ACE 46 44 CC[C@H](C)[C@@H](C(=O)N1CCC[C@@H](Cl)C1)c1ccccc1 ZINC000217593553 CI For-Sale Unstable CHRM4 16 40 CC[C@H](C)[C@@H](C(=O)N1CCC[C@@H](Cl)C1)c1ccccc1 ZINC000217593553 CI For-Sale Unstable MME 19 44 CC[C@H](C)[C@@H](C(=O)N1CCC[C@@H](Cl)C1)c1ccccc1 ZINC000217593553 CI For-Sale Unstable CCR1 27 41 CC[C@H](C)[C@@H](C(=O)N1CCC[C@@H](Cl)C1)c1ccccc1 ZINC000217593553 CI For-Sale Unstable DPP7 54 36 CC[C@H](C)[C@@H](C(=O)N1CCC[C@@H](Cl)C1)c1ccccc1 ZINC000217593553 CI For-Sale Unstable XIAP 36 40 CC[C@H](C)[C@@H](C(=O)N1CCC[C@@H](Cl)C1)c1ccccc1 ZINC000217593553 CI For-Sale Unstable RHODESAIN 0 40 Cc1cc(C)cc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217593555 EH For-Sale Unstable NPY5R 31 41 COCCNc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O ZINC000217593592 EC In-Stock Unstable CASP3 17 41 COCCNc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O ZINC000217593592 EC In-Stock Unstable BDKRB1 0 44 COc1cc2cc(C(=O)N[C@H](CO)Cc3ccccc3)[nH]c2cc1OC ZINC000217593616 FF In-Stock Unstable ADRB2 23 41 COc1cc2cc(C(=O)N[C@H](CO)Cc3ccccc3)[nH]c2cc1OC ZINC000217593616 FF In-Stock Unstable CYP51A1 22 42 COc1cc2cc(C(=O)N[C@H](CO)Cc3ccccc3)[nH]c2cc1OC ZINC000217593616 FF In-Stock Unstable PYGL 50 52 COc1cc2cc(C(=O)N[C@H](CO)Cc3ccccc3)[nH]c2cc1OC ZINC000217593616 FF In-Stock Unstable PAM 0 42 COc1cc2cc(C(=O)N[C@H](CO)Cc3ccccc3)[nH]c2cc1OC ZINC000217593616 FF In-Stock Unstable PIN1 38 40 COc1cc2cc(C(=O)N[C@H](CO)Cc3ccccc3)[nH]c2cc1OC ZINC000217593616 FF In-Stock Unstable BLA1_STEMA 23 42 COc1ccccc1NC(=O)C(F)F ZINC000217593620 BD On-Demand Unstable KCNK3 40 40 COc1ccccc1NC(=O)C(F)F ZINC000217593620 BD On-Demand Unstable KCNK9 39 40 NCc1cccc(CNC(=O)NCC2CCCCC2)c1 ZINC000217593621 CF For-Sale Unstable EPHX2 15 50 NCc1cccc(CNC(=O)NCC2CCCCC2)c1 ZINC000217593621 CF For-Sale Unstable TPSAB1 52 41 COc1ccc2cc(C(=O)N3CCC(N4CCC(Oc5nccs5)CC4)CC3)[nH]c2c1 ZINC000217593630 IH In-Stock Unstable CHRM2 51 43 COc1ccc2cc(C(=O)N3CCC(N4CCC(Oc5nccs5)CC4)CC3)[nH]c2c1 ZINC000217593630 IH In-Stock Unstable HRH1 19 41 COc1ccc2cc(C(=O)N3CCC(N4CCC(Oc5nccs5)CC4)CC3)[nH]c2c1 ZINC000217593630 IH In-Stock Unstable GRIN2B 26 48 COc1ccc2cc(C(=O)N3CCC(N4CCC(Oc5nccs5)CC4)CC3)[nH]c2c1 ZINC000217593630 IH In-Stock Unstable HRH3 30 49 COc1ccc2cc(C(=O)N3CCC(N4CCC(Oc5nccs5)CC4)CC3)[nH]c2c1 ZINC000217593630 IH In-Stock Unstable HRH4 20 40 COc1ccc2cc(C(=O)N3CCC(N4CCC(Oc5nccs5)CC4)CC3)[nH]c2c1 ZINC000217593630 IH In-Stock Unstable CCR3 33 41 COc1ccc2cc(C(=O)N3CCC(N4CCC(Oc5nccs5)CC4)CC3)[nH]c2c1 ZINC000217593630 IH In-Stock Unstable FPR2 28 44 COc1ccc2cc(C(=O)N3CCC(N4CCC(Oc5nccs5)CC4)CC3)[nH]c2c1 ZINC000217593630 IH In-Stock Unstable AKR1C3 0 41 COc1ccc2cc(C(=O)N3CCC(N4CCC(Oc5nccs5)CC4)CC3)[nH]c2c1 ZINC000217593630 IH In-Stock Unstable L3MBTL1 0 41 COc1ccc2cc(C(=O)N3CCC(N4CCC(Oc5nccs5)CC4)CC3)[nH]c2c1 ZINC000217593630 IH In-Stock Unstable L3MBTL3 76 41 Cc1cc(C)cc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217593640 EH For-Sale Unstable NPY5R 31 41 CC[C@@H](C)[C@H](C(=O)N1CCC[C@@H](Cl)C1)c1ccccc1 ZINC000217593650 CI For-Sale Unstable CHRM1 16 41 CC[C@@H](C)[C@H](C(=O)N1CCC[C@@H](Cl)C1)c1ccccc1 ZINC000217593650 CI For-Sale Unstable ACE 46 44 CC[C@@H](C)[C@H](C(=O)N1CCC[C@@H](Cl)C1)c1ccccc1 ZINC000217593650 CI For-Sale Unstable CHRM4 16 40 CC[C@@H](C)[C@H](C(=O)N1CCC[C@@H](Cl)C1)c1ccccc1 ZINC000217593650 CI For-Sale Unstable MME 19 44 CC[C@@H](C)[C@H](C(=O)N1CCC[C@@H](Cl)C1)c1ccccc1 ZINC000217593650 CI For-Sale Unstable CCR1 27 41 CC[C@@H](C)[C@H](C(=O)N1CCC[C@@H](Cl)C1)c1ccccc1 ZINC000217593650 CI For-Sale Unstable DPP7 54 36 CC[C@@H](C)[C@H](C(=O)N1CCC[C@@H](Cl)C1)c1ccccc1 ZINC000217593650 CI For-Sale Unstable XIAP 36 40 CC[C@@H](C)[C@H](C(=O)N1CCC[C@@H](Cl)C1)c1ccccc1 ZINC000217593650 CI For-Sale Unstable RHODESAIN 0 40 COCCCNc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O ZINC000217593709 EC In-Stock Unstable CASP3 17 40 COCCCNc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O ZINC000217593709 EC In-Stock Unstable BDKRB1 0 44 COc1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217593721 CG On-Demand Unstable DRD4 45 34 COc1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217593721 CG On-Demand Unstable HRH2 25 52 COc1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217593721 CG On-Demand Unstable TRPV1 0 48 COc1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217593721 CG On-Demand Unstable MTR1B_CHICK 0 40 COc1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217593721 CG On-Demand Unstable CCKAR 0 43 COc1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217593721 CG On-Demand Unstable NPY2R 0 41 COc1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217593721 CG On-Demand Unstable CCR3 61 55 COc1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217593721 CG On-Demand Unstable MTNR1A 63 49 COc1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217593721 CG On-Demand Unstable MTNR1B 44 46 COc1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217593721 CG On-Demand Unstable EPHX2 36 69 COc1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217593721 CG On-Demand Unstable Q8MMZ8_EIMTE 0 49 COc1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217593721 CG On-Demand Unstable TAAR1 35 40 COc1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217593721 CG On-Demand Unstable QRFPR 40 34 COc1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217593721 CG On-Demand Unstable PRMT3 34 40 COc1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217593721 CG On-Demand Unstable ACAT 0 61 COc1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217593721 CG On-Demand Unstable METAP2 0 60 COc1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217593721 CG On-Demand Unstable KCNK3 43 38 CCOc1ccccc1NC(=O)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217593733 II In-Stock Unstable CCR3 21 42 CCOc1ccccc1NC(=O)N1CCC(N2CCC(Oc3nccs3)CC2)CC1 ZINC000217593733 II In-Stock Unstable L3MBTL3 58 37 O=C(CN(c1ccccc1)c1ccccc1)NO ZINC000217593737 BE In-Stock Unstable HDAC8 39 46 O=C(CN(c1ccccc1)c1ccccc1)NO ZINC000217593737 BE In-Stock Unstable MMP16 0 41 O=C(CN(c1ccccc1)c1ccccc1)NO ZINC000217593737 BE In-Stock Unstable MMP2 0 41 O=C(CN(c1ccccc1)c1ccccc1)NO ZINC000217593737 BE In-Stock Unstable MMP3 0 42 O=C(CN(c1ccccc1)c1ccccc1)NO ZINC000217593737 BE In-Stock Unstable MMP8 29 41 O=C(CN(c1ccccc1)c1ccccc1)NO ZINC000217593737 BE In-Stock Unstable HDAC1 27 46 O=C(CN(c1ccccc1)c1ccccc1)NO ZINC000217593737 BE In-Stock Unstable HDAC2 31 44 O=C(CN(c1ccccc1)c1ccccc1)NO ZINC000217593737 BE In-Stock Unstable HDAC3 22 40 O=C(CN(c1ccccc1)c1ccccc1)NO ZINC000217593737 BE In-Stock Unstable HDAC6 28 41 O=C(CN(c1ccccc1)c1ccccc1)NO ZINC000217593737 BE In-Stock Unstable MMP9 0 41 O=C(CN(c1ccccc1)c1ccccc1)NO ZINC000217593737 BE In-Stock Unstable MMP1 27 42 O=C(CN(c1ccccc1)c1ccccc1)NO ZINC000217593737 BE In-Stock Unstable HDA106 0 46 O=C(CN(c1ccccc1)c1ccccc1)NO ZINC000217593737 BE In-Stock Unstable HD1B 0 46 O=C(CN(c1ccccc1)c1ccccc1)NO ZINC000217593737 BE In-Stock Unstable PFHDAC1 0 46 CC[C@H](C)[C@H](C(=O)N1CCC[C@@H](Cl)C1)c1ccccc1 ZINC000217593739 CI For-Sale Unstable CHRM1 16 41 CC[C@H](C)[C@H](C(=O)N1CCC[C@@H](Cl)C1)c1ccccc1 ZINC000217593739 CI For-Sale Unstable ACE 46 44 CC[C@H](C)[C@H](C(=O)N1CCC[C@@H](Cl)C1)c1ccccc1 ZINC000217593739 CI For-Sale Unstable CHRM4 16 40 CC[C@H](C)[C@H](C(=O)N1CCC[C@@H](Cl)C1)c1ccccc1 ZINC000217593739 CI For-Sale Unstable MME 19 44 CC[C@H](C)[C@H](C(=O)N1CCC[C@@H](Cl)C1)c1ccccc1 ZINC000217593739 CI For-Sale Unstable CCR1 27 41 CC[C@H](C)[C@H](C(=O)N1CCC[C@@H](Cl)C1)c1ccccc1 ZINC000217593739 CI For-Sale Unstable DPP7 54 36 CC[C@H](C)[C@H](C(=O)N1CCC[C@@H](Cl)C1)c1ccccc1 ZINC000217593739 CI For-Sale Unstable XIAP 36 40 CC[C@H](C)[C@H](C(=O)N1CCC[C@@H](Cl)C1)c1ccccc1 ZINC000217593739 CI For-Sale Unstable RHODESAIN 0 40 CC(C)CC(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217593747 CF For-Sale Unstable NPY5R 28 41 O=C(O)c1cc(S(=O)(=O)NCCCO)ccc1NCc1ccccc1 ZINC000217593804 FD In-Stock Unstable HTR7 15 42 O=C(O)c1cc(S(=O)(=O)NCCCO)ccc1NCc1ccccc1 ZINC000217593804 FD In-Stock Unstable CASP3 22 40 O=C(O)c1cc(S(=O)(=O)NCCCO)ccc1NCc1ccccc1 ZINC000217593804 FD In-Stock Unstable BDKRB1 0 43 CC(C)CC(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217593824 CF For-Sale Unstable NPY5R 28 41 Cn1cc(/C=C2/Oc3cc(OCC(=O)NCCn4ccnc4)ccc3C2=O)c2ccccc21 ZINC000217593840 IG In-Stock Unstable MTOR 0 43 CCOc1ccc(NC(=O)NCC2CCCCC2)cc1OCC ZINC000217593842 DI On-Demand Unstable HRH2 18 41 CCOc1ccc(NC(=O)NCC2CCCCC2)cc1OCC ZINC000217593842 DI On-Demand Unstable CCR3 40 37 CCOc1ccc(NC(=O)NCC2CCCCC2)cc1OCC ZINC000217593842 DI On-Demand Unstable EPHX2 28 58 CCOc1ccc(NC(=O)NCC2CCCCC2)cc1OCC ZINC000217593842 DI On-Demand Unstable QRFPR 41 33 CCOc1ccc(NC(=O)NCC2CCCCC2)cc1OCC ZINC000217593842 DI On-Demand Unstable PRMT3 36 44 CCOc1ccc(NC(=O)NCC2CCCCC2)cc1OCC ZINC000217593842 DI On-Demand Unstable HCN1 41 32 CCOc1ccc(NC(=O)NCC2CCCCC2)cc1OCC ZINC000217593842 DI On-Demand Unstable HCN4 41 33 CC1(C)OB(c2ccc(NS(=O)(=O)c3ccc(F)cc3)cc2)OC1(C)C ZINC000217593849 GF For-Sale Unstable MGAT1 49 34 Cc1ccc(S(=O)(=O)N2CCC(N3CCC(Oc4nccs4)CC3)CC2)cc1C ZINC000217593854 IG In-Stock Unstable CHRM2 20 42 Cc1ccc(NC(=O)C(F)F)c(C)c1 ZINC000217593860 AF On-Demand Unstable H9CNL0_SPOEX 43 35 C[C@@H](Nc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O)c1ccccc1 ZINC000217593904 GE In-Stock Unstable CASP3 19 43 C[C@@H](Nc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O)c1ccccc1 ZINC000217593904 GE In-Stock Unstable BDKRB1 0 45 O=C1O[C@@]2(CCCN(C(=O)c3ccc(Cl)cc3Cl)C2)c2ccccc21 ZINC000217593927 GI For-Sale Unstable AVPR1A 23 55 O=C1O[C@@]2(CCCN(C(=O)c3ccc(Cl)cc3Cl)C2)c2ccccc21 ZINC000217593927 GI For-Sale Unstable NPY5R 29 45 CSc1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217593956 CI On-Demand Unstable CCR3 51 52 CSc1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217593956 CI On-Demand Unstable EPHX2 23 67 CSc1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217593956 CI On-Demand Unstable ACAT 0 41 COc1cccc(S(=O)(=O)N2CCC(N3CCC(Oc4nccs4)CC3)CC2)c1 ZINC000217593960 IF In-Stock Unstable CHRM2 47 44 COc1cccc(S(=O)(=O)N2CCC(N3CCC(Oc4nccs4)CC3)CC2)c1 ZINC000217593960 IF In-Stock Unstable HRH1 18 41 COc1cccc(S(=O)(=O)N2CCC(N3CCC(Oc4nccs4)CC3)CC2)c1 ZINC000217593960 IF In-Stock Unstable CCR3 32 41 C[C@H](Nc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O)c1ccccc1 ZINC000217593981 GE In-Stock Unstable CASP3 19 43 C[C@H](Nc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O)c1ccccc1 ZINC000217593981 GE In-Stock Unstable BDKRB1 0 45 COc1cccc(CN(C)C(=O)C(F)F)c1 ZINC000217593999 BD On-Demand Unstable ACHE 0 53 COc1cccc(CN(C)C(=O)C(F)F)c1 ZINC000217593999 BD On-Demand Unstable TSPO 0 43 COc1cccc(CN(C)C(=O)C(F)F)c1 ZINC000217593999 BD On-Demand Unstable CETP 0 42 COc1cccc(CN(C)C(=O)C(F)F)c1 ZINC000217593999 BD On-Demand Unstable ROCK1 39 46 COc1cccc(CN(C)C(=O)C(F)F)c1 ZINC000217593999 BD On-Demand Unstable MTNR1A 35 44 COc1cccc(CN(C)C(=O)C(F)F)c1 ZINC000217593999 BD On-Demand Unstable MTNR1B 31 42 COc1cccc(CN(C)C(=O)C(F)F)c1 ZINC000217593999 BD On-Demand Unstable ROCK2 44 47 COc1cccc(CN(C)C(=O)C(F)F)c1 ZINC000217593999 BD On-Demand Unstable HSD17B2 48 57 COc1cccc(CN(C)C(=O)C(F)F)c1 ZINC000217593999 BD On-Demand Unstable FFAR1 18 41 COc1cccc(CN(C)C(=O)C(F)F)c1 ZINC000217593999 BD On-Demand Unstable CDC42BPA 0 47 O=C1O[C@]2(CCCN(C(=O)c3ccc(Cl)cc3Cl)C2)c2ccccc21 ZINC000217594018 GI For-Sale Unstable AVPR1A 23 55 O=C1O[C@]2(CCCN(C(=O)c3ccc(Cl)cc3Cl)C2)c2ccccc21 ZINC000217594018 GI For-Sale Unstable NPY5R 29 45 O=C(NCC1CCCCC1)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217594054 HG For-Sale Unstable LPL 50 40 O=C(NCC1CCCCC1)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217594054 HG For-Sale Unstable CNR2 0 40 O=C(NCC1CCCCC1)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217594054 HG For-Sale Unstable CASP3 0 41 O=C(NCC1CCCCC1)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217594054 HG For-Sale Unstable EPHX2 26 45 O=C(NCC1CCCCC1)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217594054 HG For-Sale Unstable PGA5 44 30 O=C(NCC1CCCCC1)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217594054 HG For-Sale Unstable MURF 0 42 O=C(NCC1CCCCC1)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217594054 HG For-Sale Unstable CACNA1I 59 36 O=C(NCC1CCCCC1)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217594054 HG For-Sale Unstable F13A1 48 37 O=C(NCC1CCCCC1)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217594054 HG For-Sale Unstable LIPG 20 40 O=C(NCC1CCCCC1)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217594054 HG For-Sale Unstable NAMPT 40 42 CC(C)[C@@H](CO)NC(=O)CC[C@@H]1NC(=O)N(Cc2ccccc2)C1=O ZINC000217594073 ED In-Stock Unstable GALR1 44 32 O=C(O)c1cc(S(=O)(=O)NCCCO)ccc1NCCc1ccccc1 ZINC000217594134 GD In-Stock Unstable TBXA2R 50 40 O=C(O)c1cc(S(=O)(=O)NCCCO)ccc1NCCc1ccccc1 ZINC000217594134 GD In-Stock Unstable HTR7 15 41 O=C(O)c1cc(S(=O)(=O)NCCCO)ccc1NCCc1ccccc1 ZINC000217594134 GD In-Stock Unstable CASP3 17 40 O=C(O)c1cc(S(=O)(=O)NCCCO)ccc1NCCc1ccccc1 ZINC000217594134 GD In-Stock Unstable BDKRB1 0 42 O=C1O[C@@]2(CCCN(C(=O)c3ccc(Cl)c(Cl)c3)C2)c2ccccc21 ZINC000217594137 GI For-Sale Unstable NPY5R 33 46 C[C@@H]1C[C@@H](C)CN(C(=O)NCC2CCCCC2)C1 ZINC000217594144 CG On-Demand Unstable DPP7 18 41 O=C(/C=C/c1ccc2c(c1)OCO2)N[C@@H]1C[C@@H]2C(=O)Nc3ccccc3N2C1 ZINC000217594149 GE In-Stock Unstable DYRK2 63 34 CN(CCOc1ccccc1)C(=O)C(F)F ZINC000217594151 BD On-Demand Unstable ALOX5 19 48 CN(CCOc1ccccc1)C(=O)C(F)F ZINC000217594151 BD On-Demand Unstable FDPS 26 45 CN(CCOc1ccccc1)C(=O)C(F)F ZINC000217594151 BD On-Demand Unstable LTA4H 27 41 CN(CCOc1ccccc1)C(=O)C(F)F ZINC000217594151 BD On-Demand Unstable ESRRG 49 37 CN(CCOc1ccccc1)C(=O)C(F)F ZINC000217594151 BD On-Demand Unstable NORA 0 42 CN(CCOc1ccccc1)C(=O)C(F)F ZINC000217594151 BD On-Demand Unstable EBPL 0 40 Cc1ccc(S(=O)(=O)NCCCCCBr)cc1 ZINC000217594168 DF For-Sale Unstable TBXAS1 30 41 Cc1ccc(S(=O)(=O)NCCCCCBr)cc1 ZINC000217594168 DF For-Sale Unstable ALOX15 46 45 Cc1ccc(S(=O)(=O)NCCCCCBr)cc1 ZINC000217594168 DF For-Sale Unstable CYP24A1 29 41 Cc1ccc(S(=O)(=O)NCCCCCBr)cc1 ZINC000217594168 DF For-Sale Unstable FFAR4 16 41 COC(=O)C[C@H](c1cc(OC)c(O)c(OC)c1)c1c(O)c2ccccc2oc1=O ZINC000217594205 HF In-Stock Unstable CYP2C9 17 41 COC(=O)C[C@H](c1cc(OC)c(O)c(OC)c1)c1c(O)c2ccccc2oc1=O ZINC000217594205 HF In-Stock Unstable NQO1 77 53 O=C(CCCCc1ccccc1)N1CCC[C@@H](c2nnc[nH]2)C1 ZINC000217594207 DF In-Stock Unstable FKBP1A 32 41 O=C(CCCCc1ccccc1)N1CCC[C@@H](c2nnc[nH]2)C1 ZINC000217594207 DF In-Stock Unstable PREP 68 48 O=C(CCCCc1ccccc1)N1CCC[C@@H](c2nnc[nH]2)C1 ZINC000217594207 DF In-Stock Unstable FAAH 46 41 O=C(CCCCc1ccccc1)N1CCC[C@@H](c2nnc[nH]2)C1 ZINC000217594207 DF In-Stock Unstable CES1 51 38 COc1ccc(CCNc2ccc(S(=O)(=O)NCCCO)cc2C(=O)O)cc1 ZINC000217594217 HD In-Stock Unstable CA2 17 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCCCO)cc2C(=O)O)cc1 ZINC000217594217 HD In-Stock Unstable TBXA2R 39 42 COc1ccc(CCNc2ccc(S(=O)(=O)NCCCO)cc2C(=O)O)cc1 ZINC000217594217 HD In-Stock Unstable TBXAS1 25 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCCCO)cc2C(=O)O)cc1 ZINC000217594217 HD In-Stock Unstable BMP1 53 36 COc1ccc(CCNc2ccc(S(=O)(=O)NCCCO)cc2C(=O)O)cc1 ZINC000217594217 HD In-Stock Unstable CA1 16 42 COc1ccc(CCNc2ccc(S(=O)(=O)NCCCO)cc2C(=O)O)cc1 ZINC000217594217 HD In-Stock Unstable MMP13 47 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCCCO)cc2C(=O)O)cc1 ZINC000217594217 HD In-Stock Unstable MMP2 27 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCCCO)cc2C(=O)O)cc1 ZINC000217594217 HD In-Stock Unstable MMP8 20 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCCCO)cc2C(=O)O)cc1 ZINC000217594217 HD In-Stock Unstable MMP9 43 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCCCO)cc2C(=O)O)cc1 ZINC000217594217 HD In-Stock Unstable MMP12 24 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCCCO)cc2C(=O)O)cc1 ZINC000217594217 HD In-Stock Unstable PTGDR 21 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCCCO)cc2C(=O)O)cc1 ZINC000217594217 HD In-Stock Unstable IAP 0 49 COc1ccc(CCNc2ccc(S(=O)(=O)NCCCO)cc2C(=O)O)cc1 ZINC000217594217 HD In-Stock Unstable CA9 23 42 COc1ccc(CCNc2ccc(S(=O)(=O)NCCCO)cc2C(=O)O)cc1 ZINC000217594217 HD In-Stock Unstable MMP1 44 36 COc1ccc(CCNc2ccc(S(=O)(=O)NCCCO)cc2C(=O)O)cc1 ZINC000217594217 HD In-Stock Unstable AKR1C3 29 45 COc1ccc(CCNc2ccc(S(=O)(=O)NCCCO)cc2C(=O)O)cc1 ZINC000217594217 HD In-Stock Unstable AKR1C2 50 37 O=C1O[C@]2(CCCN(C(=O)c3ccc(Cl)c(Cl)c3)C2)c2ccccc21 ZINC000217594236 GI For-Sale Unstable NPY5R 33 46 O=C(/C=C/c1ccc2c(c1)OCO2)N[C@@H]1C[C@H]2C(=O)Nc3ccccc3N2C1 ZINC000217594239 GE In-Stock Unstable DYRK2 63 34 C[C@H]1C[C@@H](C)CN(C(=O)NCC2CCCCC2)C1 ZINC000217594245 CG On-Demand Unstable DPP7 18 41 COC(=O)C[C@@H](c1cc(OC)c(O)c(OC)c1)c1c(O)c2ccccc2oc1=O ZINC000217594266 HF In-Stock Unstable CYP2C9 17 41 COC(=O)C[C@@H](c1cc(OC)c(O)c(OC)c1)c1c(O)c2ccccc2oc1=O ZINC000217594266 HF In-Stock Unstable NQO1 77 53 O=C(CCCCc1ccccc1)N1CCC[C@H](c2nnc[nH]2)C1 ZINC000217594276 DF In-Stock Unstable FKBP1A 32 41 O=C(CCCCc1ccccc1)N1CCC[C@H](c2nnc[nH]2)C1 ZINC000217594276 DF In-Stock Unstable PREP 68 48 O=C(CCCCc1ccccc1)N1CCC[C@H](c2nnc[nH]2)C1 ZINC000217594276 DF In-Stock Unstable FAAH 46 41 O=C(CCCCc1ccccc1)N1CCC[C@H](c2nnc[nH]2)C1 ZINC000217594276 DF In-Stock Unstable CES1 51 38 CCOc1ccc(CN(C)C(=O)C(F)F)cc1 ZINC000217594288 BE On-Demand Unstable ALOX5 15 41 C[C@H]1C[C@H](C)CN(C(=O)NCC2CCCCC2)C1 ZINC000217594306 CG On-Demand Unstable DPP7 18 41 COC(=O)[C@@H]1Cc2ccccc2CN1Cc1csc(COc2ccc(C)cc2)n1 ZINC000217594309 HI On-Demand Unstable OPRM1 0 41 COC(=O)[C@@H]1Cc2ccccc2CN1Cc1csc(COc2ccc(C)cc2)n1 ZINC000217594309 HI On-Demand Unstable OPRD1 45 32 COC(=O)[C@@H]1Cc2ccccc2CN1Cc1csc(COc2ccc(C)cc2)n1 ZINC000217594309 HI On-Demand Unstable ADAM9 61 35 COc1ccc(CCNc2ccc(S(=O)(=O)NCCCO)cc2C(=O)O)cc1OC ZINC000217594326 ID In-Stock Unstable TBXAS1 18 44 COc1ccc(CCNc2ccc(S(=O)(=O)NCCCO)cc2C(=O)O)cc1OC ZINC000217594326 ID In-Stock Unstable PTGDR 18 40 COc1ccc(CCNc2ccc(S(=O)(=O)NCCCO)cc2C(=O)O)cc1OC ZINC000217594326 ID In-Stock Unstable IAP 0 50 COc1ccc(CCNc2ccc(S(=O)(=O)NCCCO)cc2C(=O)O)cc1OC ZINC000217594326 ID In-Stock Unstable SCMU_MYCTU 0 44 O=C1O[C@@]2(CCCN(C(=O)C3CC3)C2)c2ccccc21 ZINC000217594337 CE In-Stock Unstable NPY5R 54 44 NC[C@@H]1CCCCN1C(=O)/C=C\c1ccccc1 ZINC000217594372 BE On-Demand Unstable CPT1A 64 35 NC[C@@H]1CCCCN1C(=O)/C=C\c1ccccc1 ZINC000217594372 BE On-Demand Unstable PREP 44 36 NC[C@@H]1CCCCN1C(=O)/C=C\c1ccccc1 ZINC000217594372 BE On-Demand Unstable 17HSDCL 0 40 COC(=O)[C@H]1Cc2ccccc2CN1Cc1csc(COc2ccc(C)cc2)n1 ZINC000217594389 HI On-Demand Unstable OPRM1 0 41 COC(=O)[C@H]1Cc2ccccc2CN1Cc1csc(COc2ccc(C)cc2)n1 ZINC000217594389 HI On-Demand Unstable OPRD1 45 32 COC(=O)[C@H]1Cc2ccccc2CN1Cc1csc(COc2ccc(C)cc2)n1 ZINC000217594389 HI On-Demand Unstable ADAM9 61 35 O=C(NCC1CCCCC1)Nc1ncccn1 ZINC000217594413 BE On-Demand Unstable GRIN2B 28 40 O=C1O[C@]2(CCCN(C(=O)C3CC3)C2)c2ccccc21 ZINC000217594414 CE In-Stock Unstable NPY5R 54 44 NC[C@H]1CCCCN1C(=O)/C=C\c1ccccc1 ZINC000217594463 BE On-Demand Unstable CPT1A 64 35 NC[C@H]1CCCCN1C(=O)/C=C\c1ccccc1 ZINC000217594463 BE On-Demand Unstable PREP 44 36 NC[C@H]1CCCCN1C(=O)/C=C\c1ccccc1 ZINC000217594463 BE On-Demand Unstable 17HSDCL 0 40 O=C1O[C@@]2(CCCN(C(=O)CC3CCCCC3)C2)c2ccccc21 ZINC000217594488 EH For-Sale Unstable NPY5R 40 40 CC(C)(C)C(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217594525 CF In-Stock Unstable NPY5R 33 43 CN(C(=O)NCC1CCCCC1)c1ccccc1 ZINC000217594529 BG For-Sale Unstable CHRM2 22 44 CN(C(=O)NCC1CCCCC1)c1ccccc1 ZINC000217594529 BG For-Sale Unstable CHRM1 25 44 CN(C(=O)NCC1CCCCC1)c1ccccc1 ZINC000217594529 BG For-Sale Unstable CHRM3 29 44 CN(C(=O)NCC1CCCCC1)c1ccccc1 ZINC000217594529 BG For-Sale Unstable NMBR 15 40 CN(C(=O)NCC1CCCCC1)c1ccccc1 ZINC000217594529 BG For-Sale Unstable AMY2 54 38 CN(C(=O)NCC1CCCCC1)c1ccccc1 ZINC000217594529 BG For-Sale Unstable METAP2 15 44 O=C(O)c1cc(S(=O)(=O)NCCCO)ccc1NC[C@@H]1CCCO1 ZINC000217594537 FC In-Stock Unstable BDKRB1 0 41 NC[C@@H]1CCCCN1C(=O)/C=C\c1ccc2c(c1)OCO2 ZINC000217594568 CD On-Demand Unstable DYRK2 48 33 O=C1O[C@]2(CCCN(C(=O)CC3CCCCC3)C2)c2ccccc21 ZINC000217594571 EH For-Sale Unstable NPY5R 40 40 CC(C)(C)C(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217594585 CF In-Stock Unstable NPY5R 33 43 CC[C@@H](C)[C@@H](C(=O)N1CCC[C@@H](CCl)C1)c1ccccc1 ZINC000217594605 DI For-Sale Unstable ACE 31 42 O=C(O)c1cc(S(=O)(=O)NCCCO)ccc1NC[C@H]1CCCO1 ZINC000217594609 FC In-Stock Unstable BDKRB1 0 41 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC1CCC(C(N)=O)CC1 ZINC000217594647 CG On-Demand Unstable TRPM8 0 45 NC[C@H]1CCCCN1C(=O)/C=C\c1ccc2c(c1)OCO2 ZINC000217594649 CD On-Demand Unstable DYRK2 48 33 O=C(O)/C=C\c1cccc(CNC(=O)c2cccs2)c1 ZINC000217594681 CF For-Sale Unstable HCAR2 28 42 CC[C@H](C)[C@@H](C(=O)N1CCC[C@@H](CCl)C1)c1ccccc1 ZINC000217594683 DI For-Sale Unstable ACE 31 42 COc1ccccc1CN(C)C(=O)C(F)F ZINC000217594684 BD On-Demand Unstable ACHE 0 51 COc1ccccc1CN(C)C(=O)C(F)F ZINC000217594684 BD On-Demand Unstable TACR1 29 45 COc1ccccc1CN(C)C(=O)C(F)F ZINC000217594684 BD On-Demand Unstable TSPO 45 39 COc1ccccc1CN(C)C(=O)C(F)F ZINC000217594684 BD On-Demand Unstable BCHE 0 50 Cc1nc(C)c(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)s1 ZINC000217594695 EG For-Sale Unstable NPY5R 30 42 CCCNC(=O)[C@@H]1CC[C@@H](CNC(=O)[C@@H]2Cc3ccccc3CN2)CC1 ZINC000217594704 FE In-Stock Unstable NPY2R 0 42 CCCNC(=O)[C@@H]1CC[C@@H](CNC(=O)[C@@H]2Cc3ccccc3CN2)CC1 ZINC000217594704 FE In-Stock Unstable MTNR1B 22 41 O=C(O)c1cc(S(=O)(=O)NCCCO)ccc1N1CCCC1 ZINC000217594721 EC In-Stock Unstable HTR7 21 41 O=C(O)c1cc(S(=O)(=O)NCCCO)ccc1N1CCCC1 ZINC000217594721 EC In-Stock Unstable CASP3 0 41 O=C(O)c1cc(S(=O)(=O)NCCCO)ccc1N1CCCC1 ZINC000217594721 EC In-Stock Unstable SFRP1 48 36 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC1CCC(C(N)=O)CC1 ZINC000217594729 CG On-Demand Unstable TRPM8 0 45 CC[C@@H](C)[C@H](C(=O)N1CCC[C@@H](CCl)C1)c1ccccc1 ZINC000217594757 DI For-Sale Unstable ACE 31 42 Cc1nc(C)c(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)s1 ZINC000217594768 EG For-Sale Unstable NPY5R 30 42 CCc1ccc(CN(C)C(=O)C(F)F)cc1 ZINC000217594793 BE On-Demand Unstable LIMK2 23 40 COc1ccc(/C=C\C(=O)N2CCCC[C@@H]2CN)cc1 ZINC000217594800 CE On-Demand Unstable MMP13 24 40 COc1ccc(/C=C\C(=O)N2CCCC[C@@H]2CN)cc1 ZINC000217594800 CE On-Demand Unstable MMP3 27 41 COc1ccc(/C=C\C(=O)N2CCCC[C@@H]2CN)cc1 ZINC000217594800 CE On-Demand Unstable MMP7 30 41 COc1ccc(/C=C\C(=O)N2CCCC[C@@H]2CN)cc1 ZINC000217594800 CE On-Demand Unstable GPR183 0 49 O=C(CN1CCCC[C@H]1CO)N1CCC[C@@H]1c1cccs1 ZINC000217594811 DE On-Demand Unstable COLA 78 39 O=C(CN1CCCC[C@H]1CO)N1CCC[C@@H]1c1cccs1 ZINC000217594811 DE On-Demand Unstable CPT1A 46 38 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC1CCC(C(N)=O)CC1 ZINC000217594814 CG For-Sale Unstable TRPM8 15 44 O=C(O)c1cc(S(=O)(=O)NCCCO)ccc1N1CCCCC1 ZINC000217594826 ED In-Stock Unstable HTR7 21 40 O=C(O)c1cc(S(=O)(=O)NCCCO)ccc1N1CCCCC1 ZINC000217594826 ED In-Stock Unstable CASP3 0 41 O=C(O)c1cc(S(=O)(=O)NCCCO)ccc1N1CCCCC1 ZINC000217594826 ED In-Stock Unstable SFRP1 45 36 COc1ccc(/C=C\C(=O)N2CCCC[C@H]2CN)cc1 ZINC000217594858 CE On-Demand Unstable MMP13 24 40 COc1ccc(/C=C\C(=O)N2CCCC[C@H]2CN)cc1 ZINC000217594858 CE On-Demand Unstable MMP3 27 41 COc1ccc(/C=C\C(=O)N2CCCC[C@H]2CN)cc1 ZINC000217594858 CE On-Demand Unstable GPR183 0 49 CC[C@H](C)[C@H](C(=O)N1CCC[C@@H](CCl)C1)c1ccccc1 ZINC000217594867 DI For-Sale Unstable ACE 31 42 O=C1O[C@@]2(CCCN(C(=O)c3ccc(F)cc3Cl)C2)c2ccccc21 ZINC000217594876 FH In-Stock Unstable P2RX7 19 45 O=C1O[C@@]2(CCCN(C(=O)c3ccc(F)cc3Cl)C2)c2ccccc21 ZINC000217594876 FH In-Stock Unstable NPY5R 32 44 CCOc1ccc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1OCC ZINC000217594880 GH For-Sale Unstable NPY5R 28 43 CCCCCNC(=O)NCC1CCCCC1 ZINC000217594882 BG On-Demand Unstable EPHX2 35 62 CCCCCNC(=O)NCC1CCCCC1 ZINC000217594882 BG On-Demand Unstable GNAI1 0 43 CCCCCNC(=O)NCC1CCCCC1 ZINC000217594882 BG On-Demand Unstable GNAI3 0 43 CCCCCNC(=O)NCC1CCCCC1 ZINC000217594882 BG On-Demand Unstable GNAO1 0 43 CCCCCNC(=O)NCC1CCCCC1 ZINC000217594882 BG On-Demand Unstable ASAH1 50 35 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC1CCC(C(N)=O)CC1 ZINC000217594894 CG For-Sale Unstable TRPM8 15 44 O=C(C(F)F)N1CCN(c2ccccc2[N+](=O)[O-])CC1 ZINC000217594919 CD On-Demand Unstable MC4R 22 47 O=C(C(F)F)N1CCN(c2ccccc2[N+](=O)[O-])CC1 ZINC000217594919 CD On-Demand Unstable MGLL 0 54 NC/C=C\COc1ccc(Cc2ccccc2)cc1 ZINC000217594926 CG For-Sale Unstable LTA4H 62 59 NC/C=C\COc1ccc(Cc2ccccc2)cc1 ZINC000217594926 CG For-Sale Unstable TAAR1 26 45 O=C(O)c1cc(S(=O)(=O)NCCCO)ccc1N1CCOCC1 ZINC000217594940 EB In-Stock Unstable HTR7 18 41 O=C(O)c1cc(S(=O)(=O)NCCCO)ccc1N1CCOCC1 ZINC000217594940 EB In-Stock Unstable SLC6A9 16 45 O=C1O[C@]2(CCCN(C(=O)c3ccc(F)cc3Cl)C2)c2ccccc21 ZINC000217594948 FH In-Stock Unstable P2RX7 19 45 O=C1O[C@]2(CCCN(C(=O)c3ccc(F)cc3Cl)C2)c2ccccc21 ZINC000217594948 FH In-Stock Unstable NPY5R 32 44 O=C(C[C@@H](c1ccc(O)cc1)c1c(O)c(O)c(O)c2c(=O)cc(-c3ccccc3)oc12)N1CCOCC1 ZINC000217594953 KH In-Stock Unstable RORC 41 32 CCOc1ccc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1OCC ZINC000217594955 GH For-Sale Unstable NPY5R 28 43 CCc1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217594999 CH On-Demand Unstable CCR3 46 41 CCc1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217594999 CH On-Demand Unstable EPHX2 34 42 CCc1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217594999 CH On-Demand Unstable PRMT3 41 40 O=C(C[C@H](c1ccc(O)cc1)c1c(O)c(O)c(O)c2c(=O)cc(-c3ccccc3)oc12)N1CCOCC1 ZINC000217595013 KH In-Stock Unstable RORC 41 32 CCOCCCNc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O ZINC000217595038 FC In-Stock Unstable CASP3 15 43 CCOCCCNc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O ZINC000217595038 FC In-Stock Unstable BDKRB1 0 41 CN(Cc1ccc(C(C)(C)C)cc1)C(=O)C(F)F ZINC000217595050 CG On-Demand Unstable MT-ND1 24 40 CN(Cc1ccc(C(C)(C)C)cc1)C(=O)C(F)F ZINC000217595050 CG On-Demand Unstable MLYCD 15 40 Cc1cnc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cn1 ZINC000217595071 DE In-Stock Unstable NPY5R 45 43 O=C1O[C@@]2(CCCN(C(=O)/C=C/c3ccc4c(c3)OCO4)C2)c2ccccc21 ZINC000217595072 GG In-Stock Unstable NPY5R 23 43 NC/C=C\CN1CCN(c2ccccc2)CC1 ZINC000217595138 BD For-Sale Unstable HTR1A 27 43 NC/C=C\CN1CCN(c2ccccc2)CC1 ZINC000217595138 BD For-Sale Unstable DRD1 0 48 NC/C=C\CN1CCN(c2ccccc2)CC1 ZINC000217595138 BD For-Sale Unstable DRD4 25 44 NC/C=C\CN1CCN(c2ccccc2)CC1 ZINC000217595138 BD For-Sale Unstable DRD3 22 48 NC/C=C\CN1CCN(c2ccccc2)CC1 ZINC000217595138 BD For-Sale Unstable HTR7 31 42 Cc1cnc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cn1 ZINC000217595143 DE In-Stock Unstable NPY5R 45 43 O=C1O[C@]2(CCCN(C(=O)/C=C/c3ccc4c(c3)OCO4)C2)c2ccccc21 ZINC000217595154 GG In-Stock Unstable NPY5R 23 43 CC(C)OCCCNc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O ZINC000217595163 FD In-Stock Unstable CASP3 16 41 CC(C)OCCCNc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O ZINC000217595163 FD In-Stock Unstable BDKRB1 0 41 CN(Cc1cccc(F)c1)C(=O)C(F)F ZINC000217595173 BE On-Demand Unstable HSP90AB1 15 42 CN(Cc1cccc(F)c1)C(=O)C(F)F ZINC000217595173 BE On-Demand Unstable HSD17B2 28 49 CN(Cc1cccc(F)c1)C(=O)C(F)F ZINC000217595173 BE On-Demand Unstable LIMK2 21 42 COc1cc(CCC(=O)N[C@H](CO)Cc2ccccc2)on1 ZINC000217595213 DD In-Stock Unstable CMA1 16 43 COc1cc(CCC(=O)N[C@H](CO)Cc2ccccc2)on1 ZINC000217595213 DD In-Stock Unstable PARP3 23 48 COc1cc(CCC(=O)N[C@H](CO)Cc2ccccc2)on1 ZINC000217595213 DD In-Stock Unstable PSMB8 26 42 Cc1ccc(O)c(NC(=O)NCC2CCCCC2)c1 ZINC000217595231 CG For-Sale Unstable THRA 24 45 Cc1ccc(O)c(NC(=O)NCC2CCCCC2)c1 ZINC000217595231 CG For-Sale Unstable THRB 27 45 Cc1ccc(O)c(NC(=O)NCC2CCCCC2)c1 ZINC000217595231 CG For-Sale Unstable KCNMA1 16 41 COc1ccc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c(OC)c1OC ZINC000217595243 GG For-Sale Unstable NPY5R 23 46 O=C1O[C@@]2(CCCN(C(=O)c3cc(-c4cccs4)[nH]n3)C2)c2ccccc21 ZINC000217595251 GG In-Stock Unstable NPY5R 30 41 CCCCCNc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O ZINC000217595288 ED In-Stock Unstable CASP3 17 48 NC[C@@H]1CCCCN1C(=O)/C=C\c1ccc(Cl)cc1 ZINC000217595295 CF On-Demand Unstable OPRK1 15 50 O=C1O[C@]2(CCCN(C(=O)c3cc(-c4cccs4)[nH]n3)C2)c2ccccc21 ZINC000217595317 GG In-Stock Unstable NPY5R 30 41 COc1ccc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c(OC)c1OC ZINC000217595318 GG For-Sale Unstable NPY5R 23 46 COC(=O)C[C@@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(OC(C)C)c(OC)c1 ZINC000217595326 HI In-Stock Unstable TNF 22 43 NC[C@H]1CCCCN1C(=O)/C=C\c1ccc(Cl)cc1 ZINC000217595371 CF On-Demand Unstable OPRK1 15 50 CC(C)CCNc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O ZINC000217595378 ED In-Stock Unstable CASP3 22 45 CN(C/C=C\CN)Cc1ccccc1 ZINC000217595382 AD For-Sale Unstable G6PC 51 31 COC(=O)C[C@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(OC(C)C)c(OC)c1 ZINC000217595414 HI In-Stock Unstable TNF 22 43 Cc1ccc(NC(=O)NCC2CCCCC2)cc1C ZINC000217595438 CI On-Demand Unstable LDLR 0 45 Cc1ccc(NC(=O)NCC2CCCCC2)cc1C ZINC000217595438 CI On-Demand Unstable EPHX2 30 40 Cc1ccc(NC(=O)NCC2CCCCC2)cc1C ZINC000217595438 CI On-Demand Unstable QRFPR 42 35 Cc1ccc(NC(=O)NCC2CCCCC2)cc1C ZINC000217595438 CI On-Demand Unstable PRMT3 53 47 Cc1ccc(NC(=O)NCC2CCCCC2)cc1C ZINC000217595438 CI On-Demand Unstable HSPB1 0 41 O=C1O[C@@]2(CCCN(C(=O)CSc3nc4ccccc4o3)C2)c2ccccc21 ZINC000217595445 GH For-Sale Unstable NPY5R 28 41 O=C1O[C@]2(CCCN(C(=O)CSc3nc4ccccc4o3)C2)c2ccccc21 ZINC000217595487 GH For-Sale Unstable NPY5R 28 41 CCN(Cc1ccccc1)C(=O)NCC1CCCCC1 ZINC000217595516 CH On-Demand Unstable OPRM1 16 45 CCN(Cc1ccccc1)C(=O)NCC1CCCCC1 ZINC000217595516 CH On-Demand Unstable OPRD1 21 43 CCN(Cc1ccccc1)C(=O)NCC1CCCCC1 ZINC000217595516 CH On-Demand Unstable AMY2 49 36 CCN(Cc1ccccc1)C(=O)NCC1CCCCC1 ZINC000217595516 CH On-Demand Unstable PTGES 24 57 CCN(Cc1ccccc1)C(=O)NCC1CCCCC1 ZINC000217595516 CH On-Demand Unstable LIMK2 42 36 CN(C/C=C\CN)Cc1cccnc1 ZINC000217595518 AD For-Sale Unstable NR1D1 40 35 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O ZINC000217595521 ED In-Stock Unstable CASP3 17 48 O=C1O[C@@]2(CCCN(C(=O)c3ccc(Br)o3)C2)c2ccccc21 ZINC000217595593 GG For-Sale Unstable NPY5R 25 40 CCC[C@H](C)Nc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O ZINC000217595605 ED In-Stock Unstable CASP3 17 48 O=C1O[C@]2(CCCN(C(=O)c3ccc(Br)o3)C2)c2ccccc21 ZINC000217595676 GG For-Sale Unstable NPY5R 25 40 COC[C@@H](C)Nc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O ZINC000217595695 EC In-Stock Unstable CASP3 16 40 NC[C@@H]1CCCCN1C(=O)/C=C\c1cccc([N+](=O)[O-])c1 ZINC000217595699 CD On-Demand Unstable TRPM8 0 44 COc1ccc(-c2coc3ccc(OCC(=O)N[C@@H]4CCS(=O)(=O)C4)cc23)cc1OC ZINC000217595738 IF In-Stock Unstable ALDH2 42 30 O=C(Cc1ccc2c(c1)OCO2)N1CCCn2nc(CO)cc2C1 ZINC000217595753 ED In-Stock Unstable NOS2 63 34 NC[C@H]1CCCCN1C(=O)/C=C\c1cccc([N+](=O)[O-])c1 ZINC000217595776 CD On-Demand Unstable TRPM8 0 44 COC[C@H](C)Nc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O ZINC000217595780 EC In-Stock Unstable CASP3 16 40 O=C(c1ccncc1)N1CCC(N2CCC[C@H]2COCc2ccccc2)CC1 ZINC000217595781 GG In-Stock Unstable GRIN2B 30 42 O=C(c1ccncc1)N1CCC(N2CCC[C@H]2COCc2ccccc2)CC1 ZINC000217595781 GG In-Stock Unstable PREP 43 38 O=C(c1ccncc1)N1CCC(N2CCC[C@H]2COCc2ccccc2)CC1 ZINC000217595781 GG In-Stock Unstable L3MBTL1 0 40 O=C(c1ccncc1)N1CCC(N2CCC[C@H]2COCc2ccccc2)CC1 ZINC000217595781 GG In-Stock Unstable L3MBTL3 83 40 O=C(c1ccncc1)N1CCC(N2CCC[C@H]2COCc2ccccc2)CC1 ZINC000217595781 GG In-Stock Unstable MBTD1 0 40 O=C(c1ccncc1)N1CCC(N2CCC[C@H]2COCc2ccccc2)CC1 ZINC000217595781 GG In-Stock Unstable SLC6A7 0 41 O=C1O[C@@]2(CCCN(C(=O)c3cccc(Br)c3)C2)c2ccccc21 ZINC000217595793 GH For-Sale Unstable NPY5R 29 42 O=C(NCC1CCCCC1)N(Cc1ccccc1)Cc1ccccc1 ZINC000217595796 EJ For-Sale Unstable PREP 49 35 O=C(NCC1CCCCC1)N(Cc1ccccc1)Cc1ccccc1 ZINC000217595796 EJ For-Sale Unstable AMY2 45 31 O=C(NCC1CCCCC1)N(Cc1ccccc1)Cc1ccccc1 ZINC000217595796 EJ For-Sale Unstable PTGES 27 65 O=C(NCC1CCCCC1)N(Cc1ccccc1)Cc1ccccc1 ZINC000217595796 EJ For-Sale Unstable LIMK2 42 37 COc1ccc(-c2coc3ccc(OCC(=O)N[C@H]4CCS(=O)(=O)C4)cc23)cc1OC ZINC000217595814 IF In-Stock Unstable ALDH2 42 30 O=C(O)/C=C\c1ccc(CNC(=O)[C@@H]2CCC(=O)N2)cc1 ZINC000217595839 CC For-Sale Unstable PLG 60 34 O=C(O)/C=C\c1ccc(CNC(=O)[C@@H]2CCC(=O)N2)cc1 ZINC000217595839 CC For-Sale Unstable TRYP_PIG 48 34 O=C(O)/C=C\c1ccc(CNC(=O)[C@@H]2CCC(=O)N2)cc1 ZINC000217595839 CC For-Sale Unstable LNPEP 49 38 O=C(c1ccncc1)N1CCC(N2CCC[C@@H]2COCc2ccccc2)CC1 ZINC000217595852 GG In-Stock Unstable GRIN2B 30 42 O=C(c1ccncc1)N1CCC(N2CCC[C@@H]2COCc2ccccc2)CC1 ZINC000217595852 GG In-Stock Unstable PREP 43 38 O=C(c1ccncc1)N1CCC(N2CCC[C@@H]2COCc2ccccc2)CC1 ZINC000217595852 GG In-Stock Unstable L3MBTL1 0 40 O=C(c1ccncc1)N1CCC(N2CCC[C@@H]2COCc2ccccc2)CC1 ZINC000217595852 GG In-Stock Unstable L3MBTL3 83 40 O=C(c1ccncc1)N1CCC(N2CCC[C@@H]2COCc2ccccc2)CC1 ZINC000217595852 GG In-Stock Unstable MBTD1 0 40 O=C(c1ccncc1)N1CCC(N2CCC[C@@H]2COCc2ccccc2)CC1 ZINC000217595852 GG In-Stock Unstable SLC6A7 0 41 Cn1ncc(C[C@H](N)C(=O)O)c1Br ZINC000217595855 BC For-Sale Unstable GRIA3 47 33 Cn1ncc(C[C@H](N)C(=O)O)c1Br ZINC000217595855 BC For-Sale Unstable GRIA4 47 33 Cn1ncc(C[C@H](N)C(=O)O)c1Br ZINC000217595855 BC For-Sale Unstable GRIK5 40 36 Nc1cccc2c1CN(C(=O)C(F)(F)F)CC2 ZINC000217595856 BD For-Sale Unstable AKR1C3 33 41 O=C1O[C@]2(CCCN(C(=O)c3cccc(Br)c3)C2)c2ccccc21 ZINC000217595876 GH For-Sale Unstable NPY5R 29 42 CCCNc1ccc(S(=O)(=O)NCCOC)cc1C(=O)O ZINC000217595895 DD In-Stock Unstable CASP3 15 40 CCCNc1ccc(S(=O)(=O)NCCOC)cc1C(=O)O ZINC000217595895 DD In-Stock Unstable BDKRB1 0 43 O=C(NO)[C@@H]1Cc2ccccc2N1c1ccccc1 ZINC000217595898 CE In-Stock Unstable ACE 23 43 O=C(NO)[C@@H]1Cc2ccccc2N1c1ccccc1 ZINC000217595898 CE In-Stock Unstable ADAM17 0 43 O=C(NO)[C@@H]1Cc2ccccc2N1c1ccccc1 ZINC000217595898 CE In-Stock Unstable MMP3 0 40 O=C(NO)[C@@H]1Cc2ccccc2N1c1ccccc1 ZINC000217595898 CE In-Stock Unstable MMP8 23 45 O=C(NO)[C@@H]1Cc2ccccc2N1c1ccccc1 ZINC000217595898 CE In-Stock Unstable ADAM9 75 43 O=C(NO)[C@@H]1Cc2ccccc2N1c1ccccc1 ZINC000217595898 CE In-Stock Unstable HDAC7 0 40 O=C(NO)[C@@H]1Cc2ccccc2N1c1ccccc1 ZINC000217595898 CE In-Stock Unstable MMP1 23 43 Cc1cc(Cl)ccc1NC(=O)NCC1CCCCC1 ZINC000217595905 CI On-Demand Unstable CNR1 17 50 Cc1cc(Cl)ccc1NC(=O)NCC1CCCCC1 ZINC000217595905 CI On-Demand Unstable LDLR 0 41 Cc1cc(Cl)ccc1NC(=O)NCC1CCCCC1 ZINC000217595905 CI On-Demand Unstable EPHX2 23 65 Cc1cc(Cl)ccc1NC(=O)NCC1CCCCC1 ZINC000217595905 CI On-Demand Unstable CACNA1I 63 37 Cc1cc(Cl)ccc1NC(=O)NCC1CCCCC1 ZINC000217595905 CI On-Demand Unstable METAP2 0 43 Cc1cc(Cl)ccc1NC(=O)NCC1CCCCC1 ZINC000217595905 CI On-Demand Unstable H9CNL0_SPOEX 0 43 O=C(O)/C=C\c1ccc(CNC(=O)[C@H]2CCC(=O)N2)cc1 ZINC000217595917 CC For-Sale Unstable PLG 60 34 O=C(O)/C=C\c1ccc(CNC(=O)[C@H]2CCC(=O)N2)cc1 ZINC000217595917 CC For-Sale Unstable TRYP_PIG 48 34 O=C(O)/C=C\c1ccc(CNC(=O)[C@H]2CCC(=O)N2)cc1 ZINC000217595917 CC For-Sale Unstable LNPEP 49 38 CN(Cc1ccon1)C(=O)c1ccc(CN2CCc3ccccc3C2)cc1 ZINC000217595924 FH In-Stock Unstable NOD1 36 46 CN(Cc1ccon1)C(=O)c1ccc(CN2CCc3ccccc3C2)cc1 ZINC000217595924 FH In-Stock Unstable NOD2 54 45 Cn1ncc(C[C@@H](N)C(=O)O)c1Br ZINC000217595932 BC For-Sale Unstable GRIA3 47 33 Cn1ncc(C[C@@H](N)C(=O)O)c1Br ZINC000217595932 BC For-Sale Unstable GRIA4 47 33 Cn1ncc(C[C@@H](N)C(=O)O)c1Br ZINC000217595932 BC For-Sale Unstable GRIK5 40 36 O=C(c1ccsc1)N1CCC(N2CCC[C@H]2COCc2ccccc2)CC1 ZINC000217595952 GI In-Stock Unstable L3MBTL3 80 39 O=C(NO)[C@H]1Cc2ccccc2N1c1ccccc1 ZINC000217595973 CE In-Stock Unstable ACE 23 43 O=C(NO)[C@H]1Cc2ccccc2N1c1ccccc1 ZINC000217595973 CE In-Stock Unstable ADAM17 0 43 O=C(NO)[C@H]1Cc2ccccc2N1c1ccccc1 ZINC000217595973 CE In-Stock Unstable MMP3 0 40 O=C(NO)[C@H]1Cc2ccccc2N1c1ccccc1 ZINC000217595973 CE In-Stock Unstable MMP8 23 45 O=C(NO)[C@H]1Cc2ccccc2N1c1ccccc1 ZINC000217595973 CE In-Stock Unstable ADAM9 75 43 O=C(NO)[C@H]1Cc2ccccc2N1c1ccccc1 ZINC000217595973 CE In-Stock Unstable HDAC7 0 40 O=C(NO)[C@H]1Cc2ccccc2N1c1ccccc1 ZINC000217595973 CE In-Stock Unstable MMP1 23 43 COCCNS(=O)(=O)c1ccc(NC(C)C)c(C(=O)O)c1 ZINC000217595983 DD In-Stock Unstable BDKRB1 0 41 O=C1O[C@@]2(CCCN(C(=O)c3ccc(Br)cc3)C2)c2ccccc21 ZINC000217595998 GH For-Sale Unstable NPY5R 27 42 O=C(c1ccsc1)N1CCC(N2CCC[C@@H]2COCc2ccccc2)CC1 ZINC000217596024 GI In-Stock Unstable L3MBTL3 80 39 CCn1ncc([C@H](N)C(=O)O)c1Br ZINC000217596025 BC For-Sale Unstable CACNA2D1 21 40 O=C1O[C@]2(CCCN(C(=O)c3ccc(Br)cc3)C2)c2ccccc21 ZINC000217596060 GH For-Sale Unstable NPY5R 27 42 CCCCNc1ccc(S(=O)(=O)NCCOC)cc1C(=O)O ZINC000217596068 ED In-Stock Unstable CASP3 16 41 CCn1ncc([C@@H](N)C(=O)O)c1Br ZINC000217596126 BC For-Sale Unstable CACNA2D1 21 40 Cc1cccc(CC(=O)N2CCC(N3CCC[C@@H]3COCc3ccccc3)CC2)c1 ZINC000217596131 HI In-Stock Unstable CCKAR 0 40 Cc1cccc(CC(=O)N2CCC(N3CCC[C@@H]3COCc3ccccc3)CC2)c1 ZINC000217596131 HI In-Stock Unstable GPR183 0 41 Cc1ccc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c(C)c1 ZINC000217596166 EH For-Sale Unstable NPY5R 28 45 COC(=O)c1ccc(C(=O)OC)c(NC(=O)NCC2CCCCC2)c1 ZINC000217596174 EF For-Sale Unstable METAP2 0 42 COCCNS(=O)(=O)c1ccc(NCC(C)C)c(C(=O)O)c1 ZINC000217596181 ED In-Stock Unstable CASP3 19 40 COCCNS(=O)(=O)c1ccc(NCC(C)C)c(C(=O)O)c1 ZINC000217596181 ED In-Stock Unstable BDKRB1 23 49 COc1ccc([C@@H](O)C(=O)NCCc2scnc2C)cc1 ZINC000217596197 DD In-Stock Unstable MAP1 15 41 Cc1ncsc1C(=O)NCc1ccc(/C=C\C(=O)O)cc1 ZINC000217596199 DE For-Sale Unstable VHL 40 33 Cc1cccc(CC(=O)N2CCC(N3CCC[C@H]3COCc3ccccc3)CC2)c1 ZINC000217596222 HI In-Stock Unstable CCKAR 0 40 Cc1cccc(CC(=O)N2CCC(N3CCC[C@H]3COCc3ccccc3)CC2)c1 ZINC000217596222 HI In-Stock Unstable GPR183 0 41 Cc1ccc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c(C)c1 ZINC000217596238 EH For-Sale Unstable NPY5R 28 45 COc1ccc([C@H](O)C(=O)NCCc2scnc2C)cc1 ZINC000217596267 DD In-Stock Unstable MAP1 15 41 Cc1ccc(C(=O)NCc2ccc(/C=C\C(=O)O)cc2)s1 ZINC000217596271 DG For-Sale Unstable HDAC1 16 43 CC[C@@H](C)Nc1ccc(S(=O)(=O)NCCOC)cc1C(=O)O ZINC000217596286 ED In-Stock Unstable BDKRB1 16 40 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](C2=Cc3ccccc3OC2)CC(=O)O4)cc1O ZINC000217596318 JJ In-Stock Unstable AKR1B1 0 44 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](C2=Cc3ccccc3OC2)CC(=O)O4)cc1O ZINC000217596318 JJ In-Stock Unstable CYP1B1 48 35 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](C2=Cc3ccccc3OC2)CC(=O)O4)cc1O ZINC000217596318 JJ In-Stock Unstable CYP1A1 37 44 O=C(Cc1ccc(F)cc1)N1CCC(N2CCC[C@H]2COCc2ccccc2)CC1 ZINC000217596321 HI In-Stock Unstable SIGMAR1 16 45 O=C(Cc1ccc(F)cc1)N1CCC(N2CCC[C@H]2COCc2ccccc2)CC1 ZINC000217596321 HI In-Stock Unstable CCR3 22 43 Cc1ccc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1C ZINC000217596331 EH For-Sale Unstable NPY5R 28 42 CC[C@H](C)Nc1ccc(S(=O)(=O)NCCOC)cc1C(=O)O ZINC000217596372 ED In-Stock Unstable BDKRB1 16 40 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](C2=Cc3ccccc3OC2)CC(=O)O4)cc1O ZINC000217596395 JJ In-Stock Unstable AKR1B1 0 44 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](C2=Cc3ccccc3OC2)CC(=O)O4)cc1O ZINC000217596395 JJ In-Stock Unstable CYP1B1 48 35 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](C2=Cc3ccccc3OC2)CC(=O)O4)cc1O ZINC000217596395 JJ In-Stock Unstable CYP1A1 37 44 O=C(NO)c1cc(C(F)(F)F)nc2ccccc12 ZINC000217596398 CE In-Stock Mild TACR3 30 47 O=C(Cc1ccc(F)cc1)N1CCC(N2CCC[C@@H]2COCc2ccccc2)CC1 ZINC000217596405 HI In-Stock Unstable SIGMAR1 16 45 O=C(Cc1ccc(F)cc1)N1CCC(N2CCC[C@@H]2COCc2ccccc2)CC1 ZINC000217596405 HI In-Stock Unstable CCR3 22 43 Cc1ccc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1C ZINC000217596406 EH For-Sale Unstable NPY5R 28 42 COCCNS(=O)(=O)c1ccc(NC(C)(C)C)c(C(=O)O)c1 ZINC000217596484 ED In-Stock Unstable PRTN3 47 33 O=C1O[C@@]2(CCCN(C(=O)c3ccc(I)cc3)C2)c2ccccc21 ZINC000217596515 IH For-Sale Unstable NPY5R 27 42 COC(=O)C[C@H](c1ccc(C(=O)O)cc1)c1c(O)ccc2c(=O)c(-c3ccc(O)cc3)coc12 ZINC000217596516 JI In-Stock Unstable ALDH2 99 40 Cc1occc1C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217596530 CF For-Sale Unstable PTGER2 23 42 C=CCNc1ccc(S(=O)(=O)NCCOC)cc1C(=O)O ZINC000217596580 DC In-Stock Unstable BDKRB1 0 44 COC(=O)C[C@@H](c1ccc(C(=O)O)cc1)c1c(O)ccc2c(=O)c(-c3ccc(O)cc3)coc12 ZINC000217596594 JI In-Stock Unstable ALDH2 99 40 O=C1O[C@]2(CCCN(C(=O)c3ccc(I)cc3)C2)c2ccccc21 ZINC000217596596 IH For-Sale Unstable NPY5R 27 42 Cc1ccoc1C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217596609 CF For-Sale Unstable PTGER2 0 41 OC[C@@H]1CCNC[C@H](O)[C@@H]1O ZINC000217596655 AA For-Sale Unstable PYGL 0 65 OC[C@@H]1CCNC[C@H](O)[C@@H]1O ZINC000217596655 AA For-Sale Unstable LCT 0 65 OC[C@@H]1CCNC[C@H](O)[C@@H]1O ZINC000217596655 AA For-Sale Unstable MAL62 0 40 OC[C@@H]1CCNC[C@H](O)[C@@H]1O ZINC000217596655 AA For-Sale Unstable LACA 0 44 OC[C@@H]1CCNC[C@H](O)[C@@H]1O ZINC000217596655 AA For-Sale Unstable CBG-1 0 65 OC[C@@H]1CCNC[C@H](O)[C@@H]1O ZINC000217596655 AA For-Sale Unstable AGL 0 40 OC[C@@H]1CCNC[C@H](O)[C@@H]1O ZINC000217596655 AA For-Sale Unstable Q9GPQ4_TRYVI 0 40 OC[C@@H]1CCNC[C@H](O)[C@@H]1O ZINC000217596655 AA For-Sale Unstable SGA1 0 40 CC[C@H](N)[C@H](O)COCc1ccccc1 ZINC000217596656 BD For-Sale Unstable CAPN2 41 33 CC[C@H](N)[C@H](O)COCc1ccccc1 ZINC000217596656 BD For-Sale Unstable POL 0 50 CCOCC(=O)N[C@@H](C)c1ccc(/C=C\C(=O)O)cc1 ZINC000217596686 CD For-Sale Unstable ACACA 45 40 CCOCC(=O)N[C@@H](C)c1ccc(/C=C\C(=O)O)cc1 ZINC000217596686 CD For-Sale Unstable ACACB 20 40 O=C1O[C@@]2(CCCN(C(=O)CSc3nc4ccccc4s3)C2)c2ccccc21 ZINC000217596699 HI For-Sale Unstable NPY5R 30 40 CCOc1ccccc1C(=O)N1CCC(N2CCC[C@@H]2COCc2ccccc2)CC1 ZINC000217596701 HI In-Stock Unstable CHRM2 17 49 CCOc1ccccc1C(=O)N1CCC(N2CCC[C@@H]2COCc2ccccc2)CC1 ZINC000217596701 HI In-Stock Unstable HCN1 60 39 CCOc1ccccc1C(=O)N1CCC(N2CCC[C@@H]2COCc2ccccc2)CC1 ZINC000217596701 HI In-Stock Unstable HCN4 49 39 CCOc1ccccc1C(=O)N1CCC(N2CCC[C@@H]2COCc2ccccc2)CC1 ZINC000217596701 HI In-Stock Unstable L3MBTL1 0 41 CCOc1ccccc1C(=O)N1CCC(N2CCC[C@@H]2COCc2ccccc2)CC1 ZINC000217596701 HI In-Stock Unstable L3MBTL3 64 41 CCOc1ccccc1C(=O)N1CCC(N2CCC[C@@H]2COCc2ccccc2)CC1 ZINC000217596701 HI In-Stock Unstable MBTD1 0 41 CCOc1ccccc1C(=O)N1CCC(N2CCC[C@@H]2COCc2ccccc2)CC1 ZINC000217596701 HI In-Stock Unstable TP53BP1 0 41 OC[C@@H]1CCNC[C@@H](O)[C@@H]1O ZINC000217596722 AA For-Sale Unstable PYGL 0 65 OC[C@@H]1CCNC[C@@H](O)[C@@H]1O ZINC000217596722 AA For-Sale Unstable LCT 0 65 OC[C@@H]1CCNC[C@@H](O)[C@@H]1O ZINC000217596722 AA For-Sale Unstable MAL62 0 40 OC[C@@H]1CCNC[C@@H](O)[C@@H]1O ZINC000217596722 AA For-Sale Unstable LACA 0 44 OC[C@@H]1CCNC[C@@H](O)[C@@H]1O ZINC000217596722 AA For-Sale Unstable CBG-1 0 65 OC[C@@H]1CCNC[C@@H](O)[C@@H]1O ZINC000217596722 AA For-Sale Unstable AGL 0 40 OC[C@@H]1CCNC[C@@H](O)[C@@H]1O ZINC000217596722 AA For-Sale Unstable Q9GPQ4_TRYVI 0 40 OC[C@@H]1CCNC[C@@H](O)[C@@H]1O ZINC000217596722 AA For-Sale Unstable SGA1 0 40 CC[C@@H](N)[C@H](O)COCc1ccccc1 ZINC000217596739 BD For-Sale Unstable CAPN2 41 33 CC[C@@H](N)[C@H](O)COCc1ccccc1 ZINC000217596739 BD For-Sale Unstable POL 0 50 CN(Cc1cccs1)C(=O)C(F)F ZINC000217596745 BD On-Demand Unstable ADAM17 0 48 C[C@@H](CNC(c1ccccc1)c1ccccc1)NC(=O)OC(C)(C)C ZINC000217596768 EI On-Demand Unstable PAPA1_CARPA 51 43 C[C@@H](CNC(c1ccccc1)c1ccccc1)NC(=O)OC(C)(C)C ZINC000217596768 EI On-Demand Unstable CTSK 30 40 C[C@@H](CNC(c1ccccc1)c1ccccc1)NC(=O)OC(C)(C)C ZINC000217596768 EI On-Demand Unstable CTSL 15 43 C[C@@H](CNC(c1ccccc1)c1ccccc1)NC(=O)OC(C)(C)C ZINC000217596768 EI On-Demand Unstable FPR1 52 42 CCOCC(=O)N[C@H](C)c1ccc(/C=C\C(=O)O)cc1 ZINC000217596769 CD For-Sale Unstable ACACA 45 40 CCOCC(=O)N[C@H](C)c1ccc(/C=C\C(=O)O)cc1 ZINC000217596769 CD For-Sale Unstable ACACB 20 40 COCCNS(=O)(=O)c1ccc(NC2CCCC2)c(C(=O)O)c1 ZINC000217596780 ED In-Stock Unstable CASP3 23 42 O=C1O[C@]2(CCCN(C(=O)CSc3nc4ccccc4s3)C2)c2ccccc21 ZINC000217596782 HI For-Sale Unstable NPY5R 30 40 CCOc1ccccc1C(=O)N1CCC(N2CCC[C@H]2COCc2ccccc2)CC1 ZINC000217596794 HI In-Stock Unstable CHRM2 17 49 CCOc1ccccc1C(=O)N1CCC(N2CCC[C@H]2COCc2ccccc2)CC1 ZINC000217596794 HI In-Stock Unstable HCN1 60 39 CCOc1ccccc1C(=O)N1CCC(N2CCC[C@H]2COCc2ccccc2)CC1 ZINC000217596794 HI In-Stock Unstable HCN4 49 39 CCOc1ccccc1C(=O)N1CCC(N2CCC[C@H]2COCc2ccccc2)CC1 ZINC000217596794 HI In-Stock Unstable L3MBTL1 0 41 CCOc1ccccc1C(=O)N1CCC(N2CCC[C@H]2COCc2ccccc2)CC1 ZINC000217596794 HI In-Stock Unstable L3MBTL3 64 41 CCOc1ccccc1C(=O)N1CCC(N2CCC[C@H]2COCc2ccccc2)CC1 ZINC000217596794 HI In-Stock Unstable MBTD1 0 41 CCOc1ccccc1C(=O)N1CCC(N2CCC[C@H]2COCc2ccccc2)CC1 ZINC000217596794 HI In-Stock Unstable TP53BP1 0 41 OC[C@@H]1CCNC[C@H](O)[C@H]1O ZINC000217596797 AA For-Sale Unstable PYGL 17 65 CC[C@H](N)[C@@H](O)COCc1ccccc1 ZINC000217596829 BD For-Sale Unstable CAPN2 41 33 CC[C@H](N)[C@@H](O)COCc1ccccc1 ZINC000217596829 BD For-Sale Unstable POL 0 50 OC[C@@H]1CCNC[C@@H](O)[C@H]1O ZINC000217596869 AA For-Sale Unstable PYGL 17 65 COCCNS(=O)(=O)c1ccc(NC2CCCCC2)c(C(=O)O)c1 ZINC000217596889 FE In-Stock Unstable CASP3 23 41 CC[C@@H](N)[C@@H](O)COCc1ccccc1 ZINC000217596903 BD For-Sale Unstable CAPN2 41 33 CC[C@@H](N)[C@@H](O)COCc1ccccc1 ZINC000217596903 BD For-Sale Unstable POL 0 50 COC(=O)[C@H](Cc1ccccc1)NC(=O)COc1cc2c(c3oc(=O)cc(C)c13)CCC(C)(C)O2 ZINC000217596916 JG In-Stock Unstable CTRA_BOVIN 42 33 COC(=O)[C@H](Cc1ccccc1)NC(=O)COc1cc2c(c3oc(=O)cc(C)c13)CCC(C)(C)O2 ZINC000217596916 JG In-Stock Unstable PLM2_PLAFA 44 32 NC/C=C\CN1CC[C@@H](c2ccccc2)C1 ZINC000217596946 BD For-Sale Unstable VACHT_TETCF 0 44 C[C@H]1CN(C)[C@@H](C)C[C@@H]1Nc1cccnc1Cl ZINC000217596951 CF For-Sale Unstable G2YM83_BOTF4 53 36 CCCCCC(=O)N[C@@H](C)c1ccc(/C=C\C(=O)O)cc1 ZINC000217597030 CH For-Sale Unstable ACACA 40 42 CCCCCC(=O)N[C@@H](C)c1ccc(/C=C\C(=O)O)cc1 ZINC000217597030 CH For-Sale Unstable NOD1 79 42 NC/C=C\CN1CC[C@H](c2ccccc2)C1 ZINC000217597045 BD For-Sale Unstable VACHT_TETCF 0 44 O=C1O[C@@]2(CCCN(C(=O)c3ccc4nccnc4c3)C2)c2ccccc21 ZINC000217597062 FF For-Sale Unstable NPY5R 42 42 O=C1O[C@@]2(CCCN(C(=O)c3ccc4nccnc4c3)C2)c2ccccc21 ZINC000217597062 FF For-Sale Unstable HPGD 42 38 Cc1cc(C(F)(F)F)nn1-c1ccc(C(=O)NO)cc1 ZINC000217597078 CE In-Stock Unstable HDAC8 32 40 Cc1cc(C(F)(F)F)nn1-c1ccc(C(=O)NO)cc1 ZINC000217597078 CE In-Stock Unstable HDAC6 0 40 Cc1cc(C(F)(F)F)nn1-c1ccc(C(=O)NO)cc1 ZINC000217597078 CE In-Stock Unstable CARM1 69 33 CC(C)C[C@@H](N[C@@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597085 CG For-Sale Unstable ACE 52 49 CC(C)C[C@@H](N[C@@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597085 CG For-Sale Unstable PTGS1 19 40 CC(C)C[C@@H](N[C@@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597085 CG For-Sale Unstable FOLH1 54 36 CC(C)C[C@@H](N[C@@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597085 CG For-Sale Unstable MME 94 49 CC(C)C[C@@H](N[C@@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597085 CG For-Sale Unstable ANPEP 53 43 CC(C)C[C@@H](N[C@@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597085 CG For-Sale Unstable RNPEP 37 43 CC(C)C[C@@H](N[C@@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597085 CG For-Sale Unstable CTSB 50 52 CC(C)C[C@@H](N[C@@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597085 CG For-Sale Unstable CYSP_TRYCR 47 48 CC(C)C[C@@H](N[C@@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597085 CG For-Sale Unstable CTSF 76 48 CC(C)C[C@@H](N[C@@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597085 CG For-Sale Unstable CTSK 77 70 CC(C)C[C@@H](N[C@@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597085 CG For-Sale Unstable CTSL 50 70 CC(C)C[C@@H](N[C@@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597085 CG For-Sale Unstable CPA1 41 40 CC(C)C[C@@H](N[C@@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597085 CG For-Sale Unstable CAPNS1 58 36 CC(C)C[C@@H](N[C@@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597085 CG For-Sale Unstable MMP2 17 41 CC(C)C[C@@H](N[C@@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597085 CG For-Sale Unstable MMP3 37 41 CC(C)C[C@@H](N[C@@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597085 CG For-Sale Unstable CTSS 39 63 CC(C)C[C@@H](N[C@@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597085 CG For-Sale Unstable CAPN1 67 43 CC(C)C[C@@H](N[C@@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597085 CG For-Sale Unstable MMP9 19 40 CC(C)C[C@@H](N[C@@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597085 CG For-Sale Unstable CAPN2 84 39 CC(C)C[C@@H](N[C@@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597085 CG For-Sale Unstable ACE2 83 45 CC(C)C[C@@H](N[C@@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597085 CG For-Sale Unstable LAP3 21 44 CC(C)C[C@@H](N[C@@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597085 CG For-Sale Unstable MMP1 25 40 CC(C)C[C@@H](N[C@@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597085 CG For-Sale Unstable FPR1 81 43 CC(C)C[C@@H](N[C@@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597085 CG For-Sale Unstable NPR 84 38 CC(C)C[C@@H](N[C@@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597085 CG For-Sale Unstable AMP1_PLAFQ 31 43 Cc1n[nH]c([C@@H]2CCCN2C(=O)CN2CCOC2=O)n1 ZINC000217597107 CC In-Stock Unstable COLA 85 42 Cc1n[nH]c([C@@H]2CCCN2C(=O)CN2CCOC2=O)n1 ZINC000217597107 CC In-Stock Unstable CPT1A 72 42 COCCNS(=O)(=O)c1ccc(NCCO)c(C(=O)O)c1 ZINC000217597110 DB In-Stock Unstable BDKRB1 0 43 CCCCCC(=O)N[C@H](C)c1ccc(/C=C\C(=O)O)cc1 ZINC000217597127 CH For-Sale Unstable ACACA 40 42 CCCCCC(=O)N[C@H](C)c1ccc(/C=C\C(=O)O)cc1 ZINC000217597127 CH For-Sale Unstable NOD1 79 42 O=C1O[C@]2(CCCN(C(=O)c3ccc4nccnc4c3)C2)c2ccccc21 ZINC000217597142 FF For-Sale Unstable NPY5R 42 42 O=C1O[C@]2(CCCN(C(=O)c3ccc4nccnc4c3)C2)c2ccccc21 ZINC000217597142 FF For-Sale Unstable HPGD 42 38 CC(C)C[C@@H](N[C@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597165 CG For-Sale Unstable ACE 52 49 CC(C)C[C@@H](N[C@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597165 CG For-Sale Unstable PTGS1 19 40 CC(C)C[C@@H](N[C@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597165 CG For-Sale Unstable FOLH1 54 36 CC(C)C[C@@H](N[C@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597165 CG For-Sale Unstable MME 94 49 CC(C)C[C@@H](N[C@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597165 CG For-Sale Unstable ANPEP 53 43 CC(C)C[C@@H](N[C@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597165 CG For-Sale Unstable RNPEP 37 43 CC(C)C[C@@H](N[C@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597165 CG For-Sale Unstable CTSB 50 52 CC(C)C[C@@H](N[C@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597165 CG For-Sale Unstable CYSP_TRYCR 47 48 CC(C)C[C@@H](N[C@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597165 CG For-Sale Unstable CTSF 76 48 CC(C)C[C@@H](N[C@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597165 CG For-Sale Unstable CTSK 77 70 CC(C)C[C@@H](N[C@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597165 CG For-Sale Unstable CTSL 50 70 CC(C)C[C@@H](N[C@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597165 CG For-Sale Unstable CPA1 41 40 CC(C)C[C@@H](N[C@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597165 CG For-Sale Unstable CAPNS1 58 36 CC(C)C[C@@H](N[C@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597165 CG For-Sale Unstable MMP2 17 41 CC(C)C[C@@H](N[C@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597165 CG For-Sale Unstable MMP3 37 41 CC(C)C[C@@H](N[C@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597165 CG For-Sale Unstable CTSS 39 63 CC(C)C[C@@H](N[C@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597165 CG For-Sale Unstable CAPN1 67 43 CC(C)C[C@@H](N[C@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597165 CG For-Sale Unstable MMP9 19 40 CC(C)C[C@@H](N[C@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597165 CG For-Sale Unstable CAPN2 84 39 CC(C)C[C@@H](N[C@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597165 CG For-Sale Unstable ACE2 83 45 CC(C)C[C@@H](N[C@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597165 CG For-Sale Unstable LAP3 21 44 CC(C)C[C@@H](N[C@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597165 CG For-Sale Unstable MMP1 25 40 CC(C)C[C@@H](N[C@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597165 CG For-Sale Unstable FPR1 81 43 CC(C)C[C@@H](N[C@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597165 CG For-Sale Unstable NPR 84 38 CC(C)C[C@@H](N[C@H](c1ccccc1)C(F)(F)F)C(=O)O ZINC000217597165 CG For-Sale Unstable AMP1_PLAFQ 31 43 Nc1ccc(N(C(=O)NCC2CCCCC2)c2ccccc2)cc1 ZINC000217597184 DJ For-Sale Unstable AMY2 49 33 Cc1n[nH]c([C@H]2CCCN2C(=O)CN2CCOC2=O)n1 ZINC000217597192 CC In-Stock Unstable COLA 85 42 Cc1n[nH]c([C@H]2CCCN2C(=O)CN2CCOC2=O)n1 ZINC000217597192 CC In-Stock Unstable CPT1A 72 42 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)NCCSc1ccccc1)C(=O)OC2 ZINC000217597201 JJ In-Stock Unstable IMPDH1 0 63 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)NCCSc1ccccc1)C(=O)OC2 ZINC000217597201 JJ In-Stock Unstable IMPDH2 0 63 COCCNS(=O)(=O)c1ccc(NCCCO)c(C(=O)O)c1 ZINC000217597225 EC In-Stock Unstable BDKRB1 0 44 CCOc1cc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc(OCC)c1OCC ZINC000217597247 II For-Sale Unstable NPY5R 27 41 O=C(NCC1CCCCC1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217597278 DK For-Sale Unstable ADRB1 15 40 O=C(NCC1CCCCC1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217597278 DK For-Sale Unstable LPL 42 34 O=C(NCC1CCCCC1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217597278 DK For-Sale Unstable CCR3 43 43 O=C(NCC1CCCCC1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217597278 DK For-Sale Unstable EPHX2 47 65 O=C(NCC1CCCCC1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217597278 DK For-Sale Unstable PRMT3 42 40 O=C(NCC1CCCCC1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217597278 DK For-Sale Unstable DGAT1 17 41 O=C(NCC1CCCCC1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217597278 DK For-Sale Unstable ACAT 0 49 O=C(NCC1CCCCC1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217597278 DK For-Sale Unstable NAMPT 32 43 O=C(NCC1CCCCC1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217597278 DK For-Sale Unstable P95276_MYCTO 0 44 O=C(NCc1nc2ccc(Cl)cc2[nH]1)c1ccc(O)c(F)c1 ZINC000217597290 DF In-Stock Unstable F9 27 43 COC[C@@H](Cc1ccccc1)NC(=O)c1ccccn1 ZINC000217597297 CE On-Demand Unstable MME 61 42 COC[C@@H](Cc1ccccc1)NC(=O)c1ccccn1 ZINC000217597297 CE On-Demand Unstable ANPEP 56 33 COC[C@@H](Cc1ccccc1)NC(=O)c1ccccn1 ZINC000217597297 CE On-Demand Unstable PAPA1_CARPA 46 36 COC[C@@H](Cc1ccccc1)NC(=O)c1ccccn1 ZINC000217597297 CE On-Demand Unstable CCR1 41 35 COC[C@@H](Cc1ccccc1)NC(=O)c1ccccn1 ZINC000217597297 CE On-Demand Unstable CTRB1 32 40 COC[C@@H](Cc1ccccc1)NC(=O)c1ccccn1 ZINC000217597297 CE On-Demand Unstable GRM4 49 41 COC[C@@H](Cc1ccccc1)NC(=O)c1ccccn1 ZINC000217597297 CE On-Demand Unstable CAPN1 44 33 COC[C@@H](Cc1ccccc1)NC(=O)c1ccccn1 ZINC000217597297 CE On-Demand Unstable CAPN2 45 31 COC[C@@H](Cc1ccccc1)NC(=O)c1ccccn1 ZINC000217597297 CE On-Demand Unstable ACE2 43 34 COC[C@@H](Cc1ccccc1)NC(=O)c1ccccn1 ZINC000217597297 CE On-Demand Unstable PIN1 32 42 COC[C@@H](Cc1ccccc1)NC(=O)c1ccccn1 ZINC000217597297 CE On-Demand Unstable PLM1_PLAFA 54 37 COC[C@@H](Cc1ccccc1)NC(=O)c1ccccn1 ZINC000217597297 CE On-Demand Unstable PLM2_PLAFA 28 42 COC[C@@H](Cc1ccccc1)NC(=O)c1ccccn1 ZINC000217597297 CE On-Demand Unstable PSMB5 39 40 COC[C@@H](Cc1ccccc1)NC(=O)c1ccccn1 ZINC000217597297 CE On-Demand Unstable PSMB8 25 41 O=C(CSCc1ccccc1)N1CCC(N2CCC[C@H]2COCc2ccccc2)CC1 ZINC000217597314 IJ In-Stock Unstable PREP 47 36 CCOc1cc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc(OCC)c1OCC ZINC000217597325 II For-Sale Unstable NPY5R 27 41 COCCNc1ccc(S(=O)(=O)NCCOC)cc1C(=O)O ZINC000217597356 EC In-Stock Unstable BDKRB1 0 45 O=C(NCC1CCCCC1)N1CCc2ccccc2C1 ZINC000217597371 CG On-Demand Unstable DPP8 23 43 O=C(CSCc1ccccc1)N1CCC(N2CCC[C@@H]2COCc2ccccc2)CC1 ZINC000217597378 IJ In-Stock Unstable PREP 47 36 COC[C@H](Cc1ccccc1)NC(=O)c1ccccn1 ZINC000217597391 CE On-Demand Unstable MME 61 42 COC[C@H](Cc1ccccc1)NC(=O)c1ccccn1 ZINC000217597391 CE On-Demand Unstable ANPEP 56 33 COC[C@H](Cc1ccccc1)NC(=O)c1ccccn1 ZINC000217597391 CE On-Demand Unstable PAPA1_CARPA 46 36 COC[C@H](Cc1ccccc1)NC(=O)c1ccccn1 ZINC000217597391 CE On-Demand Unstable CCR1 41 35 COC[C@H](Cc1ccccc1)NC(=O)c1ccccn1 ZINC000217597391 CE On-Demand Unstable CTRB1 32 40 COC[C@H](Cc1ccccc1)NC(=O)c1ccccn1 ZINC000217597391 CE On-Demand Unstable GRM4 49 41 COC[C@H](Cc1ccccc1)NC(=O)c1ccccn1 ZINC000217597391 CE On-Demand Unstable CAPN1 44 33 COC[C@H](Cc1ccccc1)NC(=O)c1ccccn1 ZINC000217597391 CE On-Demand Unstable CAPN2 45 31 COC[C@H](Cc1ccccc1)NC(=O)c1ccccn1 ZINC000217597391 CE On-Demand Unstable ACE2 43 34 COC[C@H](Cc1ccccc1)NC(=O)c1ccccn1 ZINC000217597391 CE On-Demand Unstable PIN1 32 42 COC[C@H](Cc1ccccc1)NC(=O)c1ccccn1 ZINC000217597391 CE On-Demand Unstable PLM1_PLAFA 54 37 COC[C@H](Cc1ccccc1)NC(=O)c1ccccn1 ZINC000217597391 CE On-Demand Unstable PLM2_PLAFA 28 42 COC[C@H](Cc1ccccc1)NC(=O)c1ccccn1 ZINC000217597391 CE On-Demand Unstable PSMB5 39 40 COC[C@H](Cc1ccccc1)NC(=O)c1ccccn1 ZINC000217597391 CE On-Demand Unstable PSMB8 25 41 CC1(C)CCCN(C/C=C\CN)C1 ZINC000217597406 AD For-Sale Unstable EBP 25 55 O=C1O[C@@]2(CCCN(C(=O)c3c[nH]c4ccccc34)C2)c2ccccc21 ZINC000217597420 EG For-Sale Unstable AVPR1A 28 61 O=C1O[C@@]2(CCCN(C(=O)c3c[nH]c4ccccc34)C2)c2ccccc21 ZINC000217597420 EG For-Sale Unstable NPY5R 30 42 COCCCNc1ccc(S(=O)(=O)NCCOC)cc1C(=O)O ZINC000217597463 EC In-Stock Unstable BDKRB1 0 46 Cc1ccc2ncccc2c1CN1CCN(C(C)C)[C@@H](C)C1 ZINC000217597465 CG In-Stock Unstable PRKCQ 40 30 Cc1cccc(NC(=O)NCC2CCCCC2)n1 ZINC000217597480 BG On-Demand Unstable GRM5 18 49 Cc1cccc(NC(=O)NCC2CCCCC2)n1 ZINC000217597480 BG On-Demand Unstable SORT1 17 42 O=C1O[C@]2(CCCN(C(=O)c3c[nH]c4ccccc34)C2)c2ccccc21 ZINC000217597493 EG For-Sale Unstable AVPR1A 28 61 O=C1O[C@]2(CCCN(C(=O)c3c[nH]c4ccccc34)C2)c2ccccc21 ZINC000217597493 EG For-Sale Unstable NPY5R 30 42 O=C(COc1ccc(Cl)cc1)N1CCC(N2CCC[C@H]2COCc2ccccc2)CC1 ZINC000217597499 II In-Stock Unstable LTA4H 21 41 O=C(COc1ccc(Cl)cc1)N1CCC(N2CCC[C@H]2COCc2ccccc2)CC1 ZINC000217597499 II In-Stock Unstable COLA 83 39 O=C(COc1ccc(Cl)cc1)N1CCC(N2CCC[C@H]2COCc2ccccc2)CC1 ZINC000217597499 II In-Stock Unstable CPT1A 76 39 O=C(COc1ccc(Cl)cc1)N1CCC(N2CCC[C@H]2COCc2ccccc2)CC1 ZINC000217597499 II In-Stock Unstable CPT2 42 39 O=C(COc1ccc(Cl)cc1)N1CCC(N2CCC[C@H]2COCc2ccccc2)CC1 ZINC000217597499 II In-Stock Unstable GPR183 0 55 CCOC(=O)c1csc(NC(=O)[C@H](C)Nc2ccc3c(cc2=O)[C@@H](NC(C)=O)CCc2cc(OC)c(OC)c(OC)c2-3)n1 ZINC000217597507 KH In-Stock Unstable TUBA1A 16 59 CCOC(=O)c1csc(NC(=O)[C@H](C)Nc2ccc3c(cc2=O)[C@@H](NC(C)=O)CCc2cc(OC)c(OC)c(OC)c2-3)n1 ZINC000217597507 KH In-Stock Unstable TPPP 0 56 CC(C)(F)C[C@@H](N[C@H](c1ccc(Br)cc1)C(F)(F)F)C(=O)O ZINC000217597521 GI For-Sale Anodyne CTSB 17 50 CC(C)(F)C[C@@H](N[C@H](c1ccc(Br)cc1)C(F)(F)F)C(=O)O ZINC000217597521 GI For-Sale Anodyne CYSP_TRYCR 35 45 CC(C)(F)C[C@@H](N[C@H](c1ccc(Br)cc1)C(F)(F)F)C(=O)O ZINC000217597521 GI For-Sale Anodyne CTSF 73 45 CC(C)(F)C[C@@H](N[C@H](c1ccc(Br)cc1)C(F)(F)F)C(=O)O ZINC000217597521 GI For-Sale Anodyne CTSK 49 55 CC(C)(F)C[C@@H](N[C@H](c1ccc(Br)cc1)C(F)(F)F)C(=O)O ZINC000217597521 GI For-Sale Anodyne CTSL 27 47 CC(C)(F)C[C@@H](N[C@H](c1ccc(Br)cc1)C(F)(F)F)C(=O)O ZINC000217597521 GI For-Sale Anodyne CTSS 19 43 O=C(NCCCCCO)NCC1CCCCC1 ZINC000217597561 BE On-Demand Unstable EPHX2 45 45 COCCNS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217597563 FD In-Stock Unstable BDKRB1 0 46 COCCNS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217597563 FD In-Stock Unstable PRTN3 44 31 COCCNS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217597563 FD In-Stock Unstable AKR1C3 16 43 O=C(COc1ccc(Cl)cc1)N1CCC(N2CCC[C@@H]2COCc2ccccc2)CC1 ZINC000217597586 II In-Stock Unstable LTA4H 21 41 O=C(COc1ccc(Cl)cc1)N1CCC(N2CCC[C@@H]2COCc2ccccc2)CC1 ZINC000217597586 II In-Stock Unstable COLA 83 39 O=C(COc1ccc(Cl)cc1)N1CCC(N2CCC[C@@H]2COCc2ccccc2)CC1 ZINC000217597586 II In-Stock Unstable CPT1A 76 39 O=C(COc1ccc(Cl)cc1)N1CCC(N2CCC[C@@H]2COCc2ccccc2)CC1 ZINC000217597586 II In-Stock Unstable CPT2 42 39 O=C(COc1ccc(Cl)cc1)N1CCC(N2CCC[C@@H]2COCc2ccccc2)CC1 ZINC000217597586 II In-Stock Unstable GPR183 0 55 COc1cc2c(cc1OC)CC(=O)N(CC(=O)N[C@H](CO)c1ccccc1)C=C2 ZINC000217597615 GD In-Stock Unstable HCN2 0 43 CC(C)C(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217597622 CE For-Sale Unstable NPY5R 32 43 COCCNS(=O)(=O)c1ccc(N[C@@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217597664 GE In-Stock Unstable BDKRB1 0 46 CN[C@@H](C)C(=O)N[C@@H]1CCC[C@@H](C)[C@@H]1C ZINC000217597665 BD On-Demand Unstable BIRC2 47 31 CCO[C@@H]1C[C@@H](NC(=O)c2cccc(C#N)c2)C1(C)C ZINC000217597672 CE For-Sale Unstable ABCC9 40 42 CCO[C@@H]1C[C@@H](NC(=O)c2cccc(C#N)c2)C1(C)C ZINC000217597672 CE For-Sale Unstable EZH2 47 35 Cc1ccc(OCc2nc(CNCCOc3ccc(Cl)cc3)cs2)cc1 ZINC000217597694 GJ On-Demand Unstable DRD4 19 41 CC(C)C(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217597704 CE For-Sale Unstable NPY5R 32 43 COCCNS(=O)(=O)c1ccc(N[C@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217597742 GE In-Stock Unstable BDKRB1 0 46 CN[C@H](C)C(=O)N[C@@H]1CCC[C@@H](C)[C@@H]1C ZINC000217597743 BD On-Demand Unstable BIRC2 47 31 CCO[C@H]1C[C@@H](NC(=O)c2cccc(C#N)c2)C1(C)C ZINC000217597747 CE For-Sale Unstable ABCC9 40 42 CCO[C@H]1C[C@@H](NC(=O)c2cccc(C#N)c2)C1(C)C ZINC000217597747 CE For-Sale Unstable EZH2 47 35 O=C(NCC1(N2CCCCC2)CCCCC1)C(F)F ZINC000217597766 CF On-Demand Unstable HCN1 60 39 O=C(NCC1(N2CCCCC2)CCCCC1)C(F)F ZINC000217597766 CF On-Demand Unstable HCN4 57 39 C=CCNC(=O)NCC1CCCCC1 ZINC000217597773 AE On-Demand Unstable ADH4 0 41 O=C([C@H]1CC=CCC1)N1CCC(N2CCC[C@@H]2COCc2ccccc2)CC1 ZINC000217597792 GI In-Stock Unstable PREP 49 43 O=C1O[C@@]2(CCCN(C(=O)c3cccc4ccccc34)C2)c2ccccc21 ZINC000217597813 FI For-Sale Unstable NPY5R 29 41 CCO[C@@H]1C[C@H](NC(=O)c2cccc(C#N)c2)C1(C)C ZINC000217597822 CE For-Sale Unstable ABCC9 40 42 CCO[C@@H]1C[C@H](NC(=O)c2cccc(C#N)c2)C1(C)C ZINC000217597822 CE For-Sale Unstable EZH2 47 35 CN[C@@H](C)C(=O)N[C@H]1CCC[C@@H](C)[C@@H]1C ZINC000217597828 BD For-Sale Unstable BIRC2 47 31 COCCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217597843 GD In-Stock Unstable CA2 20 47 COCCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217597843 GD In-Stock Unstable TBXA2R 51 40 COCCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217597843 GD In-Stock Unstable CA1 19 40 COCCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217597843 GD In-Stock Unstable BDKRB1 0 45 COCCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217597843 GD In-Stock Unstable PRTN3 44 31 COCCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217597843 GD In-Stock Unstable AKR1C3 16 50 O=C1O[C@]2(CCCN(C(=O)c3cccc4ccccc34)C2)c2ccccc21 ZINC000217597884 FI For-Sale Unstable NPY5R 29 41 CC(=O)N(C(=O)NCC1CCCCC1)c1cccc(N)c1 ZINC000217597887 CF For-Sale Unstable AMY2 43 30 O=C(CCCC(=O)N1CCC(N2CCC[C@H]2COCc2ccccc2)CC1)c1ccccc1 ZINC000217597894 IJ In-Stock Unstable PREP 56 40 O=C(CCCC(=O)N1CCC(N2CCC[C@H]2COCc2ccccc2)CC1)c1ccccc1 ZINC000217597894 IJ In-Stock Unstable CYP2J2 44 31 CCO[C@H]1C[C@H](NC(=O)c2cccc(C#N)c2)C1(C)C ZINC000217597910 CE For-Sale Unstable ABCC9 40 42 CCO[C@H]1C[C@H](NC(=O)c2cccc(C#N)c2)C1(C)C ZINC000217597910 CE For-Sale Unstable EZH2 47 35 CN[C@H](C)C(=O)N[C@H]1CCC[C@@H](C)[C@@H]1C ZINC000217597915 BD For-Sale Unstable BIRC2 47 31 COc1ccc(CCNC(=O)CCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@H]23)cc1OC ZINC000217597924 JH In-Stock Unstable MTNR1B 15 41 COCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217597944 HD In-Stock Unstable CA2 19 40 COCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217597944 HD In-Stock Unstable TBXA2R 49 43 COCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217597944 HD In-Stock Unstable TBXAS1 15 42 COCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217597944 HD In-Stock Unstable BMP1 57 36 COCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217597944 HD In-Stock Unstable CA1 20 45 COCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217597944 HD In-Stock Unstable MMP13 53 40 COCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217597944 HD In-Stock Unstable MMP2 32 40 COCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217597944 HD In-Stock Unstable MMP8 25 40 COCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217597944 HD In-Stock Unstable MMP14 17 40 COCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217597944 HD In-Stock Unstable MMP9 46 40 COCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217597944 HD In-Stock Unstable MMP12 25 40 COCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217597944 HD In-Stock Unstable PTGDR 24 42 COCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217597944 HD In-Stock Unstable IAP 0 45 COCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217597944 HD In-Stock Unstable CA9 26 45 COCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217597944 HD In-Stock Unstable MMP1 47 37 COCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217597944 HD In-Stock Unstable AKR1C3 29 46 COCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217597944 HD In-Stock Unstable AKR1C2 50 37 CC(=O)Nc1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217597963 CG On-Demand Unstable ACAT 0 44 CC(=O)Nc1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217597963 CG On-Demand Unstable METAP2 0 44 O=C(CCCC(=O)N1CCC(N2CCC[C@@H]2COCc2ccccc2)CC1)c1ccccc1 ZINC000217597969 IJ In-Stock Unstable PREP 56 40 O=C(CCCC(=O)N1CCC(N2CCC[C@@H]2COCc2ccccc2)CC1)c1ccccc1 ZINC000217597969 IJ In-Stock Unstable CYP2J2 44 31 O=C1O[C@@]2(CCCN(C(=O)COc3cccnc3)C2)c2ccccc21 ZINC000217597995 EE For-Sale Unstable COLA 41 37 O=C1O[C@@]2(CCCN(C(=O)COc3cccnc3)C2)c2ccccc21 ZINC000217597995 EE For-Sale Unstable CPT2 43 32 O=C1O[C@@]2(CCCN(C(=O)COc3cccnc3)C2)c2ccccc21 ZINC000217597995 EE For-Sale Unstable NPY5R 47 42 CCCOc1ccc([C@@H](O)CN2CCCO[C@@H](C)C2)cc1 ZINC000217597996 CF For-Sale Unstable PSMB2 46 38 CCCOc1ccc([C@@H](O)CN2CCCO[C@@H](C)C2)cc1 ZINC000217597996 CF For-Sale Unstable PSMB1 41 38 COc1ccc(CCNC(=O)CCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@@H]23)cc1OC ZINC000217598003 JH In-Stock Unstable MTNR1B 15 41 COCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217598057 ID In-Stock Unstable TBXA2R 43 39 COCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217598057 ID In-Stock Unstable IAP 0 47 COCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217598057 ID In-Stock Unstable SCMU_MYCTU 0 45 CCC(=O)CC(=O)N1C[C@H](C2CCCCC2)C[C@H]1C(=O)O ZINC000217598067 CE For-Sale Unstable ACE 27 57 O=C(CCc1cccc(Cl)c1)N1CCC(N2CCC[C@H]2COCc2ccccc2)CC1 ZINC000217598070 IJ In-Stock Unstable C3AR1 36 40 O=C1O[C@]2(CCCN(C(=O)COc3cccnc3)C2)c2ccccc21 ZINC000217598081 EE For-Sale Unstable COLA 41 37 O=C1O[C@]2(CCCN(C(=O)COc3cccnc3)C2)c2ccccc21 ZINC000217598081 EE For-Sale Unstable CPT2 43 32 O=C1O[C@]2(CCCN(C(=O)COc3cccnc3)C2)c2ccccc21 ZINC000217598081 EE For-Sale Unstable NPY5R 47 42 CCCOc1ccc([C@H](O)CN2CCCO[C@@H](C)C2)cc1 ZINC000217598082 CF For-Sale Unstable PSMB2 46 38 CCCOc1ccc([C@H](O)CN2CCCO[C@@H](C)C2)cc1 ZINC000217598082 CF For-Sale Unstable PSMB1 41 38 O=C(CCc1cccc(Cl)c1)N1CCC(N2CCC[C@@H]2COCc2ccccc2)CC1 ZINC000217598157 IJ In-Stock Unstable C3AR1 36 40 COCCNS(=O)(=O)c1ccc(NCc2ccco2)c(C(=O)O)c1 ZINC000217598170 FD In-Stock Unstable BDKRB1 0 41 O=C1O[C@@]2(CCCN(C(=O)Cc3cccc4ccccc34)C2)c2ccccc21 ZINC000217598198 FI In-Stock Unstable NPY5R 26 40 C=C(C)Cc1c(C)nn(CCC(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)c1C ZINC000217598271 GF In-Stock Unstable CHRNA4 28 49 COCCNS(=O)(=O)c1ccc(NC[C@@H]2CCCO2)c(C(=O)O)c1 ZINC000217598283 FC In-Stock Unstable BDKRB1 0 40 O=C1O[C@]2(CCCN(C(=O)Cc3cccc4ccccc34)C2)c2ccccc21 ZINC000217598289 FI In-Stock Unstable NPY5R 26 40 COCCNS(=O)(=O)c1ccc(NC[C@H]2CCCO2)c(C(=O)O)c1 ZINC000217598366 FC In-Stock Unstable BDKRB1 0 40 CCOc1ccc(NC(=O)C(F)F)cc1 ZINC000217598374 BE On-Demand Unstable CA1 31 41 CCOc1ccc(NC(=O)C(F)F)cc1 ZINC000217598374 BE On-Demand Unstable SCN2A 38 47 CCOc1ccc(NC(=O)C(F)F)cc1 ZINC000217598374 BE On-Demand Unstable PRNP 15 49 CCOc1ccc(NC(=O)C(F)F)cc1 ZINC000217598374 BE On-Demand Unstable FAAH 20 40 CCOc1ccc(NC(=O)C(F)F)cc1 ZINC000217598374 BE On-Demand Unstable CA12 17 41 CCOc1ccc(NC(=O)C(F)F)cc1 ZINC000217598374 BE On-Demand Unstable CA9 17 41 CCOc1ccc(NC(=O)C(F)F)cc1 ZINC000217598374 BE On-Demand Unstable O69638_MYCTO 0 40 C=C(CC)COc1cc(/C=C\C(=O)O)ccc1[N+](=O)[O-] ZINC000217598394 CG For-Sale Unstable AKR1C3 29 47 O=C1O[C@@]2(CCCN(C(=O)Cc3c[nH]c4ccccc34)C2)c2ccccc21 ZINC000217598400 FG For-Sale Unstable AVPR1A 15 46 O=C1O[C@]2(CCCN(C(=O)Cc3c[nH]c4ccccc34)C2)c2ccccc21 ZINC000217598477 FG For-Sale Unstable AVPR1A 15 46 COCCNS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217598481 EC In-Stock Unstable SLC6A9 17 41 COCCNS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217598481 EC In-Stock Unstable SFRP1 47 32 N#Cc1ccc(CCC(=O)N2CCC(N3CCC[C@H]3COCc3ccccc3)CC2)cc1 ZINC000217598482 II In-Stock Unstable PREP 50 39 C=C(CC)COc1ccc(/C=C\C(=O)O)cc1Br ZINC000217598502 DH For-Sale Unstable APP 44 33 C=C(CC)COc1ccc(/C=C\C(=O)O)cc1Br ZINC000217598502 DH For-Sale Unstable AKR1C3 31 47 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1ccc(N(C)C)nc1 ZINC000217598535 CI For-Sale Unstable TRPM8 15 40 Cn1ccc2cc(C(=O)N[C@H](CCCNC(N)=O)C(=O)O)ccc21 ZINC000217598558 EC In-Stock Unstable DHFR 54 40 Cn1ccc2cc(C(=O)N[C@H](CCCNC(N)=O)C(=O)O)ccc21 ZINC000217598558 EC In-Stock Unstable CA2 17 48 Cn1ccc2cc(C(=O)N[C@H](CCCNC(N)=O)C(=O)O)ccc21 ZINC000217598558 EC In-Stock Unstable FOLH1 57 35 Cn1ccc2cc(C(=O)N[C@H](CCCNC(N)=O)C(=O)O)ccc21 ZINC000217598558 EC In-Stock Unstable NPFFR2 28 40 Cn1ccc2cc(C(=O)N[C@H](CCCNC(N)=O)C(=O)O)ccc21 ZINC000217598558 EC In-Stock Unstable C3AR1 72 40 Cn1ccc2cc(C(=O)N[C@H](CCCNC(N)=O)C(=O)O)ccc21 ZINC000217598558 EC In-Stock Unstable FPGS 57 32 Cn1ccc2cc(C(=O)N[C@H](CCCNC(N)=O)C(=O)O)ccc21 ZINC000217598558 EC In-Stock Unstable PCSK5 50 32 Cn1ccc2cc(C(=O)N[C@H](CCCNC(N)=O)C(=O)O)ccc21 ZINC000217598558 EC In-Stock Unstable FURIN 59 33 Cn1ccc2cc(C(=O)N[C@H](CCCNC(N)=O)C(=O)O)ccc21 ZINC000217598558 EC In-Stock Unstable CCKBR 23 40 Cn1ccc2cc(C(=O)N[C@H](CCCNC(N)=O)C(=O)O)ccc21 ZINC000217598558 EC In-Stock Unstable NS3 28 40 Cn1ccc2cc(C(=O)N[C@H](CCCNC(N)=O)C(=O)O)ccc21 ZINC000217598558 EC In-Stock Unstable GART 61 33 Cn1ccc2cc(C(=O)N[C@H](CCCNC(N)=O)C(=O)O)ccc21 ZINC000217598558 EC In-Stock Unstable POLG_WNV 46 39 Cn1ccc2cc(C(=O)N[C@H](CCCNC(N)=O)C(=O)O)ccc21 ZINC000217598558 EC In-Stock Unstable F2RL1 44 38 Cn1ccc2cc(C(=O)N[C@H](CCCNC(N)=O)C(=O)O)ccc21 ZINC000217598558 EC In-Stock Unstable NPFFR1 44 38 Cn1ccc2cc(C(=O)N[C@H](CCCNC(N)=O)C(=O)O)ccc21 ZINC000217598558 EC In-Stock Unstable PADI4 0 40 Cn1ccc2cc(C(=O)N[C@H](CCCNC(N)=O)C(=O)O)ccc21 ZINC000217598558 EC In-Stock Unstable PADI1 0 40 Cn1ccc2cc(C(=O)N[C@H](CCCNC(N)=O)C(=O)O)ccc21 ZINC000217598558 EC In-Stock Unstable PADI3 0 40 N#Cc1ccc(CCC(=O)N2CCC(N3CCC[C@@H]3COCc3ccccc3)CC2)cc1 ZINC000217598570 II In-Stock Unstable PREP 50 39 COCCNS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217598581 ED In-Stock Unstable SLC6A9 15 43 CCC(CC)C(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217598583 DG For-Sale Unstable NPY5R 27 41 O=C(Nc1ccccc1Cl)C(F)F ZINC000217598589 BF On-Demand Anodyne CXCL8 63 47 O=C(Nc1ccccc1Cl)C(F)F ZINC000217598589 BF On-Demand Anodyne KCNQ2 64 41 O=C(Nc1ccccc1Cl)C(F)F ZINC000217598589 BF On-Demand Anodyne EPHB3 53 40 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1ccc(N(C)C)nc1 ZINC000217598621 CI For-Sale Unstable TRPM8 15 40 C=C(CC)COc1ccc(/C=C\C(=O)O)cc1C(F)(F)F ZINC000217598625 DI For-Sale Unstable RXRA 15 41 C=C(CC)COc1ccc(/C=C\C(=O)O)cc1C(F)(F)F ZINC000217598625 DI For-Sale Unstable AKR1C3 31 46 CCc1nnc(N2CCN(S(=O)(=O)c3cccc4cnccc34)[C@@H](C)C2)o1 ZINC000217598638 GE In-Stock Unstable Q95J97_RABIT 0 54 CCC(CC)C(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217598648 DG For-Sale Unstable NPY5R 27 41 CC(C)[C@H](NC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000217598665 JF In-Stock Unstable SSTR2 60 35 CC(C)[C@H](NC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000217598665 JF In-Stock Unstable EDNRA 28 40 CC(C)[C@H](NC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000217598665 JF In-Stock Unstable TACR1 37 41 CC(C)[C@H](NC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000217598665 JF In-Stock Unstable MC4R 32 40 CC(C)[C@H](NC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000217598665 JF In-Stock Unstable CCKAR 51 39 CC(C)[C@H](NC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000217598665 JF In-Stock Unstable CHRNA4 23 41 CC(C)[C@H](NC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000217598665 JF In-Stock Unstable BRS3 25 40 CC(C)[C@H](NC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000217598665 JF In-Stock Unstable NMBR 35 40 CC(C)[C@H](NC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000217598665 JF In-Stock Unstable MC3R 41 35 CC(C)[C@H](NC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000217598665 JF In-Stock Unstable MMP14 46 33 CC(C)[C@H](NC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000217598665 JF In-Stock Unstable GRPR 71 34 CC(C)[C@H](NC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000217598665 JF In-Stock Unstable ECE1 40 35 CC(C)[C@H](NC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000217598665 JF In-Stock Unstable CCKBR 63 38 CC(C)[C@H](NC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000217598665 JF In-Stock Unstable GHSR 40 34 CC(C)[C@H](NC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000217598665 JF In-Stock Unstable KISS1R 62 31 CC(=O)Nc1ccc(CC(=O)N2CCC(N3CCC[C@@H]3COCc3ccccc3)CC2)cc1 ZINC000217598681 IH In-Stock Unstable TSHR 42 32 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1ccc(N(C)C)nc1 ZINC000217598695 CI For-Sale Unstable TRPM8 15 40 COCCNS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1 ZINC000217598700 EC In-Stock Unstable BDKRB1 0 41 COCCNS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1 ZINC000217598700 EC In-Stock Unstable SLC6A9 20 46 COc1cc(/C=C/C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc(OC)c1OC ZINC000217598758 HG For-Sale Unstable NPY5R 24 44 CC(=O)Nc1ccc(CC(=O)N2CCC(N3CCC[C@H]3COCc3ccccc3)CC2)cc1 ZINC000217598771 IH In-Stock Unstable TSHR 42 32 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1ccc(N(C)C)nc1 ZINC000217598773 CI For-Sale Unstable TRPM8 15 40 CCOCCCNc1ccc(S(=O)(=O)NCCOC)cc1C(=O)O ZINC000217598791 FD In-Stock Unstable CASP3 0 40 CCOCCCNc1ccc(S(=O)(=O)NCCOC)cc1C(=O)O ZINC000217598791 FD In-Stock Unstable BDKRB1 0 44 COc1ccc(OC)c(NS(=O)(=O)[C@@H](C)CO)c1 ZINC000217598808 CC For-Sale Unstable CYP1B1 35 40 COc1ccc(OC)c(NS(=O)(=O)[C@@H](C)CO)c1 ZINC000217598808 CC For-Sale Unstable AKR1C2 48 35 COc1cc(/C=C/C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc(OC)c1OC ZINC000217598840 HG For-Sale Unstable NPY5R 24 44 CCN(CCc1ccncc1)C(=O)NCC1CCCCC1 ZINC000217598870 CG For-Sale Unstable USP1 0 40 Cc1nc2ccc(C(=O)N3CCC(N4CCC[C@@H]4COCc4ccccc4)CC3)cc2s1 ZINC000217598883 IJ In-Stock Unstable NMT1 17 41 Cc1nc2ccc(C(=O)N3CCC(N4CCC[C@@H]4COCc4ccccc4)CC3)cc2s1 ZINC000217598883 IJ In-Stock Unstable L3MBTL3 62 39 Cc1ccc(NC(=O)C(F)F)cc1 ZINC000217598885 AE On-Demand Unstable PSBA 0 52 COc1ccc(OC)c(NS(=O)(=O)[C@H](C)CO)c1 ZINC000217598893 CC For-Sale Unstable CYP1B1 35 40 COc1ccc(OC)c(NS(=O)(=O)[C@H](C)CO)c1 ZINC000217598893 CC For-Sale Unstable AKR1C2 48 35 COCCNS(=O)(=O)c1ccc(NCCCOC(C)C)c(C(=O)O)c1 ZINC000217598908 FD In-Stock Unstable BDKRB1 0 44 COc1ccc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c(OC)c1 ZINC000217598953 FG For-Sale Unstable OXTR 25 44 COc1ccc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c(OC)c1 ZINC000217598953 FG For-Sale Unstable NPY5R 24 47 COc1ccc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c(OC)c1 ZINC000217598953 FG For-Sale Unstable SCN5A 23 40 O=C(NCC1CCCCC1)Nc1ccccc1N1CCOCC1 ZINC000217598975 DG For-Sale Unstable KCNQ2 91 44 O=C(NCC1CCCCC1)Nc1ccccc1N1CCOCC1 ZINC000217598975 DG For-Sale Unstable KCNQ4 0 41 O=C(NCC1CCCCC1)Nc1ccccc1N1CCOCC1 ZINC000217598975 DG For-Sale Unstable MTOR 43 37 O=C(NCC1CCCCC1)Nc1ccccc1N1CCOCC1 ZINC000217598975 DG For-Sale Unstable EPHX2 15 45 O=C(NCC1CCCCC1)Nc1ccccc1N1CCOCC1 ZINC000217598975 DG For-Sale Unstable PGA5 43 31 O=C(NCC1CCCCC1)Nc1ccccc1N1CCOCC1 ZINC000217598975 DG For-Sale Unstable CSF1R 28 47 O=C(NCC1CCCCC1)Nc1ccccc1N1CCOCC1 ZINC000217598975 DG For-Sale Unstable AKR1C3 22 42 Cc1nc2ccc(C(=O)N3CCC(N4CCC[C@H]4COCc4ccccc4)CC3)cc2s1 ZINC000217598980 IJ In-Stock Unstable NMT1 17 41 Cc1nc2ccc(C(=O)N3CCC(N4CCC[C@H]4COCc4ccccc4)CC3)cc2s1 ZINC000217598980 IJ In-Stock Unstable L3MBTL3 62 39 O=C(NO)c1nc(N2CCOCC2)ncc1Cl ZINC000217599007 CC In-Stock Unstable PIK3CA 19 40 O=C(NO)c1nc(N2CCOCC2)ncc1Cl ZINC000217599007 CC In-Stock Unstable MTOR 15 40 O=C(Nc1cc(Cl)ccc1Cl)C(F)F ZINC000217599010 BG On-Demand Anodyne KCNMA1 18 40 CCCCCNc1ccc(S(=O)(=O)NCCOC)cc1C(=O)O ZINC000217599012 ED In-Stock Unstable CASP3 17 42 COc1ccc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c(OC)c1 ZINC000217599043 FG For-Sale Unstable OXTR 25 44 COc1ccc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c(OC)c1 ZINC000217599043 FG For-Sale Unstable NPY5R 24 47 COc1ccc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c(OC)c1 ZINC000217599043 FG For-Sale Unstable SCN5A 23 40 CC(=O)Nc1ccc(C(=O)N2CCC(N3CCC[C@@H]3COCc3ccccc3)CC2)cc1 ZINC000217599087 IH In-Stock Unstable AVPR2 42 36 CC(=O)Nc1ccc(C(=O)N2CCC(N3CCC[C@@H]3COCc3ccccc3)CC2)cc1 ZINC000217599087 IH In-Stock Unstable AVPR1A 45 38 CC(=O)Nc1ccc(C(=O)N2CCC(N3CCC[C@@H]3COCc3ccccc3)CC2)cc1 ZINC000217599087 IH In-Stock Unstable GRIN2B 18 41 CC(=O)Nc1ccc(C(=O)N2CCC(N3CCC[C@@H]3COCc3ccccc3)CC2)cc1 ZINC000217599087 IH In-Stock Unstable L3MBTL3 90 39 CN1CCN(c2ccc(NC(=O)NCC3CCCCC3)cc2)CC1 ZINC000217599088 EG For-Sale Unstable HTR1D 16 40 CN1CCN(c2ccc(NC(=O)NCC3CCCCC3)cc2)CC1 ZINC000217599088 EG For-Sale Unstable HTR1B 21 41 CN1CCN(c2ccc(NC(=O)NCC3CCCCC3)cc2)CC1 ZINC000217599088 EG For-Sale Unstable F10 0 43 CN1CCN(c2ccc(NC(=O)NCC3CCCCC3)cc2)CC1 ZINC000217599088 EG For-Sale Unstable LCK 19 66 CN1CCN(c2ccc(NC(=O)NCC3CCCCC3)cc2)CC1 ZINC000217599088 EG For-Sale Unstable HRH3 27 43 CN1CCN(c2ccc(NC(=O)NCC3CCCCC3)cc2)CC1 ZINC000217599088 EG For-Sale Unstable CCR3 49 38 CN1CCN(c2ccc(NC(=O)NCC3CCCCC3)cc2)CC1 ZINC000217599088 EG For-Sale Unstable PIK3CA 23 47 CN1CCN(c2ccc(NC(=O)NCC3CCCCC3)cc2)CC1 ZINC000217599088 EG For-Sale Unstable PRNP 41 47 CN1CCN(c2ccc(NC(=O)NCC3CCCCC3)cc2)CC1 ZINC000217599088 EG For-Sale Unstable MTOR 61 48 CN1CCN(c2ccc(NC(=O)NCC3CCCCC3)cc2)CC1 ZINC000217599088 EG For-Sale Unstable EPHX2 51 62 CN1CCN(c2ccc(NC(=O)NCC3CCCCC3)cc2)CC1 ZINC000217599088 EG For-Sale Unstable HCK 37 66 CN1CCN(c2ccc(NC(=O)NCC3CCCCC3)cc2)CC1 ZINC000217599088 EG For-Sale Unstable PIK3CG 17 43 CN1CCN(c2ccc(NC(=O)NCC3CCCCC3)cc2)CC1 ZINC000217599088 EG For-Sale Unstable FLT3 20 47 CN1CCN(c2ccc(NC(=O)NCC3CCCCC3)cc2)CC1 ZINC000217599088 EG For-Sale Unstable AURKA 18 42 CN1CCN(c2ccc(NC(=O)NCC3CCCCC3)cc2)CC1 ZINC000217599088 EG For-Sale Unstable CACNA1I 40 36 O=C(NO)c1nc(N2CCCCC2)ncc1Cl ZINC000217599098 CD In-Stock Unstable CNR1 50 31 COCCNS(=O)(=O)c1ccc(NCCC(C)C)c(C(=O)O)c1 ZINC000217599105 ED In-Stock Unstable CASP3 16 42 COCCNS(=O)(=O)c1ccc(NCCC(C)C)c(C(=O)O)c1 ZINC000217599105 ED In-Stock Unstable BDKRB1 17 44 COc1ccc(NC(=O)C(F)F)cc1 ZINC000217599130 BD On-Demand Unstable CA1 35 40 COc1ccc(NC(=O)C(F)F)cc1 ZINC000217599130 BD On-Demand Unstable MTNR1A 25 45 COc1ccc(NC(=O)C(F)F)cc1 ZINC000217599130 BD On-Demand Unstable MTNR1B 23 45 COc1ccc(NC(=O)C(F)F)cc1 ZINC000217599130 BD On-Demand Unstable MMP9 26 43 COc1ccc(NC(=O)C(F)F)cc1 ZINC000217599130 BD On-Demand Unstable MMP12 22 40 COc1ccc(NC(=O)C(F)F)cc1 ZINC000217599130 BD On-Demand Unstable ACR 42 33 COc1ccc(NC(=O)C(F)F)cc1 ZINC000217599130 BD On-Demand Unstable MMP1 22 41 COc1ccc(NC(=O)C(F)F)cc1 ZINC000217599130 BD On-Demand Unstable PDE9A 0 41 COc1ccc(NC(=O)C(F)F)cc1 ZINC000217599130 BD On-Demand Unstable AKR1C2 47 41 COc1ccc(NC(=O)C(F)F)cc1 ZINC000217599130 BD On-Demand Unstable PSBA 0 56 CS(=O)(=O)c1ccc(SC/C=C\CN)cc1 ZINC000217599136 CD For-Sale Unstable O49150_SOLTU 51 37 O=C1O[C@@]2(CCCN(C(=O)c3ccc4ccccc4c3)C2)c2ccccc21 ZINC000217599148 FI For-Sale Unstable NPY5R 31 41 O=C(NCC1CCCCC1)Nc1ccc(N2CCCCC2)cc1 ZINC000217599165 DI For-Sale Unstable HRH3 24 42 O=C(NCC1CCCCC1)Nc1ccc(N2CCCCC2)cc1 ZINC000217599165 DI For-Sale Unstable CCR3 39 40 O=C(NCC1CCCCC1)Nc1ccc(N2CCCCC2)cc1 ZINC000217599165 DI For-Sale Unstable MTOR 43 39 O=C(NCC1CCCCC1)Nc1ccc(N2CCCCC2)cc1 ZINC000217599165 DI For-Sale Unstable EPHX2 48 62 O=C(NCC1CCCCC1)Nc1ccc(N2CCCCC2)cc1 ZINC000217599165 DI For-Sale Unstable HCK 25 56 CC(=O)Nc1ccc(C(=O)N2CCC(N3CCC[C@H]3COCc3ccccc3)CC2)cc1 ZINC000217599170 IH In-Stock Unstable AVPR2 42 36 CC(=O)Nc1ccc(C(=O)N2CCC(N3CCC[C@H]3COCc3ccccc3)CC2)cc1 ZINC000217599170 IH In-Stock Unstable AVPR1A 45 38 CC(=O)Nc1ccc(C(=O)N2CCC(N3CCC[C@H]3COCc3ccccc3)CC2)cc1 ZINC000217599170 IH In-Stock Unstable GRIN2B 18 41 CC(=O)Nc1ccc(C(=O)N2CCC(N3CCC[C@H]3COCc3ccccc3)CC2)cc1 ZINC000217599170 IH In-Stock Unstable L3MBTL3 90 39 CC[C@@H](C)[C@@H](C(=O)N1CC[C@@H](Cl)C1)c1ccccc1 ZINC000217599175 CH For-Sale Unstable CHRM1 15 42 CC[C@@H](C)[C@@H](C(=O)N1CC[C@@H](Cl)C1)c1ccccc1 ZINC000217599175 CH For-Sale Unstable ACE 32 41 CC[C@@H](C)[C@@H](C(=O)N1CC[C@@H](Cl)C1)c1ccccc1 ZINC000217599175 CH For-Sale Unstable MME 17 41 CC[C@@H](C)[C@@H](C(=O)N1CC[C@@H](Cl)C1)c1ccccc1 ZINC000217599175 CH For-Sale Unstable CCR1 38 45 CC[C@@H](C)[C@@H](C(=O)N1CC[C@@H](Cl)C1)c1ccccc1 ZINC000217599175 CH For-Sale Unstable CCR5 39 40 CC[C@@H](C)[C@@H](C(=O)N1CC[C@@H](Cl)C1)c1ccccc1 ZINC000217599175 CH For-Sale Unstable DPP4 19 40 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NCCOC)cc1C(=O)O ZINC000217599209 ED In-Stock Unstable CASP3 17 41 O=C1O[C@]2(CCCN(C(=O)c3ccc4ccccc4c3)C2)c2ccccc21 ZINC000217599230 FI For-Sale Unstable NPY5R 31 41 COc1cccc([C@H](O)CN2CCCO[C@@H](C)C2)c1 ZINC000217599239 CD For-Sale Unstable OPRK1 0 43 O=C(Nc1cccc(Cl)c1)C(F)F ZINC000217599247 BF On-Demand Anodyne PPIA 23 46 O=C(Nc1cccc(Cl)c1)C(F)F ZINC000217599247 BF On-Demand Anodyne PTGER3 15 41 O=C(Nc1cccc(Cl)c1)C(F)F ZINC000217599247 BF On-Demand Anodyne GRM5 16 54 O=C(Nc1cccc(Cl)c1)C(F)F ZINC000217599247 BF On-Demand Anodyne TAAR1 17 51 O=C(Nc1cccc(Cl)c1)C(F)F ZINC000217599247 BF On-Demand Anodyne IMDH_CRYPV 18 43 O=C(Nc1cccc(Cl)c1)C(F)F ZINC000217599247 BF On-Demand Anodyne PSBA 0 56 O=C(Nc1cccc(Cl)c1)C(F)F ZINC000217599247 BF On-Demand Anodyne KCNK3 79 49 O=C(Nc1cccc(Cl)c1)C(F)F ZINC000217599247 BF On-Demand Anodyne KCNK9 51 45 CC[C@H](C)[C@@H](C(=O)N1CC[C@@H](Cl)C1)c1ccccc1 ZINC000217599251 CH For-Sale Unstable CHRM1 15 42 CC[C@H](C)[C@@H](C(=O)N1CC[C@@H](Cl)C1)c1ccccc1 ZINC000217599251 CH For-Sale Unstable ACE 32 41 CC[C@H](C)[C@@H](C(=O)N1CC[C@@H](Cl)C1)c1ccccc1 ZINC000217599251 CH For-Sale Unstable MME 17 41 CC[C@H](C)[C@@H](C(=O)N1CC[C@@H](Cl)C1)c1ccccc1 ZINC000217599251 CH For-Sale Unstable CCR1 38 45 CC[C@H](C)[C@@H](C(=O)N1CC[C@@H](Cl)C1)c1ccccc1 ZINC000217599251 CH For-Sale Unstable CCR5 39 40 CC[C@H](C)[C@@H](C(=O)N1CC[C@@H](Cl)C1)c1ccccc1 ZINC000217599251 CH For-Sale Unstable DPP4 19 40 O=C(c1cc(-c2ccccc2)n[nH]1)N1CCC(N2CCC[C@H]2COCc2ccccc2)CC1 ZINC000217599280 II In-Stock Unstable TACR3 19 46 CCC[C@H](C)Nc1ccc(S(=O)(=O)NCCOC)cc1C(=O)O ZINC000217599299 ED In-Stock Unstable CASP3 17 41 Cc1ccc(/C=C\C(=O)O)cc1NC(=O)OCC(C)C ZINC000217599311 CG For-Sale Unstable AKR1C3 28 43 O=C1O[C@@]2(CCCN(C(=O)c3ccc4ccccc4n3)C2)c2ccccc21 ZINC000217599328 FH For-Sale Unstable NPY5R 34 41 CC[C@@H](C)[C@H](C(=O)N1CC[C@@H](Cl)C1)c1ccccc1 ZINC000217599334 CH For-Sale Unstable CHRM1 15 42 CC[C@@H](C)[C@H](C(=O)N1CC[C@@H](Cl)C1)c1ccccc1 ZINC000217599334 CH For-Sale Unstable ACE 32 41 CC[C@@H](C)[C@H](C(=O)N1CC[C@@H](Cl)C1)c1ccccc1 ZINC000217599334 CH For-Sale Unstable MME 17 41 CC[C@@H](C)[C@H](C(=O)N1CC[C@@H](Cl)C1)c1ccccc1 ZINC000217599334 CH For-Sale Unstable CCR1 38 45 CC[C@@H](C)[C@H](C(=O)N1CC[C@@H](Cl)C1)c1ccccc1 ZINC000217599334 CH For-Sale Unstable CCR5 39 40 CC[C@@H](C)[C@H](C(=O)N1CC[C@@H](Cl)C1)c1ccccc1 ZINC000217599334 CH For-Sale Unstable DPP4 19 40 O=C(Nc1cccc(F)c1)C(F)F ZINC000217599365 AE On-Demand Anodyne PPIA 16 41 O=C(Nc1cccc(F)c1)C(F)F ZINC000217599365 AE On-Demand Anodyne TAAR1 17 40 O=C(Nc1cccc(F)c1)C(F)F ZINC000217599365 AE On-Demand Anodyne PARP15 43 31 O=C(Nc1cccc(F)c1)C(F)F ZINC000217599365 AE On-Demand Anodyne PSBA 0 59 O=C(Nc1cccc(F)c1)C(F)F ZINC000217599365 AE On-Demand Anodyne KCNK3 100 51 O=C(Nc1cccc(F)c1)C(F)F ZINC000217599365 AE On-Demand Anodyne KCNK9 65 48 O=C(Nc1cccc(F)c1)C(F)F ZINC000217599365 AE On-Demand Anodyne PARP10 65 36 O=C(c1cc(-c2ccccc2)n[nH]1)N1CCC(N2CCC[C@@H]2COCc2ccccc2)CC1 ZINC000217599369 II In-Stock Unstable TACR3 19 46 CN(C)c1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217599379 CG On-Demand Unstable CCR3 18 42 CN(C)c1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217599379 CG On-Demand Unstable EPHX2 33 67 CN(C)c1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217599379 CG On-Demand Unstable PRMT3 34 40 CN(C)S(=O)(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217599392 CD For-Sale Unstable PTGER2 24 43 CN(C)S(=O)(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217599392 CD For-Sale Unstable AKR1C3 32 41 O=C1O[C@]2(CCCN(C(=O)c3ccc4ccccc4n3)C2)c2ccccc21 ZINC000217599406 FH For-Sale Unstable NPY5R 34 41 COCCNS(=O)(=O)c1ccc(N[C@@H](C)COC)c(C(=O)O)c1 ZINC000217599411 EC In-Stock Unstable BDKRB1 0 40 CC[C@H](C)[C@H](C(=O)N1CC[C@@H](Cl)C1)c1ccccc1 ZINC000217599414 CH For-Sale Unstable CHRM1 15 42 CC[C@H](C)[C@H](C(=O)N1CC[C@@H](Cl)C1)c1ccccc1 ZINC000217599414 CH For-Sale Unstable ACE 32 41 CC[C@H](C)[C@H](C(=O)N1CC[C@@H](Cl)C1)c1ccccc1 ZINC000217599414 CH For-Sale Unstable MME 17 41 CC[C@H](C)[C@H](C(=O)N1CC[C@@H](Cl)C1)c1ccccc1 ZINC000217599414 CH For-Sale Unstable CCR1 38 45 CC[C@H](C)[C@H](C(=O)N1CC[C@@H](Cl)C1)c1ccccc1 ZINC000217599414 CH For-Sale Unstable CCR5 39 40 CC[C@H](C)[C@H](C(=O)N1CC[C@@H](Cl)C1)c1ccccc1 ZINC000217599414 CH For-Sale Unstable DPP4 19 40 C[C@@H](NC(=O)CN1CCOc2ccccc2C1)c1ccc2c(c1)OCCO2 ZINC000217599465 FF In-Stock Unstable KCNQ2 24 42 CCOc1ccccc1[C@@H](O)CN1CCCO[C@@H](C)C1 ZINC000217599478 CE For-Sale Unstable ABCB1 16 43 CCOc1ccccc1[C@@H](O)CN1CCCO[C@@H](C)C1 ZINC000217599478 CE For-Sale Unstable HCN1 41 32 CCOc1ccccc1[C@@H](O)CN1CCCO[C@@H](C)C1 ZINC000217599478 CE For-Sale Unstable HCN4 41 32 CN(Cc1cccc(/C=C\C(=O)O)c1)S(=O)(=O)C(F)F ZINC000217599486 DD For-Sale Unstable PTGER2 23 41 CN(Cc1cccc(/C=C\C(=O)O)c1)S(=O)(=O)C(F)F ZINC000217599486 DD For-Sale Unstable AKR1C3 35 43 Cc1ccc(NC(=O)C(F)F)cc1Cl ZINC000217599488 BF On-Demand Unstable DHODH 15 46 Cc1ccc(NC(=O)C(F)F)cc1Cl ZINC000217599488 BF On-Demand Unstable PPIA 16 47 Cc1ccc(NC(=O)C(F)F)cc1Cl ZINC000217599488 BF On-Demand Unstable NPY2R 45 37 Cc1ccc(NC(=O)C(F)F)cc1Cl ZINC000217599488 BF On-Demand Unstable P95276_MYCTO 0 40 Cc1ccc(NC(=O)C(F)F)cc1Cl ZINC000217599488 BF On-Demand Unstable PSBA 0 43 Cc1ccc(NC(=O)C(F)F)cc1Cl ZINC000217599488 BF On-Demand Unstable PPX1 0 43 O=C(NCC1CCCCC1)N(Cc1ccccc1)c1ccccc1 ZINC000217599495 DJ For-Sale Unstable CHRM2 28 45 O=C(NCC1CCCCC1)N(Cc1ccccc1)c1ccccc1 ZINC000217599495 DJ For-Sale Unstable CHRM1 26 47 O=C(NCC1CCCCC1)N(Cc1ccccc1)c1ccccc1 ZINC000217599495 DJ For-Sale Unstable CHRM3 30 47 O=C(NCC1CCCCC1)N(Cc1ccccc1)c1ccccc1 ZINC000217599495 DJ For-Sale Unstable AMY2 46 32 O=C(NCC1CCCCC1)N(Cc1ccccc1)c1ccccc1 ZINC000217599495 DJ For-Sale Unstable NR1H4 27 41 COCCNS(=O)(=O)c1ccc(N[C@H](C)COC)c(C(=O)O)c1 ZINC000217599500 EC In-Stock Unstable BDKRB1 0 40 Cc1ccc(OCC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217599534 FG For-Sale Unstable COLA 43 35 Cc1ccc(OCC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217599534 FG For-Sale Unstable NPY5R 26 40 C[C@H](NC(=O)CN1CCOc2ccccc2C1)c1ccc2c(c1)OCCO2 ZINC000217599552 FF In-Stock Unstable KCNQ2 24 42 CCOc1ccccc1[C@H](O)CN1CCCO[C@@H](C)C1 ZINC000217599564 CE For-Sale Unstable ABCB1 16 43 CCOc1ccccc1[C@H](O)CN1CCCO[C@@H](C)C1 ZINC000217599564 CE For-Sale Unstable HCN1 41 32 CCOc1ccccc1[C@H](O)CN1CCCO[C@@H](C)C1 ZINC000217599564 CE For-Sale Unstable HCN4 41 32 CC(C)COC(=O)N[C@@H](C)c1ccc(/C=C\C(=O)O)cc1 ZINC000217599574 CG For-Sale Unstable AKR1C3 26 41 CCCNc1ccc(S(=O)(=O)NCCCOC)cc1C(=O)O ZINC000217599604 ED In-Stock Unstable CASP3 22 43 Cc1ccc(OCC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217599618 FG For-Sale Unstable COLA 43 35 Cc1ccc(OCC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217599618 FG For-Sale Unstable NPY5R 26 40 COc1ccc2nc(C(=O)Nc3ccc(-c4nc5ccccc5s4)cn3)ccc2c1 ZINC000217599619 HK On-Demand Unstable APP 19 44 COc1ccc2nc(C(=O)Nc3ccc(-c4nc5ccccc5s4)cn3)ccc2c1 ZINC000217599619 HK On-Demand Unstable MTTP 44 35 COc1ccc2nc(C(=O)Nc3ccc(-c4nc5ccccc5s4)cn3)ccc2c1 ZINC000217599619 HK On-Demand Unstable LUCI_LUCLA 46 51 COc1ccc2nc(C(=O)Nc3ccc(-c4nc5ccccc5s4)cn3)ccc2c1 ZINC000217599619 HK On-Demand Unstable LUCI_PHOPY 17 50 COc1ccc2nc(C(=O)Nc3ccc(-c4nc5ccccc5s4)cn3)ccc2c1 ZINC000217599619 HK On-Demand Unstable LUCI_PHOPE 36 50 COc1ccc2nc(C(=O)Nc3ccc(-c4nc5ccccc5s4)cn3)ccc2c1 ZINC000217599619 HK On-Demand Unstable ETHR 20 51 CC(C)COC(=O)N[C@H](C)c1ccc(/C=C\C(=O)O)cc1 ZINC000217599654 CG For-Sale Unstable AKR1C3 26 41 NS(=O)(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217599677 CC On-Demand Unstable CA2 100 64 NS(=O)(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217599677 CC On-Demand Unstable CA1 86 52 NS(=O)(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217599677 CC On-Demand Unstable CA7 56 43 NS(=O)(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217599677 CC On-Demand Unstable CA5B 62 38 NS(=O)(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217599677 CC On-Demand Unstable CA4 97 64 NS(=O)(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217599677 CC On-Demand Unstable CA5A 67 38 NS(=O)(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217599677 CC On-Demand Unstable CA14 37 44 NS(=O)(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217599677 CC On-Demand Unstable CA12 57 63 NS(=O)(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217599677 CC On-Demand Unstable CA9 61 63 NS(=O)(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217599677 CC On-Demand Unstable CAH_METTE 36 43 NS(=O)(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217599677 CC On-Demand Unstable TTK 36 41 NS(=O)(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217599677 CC On-Demand Unstable CYNT 35 55 NS(=O)(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217599677 CC On-Demand Unstable NCE103 43 35 NS(=O)(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217599677 CC On-Demand Unstable MTCA1 53 44 NS(=O)(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217599677 CC On-Demand Unstable P96878_MYCTU 63 44 NS(=O)(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217599677 CC On-Demand Unstable Q5TU56_ANOGA 0 48 O=C(C[C@@H]1NC(=O)N(Cc2ccccc2)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217599684 GD In-Stock Unstable MME 52 42 CC[C@H](O)[C@H](N)COCc1ccccc1 ZINC000217599686 BD For-Sale Unstable TACR1 0 58 CC[C@H](O)[C@H](N)COCc1ccccc1 ZINC000217599686 BD For-Sale Unstable CAPN2 51 33 CC[C@H](O)[C@H](N)COCc1ccccc1 ZINC000217599686 BD For-Sale Unstable POL 0 50 Cc1cc2cc(Cl)cc(C(=O)O)c2s1 ZINC000217599696 BH For-Sale Unstable AKR1C2 21 42 Cc1cc2cc(Cl)cc(C(=O)O)c2s1 ZINC000217599696 BH For-Sale Unstable AKR1C1 23 42 COCCCNS(=O)(=O)c1ccc(NC(C)C)c(C(=O)O)c1 ZINC000217599705 ED In-Stock Unstable CASP3 25 42 NC(=O)c1cc(C(F)(F)F)n(-c2ccccc2)n1 ZINC000217599709 CD In-Stock Unstable SCN10A 21 52 NC(=O)c1cc(C(F)(F)F)n(-c2ccccc2)n1 ZINC000217599709 CD In-Stock Unstable RPA1 44 35 O=C1O[C@@]2(CCCN(C(=O)c3ccc(Cn4ccnc4)cc3)C2)c2ccccc21 ZINC000217599716 GG For-Sale Unstable CYP19A1 15 46 O=C1O[C@@]2(CCCN(C(=O)c3ccc(Cn4ccnc4)cc3)C2)c2ccccc21 ZINC000217599716 GG For-Sale Unstable TBXAS1 25 42 CN1C(=O)c2ccc(C(=O)Nc3ccc(-c4nc5ccccc5s4)cn3)cc2C1=O ZINC000217599723 HH On-Demand Unstable MTTP 50 34 CN1C(=O)c2ccc(C(=O)Nc3ccc(-c4nc5ccccc5s4)cn3)cc2C1=O ZINC000217599723 HH On-Demand Unstable RPS6KA3 45 39 CN1C(=O)c2ccc(C(=O)Nc3ccc(-c4nc5ccccc5s4)cn3)cc2C1=O ZINC000217599723 HH On-Demand Unstable LUCI_LUCLA 37 41 CC(C)COC(=O)Nc1ccc(/C=C\C(=O)O)cc1F ZINC000217599741 CG For-Sale Unstable AKR1C3 29 42 CC[C@@H](O)[C@H](N)COCc1ccccc1 ZINC000217599761 BD For-Sale Unstable TACR1 0 58 CC[C@@H](O)[C@H](N)COCc1ccccc1 ZINC000217599761 BD For-Sale Unstable CAPN2 51 33 CC[C@@H](O)[C@H](N)COCc1ccccc1 ZINC000217599761 BD For-Sale Unstable POL 0 50 CCCCNc1ccc(S(=O)(=O)NCCCOC)cc1C(=O)O ZINC000217599791 ED In-Stock Unstable CASP3 22 42 CCO[C@@H]1C[C@@H](NC(=O)c2cc(Cl)ccc2O)C1(C)C ZINC000217599797 CF For-Sale Unstable KCNMA1 26 42 O=C1O[C@]2(CCCN(C(=O)c3ccc(Cn4ccnc4)cc3)C2)c2ccccc21 ZINC000217599800 GG For-Sale Unstable CYP19A1 15 46 O=C1O[C@]2(CCCN(C(=O)c3ccc(Cn4ccnc4)cc3)C2)c2ccccc21 ZINC000217599800 GG For-Sale Unstable TBXAS1 25 42 O=C(C[C@@H](c1cccc(O)c1)c1c(O)c(O)c(O)c2c(=O)cc(-c3ccccc3)oc12)N1CCOCC1 ZINC000217599802 KH In-Stock Unstable PRKDC 21 45 CCCS(=O)(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217599827 CD For-Sale Unstable PTGER2 0 41 CCCS(=O)(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217599827 CD For-Sale Unstable AKR1C3 31 40 CC(C)N(C)S(=O)(=O)c1ccc(C(=O)Nc2ccc(-c3nc4ccccc4s3)cn2)cc1 ZINC000217599828 JJ On-Demand Unstable PRNP 21 40 CC(C)N(C)S(=O)(=O)c1ccc(C(=O)Nc2ccc(-c3nc4ccccc4s3)cn2)cc1 ZINC000217599828 JJ On-Demand Unstable ATR 19 40 CC(C)N(C)S(=O)(=O)c1ccc(C(=O)Nc2ccc(-c3nc4ccccc4s3)cn2)cc1 ZINC000217599828 JJ On-Demand Unstable LUCI_LUCLA 36 42 CC[C@H](O)[C@@H](N)COCc1ccccc1 ZINC000217599855 BD For-Sale Unstable TACR1 0 58 CC[C@H](O)[C@@H](N)COCc1ccccc1 ZINC000217599855 BD For-Sale Unstable CAPN2 51 33 CC[C@H](O)[C@@H](N)COCc1ccccc1 ZINC000217599855 BD For-Sale Unstable POL 0 50 CCO[C@H]1C[C@@H](NC(=O)c2cc(Cl)ccc2O)C1(C)C ZINC000217599868 CF For-Sale Unstable KCNMA1 26 42 NS(=O)(=O)c1cccc(NC(=O)c2ccc(=O)[nH]n2)c1 ZINC000217599881 CB For-Sale Unstable CA2 47 60 NS(=O)(=O)c1cccc(NC(=O)c2ccc(=O)[nH]n2)c1 ZINC000217599881 CB For-Sale Unstable CA1 40 44 NS(=O)(=O)c1cccc(NC(=O)c2ccc(=O)[nH]n2)c1 ZINC000217599881 CB For-Sale Unstable CA5B 46 33 NS(=O)(=O)c1cccc(NC(=O)c2ccc(=O)[nH]n2)c1 ZINC000217599881 CB For-Sale Unstable CA4 46 60 NS(=O)(=O)c1cccc(NC(=O)c2ccc(=O)[nH]n2)c1 ZINC000217599881 CB For-Sale Unstable CA5A 52 33 NS(=O)(=O)c1cccc(NC(=O)c2ccc(=O)[nH]n2)c1 ZINC000217599881 CB For-Sale Unstable GRM4 40 33 NS(=O)(=O)c1cccc(NC(=O)c2ccc(=O)[nH]n2)c1 ZINC000217599881 CB For-Sale Unstable CA12 29 52 NS(=O)(=O)c1cccc(NC(=O)c2ccc(=O)[nH]n2)c1 ZINC000217599881 CB For-Sale Unstable CA9 34 52 NS(=O)(=O)c1cccc(NC(=O)c2ccc(=O)[nH]n2)c1 ZINC000217599881 CB For-Sale Unstable TTK 39 41 NS(=O)(=O)c1cccc(NC(=O)c2ccc(=O)[nH]n2)c1 ZINC000217599881 CB For-Sale Unstable CYNT 15 52 NS(=O)(=O)c1cccc(NC(=O)c2ccc(=O)[nH]n2)c1 ZINC000217599881 CB For-Sale Unstable MTCA1 40 38 NS(=O)(=O)c1cccc(NC(=O)c2ccc(=O)[nH]n2)c1 ZINC000217599881 CB For-Sale Unstable P96878_MYCTU 44 38 NS(=O)(=O)c1cccc(NC(=O)c2ccc(=O)[nH]n2)c1 ZINC000217599881 CB For-Sale Unstable KCNK3 51 36 O=C(C[C@H](c1cccc(O)c1)c1c(O)c(O)c(O)c2c(=O)cc(-c3ccccc3)oc12)N1CCOCC1 ZINC000217599887 KH In-Stock Unstable PRKDC 21 45 O=C(NCCc1cccnc1)[C@@H](O)Cc1ccccc1 ZINC000217599892 CD In-Stock Unstable ADRB2 21 40 O=C(NCCc1cccnc1)[C@@H](O)Cc1ccccc1 ZINC000217599892 CD In-Stock Unstable ADRB1 24 40 O=C(NCCc1cccnc1)[C@@H](O)Cc1ccccc1 ZINC000217599892 CD In-Stock Unstable ADRB3 48 41 O=C(NCCc1cccnc1)[C@@H](O)Cc1ccccc1 ZINC000217599892 CD In-Stock Unstable MME 67 40 O=C(NCCc1cccnc1)[C@@H](O)Cc1ccccc1 ZINC000217599892 CD In-Stock Unstable ANPEP 59 47 O=C(NCCc1cccnc1)[C@@H](O)Cc1ccccc1 ZINC000217599892 CD In-Stock Unstable TBXAS1 66 50 O=C(NCCc1cccnc1)[C@@H](O)Cc1ccccc1 ZINC000217599892 CD In-Stock Unstable PTAFR 40 50 O=C(NCCc1cccnc1)[C@@H](O)Cc1ccccc1 ZINC000217599892 CD In-Stock Unstable KCNA5 24 48 O=C(NCCc1cccnc1)[C@@H](O)Cc1ccccc1 ZINC000217599892 CD In-Stock Unstable CYSP_TRYCR 34 41 O=C(NCCc1cccnc1)[C@@H](O)Cc1ccccc1 ZINC000217599892 CD In-Stock Unstable BRS3 21 46 O=C(NCCc1cccnc1)[C@@H](O)Cc1ccccc1 ZINC000217599892 CD In-Stock Unstable C3AR1 45 40 O=C(NCCc1cccnc1)[C@@H](O)Cc1ccccc1 ZINC000217599892 CD In-Stock Unstable DNPEP 0 41 O=C(NCCc1cccnc1)[C@@H](O)Cc1ccccc1 ZINC000217599892 CD In-Stock Unstable MMP9 15 41 O=C(NCCc1cccnc1)[C@@H](O)Cc1ccccc1 ZINC000217599892 CD In-Stock Unstable LAP3 42 47 O=C(NCCc1cccnc1)[C@@H](O)Cc1ccccc1 ZINC000217599892 CD In-Stock Unstable POL 0 52 O=C(NCCc1cccnc1)[C@@H](O)Cc1ccccc1 ZINC000217599892 CD In-Stock Unstable AMP1_PLAFQ 63 50 O=C(NCCc1cccnc1)[C@@H](O)Cc1ccccc1 ZINC000217599892 CD In-Stock Unstable NAMPT 40 37 O=C(NCCc1cccnc1)[C@@H](O)Cc1ccccc1 ZINC000217599892 CD In-Stock Unstable GPR142 42 35 COCCCNS(=O)(=O)c1ccc(NCC(C)C)c(C(=O)O)c1 ZINC000217599901 ED In-Stock Unstable CASP3 18 43 O=C1O[C@@]2(CCCN(C(=O)COc3ccc(Cl)cc3Cl)C2)c2ccccc21 ZINC000217599905 HI For-Sale Unstable NPY5R 27 44 CCCCS(=O)(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217599912 DE For-Sale Unstable PTGER2 17 42 CCCCS(=O)(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217599912 DE For-Sale Unstable AKR1C3 29 44 CC[C@@H](O)[C@@H](N)COCc1ccccc1 ZINC000217599924 BD For-Sale Unstable TACR1 0 58 CC[C@@H](O)[C@@H](N)COCc1ccccc1 ZINC000217599924 BD For-Sale Unstable CAPN2 51 33 CC[C@@H](O)[C@@H](N)COCc1ccccc1 ZINC000217599924 BD For-Sale Unstable POL 0 50 CCO[C@@H]1C[C@H](NC(=O)c2cc(Cl)ccc2O)C1(C)C ZINC000217599937 CF For-Sale Unstable KCNMA1 26 42 CCc1cccc(OC/C=C\CN)c1 ZINC000217599946 AE For-Sale Unstable SQLE 43 32 COC(=O)C[C@H](c1ccc2c(c1)OCCO2)c1c(O)ccc2c(=O)c(-c3ccc(O)cc3)coc12 ZINC000217599982 JI In-Stock Unstable ALDH2 96 39 O=C1O[C@]2(CCCN(C(=O)COc3ccc(Cl)cc3Cl)C2)c2ccccc21 ZINC000217599986 HI For-Sale Unstable NPY5R 27 44 O=CNCCCNC(=O)NCC1CCCCC1 ZINC000217600002 BD For-Sale Unstable ADH1A 0 53 O=CNCCCNC(=O)NCC1CCCCC1 ZINC000217600002 BD For-Sale Unstable ADH1B 0 53 O=CNCCCNC(=O)NCC1CCCCC1 ZINC000217600002 BD For-Sale Unstable ADH1C 0 53 O=CNCCCNC(=O)NCC1CCCCC1 ZINC000217600002 BD For-Sale Unstable ADH4 0 53 CCO[C@H]1C[C@H](NC(=O)c2cc(Cl)ccc2O)C1(C)C ZINC000217600007 CF For-Sale Unstable KCNMA1 26 42 CC[C@@H](C)Nc1ccc(S(=O)(=O)NCCCOC)cc1C(=O)O ZINC000217600010 ED In-Stock Unstable CASP3 17 40 CNS(=O)(=O)c1ccc(C)c(C(=O)N2CCN([C@@H](C#N)c3ccccc3)CC2)c1 ZINC000217600059 HD On-Demand Unstable PTAFR 52 45 COC(=O)C[C@@H](c1ccc2c(c1)OCCO2)c1c(O)ccc2c(=O)c(-c3ccc(O)cc3)coc12 ZINC000217600066 JI In-Stock Unstable ALDH2 96 39 Cc1cnc(C(=O)N2CCC(N3CCC[C@@H]3COCc3ccccc3)CC2)cn1 ZINC000217600072 GG In-Stock Unstable PREP 49 39 CC[C@H](C)Nc1ccc(S(=O)(=O)NCCCOC)cc1C(=O)O ZINC000217600082 ED In-Stock Unstable CASP3 17 40 O=C1O[C@@]2(CCCN(C(=O)Cn3ncccc3=O)C2)c2ccccc21 ZINC000217600092 EC For-Sale Unstable NPY5R 33 41 CNS(=O)(=O)c1ccc(C)c(C(=O)N2CCN([C@H](C#N)c3ccccc3)CC2)c1 ZINC000217600141 HD On-Demand Unstable PTAFR 52 45 Cc1cnc(C(=O)N2CCC(N3CCC[C@H]3COCc3ccccc3)CC2)cn1 ZINC000217600151 GG In-Stock Unstable PREP 52 39 C[C@@H](CN[C@@H]1CCc2cc(O)ccc21)N(C)C1CC1 ZINC000217600157 CE For-Sale Unstable STS 40 36 O=C1O[C@]2(CCCN(C(=O)Cn3ncccc3=O)C2)c2ccccc21 ZINC000217600186 EC For-Sale Unstable NPY5R 33 41 COCCCNS(=O)(=O)c1ccc(NC(C)(C)C)c(C(=O)O)c1 ZINC000217600210 ED In-Stock Unstable PRTN3 45 32 Cc1nn(-c2cccc(C(=O)N(C)Cc3ccon3)c2)c(=O)c2ccccc12 ZINC000217600216 FF In-Stock Unstable PHOSPHO1 0 40 C[C@H](CN[C@@H]1CCc2cc(O)ccc21)N(C)C1CC1 ZINC000217600226 CE For-Sale Unstable STS 40 36 Cc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)N1CCN([C@@H](C#N)c2ccccc2)CC1 ZINC000217600255 IE On-Demand Unstable PTAFR 50 42 Cc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)N1CCN([C@@H](C#N)c2ccccc2)CC1 ZINC000217600255 IE On-Demand Unstable CCR8 75 35 Cc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)N1CCN([C@@H](C#N)c2ccccc2)CC1 ZINC000217600255 IE On-Demand Unstable SFRP1 122 38 Cc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)N1CCN([C@@H](C#N)c2ccccc2)CC1 ZINC000217600255 IE On-Demand Unstable WNT3 82 35 O=C(O)c1cnc(NCC2CC2)nc1 ZINC000217600259 AC On-Demand Unstable GRIN2B 25 40 O=C(O)c1cnc(NCC2CC2)nc1 ZINC000217600259 AC On-Demand Unstable PRKCQ 41 35 O=C(O)c1cnc(NCC2CC2)nc1 ZINC000217600259 AC On-Demand Unstable VCP 65 46 CC(C)(C)c1ccc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217600289 FI For-Sale Unstable NPY5R 26 41 C[C@@H](CN[C@H]1CCc2cc(O)ccc21)N(C)C1CC1 ZINC000217600298 CE For-Sale Unstable STS 40 36 C[C@H]1CN([C@@H](C)[C@@H](O)c2ccccc2)CCCO1 ZINC000217600303 BE For-Sale Unstable GRIN2C 17 41 C=CCNc1ccc(S(=O)(=O)NCCCOC)cc1C(=O)O ZINC000217600317 ED In-Stock Unstable CASP3 0 40 Cc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)N1CCN([C@H](C#N)c2ccccc2)CC1 ZINC000217600326 IE On-Demand Unstable PTAFR 50 42 Cc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)N1CCN([C@H](C#N)c2ccccc2)CC1 ZINC000217600326 IE On-Demand Unstable CCR8 75 35 Cc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)N1CCN([C@H](C#N)c2ccccc2)CC1 ZINC000217600326 IE On-Demand Unstable SFRP1 122 38 Cc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)N1CCN([C@H](C#N)c2ccccc2)CC1 ZINC000217600326 IE On-Demand Unstable WNT3 82 35 C[C@H](CN[C@H]1CCc2cc(O)ccc21)N(C)C1CC1 ZINC000217600372 CE For-Sale Unstable STS 40 36 CC(C)(C)c1ccc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217600373 FI For-Sale Unstable NPY5R 26 41 C[C@H]1CN([C@H](C)[C@@H](O)c2ccccc2)CCCO1 ZINC000217600394 BE For-Sale Unstable GRIN2C 17 41 COCCCNS(=O)(=O)c1ccc(NC2CC2)c(C(=O)O)c1 ZINC000217600425 ED In-Stock Unstable CASP3 24 42 O=C(Nc1ccc(Cl)cc1)C(F)F ZINC000217600441 BF On-Demand Anodyne GUAB 0 45 O=C(Nc1ccc(Cl)cc1)C(F)F ZINC000217600441 BF On-Demand Anodyne IMDH_CRYPV 25 42 O=C(Nc1ccc(Cl)cc1)C(F)F ZINC000217600441 BF On-Demand Anodyne P95276_MYCTO 0 47 O=C(Nc1ccc(Cl)cc1)C(F)F ZINC000217600441 BF On-Demand Anodyne PSBA 0 50 CN(C)c1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217600448 CG For-Sale Unstable CCKAR 22 40 CN(C)c1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217600448 CG For-Sale Unstable CCR3 60 39 CN(C)c1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217600448 CG For-Sale Unstable CCKBR 36 40 CN(C)c1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217600448 CG For-Sale Unstable EPHX2 25 67 CN(C)c1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217600448 CG For-Sale Unstable ACAT 0 43 COc1ccc2cc(C(=O)N3CCC(N4CCC[C@@H]4COCc4ccccc4)CC3)[nH]c2c1 ZINC000217600452 II In-Stock Unstable GRIN2B 46 53 COc1ccc2cc(C(=O)N3CCC(N4CCC[C@@H]4COCc4ccccc4)CC3)[nH]c2c1 ZINC000217600452 II In-Stock Unstable HRH4 15 43 COc1ccc2cc(C(=O)N3CCC(N4CCC[C@@H]4COCc4ccccc4)CC3)[nH]c2c1 ZINC000217600452 II In-Stock Unstable FPR2 31 47 COc1ccc2cc(C(=O)N3CCC(N4CCC[C@@H]4COCc4ccccc4)CC3)[nH]c2c1 ZINC000217600452 II In-Stock Unstable AKR1C3 18 41 CCCCNC(=O)Nc1cc(/C=C\C(=O)O)ccc1C ZINC000217600470 CG For-Sale Unstable ACAT 0 54 C[C@H]1CN([C@H](C)[C@H](O)c2ccccc2)CCCO1 ZINC000217600473 BE For-Sale Unstable GRIN2C 17 41 O=C1O[C@@]2(CCCN(C(=O)C3CCCCC3)C2)c2ccccc21 ZINC000217600500 DG For-Sale Unstable NPY5R 51 43 C[C@H](/C=C/CO)NC(=O)OC(C)(C)C ZINC000217600521 BD For-Sale Unstable PAPA1_CARPA 43 36 C[C@H](/C=C/CO)NC(=O)OC(C)(C)C ZINC000217600521 BD For-Sale Unstable CTSK 24 61 COCCCNS(=O)(=O)c1ccc(NC2CCCC2)c(C(=O)O)c1 ZINC000217600529 FE In-Stock Unstable CASP3 25 45 O=C(NCCc1cn[nH]c1)[C@@H]1CCCN1C(=O)C1CCCCC1 ZINC000217600532 DD In-Stock Unstable PREP 57 34 O=C(NCCc1cn[nH]c1)[C@@H]1CCCN1C(=O)C1CCCCC1 ZINC000217600532 DD In-Stock Unstable LGMN 55 32 COc1ccc2cc(C(=O)N3CCC(N4CCC[C@H]4COCc4ccccc4)CC3)[nH]c2c1 ZINC000217600537 II In-Stock Unstable GRIN2B 46 53 COc1ccc2cc(C(=O)N3CCC(N4CCC[C@H]4COCc4ccccc4)CC3)[nH]c2c1 ZINC000217600537 II In-Stock Unstable HRH4 15 43 COc1ccc2cc(C(=O)N3CCC(N4CCC[C@H]4COCc4ccccc4)CC3)[nH]c2c1 ZINC000217600537 II In-Stock Unstable FPR2 31 47 COc1ccc2cc(C(=O)N3CCC(N4CCC[C@H]4COCc4ccccc4)CC3)[nH]c2c1 ZINC000217600537 II In-Stock Unstable AKR1C3 18 41 CN1CCc2nc(NC(=O)NCC3CCCCC3)sc2C1 ZINC000217600566 DF For-Sale Unstable F10 26 47 O=C1O[C@]2(CCCN(C(=O)C3CCCCC3)C2)c2ccccc21 ZINC000217600586 DG For-Sale Unstable NPY5R 51 43 COc1ccc(CN2C(=O)N[C@@H](CC(=O)NCc3ccncc3)C2=O)cc1OC ZINC000217600594 GD In-Stock Unstable ENPP1 63 33 COCCCNS(=O)(=O)c1ccc(NC2CCCCC2)c(C(=O)O)c1 ZINC000217600637 FE In-Stock Unstable CASP3 23 44 Cn1c(=O)c2c(ncn2CCN2CCN(CCOc3ccccc3Cl)CC2)n(C)c1=O ZINC000217600647 IC On-Demand Unstable HTR1A 33 58 Cn1c(=O)c2c(ncn2CCN2CCN(CCOc3ccccc3Cl)CC2)n(C)c1=O ZINC000217600647 IC On-Demand Unstable HTR2A 22 58 Cn1c(=O)c2c(ncn2CCN2CCN(CCOc3ccccc3Cl)CC2)n(C)c1=O ZINC000217600647 IC On-Demand Unstable ADORA2A 0 50 Cn1c(=O)c2c(ncn2CCN2CCN(CCOc3ccccc3Cl)CC2)n(C)c1=O ZINC000217600647 IC On-Demand Unstable HTR7 31 58 O=C(Nc1ccccc1)N1CCC(N2CCC[C@H]2COCc2ccccc2)CC1 ZINC000217600656 GI In-Stock Unstable HRH3 26 45 O=C(Nc1ccccc1)N1CCC(N2CCC[C@H]2COCc2ccccc2)CC1 ZINC000217600656 GI In-Stock Unstable EPHX2 21 41 O=C(NCC1CCCCC1)Nc1ccc2nc[nH]c2c1 ZINC000217600672 CG For-Sale Unstable QPCT 16 40 O=C(NCC1CCCCC1)Nc1ccc2nc[nH]c2c1 ZINC000217600672 CG For-Sale Unstable PRMT3 71 47 Cc1cccc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217600704 DG For-Sale Unstable NPY5R 29 42 Cc1cccc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217600704 DG For-Sale Unstable HPGD 17 42 O=C(Nc1cccc(C(F)(F)F)c1)C(F)F ZINC000217600706 BF On-Demand Anodyne DHODH 0 48 O=C(Nc1cccc(C(F)(F)F)c1)C(F)F ZINC000217600706 BF On-Demand Anodyne KIT 17 44 O=C(Nc1cccc(C(F)(F)F)c1)C(F)F ZINC000217600706 BF On-Demand Anodyne LCK 27 40 O=C(Nc1cccc(C(F)(F)F)c1)C(F)F ZINC000217600706 BF On-Demand Anodyne TRPV1 21 50 O=C(Nc1cccc(C(F)(F)F)c1)C(F)F ZINC000217600706 BF On-Demand Anodyne KDR 19 44 O=C(Nc1cccc(C(F)(F)F)c1)C(F)F ZINC000217600706 BF On-Demand Anodyne NPY5R 18 41 O=C(Nc1cccc(C(F)(F)F)c1)C(F)F ZINC000217600706 BF On-Demand Anodyne SLC1A1 21 41 O=C(Nc1cccc(C(F)(F)F)c1)C(F)F ZINC000217600706 BF On-Demand Anodyne SLC1A3 18 41 O=C(Nc1cccc(C(F)(F)F)c1)C(F)F ZINC000217600706 BF On-Demand Anodyne EPHX2 18 52 O=C(Nc1cccc(C(F)(F)F)c1)C(F)F ZINC000217600706 BF On-Demand Anodyne SLC1A2 34 41 O=C(Nc1cccc(C(F)(F)F)c1)C(F)F ZINC000217600706 BF On-Demand Anodyne TEK 32 43 O=C(Nc1cccc(C(F)(F)F)c1)C(F)F ZINC000217600706 BF On-Demand Anodyne EPHA3 23 41 O=C(Nc1cccc(C(F)(F)F)c1)C(F)F ZINC000217600706 BF On-Demand Anodyne BTK 20 43 O=C(Nc1cccc(C(F)(F)F)c1)C(F)F ZINC000217600706 BF On-Demand Anodyne BRAF 33 40 O=C(Nc1cccc(C(F)(F)F)c1)C(F)F ZINC000217600706 BF On-Demand Anodyne EPHB4 28 41 O=C(Nc1cccc(C(F)(F)F)c1)C(F)F ZINC000217600706 BF On-Demand Anodyne AKR1C3 17 54 O=C(Nc1cccc(C(F)(F)F)c1)C(F)F ZINC000217600706 BF On-Demand Anodyne RIPK1 54 43 O=C(Nc1cccc(C(F)(F)F)c1)C(F)F ZINC000217600706 BF On-Demand Anodyne TRPM4 0 49 O=C(Nc1cccc(C(F)(F)F)c1)C(F)F ZINC000217600706 BF On-Demand Anodyne PSBA 0 61 O=C(Nc1cccc(C(F)(F)F)c1)C(F)F ZINC000217600706 BF On-Demand Anodyne KCNK3 75 54 O=C(Nc1cccc(C(F)(F)F)c1)C(F)F ZINC000217600706 BF On-Demand Anodyne KCNK9 55 35 O=C(Nc1cccc(C(F)(F)F)c1)C(F)F ZINC000217600706 BF On-Demand Anodyne PDS 43 41 NC/C=C\COc1cc(Cl)ccc1[N+](=O)[O-] ZINC000217600722 BE For-Sale Unstable PDE7A 0 44 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1ccc2[nH]ncc2c1 ZINC000217600740 CI For-Sale Unstable ROCK2 26 44 O=C(Nc1ccccc1)N1CCC(N2CCC[C@@H]2COCc2ccccc2)CC1 ZINC000217600749 GI In-Stock Unstable HRH3 26 45 O=C(Nc1ccccc1)N1CCC(N2CCC[C@@H]2COCc2ccccc2)CC1 ZINC000217600749 GI In-Stock Unstable EPHX2 21 41 COCCCNS(=O)(=O)c1ccc(NCCC2=CCCCC2)c(C(=O)O)c1 ZINC000217600767 GG In-Stock Unstable BDKRB1 16 40 Cc1cccc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217600788 DG For-Sale Unstable NPY5R 29 42 Cc1cccc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217600788 DG For-Sale Unstable HPGD 17 42 O=C(Cc1cccs1)N1C[C@H]2CNC[C@@H](C2)C1 ZINC000217600816 CD For-Sale Unstable ETHR 32 43 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1ccc2[nH]ncc2c1 ZINC000217600823 CI For-Sale Unstable ROCK2 26 44 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)N1CCN(C(c3ccccc3)c3ccccc3)CC1)C(=O)OC2 ZINC000217600836 KK In-Stock Unstable IMPDH2 51 48 COCCCNS(=O)(=O)c1ccc(NCCO)c(C(=O)O)c1 ZINC000217600884 EC In-Stock Unstable BDKRB1 0 44 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1ccc2[nH]ncc2c1 ZINC000217600900 CI For-Sale Unstable ROCK2 26 44 CCCC(CCC)C(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217600906 EH For-Sale Unstable NPY5R 25 40 COCCCNS(=O)(=O)c1ccc(NCCCO)c(C(=O)O)c1 ZINC000217600956 EC In-Stock Unstable CASP3 17 40 COCCCNS(=O)(=O)c1ccc(NCCCO)c(C(=O)O)c1 ZINC000217600956 EC In-Stock Unstable BDKRB1 0 44 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1ccc2[nH]ncc2c1 ZINC000217600963 CI For-Sale Unstable ROCK2 26 44 CCCC(CCC)C(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217600997 EH For-Sale Unstable NPY5R 25 40 C[C@@H]1CCCN(C(=O)C(F)F)C1 ZINC000217601025 AD On-Demand Unstable DPP7 28 41 c1cc2[nH]ncc2cc1N[C@@H]1C[C@@H]2C[C@H]1[C@@H]1CCC[C@H]21 ZINC000217601042 CH For-Sale Unstable ROCK2 0 43 COCCCNS(=O)(=O)c1ccc(NCCOC)c(C(=O)O)c1 ZINC000217601066 EC In-Stock Unstable CASP3 24 41 COCCCNS(=O)(=O)c1ccc(NCCOC)c(C(=O)O)c1 ZINC000217601066 EC In-Stock Unstable BDKRB1 0 46 O=C(NCC1CCCCC1)Nc1cccc(Br)c1 ZINC000217601101 DI On-Demand Unstable CCR3 45 38 O=C(NCC1CCCCC1)Nc1cccc(Br)c1 ZINC000217601101 DI On-Demand Unstable EPHX2 24 45 O=C(NCC1CCCCC1)Nc1cccc(Br)c1 ZINC000217601101 DI On-Demand Unstable PRMT3 35 41 O=C(NCC1CCCCC1)Nc1cccc(Br)c1 ZINC000217601101 DI On-Demand Unstable ACAT 0 43 Cc1ccc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217601112 DG For-Sale Unstable CHRM5 22 40 Cc1ccc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217601112 DG For-Sale Unstable NPY5R 30 44 C[C@H]1CCCN(C(=O)C(F)F)C1 ZINC000217601113 AD On-Demand Unstable DPP7 28 41 c1cc2[nH]ncc2cc1N[C@@H]1C[C@@H]2C[C@H]1[C@@H]1CCC[C@@H]21 ZINC000217601125 CH For-Sale Unstable ROCK2 0 43 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1cccc(OC)c1 ZINC000217601157 JH In-Stock Unstable CACNA1C 42 40 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1cccc(OC)c1 ZINC000217601157 JH In-Stock Unstable CACNA1D 76 40 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1cccc(OC)c1 ZINC000217601157 JH In-Stock Unstable TGFBR2 50 40 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1cccc(OC)c1 ZINC000217601157 JH In-Stock Unstable HISG 0 47 COCCCNc1ccc(S(=O)(=O)NCCCOC)cc1C(=O)O ZINC000217601168 FD In-Stock Unstable CASP3 18 41 COCCCNc1ccc(S(=O)(=O)NCCCOC)cc1C(=O)O ZINC000217601168 FD In-Stock Unstable BDKRB1 0 46 COCCCNc1ccc(S(=O)(=O)NCCCOC)cc1C(=O)O ZINC000217601168 FD In-Stock Unstable AKR1C3 28 40 O=C(NCC1C[C@@H]2CC[C@H](C1)N2)c1cccs1 ZINC000217601183 CE For-Sale Unstable GLRA1 30 54 Cc1ccc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217601187 DG For-Sale Unstable CHRM5 22 40 Cc1ccc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217601187 DG For-Sale Unstable NPY5R 30 44 COc1ccc(N2C(=O)[C@@H]3[C@@H](C(=O)c4ccc(F)cc4)N4CCC[C@@H]4[C@@H]3C2=O)cc1 ZINC000217601193 HF In-Stock Unstable SLC18A3 33 45 c1cc2[nH]ncc2cc1N[C@@H]1C[C@H]2C[C@H]1[C@@H]1CCC[C@H]21 ZINC000217601210 CH For-Sale Unstable ROCK2 0 43 CCOc1ccc(CCNC(=O)NCC2CCCCC2)cc1OCC ZINC000217601218 EH On-Demand Unstable SSTR5 69 37 CNc1nc(C2CC2)nc(N2CCN(C)[C@@H](C)C2)c1C ZINC000217601223 CD For-Sale Unstable CHRM3 16 50 CCC[C@H](CN(C=O)OCc1ccccc1)C(=O)O ZINC000217601230 CE For-Sale Unstable FOLH1 16 40 CCC[C@H](CN(C=O)OCc1ccccc1)C(=O)O ZINC000217601230 CE For-Sale Unstable CPA1 35 45 C[C@@H]1CN(C[C@@H](O)c2ccc3c(c2)OCO3)CCCO1 ZINC000217601239 CD For-Sale Unstable SSTR3 100 33 COC(=O)C[C@H](C1=C(O)C(=O)c2ccccc2C1=O)c1coc2ccc(OC)cc2c1=O ZINC000217601255 IG In-Stock Unstable ALDH2 54 33 COC(=O)C[C@H](C1=C(O)C(=O)c2ccccc2C1=O)c1coc2ccc(OC)cc2c1=O ZINC000217601255 IG In-Stock Unstable NQO2 22 44 COC(=O)C[C@H](C1=C(O)C(=O)c2ccccc2C1=O)c1coc2ccc(OC)cc2c1=O ZINC000217601255 IG In-Stock Unstable MTNR1A 46 44 COC(=O)C[C@H](C1=C(O)C(=O)c2ccccc2C1=O)c1coc2ccc(OC)cc2c1=O ZINC000217601255 IG In-Stock Unstable MTNR1B 37 44 COc1ccc(N2C(=O)[C@H]3[C@H](C2=O)[C@H]2CCCN2[C@@H]3C(=O)c2ccc(F)cc2)cc1 ZINC000217601270 HF In-Stock Unstable SLC18A3 33 45 CCN(C/C=C\CN)c1cccc2ccccc12 ZINC000217601273 BG For-Sale Unstable CHAT 44 31 O=C1O[C@@]2(CCCN(C(=O)c3ccc(S(=O)(=O)N4CCCC4)cc3)C2)c2ccccc21 ZINC000217601284 IF For-Sale Unstable NPY5R 23 40 COCCCNS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217601287 GE In-Stock Unstable BDKRB1 0 46 c1cc2[nH]ncc2cc1N[C@@H]1C[C@H]2C[C@H]1[C@@H]1CCC[C@@H]21 ZINC000217601295 CH For-Sale Unstable ROCK2 0 43 N#Cc1ccc(OCC(=O)Nc2cccc(O)c2)cc1 ZINC000217601309 CE On-Demand Unstable ADORA2B 40 45 N#Cc1ccc(OCC(=O)Nc2cccc(O)c2)cc1 ZINC000217601309 CE On-Demand Unstable HIF1A 23 47 C[C@H]1CN(C[C@@H](O)c2ccc3c(c2)OCO3)CCCO1 ZINC000217601322 CD For-Sale Unstable SSTR3 100 33 COC(=O)C[C@@H](C1=C(O)C(=O)c2ccccc2C1=O)c1coc2ccc(OC)cc2c1=O ZINC000217601333 IG In-Stock Unstable ALDH2 54 33 COC(=O)C[C@@H](C1=C(O)C(=O)c2ccccc2C1=O)c1coc2ccc(OC)cc2c1=O ZINC000217601333 IG In-Stock Unstable NQO2 22 44 COC(=O)C[C@@H](C1=C(O)C(=O)c2ccccc2C1=O)c1coc2ccc(OC)cc2c1=O ZINC000217601333 IG In-Stock Unstable MTNR1A 46 44 COC(=O)C[C@@H](C1=C(O)C(=O)c2ccccc2C1=O)c1coc2ccc(OC)cc2c1=O ZINC000217601333 IG In-Stock Unstable MTNR1B 37 44 CC(C)(C)c1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217601336 CJ For-Sale Unstable TRPV1 26 40 CC(C)(C)c1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217601336 CJ For-Sale Unstable CCR3 21 49 CC(C)(C)c1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217601336 CJ For-Sale Unstable AMY2 45 31 CC(C)(C)c1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217601336 CJ For-Sale Unstable EPHX2 57 69 CC(C)(C)c1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217601336 CJ For-Sale Unstable CACNA1I 52 46 CC(C)(C)c1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217601336 CJ For-Sale Unstable PRMT3 35 43 CC(C)(C)c1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217601336 CJ For-Sale Unstable DOT1L 44 32 O=C1O[C@]2(CCCN(C(=O)c3ccc(S(=O)(=O)N4CCCC4)cc3)C2)c2ccccc21 ZINC000217601361 IF For-Sale Unstable NPY5R 23 40 NC[C@@H]1CCCCN1C[C@@H]1COc2ccccc2O1 ZINC000217601366 CD On-Demand Unstable ADRA2B 23 45 C[C@@H](C(=O)NCCc1ccncc1)N(c1ccccc1)S(C)(=O)=O ZINC000217601385 ED In-Stock Unstable KCNA5 16 40 C[C@@H](C(=O)NCCc1ccncc1)N(c1ccccc1)S(C)(=O)=O ZINC000217601385 ED In-Stock Unstable CA5B 17 42 C[C@@H](C(=O)NCCc1ccncc1)N(c1ccccc1)S(C)(=O)=O ZINC000217601385 ED In-Stock Unstable CA5A 15 42 C[C@@H](C(=O)NCCc1ccncc1)N(c1ccccc1)S(C)(=O)=O ZINC000217601385 ED In-Stock Unstable AMP1_PLAFQ 27 41 O=C(COc1cc(C(F)(F)F)cc(C(F)(F)F)c1)Nc1nc(-c2ccccn2)cs1 ZINC000217601391 IK On-Demand Unstable MPL 57 38 O=C(COc1cc(C(F)(F)F)cc(C(F)(F)F)c1)Nc1nc(-c2ccccn2)cs1 ZINC000217601391 IK On-Demand Unstable NPY5R 23 54 O=C(COc1cc(C(F)(F)F)cc(C(F)(F)F)c1)Nc1nc(-c2ccccn2)cs1 ZINC000217601391 IK On-Demand Unstable KCNN1 28 44 O=C(COc1cc(C(F)(F)F)cc(C(F)(F)F)c1)Nc1nc(-c2ccccn2)cs1 ZINC000217601391 IK On-Demand Unstable TRPA1 23 40 COCCCNS(=O)(=O)c1ccc(N[C@@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217601401 GF In-Stock Unstable CASP3 20 41 C[C@@H]1CN([C@@H]2C[C@@H](c3ccccc3)CC[C@@H]2O)CCCO1 ZINC000217601417 CF For-Sale Unstable SLC18A3 85 49 CCCC1=C(C(=O)OCC)[C@H](c2cccc(Cl)c2Cl)C2=C(C[C@@H](c3cccs3)[C@@H](C(=O)OCC)C2=O)N1 ZINC000217601451 KK In-Stock Unstable TGFBR2 15 40 C[C@H](C(=O)NCCc1ccncc1)N(c1ccccc1)S(C)(=O)=O ZINC000217601482 ED In-Stock Unstable KCNA5 16 40 C[C@H](C(=O)NCCc1ccncc1)N(c1ccccc1)S(C)(=O)=O ZINC000217601482 ED In-Stock Unstable CA5B 17 42 C[C@H](C(=O)NCCc1ccncc1)N(c1ccccc1)S(C)(=O)=O ZINC000217601482 ED In-Stock Unstable CA5A 15 42 C[C@H](C(=O)NCCc1ccncc1)N(c1ccccc1)S(C)(=O)=O ZINC000217601482 ED In-Stock Unstable AMP1_PLAFQ 27 41 CCNc1nc(C2CC2)nc(N2CCN(C)[C@@H](C)C2)c1C ZINC000217601487 CE For-Sale Unstable CHRM3 21 47 COCCCNS(=O)(=O)c1ccc(N[C@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217601504 GF In-Stock Unstable CASP3 20 41 CCCC1=C(C(=O)OCC)[C@H](c2cccc(Cl)c2Cl)C2=C(C[C@H](c3cccs3)[C@@H](C(=O)OCC)C2=O)N1 ZINC000217601539 KK In-Stock Unstable TGFBR2 15 40 O=C(Nc1cccc(O)c1)C(F)F ZINC000217601544 AD On-Demand Anodyne KYNU 45 32 O=C(Nc1cccc(O)c1)C(F)F ZINC000217601544 AD On-Demand Anodyne PARP14 41 35 O=C(Nc1cccc(O)c1)C(F)F ZINC000217601544 AD On-Demand Anodyne PARP15 46 33 O=C(Nc1cccc(O)c1)C(F)F ZINC000217601544 AD On-Demand Anodyne PSBA 0 41 O=C(Nc1cccc(O)c1)C(F)F ZINC000217601544 AD On-Demand Anodyne KCNK9 50 36 O=C(Nc1cccc(O)c1)C(F)F ZINC000217601544 AD On-Demand Anodyne PARP10 74 38 Cc1ccc(NC(=O)Nc2ncc(/C=C\C(=O)O)s2)cc1 ZINC000217601605 DG For-Sale Unstable KIT 27 42 Cc1ccc(NC(=O)Nc2ncc(/C=C\C(=O)O)s2)cc1 ZINC000217601605 DG For-Sale Unstable KDR 23 42 Cc1ccc(NC(=O)Nc2ncc(/C=C\C(=O)O)s2)cc1 ZINC000217601605 DG For-Sale Unstable TEK 32 42 COCCCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217601617 GE In-Stock Unstable CA2 16 43 COCCCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217601617 GE In-Stock Unstable TBXA2R 49 39 COCCCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217601617 GE In-Stock Unstable CASP3 17 40 COCCCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217601617 GE In-Stock Unstable BDKRB1 0 46 COC(=O)[C@H]1C[C@@H](OC)CN1C(=O)CCc1ccccc1 ZINC000217601623 CD In-Stock Unstable ACE 47 40 COC(=O)[C@H]1C[C@@H](OC)CN1C(=O)CCc1ccccc1 ZINC000217601623 CD In-Stock Unstable FKBP1A 41 37 COC(=O)[C@H]1C[C@@H](OC)CN1C(=O)CCc1ccccc1 ZINC000217601623 CD In-Stock Unstable PREP 44 37 COC(=O)[C@H]1C[C@@H](OC)CN1C(=O)CCc1ccccc1 ZINC000217601623 CD In-Stock Unstable CES1 43 31 COC(=O)[C@H]1C[C@@H](OC)CN1C(=O)CCc1ccccc1 ZINC000217601623 CD In-Stock Unstable ACHP_LYMST 17 40 COC(=O)[C@H]1C[C@@H](OC)CN1C(=O)CCc1ccccc1 ZINC000217601623 CD In-Stock Unstable Q8WSF8_APLCA 25 40 Cc1c(N)nc(C2CC2)nc1N1CCN(C)[C@@H](C)C1 ZINC000217601657 CD For-Sale Unstable CHRM3 0 48 O=C(c1cccc(CN2CCCCCC2)c1)N1CCN2CCC[C@@H]2C1 ZINC000217601674 EF In-Stock Unstable PREP 22 40 O=C(c1cccc(CN2CCCCCC2)c1)N1CCN2CCC[C@@H]2C1 ZINC000217601674 EF In-Stock Unstable PARP1 15 42 O=C(c1cccc(CN2CCCCCC2)c1)N1CCN2CCC[C@@H]2C1 ZINC000217601674 EF In-Stock Unstable MGLL 0 48 O=C(c1cccc(CN2CCCCCC2)c1)N1CCN2CCC[C@@H]2C1 ZINC000217601674 EF In-Stock Unstable L3MBTL1 0 52 O=C(c1cccc(CN2CCCCCC2)c1)N1CCN2CCC[C@@H]2C1 ZINC000217601674 EF In-Stock Unstable L3MBTL3 94 52 O=C(c1cccc(CN2CCCCCC2)c1)N1CCN2CCC[C@@H]2C1 ZINC000217601674 EF In-Stock Unstable MBTD1 0 50 O=C(c1cccc(CN2CCCCCC2)c1)N1CCN2CCC[C@@H]2C1 ZINC000217601674 EF In-Stock Unstable TP53BP1 0 42 O=C(O)/C=C\c1cccc(NC(=O)NC2CCCCC2)n1 ZINC000217601684 CF For-Sale Unstable EPHX2 22 50 COC(=O)[C@H]1C[C@H](OC)CN1C(=O)CCc1ccccc1 ZINC000217601703 CD In-Stock Unstable ACE 47 40 COC(=O)[C@H]1C[C@H](OC)CN1C(=O)CCc1ccccc1 ZINC000217601703 CD In-Stock Unstable FKBP1A 41 37 COC(=O)[C@H]1C[C@H](OC)CN1C(=O)CCc1ccccc1 ZINC000217601703 CD In-Stock Unstable PREP 44 37 COC(=O)[C@H]1C[C@H](OC)CN1C(=O)CCc1ccccc1 ZINC000217601703 CD In-Stock Unstable CES1 43 31 COC(=O)[C@H]1C[C@H](OC)CN1C(=O)CCc1ccccc1 ZINC000217601703 CD In-Stock Unstable ACHP_LYMST 17 40 COC(=O)[C@H]1C[C@H](OC)CN1C(=O)CCc1ccccc1 ZINC000217601703 CD In-Stock Unstable Q8WSF8_APLCA 25 40 COCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217601750 HE In-Stock Unstable CA2 16 44 COCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217601750 HE In-Stock Unstable TBXA2R 38 42 COCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217601750 HE In-Stock Unstable TBXAS1 22 42 COCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217601750 HE In-Stock Unstable BMP1 58 35 COCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217601750 HE In-Stock Unstable CA1 17 44 COCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217601750 HE In-Stock Unstable MMP13 46 38 COCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217601750 HE In-Stock Unstable PTGDR 20 41 COCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217601750 HE In-Stock Unstable IAP 0 48 COCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217601750 HE In-Stock Unstable CA9 23 44 COCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217601750 HE In-Stock Unstable MMP1 40 36 COCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217601750 HE In-Stock Unstable AKR1C3 27 45 COCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217601750 HE In-Stock Unstable AKR1C2 46 36 O=C(c1cccc(CN2CCCCCC2)c1)N1CCN2CCC[C@H]2C1 ZINC000217601757 EF In-Stock Unstable PREP 22 40 O=C(c1cccc(CN2CCCCCC2)c1)N1CCN2CCC[C@H]2C1 ZINC000217601757 EF In-Stock Unstable PARP1 15 42 O=C(c1cccc(CN2CCCCCC2)c1)N1CCN2CCC[C@H]2C1 ZINC000217601757 EF In-Stock Unstable MGLL 0 48 O=C(c1cccc(CN2CCCCCC2)c1)N1CCN2CCC[C@H]2C1 ZINC000217601757 EF In-Stock Unstable L3MBTL1 0 52 O=C(c1cccc(CN2CCCCCC2)c1)N1CCN2CCC[C@H]2C1 ZINC000217601757 EF In-Stock Unstable L3MBTL3 94 52 O=C(c1cccc(CN2CCCCCC2)c1)N1CCN2CCC[C@H]2C1 ZINC000217601757 EF In-Stock Unstable MBTD1 0 50 O=C(c1cccc(CN2CCCCCC2)c1)N1CCN2CCC[C@H]2C1 ZINC000217601757 EF In-Stock Unstable TP53BP1 0 42 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable ACE 20 48 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable TYR 15 42 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable SSTR2 80 51 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable GNRHR 23 44 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable OPRM1 21 54 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable OPRD1 22 54 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable GHRHR 33 44 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable MME 29 46 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable EDNRB 56 41 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable EDNRA 65 66 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable TACR1 59 65 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable PGC 50 36 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable MC4R 63 44 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable BMP1 38 49 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable TACR2 25 57 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable CTSB 25 56 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable PAPA1_CARPA 65 48 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable CCKAR 166 57 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable CTSK 19 40 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable CTSL 42 57 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable PGA 35 56 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable BRS3 49 49 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable TIMP3 17 45 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable TACR3 18 41 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable NMBR 55 60 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable MC3R 78 42 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable MC5R 77 42 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable MMP2 31 47 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable MMP8 70 49 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable GRIA1 30 42 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable MMP14 105 44 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable GRPR 95 45 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable ECE1 80 49 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable HLA-DRB1 49 42 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable REN 70 56 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable REN1 37 56 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable LNPEP 19 40 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable SSTR3 23 54 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable MMP11 106 41 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable CCKBR 127 61 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable CTSS 18 73 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable GHSR 74 52 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable CAPN1 23 49 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable MMP9 30 47 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable CAPN2 38 42 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable MC1R 110 46 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable ADAM9 42 44 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable AKT1 42 35 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable MMP7 32 47 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable MMP1 26 47 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable FPR1 57 62 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable NPR 34 46 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable KISS1R 87 41 CCOC(=O)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C ZINC000217601770 GE On-Demand Unstable ERAP2 45 40 COC(=O)[C@@H]1C[C@@H](OC)CN1C(=O)CCc1ccccc1 ZINC000217601776 CD In-Stock Unstable ACE 47 40 COC(=O)[C@@H]1C[C@@H](OC)CN1C(=O)CCc1ccccc1 ZINC000217601776 CD In-Stock Unstable FKBP1A 41 37 COC(=O)[C@@H]1C[C@@H](OC)CN1C(=O)CCc1ccccc1 ZINC000217601776 CD In-Stock Unstable PREP 44 37 COC(=O)[C@@H]1C[C@@H](OC)CN1C(=O)CCc1ccccc1 ZINC000217601776 CD In-Stock Unstable CES1 43 31 COC(=O)[C@@H]1C[C@@H](OC)CN1C(=O)CCc1ccccc1 ZINC000217601776 CD In-Stock Unstable ACHP_LYMST 17 40 COC(=O)[C@@H]1C[C@@H](OC)CN1C(=O)CCc1ccccc1 ZINC000217601776 CD In-Stock Unstable Q8WSF8_APLCA 25 40 Cc1cc(NC(=O)c2ccc(C(C)(C)C)c([N+](=O)[O-])c2)ccn1 ZINC000217601796 DH On-Demand Unstable TYK2 51 33 Cc1cc(NC(=O)c2ccc(C(C)(C)C)c([N+](=O)[O-])c2)ccn1 ZINC000217601796 DH On-Demand Unstable TAAR1 39 43 Cc1cc(NC(=O)c2ccc(C(C)(C)C)c([N+](=O)[O-])c2)ccn1 ZINC000217601796 DH On-Demand Unstable KCNK3 47 39 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1ccccn1 ZINC000217601817 IG In-Stock Unstable TGFBR2 48 40 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1ccccn1 ZINC000217601817 IG In-Stock Unstable HISG 0 43 O=C(NCC1CCCCC1)Nc1ccc2cn[nH]c2c1 ZINC000217601822 CG For-Sale Unstable CCR3 19 46 O=C(NCC1CCCCC1)Nc1ccc2cn[nH]c2c1 ZINC000217601822 CG For-Sale Unstable ROCK2 22 58 O=C(NCC1CCCCC1)Nc1ccc2cn[nH]c2c1 ZINC000217601822 CG For-Sale Unstable PRMT3 36 42 O=C(NCC1CCCCC1)Nc1ccc2cn[nH]c2c1 ZINC000217601822 CG For-Sale Unstable PHLPP2 0 50 COC(=O)C[C@H](c1cc(OC)c2c(c1)OCCO2)c1c(O)c2ccccc2oc1=O ZINC000217601843 HF In-Stock Unstable NQO1 48 45 O=C1O[C@@]2(CCCN(C(=O)CSc3ncccn3)C2)c2ccccc21 ZINC000217601851 FE For-Sale Unstable NPY5R 48 42 COCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217601859 JE In-Stock Unstable BDKRB1 0 41 COCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217601859 JE In-Stock Unstable IAP 0 49 COCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217601859 JE In-Stock Unstable SCMU_MYCTU 0 44 COC(=O)[C@@H]1C[C@H](OC)CN1C(=O)CCc1ccccc1 ZINC000217601860 CD In-Stock Unstable ACE 47 40 COC(=O)[C@@H]1C[C@H](OC)CN1C(=O)CCc1ccccc1 ZINC000217601860 CD In-Stock Unstable FKBP1A 41 37 COC(=O)[C@@H]1C[C@H](OC)CN1C(=O)CCc1ccccc1 ZINC000217601860 CD In-Stock Unstable PREP 44 37 COC(=O)[C@@H]1C[C@H](OC)CN1C(=O)CCc1ccccc1 ZINC000217601860 CD In-Stock Unstable CES1 43 31 COC(=O)[C@@H]1C[C@H](OC)CN1C(=O)CCc1ccccc1 ZINC000217601860 CD In-Stock Unstable ACHP_LYMST 17 40 COC(=O)[C@@H]1C[C@H](OC)CN1C(=O)CCc1ccccc1 ZINC000217601860 CD In-Stock Unstable Q8WSF8_APLCA 25 40 O=C(O)/C=C\c1cnc(NC(=O)Nc2cccc(Cl)c2)s1 ZINC000217601861 DH For-Sale Anodyne PPIA 19 41 O=C(O)/C=C\c1cnc(NC(=O)Nc2cccc(Cl)c2)s1 ZINC000217601861 DH For-Sale Anodyne KIT 18 42 O=C(O)/C=C\c1cnc(NC(=O)Nc2cccc(Cl)c2)s1 ZINC000217601861 DH For-Sale Anodyne KDR 19 42 O=C(O)/C=C\c1cnc(NC(=O)Nc2cccc(Cl)c2)s1 ZINC000217601861 DH For-Sale Anodyne TEK 24 42 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@H](c3cccs3)C2)[C@@H]1c1ccccn1 ZINC000217601901 IG In-Stock Unstable TGFBR2 48 40 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@H](c3cccs3)C2)[C@@H]1c1ccccn1 ZINC000217601901 IG In-Stock Unstable HISG 0 43 NS(=O)(=O)c1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217601905 ED On-Demand Unstable CA2 115 55 NS(=O)(=O)c1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217601905 ED On-Demand Unstable CA6 25 42 NS(=O)(=O)c1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217601905 ED On-Demand Unstable CA1 95 55 NS(=O)(=O)c1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217601905 ED On-Demand Unstable CA7 71 51 NS(=O)(=O)c1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217601905 ED On-Demand Unstable CA13 26 41 NS(=O)(=O)c1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217601905 ED On-Demand Unstable CA5B 57 51 NS(=O)(=O)c1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217601905 ED On-Demand Unstable CA4 80 55 NS(=O)(=O)c1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217601905 ED On-Demand Unstable CA5A 55 51 NS(=O)(=O)c1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217601905 ED On-Demand Unstable CA14 62 44 NS(=O)(=O)c1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217601905 ED On-Demand Unstable MMP2 68 48 NS(=O)(=O)c1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217601905 ED On-Demand Unstable MMP3 16 48 NS(=O)(=O)c1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217601905 ED On-Demand Unstable CA12 83 54 NS(=O)(=O)c1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217601905 ED On-Demand Unstable CA9 78 54 NS(=O)(=O)c1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217601905 ED On-Demand Unstable CAH_METTE 24 41 NS(=O)(=O)c1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217601905 ED On-Demand Unstable CYNT 32 48 NS(=O)(=O)c1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217601905 ED On-Demand Unstable NCE103 41 52 NS(=O)(=O)c1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217601905 ED On-Demand Unstable ALPI 17 51 NS(=O)(=O)c1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217601905 ED On-Demand Unstable LIG1 0 45 NS(=O)(=O)c1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217601905 ED On-Demand Unstable CA15 15 42 NS(=O)(=O)c1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217601905 ED On-Demand Unstable MTCA1 38 43 NS(=O)(=O)c1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217601905 ED On-Demand Unstable P96878_MYCTU 51 46 NS(=O)(=O)c1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217601905 ED On-Demand Unstable CA 0 43 NS(=O)(=O)c1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217601905 ED On-Demand Unstable A6YCJ1_9METZ 28 54 NS(=O)(=O)c1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217601905 ED On-Demand Unstable Q5TU56_ANOGA 0 42 COC(=O)C[C@@H](c1cc(OC)c2c(c1)OCCO2)c1c(O)c2ccccc2oc1=O ZINC000217601922 HF In-Stock Unstable NQO1 48 45 O=C1O[C@]2(CCCN(C(=O)CSc3ncccn3)C2)c2ccccc21 ZINC000217601932 FE For-Sale Unstable NPY5R 48 42 O=C(O)/C=C\c1cnc(NC(=O)NC2CCCCC2)s1 ZINC000217601939 CF For-Sale Unstable EPHX2 17 45 O=C(O)/C=C\c1cnc(NC(=O)NC2CCCCC2)s1 ZINC000217601939 CF For-Sale Unstable CDK5 46 39 COC(=O)[C@H]1C[C@@H](OC)CN1C(=O)c1cccc(OC)c1 ZINC000217601951 CD In-Stock Unstable DRD4 46 35 COC(=O)[C@H]1C[C@@H](OC)CN1C(=O)c1cccc(OC)c1 ZINC000217601951 CD In-Stock Unstable CFTR 42 41 COC(=O)[C@H]1C[C@@H](OC)CN1C(=O)c1cccc(OC)c1 ZINC000217601951 CD In-Stock Unstable BRPF1 0 40 COCCCNS(=O)(=O)c1ccc(NCc2ccco2)c(C(=O)O)c1 ZINC000217601971 FD In-Stock Unstable BDKRB1 0 42 COc1ccc(NC(=O)[C@@H]2CC[C@@H](CNC(=O)[C@@H]3Cc4ccccc4CN3)CC2)cc1 ZINC000217601988 HG In-Stock Unstable HDAC8 0 44 COc1ccc(NC(=O)[C@@H]2CC[C@@H](CNC(=O)[C@@H]3Cc4ccccc4CN3)CC2)cc1 ZINC000217601988 HG In-Stock Unstable MTNR1A 32 47 COc1ccc(NC(=O)[C@@H]2CC[C@@H](CNC(=O)[C@@H]3Cc4ccccc4CN3)CC2)cc1 ZINC000217601988 HG In-Stock Unstable MTNR1B 32 47 COc1ccc(NC(=O)[C@@H]2CC[C@@H](CNC(=O)[C@@H]3Cc4ccccc4CN3)CC2)cc1 ZINC000217601988 HG In-Stock Unstable ROCK2 18 48 COc1ccc(NC(=O)[C@@H]2CC[C@@H](CNC(=O)[C@@H]3Cc4ccccc4CN3)CC2)cc1 ZINC000217601988 HG In-Stock Unstable NPY5R 15 42 COc1ccc(NC(=O)[C@@H]2CC[C@@H](CNC(=O)[C@@H]3Cc4ccccc4CN3)CC2)cc1 ZINC000217601988 HG In-Stock Unstable PFKFB3 42 32 C[C@H]1CN(C)[C@@H](C)C[C@@H]1Nc1ccc2[nH]ncc2c1 ZINC000217601994 CF For-Sale Unstable ROCK2 32 40 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1cccs1 ZINC000217602005 IH In-Stock Unstable CACNA1C 42 36 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1cccs1 ZINC000217602005 IH In-Stock Unstable CACNA1D 43 36 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1cccs1 ZINC000217602005 IH In-Stock Unstable TGFBR2 53 44 O=C(NCC1CCCCC1)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217602028 FK For-Sale Unstable CCR3 16 42 O=C(NCC1CCCCC1)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217602028 FK For-Sale Unstable EPHX2 30 55 O=C(NCC1CCCCC1)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217602028 FK For-Sale Unstable CACNA1I 34 45 O=C(NCC1CCCCC1)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217602028 FK For-Sale Unstable PTPA 0 43 O=C(NCC1CCCCC1)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217602028 FK For-Sale Unstable PRMT3 25 40 COC(=O)[C@H]1C[C@H](OC)CN1C(=O)c1cccc(OC)c1 ZINC000217602040 CD In-Stock Unstable DRD4 46 35 COC(=O)[C@H]1C[C@H](OC)CN1C(=O)c1cccc(OC)c1 ZINC000217602040 CD In-Stock Unstable CFTR 42 41 COC(=O)[C@H]1C[C@H](OC)CN1C(=O)c1cccc(OC)c1 ZINC000217602040 CD In-Stock Unstable BRPF1 0 40 Cc1nc(-n2cccc2)sc1C(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217602049 GH For-Sale Unstable NPY5R 25 41 C[C@@H](C1CC1)N(C)C[C@@H](O)c1ccc2c(c1)OCCO2 ZINC000217602050 CE For-Sale Unstable AOC3 15 62 COCCCNS(=O)(=O)c1ccc(NC[C@@H]2CCCO2)c(C(=O)O)c1 ZINC000217602081 FD In-Stock Unstable BDKRB1 0 40 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@H](c3cccs3)C2)[C@@H]1c1cccs1 ZINC000217602097 IH In-Stock Unstable CACNA1C 42 36 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@H](c3cccs3)C2)[C@@H]1c1cccs1 ZINC000217602097 IH In-Stock Unstable CACNA1D 43 36 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@H](c3cccs3)C2)[C@@H]1c1cccs1 ZINC000217602097 IH In-Stock Unstable TGFBR2 53 44 COC(=O)[C@@H]1C[C@@H](OC)CN1C(=O)c1cccc(OC)c1 ZINC000217602108 CD In-Stock Unstable DRD4 46 35 COC(=O)[C@@H]1C[C@@H](OC)CN1C(=O)c1cccc(OC)c1 ZINC000217602108 CD In-Stock Unstable CFTR 42 41 COC(=O)[C@@H]1C[C@@H](OC)CN1C(=O)c1cccc(OC)c1 ZINC000217602108 CD In-Stock Unstable BRPF1 0 40 Cc1nc(-n2cccc2)sc1C(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217602120 GH For-Sale Unstable NPY5R 25 41 C[C@H](C1CC1)N(C)C[C@@H](O)c1ccc2c(c1)OCCO2 ZINC000217602123 CE For-Sale Unstable AOC3 15 62 Cc1cc(NC(=O)NC(C)(C)C)ccc1/C=C\C(=O)O ZINC000217602133 CG For-Sale Unstable IMDH_CRYPV 60 37 CCc1ccccc1NC(=O)NCC1CCCCC1 ZINC000217602141 CH On-Demand Unstable KCNQ2 49 32 CCc1ccccc1NC(=O)NCC1CCCCC1 ZINC000217602141 CH On-Demand Unstable NMBR 21 40 CCc1ccccc1NC(=O)NCC1CCCCC1 ZINC000217602141 CH On-Demand Unstable AMY2 43 31 CCc1ccccc1NC(=O)NCC1CCCCC1 ZINC000217602141 CH On-Demand Unstable ACAT 0 42 CCCN(C(=O)c1ccc(=O)n(Cc2ccccc2Cl)c1)[C@@H]1CCS(=O)(=O)C1 ZINC000217602152 HF On-Demand Unstable MBTPS1 62 38 COCCCNS(=O)(=O)c1ccc(NC[C@H]2CCCO2)c(C(=O)O)c1 ZINC000217602160 FD In-Stock Unstable BDKRB1 0 40 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@H](c3cccs3)C2)[C@@H]1c1ccsc1 ZINC000217602183 IH In-Stock Unstable CACNA1D 52 38 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@H](c3cccs3)C2)[C@@H]1c1ccsc1 ZINC000217602183 IH In-Stock Unstable TGFBR2 52 42 COC(=O)[C@@H]1C[C@H](OC)CN1C(=O)c1cccc(OC)c1 ZINC000217602187 CD In-Stock Unstable DRD4 46 35 COC(=O)[C@@H]1C[C@H](OC)CN1C(=O)c1cccc(OC)c1 ZINC000217602187 CD In-Stock Unstable CFTR 42 41 COC(=O)[C@@H]1C[C@H](OC)CN1C(=O)c1cccc(OC)c1 ZINC000217602187 CD In-Stock Unstable BRPF1 0 40 CCCCNC(=O)Nc1ccc(/C=C\C(=O)O)c(C)c1 ZINC000217602228 CG For-Sale Unstable PRMT3 44 32 CCCCNC(=O)Nc1ccc(/C=C\C(=O)O)c(C)c1 ZINC000217602228 CG For-Sale Unstable ACAT 0 43 COc1cc(-c2cc(C(=O)N3CCC[C@]4(C3)OC(=O)c3ccccc34)[nH]n2)cc(OC)c1OC ZINC000217602230 JG For-Sale Unstable TACR3 23 44 COc1cc(-c2cc(C(=O)N3CCC[C@]4(C3)OC(=O)c3ccccc34)[nH]n2)cc(OC)c1OC ZINC000217602230 JG For-Sale Unstable NPY5R 30 47 CCCN(C(=O)c1ccc(=O)n(Cc2ccccc2Cl)c1)[C@H]1CCS(=O)(=O)C1 ZINC000217602238 HF On-Demand Unstable MBTPS1 62 38 COCCCNS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217602261 ED In-Stock Unstable HTR7 22 40 COCCCNS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217602261 ED In-Stock Unstable HTR6 0 42 COc1cc([C@H](C)N)c(F)cc1Br ZINC000217602263 BF For-Sale Unstable P2RX2 15 40 COC(=O)[C@H]1C[C@@H](OC)CN1C(=O)COc1ccc(F)cc1 ZINC000217602297 DC In-Stock Unstable COLA 40 36 COc1cc(-c2cc(C(=O)N3CCC[C@@]4(C3)OC(=O)c3ccccc34)[nH]n2)cc(OC)c1OC ZINC000217602302 JG For-Sale Unstable TACR3 23 44 COc1cc(-c2cc(C(=O)N3CCC[C@@]4(C3)OC(=O)c3ccccc34)[nH]n2)cc(OC)c1OC ZINC000217602302 JG For-Sale Unstable NPY5R 30 47 C[C@@H]1CN(C[C@@H](O)c2ccc(C(C)(C)C)cc2)CCCO1 ZINC000217602307 CG For-Sale Unstable LOC100281352 0 42 C[C@@H]1CN(C[C@@H](O)c2ccc(C(C)(C)C)cc2)CCCO1 ZINC000217602307 CG For-Sale Unstable ZM.86993 0 42 C[C@@H]1CN(C[C@@H](O)c2ccc(C(C)(C)C)cc2)CCCO1 ZINC000217602307 CG For-Sale Unstable Q2TU57_MAIZE 21 42 CCN(CC)S(=O)(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217602308 DD For-Sale Unstable PTGER2 23 41 CCN(CC)S(=O)(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217602308 DD For-Sale Unstable AKR1C3 32 40 C[C@@H](N(C)C[C@@H](O)c1ccc2c(c1)OCCO2)C(C)(C)C ZINC000217602325 CF For-Sale Unstable AOC3 17 68 COc1cc([C@@H](C)N)c(F)cc1Br ZINC000217602336 BF For-Sale Unstable P2RX2 15 40 COCCCNS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217602358 FD In-Stock Unstable HTR6 0 42 O=C(NCC1CCCCC1)Nc1ccc(F)c(Cl)c1 ZINC000217602374 CI For-Sale Unstable DPEP1 16 43 O=C(NCC1CCCCC1)Nc1ccc(F)c(Cl)c1 ZINC000217602374 CI For-Sale Unstable CCR3 45 39 O=C(NCC1CCCCC1)Nc1ccc(F)c(Cl)c1 ZINC000217602374 CI For-Sale Unstable EPHX2 43 69 O=C(NCC1CCCCC1)Nc1ccc(F)c(Cl)c1 ZINC000217602374 CI For-Sale Unstable ERBB4 52 34 O=C(NCC1CCCCC1)Nc1ccc(F)c(Cl)c1 ZINC000217602374 CI For-Sale Unstable ENV 44 34 O=C(NCC1CCCCC1)Nc1ccc(F)c(Cl)c1 ZINC000217602374 CI For-Sale Unstable MCHR1 35 48 O=C(NCC1CCCCC1)Nc1ccc(F)c(Cl)c1 ZINC000217602374 CI For-Sale Unstable CACNA1I 58 34 O=C(NCC1CCCCC1)Nc1ccc(F)c(Cl)c1 ZINC000217602374 CI For-Sale Unstable PRMT3 43 42 O=C(NCC1CCCCC1)Nc1ccc(F)c(Cl)c1 ZINC000217602374 CI For-Sale Unstable P95276_MYCTO 0 44 COC(=O)[C@H]1C[C@H](OC)CN1C(=O)COc1ccc(F)cc1 ZINC000217602379 DC In-Stock Unstable COLA 40 36 C[C@H]1CN(C[C@@H](O)c2ccc(C(C)(C)C)cc2)CCCO1 ZINC000217602380 CG For-Sale Unstable LOC100281352 0 42 C[C@H]1CN(C[C@@H](O)c2ccc(C(C)(C)C)cc2)CCCO1 ZINC000217602380 CG For-Sale Unstable ZM.86993 0 42 C[C@H]1CN(C[C@@H](O)c2ccc(C(C)(C)C)cc2)CCCO1 ZINC000217602380 CG For-Sale Unstable Q2TU57_MAIZE 21 42 O=C(O)/C=C\c1cccc(CNS(=O)(=O)N2CCCC2)c1 ZINC000217602393 DD For-Sale Unstable HDAC8 40 36 O=C1O[C@@]2(CCCN(C(=O)c3cc(-c4ccco4)[nH]n3)C2)c2ccccc21 ZINC000217602413 FF For-Sale Unstable NPY5R 29 42 C[C@H](N(C)C[C@@H](O)c1ccc2c(c1)OCCO2)C(C)(C)C ZINC000217602414 CF For-Sale Unstable AOC3 17 68 COC(=O)[C@@H]1C[C@@H](OC)CN1C(=O)COc1ccc(F)cc1 ZINC000217602462 DC In-Stock Unstable COLA 40 36 COCCCNS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1 ZINC000217602472 FC In-Stock Unstable BDKRB1 0 42 CCN(CC)c1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217602480 DI For-Sale Unstable GHSR 0 45 CCN(CC)c1ccc(NC(=O)NCC2CCCCC2)cc1 ZINC000217602480 DI For-Sale Unstable EPHX2 30 66 O=C(O)/C=C\c1cnc(NC(=O)Nc2ccccc2F)s1 ZINC000217602484 DG For-Sale Anodyne CDK5 42 41 CC(C)C[C@@H](C)N(C)C[C@@H](O)c1ccc2c(c1)OCCO2 ZINC000217602493 CF For-Sale Unstable AOC3 16 63 O=C1O[C@]2(CCCN(C(=O)c3cc(-c4ccco4)[nH]n3)C2)c2ccccc21 ZINC000217602494 FF For-Sale Unstable NPY5R 29 42 CNS(=O)(=O)c1ccc(C)c(C(=O)Nc2nc(-c3cccc(Br)c3)cs2)c1 ZINC000217602505 JI On-Demand Unstable MPL 24 47 COC(=O)[C@@H]1C[C@H](OC)CN1C(=O)COc1ccc(F)cc1 ZINC000217602557 DC In-Stock Unstable COLA 40 36 CC(C)C[C@H](C)N(C)C[C@@H](O)c1ccc2c(c1)OCCO2 ZINC000217602579 CF For-Sale Unstable AOC3 16 63 O=C1O[C@@]2(CCCN(C(=O)c3cccc(-n4cnnn4)c3)C2)c2ccccc21 ZINC000217602600 GD For-Sale Unstable NPY5R 29 42 CCOCCCNc1ccc(S(=O)(=O)NCCCOC)cc1C(=O)O ZINC000217602601 FD In-Stock Unstable CASP3 23 42 CCOCCCNc1ccc(S(=O)(=O)NCCCOC)cc1C(=O)O ZINC000217602601 FD In-Stock Unstable BDKRB1 0 44 Cc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)Nc1nc(-c2cccc(Br)c2)cs1 ZINC000217602612 JJ On-Demand Unstable MPL 20 44 Cc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)Nc1nc(-c2cccc(Br)c2)cs1 ZINC000217602612 JJ On-Demand Unstable CCR8 50 32 Cc1cccc(NC(=O)Nc2ncc(/C=C\C(=O)O)s2)c1 ZINC000217602664 DG For-Sale Unstable KIT 33 44 Cc1cccc(NC(=O)Nc2ncc(/C=C\C(=O)O)s2)c1 ZINC000217602664 DG For-Sale Unstable CCKAR 24 43 Cc1cccc(NC(=O)Nc2ncc(/C=C\C(=O)O)s2)c1 ZINC000217602664 DG For-Sale Unstable KDR 31 45 Cc1cccc(NC(=O)Nc2ncc(/C=C\C(=O)O)s2)c1 ZINC000217602664 DG For-Sale Unstable FBP1 24 40 Cc1cccc(NC(=O)Nc2ncc(/C=C\C(=O)O)s2)c1 ZINC000217602664 DG For-Sale Unstable TEK 31 44 Cc1cccc(NC(=O)Nc2ncc(/C=C\C(=O)O)s2)c1 ZINC000217602664 DG For-Sale Unstable CDK5 40 38 Cc1cccc(NC(=O)Nc2ncc(/C=C\C(=O)O)s2)c1 ZINC000217602664 DG For-Sale Unstable RIPK1 16 43 Cc1cccc(NC(=O)Nc2ncc(/C=C\C(=O)O)s2)c1 ZINC000217602664 DG For-Sale Unstable KCNK3 62 38 Cc1cccc(NC(=O)Nc2ncc(/C=C\C(=O)O)s2)c1 ZINC000217602664 DG For-Sale Unstable KCNK9 48 38 COC(=O)[C@H]1C[C@@H](OC)CN1C(=O)c1ccc(F)cc1Cl ZINC000217602669 DD In-Stock Unstable P2RX7 23 41 O=C1O[C@]2(CCCN(C(=O)c3cccc(-n4cnnn4)c3)C2)c2ccccc21 ZINC000217602694 GD For-Sale Unstable NPY5R 29 42 COCCCNS(=O)(=O)c1ccc(NCCCOC(C)C)c(C(=O)O)c1 ZINC000217602708 GD In-Stock Unstable CASP3 17 41 COCCCNS(=O)(=O)c1ccc(NCCCOC(C)C)c(C(=O)O)c1 ZINC000217602708 GD In-Stock Unstable BDKRB1 0 44 Cc1cc(/C=C\C(=O)O)ccc1NC(=O)OCC(C)C ZINC000217602732 CG For-Sale Unstable AKR1C3 28 43 C[C@H]1CCC[C@H](C)C1N[C@H](C)Cn1ccnc1 ZINC000217602735 BF For-Sale Unstable CAMC 0 41 COC(=O)[C@H]1C[C@H](OC)CN1C(=O)c1ccc(F)cc1Cl ZINC000217602742 DD In-Stock Unstable P2RX7 23 41 CNS(=O)(=O)c1ccc(C)c(C(=O)Nc2nc(-c3ccc(C)cc3C)cs2)c1 ZINC000217602748 HH On-Demand Unstable MPL 40 36 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1cnc2ccccc2c1 ZINC000217602793 CK For-Sale Unstable TRPM8 15 42 CC[C@@H](C)[C@@H](C(=O)N1CC[C@@H](CCl)C1)c1ccccc1 ZINC000217602800 CH For-Sale Unstable GRIN2B 23 43 CC[C@@H](C)[C@@H](C(=O)N1CC[C@@H](CCl)C1)c1ccccc1 ZINC000217602800 CH For-Sale Unstable CCR1 32 43 O=C1O[C@@]2(CCCN(C(=O)Cn3cnc4ccccc4c3=O)C2)c2ccccc21 ZINC000217602805 GE For-Sale Unstable NPY5R 28 42 O=CN1CCN(C(=O)NCC2CCCCC2)CC1 ZINC000217602822 CD For-Sale Unstable ADH4 0 41 CCCCCNc1ccc(S(=O)(=O)NCCCOC)cc1C(=O)O ZINC000217602826 FE In-Stock Unstable CASP3 0 44 C[C@H]1CCC[C@@H](C)C1N[C@H](C)Cn1ccnc1 ZINC000217602829 BF For-Sale Unstable CAMC 0 41 COc1ccc(/C=C\C(=O)O)cc1NC(=O)NC(C)C ZINC000217602830 CE For-Sale Unstable NR1H4 29 40 COc1ccc(/C=C\C(=O)O)cc1NC(=O)NC(C)C ZINC000217602830 CE For-Sale Unstable TUBB1 48 39 COc1ccc(/C=C\C(=O)O)cc1NC(=O)NC(C)C ZINC000217602830 CE For-Sale Unstable ABCG2 15 41 COC(=O)[C@@H]1C[C@@H](OC)CN1C(=O)c1ccc(F)cc1Cl ZINC000217602833 DD In-Stock Unstable P2RX7 23 41 NC/C=C\CN1CCN(C2CCCC2)CC1 ZINC000217602859 BD For-Sale Unstable EBP 15 48 Cc1ccc(-c2csc(NC(=O)c3cc(S(=O)(=O)NC4CC4)ccc3C)n2)c(C)c1 ZINC000217602864 II On-Demand Unstable CCR8 47 31 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1cnc2ccccc2c1 ZINC000217602873 CK For-Sale Unstable TRPM8 15 42 CC[C@H](C)[C@@H](C(=O)N1CC[C@@H](CCl)C1)c1ccccc1 ZINC000217602874 CH For-Sale Unstable GRIN2B 23 43 CC[C@H](C)[C@@H](C(=O)N1CC[C@@H](CCl)C1)c1ccccc1 ZINC000217602874 CH For-Sale Unstable CCR1 32 43 O=C1O[C@]2(CCCN(C(=O)Cn3cnc4ccccc4c3=O)C2)c2ccccc21 ZINC000217602896 GE For-Sale Unstable NPY5R 28 42 O=C(NCC1CCCCC1)NC1CCCCCC1 ZINC000217602911 CH On-Demand Unstable ADH1B 0 41 O=C(NCC1CCCCC1)NC1CCCCCC1 ZINC000217602911 CH On-Demand Unstable ADH1C 0 41 O=C(NCC1CCCCC1)NC1CCCCCC1 ZINC000217602911 CH On-Demand Unstable ADH4 0 41 O=C(NCC1CCCCC1)NC1CCCCCC1 ZINC000217602911 CH On-Demand Unstable EPHX2 31 56 O=C(NCC1CCCCC1)NC1CCCCCC1 ZINC000217602911 CH On-Demand Unstable P95276_MYCTO 0 43 COc1ccc(/C=C\C(=O)O)cc1NC(=O)OCC(C)C ZINC000217602915 CF For-Sale Unstable TUBB1 43 36 COc1ccc(/C=C\C(=O)O)cc1NC(=O)OCC(C)C ZINC000217602915 CF For-Sale Unstable AKR1C3 39 46 COC(=O)[C@@H]1C[C@H](OC)CN1C(=O)c1ccc(F)cc1Cl ZINC000217602926 DD In-Stock Unstable P2RX7 23 41 COCCCNS(=O)(=O)c1ccc(NCCC(C)C)c(C(=O)O)c1 ZINC000217602937 FE In-Stock Unstable CASP3 22 42 CC[C@@H](C)[C@H](C(=O)N1CC[C@@H](CCl)C1)c1ccccc1 ZINC000217602947 CH For-Sale Unstable GRIN2B 23 43 CC[C@@H](C)[C@H](C(=O)N1CC[C@@H](CCl)C1)c1ccccc1 ZINC000217602947 CH For-Sale Unstable CCR1 32 43 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1cnc2ccccc2c1 ZINC000217602958 CK For-Sale Unstable TRPM8 15 42 O=C1O[C@@]2(CCCN(C(=O)c3cc(-c4ccc5c(c4)OCO5)n[nH]3)C2)c2ccccc21 ZINC000217602999 HG For-Sale Unstable NPY5R 28 47 Cc1ccc(C)c(NC(=O)NCC2CCCCC2)c1 ZINC000217603016 CI On-Demand Unstable LDLR 0 47 Cc1ccc(C)c(NC(=O)NCC2CCCCC2)c1 ZINC000217603016 CI On-Demand Unstable EPHX2 15 42 Cc1ccc(C)c(NC(=O)NCC2CCCCC2)c1 ZINC000217603016 CI On-Demand Unstable ACAT 0 55 CC[C@H](C)[C@H](C(=O)N1CC[C@@H](CCl)C1)c1ccccc1 ZINC000217603026 CH For-Sale Unstable GRIN2B 23 43 CC[C@H](C)[C@H](C(=O)N1CC[C@@H](CCl)C1)c1ccccc1 ZINC000217603026 CH For-Sale Unstable CCR1 32 43 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1cnc2ccccc2c1 ZINC000217603032 CK For-Sale Unstable TRPM8 15 42 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NCCCOC)cc1C(=O)O ZINC000217603063 FE In-Stock Unstable CASP3 23 44 CC[C@H]1CCCN(C[C@@H](O)c2ccc3c(c2)OCCO3)C1 ZINC000217603065 CF For-Sale Unstable SSTR3 82 33 O=C1O[C@]2(CCCN(C(=O)c3cc(-c4ccc5c(c4)OCO5)n[nH]3)C2)c2ccccc21 ZINC000217603077 HG For-Sale Unstable NPY5R 28 47 Cc1ccc(-c2csc(NC(=O)c3cc(S(=O)(=O)NC4CC4)ccc3C)n2)s1 ZINC000217603081 II On-Demand Unstable CCR8 50 32 O=C(O)/C=C\c1cccc(CNS(=O)(=O)c2cccs2)c1 ZINC000217603086 DE For-Sale Unstable PTGER2 32 46 O=C(O)/C=C\c1cccc(CNS(=O)(=O)c2cccs2)c1 ZINC000217603086 DE For-Sale Unstable PTGER4 22 46 O=C(O)/C=C\c1cccc(CNS(=O)(=O)c2cccs2)c1 ZINC000217603086 DE For-Sale Unstable PTGER3 25 46 O=C(O)/C=C\c1cccc(CNS(=O)(=O)c2cccs2)c1 ZINC000217603086 DE For-Sale Unstable HCAR2 0 40 COc1ccc2c(c1OC)C(=O)O[C@@H]2CC(=O)Nc1ccc2c(C)cc(=O)oc2c1 ZINC000217603127 HG In-Stock Unstable MAOA 42 40 CCOc1ccccc1NC(=O)NCC1CCCCC1 ZINC000217603136 CH On-Demand Unstable DEF 0 43 CCOc1ccccc1NC(=O)NCC1CCCCC1 ZINC000217603136 CH On-Demand Unstable NMBR 21 40 CCOc1ccccc1NC(=O)NCC1CCCCC1 ZINC000217603136 CH On-Demand Unstable ACAT 0 45 CCOc1ccccc1NC(=O)NCC1CCCCC1 ZINC000217603136 CH On-Demand Unstable HCN1 49 38 CCOc1ccccc1NC(=O)NCC1CCCCC1 ZINC000217603136 CH On-Demand Unstable HCN4 50 40 CCC[C@H](C)Nc1ccc(S(=O)(=O)NCCCOC)cc1C(=O)O ZINC000217603137 FE In-Stock Unstable CASP3 23 44 CC(C)[C@@H](C)N(C)C[C@@H](O)c1ccc2c(c1)OCCO2 ZINC000217603155 CE For-Sale Unstable AOC3 17 71 CC(C)N(C)S(=O)(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217603171 DD For-Sale Unstable AKR1C3 33 40 COc1ccccc1-c1cc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)[nH]n1 ZINC000217603175 HG For-Sale Unstable TACR3 21 43 COc1ccccc1-c1cc(C(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)[nH]n1 ZINC000217603175 HG For-Sale Unstable NPY5R 31 48 COc1ccc2c(c1OC)C(=O)O[C@H]2CC(=O)Nc1ccc2c(C)cc(=O)oc2c1 ZINC000217603200 HG In-Stock Unstable MAOA 42 40 CC(C)[C@H](C)N(C)C[C@@H](O)c1ccc2c(c1)OCCO2 ZINC000217603216 CE For-Sale Unstable AOC3 17 71 Cc1cc(C)cc(NC(=O)NCC2CCCCC2)c1 ZINC000217603230 CI On-Demand Unstable CACNA1I 46 32 COCCCNS(=O)(=O)c1ccc(N[C@@H](C)COC)c(C(=O)O)c1 ZINC000217603238 FD In-Stock Unstable CASP3 16 40 COCCCNS(=O)(=O)c1ccc(N[C@@H](C)COC)c(C(=O)O)c1 ZINC000217603238 FD In-Stock Unstable BDKRB1 0 41 COc1ccccc1-c1cc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)[nH]n1 ZINC000217603251 HG For-Sale Unstable TACR3 21 43 COc1ccccc1-c1cc(C(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)[nH]n1 ZINC000217603251 HG For-Sale Unstable NPY5R 31 48 COC(=O)CS(=O)(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217603252 DC For-Sale Unstable AKR1C3 34 40 Cc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)Nc1nc(-c2cc3ccccc3o2)cs1 ZINC000217603305 JJ On-Demand Unstable CDC25C 0 45 Cc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)Nc1nc(-c2cc3ccccc3o2)cs1 ZINC000217603305 JJ On-Demand Unstable CCR8 58 33 CCC[C@@H](C)N(C)C[C@@H](O)c1ccc2c(c1)OCCO2 ZINC000217603312 CF For-Sale Unstable AOC3 17 63 COCCCNS(=O)(=O)c1ccc(N[C@H](C)COC)c(C(=O)O)c1 ZINC000217603321 FD In-Stock Unstable CASP3 16 40 COCCCNS(=O)(=O)c1ccc(N[C@H](C)COC)c(C(=O)O)c1 ZINC000217603321 FD In-Stock Unstable BDKRB1 0 41 O=C(O)/C=C\c1cnc(NC(=O)Nc2ccccc2Cl)s1 ZINC000217603337 DH For-Sale Anodyne EPHB3 59 39 COc1ccc(OCCNC(=O)NCC2CCCCC2)cc1 ZINC000217603338 DF On-Demand Unstable HRH2 24 43 COc1ccc(OCCNC(=O)NCC2CCCCC2)cc1 ZINC000217603338 DF On-Demand Unstable MTNR1B 36 43 O=C1O[C@@]2(CCCN(C(=O)Cn3nnc4ccccc43)C2)c2ccccc21 ZINC000217603369 FE For-Sale Unstable NPY5R 29 41 CCC[C@H](C)N(C)C[C@@H](O)c1ccc2c(c1)OCCO2 ZINC000217603388 CF For-Sale Unstable AOC3 17 63 CCCCS(=O)(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217603420 CE For-Sale Unstable HDAC8 40 36 CCCCS(=O)(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217603420 CE For-Sale Unstable HDAC1 18 41 CCCCS(=O)(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217603420 CE For-Sale Unstable AKR1C3 28 42 CCCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217603435 EF In-Stock Unstable CA2 20 42 CCCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217603435 EF In-Stock Unstable GNRHR 18 45 CCCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217603435 EF In-Stock Unstable CASP3 21 42 CCCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217603435 EF In-Stock Unstable CA4 15 42 CCCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217603435 EF In-Stock Unstable CASP6 18 42 CCCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217603435 EF In-Stock Unstable AKR1C3 15 43 O=C1O[C@]2(CCCN(C(=O)Cn3nnc4ccccc43)C2)c2ccccc21 ZINC000217603454 FE For-Sale Unstable NPY5R 29 41 O=C(CCCn1cnc2ccccc2c1=O)NO ZINC000217603515 BC In-Stock Unstable HTR7 26 54 O=C(CCCn1cnc2ccccc2c1=O)NO ZINC000217603515 BC In-Stock Unstable HDAC10 41 38 O=C(CCCn1cnc2ccccc2c1=O)NO ZINC000217603515 BC In-Stock Unstable HDAC1 34 48 O=C(CCCn1cnc2ccccc2c1=O)NO ZINC000217603515 BC In-Stock Unstable HDAC2 27 40 O=C(CCCn1cnc2ccccc2c1=O)NO ZINC000217603515 BC In-Stock Unstable HDAC3 42 38 O=C(CCCn1cnc2ccccc2c1=O)NO ZINC000217603515 BC In-Stock Unstable HDAC6 44 36 OCc1cc2n(n1)CCN(CCN1CCN(c3ccccc3)CC1)C2 ZINC000217603523 ED In-Stock Unstable HTR1A 35 43 OCc1cc2n(n1)CCN(CCN1CCN(c3ccccc3)CC1)C2 ZINC000217603523 ED In-Stock Unstable DRD2 23 44 OCc1cc2n(n1)CCN(CCN1CCN(c3ccccc3)CC1)C2 ZINC000217603523 ED In-Stock Unstable DRD4 20 40 OCc1cc2n(n1)CCN(CCN1CCN(c3ccccc3)CC1)C2 ZINC000217603523 ED In-Stock Unstable HTR2A 27 42 OCc1cc2n(n1)CCN(CCN1CCN(c3ccccc3)CC1)C2 ZINC000217603523 ED In-Stock Unstable HTR7 43 42 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)NCCN3CCOCC3)[C@H]21 ZINC000217603525 JD In-Stock Unstable DRD4 40 32 COC[C@@H](C)N(C)C[C@@H](O)c1ccc2c(c1)OCCO2 ZINC000217603529 CD For-Sale Unstable AOC3 15 62 COC[C@@H](C)N(C)C[C@@H](O)c1ccc2c(c1)OCCO2 ZINC000217603529 CD For-Sale Unstable PDE10A 23 40 CC(C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217603544 EF In-Stock Unstable CA2 18 43 CC(C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217603544 EF In-Stock Unstable GNRHR 17 44 CC(C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217603544 EF In-Stock Unstable CASP3 24 44 CC(C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217603544 EF In-Stock Unstable CA1 15 40 CC(C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217603544 EF In-Stock Unstable CA4 16 43 CC(C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217603544 EF In-Stock Unstable CASP6 19 44 CC(C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217603544 EF In-Stock Unstable ACPS 0 40 CC(C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217603544 EF In-Stock Unstable AKR1C3 17 41 COc1cccc(-c2cc(C(=O)N3CCC[C@]4(C3)OC(=O)c3ccccc34)n(C)n2)c1 ZINC000217603555 HG For-Sale Unstable NPY5R 29 51 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)NCCN3CCOCC3)[C@@H]21 ZINC000217603604 JD In-Stock Unstable DRD4 40 32 COC[C@H](C)N(C)C[C@@H](O)c1ccc2c(c1)OCCO2 ZINC000217603611 CD For-Sale Unstable AOC3 15 62 COC[C@H](C)N(C)C[C@@H](O)c1ccc2c(c1)OCCO2 ZINC000217603611 CD For-Sale Unstable PDE10A 23 40 CC[C@H](C(=O)NO)n1cnc2ccccc2c1=O ZINC000217603635 BC In-Stock Unstable CASP8 40 31 CCCCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217603640 FG In-Stock Unstable GNRHR 17 44 CCCCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217603640 FG In-Stock Unstable CASP3 21 40 CCCCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217603640 FG In-Stock Unstable CASP6 18 40 COc1cccc(-c2cc(C(=O)N3CCC[C@@]4(C3)OC(=O)c3ccccc34)n(C)n2)c1 ZINC000217603643 HG For-Sale Unstable NPY5R 29 51 O=C(NCC1CCCCC1)Nc1cccc2cccnc12 ZINC000217603668 CH On-Demand Unstable TRPV1 31 40 O=C(NCC1CCCCC1)Nc1cccc2cccnc12 ZINC000217603668 CH On-Demand Unstable WNT3 20 44 O=C(NCC1CCCCC1)Nc1cccc2cccnc12 ZINC000217603668 CH On-Demand Unstable TNKS 18 41 CCCC1=C(C(=O)OCC)[C@H](c2cc(OC)c(OC)c(OC)c2)C2=C(C[C@H](c3cccs3)[C@@H](C(=O)OCC)C2=O)N1 ZINC000217603691 KK In-Stock Unstable TGFBR2 22 41 COC(=O)[C@H]1C[C@@H](OC)CN1C(=O)Cc1ccc(NC(C)=O)cc1 ZINC000217603703 EC In-Stock Unstable TSHR 59 32 CC[C@@H](C(=O)NO)n1cnc2ccccc2c1=O ZINC000217603719 BC In-Stock Unstable CASP8 40 31 CC(C)CNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217603737 FF In-Stock Unstable CA2 17 41 CC(C)CNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217603737 FF In-Stock Unstable GNRHR 17 42 CC(C)CNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217603737 FF In-Stock Unstable CASP3 23 43 CC(C)CNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217603737 FF In-Stock Unstable BDKRB1 27 45 CC(C)CNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217603737 FF In-Stock Unstable CASP6 19 43 CC(C)CNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217603737 FF In-Stock Unstable MTNN 71 35 NC[C@@H]1CCCCN1CC(=O)N1CCC[C@@H]1c1cccs1 ZINC000217603769 DE For-Sale Unstable COLA 73 40 NC[C@@H]1CCCCN1CC(=O)N1CCC[C@@H]1c1cccs1 ZINC000217603769 DE For-Sale Unstable CPT1A 69 40 COC(=O)[C@H]1C[C@H](OC)CN1C(=O)Cc1ccc(NC(C)=O)cc1 ZINC000217603787 EC In-Stock Unstable TSHR 59 32 Cc1ccc2nc(-c3ccc(NC(=O)NCC4CCCCC4)cc3)sc2c1 ZINC000217603810 GK For-Sale Unstable PPARA 0 40 Cc1ccc2nc(-c3ccc(NC(=O)NCC4CCCCC4)cc3)sc2c1 ZINC000217603810 GK For-Sale Unstable LCK 24 40 Cc1ccc2nc(-c3ccc(NC(=O)NCC4CCCCC4)cc3)sc2c1 ZINC000217603810 GK For-Sale Unstable CSNK1D 27 41 Cc1ccc2nc(-c3ccc(NC(=O)NCC4CCCCC4)cc3)sc2c1 ZINC000217603810 GK For-Sale Unstable NMT1 30 40 Cc1ccc2nc(-c3ccc(NC(=O)NCC4CCCCC4)cc3)sc2c1 ZINC000217603810 GK For-Sale Unstable APP 26 53 Cc1ccc2nc(-c3ccc(NC(=O)NCC4CCCCC4)cc3)sc2c1 ZINC000217603810 GK For-Sale Unstable PRMT3 68 45 Cc1ccc2nc(-c3ccc(NC(=O)NCC4CCCCC4)cc3)sc2c1 ZINC000217603810 GK For-Sale Unstable ETHR 18 41 O=C(CCc1c[nH]c2ccccc12)NCCn1ccc2ccccc21 ZINC000217603821 EH In-Stock Unstable ACHE 32 49 O=C(CCc1c[nH]c2ccccc12)NCCn1ccc2ccccc21 ZINC000217603821 EH In-Stock Unstable MC4R 33 40 O=C(CCc1c[nH]c2ccccc12)NCCn1ccc2ccccc21 ZINC000217603821 EH In-Stock Unstable CTSL 0 40 O=C(CCc1c[nH]c2ccccc12)NCCn1ccc2ccccc21 ZINC000217603821 EH In-Stock Unstable BCHE 15 44 O=C(CCc1c[nH]c2ccccc12)NCCn1ccc2ccccc21 ZINC000217603821 EH In-Stock Unstable BRS3 22 40 O=C(CCc1c[nH]c2ccccc12)NCCn1ccc2ccccc21 ZINC000217603821 EH In-Stock Unstable MC5R 34 42 CC[C@@H](C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217603835 FG In-Stock Unstable CA2 18 41 CC[C@@H](C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217603835 FG In-Stock Unstable GNRHR 17 42 CC[C@@H](C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217603835 FG In-Stock Unstable CASP3 22 43 CC[C@@H](C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217603835 FG In-Stock Unstable CA4 15 41 CC[C@@H](C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217603835 FG In-Stock Unstable CASP6 19 43 O=C(NCc1ccc(-c2nc3ccccc3s2)o1)c1cc(N2CCOCC2)ccn1 ZINC000217603860 HH On-Demand Unstable CASR 25 41 COC(=O)[C@@H]1C[C@@H](OC)CN1C(=O)Cc1ccc(NC(C)=O)cc1 ZINC000217603868 EC In-Stock Unstable TSHR 59 32 O=C(NCC1CCCCC1)Nc1cccc(F)c1 ZINC000217603906 CH On-Demand Unstable CCR3 75 47 O=C(NCC1CCCCC1)Nc1cccc(F)c1 ZINC000217603906 CH On-Demand Unstable EPHX2 28 48 O=C(NCC1CCCCC1)Nc1cccc(F)c1 ZINC000217603906 CH On-Demand Unstable PRMT3 43 41 O=C(NCC1CCCCC1)Nc1cccc(F)c1 ZINC000217603906 CH On-Demand Unstable ACAT 0 40 O=C(NCC1CCCCC1)Nc1cccc(F)c1 ZINC000217603906 CH On-Demand Unstable KCNK3 16 40 O=C1O[C@@]2(CCCN(C(=O)c3ccoc3)C2)c2ccccc21 ZINC000217603917 CF In-Stock Unstable NPY5R 27 42 CC[C@H](C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217603927 FG In-Stock Unstable CA2 18 41 CC[C@H](C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217603927 FG In-Stock Unstable GNRHR 17 42 CC[C@H](C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217603927 FG In-Stock Unstable CASP3 22 43 CC[C@H](C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217603927 FG In-Stock Unstable CA4 15 41 CC[C@H](C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217603927 FG In-Stock Unstable CASP6 19 43 CC[C@@H](C)[C@@H](CO)NC(=O)Cn1c(=O)[nH]c2ccccc2c1=O ZINC000217603934 DC In-Stock Unstable ELANE 26 41 CC[C@@H](C)[C@@H](CO)NC(=O)Cn1c(=O)[nH]c2ccccc2c1=O ZINC000217603934 DC In-Stock Unstable NPEPPS 0 42 CC[C@@H](C)[C@@H](CO)NC(=O)Cn1c(=O)[nH]c2ccccc2c1=O ZINC000217603934 DC In-Stock Unstable PSMB5 16 40 CC[C@@H](C)[C@@H](CO)NC(=O)Cn1c(=O)[nH]c2ccccc2c1=O ZINC000217603934 DC In-Stock Unstable PSMB1 15 40 COC(=O)[C@@H]1C[C@H](OC)CN1C(=O)Cc1ccc(NC(C)=O)cc1 ZINC000217603942 EC In-Stock Unstable TSHR 59 32 O=C1O[C@]2(CCCN(C(=O)c3ccoc3)C2)c2ccccc21 ZINC000217604008 CF In-Stock Unstable NPY5R 27 42 O=C(NCCc1ccc(F)cc1)NCC1CCCCC1 ZINC000217604019 CG On-Demand Unstable CCR3 64 38 O=C(CCCn1nnc2ccccc2c1=O)NO ZINC000217604021 BC In-Stock Unstable HTR7 17 40 O=C(CCCn1nnc2ccccc2c1=O)NO ZINC000217604021 BC In-Stock Unstable HDAC10 53 38 O=C(CCCn1nnc2ccccc2c1=O)NO ZINC000217604021 BC In-Stock Unstable HDAC1 35 44 O=C(CCCn1nnc2ccccc2c1=O)NO ZINC000217604021 BC In-Stock Unstable HDAC2 29 40 O=C(CCCn1nnc2ccccc2c1=O)NO ZINC000217604021 BC In-Stock Unstable HDAC3 51 38 O=C(CCCn1nnc2ccccc2c1=O)NO ZINC000217604021 BC In-Stock Unstable HDAC6 60 38 CCCC1=C(C(=O)OCC)[C@H](c2ccc(N(C)C)cc2)C2=C(C[C@H](c3cccs3)[C@@H](C(=O)OCC)C2=O)N1 ZINC000217604028 KK In-Stock Unstable TGFBR2 32 45 CC(C)(C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217604050 FG In-Stock Unstable CA2 15 43 CC(C)(C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217604050 FG In-Stock Unstable GNRHR 18 48 CC(C)(C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217604050 FG In-Stock Unstable CASP3 21 42 CC(C)(C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217604050 FG In-Stock Unstable PRTN3 53 35 CC(C)(C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217604050 FG In-Stock Unstable CASP6 18 42 CC(C)(C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217604050 FG In-Stock Unstable AKR1C3 22 43 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)Nc3ccc4c(c3)OCO4)[C@H]21 ZINC000217604051 JG In-Stock Unstable TSHR 49 33 O=C1O[C@@]2(CCCN(C(=O)c3cccc(I)c3)C2)c2ccccc21 ZINC000217604122 IH For-Sale Unstable NPY5R 29 41 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)Nc3ccc4c(c3)OCO4)[C@@H]21 ZINC000217604125 JG In-Stock Unstable TSHR 49 33 O=C(NCC1CCCCC1)Nc1ccc(I)cc1 ZINC000217604141 FH For-Sale Unstable EPHX2 28 68 O=C(NCC1CCCCC1)Nc1ccc(I)cc1 ZINC000217604141 FH For-Sale Unstable NCE103 24 43 O=C(NCC1CCCCC1)Nc1ccc(I)cc1 ZINC000217604141 FH For-Sale Unstable PRMT3 38 44 C=CCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217604172 EE In-Stock Unstable CASP3 0 43 O=C1O[C@]2(CCCN(C(=O)c3cccc(I)c3)C2)c2ccccc21 ZINC000217604209 IH For-Sale Unstable NPY5R 29 41 O=C(Cc1ccc(F)cc1Cl)N1CCCn2nc([C@@H](O)CO)cc2C1 ZINC000217604220 FD In-Stock Unstable P2RX7 50 37 Cn1cccc1C(=O)Nc1ncc(Cc2ccc(Br)cc2)s1 ZINC000217604242 GI On-Demand Unstable CDK5 20 40 Cn1cccc1C(=O)Nc1ncc(Cc2ccc(Br)cc2)s1 ZINC000217604242 GI On-Demand Unstable SCD1 41 41 Cn1cccc1C(=O)Nc1ncc(Cc2ccc(Br)cc2)s1 ZINC000217604242 GI On-Demand Unstable SCD 35 41 O=C(NCCc1c[nH]c2ccccc12)NCC1CCCCC1 ZINC000217604261 CH On-Demand Unstable HTR1B 26 42 O=C(NCCc1c[nH]c2ccccc12)NCC1CCCCC1 ZINC000217604261 CH On-Demand Unstable SSTR2 38 43 O=C(NCCc1c[nH]c2ccccc12)NCC1CCCCC1 ZINC000217604261 CH On-Demand Unstable EDNRA 24 44 O=C(NCCc1c[nH]c2ccccc12)NCC1CCCCC1 ZINC000217604261 CH On-Demand Unstable TACR1 26 46 O=C(NCCc1c[nH]c2ccccc12)NCC1CCCCC1 ZINC000217604261 CH On-Demand Unstable CCKAR 63 49 O=C(NCCc1c[nH]c2ccccc12)NCC1CCCCC1 ZINC000217604261 CH On-Demand Unstable BCHE 15 42 O=C(NCCc1c[nH]c2ccccc12)NCC1CCCCC1 ZINC000217604261 CH On-Demand Unstable BRS3 23 42 O=C(NCCc1c[nH]c2ccccc12)NCC1CCCCC1 ZINC000217604261 CH On-Demand Unstable NMBR 71 35 O=C(NCCc1c[nH]c2ccccc12)NCC1CCCCC1 ZINC000217604261 CH On-Demand Unstable MC5R 37 46 O=C(NCCc1c[nH]c2ccccc12)NCC1CCCCC1 ZINC000217604261 CH On-Demand Unstable MTNR1A 18 50 O=C(NCCc1c[nH]c2ccccc12)NCC1CCCCC1 ZINC000217604261 CH On-Demand Unstable GRPR 43 33 O=C(NCCc1c[nH]c2ccccc12)NCC1CCCCC1 ZINC000217604261 CH On-Demand Unstable ECE1 41 37 O=C(NCCc1c[nH]c2ccccc12)NCC1CCCCC1 ZINC000217604261 CH On-Demand Unstable SSTR3 23 43 O=C(NCCc1c[nH]c2ccccc12)NCC1CCCCC1 ZINC000217604261 CH On-Demand Unstable CCKBR 54 49 O=C(NCCc1c[nH]c2ccccc12)NCC1CCCCC1 ZINC000217604261 CH On-Demand Unstable GHSR 46 35 O=C(NCCc1c[nH]c2ccccc12)NCC1CCCCC1 ZINC000217604261 CH On-Demand Unstable ALOX15 21 40 O=C(NCCc1c[nH]c2ccccc12)NCC1CCCCC1 ZINC000217604261 CH On-Demand Unstable SLC15A2 0 40 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NC1CC1 ZINC000217604271 EE In-Stock Unstable CASP3 18 42 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NC1CC1 ZINC000217604271 EE In-Stock Unstable NPY2R 27 41 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NC1CC1 ZINC000217604271 EE In-Stock Unstable CASP6 18 42 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NC1CC1 ZINC000217604271 EE In-Stock Unstable SFRP1 78 33 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NC1CC1 ZINC000217604271 EE In-Stock Unstable WNT3 50 32 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1ccccc1 ZINC000217604288 IH In-Stock Unstable CACNA1C 50 35 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1ccccc1 ZINC000217604288 IH In-Stock Unstable CACNA1D 65 37 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1ccccc1 ZINC000217604288 IH In-Stock Unstable TGFBR2 62 49 O=C(NCC(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12)OCc1ccccc1 ZINC000217604300 GF For-Sale Unstable GHRHR 44 33 O=C(NCC(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12)OCc1ccccc1 ZINC000217604300 GF For-Sale Unstable PREP 16 46 O=C(NCC(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12)OCc1ccccc1 ZINC000217604300 GF For-Sale Unstable NPY5R 24 40 O=C(NCC(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12)OCc1ccccc1 ZINC000217604300 GF For-Sale Unstable NPR 59 33 O=C(NCC(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12)OCc1ccccc1 ZINC000217604300 GF For-Sale Unstable SLC12A5 63 36 O=C(Cc1ccc(F)cc1Cl)N1CCCn2nc([C@H](O)CO)cc2C1 ZINC000217604312 FD In-Stock Unstable P2RX7 50 37 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NC1CCCC1 ZINC000217604371 FG In-Stock Unstable CASP3 16 40 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NC1CCCC1 ZINC000217604371 FG In-Stock Unstable CASP6 18 40 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NC1CCCC1 ZINC000217604371 FG In-Stock Unstable SFRP1 77 32 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NC1CCCC1 ZINC000217604371 FG In-Stock Unstable WNT3 62 33 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@H](c3cccs3)C2)[C@@H]1c1ccccc1 ZINC000217604382 IH In-Stock Unstable CACNA1C 50 35 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@H](c3cccs3)C2)[C@@H]1c1ccccc1 ZINC000217604382 IH In-Stock Unstable CACNA1D 65 37 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@H](c3cccs3)C2)[C@@H]1c1ccccc1 ZINC000217604382 IH In-Stock Unstable TGFBR2 62 49 O=C(NCC(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12)OCc1ccccc1 ZINC000217604385 GF For-Sale Unstable GHRHR 44 33 O=C(NCC(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12)OCc1ccccc1 ZINC000217604385 GF For-Sale Unstable PREP 16 46 O=C(NCC(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12)OCc1ccccc1 ZINC000217604385 GF For-Sale Unstable NPY5R 24 40 O=C(NCC(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12)OCc1ccccc1 ZINC000217604385 GF For-Sale Unstable NPR 59 33 O=C(NCC(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12)OCc1ccccc1 ZINC000217604385 GF For-Sale Unstable SLC12A5 63 36 COC(=O)[C@H]1C[C@@H](OC)CN1S(=O)(=O)c1cc(F)ccc1OC ZINC000217604396 EC In-Stock Unstable COLA 44 38 CCCC[C@H]1NC(=O)[C@H]1O ZINC000217604454 AC For-Sale Unstable GAA 20 42 CCCC[C@H]1NC(=O)[C@H]1O ZINC000217604454 AC For-Sale Unstable SI 19 42 CCCC[C@H]1NC(=O)[C@H]1O ZINC000217604454 AC For-Sale Unstable P0504H10.9 42 35 O=C(O)/C=C\c1cnc(NC(=O)Nc2cccc(F)c2)s1 ZINC000217604456 DG For-Sale Anodyne KIT 16 42 O=C(O)/C=C\c1cnc(NC(=O)Nc2cccc(F)c2)s1 ZINC000217604456 DG For-Sale Anodyne KDR 20 42 O=C(O)/C=C\c1cnc(NC(=O)Nc2cccc(F)c2)s1 ZINC000217604456 DG For-Sale Anodyne TEK 23 42 O=C(O)/C=C\c1cnc(NC(=O)Nc2cccc(F)c2)s1 ZINC000217604456 DG For-Sale Anodyne CDK5 40 40 COC(=O)[C@H]1C[C@H](OC)CN1S(=O)(=O)c1cc(F)ccc1OC ZINC000217604466 EC In-Stock Unstable COLA 44 38 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@H](c3cccs3)C2)[C@@H]1c1ccccc1C ZINC000217604468 JH In-Stock Unstable NR3C2 0 40 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@H](c3cccs3)C2)[C@@H]1c1ccccc1C ZINC000217604468 JH In-Stock Unstable TGFBR2 50 41 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@H](c3cccs3)C2)[C@@H]1c1ccccc1C ZINC000217604468 JH In-Stock Unstable HISG 0 46 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NC1CCCCC1 ZINC000217604481 GH In-Stock Unstable CASP3 15 40 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NC1CCCCC1 ZINC000217604481 GH In-Stock Unstable CASP6 18 40 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NC1CCCCC1 ZINC000217604481 GH In-Stock Unstable SFRP1 73 32 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NC1CCCCC1 ZINC000217604481 GH In-Stock Unstable WNT3 51 34 Cc1ccc(NC(=O)NCC2CCCCC2)c(O)c1 ZINC000217604487 CG For-Sale Unstable THRB 15 43 Cc1ccc(NC(=O)NCC2CCCCC2)c(O)c1 ZINC000217604487 CG For-Sale Unstable LDLR 0 41 Cc1ccc(NC(=O)NCC2CCCCC2)c(O)c1 ZINC000217604487 CG For-Sale Unstable EPHX2 15 51 COc1ccc2cc(C(=O)N3CCC[C@]4(C3)OC(=O)c3ccccc34)[nH]c2c1 ZINC000217604502 GG For-Sale Unstable GRIN2B 19 41 COc1ccc2cc(C(=O)N3CCC[C@]4(C3)OC(=O)c3ccccc34)[nH]c2c1 ZINC000217604502 GG For-Sale Unstable HRH4 15 43 COc1ccc2cc(C(=O)N3CCC[C@]4(C3)OC(=O)c3ccccc34)[nH]c2c1 ZINC000217604502 GG For-Sale Unstable SYK 27 46 COc1ccc2cc(C(=O)N3CCC[C@]4(C3)OC(=O)c3ccccc34)[nH]c2c1 ZINC000217604502 GG For-Sale Unstable NPY5R 29 43 CCCC[C@@H]1NC(=O)[C@H]1O ZINC000217604517 AC For-Sale Unstable GAA 20 42 CCCC[C@@H]1NC(=O)[C@H]1O ZINC000217604517 AC For-Sale Unstable SI 19 42 CCCC[C@@H]1NC(=O)[C@H]1O ZINC000217604517 AC For-Sale Unstable P0504H10.9 42 35 C=C(CC)COc1ccc(C)cc1/C=C\C(=O)O ZINC000217604529 BG For-Sale Unstable PTGER2 49 51 C=C(CC)COc1ccc(C)cc1/C=C\C(=O)O ZINC000217604529 BG For-Sale Unstable PTGER4 24 47 C=C(CC)COc1ccc(C)cc1/C=C\C(=O)O ZINC000217604529 BG For-Sale Unstable PTGER3 19 51 C=C(CC)COc1ccc(C)cc1/C=C\C(=O)O ZINC000217604529 BG For-Sale Unstable AKR1C3 31 41 O=C(C(F)F)N1CCN(c2ccc(O)cc2)CC1 ZINC000217604532 CD On-Demand Unstable AKR1C3 26 44 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1cccnc1 ZINC000217604545 IG In-Stock Unstable CACNA1D 58 36 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1cccnc1 ZINC000217604545 IG In-Stock Unstable TGFBR2 50 42 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1cccnc1 ZINC000217604545 IG In-Stock Unstable HISG 0 41 COc1ccc2cc(C(=O)N3CCC[C@@]4(C3)OC(=O)c3ccccc34)[nH]c2c1 ZINC000217604579 GG For-Sale Unstable GRIN2B 19 41 COc1ccc2cc(C(=O)N3CCC[C@@]4(C3)OC(=O)c3ccccc34)[nH]c2c1 ZINC000217604579 GG For-Sale Unstable HRH4 15 43 COc1ccc2cc(C(=O)N3CCC[C@@]4(C3)OC(=O)c3ccccc34)[nH]c2c1 ZINC000217604579 GG For-Sale Unstable SYK 27 46 COc1ccc2cc(C(=O)N3CCC[C@@]4(C3)OC(=O)c3ccccc34)[nH]c2c1 ZINC000217604579 GG For-Sale Unstable NPY5R 29 43 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NCCC1=CCCCC1 ZINC000217604584 HI In-Stock Unstable GNRHR 15 41 CCCCNC(=O)Nc1ccc(/C=C\C(=O)O)cc1C ZINC000217604604 CG For-Sale Unstable ACAT 0 47 O=C(NCC1CCCCC1)Nc1ccc(Cl)cc1C(F)(F)F ZINC000217604607 EK For-Sale Unstable TRPV1 16 50 O=C(NCC1CCCCC1)Nc1ccc(Cl)cc1C(F)(F)F ZINC000217604607 EK For-Sale Unstable NR1H4 31 41 O=C(NCC1CCCCC1)Nc1ccc(Cl)cc1C(F)(F)F ZINC000217604607 EK For-Sale Unstable EPHX2 18 59 O=C(NCC1CCCCC1)Nc1ccc(Cl)cc1C(F)(F)F ZINC000217604607 EK For-Sale Unstable CACNA1I 72 38 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@H](c3cccs3)C2)[C@@H]1c1cccnc1 ZINC000217604623 IG In-Stock Unstable CACNA1D 58 36 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@H](c3cccs3)C2)[C@@H]1c1cccnc1 ZINC000217604623 IG In-Stock Unstable TGFBR2 50 42 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@H](c3cccs3)C2)[C@@H]1c1cccnc1 ZINC000217604623 IG In-Stock Unstable HISG 0 41 CC(C)(C)c1ccc(NC(=O)C(F)F)cc1 ZINC000217604636 BG On-Demand Unstable DHODH 32 40 CC(C)(C)c1ccc(NC(=O)C(F)F)cc1 ZINC000217604636 BG On-Demand Unstable TRPV1 33 54 CC(C)(C)c1ccc(NC(=O)C(F)F)cc1 ZINC000217604636 BG On-Demand Unstable CYNT 43 45 CC(C)(C)c1ccc(NC(=O)C(F)F)cc1 ZINC000217604636 BG On-Demand Unstable PSBA 0 43 COc1ccc(OC)c(CC(=O)Nc2ncc(Cc3ccc(Br)cc3)s2)c1 ZINC000217604650 IJ On-Demand Unstable PDGFRB 36 45 COc1ccc(OC)c(CC(=O)Nc2ncc(Cc3ccc(Br)cc3)s2)c1 ZINC000217604650 IJ On-Demand Unstable CSNK1D 30 48 COc1ccc(OC)c(CC(=O)Nc2ncc(Cc3ccc(Br)cc3)s2)c1 ZINC000217604650 IJ On-Demand Unstable SCD1 44 46 COc1ccc(OC)c(CC(=O)Nc2ncc(Cc3ccc(Br)cc3)s2)c1 ZINC000217604650 IJ On-Demand Unstable SCD 39 46 COc1ccc(/C=C\C(=O)O)cc1NC(=O)NC(C)(C)C ZINC000217604671 CF For-Sale Unstable TUBB1 47 38 COc1ccc(/C=C\C(=O)O)cc1NC(=O)NC(C)(C)C ZINC000217604671 CF For-Sale Unstable ABCG2 15 40 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NCCO ZINC000217604676 FD In-Stock Unstable GNRHR 17 43 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NCCO ZINC000217604676 FD In-Stock Unstable CASP3 21 42 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NCCO ZINC000217604676 FD In-Stock Unstable BDKRB1 0 40 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NCCO ZINC000217604676 FD In-Stock Unstable CASP6 18 42 Fc1cc(CN2CCNCC2)ccc1C(F)F ZINC000217604677 BE On-Demand Anodyne CXCR4 24 48 COc1cc(NC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc(OC)c1OC ZINC000217604693 HG For-Sale Unstable NPY5R 43 54 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1cc(OC)c(OC)c(OC)c1 ZINC000217604717 KH In-Stock Unstable TGFBR2 50 40 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1cc(OC)c(OC)c(OC)c1 ZINC000217604717 KH In-Stock Unstable HISG 0 43 Cc1cc(C)c(NC(=O)NCC2CCCCC2)c(Cl)c1 ZINC000217604720 CJ On-Demand Unstable EPHX2 15 48 Cc1cc(C)c(NC(=O)NCC2CCCCC2)c(Cl)c1 ZINC000217604720 CJ On-Demand Unstable CACNA1I 46 34 CCCCNC(=O)Nc1cc(/C=C\C(=O)O)ccc1OC ZINC000217604742 CF For-Sale Unstable TUBB1 41 36 CCCCNC(=O)Nc1cc(/C=C\C(=O)O)ccc1OC ZINC000217604742 CF For-Sale Unstable AKR1C3 37 42 COc1cc(NC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc(OC)c1OC ZINC000217604759 HG For-Sale Unstable NPY5R 43 54 O=C(Nc1ccccc1F)C(F)F ZINC000217604762 AE On-Demand Anodyne CXCL8 23 49 COC(=O)[C@H]1C[C@@H](OC)CN1S(=O)(=O)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217604773 IG In-Stock Unstable MMP13 43 41 COC(=O)[C@H]1C[C@@H](OC)CN1S(=O)(=O)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217604773 IG In-Stock Unstable CACNA1B 54 33 COC(=O)[C@H]1C[C@@H](OC)CN1S(=O)(=O)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217604773 IG In-Stock Unstable ADAM17 18 47 COC(=O)[C@H]1C[C@@H](OC)CN1S(=O)(=O)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217604773 IG In-Stock Unstable MMP2 21 53 COC(=O)[C@H]1C[C@@H](OC)CN1S(=O)(=O)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217604773 IG In-Stock Unstable MMP3 54 38 COC(=O)[C@H]1C[C@@H](OC)CN1S(=O)(=O)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217604773 IG In-Stock Unstable MMP8 22 41 COC(=O)[C@H]1C[C@@H](OC)CN1S(=O)(=O)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217604773 IG In-Stock Unstable MMP7 49 37 COC(=O)[C@H]1C[C@@H](OC)CN1S(=O)(=O)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217604773 IG In-Stock Unstable MMP1 40 38 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@H](c3cccs3)C2)[C@@H]1c1cc(OC)c(OC)c(OC)c1 ZINC000217604795 KH In-Stock Unstable TGFBR2 50 40 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@H](c3cccs3)C2)[C@@H]1c1cc(OC)c(OC)c(OC)c1 ZINC000217604795 KH In-Stock Unstable HISG 0 43 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NCCCO ZINC000217604800 FD In-Stock Unstable GNRHR 17 42 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NCCCO ZINC000217604800 FD In-Stock Unstable CASP3 20 41 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NCCCO ZINC000217604800 FD In-Stock Unstable BDKRB1 0 41 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NCCCO ZINC000217604800 FD In-Stock Unstable CASP6 18 41 CCCNC(=O)Nc1cc(/C=C\C(=O)O)ccc1OC ZINC000217604826 CE For-Sale Unstable TUBB1 47 37 CCCNC(=O)Nc1cc(/C=C\C(=O)O)ccc1OC ZINC000217604826 CE For-Sale Unstable AKR1C3 29 41 CC(C)(C)[C@@H]1CC[C@@H](O)[C@@H](N2CCCOCC2)C1 ZINC000217604828 CE For-Sale Unstable SLC18A3 18 53 COc1cc(NC(=O)NCC2CCCCC2)c(OC)cc1Cl ZINC000217604829 EI On-Demand Unstable DRD3 0 44 COc1cc(NC(=O)NCC2CCCCC2)c(OC)cc1Cl ZINC000217604829 EI On-Demand Unstable HTR4 52 48 COc1cc(NC(=O)NCC2CCCCC2)c(OC)cc1Cl ZINC000217604829 EI On-Demand Unstable CACNA1I 46 33 COC(=O)[C@H]1C[C@H](OC)CN1S(=O)(=O)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217604851 IG In-Stock Unstable MMP13 43 41 COC(=O)[C@H]1C[C@H](OC)CN1S(=O)(=O)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217604851 IG In-Stock Unstable CACNA1B 54 33 COC(=O)[C@H]1C[C@H](OC)CN1S(=O)(=O)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217604851 IG In-Stock Unstable ADAM17 18 47 COC(=O)[C@H]1C[C@H](OC)CN1S(=O)(=O)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217604851 IG In-Stock Unstable MMP2 21 53 COC(=O)[C@H]1C[C@H](OC)CN1S(=O)(=O)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217604851 IG In-Stock Unstable MMP3 54 38 COC(=O)[C@H]1C[C@H](OC)CN1S(=O)(=O)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217604851 IG In-Stock Unstable MMP8 22 41 COC(=O)[C@H]1C[C@H](OC)CN1S(=O)(=O)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217604851 IG In-Stock Unstable MMP7 49 37 COC(=O)[C@H]1C[C@H](OC)CN1S(=O)(=O)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217604851 IG In-Stock Unstable MMP1 40 38 O=C1O[C@@]2(CCCN(C(=O)Nc3ccccc3)C2)c2ccccc21 ZINC000217604880 DG For-Sale Unstable NPY5R 67 57 O=C1O[C@@]2(CCCN(C(=O)Nc3ccccc3)C2)c2ccccc21 ZINC000217604880 DG For-Sale Unstable EPHX2 34 48 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1cc(OC)ccc1OC ZINC000217604884 JH In-Stock Unstable HISG 0 48 CC(=O)N1CCc2ccccc2[C@@H]1CC(=O)Nc1ncc(Cc2ccc(Br)cc2)s1 ZINC000217604895 JJ On-Demand Unstable MGEA5 34 41 Cc1c(Cl)cccc1NC(=O)C(F)F ZINC000217604902 BF On-Demand Unstable CXCL8 49 41 Cc1c(Cl)cccc1NC(=O)C(F)F ZINC000217604902 BF On-Demand Unstable KCNQ2 43 35 COCCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217604930 FD In-Stock Unstable GNRHR 17 43 COCCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217604930 FD In-Stock Unstable CASP3 21 42 COCCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217604930 FD In-Stock Unstable BDKRB1 0 44 COCCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217604930 FD In-Stock Unstable PRTN3 44 31 COCCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217604930 FD In-Stock Unstable CASP6 18 42 NC[C@@H]1CCCCN1C[C@@H](O)c1ccccc1 ZINC000217604931 BD On-Demand Unstable SLC18A2 56 40 NC[C@@H]1CCCCN1C[C@@H](O)c1ccccc1 ZINC000217604931 BD On-Demand Unstable SLC18A3 25 43 COC(=O)[C@@H]1C[C@@H](OC)CN1S(=O)(=O)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217604939 IG In-Stock Unstable MMP13 43 41 COC(=O)[C@@H]1C[C@@H](OC)CN1S(=O)(=O)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217604939 IG In-Stock Unstable CACNA1B 54 33 COC(=O)[C@@H]1C[C@@H](OC)CN1S(=O)(=O)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217604939 IG In-Stock Unstable ADAM17 18 47 COC(=O)[C@@H]1C[C@@H](OC)CN1S(=O)(=O)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217604939 IG In-Stock Unstable MMP2 21 53 COC(=O)[C@@H]1C[C@@H](OC)CN1S(=O)(=O)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217604939 IG In-Stock Unstable MMP3 54 38 COC(=O)[C@@H]1C[C@@H](OC)CN1S(=O)(=O)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217604939 IG In-Stock Unstable MMP8 22 41 COC(=O)[C@@H]1C[C@@H](OC)CN1S(=O)(=O)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217604939 IG In-Stock Unstable MMP7 49 37 COC(=O)[C@@H]1C[C@@H](OC)CN1S(=O)(=O)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217604939 IG In-Stock Unstable MMP1 40 38 O=C(NCC1CCCCC1)Nc1c(Cl)cccc1Cl ZINC000217604941 DJ For-Sale Unstable EPHX2 17 65 O=C(NCC1CCCCC1)Nc1c(Cl)cccc1Cl ZINC000217604941 DJ For-Sale Unstable CACNA1I 41 34 O=C(NCC1CCCCC1)Nc1c(Cl)cccc1Cl ZINC000217604941 DJ For-Sale Unstable ACAT 0 51 O=C1O[C@]2(CCCN(C(=O)Nc3ccccc3)C2)c2ccccc21 ZINC000217604966 DG For-Sale Unstable NPY5R 67 57 O=C1O[C@]2(CCCN(C(=O)Nc3ccccc3)C2)c2ccccc21 ZINC000217604966 DG For-Sale Unstable EPHX2 34 48 CC(=O)N1CCc2ccccc2[C@H]1CC(=O)Nc1ncc(Cc2ccc(Br)cc2)s1 ZINC000217604984 JJ On-Demand Unstable MGEA5 34 41 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1cccc(F)c1 ZINC000217604986 JH In-Stock Unstable CACNA1C 44 41 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1cccc(F)c1 ZINC000217604986 JH In-Stock Unstable CACNA1D 79 41 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1cccc(F)c1 ZINC000217604986 JH In-Stock Unstable TGFBR2 51 42 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1cccc(F)c1 ZINC000217604986 JH In-Stock Unstable HISG 0 41 CC(C)(C)[C@@H]1CC[C@H](O)[C@@H](N2CCCOCC2)C1 ZINC000217604996 CE For-Sale Unstable SLC18A3 18 53 O=C(Nc1ccc(Cl)cc1Cl)C(F)F ZINC000217605025 BG On-Demand Anodyne PYGL 21 48 O=C(Nc1ccc(Cl)cc1Cl)C(F)F ZINC000217605025 BG On-Demand Anodyne ACPS 0 40 COC(=O)[C@@H]1C[C@H](OC)CN1S(=O)(=O)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217605027 IG In-Stock Unstable MMP13 43 41 COC(=O)[C@@H]1C[C@H](OC)CN1S(=O)(=O)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217605027 IG In-Stock Unstable CACNA1B 54 33 COC(=O)[C@@H]1C[C@H](OC)CN1S(=O)(=O)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217605027 IG In-Stock Unstable ADAM17 18 47 COC(=O)[C@@H]1C[C@H](OC)CN1S(=O)(=O)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217605027 IG In-Stock Unstable MMP2 21 53 COC(=O)[C@@H]1C[C@H](OC)CN1S(=O)(=O)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217605027 IG In-Stock Unstable MMP3 54 38 COC(=O)[C@@H]1C[C@H](OC)CN1S(=O)(=O)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217605027 IG In-Stock Unstable MMP8 22 41 COC(=O)[C@@H]1C[C@H](OC)CN1S(=O)(=O)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217605027 IG In-Stock Unstable MMP7 49 37 COC(=O)[C@@H]1C[C@H](OC)CN1S(=O)(=O)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217605027 IG In-Stock Unstable MMP1 40 38 COCCCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217605050 GE In-Stock Unstable GNRHR 16 42 COCCCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217605050 GE In-Stock Unstable CASP3 22 41 COCCCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217605050 GE In-Stock Unstable BDKRB1 0 44 COCCCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217605050 GE In-Stock Unstable CASP6 18 41 Cc1cccc(N2CCN(C(=O)NCC3CCCCC3)CC2)c1C ZINC000217605059 EH For-Sale Unstable HTR1A 32 43 Cc1cccc(N2CCN(C(=O)NCC3CCCCC3)CC2)c1C ZINC000217605059 EH For-Sale Unstable DRD2 22 43 Cc1cccc(N2CCN(C(=O)NCC3CCCCC3)CC2)c1C ZINC000217605059 EH For-Sale Unstable HTR1B 17 41 Cc1cccc(N2CCN(C(=O)NCC3CCCCC3)CC2)c1C ZINC000217605059 EH For-Sale Unstable HTR2A 24 43 Cc1cccc(N2CCN(C(=O)NCC3CCCCC3)CC2)c1C ZINC000217605059 EH For-Sale Unstable HTR2C 29 47 Cc1cccc(N2CCN(C(=O)NCC3CCCCC3)CC2)c1C ZINC000217605059 EH For-Sale Unstable DRD3 21 43 Cc1cccc(N2CCN(C(=O)NCC3CCCCC3)CC2)c1C ZINC000217605059 EH For-Sale Unstable ABCB1 20 41 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@H](c3cccs3)C2)[C@@H]1c1cccc(F)c1 ZINC000217605070 JH In-Stock Unstable CACNA1C 44 41 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@H](c3cccs3)C2)[C@@H]1c1cccc(F)c1 ZINC000217605070 JH In-Stock Unstable CACNA1D 79 41 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@H](c3cccs3)C2)[C@@H]1c1cccc(F)c1 ZINC000217605070 JH In-Stock Unstable TGFBR2 51 42 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@H](c3cccs3)C2)[C@@H]1c1cccc(F)c1 ZINC000217605070 JH In-Stock Unstable HISG 0 41 NC[C@@H]1CCCCN1[C@@H]1CCCC[C@@H]1O ZINC000217605071 BD For-Sale Unstable SLC18A3 28 41 O=C1O[C@@]2(CCCN(C(=O)Nc3ccc(Cl)cc3)C2)c2ccccc21 ZINC000217605081 FI For-Sale Unstable NPY5R 51 56 O=C1O[C@@]2(CCCN(C(=O)Nc3ccc(Cl)cc3)C2)c2ccccc21 ZINC000217605081 FI For-Sale Unstable EPHX2 37 57 O=C1O[C@@]2(CCCN(C(=O)Nc3ccc(Cl)cc3)C2)c2ccccc21 ZINC000217605081 FI For-Sale Unstable TRPM8 28 40 C[C@@H](c1cccc(CN2CCN(CCN3CCOCC3)CC2)c1)N(C)C ZINC000217605122 FD In-Stock Unstable SLC6A4 15 41 C[C@@H](c1cccc(CN2CCN(CCN3CCOCC3)CC2)c1)N(C)C ZINC000217605122 FD In-Stock Unstable SLC6A3 21 41 C[C@@H](c1cccc(CN2CCN(CCN3CCOCC3)CC2)c1)N(C)C ZINC000217605122 FD In-Stock Unstable CASR 48 38 O=C(C(F)F)N1CCN(c2ccccc2F)CC1 ZINC000217605146 CD On-Demand Unstable MC4R 48 40 O=C(C(F)F)N1CCN(c2ccccc2F)CC1 ZINC000217605146 CD On-Demand Unstable KCNQ2 43 37 O=C(C(F)F)N1CCN(c2ccccc2F)CC1 ZINC000217605146 CD On-Demand Unstable NPY2R 42 36 O=C1O[C@]2(CCCN(C(=O)Nc3ccc(Cl)cc3)C2)c2ccccc21 ZINC000217605157 FI For-Sale Unstable NPY5R 51 56 O=C1O[C@]2(CCCN(C(=O)Nc3ccc(Cl)cc3)C2)c2ccccc21 ZINC000217605157 FI For-Sale Unstable EPHX2 37 57 O=C1O[C@]2(CCCN(C(=O)Nc3ccc(Cl)cc3)C2)c2ccccc21 ZINC000217605157 FI For-Sale Unstable TRPM8 28 40 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NCc1ccccc1 ZINC000217605159 GG In-Stock Unstable CA2 24 47 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NCc1ccccc1 ZINC000217605159 GG In-Stock Unstable GNRHR 18 44 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NCc1ccccc1 ZINC000217605159 GG In-Stock Unstable CASP3 21 45 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NCc1ccccc1 ZINC000217605159 GG In-Stock Unstable CA1 23 47 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NCc1ccccc1 ZINC000217605159 GG In-Stock Unstable CA7 15 40 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NCc1ccccc1 ZINC000217605159 GG In-Stock Unstable CA5B 31 40 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NCc1ccccc1 ZINC000217605159 GG In-Stock Unstable CA4 18 47 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NCc1ccccc1 ZINC000217605159 GG In-Stock Unstable CA5A 35 40 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NCc1ccccc1 ZINC000217605159 GG In-Stock Unstable CASP6 19 45 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NCc1ccccc1 ZINC000217605159 GG In-Stock Unstable CA9 16 51 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NCc1ccccc1 ZINC000217605159 GG In-Stock Unstable AKR1C3 21 44 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NCc1ccccc1 ZINC000217605159 GG In-Stock Unstable NAMPT 20 40 C[C@H](c1cccc(CN2CCN(CCN3CCOCC3)CC2)c1)N(C)C ZINC000217605194 FD In-Stock Unstable SLC6A4 15 41 C[C@H](c1cccc(CN2CCN(CCN3CCOCC3)CC2)c1)N(C)C ZINC000217605194 FD In-Stock Unstable SLC6A3 21 41 C[C@H](c1cccc(CN2CCN(CCN3CCOCC3)CC2)c1)N(C)C ZINC000217605194 FD In-Stock Unstable CASR 48 38 C[C@@H]1Oc2ccccc2N(CC(=O)Nc2ccccc2Nc2ccccc2)C1=O ZINC000217605214 GI On-Demand Unstable CCKAR 26 44 C[C@@H]1Oc2ccccc2N(CC(=O)Nc2ccccc2Nc2ccccc2)C1=O ZINC000217605214 GI On-Demand Unstable CCKBR 37 44 C[C@@H](Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217605243 HI In-Stock Unstable GNRHR 17 42 C[C@@H](Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217605243 HI In-Stock Unstable CASP3 22 42 C[C@@H](Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217605243 HI In-Stock Unstable BDKRB1 0 40 C[C@@H](Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217605243 HI In-Stock Unstable CASP6 19 42 C[C@@H](Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217605243 HI In-Stock Unstable ACPS 0 41 CCCNC(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217605258 CE For-Sale Unstable NPY5R 33 43 C[C@H]1Oc2ccccc2N(CC(=O)Nc2ccccc2Nc2ccccc2)C1=O ZINC000217605286 GI On-Demand Unstable CCKAR 26 44 C[C@H]1Oc2ccccc2N(CC(=O)Nc2ccccc2Nc2ccccc2)C1=O ZINC000217605286 GI On-Demand Unstable CCKBR 37 44 COc1ccc([N+](=O)[O-])cc1NC(=O)NCC1CCCCC1 ZINC000217605307 DG On-Demand Unstable TBXA2R 21 41 COc1ccc([N+](=O)[O-])cc1NC(=O)NCC1CCCCC1 ZINC000217605307 DG On-Demand Unstable CACNA1D 65 36 COc1ccc([N+](=O)[O-])cc1NC(=O)NCC1CCCCC1 ZINC000217605307 DG On-Demand Unstable KCNMA1 23 52 COc1ccc([N+](=O)[O-])cc1NC(=O)NCC1CCCCC1 ZINC000217605307 DG On-Demand Unstable STK17B 41 36 COc1ccc([N+](=O)[O-])cc1NC(=O)NCC1CCCCC1 ZINC000217605307 DG On-Demand Unstable WDR5 31 40 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)NCc3cccnc3)[C@H]21 ZINC000217605311 JF In-Stock Unstable TSHR 41 31 O=C(CN1C(=O)c2cccc3cccc(c23)C1=O)NC1CCCC1 ZINC000217605321 DE For-Sale Unstable EPHX2 22 45 C[C@H](Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217605338 HI In-Stock Unstable GNRHR 17 42 C[C@H](Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217605338 HI In-Stock Unstable CASP3 22 42 C[C@H](Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217605338 HI In-Stock Unstable BDKRB1 0 40 C[C@H](Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217605338 HI In-Stock Unstable CASP6 19 42 C[C@H](Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217605338 HI In-Stock Unstable ACPS 0 41 CCCNC(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217605348 CE For-Sale Unstable NPY5R 33 43 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)NCc3cccnc3)[C@@H]21 ZINC000217605379 JF In-Stock Unstable TSHR 41 31 O=C(C(F)F)N1CCC(Cc2ccccc2)CC1 ZINC000217605391 CF On-Demand Unstable F2 22 44 O=C(C(F)F)N1CCC(Cc2ccccc2)CC1 ZINC000217605391 CF On-Demand Unstable CHRM2 22 41 O=C(C(F)F)N1CCC(Cc2ccccc2)CC1 ZINC000217605391 CF On-Demand Unstable ACE 57 38 O=C(C(F)F)N1CCC(Cc2ccccc2)CC1 ZINC000217605391 CF On-Demand Unstable GRIN2B 90 52 O=C(C(F)F)N1CCC(Cc2ccccc2)CC1 ZINC000217605391 CF On-Demand Unstable SIGMAR1 41 49 O=C(C(F)F)N1CCC(Cc2ccccc2)CC1 ZINC000217605391 CF On-Demand Unstable CCR3 61 50 O=C(C(F)F)N1CCC(Cc2ccccc2)CC1 ZINC000217605391 CF On-Demand Unstable CCR5 22 44 O=C(C(F)F)N1CCC(Cc2ccccc2)CC1 ZINC000217605391 CF On-Demand Unstable ST14 49 39 O=C(C(F)F)N1CCC(Cc2ccccc2)CC1 ZINC000217605391 CF On-Demand Unstable GRIN2C 23 47 O=C(C(F)F)N1CCC(Cc2ccccc2)CC1 ZINC000217605391 CF On-Demand Unstable GRIN3A 0 44 O=C(C(F)F)N1CCC(Cc2ccccc2)CC1 ZINC000217605391 CF On-Demand Unstable AMP1_PLAFQ 30 64 COc1cc(Cl)c(C)cc1NC(=O)NCC1CCCCC1 ZINC000217605410 DI For-Sale Unstable HTR4 36 44 COc1cc(Cl)c(C)cc1NC(=O)NCC1CCCCC1 ZINC000217605410 DI For-Sale Unstable CACNA1I 44 32 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NCCc1ccccc1 ZINC000217605437 HH In-Stock Unstable CA2 26 43 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NCCc1ccccc1 ZINC000217605437 HH In-Stock Unstable GNRHR 17 46 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NCCc1ccccc1 ZINC000217605437 HH In-Stock Unstable TBXA2R 44 40 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NCCc1ccccc1 ZINC000217605437 HH In-Stock Unstable CASP3 21 42 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NCCc1ccccc1 ZINC000217605437 HH In-Stock Unstable CA1 27 43 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NCCc1ccccc1 ZINC000217605437 HH In-Stock Unstable BDKRB1 0 40 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NCCc1ccccc1 ZINC000217605437 HH In-Stock Unstable CA4 17 43 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NCCc1ccccc1 ZINC000217605437 HH In-Stock Unstable CASP6 18 42 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NCCc1ccccc1 ZINC000217605437 HH In-Stock Unstable CA12 16 43 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NCCc1ccccc1 ZINC000217605437 HH In-Stock Unstable CA9 22 41 COC(=O)c1ccc2cc(NC(=O)OC(C)(C)C)ccc2n1 ZINC000217605468 DG In-Stock Unstable LEF1 0 44 CC(C)(C)NC(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217605478 DF For-Sale Unstable NPY5R 35 45 Cc1cccnc1NC(=O)NCC1CCCCC1 ZINC000217605523 BG On-Demand Unstable GCK 0 42 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccccc3)cc2C(=O)O)cc1 ZINC000217605549 IH In-Stock Unstable CA2 25 44 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccccc3)cc2C(=O)O)cc1 ZINC000217605549 IH In-Stock Unstable GNRHR 18 53 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccccc3)cc2C(=O)O)cc1 ZINC000217605549 IH In-Stock Unstable TBXA2R 34 40 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccccc3)cc2C(=O)O)cc1 ZINC000217605549 IH In-Stock Unstable TBXAS1 23 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccccc3)cc2C(=O)O)cc1 ZINC000217605549 IH In-Stock Unstable BMP1 76 40 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccccc3)cc2C(=O)O)cc1 ZINC000217605549 IH In-Stock Unstable CA1 26 44 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccccc3)cc2C(=O)O)cc1 ZINC000217605549 IH In-Stock Unstable KCNA5 22 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccccc3)cc2C(=O)O)cc1 ZINC000217605549 IH In-Stock Unstable MMP13 71 45 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccccc3)cc2C(=O)O)cc1 ZINC000217605549 IH In-Stock Unstable ADAM17 52 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccccc3)cc2C(=O)O)cc1 ZINC000217605549 IH In-Stock Unstable CA14 19 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccccc3)cc2C(=O)O)cc1 ZINC000217605549 IH In-Stock Unstable MMP2 42 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccccc3)cc2C(=O)O)cc1 ZINC000217605549 IH In-Stock Unstable MMP3 50 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccccc3)cc2C(=O)O)cc1 ZINC000217605549 IH In-Stock Unstable PRTN3 46 32 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccccc3)cc2C(=O)O)cc1 ZINC000217605549 IH In-Stock Unstable ALOX15 43 38 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccccc3)cc2C(=O)O)cc1 ZINC000217605549 IH In-Stock Unstable MMP9 61 45 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccccc3)cc2C(=O)O)cc1 ZINC000217605549 IH In-Stock Unstable CA12 17 44 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccccc3)cc2C(=O)O)cc1 ZINC000217605549 IH In-Stock Unstable PTGDR 23 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccccc3)cc2C(=O)O)cc1 ZINC000217605549 IH In-Stock Unstable MMP7 34 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccccc3)cc2C(=O)O)cc1 ZINC000217605549 IH In-Stock Unstable IAP 0 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccccc3)cc2C(=O)O)cc1 ZINC000217605549 IH In-Stock Unstable CA9 25 42 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccccc3)cc2C(=O)O)cc1 ZINC000217605549 IH In-Stock Unstable MMP1 61 42 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccccc3)cc2C(=O)O)cc1 ZINC000217605549 IH In-Stock Unstable AKR1C3 31 48 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccccc3)cc2C(=O)O)cc1 ZINC000217605549 IH In-Stock Unstable AKR1C2 51 37 CC(C)(C)NC(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217605556 DF For-Sale Unstable NPY5R 35 45 CCN(C(=O)NCC1CCCCC1)c1cccc(C)c1 ZINC000217605640 CI For-Sale Unstable AMY2 47 34 CCN(C(=O)NCC1CCCCC1)c1cccc(C)c1 ZINC000217605640 CI For-Sale Unstable NR1H4 29 40 O=C(c1ccco1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217605650 DD In-Stock Unstable HSP90AB1 0 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccccc3)cc2C(=O)O)cc1OC ZINC000217605653 JH In-Stock Unstable GNRHR 17 44 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccccc3)cc2C(=O)O)cc1OC ZINC000217605653 JH In-Stock Unstable TBXA2R 38 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccccc3)cc2C(=O)O)cc1OC ZINC000217605653 JH In-Stock Unstable CA7 17 45 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccccc3)cc2C(=O)O)cc1OC ZINC000217605653 JH In-Stock Unstable BDKRB1 0 40 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccccc3)cc2C(=O)O)cc1OC ZINC000217605653 JH In-Stock Unstable PTGDR 16 40 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccccc3)cc2C(=O)O)cc1OC ZINC000217605653 JH In-Stock Unstable IAP 0 44 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccccc3)cc2C(=O)O)cc1OC ZINC000217605653 JH In-Stock Unstable AKR1C3 16 44 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccccc3)cc2C(=O)O)cc1OC ZINC000217605653 JH In-Stock Unstable SCMU_MYCTU 0 44 COc1cccc(NC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217605656 FG For-Sale Unstable NPY5R 60 57 Cc1cccc(C(=O)N2CCN(CCOc3ccccc3Cl)CC2)c1O ZINC000217605711 FG On-Demand Unstable HTR2C 26 40 Cc1cccc(C(=O)N2CCN(CCOc3ccccc3Cl)CC2)c1O ZINC000217605711 FG On-Demand Unstable SLC6A1 50 38 Cc1cccc(C(=O)N2CCN(CCOc3ccccc3Cl)CC2)c1O ZINC000217605711 FG On-Demand Unstable THRB 0 40 Cc1cccc(C(=O)N2CCN(CCOc3ccccc3Cl)CC2)c1O ZINC000217605711 FG On-Demand Unstable P2RX7 0 40 COc1cccc(NC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217605735 FG For-Sale Unstable NPY5R 60 57 O=C(c1ccno1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217605750 DC In-Stock Unstable HSP90AB1 0 43 CC(C)NC(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217605810 CE For-Sale Unstable NR1H4 49 48 CC(C)NC(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217605810 CE For-Sale Unstable AKR1C3 32 44 CC(C)NC(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217605810 CE For-Sale Unstable PTGES 30 49 Cn1c(N2CC[C@H](O)C2)nc2cc(C(=O)NCCn3cccn3)ccc21 ZINC000217605811 FC In-Stock Unstable DRD4 42 33 Cn1c(N2CC[C@H](O)C2)nc2cc(C(=O)NCCn3cccn3)ccc21 ZINC000217605811 FC In-Stock Unstable PLD2 50 36 O=C1C[C@@]2(N1)C(=O)Nc1ccccc12 ZINC000217605819 AC For-Sale Unstable AKR1B1 0 50 COc1ccc(O)cc1OC1CS(=O)(=O)C1 ZINC000217605842 BC For-Sale Unstable PDE4A 21 40 COc1ccc(O)cc1OC1CS(=O)(=O)C1 ZINC000217605842 BC For-Sale Unstable PDE4D 18 40 CC(C)(C)c1ccc(NC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217605843 GJ For-Sale Unstable NPY5R 45 49 CC(C)(C)c1ccc(NC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217605843 GJ For-Sale Unstable EPHX2 37 46 CC(C)(C)c1ccc(NC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217605843 GJ For-Sale Unstable TRPM8 30 41 O=C(c1cccnc1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217605859 DC In-Stock Unstable PIK3CA 26 41 O=C(c1cccnc1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217605859 DC In-Stock Unstable MTOR 36 45 O=C(c1cccnc1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217605859 DC In-Stock Unstable HSP90AB1 0 45 O=C(c1cccnc1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217605859 DC In-Stock Unstable PIK3CG 24 45 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)Nc1cccc(Br)c1)C(=O)OC2 ZINC000217605861 JK In-Stock Unstable IMPDH1 0 63 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)Nc1cccc(Br)c1)C(=O)OC2 ZINC000217605861 JK In-Stock Unstable IMPDH2 0 63 O=C(NCC1CCCCC1)NC[C@@H]1COc2ccccc2O1 ZINC000217605862 DF On-Demand Unstable HTR1A 0 52 O=C1C[C@]2(N1)C(=O)Nc1ccccc12 ZINC000217605886 AC For-Sale Unstable AKR1B1 0 50 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NC[C@@H]1CCCO1 ZINC000217605892 GE In-Stock Unstable BDKRB1 0 44 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NC[C@@H]1CCCO1 ZINC000217605892 GE In-Stock Unstable TNK2 46 38 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NC[C@@H]1CCCO1 ZINC000217605892 GE In-Stock Unstable SFRP1 42 31 CC(C)COC(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217605899 CG For-Sale Unstable PTGER2 0 40 CC(C)COC(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217605899 CG For-Sale Unstable AKR1C3 34 55 CC(C)(C)c1ccc(NC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217605923 GJ For-Sale Unstable NPY5R 45 49 CC(C)(C)c1ccc(NC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217605923 GJ For-Sale Unstable EPHX2 37 46 CC(C)(C)c1ccc(NC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217605923 GJ For-Sale Unstable TRPM8 30 41 COc1ccc(NC(=O)c2sc(NC(=O)c3ccco3)cc2C)c([N+](=O)[O-])c1 ZINC000217605940 HI On-Demand Unstable TAAR1 20 40 O=C(NCC1CCCCC1)NC[C@H]1COc2ccccc2O1 ZINC000217605945 DF On-Demand Unstable HTR1A 0 52 O=C(c1ccccn1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217605960 DC In-Stock Unstable HSP90AB1 0 48 Cn1cncc1CN1CCN(c2cccnc2)CC1 ZINC000217605964 CD In-Stock Unstable HTR1A 17 47 Cn1cncc1CN1CCN(c2cccnc2)CC1 ZINC000217605964 CD In-Stock Unstable DRD4 29 41 Cn1cncc1CN1CCN(c2cccnc2)CC1 ZINC000217605964 CD In-Stock Unstable DRD3 17 49 Cn1cncc1CN1CCN(c2cccnc2)CC1 ZINC000217605964 CD In-Stock Unstable CHRNA4 17 44 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NC[C@H]1CCCO1 ZINC000217605975 GE In-Stock Unstable BDKRB1 0 44 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NC[C@H]1CCCO1 ZINC000217605975 GE In-Stock Unstable TNK2 46 38 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1NC[C@H]1CCCO1 ZINC000217605975 GE In-Stock Unstable SFRP1 42 31 O=C1O[C@@]2(CCCN(C(=O)NCCc3ccccc3)C2)c2ccccc21 ZINC000217606023 FG For-Sale Unstable NPY5R 35 46 C[C@@H]1CCc2ccc(C(F)(F)F)cc2N1 ZINC000217606027 BG In-Stock Unstable HTR5B 0 43 CC(C)COC(=O)NCc1cc(/C=C\C(=O)O)ccc1F ZINC000217606058 CF For-Sale Unstable AKR1C3 37 41 CC(C)COC(=O)NCc1cc(/C=C\C(=O)O)ccc1F ZINC000217606058 CF For-Sale Unstable PDS 44 33 O=C(CCC(=O)c1ccccc1)Nc1nc(-c2ccc3c(c2)CCO3)cs1 ZINC000217606059 GI On-Demand Unstable HDAC9 20 48 O=C(c1cnccn1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217606069 DC In-Stock Unstable HSP90AB1 0 42 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1N1CCCC1 ZINC000217606072 FE In-Stock Unstable CASP3 23 42 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1N1CCCC1 ZINC000217606072 FE In-Stock Unstable KCNQ2 75 42 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1N1CCCC1 ZINC000217606072 FE In-Stock Unstable TRY2_BOVIN 56 34 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1N1CCCC1 ZINC000217606072 FE In-Stock Unstable CASP7 0 42 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1N1CCCC1 ZINC000217606072 FE In-Stock Unstable SFRP1 113 36 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1N1CCCC1 ZINC000217606072 FE In-Stock Unstable WNT3 80 36 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1N1CCCC1 ZINC000217606072 FE In-Stock Unstable NAMPT 39 41 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1N1CCCC1 ZINC000217606072 FE In-Stock Unstable BRPF1 0 40 O[C@@H]1CC[C@@H](c2ccccc2)C[C@@H]1N1CCCOCC1 ZINC000217606097 CE For-Sale Unstable SLC18A3 97 51 O=C1O[C@]2(CCCN(C(=O)NCCc3ccccc3)C2)c2ccccc21 ZINC000217606102 FG For-Sale Unstable NPY5R 35 46 C[C@H]1CCc2ccc(C(F)(F)F)cc2N1 ZINC000217606111 BG In-Stock Unstable HTR5B 0 43 CC(C)COC(=O)NCc1ccc(/C=C\C(=O)O)cc1 ZINC000217606130 CF For-Sale Unstable AKR1C3 35 42 CC(C)COC(=O)NCc1ccc(/C=C\C(=O)O)cc1 ZINC000217606130 CF For-Sale Unstable PDS 57 37 COc1cc2c(cc1OC)CN(Cc1cc(=O)c(O)c(CN(C)Cc3ccccc3)o1)CC2 ZINC000217606145 JH In-Stock Unstable ACHE 20 42 COc1cc2c(cc1OC)CN(Cc1cc(=O)c(O)c(CN(C)Cc3ccccc3)o1)CC2 ZINC000217606145 JH In-Stock Unstable ADRA2B 0 44 COc1cc2c(cc1OC)CN(Cc1cc(=O)c(O)c(CN(C)Cc3ccccc3)o1)CC2 ZINC000217606145 JH In-Stock Unstable ADRA2C 18 44 COc1cc2c(cc1OC)CN(Cc1cc(=O)c(O)c(CN(C)Cc3ccccc3)o1)CC2 ZINC000217606145 JH In-Stock Unstable ABCB1B 65 37 COc1cc2c(cc1OC)CN(Cc1cc(=O)c(O)c(CN(C)Cc3ccccc3)o1)CC2 ZINC000217606145 JH In-Stock Unstable ABCB1 25 48 COc1cc2c(cc1OC)CN(Cc1cc(=O)c(O)c(CN(C)Cc3ccccc3)o1)CC2 ZINC000217606145 JH In-Stock Unstable HCRTR2 15 42 Cc1cc(Br)ccc1NC(=O)NCC1CCCCC1 ZINC000217606163 EI On-Demand Unstable LDLR 0 41 Cc1cc(C(=O)N2Cc3cnc(N4CCOCC4)nc3C2)no1 ZINC000217606175 DC In-Stock Unstable HSP90AB1 0 41 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1N1CCCCC1 ZINC000217606184 FF In-Stock Unstable WNT3 49 30 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1N1CCCCC1 ZINC000217606184 FF In-Stock Unstable BRPF1 0 41 O[C@H]1CC[C@@H](c2ccccc2)C[C@@H]1N1CCCOCC1 ZINC000217606188 CE For-Sale Unstable SLC18A3 97 51 O=C1O[C@@]2(CCCN(C(=O)NCCCl)C2)c2ccccc21 ZINC000217606218 DE For-Sale Unstable NPY5R 32 43 CC[C@@H](C)[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217606247 HD In-Stock Unstable EDNRA 40 39 CC[C@@H](C)[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217606247 HD In-Stock Unstable CCKAR 49 37 CC[C@@H](C)[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217606247 HD In-Stock Unstable CTSL 28 41 CC[C@@H](C)[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217606247 HD In-Stock Unstable CCKBR 51 37 CC[C@@H](C)[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217606247 HD In-Stock Unstable GHSR 61 39 Cc1cc(NC(=O)NCC2CCCCC2)ccc1Br ZINC000217606256 EI For-Sale Unstable DHODH 0 46 Cc1cc(NC(=O)NCC2CCCCC2)ccc1Br ZINC000217606256 EI For-Sale Unstable LDLR 0 40 Cc1cc(NC(=O)NCC2CCCCC2)ccc1Br ZINC000217606256 EI For-Sale Unstable EPHX2 16 60 Cc1cc(NC(=O)NCC2CCCCC2)ccc1Br ZINC000217606256 EI For-Sale Unstable PRMT3 36 42 O[C@@H]1CC[C@H](c2ccccc2)C[C@@H]1N1CCCOCC1 ZINC000217606267 CE For-Sale Unstable SLC18A3 97 51 O=C(c1cccs1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217606273 DD In-Stock Unstable PIK3CA 17 40 O=C(c1cccs1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217606273 DD In-Stock Unstable MTOR 24 40 O=C(c1cccs1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217606273 DD In-Stock Unstable HSP90AB1 0 43 O=C(c1cccs1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217606273 DD In-Stock Unstable PIK3CG 18 40 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1N1CCOCC1 ZINC000217606287 GD In-Stock Unstable GNRHR 18 46 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1N1CCOCC1 ZINC000217606287 GD In-Stock Unstable CASP3 25 40 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1N1CCOCC1 ZINC000217606287 GD In-Stock Unstable SLC6A9 18 45 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1N1CCOCC1 ZINC000217606287 GD In-Stock Unstable CASP6 18 40 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1N1CCOCC1 ZINC000217606287 GD In-Stock Unstable CASP7 0 40 O=C(O)c1cc(S(=O)(=O)NCc2ccccc2)ccc1N1CCOCC1 ZINC000217606287 GD In-Stock Unstable SFRP1 51 34 O=C1O[C@]2(CCCN(C(=O)NCCCl)C2)c2ccccc21 ZINC000217606297 DE For-Sale Unstable NPY5R 32 43 COc1ccc([C@@H]2CC(=O)Oc3ccc4c(c32)OC(=C(C)C)C4=O)c(OC)c1OC ZINC000217606352 HI In-Stock Unstable MT-ND4 42 32 O[C@H]1CC[C@H](c2ccccc2)C[C@@H]1N1CCCOCC1 ZINC000217606358 CE For-Sale Unstable SLC18A3 97 51 CCOCCCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217606388 GF In-Stock Unstable GNRHR 16 41 Cc1ccc2cccc(OC/C=C\CN)c2n1 ZINC000217606396 BE For-Sale Unstable BDKRB2 58 34 Cc1ccc2cccc(OC/C=C\CN)c2n1 ZINC000217606396 BE For-Sale Unstable MCHR1 25 44 O=C(c1ccsc1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217606407 DD In-Stock Unstable MTOR 28 40 O=C(c1ccsc1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217606407 DD In-Stock Unstable HSP90AB1 0 43 CCCCOc1ccc(NC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217606408 GJ For-Sale Unstable FAAH 22 42 CCCCOc1ccc(NC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217606408 GJ For-Sale Unstable NPY5R 43 47 CCCCOc1ccc(NC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217606408 GJ For-Sale Unstable EPHX2 39 44 O=C(Nc1ccc(-c2ccccc2)cc1)C(F)F ZINC000217606413 BH On-Demand Anodyne EPHX1 0 43 O=C(Nc1ccc(-c2ccccc2)cc1)C(F)F ZINC000217606413 BH On-Demand Anodyne DHODH 19 47 O=C(Nc1ccc(-c2ccccc2)cc1)C(F)F ZINC000217606413 BH On-Demand Anodyne MME 46 45 O=C(Nc1ccc(-c2ccccc2)cc1)C(F)F ZINC000217606413 BH On-Demand Anodyne CA1 19 44 O=C(Nc1ccc(-c2ccccc2)cc1)C(F)F ZINC000217606413 BH On-Demand Anodyne GUAB 0 50 O=C(Nc1ccc(-c2ccccc2)cc1)C(F)F ZINC000217606413 BH On-Demand Anodyne PRNP 36 49 O=C(Nc1ccc(-c2ccccc2)cc1)C(F)F ZINC000217606413 BH On-Demand Anodyne MMP2 23 40 O=C(Nc1ccc(-c2ccccc2)cc1)C(F)F ZINC000217606413 BH On-Demand Anodyne MMP3 19 42 O=C(Nc1ccc(-c2ccccc2)cc1)C(F)F ZINC000217606413 BH On-Demand Anodyne HDAC1 17 46 O=C(Nc1ccc(-c2ccccc2)cc1)C(F)F ZINC000217606413 BH On-Demand Anodyne HDAC3 18 46 O=C(Nc1ccc(-c2ccccc2)cc1)C(F)F ZINC000217606413 BH On-Demand Anodyne HDAC6 18 46 O=C(Nc1ccc(-c2ccccc2)cc1)C(F)F ZINC000217606413 BH On-Demand Anodyne SLC1A1 17 50 O=C(Nc1ccc(-c2ccccc2)cc1)C(F)F ZINC000217606413 BH On-Demand Anodyne ACE2 41 36 O=C(Nc1ccc(-c2ccccc2)cc1)C(F)F ZINC000217606413 BH On-Demand Anodyne SLC1A2 25 50 O=C(Nc1ccc(-c2ccccc2)cc1)C(F)F ZINC000217606413 BH On-Demand Anodyne E1 0 46 O=C(Nc1ccc(-c2ccccc2)cc1)C(F)F ZINC000217606413 BH On-Demand Anodyne SMO 27 41 O=C(Nc1ccc(-c2ccccc2)cc1)C(F)F ZINC000217606413 BH On-Demand Anodyne Q25615_ONCVO 23 42 O=C(Nc1ccc(-c2ccccc2)cc1)C(F)F ZINC000217606413 BH On-Demand Anodyne P95276_MYCTO 0 43 COc1ccc([C@H]2CC(=O)Oc3ccc4c(c32)OC(=C(C)C)C4=O)c(OC)c1OC ZINC000217606442 HI In-Stock Unstable MT-ND4 42 32 CC(C)OCCCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217606488 HG In-Stock Unstable GNRHR 16 41 CC(C)OCCCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217606488 HG In-Stock Unstable CASP3 21 41 CC(C)OCCCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217606488 HG In-Stock Unstable BDKRB1 0 41 CC(C)OCCCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217606488 HG In-Stock Unstable CASP6 18 41 CCCCOc1ccc(NC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217606491 GJ For-Sale Unstable FAAH 22 42 CCCCOc1ccc(NC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217606491 GJ For-Sale Unstable NPY5R 43 47 CCCCOc1ccc(NC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217606491 GJ For-Sale Unstable EPHX2 39 44 Cc1ccc(C(=O)CCC(=O)Nc2nc(-c3ccc4c(c3)CCO4)cs2)cc1 ZINC000217606497 GJ On-Demand Unstable HDAC9 18 51 Cc1ccccc1C(=O)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217606519 DD In-Stock Unstable HSP90AB1 0 47 O=C(Nc1cc(Cl)cc(Cl)c1)C(F)F ZINC000217606544 BG On-Demand Anodyne ATF1 24 40 O=C(Nc1cc(Cl)cc(Cl)c1)C(F)F ZINC000217606544 BG On-Demand Anodyne NFKB1 22 40 O=C(Nc1cc(Cl)cc(Cl)c1)C(F)F ZINC000217606544 BG On-Demand Anodyne PROC1 0 41 O=C(Nc1cc(Cl)cc(Cl)c1)C(F)F ZINC000217606544 BG On-Demand Anodyne GLN2 0 41 O=C(Nc1cc(Cl)cc(Cl)c1)C(F)F ZINC000217606544 BG On-Demand Anodyne OSIGBA0132E09-OSIGBA0108L24.11 0 41 O=C1O[C@@]2(CCCN(C(=O)Nc3cccc(Cl)c3)C2)c2ccccc21 ZINC000217606588 FI For-Sale Unstable NPY5R 55 49 O=C1O[C@@]2(CCCN(C(=O)Nc3cccc(Cl)c3)C2)c2ccccc21 ZINC000217606588 FI For-Sale Unstable EPHX2 20 44 CCCCCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217606599 GG In-Stock Unstable GNRHR 17 43 CCCCCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217606599 GG In-Stock Unstable CASP3 19 40 CCCCCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217606599 GG In-Stock Unstable CASP6 17 40 O=C1O[C@]2(CCCN(C(=O)Nc3cccc(Cl)c3)C2)c2ccccc21 ZINC000217606667 FI For-Sale Unstable NPY5R 55 49 O=C1O[C@]2(CCCN(C(=O)Nc3cccc(Cl)c3)C2)c2ccccc21 ZINC000217606667 FI For-Sale Unstable EPHX2 20 44 CC(C)CCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217606703 GG In-Stock Unstable GNRHR 17 43 CC(C)CCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217606703 GG In-Stock Unstable CASP3 22 42 CC(C)CCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217606703 GG In-Stock Unstable CASP6 18 42 CC[C@@H](C)c1ccccc1NC(=O)NCC1CCCCC1 ZINC000217606721 CJ For-Sale Unstable KCNQ2 43 35 CC[C@@H](C)c1ccccc1NC(=O)NCC1CCCCC1 ZINC000217606721 CJ For-Sale Unstable NMBR 15 43 CC[C@@H](C)c1ccccc1NC(=O)NCC1CCCCC1 ZINC000217606721 CJ For-Sale Unstable SOAT1 21 41 CC[C@@H](C)c1ccccc1NC(=O)NCC1CCCCC1 ZINC000217606721 CJ For-Sale Unstable ACAT 0 46 CC[C@@H](C)c1ccccc1NC(=O)NCC1CCCCC1 ZINC000217606721 CJ For-Sale Unstable AO-ACHE 0 43 O=C(Nc1nc(-c2ccc3c(c2)CCO3)cs1)c1ccc(Cl)c(NC(=O)c2cccs2)c1 ZINC000217606731 JK On-Demand Unstable ITGAL 16 40 O=C(Nc1nc(-c2ccc3c(c2)CCO3)cs1)c1ccc(Cl)c(NC(=O)c2cccs2)c1 ZINC000217606731 JK On-Demand Unstable MPL 51 41 Cc1cc(C(=O)N2Cc3cnc(N4CCOCC4)nc3C2)c(C)o1 ZINC000217606756 ED In-Stock Unstable HSP90AB1 16 44 O=C1O[C@@]2(CCCN(C(=O)NCc3ccc(Cl)cc3)C2)c2ccccc21 ZINC000217606775 FH For-Sale Unstable NPY5R 29 49 O=C1O[C@@]2(CCCN(C(=O)NCc3ccc(Cl)cc3)C2)c2ccccc21 ZINC000217606775 FH For-Sale Unstable NPSR1 26 40 CC[C@H](C)c1ccccc1NC(=O)NCC1CCCCC1 ZINC000217606788 CJ For-Sale Unstable KCNQ2 43 35 CC[C@H](C)c1ccccc1NC(=O)NCC1CCCCC1 ZINC000217606788 CJ For-Sale Unstable NMBR 15 43 CC[C@H](C)c1ccccc1NC(=O)NCC1CCCCC1 ZINC000217606788 CJ For-Sale Unstable SOAT1 21 41 CC[C@H](C)c1ccccc1NC(=O)NCC1CCCCC1 ZINC000217606788 CJ For-Sale Unstable ACAT 0 46 CC[C@H](C)c1ccccc1NC(=O)NCC1CCCCC1 ZINC000217606788 CJ For-Sale Unstable AO-ACHE 0 43 CCOC(=O)/C=C(/N)C(C)=O ZINC000217606792 AB For-Sale Unstable HCAR2 15 45 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217606806 GG In-Stock Unstable GNRHR 16 41 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217606806 GG In-Stock Unstable CASP3 21 41 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217606806 GG In-Stock Unstable CASP6 18 41 O=C1O[C@]2(CCCN(C(=O)NCc3ccc(Cl)cc3)C2)c2ccccc21 ZINC000217606856 FH For-Sale Unstable NPY5R 29 49 O=C1O[C@]2(CCCN(C(=O)NCc3ccc(Cl)cc3)C2)c2ccccc21 ZINC000217606856 FH For-Sale Unstable NPSR1 26 40 O=C(Cc1cccs1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217606871 ED In-Stock Unstable MTOR 19 40 CCC[C@H](C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217606880 GG In-Stock Unstable GNRHR 16 41 CCC[C@H](C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217606880 GG In-Stock Unstable CASP3 21 41 CCC[C@H](C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217606880 GG In-Stock Unstable CASP6 18 41 O=C1O[C@@]2(CCCN(C(=O)NC3CCCCC3)C2)c2ccccc21 ZINC000217606949 EG For-Sale Unstable NPY5R 51 46 O=C1O[C@@]2(CCCN(C(=O)NC3CCCCC3)C2)c2ccccc21 ZINC000217606949 EG For-Sale Unstable EPHX2 24 44 CC(C)COC(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217606954 CF For-Sale Unstable PTGER2 0 40 CC(C)COC(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217606954 CF For-Sale Unstable NPR 57 33 CC(C)COC(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217606954 CF For-Sale Unstable AKR1C3 41 50 CC(C)COC(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217606954 CF For-Sale Unstable PDS 75 40 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1ccccc1CN(C)C ZINC000217606960 CJ For-Sale Unstable TRPM8 16 45 COC[C@@H](C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217607003 GE In-Stock Unstable GNRHR 16 40 COC[C@@H](C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217607003 GE In-Stock Unstable CASP3 19 41 COC[C@@H](C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217607003 GE In-Stock Unstable CASP6 18 41 O=C(NCC1CCCCC1)Nc1ccc(F)c(F)c1F ZINC000217607016 CH On-Demand Unstable EPHX2 15 64 O=C1O[C@]2(CCCN(C(=O)NC3CCCCC3)C2)c2ccccc21 ZINC000217607026 EG For-Sale Unstable NPY5R 51 46 O=C1O[C@]2(CCCN(C(=O)NC3CCCCC3)C2)c2ccccc21 ZINC000217607026 EG For-Sale Unstable EPHX2 24 44 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1ccccc1CN(C)C ZINC000217607039 CJ For-Sale Unstable TRPM8 16 45 O=C(Nc1nc(-c2ccc3c(c2)CCO3)cs1)c1cc(N2CCOCC2)ccn1 ZINC000217607061 HG On-Demand Unstable EPHB4 55 32 O=C(Nc1nc(-c2ccc3c(c2)CCO3)cs1)c1cc(N2CCOCC2)ccn1 ZINC000217607061 HG On-Demand Unstable SMG1 41 34 N#Cc1cccc(C(=O)N2Cc3cnc(N4CCOCC4)nc3C2)c1 ZINC000217607069 ED In-Stock Unstable SLC6A7 0 43 O=C(Nc1cccnc1)C(F)F ZINC000217607072 AD On-Demand Anodyne NAMPT 33 51 COC[C@H](C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217607101 GE In-Stock Unstable GNRHR 16 40 COC[C@H](C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217607101 GE In-Stock Unstable CASP3 19 41 COC[C@H](C)Nc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217607101 GE In-Stock Unstable CASP6 18 41 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1ccccc1CN(C)C ZINC000217607120 CJ For-Sale Unstable TRPM8 16 45 CCOc1ccc(NC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217607129 FH For-Sale Unstable NPY5R 48 49 CCOc1ccc(NC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217607129 FH For-Sale Unstable EPHX2 39 42 O=C(NCC1CCCCC1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217607135 FF For-Sale Unstable HRH2 24 45 O=C(NCC1CCCCC1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217607135 FF For-Sale Unstable KCNH2 17 47 O=C(NCC1CCCCC1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217607135 FF For-Sale Unstable EDNRB 19 41 O=C(NCC1CCCCC1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217607135 FF For-Sale Unstable EDNRA 18 41 O=C(NCC1CCCCC1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217607135 FF For-Sale Unstable BMP1 26 43 O=C(NCC1CCCCC1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217607135 FF For-Sale Unstable SIGMAR1 18 53 O=C(NCC1CCCCC1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217607135 FF For-Sale Unstable CCR3 18 41 O=C(NCC1CCCCC1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217607135 FF For-Sale Unstable NOS2 94 35 O=C(NCC1CCCCC1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217607135 FF For-Sale Unstable SSTR3 116 38 O=C(NCC1CCCCC1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217607135 FF For-Sale Unstable MCHR1 43 54 O=C(/C=C/c1ccccc1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217607185 ED In-Stock Unstable ITGAL 41 31 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1ccccc1CN(C)C ZINC000217607200 CJ For-Sale Unstable TRPM8 16 45 CCCNc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O ZINC000217607203 FG In-Stock Unstable BDKRB1 16 42 CC(C)C[C@@H](CO)NC(=O)CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217607213 HD In-Stock Unstable EDNRA 38 42 CC(C)C[C@@H](CO)NC(=O)CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217607213 HD In-Stock Unstable CCKAR 40 37 CC(C)C[C@@H](CO)NC(=O)CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217607213 HD In-Stock Unstable NMBR 50 36 CC(C)C[C@@H](CO)NC(=O)CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217607213 HD In-Stock Unstable GRPR 78 37 CC(C)C[C@@H](CO)NC(=O)CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217607213 HD In-Stock Unstable HDAC2 15 43 CC(C)C[C@@H](CO)NC(=O)CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217607213 HD In-Stock Unstable GHSR 54 38 CC(C)C[C@@H](CO)NC(=O)CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217607213 HD In-Stock Unstable SLC15A2 0 41 CC(C)C[C@@H](CO)NC(=O)CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217607213 HD In-Stock Unstable KISS1R 52 32 CCOc1ccc(NC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217607220 FH For-Sale Unstable NPY5R 48 49 CCOc1ccc(NC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217607220 FH For-Sale Unstable EPHX2 39 42 CCCNc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O ZINC000217607288 FG In-Stock Unstable BDKRB1 16 42 O=C(Nc1nc(-c2ccc3c(c2)CCO3)cs1)c1cc(N2CCCC2)ccn1 ZINC000217607294 GH On-Demand Unstable MPL 42 40 O=C(CCc1ccccc1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217607301 ED In-Stock Unstable FAAH 18 40 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217607328 JF In-Stock Unstable MC4R 42 35 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217607328 JF In-Stock Unstable HDAC8 0 40 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217607328 JF In-Stock Unstable MC3R 30 40 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217607328 JF In-Stock Unstable MC5R 36 43 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217607328 JF In-Stock Unstable MC1R 18 40 O=C1O[C@@]2(CCCN(C(=O)Nc3ccccc3Cl)C2)c2ccccc21 ZINC000217607334 FI For-Sale Unstable NPY5R 49 55 O=C1O[C@@]2(CCCN(C(=O)Nc3ccccc3Cl)C2)c2ccccc21 ZINC000217607334 FI For-Sale Unstable EPHX2 15 40 Cc1ccc(NC(=O)NCC2CCCCC2)c(N)c1 ZINC000217607348 CG For-Sale Unstable LDLR 0 41 NC/C=C\CN1CCN(c2ccc(F)cc2)CC1 ZINC000217607376 BD For-Sale Unstable DRD4 25 43 O=C(O)/C=C\c1cnc(NS(=O)(=O)c2ccc(Cl)s2)s1 ZINC000217607383 FF For-Sale Anodyne CCR4 52 33 CC(C)Nc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O ZINC000217607387 FG In-Stock Unstable LEF 30 42 O=C(CNC(=O)c1ccc(C(F)(F)F)cc1)Nc1nc(-c2ccc3c(c2)CCO3)cs1 ZINC000217607408 II On-Demand Unstable GCGR 18 44 O=C(CNC(=O)c1ccc(C(F)(F)F)cc1)Nc1nc(-c2ccc3c(c2)CCO3)cs1 ZINC000217607408 II On-Demand Unstable MPL 54 43 O=C(CNC(=O)c1ccc(C(F)(F)F)cc1)Nc1nc(-c2ccc3c(c2)CCO3)cs1 ZINC000217607408 II On-Demand Unstable GIPR 55 44 O=C1O[C@]2(CCCN(C(=O)Nc3ccccc3Cl)C2)c2ccccc21 ZINC000217607409 FI For-Sale Unstable NPY5R 49 55 O=C1O[C@]2(CCCN(C(=O)Nc3ccccc3Cl)C2)c2ccccc21 ZINC000217607409 FI For-Sale Unstable EPHX2 15 40 O=C(COc1ccccc1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217607415 ED In-Stock Unstable COLA 129 47 O=C(COc1ccccc1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217607415 ED In-Stock Unstable CPT1A 106 41 O=C(COc1ccccc1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217607415 ED In-Stock Unstable CPT2 52 42 O=C(NCCCn1ccnc1)C(F)F ZINC000217607460 BC On-Demand Unstable TBXAS1 65 54 O=C(NCCCn1ccnc1)C(F)F ZINC000217607460 BC On-Demand Unstable HMOX2 47 37 O=C(NCCCn1ccnc1)C(F)F ZINC000217607460 BC On-Demand Unstable CAMC 0 40 O=C(NCCCn1ccnc1)C(F)F ZINC000217607460 BC On-Demand Unstable QPCT 52 50 O=C(NCCCn1ccnc1)C(F)F ZINC000217607460 BC On-Demand Unstable NAMPT 24 42 O=C(NCC1CCCCC1)Nc1ccc(C(F)(F)F)cc1 ZINC000217607471 DI For-Sale Unstable DHODH 45 44 O=C(NCC1CCCCC1)Nc1ccc(C(F)(F)F)cc1 ZINC000217607471 DI For-Sale Unstable TRPV1 23 42 O=C(NCC1CCCCC1)Nc1ccc(C(F)(F)F)cc1 ZINC000217607471 DI For-Sale Unstable CCR3 22 50 O=C(NCC1CCCCC1)Nc1ccc(C(F)(F)F)cc1 ZINC000217607471 DI For-Sale Unstable EPHX2 73 64 O=C(NCC1CCCCC1)Nc1ccc(C(F)(F)F)cc1 ZINC000217607471 DI For-Sale Unstable MCHR1 19 43 O=C(NCC1CCCCC1)Nc1ccc(C(F)(F)F)cc1 ZINC000217607471 DI For-Sale Unstable PTPA 0 40 O=C(NCC1CCCCC1)Nc1ccc(C(F)(F)F)cc1 ZINC000217607471 DI For-Sale Unstable TRPM8 40 34 O=C(NCC1CCCCC1)Nc1ccc(C(F)(F)F)cc1 ZINC000217607471 DI For-Sale Unstable PRMT3 34 42 CC(C)Nc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O ZINC000217607487 FG In-Stock Unstable LEF 30 42 NC/C=C\CN1CCN(c2ccccn2)CC1 ZINC000217607494 BC For-Sale Unstable DRD2 17 57 NC/C=C\CN1CCN(c2ccccn2)CC1 ZINC000217607494 BC For-Sale Unstable DRD4 38 49 NC/C=C\CN1CCN(c2ccccn2)CC1 ZINC000217607494 BC For-Sale Unstable EBP 27 41 O=C(CNC(=O)c1ccc(Cl)c(Cl)c1)Nc1nc(-c2ccc3c(c2)CCO3)cs1 ZINC000217607502 II On-Demand Unstable MPL 25 42 O=C(CNC(=O)c1ccc(Cl)c(Cl)c1)Nc1nc(-c2ccc3c(c2)CCO3)cs1 ZINC000217607502 II On-Demand Unstable GIPR 31 41 O=C(CNC(=O)c1ccc(Cl)c(Cl)c1)Nc1nc(-c2ccc3c(c2)CCO3)cs1 ZINC000217607502 II On-Demand Unstable TRPA1 15 41 COCCNC(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217607516 DD For-Sale Unstable NPY5R 28 46 COc1ccccc1C(=O)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217607525 ED In-Stock Unstable BRPF1 0 40 O=C(O)/C=C\c1cnc(NS(=O)(=O)c2ccccc2)s1 ZINC000217607555 DE For-Sale Anodyne NCE103 17 43 O=C(O)/C=C\c1cnc(NS(=O)(=O)c2ccccc2)s1 ZINC000217607555 DE For-Sale Anodyne A6YCJ1_9METZ 15 43 CCCCNc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O ZINC000217607592 GH In-Stock Unstable BDKRB1 17 43 COCCNC(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217607599 DD For-Sale Unstable NPY5R 28 46 O=C(Nc1nc(-c2ccc3c(c2)CCO3)cs1)[C@@H]1CCCN(C(=O)Nc2ccccc2)C1 ZINC000217607626 IJ On-Demand Unstable RHOA 0 44 O=C(Nc1nc(-c2ccc3c(c2)CCO3)cs1)[C@@H]1CCCN(C(=O)Nc2ccccc2)C1 ZINC000217607626 IJ On-Demand Unstable TRPC6 43 35 O=C(Nc1nc(-c2ccc3c(c2)CCO3)cs1)[C@@H]1CCCN(C(=O)Nc2ccccc2)C1 ZINC000217607626 IJ On-Demand Unstable TRPC3 42 35 Cn1cccc(C(=O)N2Cc3cnc(N4CCOCC4)nc3C2)c1=O ZINC000217607634 EC In-Stock Unstable HSP90AB1 0 46 CC(C)(C)NC(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217607640 CE For-Sale Unstable PTGER2 23 42 CC(C)(C)NC(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217607640 CE For-Sale Unstable ANPEP 15 40 CC(=O)c1cccc(S(=O)(=O)C[C@H](C)F)c1 ZINC000217607643 BE For-Sale Unstable IMDH_CRYPV 43 37 CC1(C)CCCN(c2ccc(CBr)cc2C(F)(F)F)C1 ZINC000217607644 FK For-Sale Unstable TAAR1 22 40 COc1cccc2c(O)c(C(=O)N3CCc4ccccc4C3)cnc12 ZINC000217607659 EG In-Stock Unstable BCL2 23 47 COc1cccc2c(O)c(C(=O)N3CCc4ccccc4C3)cnc12 ZINC000217607659 EG In-Stock Unstable TRPC6 17 41 CCCCNc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O ZINC000217607676 GH In-Stock Unstable BDKRB1 17 43 CC(=O)c1cccc(S(=O)(=O)C[C@@H](C)F)c1 ZINC000217607710 BE For-Sale Unstable IMDH_CRYPV 43 37 O=C(Nc1nc(-c2ccc3c(c2)CCO3)cs1)[C@H]1CCCN(C(=O)Nc2ccccc2)C1 ZINC000217607718 IJ On-Demand Unstable RHOA 0 44 O=C(Nc1nc(-c2ccc3c(c2)CCO3)cs1)[C@H]1CCCN(C(=O)Nc2ccccc2)C1 ZINC000217607718 IJ On-Demand Unstable TRPC6 43 35 O=C(Nc1nc(-c2ccc3c(c2)CCO3)cs1)[C@H]1CCCN(C(=O)Nc2ccccc2)C1 ZINC000217607718 IJ On-Demand Unstable TRPC3 42 35 O=C1O[C@@]2(CCCN(C(=O)NC34CC5CC(CC(C5)C3)C4)C2)c2ccccc21 ZINC000217607730 GH For-Sale Unstable NPY5R 36 43 O=C1O[C@@]2(CCCN(C(=O)NC34CC5CC(CC(C5)C3)C4)C2)c2ccccc21 ZINC000217607730 GH For-Sale Unstable EPHX2 43 45 CCCCNC(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217607738 CE For-Sale Unstable AKR1C3 28 43 O=C(Cc1ccc(F)cc1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217607741 ED In-Stock Unstable MTOR 16 41 O=C(Cc1ccc(F)cc1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217607741 ED In-Stock Unstable STAT6 43 32 CC(C)(CO)NC(=O)NCC1CCCCC1 ZINC000217607747 BD For-Sale Unstable CACNA1I 41 33 COC(=O)C[C@@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccccc1 ZINC000217607753 EG In-Stock Unstable KCNA5 39 45 CC(C)CNc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O ZINC000217607777 GG In-Stock Unstable KCNA5 0 40 CC(C)CNc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O ZINC000217607777 GG In-Stock Unstable BDKRB1 16 45 CC(C)CNc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O ZINC000217607777 GG In-Stock Unstable MTNN 71 35 CC(C)CNc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O ZINC000217607777 GG In-Stock Unstable LEF 29 40 Cn1ccnc1CN1CCN(C(=O)c2ccccc2OC(F)F)CC1 ZINC000217607786 FD In-Stock Unstable HTR1A 16 43 O=C1O[C@]2(CCCN(C(=O)NC34CC5CC(CC(C5)C3)C4)C2)c2ccccc21 ZINC000217607805 GH For-Sale Unstable NPY5R 36 43 O=C1O[C@]2(CCCN(C(=O)NC34CC5CC(CC(C5)C3)C4)C2)c2ccccc21 ZINC000217607805 GH For-Sale Unstable EPHX2 43 45 CN(Cc1cccc(/C=C\C(=O)O)c1)C(=O)NC(C)(C)C ZINC000217607814 CF For-Sale Unstable PTGER2 0 44 CN(Cc1cccc(/C=C\C(=O)O)c1)C(=O)NC(C)(C)C ZINC000217607814 CF For-Sale Unstable NR1H4 42 38 CN(Cc1cccc(/C=C\C(=O)O)c1)C(=O)NC(C)(C)C ZINC000217607814 CF For-Sale Unstable AKR1C3 40 39 O=C(CCn1cnc2ccccc21)Nc1nc(-c2ccc3c(c2)CCO3)cs1 ZINC000217607829 GI On-Demand Unstable HDAC9 15 40 O=C(CCn1cnc2ccccc21)Nc1nc(-c2ccc3c(c2)CCO3)cs1 ZINC000217607829 GI On-Demand Unstable TRPA1 20 40 COC(=O)C[C@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccccc1 ZINC000217607855 EG In-Stock Unstable KCNA5 39 45 CC(C)CNc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O ZINC000217607859 GG In-Stock Unstable KCNA5 0 40 CC(C)CNc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O ZINC000217607859 GG In-Stock Unstable BDKRB1 18 45 CC(C)CNc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O ZINC000217607859 GG In-Stock Unstable MTNN 74 36 CC(C)CNc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O ZINC000217607859 GG In-Stock Unstable LEF 29 40 CCOc1ccccc1N1CCN(C(=O)C(F)F)CC1 ZINC000217607873 CD On-Demand Unstable HTR1A 68 45 CCOc1ccccc1N1CCN(C(=O)C(F)F)CC1 ZINC000217607873 CD On-Demand Unstable DRD2 65 49 CCOc1ccccc1N1CCN(C(=O)C(F)F)CC1 ZINC000217607873 CD On-Demand Unstable DRD4 27 45 CCOc1ccccc1N1CCN(C(=O)C(F)F)CC1 ZINC000217607873 CD On-Demand Unstable ADRA1D 73 45 CCOc1ccccc1N1CCN(C(=O)C(F)F)CC1 ZINC000217607873 CD On-Demand Unstable HTR2A 28 41 CCOc1ccccc1N1CCN(C(=O)C(F)F)CC1 ZINC000217607873 CD On-Demand Unstable ADRA1A 51 45 CCOc1ccccc1N1CCN(C(=O)C(F)F)CC1 ZINC000217607873 CD On-Demand Unstable ADRA1B 47 45 CCOc1ccccc1N1CCN(C(=O)C(F)F)CC1 ZINC000217607873 CD On-Demand Unstable DRD3 53 41 CCOc1ccccc1N1CCN(C(=O)C(F)F)CC1 ZINC000217607873 CD On-Demand Unstable HTR7 61 44 CCOc1ccccc1N1CCN(C(=O)C(F)F)CC1 ZINC000217607873 CD On-Demand Unstable MC4R 49 48 CCOc1ccccc1N1CCN(C(=O)C(F)F)CC1 ZINC000217607873 CD On-Demand Unstable KCNQ2 52 35 CCOc1ccccc1N1CCN(C(=O)C(F)F)CC1 ZINC000217607873 CD On-Demand Unstable HCN1 42 33 CCOc1ccccc1N1CCN(C(=O)C(F)F)CC1 ZINC000217607873 CD On-Demand Unstable HCN4 42 33 O=C1O[C@@]2(CCCN(C(=O)NC3CCCC3)C2)c2ccccc21 ZINC000217607910 DF For-Sale Unstable NPY5R 53 46 O=C1O[C@@]2(CCCN(C(=O)NC3CCCC3)C2)c2ccccc21 ZINC000217607910 DF For-Sale Unstable EPHX2 21 44 CCCCNC(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217607912 CF For-Sale Unstable NR1H4 42 36 CCCCNC(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217607912 CF For-Sale Unstable AKR1C3 37 44 C[C@@H]1CN(S(=O)(=O)Nc2cccnc2Cl)C[C@@H](C)O1 ZINC000217607932 DD For-Sale Unstable G2YM83_BOTF4 60 36 CC[C@@H](C)Nc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O ZINC000217607952 GH In-Stock Unstable BDKRB1 17 40 CC[C@@H](C)Nc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O ZINC000217607952 GH In-Stock Unstable LEF 30 40 CCOC(=O)CCNC(=O)NCC1CCCCC1 ZINC000217607963 CD For-Sale Unstable EPHX2 15 44 COc1cc2c(c(OC)c1OC)-c1ccc(NCCCCCC(=O)Nc3cccc(-c4nnn(C)n4)c3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217607967 KJ In-Stock Unstable TUBA1A 15 55 Cc1ccc(NC(=O)C(F)F)cc1C ZINC000217607986 AF On-Demand Unstable LEF 41 33 O=C1O[C@]2(CCCN(C(=O)NC3CCCC3)C2)c2ccccc21 ZINC000217607991 DF For-Sale Unstable NPY5R 53 46 O=C1O[C@]2(CCCN(C(=O)NC3CCCC3)C2)c2ccccc21 ZINC000217607991 DF For-Sale Unstable EPHX2 21 44 CCCNC(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217607996 CE For-Sale Unstable NR1H4 48 37 CCCNC(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217607996 CE For-Sale Unstable AKR1C3 31 40 C[C@H]1CN(S(=O)(=O)Nc2cccnc2Cl)C[C@@H](C)O1 ZINC000217608012 DD For-Sale Unstable G2YM83_BOTF4 60 36 O=C(N[C@@H](Cn1cccn1)c1ccccc1)[C@@H]1CC[C@H](O)CC1 ZINC000217608025 DE In-Stock Unstable CCR5 22 42 O=C(N[C@@H](Cn1cccn1)c1ccccc1)[C@@H]1CC[C@H](O)CC1 ZINC000217608025 DE In-Stock Unstable F11 50 40 CC[C@H](C)Nc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O ZINC000217608030 GH In-Stock Unstable BDKRB1 17 40 CC[C@H](C)Nc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O ZINC000217608030 GH In-Stock Unstable LEF 30 40 COC(=O)C[C@H](c1cccc(O)c1)c1c(O)c2ccccc2oc1=O ZINC000217608078 EF In-Stock Unstable NQO1 57 40 COC(=O)C[C@H](c1cccc(O)c1)c1c(O)c2ccccc2oc1=O ZINC000217608078 EF In-Stock Unstable POL 0 48 CN(C)c1cccc(C(=O)N2Cc3cnc(N4CCOCC4)nc3C2)c1 ZINC000217608094 FD In-Stock Unstable MTOR 41 39 C[C@H]1CN(S(=O)(=O)Nc2cccnc2Cl)C[C@H](C)O1 ZINC000217608109 DD For-Sale Unstable G2YM83_BOTF4 60 36 O=C(Nc1ccc(F)cc1)C(F)F ZINC000217608113 AE On-Demand Anodyne MTCA1 29 47 O=C(Nc1ccc(F)cc1)C(F)F ZINC000217608113 AE On-Demand Anodyne P96878_MYCTU 20 47 O=C(Nc1ccc(F)cc1)C(F)F ZINC000217608113 AE On-Demand Anodyne PSBA 0 53 Cc1ccc(NC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1C ZINC000217608116 FH For-Sale Unstable NPY5R 56 48 Cc1ccc(NC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1C ZINC000217608116 FH For-Sale Unstable EPHX2 23 42 CC[C@@H](C)Nc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O ZINC000217608117 GH In-Stock Unstable BDKRB1 17 40 CC[C@@H](C)Nc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O ZINC000217608117 GH In-Stock Unstable LEF 30 40 O=C(N[C@H](Cn1cccn1)c1ccccc1)[C@@H]1CC[C@H](O)CC1 ZINC000217608121 DE In-Stock Unstable CCR5 22 42 O=C(N[C@H](Cn1cccn1)c1ccccc1)[C@@H]1CC[C@H](O)CC1 ZINC000217608121 DE In-Stock Unstable F11 50 40 COC(=O)C[C@@H](c1cccc(O)c1)c1c(O)c2ccccc2oc1=O ZINC000217608152 EF In-Stock Unstable NQO1 57 40 COC(=O)C[C@@H](c1cccc(O)c1)c1c(O)c2ccccc2oc1=O ZINC000217608152 EF In-Stock Unstable POL 0 48 COC(=O)c1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217608177 CG On-Demand Unstable CCKAR 30 43 COC(=O)c1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217608177 CG On-Demand Unstable CCKBR 37 43 COC(=O)c1cccc(NC(=O)NCC2CCCCC2)c1 ZINC000217608177 CG On-Demand Unstable ACAT 0 44 CC[C@H](C)Nc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O ZINC000217608178 GH In-Stock Unstable LEF 30 40 Cc1ccc(NC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1C ZINC000217608195 FH For-Sale Unstable NPY5R 56 48 Cc1ccc(NC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1C ZINC000217608195 FH For-Sale Unstable EPHX2 23 42 O=C(Cc1ccccc1Cl)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217608207 FE In-Stock Unstable AKR1C3 0 40 O=C(Cc1ccccc1Cl)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217608207 FE In-Stock Unstable STAT6 23 41 CN(Cc1ccc(Br)cc1)C(=O)C(F)F ZINC000217608239 CF On-Demand Unstable SHC 17 44 CNc1nc(C2CC2)nc(N[C@@H]2CC[C@@H](C)[C@@H](C)C2)c1C ZINC000217608259 CH For-Sale Unstable CHRM3 0 57 C[C@@H](NS(=O)(=O)c1ccc(NC(C)(C)C)c(C(=O)O)c1)c1ccccc1 ZINC000217608273 GH In-Stock Unstable PRTN3 52 35 C[C@@H](NS(=O)(=O)c1ccc(NC(C)(C)C)c(C(=O)O)c1)c1ccccc1 ZINC000217608273 GH In-Stock Unstable MMP12 40 37 C[C@@H](NS(=O)(=O)c1ccc(NC(C)(C)C)c(C(=O)O)c1)c1ccccc1 ZINC000217608273 GH In-Stock Unstable LEF 29 41 CCOC(=O)c1ccc(CNC(=O)NCC2CCCCC2)cc1 ZINC000217608287 DG On-Demand Unstable PROC 52 36 CCOc1ccccc1NC(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217608290 FH For-Sale Unstable NPY5R 43 52 CCOc1ccccc1NC(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217608290 FH For-Sale Unstable HCN1 43 33 CCOc1ccccc1NC(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217608290 FH For-Sale Unstable HCN4 43 33 CN1CCCC[C@@H]1CN[C@H](c1ccccc1)C1CC1 ZINC000217608295 CG For-Sale Unstable CHRM5 19 41 CN1CCCC[C@@H]1CN[C@H](c1ccccc1)C1CC1 ZINC000217608295 CG For-Sale Unstable CHRNA10 61 43 CNc1nc(C2CC2)nc(N[C@H]2CC[C@@H](C)[C@@H](C)C2)c1C ZINC000217608349 CH For-Sale Unstable CHRM3 0 57 C[C@H](NS(=O)(=O)c1ccc(NC(C)(C)C)c(C(=O)O)c1)c1ccccc1 ZINC000217608366 GH In-Stock Unstable BDKRB1 22 41 C[C@H](NS(=O)(=O)c1ccc(NC(C)(C)C)c(C(=O)O)c1)c1ccccc1 ZINC000217608366 GH In-Stock Unstable PRTN3 52 35 C[C@H](NS(=O)(=O)c1ccc(NC(C)(C)C)c(C(=O)O)c1)c1ccccc1 ZINC000217608366 GH In-Stock Unstable MMP12 41 37 C[C@H](NS(=O)(=O)c1ccc(NC(C)(C)C)c(C(=O)O)c1)c1ccccc1 ZINC000217608366 GH In-Stock Unstable LEF 29 41 CCOc1ccccc1NC(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217608370 FH For-Sale Unstable NPY5R 43 52 CCOc1ccccc1NC(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217608370 FH For-Sale Unstable HCN1 43 33 CCOc1ccccc1NC(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217608370 FH For-Sale Unstable HCN4 43 33 COc1cccc(CCC(=O)Nc2nc(-c3ccc4c(c3)CCO4)cs2)c1 ZINC000217608371 GI On-Demand Unstable ROCK1 48 50 COc1cccc(CCC(=O)Nc2nc(-c3ccc4c(c3)CCO4)cs2)c1 ZINC000217608371 GI On-Demand Unstable MTNR1A 19 40 COc1cccc(CCC(=O)Nc2nc(-c3ccc4c(c3)CCO4)cs2)c1 ZINC000217608371 GI On-Demand Unstable ROCK2 57 50 COc1cccc(CCC(=O)Nc2nc(-c3ccc4c(c3)CCO4)cs2)c1 ZINC000217608371 GI On-Demand Unstable HDAC9 16 41 COc1cccc(CCC(=O)Nc2nc(-c3ccc4c(c3)CCO4)cs2)c1 ZINC000217608371 GI On-Demand Unstable TRPA1 17 43 CN1CCCC[C@H]1CN[C@H](c1ccccc1)C1CC1 ZINC000217608373 CG For-Sale Unstable CHRM5 19 41 CN1CCCC[C@H]1CN[C@H](c1ccccc1)C1CC1 ZINC000217608373 CG For-Sale Unstable CHRNA10 61 43 COC(=O)c1ccc(C(=O)N2Cc3cnc(N4CCOCC4)nc3C2)cc1 ZINC000217608401 FD In-Stock Unstable PIK3CA 27 51 COC(=O)c1ccc(C(=O)N2Cc3cnc(N4CCOCC4)nc3C2)cc1 ZINC000217608401 FD In-Stock Unstable MTOR 45 41 COC(=O)c1ccc(C(=O)N2Cc3cnc(N4CCOCC4)nc3C2)cc1 ZINC000217608401 FD In-Stock Unstable PIK3CG 29 51 CCN1C[C@H](O)[C@H](O)[C@@H]1CO ZINC000217608428 AA For-Sale Unstable MGAM 49 57 CCN1C[C@H](O)[C@H](O)[C@@H]1CO ZINC000217608428 AA For-Sale Unstable UGCG 102 49 CCN1C[C@H](O)[C@H](O)[C@@H]1CO ZINC000217608428 AA For-Sale Unstable GBA 67 56 CCN1C[C@H](O)[C@H](O)[C@@H]1CO ZINC000217608428 AA For-Sale Unstable GAA 29 59 CCN1C[C@H](O)[C@H](O)[C@@H]1CO ZINC000217608428 AA For-Sale Unstable GBA2 170 59 CCN1C[C@H](O)[C@H](O)[C@@H]1CO ZINC000217608428 AA For-Sale Unstable SI 66 59 CNc1nc(C2CC2)nc(N[C@@H]2CC[C@H](C)[C@@H](C)C2)c1C ZINC000217608439 CH For-Sale Unstable CHRM3 0 57 O=C(O)/C=C\c1cnc(NS(=O)(=O)c2cccc(Cl)c2)s1 ZINC000217608476 EF For-Sale Anodyne FBP1 23 49 O=C(O)/C=C\c1cnc(NS(=O)(=O)c2cccc(Cl)c2)s1 ZINC000217608476 EF For-Sale Anodyne CCR2 0 40 C=CCNc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O ZINC000217608483 FG In-Stock Unstable BDKRB1 0 41 C=CCNc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O ZINC000217608483 FG In-Stock Unstable ADAMTS4 44 35 COc1cc(NC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc(OC)c1 ZINC000217608494 GG For-Sale Unstable NPY5R 51 53 CN(Cc1ccccc1Cl)C(=O)C(F)F ZINC000217608502 BF On-Demand Unstable DXS 0 49 Cc1ccccc1CNC(=O)NCC1CCCCC1 ZINC000217608508 CG On-Demand Unstable P2RX7 22 46 Cc1ccccc1CNC(=O)NCC1CCCCC1 ZINC000217608508 CG On-Demand Unstable EPHX2 15 40 O=C(O)Cc1cnc2ccccc2c1-c1ccccc1 ZINC000217608519 CH In-Stock Unstable TSPO 29 42 O=C(O)Cc1cnc2ccccc2c1-c1ccccc1 ZINC000217608519 CH In-Stock Unstable TACR3 48 40 O=C(O)Cc1cnc2ccccc2c1-c1ccccc1 ZINC000217608519 CH In-Stock Unstable NR1H3 27 49 O=C(O)Cc1cnc2ccccc2c1-c1ccccc1 ZINC000217608519 CH In-Stock Unstable NR1H2 46 41 O=C(O)Cc1cnc2ccccc2c1-c1ccccc1 ZINC000217608519 CH In-Stock Unstable PTGDR2 24 43 CNc1nc(C2CC2)nc(N[C@H]2CC[C@H](C)[C@@H](C)C2)c1C ZINC000217608531 CH For-Sale Unstable CHRM3 0 57 O=C(O)/C=C\c1cnc(NS(=O)(=O)c2cccnc2)s1 ZINC000217608556 DD For-Sale Anodyne TBXAS1 25 45 C=CCNc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O ZINC000217608563 FG In-Stock Unstable BDKRB1 0 41 C=CCNc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O ZINC000217608563 FG In-Stock Unstable ADAMTS4 44 35 COc1cc(NC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc(OC)c1 ZINC000217608582 GG For-Sale Unstable NPY5R 51 53 COc1ccc(CN(C)C(=O)C(F)F)cc1OC ZINC000217608626 CD On-Demand Unstable MT-ND1 30 51 CN1CCCC[C@@H]1CN[C@H](c1cccs1)C1CC1 ZINC000217608631 CG For-Sale Unstable CHRNA10 50 35 O=C(c1cccs1)N1CCC(N2CCCn3nc(CO)cc3C2)CC1 ZINC000217608632 FD In-Stock Unstable L3MBTL1 0 45 O=C(c1cccs1)N1CCC(N2CCCn3nc(CO)cc3C2)CC1 ZINC000217608632 FD In-Stock Unstable L3MBTL3 69 45 O=C(O)Cc1c(Cl)nc2ccccc2c1-c1ccccc1 ZINC000217608636 CI In-Stock Unstable TSPO 44 46 O=C(O)Cc1c(Cl)nc2ccccc2c1-c1ccccc1 ZINC000217608636 CI In-Stock Unstable TACR3 46 36 O=C(O)Cc1c(Cl)nc2ccccc2c1-c1ccccc1 ZINC000217608636 CI In-Stock Unstable PTGDR2 25 41 Cc1cccc(S(=O)(=O)Nc2ncc(/C=C\C(=O)O)s2)c1 ZINC000217608648 DE For-Sale Unstable FBP1 32 47 C[C@@H](NS(=O)(=O)c1ccc(NC2CC2)c(C(=O)O)c1)c1ccccc1 ZINC000217608690 FF In-Stock Unstable MMP13 19 41 C[C@@H](NS(=O)(=O)c1ccc(NC2CC2)c(C(=O)O)c1)c1ccccc1 ZINC000217608690 FF In-Stock Unstable MMP2 18 41 C[C@@H](NS(=O)(=O)c1ccc(NC2CC2)c(C(=O)O)c1)c1ccccc1 ZINC000217608690 FF In-Stock Unstable CCR8 42 33 COc1ccc(NC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217608699 FG For-Sale Unstable NPY5R 50 51 COc1ccc(NC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217608699 FG For-Sale Unstable EPHX2 38 44 COc1ccc(NC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217608699 FG For-Sale Unstable TRPM8 26 40 CN1CCCC[C@H]1CN[C@H](c1cccs1)C1CC1 ZINC000217608714 CG For-Sale Unstable CHRNA10 50 35 Cc1cccc(CNC(=O)NCC2CCCCC2)c1 ZINC000217608733 CG On-Demand Unstable GNRHR 0 43 C[C@@H](CNCCCc1ccccc1)N(C)C1CC1 ZINC000217608736 BF For-Sale Unstable SLC18A2 35 40 C[C@@H](CNCCCc1ccccc1)N(C)C1CC1 ZINC000217608736 BF For-Sale Unstable SIGMAR1 21 45 C[C@H](NS(=O)(=O)c1ccc(NC2CC2)c(C(=O)O)c1)c1ccccc1 ZINC000217608763 FF In-Stock Unstable MMP13 19 41 C[C@H](NS(=O)(=O)c1ccc(NC2CC2)c(C(=O)O)c1)c1ccccc1 ZINC000217608763 FF In-Stock Unstable MMP2 18 41 C[C@H](NS(=O)(=O)c1ccc(NC2CC2)c(C(=O)O)c1)c1ccccc1 ZINC000217608763 FF In-Stock Unstable CCR8 42 33 COc1ccc(NC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217608790 FG For-Sale Unstable NPY5R 50 51 COc1ccc(NC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217608790 FG For-Sale Unstable EPHX2 38 44 COc1ccc(NC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217608790 FG For-Sale Unstable TRPM8 26 40 C[C@H](CNCCCc1ccccc1)N(C)C1CC1 ZINC000217608818 BF For-Sale Unstable SLC18A2 35 40 C[C@H](CNCCCc1ccccc1)N(C)C1CC1 ZINC000217608818 BF For-Sale Unstable SIGMAR1 21 45 CC(C)NC(=O)N(C)Cc1ccc(/C=C\C(=O)O)cc1 ZINC000217608835 CE For-Sale Unstable NR1H4 36 46 O=C(NCc1cccc(F)c1)NCC1CCCCC1 ZINC000217608848 CG On-Demand Unstable GRIN2B 28 43 COC(=O)C1(N(C)C)CC1 ZINC000217608862 AC In-Stock Unstable CPT1 64 30 C[C@@H](NS(=O)(=O)c1ccc(NC2CCCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217608871 GH In-Stock Unstable BDKRB1 26 40 C[C@@H](NS(=O)(=O)c1ccc(NC2CCCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217608871 GH In-Stock Unstable CCR8 42 35 O=C(c1cccc(C(F)(F)F)c1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217608884 GE In-Stock Unstable BRAF 18 45 O=C(c1cccc(C(F)(F)F)c1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217608884 GE In-Stock Unstable MAP3K12 15 40 O=C(c1cccc(C(F)(F)F)c1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217608884 GE In-Stock Unstable SLC6A7 0 43 COc1ccc(CNC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217608889 FG For-Sale Unstable MMP13 15 41 COc1ccc(CNC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217608889 FG For-Sale Unstable NPY5R 28 45 CC(C)(C)OC(=O)N[C@@H](CC1CNC1)C(=O)O ZINC000217608900 BC For-Sale Unstable PAPA1_CARPA 53 44 CC(C)(C)OC(=O)N[C@@H](CC1CNC1)C(=O)O ZINC000217608900 BC For-Sale Unstable CTSK 22 44 CC(C)(C)OC(=O)N[C@@H](CC1CNC1)C(=O)O ZINC000217608900 BC For-Sale Unstable REN 42 39 CC(C)(C)OC(=O)N[C@@H](CC1CNC1)C(=O)O ZINC000217608900 BC For-Sale Unstable FPR1 50 47 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)COCC(=O)O ZINC000217608902 CD For-Sale Unstable TRPM8 20 53 C[C@H](NS(=O)(=O)c1ccc(NC2CCCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217608936 GH In-Stock Unstable BDKRB1 26 40 C[C@H](NS(=O)(=O)c1ccc(NC2CCCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217608936 GH In-Stock Unstable CCR8 42 35 O=C(NCc1cccc(Cl)c1)NCC1CCCCC1 ZINC000217608953 CH On-Demand Unstable GRIN2B 18 49 O=C(NCc1cccc(Cl)c1)NCC1CCCCC1 ZINC000217608953 CH On-Demand Unstable ROCK2 15 46 O=C(NCc1cccc(Cl)c1)NCC1CCCCC1 ZINC000217608953 CH On-Demand Unstable EPHX2 21 54 O=C(NCc1cccc(Cl)c1)NCC1CCCCC1 ZINC000217608953 CH On-Demand Unstable CACNA1I 52 42 O=C(CCCc1nc(-c2ccccc2)no1)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217608959 GG In-Stock Unstable HCAR2 18 41 CC(C)(C)OC(=O)N[C@H](CC1CNC1)C(=O)O ZINC000217608981 BC For-Sale Unstable PAPA1_CARPA 53 44 CC(C)(C)OC(=O)N[C@H](CC1CNC1)C(=O)O ZINC000217608981 BC For-Sale Unstable CTSK 22 44 CC(C)(C)OC(=O)N[C@H](CC1CNC1)C(=O)O ZINC000217608981 BC For-Sale Unstable REN 42 39 CC(C)(C)OC(=O)N[C@H](CC1CNC1)C(=O)O ZINC000217608981 BC For-Sale Unstable FPR1 50 47 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)COCC(=O)O ZINC000217608991 CD For-Sale Unstable TRPM8 20 53 COc1ccc(CNC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217608992 FG For-Sale Unstable MMP13 15 41 COc1ccc(CNC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217608992 FG For-Sale Unstable NPY5R 28 45 O=C(c1cc(=O)c2ccccc2o1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217608995 GD In-Stock Unstable PRKDC 58 38 O=C(CCC(=O)c1ccc(F)cc1)Nc1nc(-c2ccc3c(c2)CCO3)cs1 ZINC000217609032 GI On-Demand Unstable HDAC9 18 52 C[C@@H](NS(=O)(=O)c1ccc(NC2CCCCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217609046 HI In-Stock Unstable BDKRB1 26 41 C[C@@H](NS(=O)(=O)c1ccc(NC2CCCCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217609046 HI In-Stock Unstable CCR8 40 37 C[C@@H](NS(=O)(=O)c1ccc(NC2CCCCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217609046 HI In-Stock Unstable LEF 25 40 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)COCC(=O)O ZINC000217609069 CD For-Sale Unstable TRPM8 20 53 Cc1cccc(NC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217609085 EH For-Sale Unstable NPY5R 56 48 Cc1cccc(NC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217609085 EH For-Sale Unstable EPHX2 20 41 Cc1cccc(NC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217609085 EH For-Sale Unstable KCNK3 48 36 Cc1cccc(NC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217609085 EH For-Sale Unstable KCNK9 41 36 CC(C)COC(=O)N[C@@H](C)c1cccc(/C=C\C(=O)O)c1 ZINC000217609095 CG For-Sale Unstable AKR1C3 28 45 COC(=O)C1(CNC(C)=O)CC1 ZINC000217609096 AC In-Stock Unstable CPT1 72 33 O=C(c1cc2ccccc2oc1=O)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217609104 GD In-Stock Unstable PRKDC 15 44 O=C(c1cc2ccccc2oc1=O)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217609104 GD In-Stock Unstable HSP90AB1 0 46 O=C(c1cc2ccccc2oc1=O)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217609104 GD In-Stock Unstable SLC16A3 0 44 CC(C)(C)OC(=O)N1CCCN[C@H](C(=O)O)C1 ZINC000217609106 BC For-Sale Unstable GPR119 27 40 C[C@H](NS(=O)(=O)c1ccc(NC2CCCCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217609128 HI In-Stock Unstable BDKRB1 26 41 C[C@H](NS(=O)(=O)c1ccc(NC2CCCCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217609128 HI In-Stock Unstable CCR8 40 37 C[C@H](NS(=O)(=O)c1ccc(NC2CCCCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217609128 HI In-Stock Unstable LEF 25 40 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)COCC(=O)O ZINC000217609141 CD For-Sale Unstable TRPM8 20 53 Cc1cccc(NC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217609156 EH For-Sale Unstable NPY5R 56 48 Cc1cccc(NC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217609156 EH For-Sale Unstable EPHX2 20 41 Cc1cccc(NC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217609156 EH For-Sale Unstable KCNK3 48 36 Cc1cccc(NC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217609156 EH For-Sale Unstable KCNK9 41 36 O=C(NCc1ccc(Br)cc1)NCC1CCCCC1 ZINC000217609171 EH On-Demand Unstable TPSAB1 16 40 O=C(NCc1ccc(Br)cc1)NCC1CCCCC1 ZINC000217609171 EH On-Demand Unstable PROC 45 33 CC(C)COC(=O)N[C@H](C)c1cccc(/C=C\C(=O)O)c1 ZINC000217609175 CG For-Sale Unstable AKR1C3 28 45 CC(C)(C)OC(=O)N1CCCN[C@@H](C(=O)O)C1 ZINC000217609177 BC For-Sale Unstable GPR119 27 40 COc1cccc2cc(C(=O)N3Cc4cnc(N5CCOCC5)nc4C3)oc12 ZINC000217609209 GE In-Stock Unstable HSP90AB1 0 46 COc1ccc2c(c1)[C@@H](NC[C@@H]1CCCCN1C)CCO2 ZINC000217609216 CF For-Sale Unstable CHRNA10 63 42 Cc1ccc(NC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217609258 EH For-Sale Unstable NPY5R 56 53 Cc1ccc(NC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217609258 EH For-Sale Unstable EPHX2 35 50 Cc1ccc(NC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217609258 EH For-Sale Unstable TRPM8 25 44 Cc1ccc(S(=O)(=O)Nc2ncc(/C=C\C(=O)O)s2)cc1 ZINC000217609272 DE For-Sale Unstable CA1 16 44 Cc1ccc(S(=O)(=O)Nc2ncc(/C=C\C(=O)O)s2)cc1 ZINC000217609272 DE For-Sale Unstable CA4 29 44 NC/C=C\CN1CCc2ccccc2CC1 ZINC000217609281 BD For-Sale Unstable CHRNA6 0 46 COc1ccc2c(c1)[C@@H](NC[C@H]1CCCCN1C)CCO2 ZINC000217609287 CF For-Sale Unstable CHRNA10 63 42 Cc1ccccc1CCNC(=O)NCC1CCCCC1 ZINC000217609293 CG For-Sale Unstable MTNR1A 37 41 Cc1ccccc1CCNC(=O)NCC1CCCCC1 ZINC000217609293 CG For-Sale Unstable METAP2 0 42 O=C(/C=C/c1ccc2c(c1)OCO2)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217609307 GD In-Stock Unstable ITGAL 16 41 Cc1ccc(NC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217609334 EH For-Sale Unstable NPY5R 56 53 Cc1ccc(NC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217609334 EH For-Sale Unstable EPHX2 35 50 Cc1ccc(NC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217609334 EH For-Sale Unstable TRPM8 25 44 COc1ccccc1CCNC(=O)NCC1CCCCC1 ZINC000217609397 CG On-Demand Unstable DEF 0 40 COc1ccccc1CCNC(=O)NCC1CCCCC1 ZINC000217609397 CG On-Demand Unstable METAP2 26 43 C[C@@H](NS(=O)(=O)c1ccc(NCCO)c(C(=O)O)c1)c1ccccc1 ZINC000217609442 FD In-Stock Unstable BDKRB1 16 42 O=C(COC[C@@H]1CCCO1)NCc1nc(-c2ccccc2)n[nH]1 ZINC000217609451 DD In-Stock Unstable TNK2 43 35 O=C1O[C@@]2(CCCN(C(=O)NCCCc3ccccc3)C2)c2ccccc21 ZINC000217609456 FG For-Sale Unstable GHRHR 42 35 O=C1O[C@@]2(CCCN(C(=O)NCCCc3ccccc3)C2)c2ccccc21 ZINC000217609456 FG For-Sale Unstable NPY5R 31 45 O=C(NCCc1ccccc1F)NCC1CCCCC1 ZINC000217609499 CG On-Demand Unstable METAP2 0 42 O=C(N1Cc2cnc(N3CCOCC3)nc2C1)C1(c2ccc(Cl)cc2)CCCC1 ZINC000217609515 HG In-Stock Unstable AKR1C3 24 40 C[C@H](NS(=O)(=O)c1ccc(NCCO)c(C(=O)O)c1)c1ccccc1 ZINC000217609527 FD In-Stock Unstable BDKRB1 16 42 O=C(COC[C@H]1CCCO1)NCc1nc(-c2ccccc2)n[nH]1 ZINC000217609536 DD In-Stock Unstable TNK2 43 35 O=C(O)/C=C\c1cnc(NS(=O)(=O)c2ccc(F)cc2)s1 ZINC000217609539 EE For-Sale Anodyne PIK3C3 45 37 O=C1O[C@]2(CCCN(C(=O)NCCCc3ccccc3)C2)c2ccccc21 ZINC000217609540 FG For-Sale Unstable GHRHR 42 35 O=C1O[C@]2(CCCN(C(=O)NCCCc3ccccc3)C2)c2ccccc21 ZINC000217609540 FG For-Sale Unstable NPY5R 31 45 Cc1c(N)nc(C2CC2)nc1N[C@@H]1CC[C@@H](C)[C@@H](C)C1 ZINC000217609552 CG For-Sale Unstable CHRM3 0 54 CC(C)(CNC(=O)OCc1ccccc1)N=C=O ZINC000217609562 BE For-Sale Unstable CASP3 17 42 CC(C)(CNC(=O)OCc1ccccc1)N=C=O ZINC000217609562 BE For-Sale Unstable BMP1 43 34 CC(C)(CNC(=O)OCc1ccccc1)N=C=O ZINC000217609562 BE For-Sale Unstable KLK3 77 38 CC(C)(CNC(=O)OCc1ccccc1)N=C=O ZINC000217609562 BE For-Sale Unstable CTSB 61 39 CC(C)(CNC(=O)OCc1ccccc1)N=C=O ZINC000217609562 BE For-Sale Unstable PAPA1_CARPA 69 39 CC(C)(CNC(=O)OCc1ccccc1)N=C=O ZINC000217609562 BE For-Sale Unstable CYSP_TRYCR 57 41 CC(C)(CNC(=O)OCc1ccccc1)N=C=O ZINC000217609562 BE For-Sale Unstable CTSK 36 47 CC(C)(CNC(=O)OCc1ccccc1)N=C=O ZINC000217609562 BE For-Sale Unstable CTSL 41 47 CC(C)(CNC(=O)OCc1ccccc1)N=C=O ZINC000217609562 BE For-Sale Unstable CAPNS1 65 38 CC(C)(CNC(=O)OCc1ccccc1)N=C=O ZINC000217609562 BE For-Sale Unstable CTSS 25 47 CC(C)(CNC(=O)OCc1ccccc1)N=C=O ZINC000217609562 BE For-Sale Unstable CAPN1 86 42 CC(C)(CNC(=O)OCc1ccccc1)N=C=O ZINC000217609562 BE For-Sale Unstable CASP1 23 42 CC(C)(CNC(=O)OCc1ccccc1)N=C=O ZINC000217609562 BE For-Sale Unstable CAPN2 125 41 CC(C)(CNC(=O)OCc1ccccc1)N=C=O ZINC000217609562 BE For-Sale Unstable CASP6 23 42 CC(C)(CNC(=O)OCc1ccccc1)N=C=O ZINC000217609562 BE For-Sale Unstable CASP9 30 42 CC(C)(CNC(=O)OCc1ccccc1)N=C=O ZINC000217609562 BE For-Sale Unstable NPR 81 43 CC(C)(CNC(=O)OCc1ccccc1)N=C=O ZINC000217609562 BE For-Sale Unstable NAAA 22 40 CC(C)(CNC(=O)OCc1ccccc1)N=C=O ZINC000217609562 BE For-Sale Unstable PSMB5 38 40 COc1cc2c(cc1OC)CN(Cc1cc(=O)c(O)c(CN3CCN(C)CC3)o1)CC2 ZINC000217609567 ID In-Stock Unstable ABCB1B 64 36 COc1cc2c(cc1OC)CN(Cc1cc(=O)c(O)c(CN3CCN(C)CC3)o1)CC2 ZINC000217609567 ID In-Stock Unstable ABCB1 24 47 O=C(NCCc1ccccc1Cl)NCC1CCCCC1 ZINC000217609615 CH On-Demand Unstable P2RX7 17 42 O=C(NCCc1ccccc1Cl)NCC1CCCCC1 ZINC000217609615 CH On-Demand Unstable EPHX2 15 50 O=C(NCCc1ccccc1Cl)NCC1CCCCC1 ZINC000217609615 CH On-Demand Unstable METAP2 19 49 COCCOCC(=O)Nc1nc(-c2cc(C)n(CCc3ccccc3)c2C)cs1 ZINC000217609619 HI On-Demand Unstable MPL 42 33 COCCOCC(=O)Nc1nc(-c2cc(C)n(CCc3ccccc3)c2C)cs1 ZINC000217609619 HI On-Demand Unstable ROCK1 17 41 Cc1onc(-c2ccccc2Cl)c1C(=O)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217609631 IG In-Stock Unstable GPBAR1 28 41 Cc1c(N)nc(C2CC2)nc1N[C@H]1CC[C@@H](C)[C@@H](C)C1 ZINC000217609637 CG For-Sale Unstable CHRM3 0 54 C[C@@H](NS(=O)(=O)c1ccc(NCCCO)c(C(=O)O)c1)c1ccccc1 ZINC000217609649 GE In-Stock Unstable BDKRB1 18 43 O=C1O[C@@]2(CCCN(C(=O)Nc3ccc4c(c3)OCO4)C2)c2ccccc21 ZINC000217609650 FG For-Sale Unstable NPY5R 48 47 CC[C@@H]1C=CCN1C(=O)c1cccc(S(=O)(=O)N[C@@H]2CC[C@@H](O)CC2)c1 ZINC000217609653 GE In-Stock Unstable SFRP1 95 36 CC[C@@H]1C=CCN1C(=O)c1cccc(S(=O)(=O)N[C@@H]2CC[C@@H](O)CC2)c1 ZINC000217609653 GE In-Stock Unstable WNT3 54 35 C[C@@H](CN=C=O)N(C)C(=O)OCc1ccccc1 ZINC000217609685 BD For-Sale Unstable CTSB 58 44 C[C@@H](CN=C=O)N(C)C(=O)OCc1ccccc1 ZINC000217609685 BD For-Sale Unstable PAPA1_CARPA 61 43 C[C@@H](CN=C=O)N(C)C(=O)OCc1ccccc1 ZINC000217609685 BD For-Sale Unstable CTSK 15 44 C[C@@H](CN=C=O)N(C)C(=O)OCc1ccccc1 ZINC000217609685 BD For-Sale Unstable CTSL 26 43 C[C@@H](CN=C=O)N(C)C(=O)OCc1ccccc1 ZINC000217609685 BD For-Sale Unstable CAPNS1 48 35 C[C@@H](CN=C=O)N(C)C(=O)OCc1ccccc1 ZINC000217609685 BD For-Sale Unstable CAPN1 42 41 C[C@@H](CN=C=O)N(C)C(=O)OCc1ccccc1 ZINC000217609685 BD For-Sale Unstable CAPN2 74 36 C[C@@H](CN=C=O)N(C)C(=O)OCc1ccccc1 ZINC000217609685 BD For-Sale Unstable NPR 56 35 Cc1c(N)nc(C2CC2)nc1N[C@@H]1CC[C@H](C)[C@@H](C)C1 ZINC000217609715 CG For-Sale Unstable CHRM3 0 54 C[C@H](NS(=O)(=O)c1ccc(NCCCO)c(C(=O)O)c1)c1ccccc1 ZINC000217609719 GE In-Stock Unstable BDKRB1 18 43 O=C1O[C@]2(CCCN(C(=O)Nc3ccc4c(c3)OCO4)C2)c2ccccc21 ZINC000217609720 FG For-Sale Unstable NPY5R 48 47 CN1CCCC[C@@H]1CN[C@H](c1ccc(F)cc1)C1CC1 ZINC000217609735 CG For-Sale Unstable CHRNA10 59 38 CC[C@H]1C=CCN1C(=O)c1cccc(S(=O)(=O)N[C@@H]2CC[C@@H](O)CC2)c1 ZINC000217609737 GE In-Stock Unstable SFRP1 95 36 CC[C@H]1C=CCN1C(=O)c1cccc(S(=O)(=O)N[C@@H]2CC[C@@H](O)CC2)c1 ZINC000217609737 GE In-Stock Unstable WNT3 54 35 C[C@H](CN=C=O)N(C)C(=O)OCc1ccccc1 ZINC000217609775 BD For-Sale Unstable CTSB 58 44 C[C@H](CN=C=O)N(C)C(=O)OCc1ccccc1 ZINC000217609775 BD For-Sale Unstable PAPA1_CARPA 61 43 C[C@H](CN=C=O)N(C)C(=O)OCc1ccccc1 ZINC000217609775 BD For-Sale Unstable CTSK 15 44 C[C@H](CN=C=O)N(C)C(=O)OCc1ccccc1 ZINC000217609775 BD For-Sale Unstable CTSL 26 43 C[C@H](CN=C=O)N(C)C(=O)OCc1ccccc1 ZINC000217609775 BD For-Sale Unstable CAPNS1 48 35 C[C@H](CN=C=O)N(C)C(=O)OCc1ccccc1 ZINC000217609775 BD For-Sale Unstable CAPN1 42 41 C[C@H](CN=C=O)N(C)C(=O)OCc1ccccc1 ZINC000217609775 BD For-Sale Unstable CAPN2 74 36 C[C@H](CN=C=O)N(C)C(=O)OCc1ccccc1 ZINC000217609775 BD For-Sale Unstable NPR 56 35 Cc1c(N)nc(C2CC2)nc1N[C@H]1CC[C@H](C)[C@@H](C)C1 ZINC000217609807 CG For-Sale Unstable CHRM3 0 54 CN1CCCC[C@H]1CN[C@H](c1ccc(F)cc1)C1CC1 ZINC000217609824 CG For-Sale Unstable CHRNA10 59 38 COc1ccccc1NC(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217609830 FG For-Sale Unstable NPY5R 42 59 COCCNc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O ZINC000217609837 GE In-Stock Unstable KCNA5 0 40 COCCNc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O ZINC000217609837 GE In-Stock Unstable BDKRB1 17 44 COCCNc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O ZINC000217609837 GE In-Stock Unstable ADAMTS4 41 32 Cc1cccc(CCNC(=O)NCC2CCCCC2)c1 ZINC000217609852 CG On-Demand Unstable FAAH 15 45 C[C@@H](CN(C)C(=O)OCc1ccccc1)N=C=O ZINC000217609888 BD For-Sale Unstable KLK3 62 33 C[C@@H](CN(C)C(=O)OCc1ccccc1)N=C=O ZINC000217609888 BD For-Sale Unstable CTSB 47 40 C[C@@H](CN(C)C(=O)OCc1ccccc1)N=C=O ZINC000217609888 BD For-Sale Unstable PAPA1_CARPA 50 40 C[C@@H](CN(C)C(=O)OCc1ccccc1)N=C=O ZINC000217609888 BD For-Sale Unstable CTSL 25 40 C[C@@H](CN(C)C(=O)OCc1ccccc1)N=C=O ZINC000217609888 BD For-Sale Unstable CAPNS1 53 34 C[C@@H](CN(C)C(=O)OCc1ccccc1)N=C=O ZINC000217609888 BD For-Sale Unstable CAPN2 61 34 C[C@@H](CN(C)C(=O)OCc1ccccc1)N=C=O ZINC000217609888 BD For-Sale Unstable NPR 59 35 C[C@@H](CN(C)C(=O)OCc1ccccc1)N=C=O ZINC000217609888 BD For-Sale Unstable Q6PRC7_IXORI 41 32 COCCNc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O ZINC000217609919 GE In-Stock Unstable KCNA5 0 40 COCCNc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O ZINC000217609919 GE In-Stock Unstable BDKRB1 17 44 COCCNc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O ZINC000217609919 GE In-Stock Unstable ADAMTS4 41 32 COc1ccccc1NC(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217609924 FG For-Sale Unstable NPY5R 42 59 CC(C)COC(=O)N(C)Cc1ccc(/C=C\C(=O)O)cc1 ZINC000217609948 CG For-Sale Unstable AKR1C3 28 45 COc1cccc(CCNC(=O)NCC2CCCCC2)c1 ZINC000217609951 CG On-Demand Unstable TRPV1 0 40 C[C@H](CN(C)C(=O)OCc1ccccc1)N=C=O ZINC000217609959 BD For-Sale Unstable KLK3 62 33 C[C@H](CN(C)C(=O)OCc1ccccc1)N=C=O ZINC000217609959 BD For-Sale Unstable CTSB 47 40 C[C@H](CN(C)C(=O)OCc1ccccc1)N=C=O ZINC000217609959 BD For-Sale Unstable PAPA1_CARPA 50 40 C[C@H](CN(C)C(=O)OCc1ccccc1)N=C=O ZINC000217609959 BD For-Sale Unstable CTSL 25 40 C[C@H](CN(C)C(=O)OCc1ccccc1)N=C=O ZINC000217609959 BD For-Sale Unstable CAPNS1 53 34 C[C@H](CN(C)C(=O)OCc1ccccc1)N=C=O ZINC000217609959 BD For-Sale Unstable CAPN2 61 34 C[C@H](CN(C)C(=O)OCc1ccccc1)N=C=O ZINC000217609959 BD For-Sale Unstable NPR 59 35 C[C@H](CN(C)C(=O)OCc1ccccc1)N=C=O ZINC000217609959 BD For-Sale Unstable Q6PRC7_IXORI 41 32 CO[C@@H](CCO)C(=O)N1CCCCC1 ZINC000217609966 BC In-Stock Unstable DPP7 49 37 CN1CCCC[C@@H]1CN[C@H](c1cccs1)C1CCCC1 ZINC000217609995 CI For-Sale Unstable CHRNA10 50 35 COCCCNc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O ZINC000217610023 GF In-Stock Unstable BDKRB1 27 45 O=C(O)/C=C\c1cccc(NC(=O)Oc2ccccc2)c1 ZINC000217610035 CG For-Sale Anodyne HDAC8 19 44 O=C(O)/C=C\c1cccc(NC(=O)Oc2ccccc2)c1 ZINC000217610035 CG For-Sale Anodyne MMP2 0 51 O=C(O)/C=C\c1cccc(NC(=O)Oc2ccccc2)c1 ZINC000217610035 CG For-Sale Anodyne FAAH 19 50 O=C(O)/C=C\c1cccc(NC(=O)Oc2ccccc2)c1 ZINC000217610035 CG For-Sale Anodyne MMP9 0 51 O=C(O)/C=C\c1cccc(NC(=O)Oc2ccccc2)c1 ZINC000217610035 CG For-Sale Anodyne MMP1 0 49 O=C(O)/C=C\c1cccc(NC(=O)Oc2ccccc2)c1 ZINC000217610035 CG For-Sale Anodyne AKR1C3 49 38 O=C(O)/C=C\c1cccc(NC(=O)Oc2ccccc2)c1 ZINC000217610035 CG For-Sale Anodyne TRPM8 0 43 O=C(O)/C=C\c1cccc(NC(=O)Oc2ccccc2)c1 ZINC000217610035 CG For-Sale Anodyne RHOA 0 50 O=C(O)/C=C\c1cccc(NC(=O)Oc2ccccc2)c1 ZINC000217610035 CG For-Sale Anodyne PARP14 0 40 O=C(O)/C=C\c1cccc(NC(=O)Oc2ccccc2)c1 ZINC000217610035 CG For-Sale Anodyne KCNK3 82 38 O=C(O)/C=C\c1cccc(NC(=O)Oc2ccccc2)c1 ZINC000217610035 CG For-Sale Anodyne KCNK9 52 35 O=C(O)/C=C\c1cccc(NC(=O)Oc2ccccc2)c1 ZINC000217610035 CG For-Sale Anodyne PARP10 0 40 O=C1O[C@@]2(CCCN(C(=O)NCc3cccs3)C2)c2ccccc21 ZINC000217610037 EG In-Stock Unstable NPY5R 25 42 CO[C@H](CCO)C(=O)N1CCCCC1 ZINC000217610052 BC In-Stock Unstable DPP7 49 37 O=C(c1ccc(OC(F)(F)F)cc1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217610054 GE In-Stock Unstable SLC6A7 0 42 O=C(NCCc1cccc(F)c1)NCC1CCCCC1 ZINC000217610068 CG On-Demand Unstable CCR3 33 41 COc1ccc(CCN2C(=O)N[C@@H](CC(=O)N3CCc4cc(OC)c(OC)cc4C3)C2=O)cc1OC ZINC000217610073 JE In-Stock Unstable ABCB1B 45 40 COc1ccc(CCN2C(=O)N[C@@H](CC(=O)N3CCc4cc(OC)c(OC)cc4C3)C2=O)cc1OC ZINC000217610073 JE In-Stock Unstable MTNR1B 22 41 COc1ccc(CCN2C(=O)N[C@@H](CC(=O)N3CCc4cc(OC)c(OC)cc4C3)C2=O)cc1OC ZINC000217610073 JE In-Stock Unstable ABCB1 23 48 COc1ccc(CCN2C(=O)N[C@@H](CC(=O)N3CCc4cc(OC)c(OC)cc4C3)C2=O)cc1OC ZINC000217610073 JE In-Stock Unstable HCRTR2 17 42 COc1ccc(CCN2C(=O)N[C@@H](CC(=O)N3CCc4cc(OC)c(OC)cc4C3)C2=O)cc1OC ZINC000217610073 JE In-Stock Unstable ABCG2 33 43 COc1ccc(CCN2C(=O)N[C@@H](CC(=O)N3CCc4cc(OC)c(OC)cc4C3)C2=O)cc1OC ZINC000217610073 JE In-Stock Unstable HCN2 0 43 CC(C)(C)OC(=O)Nc1ccc(O)c(CC#N)c1 ZINC000217610083 BF For-Sale Unstable PAPA1_CARPA 48 38 CN1CCCC[C@H]1CN[C@H](c1cccs1)C1CCCC1 ZINC000217610091 CI For-Sale Unstable CHRNA10 50 35 COCCCNc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O ZINC000217610110 GF In-Stock Unstable BDKRB1 27 45 O=C1O[C@]2(CCCN(C(=O)NCc3cccs3)C2)c2ccccc21 ZINC000217610130 EG In-Stock Unstable NPY5R 25 42 COc1ccc(CN2C(=O)N[C@@H](CCC(=O)N[C@H](CO)c3ccccc3)C2=O)cc1 ZINC000217610172 HD In-Stock Unstable GHSR 16 40 COc1ccc(CN2C(=O)N[C@@H](CCC(=O)N[C@H](CO)c3ccccc3)C2=O)cc1 ZINC000217610172 HD In-Stock Unstable GPR88 0 47 O=C(c1ccc(-c2ccsc2)cc1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217610175 GG In-Stock Unstable PIK3CA 26 41 O=C(c1ccc(-c2ccsc2)cc1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217610175 GG In-Stock Unstable MTOR 45 45 O=C(c1ccc(-c2ccsc2)cc1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217610175 GG In-Stock Unstable PIK3CG 29 41 O=C(NCCc1cccc(Cl)c1)NCC1CCCCC1 ZINC000217610184 CH On-Demand Unstable EPHX2 21 52 O=C(NCCc1cccc(Cl)c1)NCC1CCCCC1 ZINC000217610184 CH On-Demand Unstable CACNA1I 51 41 O=C(NCCc1cccc(Cl)c1)NCC1CCCCC1 ZINC000217610184 CH On-Demand Unstable LMGT2 0 46 C[C@@H](NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1)c1ccccc1 ZINC000217610220 HI In-Stock Unstable TRY2_BOVIN 62 32 C[C@@H](NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1)c1ccccc1 ZINC000217610220 HI In-Stock Unstable BDKRB1 23 40 C[C@@H](NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1)c1ccccc1 ZINC000217610220 HI In-Stock Unstable ADAMTS4 50 36 C[C@@H](NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1)c1ccccc1 ZINC000217610220 HI In-Stock Unstable ACPS 0 41 COc1ccc(NC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c(OC)c1 ZINC000217610230 GG For-Sale Unstable NPY5R 46 55 Cn1cc(C(=O)N2CCC[C@@H]2c2nc3cc(F)ccc3[nH]2)c(=O)[nH]c1=O ZINC000217610258 FD In-Stock Unstable PRCP 51 42 COc1ccc(NC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c(OC)c1 ZINC000217610282 GG For-Sale Unstable NPY5R 46 55 COC(=O)C[C@H](c1cccc(O)c1)c1c(O)ccc2c(=O)c(-c3ccc(O)cc3)coc12 ZINC000217610291 II In-Stock Unstable ALDH2 102 42 C[C@H](NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1)c1ccccc1 ZINC000217610309 HI In-Stock Unstable TRY2_BOVIN 62 32 C[C@H](NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1)c1ccccc1 ZINC000217610309 HI In-Stock Unstable BDKRB1 23 40 C[C@H](NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1)c1ccccc1 ZINC000217610309 HI In-Stock Unstable ADAMTS4 50 36 C[C@H](NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1)c1ccccc1 ZINC000217610309 HI In-Stock Unstable ACPS 0 41 Cn1cc(C(=O)N2CCC[C@H]2c2nc3cc(F)ccc3[nH]2)c(=O)[nH]c1=O ZINC000217610338 FD In-Stock Unstable PRCP 51 42 C=CCOc1ccc(CN(C)C(=O)C(F)F)cc1 ZINC000217610377 CE For-Sale Unstable SHC 29 40 C=CCOc1ccc(CN(C)C(=O)C(F)F)cc1 ZINC000217610377 CE For-Sale Unstable LSS 37 40 COC(=O)C[C@@H](c1cccc(O)c1)c1c(O)ccc2c(=O)c(-c3ccc(O)cc3)coc12 ZINC000217610383 II In-Stock Unstable ALDH2 102 42 COc1ccc(CNC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1OC ZINC000217610398 GG For-Sale Unstable NPY5R 25 47 Cc1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217610408 CG On-Demand Unstable MMP2 66 42 Cc1ccc(CCNC(=O)NCC2CCCCC2)cc1 ZINC000217610408 CG On-Demand Unstable GPBAR1 0 43 C[C@H](NS(=O)(=O)c1ccc(N[C@H](C)c2ccccc2)c(C(=O)O)c1)c1ccccc1 ZINC000217610412 HJ In-Stock Unstable MMP13 26 40 C[C@H](NS(=O)(=O)c1ccc(N[C@H](C)c2ccccc2)c(C(=O)O)c1)c1ccccc1 ZINC000217610412 HJ In-Stock Unstable BDKRB1 17 40 C[C@H](NS(=O)(=O)c1ccc(N[C@H](C)c2ccccc2)c(C(=O)O)c1)c1ccccc1 ZINC000217610412 HJ In-Stock Unstable MMP2 20 40 C[C@H](NS(=O)(=O)c1ccc(N[C@H](C)c2ccccc2)c(C(=O)O)c1)c1ccccc1 ZINC000217610412 HJ In-Stock Unstable MMP12 46 39 C[C@H](NS(=O)(=O)c1ccc(N[C@H](C)c2ccccc2)c(C(=O)O)c1)c1ccccc1 ZINC000217610412 HJ In-Stock Unstable LEF 36 43 O=C(CCc1ccc(OCc2ccccc2)cc1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217610420 IG In-Stock Unstable FAAH 22 41 O=C(CCc1ccc(OCc2ccccc2)cc1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217610420 IG In-Stock Unstable ABCB1 0 41 O=C(CCc1ccc(OCc2ccccc2)cc1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217610420 IG In-Stock Unstable FFAR1 25 43 O=C(O)CCCCCN1C(=O)[C@@H]2[C@@H]3C[C@@H]([C@H]4Sc5[nH]c(=O)sc5[C@H](c5cccnc5)[C@H]34)[C@@H]2C1=O ZINC000217610425 JF In-Stock Unstable TBXAS1 24 41 CNC(=O)[C@@H](CC(C)C)N[C@@H]1CCCC[C@@H]1C ZINC000217610441 BE For-Sale Unstable MMP1 0 41 COc1ccc(CNC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1OC ZINC000217610469 GG For-Sale Unstable NPY5R 25 47 C[C@H](Nc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217610475 HJ In-Stock Unstable MMP13 26 40 C[C@H](Nc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217610475 HJ In-Stock Unstable BDKRB1 17 40 C[C@H](Nc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217610475 HJ In-Stock Unstable MMP2 20 40 C[C@H](Nc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217610475 HJ In-Stock Unstable MMP12 46 39 C[C@H](Nc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217610475 HJ In-Stock Unstable LEF 36 43 O=C(NCCc1ccc(Cl)cc1)NCC1CCCCC1 ZINC000217610507 CH On-Demand Unstable CNR1 15 47 O=C(NCCc1ccc(Cl)cc1)NCC1CCCCC1 ZINC000217610507 CH On-Demand Unstable MMP2 55 41 O=C(NCCc1ccc(Cl)cc1)NCC1CCCCC1 ZINC000217610507 CH On-Demand Unstable MMP3 18 44 O=C(NCCc1ccc(Cl)cc1)NCC1CCCCC1 ZINC000217610507 CH On-Demand Unstable CACNA1I 57 36 O=C(O)CCCCCN1C(=O)[C@@H]2[C@@H]3C[C@@H]([C@H]4Sc5[nH]c(=O)sc5[C@H](c5cccnc5)[C@@H]34)[C@@H]2C1=O ZINC000217610510 JF In-Stock Unstable TBXAS1 24 41 CNC(=O)[C@@H](CC(C)C)N[C@H]1CCCC[C@@H]1C ZINC000217610526 BE For-Sale Unstable MMP1 0 41 O=C(O)/C=C\c1cccc(NC(=O)NC2CCCCC2)c1 ZINC000217610527 CG For-Sale Unstable FAAH 15 43 O=C(O)/C=C\c1cccc(NC(=O)NC2CCCCC2)c1 ZINC000217610527 CG For-Sale Unstable EPHX2 51 62 O=C(O)/C=C\c1cccc(NC(=O)NC2CCCCC2)c1 ZINC000217610527 CG For-Sale Unstable MMP1 0 42 C[C@@H](Nc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217610562 HJ In-Stock Unstable MMP13 26 40 C[C@@H](Nc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217610562 HJ In-Stock Unstable BDKRB1 17 40 C[C@@H](Nc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217610562 HJ In-Stock Unstable MMP2 20 40 C[C@@H](Nc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217610562 HJ In-Stock Unstable MMP12 46 39 C[C@@H](Nc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217610562 HJ In-Stock Unstable LEF 36 43 COc1cccc(NC(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1OC ZINC000217610575 GG For-Sale Unstable NPY5R 33 57 O=C(O)CCCCCN1C(=O)[C@@H]2[C@@H]3C[C@@H]([C@H]4Sc5[nH]c(=O)sc5[C@@H](c5cccnc5)[C@H]34)[C@@H]2C1=O ZINC000217610591 JF In-Stock Unstable TBXAS1 24 41 O=C(NCCc1ccc(Br)cc1)NCC1CCCCC1 ZINC000217610602 EH For-Sale Unstable MMP2 50 37 O=C(O)/C=C\c1cccc(NC(=O)Nc2ccccc2)c1 ZINC000217610613 CG For-Sale Anodyne EPHX1 0 55 O=C(O)/C=C\c1cccc(NC(=O)Nc2ccccc2)c1 ZINC000217610613 CG For-Sale Anodyne LPL 42 39 O=C(O)/C=C\c1cccc(NC(=O)Nc2ccccc2)c1 ZINC000217610613 CG For-Sale Anodyne CA1 31 41 O=C(O)/C=C\c1cccc(NC(=O)Nc2ccccc2)c1 ZINC000217610613 CG For-Sale Anodyne CCKAR 16 45 O=C(O)/C=C\c1cccc(NC(=O)Nc2ccccc2)c1 ZINC000217610613 CG For-Sale Anodyne HDAC8 40 52 O=C(O)/C=C\c1cccc(NC(=O)Nc2ccccc2)c1 ZINC000217610613 CG For-Sale Anodyne MMP2 22 57 O=C(O)/C=C\c1cccc(NC(=O)Nc2ccccc2)c1 ZINC000217610613 CG For-Sale Anodyne HDAC1 16 49 O=C(O)/C=C\c1cccc(NC(=O)Nc2ccccc2)c1 ZINC000217610613 CG For-Sale Anodyne HDAC6 30 52 O=C(O)/C=C\c1cccc(NC(=O)Nc2ccccc2)c1 ZINC000217610613 CG For-Sale Anodyne MMP9 22 57 O=C(O)/C=C\c1cccc(NC(=O)Nc2ccccc2)c1 ZINC000217610613 CG For-Sale Anodyne EPHX2 17 55 O=C(O)/C=C\c1cccc(NC(=O)Nc2ccccc2)c1 ZINC000217610613 CG For-Sale Anodyne CA12 15 49 O=C(O)/C=C\c1cccc(NC(=O)Nc2ccccc2)c1 ZINC000217610613 CG For-Sale Anodyne IMPDH2 0 46 O=C(O)/C=C\c1cccc(NC(=O)Nc2ccccc2)c1 ZINC000217610613 CG For-Sale Anodyne MMP1 27 54 O=C(O)/C=C\c1cccc(NC(=O)Nc2ccccc2)c1 ZINC000217610613 CG For-Sale Anodyne AKR1C3 53 38 O=C(O)/C=C\c1cccc(NC(=O)Nc2ccccc2)c1 ZINC000217610613 CG For-Sale Anodyne MTCA1 26 41 O=C(O)/C=C\c1cccc(NC(=O)Nc2ccccc2)c1 ZINC000217610613 CG For-Sale Anodyne P96878_MYCTU 30 41 O=C(O)/C=C\c1cccc(NC(=O)Nc2ccccc2)c1 ZINC000217610613 CG For-Sale Anodyne RHOA 0 56 O=C(O)/C=C\c1cccc(NC(=O)Nc2ccccc2)c1 ZINC000217610613 CG For-Sale Anodyne P95276_MYCTO 0 55 O=C(O)/C=C\c1cccc(NC(=O)Nc2ccccc2)c1 ZINC000217610613 CG For-Sale Anodyne PARP14 0 44 O=C(O)/C=C\c1cccc(NC(=O)Nc2ccccc2)c1 ZINC000217610613 CG For-Sale Anodyne KCNK3 96 39 O=C(O)/C=C\c1cccc(NC(=O)Nc2ccccc2)c1 ZINC000217610613 CG For-Sale Anodyne KCNK9 54 39 O=C(O)/C=C\c1cccc(NC(=O)Nc2ccccc2)c1 ZINC000217610613 CG For-Sale Anodyne PARP10 0 44 C[C@H](Nc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217610636 HJ In-Stock Unstable MMP13 26 40 C[C@H](Nc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217610636 HJ In-Stock Unstable BDKRB1 17 40 C[C@H](Nc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217610636 HJ In-Stock Unstable MMP2 20 40 C[C@H](Nc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217610636 HJ In-Stock Unstable MMP12 46 39 C[C@H](Nc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217610636 HJ In-Stock Unstable LEF 36 43 COc1cccc(NC(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1OC ZINC000217610664 GG For-Sale Unstable NPY5R 33 57 CNC(=O)[C@@H](CC(C)C)N[C@@H]1CCC[C@@H](C)C1 ZINC000217610673 BE For-Sale Unstable MMP1 15 45 O=C(O)CCCCCN1C(=O)[C@@H]2[C@@H]3C[C@@H]([C@H]4Sc5[nH]c(=O)sc5[C@@H](c5cccnc5)[C@@H]34)[C@@H]2C1=O ZINC000217610682 JF In-Stock Unstable TBXAS1 24 41 Cc1ccc(NC(=O)NCC2CCCCC2)cn1 ZINC000217610708 BG On-Demand Unstable PRMT3 34 41 C[C@@H](NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1)c1ccccc1 ZINC000217610745 HI In-Stock Unstable ADRB1 29 40 C[C@@H](NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1)c1ccccc1 ZINC000217610745 HI In-Stock Unstable ADRB3 52 40 C[C@@H](NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1)c1ccccc1 ZINC000217610745 HI In-Stock Unstable MMP13 22 41 C[C@@H](NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1)c1ccccc1 ZINC000217610745 HI In-Stock Unstable TRY2_BOVIN 56 32 C[C@@H](NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1)c1ccccc1 ZINC000217610745 HI In-Stock Unstable BDKRB1 18 41 C[C@@H](NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1)c1ccccc1 ZINC000217610745 HI In-Stock Unstable MMP2 24 41 C[C@@H](NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1)c1ccccc1 ZINC000217610745 HI In-Stock Unstable MMP8 16 41 C[C@@H](NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1)c1ccccc1 ZINC000217610745 HI In-Stock Unstable ADAMTS4 44 33 CNC(=O)[C@@H](CC(C)C)N[C@H]1CCC[C@@H](C)C1 ZINC000217610754 BE For-Sale Unstable MMP1 15 45 CCS(=O)(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217610774 CD For-Sale Unstable NPY5R 30 40 Cc1ccc(NC(=O)NCC2CCCCC2)nc1 ZINC000217610804 BG On-Demand Unstable GYRB 0 40 Cc1ccc(NC(=O)NCC2CCCCC2)nc1 ZINC000217610804 BG On-Demand Unstable GCK 32 47 Cc1ccc(NC(=O)NCC2CCCCC2)nc1 ZINC000217610804 BG On-Demand Unstable LUCI_LUCLA 23 43 C[C@H](NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1)c1ccccc1 ZINC000217610831 HI In-Stock Unstable ADRB1 29 40 C[C@H](NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1)c1ccccc1 ZINC000217610831 HI In-Stock Unstable ADRB3 52 40 C[C@H](NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1)c1ccccc1 ZINC000217610831 HI In-Stock Unstable MMP13 22 41 C[C@H](NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1)c1ccccc1 ZINC000217610831 HI In-Stock Unstable TRY2_BOVIN 56 32 C[C@H](NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1)c1ccccc1 ZINC000217610831 HI In-Stock Unstable BDKRB1 18 41 C[C@H](NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1)c1ccccc1 ZINC000217610831 HI In-Stock Unstable MMP2 24 41 C[C@H](NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1)c1ccccc1 ZINC000217610831 HI In-Stock Unstable MMP8 16 41 C[C@H](NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1)c1ccccc1 ZINC000217610831 HI In-Stock Unstable ADAMTS4 44 33 COc1ccccc1[C@@H](C)NC(=O)C(F)F ZINC000217610854 BE On-Demand Unstable KCNK3 39 43 COc1ccccc1[C@@H](C)NC(=O)C(F)F ZINC000217610854 BE On-Demand Unstable KCNK9 35 43 CCS(=O)(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217610858 CD For-Sale Unstable NPY5R 30 40 COc1ccc([C@@H](NC[C@@H]2CCCCN2C)C2CC2)cc1 ZINC000217610886 CG For-Sale Unstable CHRNA10 65 42 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217610936 JI In-Stock Unstable ADRB1 43 40 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217610936 JI In-Stock Unstable ADRB3 60 40 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217610936 JI In-Stock Unstable BMP1 86 45 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217610936 JI In-Stock Unstable KCNA5 26 41 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217610936 JI In-Stock Unstable MMP13 69 43 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217610936 JI In-Stock Unstable TRY2_BOVIN 41 34 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217610936 JI In-Stock Unstable BDKRB1 17 42 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217610936 JI In-Stock Unstable MMP2 51 41 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217610936 JI In-Stock Unstable MMP3 45 41 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217610936 JI In-Stock Unstable MMP8 31 43 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217610936 JI In-Stock Unstable PRTN3 44 31 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217610936 JI In-Stock Unstable MMP9 53 43 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217610936 JI In-Stock Unstable MMP12 41 40 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217610936 JI In-Stock Unstable PTGDR 27 40 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217610936 JI In-Stock Unstable ADAMTS4 63 38 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217610936 JI In-Stock Unstable CA9 21 40 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217610936 JI In-Stock Unstable MMP1 47 40 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217610936 JI In-Stock Unstable AKR1C2 49 35 COc1ccccc1[C@H](C)NC(=O)C(F)F ZINC000217610941 BE On-Demand Unstable KCNK3 39 43 COc1ccccc1[C@H](C)NC(=O)C(F)F ZINC000217610941 BE On-Demand Unstable KCNK9 35 43 COc1cccc(C(=O)NCC(=O)Nc2nc(CN3CCC[C@@H](C)C3)cs2)c1 ZINC000217610948 HF On-Demand Unstable DRD4 51 40 COc1cccc(C(=O)NCC(=O)Nc2nc(CN3CCC[C@@H](C)C3)cs2)c1 ZINC000217610948 HF On-Demand Unstable CCR3 17 42 COc1cccc(C(=O)NCC(=O)Nc2nc(CN3CCC[C@@H](C)C3)cs2)c1 ZINC000217610948 HF On-Demand Unstable CCR2 38 44 COc1ccc([C@@H](NC[C@H]2CCCCN2C)C2CC2)cc1 ZINC000217610986 CG For-Sale Unstable CHRNA10 65 42 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217611012 JI In-Stock Unstable ADRB1 43 40 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217611012 JI In-Stock Unstable ADRB3 60 40 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217611012 JI In-Stock Unstable BMP1 86 45 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217611012 JI In-Stock Unstable KCNA5 26 41 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217611012 JI In-Stock Unstable MMP13 69 43 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217611012 JI In-Stock Unstable TRY2_BOVIN 41 34 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217611012 JI In-Stock Unstable BDKRB1 17 42 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217611012 JI In-Stock Unstable MMP2 51 41 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217611012 JI In-Stock Unstable MMP3 45 41 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217611012 JI In-Stock Unstable MMP8 31 43 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217611012 JI In-Stock Unstable PRTN3 44 31 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217611012 JI In-Stock Unstable MMP9 53 43 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217611012 JI In-Stock Unstable MMP12 41 40 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217611012 JI In-Stock Unstable PTGDR 27 40 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217611012 JI In-Stock Unstable ADAMTS4 63 38 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217611012 JI In-Stock Unstable CA9 21 40 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217611012 JI In-Stock Unstable MMP1 47 40 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@H](C)c3ccccc3)cc2C(=O)O)cc1 ZINC000217611012 JI In-Stock Unstable AKR1C2 49 35 COc1cccc(C(=O)NCC(=O)Nc2nc(CN3CCC[C@H](C)C3)cs2)c1 ZINC000217611037 HF On-Demand Unstable DRD4 51 40 COc1cccc(C(=O)NCC(=O)Nc2nc(CN3CCC[C@H](C)C3)cs2)c1 ZINC000217611037 HF On-Demand Unstable CCR3 17 42 COc1cccc(C(=O)NCC(=O)Nc2nc(CN3CCC[C@H](C)C3)cs2)c1 ZINC000217611037 HF On-Demand Unstable CCR2 38 44 CNC(=O)[C@@H](CC(C)C)N[C@@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217611066 CG For-Sale Unstable TRPM8 15 43 CC(C)Cc1ccc([C@@H](C)NC(=O)C(F)F)cc1 ZINC000217611068 CG On-Demand Unstable MME 64 38 CC(C)Cc1ccc([C@@H](C)NC(=O)C(F)F)cc1 ZINC000217611068 CG On-Demand Unstable ACACA 51 38 CC(C)Cc1ccc([C@@H](C)NC(=O)C(F)F)cc1 ZINC000217611068 CG On-Demand Unstable CAPNS1 51 31 CC(C)Cc1ccc([C@@H](C)NC(=O)C(F)F)cc1 ZINC000217611068 CG On-Demand Unstable ACE2 55 35 CC(C)Cc1ccc([C@@H](C)NC(=O)C(F)F)cc1 ZINC000217611068 CG On-Demand Unstable SLC22A20 0 51 CN1CCCC[C@@H]1CN[C@H](c1ccc(Cl)cc1)C1CC1 ZINC000217611114 CH For-Sale Unstable CHRNA10 55 45 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@@H](C)c3ccccc3)cc2C(=O)O)cc1OC ZINC000217611126 JI In-Stock Unstable ADRB3 46 39 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@@H](C)c3ccccc3)cc2C(=O)O)cc1OC ZINC000217611126 JI In-Stock Unstable BDKRB1 19 40 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@@H](C)c3ccccc3)cc2C(=O)O)cc1OC ZINC000217611126 JI In-Stock Unstable ADAMTS4 47 35 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@@H](C)c3ccccc3)cc2C(=O)O)cc1OC ZINC000217611126 JI In-Stock Unstable SCMU_MYCTU 0 43 O=C(NCC1CCCCC1)Nc1ccc(Cl)cn1 ZINC000217611129 CG On-Demand Unstable F10 53 34 O=C(NCC1CCCCC1)Nc1ccc(Cl)cn1 ZINC000217611129 CG On-Demand Unstable GCK 22 43 CNC(=O)[C@@H](CC(C)C)N[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217611139 CG For-Sale Unstable TRPM8 15 43 COc1ccccc1C(=O)NCC(=O)Nc1nc(CN2CCC[C@@H](C)C2)cs1 ZINC000217611149 HF On-Demand Unstable KCNA3 41 36 COc1ccccc1C(=O)NCC(=O)Nc1nc(CN2CCC[C@@H](C)C2)cs1 ZINC000217611149 HF On-Demand Unstable HCN1 48 36 COc1ccccc1C(=O)NCC(=O)Nc1nc(CN2CCC[C@@H](C)C2)cs1 ZINC000217611149 HF On-Demand Unstable HCN4 42 35 CC(C)Cc1ccc([C@H](C)NC(=O)C(F)F)cc1 ZINC000217611154 CG On-Demand Unstable MME 64 38 CC(C)Cc1ccc([C@H](C)NC(=O)C(F)F)cc1 ZINC000217611154 CG On-Demand Unstable ACACA 51 38 CC(C)Cc1ccc([C@H](C)NC(=O)C(F)F)cc1 ZINC000217611154 CG On-Demand Unstable CAPNS1 51 31 CC(C)Cc1ccc([C@H](C)NC(=O)C(F)F)cc1 ZINC000217611154 CG On-Demand Unstable ACE2 55 35 CC(C)Cc1ccc([C@H](C)NC(=O)C(F)F)cc1 ZINC000217611154 CG On-Demand Unstable SLC22A20 0 51 CN1CCCC[C@H]1CN[C@H](c1ccc(Cl)cc1)C1CC1 ZINC000217611194 CH For-Sale Unstable CHRNA10 55 45 O=C(CCc1cccc(Oc2ccc(F)cc2)c1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217611203 IH In-Stock Unstable BRS3 20 44 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@H](C)c3ccccc3)cc2C(=O)O)cc1OC ZINC000217611212 JI In-Stock Unstable ADRB3 46 39 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@H](C)c3ccccc3)cc2C(=O)O)cc1OC ZINC000217611212 JI In-Stock Unstable BDKRB1 19 40 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@H](C)c3ccccc3)cc2C(=O)O)cc1OC ZINC000217611212 JI In-Stock Unstable ADAMTS4 47 35 COc1ccc(CCNc2ccc(S(=O)(=O)N[C@H](C)c3ccccc3)cc2C(=O)O)cc1OC ZINC000217611212 JI In-Stock Unstable SCMU_MYCTU 0 43 COc1ccccc1C(=O)NCC(=O)Nc1nc(CN2CCC[C@H](C)C2)cs1 ZINC000217611229 HF On-Demand Unstable KCNA3 41 36 COc1ccccc1C(=O)NCC(=O)Nc1nc(CN2CCC[C@H](C)C2)cs1 ZINC000217611229 HF On-Demand Unstable HCN1 48 36 COc1ccccc1C(=O)NCC(=O)Nc1nc(CN2CCC[C@H](C)C2)cs1 ZINC000217611229 HF On-Demand Unstable HCN4 42 35 CNC(=O)[C@H](CC(C)C)N[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217611236 CG For-Sale Unstable TRPM8 15 43 CC(=O)Nc1cccc2c1ccn2CC(=O)NCCc1ccc(O)cc1 ZINC000217611237 FF In-Stock Unstable NR5A1 24 42 O=C(NCC1CCCCC1)Nc1cc(Cl)ccn1 ZINC000217611247 CG For-Sale Unstable EPHX2 15 63 O=C(NCC1CCCCC1)Nc1cc(Cl)ccn1 ZINC000217611247 CG For-Sale Unstable TYK2 62 38 O=C(NCC1CCCCC1)Nc1cc(Cl)ccn1 ZINC000217611247 CG For-Sale Unstable CACNA1I 55 35 COC(=O)[C@@H](O)[C@H](O)Cc1ccccc1 ZINC000217611304 BC For-Sale Unstable ACE 43 40 COC(=O)[C@@H](O)[C@H](O)Cc1ccccc1 ZINC000217611304 BC For-Sale Unstable PPARA 15 40 COC(=O)[C@@H](O)[C@H](O)Cc1ccccc1 ZINC000217611304 BC For-Sale Unstable MME 104 44 COC(=O)[C@@H](O)[C@H](O)Cc1ccccc1 ZINC000217611304 BC For-Sale Unstable LTA4H 20 44 COC(=O)[C@@H](O)[C@H](O)Cc1ccccc1 ZINC000217611304 BC For-Sale Unstable ANPEP 88 36 COC(=O)[C@@H](O)[C@H](O)Cc1ccccc1 ZINC000217611304 BC For-Sale Unstable CTSD 19 40 COC(=O)[C@@H](O)[C@H](O)Cc1ccccc1 ZINC000217611304 BC For-Sale Unstable FCER2 69 36 COC(=O)[C@@H](O)[C@H](O)Cc1ccccc1 ZINC000217611304 BC For-Sale Unstable CTSB 49 40 COC(=O)[C@@H](O)[C@H](O)Cc1ccccc1 ZINC000217611304 BC For-Sale Unstable PAPA1_CARPA 63 42 COC(=O)[C@@H](O)[C@H](O)Cc1ccccc1 ZINC000217611304 BC For-Sale Unstable CYSP_TRYCR 50 38 COC(=O)[C@@H](O)[C@H](O)Cc1ccccc1 ZINC000217611304 BC For-Sale Unstable CPA1 71 43 COC(=O)[C@@H](O)[C@H](O)Cc1ccccc1 ZINC000217611304 BC For-Sale Unstable CTRB1 38 43 COC(=O)[C@@H](O)[C@H](O)Cc1ccccc1 ZINC000217611304 BC For-Sale Unstable CAPNS1 58 39 COC(=O)[C@@H](O)[C@H](O)Cc1ccccc1 ZINC000217611304 BC For-Sale Unstable HLA-DRB1 43 31 COC(=O)[C@@H](O)[C@H](O)Cc1ccccc1 ZINC000217611304 BC For-Sale Unstable PTPRB 21 40 COC(=O)[C@@H](O)[C@H](O)Cc1ccccc1 ZINC000217611304 BC For-Sale Unstable CTSS 23 43 COC(=O)[C@@H](O)[C@H](O)Cc1ccccc1 ZINC000217611304 BC For-Sale Unstable CAPN1 71 42 COC(=O)[C@@H](O)[C@H](O)Cc1ccccc1 ZINC000217611304 BC For-Sale Unstable CAPN2 60 37 COC(=O)[C@@H](O)[C@H](O)Cc1ccccc1 ZINC000217611304 BC For-Sale Unstable ACE2 66 39 COC(=O)[C@@H](O)[C@H](O)Cc1ccccc1 ZINC000217611304 BC For-Sale Unstable LAP3 55 47 COC(=O)[C@@H](O)[C@H](O)Cc1ccccc1 ZINC000217611304 BC For-Sale Unstable MMP1 22 43 COC(=O)[C@@H](O)[C@H](O)Cc1ccccc1 ZINC000217611304 BC For-Sale Unstable FPR1 42 38 COC(=O)[C@@H](O)[C@H](O)Cc1ccccc1 ZINC000217611304 BC For-Sale Unstable NPR 54 48 COC(=O)[C@@H](O)[C@H](O)Cc1ccccc1 ZINC000217611304 BC For-Sale Unstable AMP1_PLAFQ 63 44 COC(=O)[C@@H](O)[C@H](O)Cc1ccccc1 ZINC000217611304 BC For-Sale Unstable KIF11 18 43 COC(=O)[C@@H](O)[C@H](O)Cc1ccccc1 ZINC000217611304 BC For-Sale Unstable NPFFR1 43 33 COC(=O)[C@@H](O)[C@H](O)Cc1ccccc1 ZINC000217611304 BC For-Sale Unstable PDS 41 34 COC(=O)[C@@H](O)[C@H](O)Cc1ccccc1 ZINC000217611304 BC For-Sale Unstable H9B8T9_CAPHI 21 40 CC(C)CS(=O)(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217611368 DE For-Sale Unstable NPY5R 24 40 CN(Cc1ccc(C(F)(F)F)cc1)C(=O)C(F)F ZINC000217611409 CF On-Demand Unstable TACR1 22 51 CN(Cc1ccc(C(F)(F)F)cc1)C(=O)C(F)F ZINC000217611409 CF On-Demand Unstable MTTP 27 46 CN(Cc1ccc(C(F)(F)F)cc1)C(=O)C(F)F ZINC000217611409 CF On-Demand Unstable MLYCD 23 43 Cc1ccc2cccc(C(=O)N3Cc4cnc(N5CCOCC5)nc4C3)c2n1 ZINC000217611430 GE In-Stock Unstable HSP90AB1 0 43 CC(C)CS(=O)(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217611456 DE For-Sale Unstable NPY5R 24 40 O=C(NCCCc1ccccc1)NCC1CCCCC1 ZINC000217611482 CG On-Demand Unstable DEF 0 45 O=C(NCCCc1ccccc1)NCC1CCCCC1 ZINC000217611482 CG On-Demand Unstable MMP2 48 34 C[C@@H](NS(=O)(=O)c1ccc(NC[C@@H]2CCCO2)c(C(=O)O)c1)c1ccccc1 ZINC000217611529 HG In-Stock Unstable BDKRB1 28 40 C[C@@H](NS(=O)(=O)c1ccc(NC[C@@H]2CCCO2)c(C(=O)O)c1)c1ccccc1 ZINC000217611529 HG In-Stock Unstable TNK2 45 39 C[C@@H](NS(=O)(=O)c1ccc(NC[C@@H]2CCCO2)c(C(=O)O)c1)c1ccccc1 ZINC000217611529 HG In-Stock Unstable CCR8 43 31 CN(C[C@@H]1COc2ccccc2O1)C(=O)C(F)F ZINC000217611533 CD On-Demand Unstable ADRA2B 17 41 O=C(c1ccc(-c2cccs2)cc1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217611539 GG In-Stock Unstable PIK3CA 22 43 O=C(c1ccc(-c2cccs2)cc1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217611539 GG In-Stock Unstable MTOR 41 44 O=C(c1ccc(-c2cccs2)cc1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217611539 GG In-Stock Unstable PIK3CG 26 43 O=C(NCCCCc1ccccc1)NCC1CCCCC1 ZINC000217611596 CH For-Sale Unstable FKBP1A 45 49 O=C(NCCCCc1ccccc1)NCC1CCCCC1 ZINC000217611596 CH For-Sale Unstable HRH2 34 40 O=C(NCCCCc1ccccc1)NCC1CCCCC1 ZINC000217611596 CH For-Sale Unstable GRIN2B 31 42 O=C(NCCCCc1ccccc1)NCC1CCCCC1 ZINC000217611596 CH For-Sale Unstable SIGMAR1 21 44 O=C(NCCCCc1ccccc1)NCC1CCCCC1 ZINC000217611596 CH For-Sale Unstable CCR3 23 46 O=C(NCCCCc1ccccc1)NCC1CCCCC1 ZINC000217611596 CH For-Sale Unstable SCN2A 18 40 O=C(NCCCCc1ccccc1)NCC1CCCCC1 ZINC000217611596 CH For-Sale Unstable PREP 54 38 O=C(NCCCCc1ccccc1)NCC1CCCCC1 ZINC000217611596 CH For-Sale Unstable MTNR1A 31 42 O=C(NCCCCc1ccccc1)NCC1CCCCC1 ZINC000217611596 CH For-Sale Unstable MTNR1B 42 42 O=C(NCCCCc1ccccc1)NCC1CCCCC1 ZINC000217611596 CH For-Sale Unstable MMP2 52 43 O=C(NCCCCc1ccccc1)NCC1CCCCC1 ZINC000217611596 CH For-Sale Unstable MMP3 23 46 O=C(NCCCCc1ccccc1)NCC1CCCCC1 ZINC000217611596 CH For-Sale Unstable REN 32 40 O=C(NCCCCc1ccccc1)NCC1CCCCC1 ZINC000217611596 CH For-Sale Unstable FAAH 53 44 O=C(NCCCCc1ccccc1)NCC1CCCCC1 ZINC000217611596 CH For-Sale Unstable SCN5A 0 41 O=C(NCCCCc1ccccc1)NCC1CCCCC1 ZINC000217611596 CH For-Sale Unstable CES1 54 35 O=C(NCCCCc1ccccc1)NCC1CCCCC1 ZINC000217611596 CH For-Sale Unstable EPHX2 23 49 O=C(NCCCCc1ccccc1)NCC1CCCCC1 ZINC000217611596 CH For-Sale Unstable AMP1_PLAFQ 25 44 C[C@H](NS(=O)(=O)c1ccc(NC[C@@H]2CCCO2)c(C(=O)O)c1)c1ccccc1 ZINC000217611600 HG In-Stock Unstable BDKRB1 28 40 C[C@H](NS(=O)(=O)c1ccc(NC[C@@H]2CCCO2)c(C(=O)O)c1)c1ccccc1 ZINC000217611600 HG In-Stock Unstable TNK2 45 39 C[C@H](NS(=O)(=O)c1ccc(NC[C@@H]2CCCO2)c(C(=O)O)c1)c1ccccc1 ZINC000217611600 HG In-Stock Unstable CCR8 43 31 CN(C[C@H]1COc2ccccc2O1)C(=O)C(F)F ZINC000217611615 CD On-Demand Unstable ADRA2B 17 41 C[C@@H](NS(=O)(=O)c1ccc(NC[C@H]2CCCO2)c(C(=O)O)c1)c1ccccc1 ZINC000217611688 HG In-Stock Unstable BDKRB1 28 40 C[C@@H](NS(=O)(=O)c1ccc(NC[C@H]2CCCO2)c(C(=O)O)c1)c1ccccc1 ZINC000217611688 HG In-Stock Unstable TNK2 45 39 C[C@@H](NS(=O)(=O)c1ccc(NC[C@H]2CCCO2)c(C(=O)O)c1)c1ccccc1 ZINC000217611688 HG In-Stock Unstable CCR8 43 31 CC(=O)N[C@@H](CCO)c1nc2ccccc2s1 ZINC000217611695 CD In-Stock Unstable PRSS3 0 41 CC(=O)N[C@@H](CCO)c1nc2ccccc2s1 ZINC000217611695 CD In-Stock Unstable TPSAB1 19 42 CC(=O)N[C@@H](CCO)c1nc2ccccc2s1 ZINC000217611695 CD In-Stock Unstable TMPRSS6 49 34 O=c1cc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)oc(CN2CCN(Cc3ccc4c(c3)OCO4)CC2)c1O ZINC000217611757 KE In-Stock Unstable CHRNA4 29 50 O=c1cc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)oc(CN2CCN(Cc3ccc4c(c3)OCO4)CC2)c1O ZINC000217611757 KE In-Stock Unstable MCHR1 19 40 C[C@H](NS(=O)(=O)c1ccc(NC[C@H]2CCCO2)c(C(=O)O)c1)c1ccccc1 ZINC000217611761 HG In-Stock Unstable BDKRB1 28 40 C[C@H](NS(=O)(=O)c1ccc(NC[C@H]2CCCO2)c(C(=O)O)c1)c1ccccc1 ZINC000217611761 HG In-Stock Unstable TNK2 45 39 C[C@H](NS(=O)(=O)c1ccc(NC[C@H]2CCCO2)c(C(=O)O)c1)c1ccccc1 ZINC000217611761 HG In-Stock Unstable CCR8 43 31 CC(=O)N[C@H](CCO)c1nc2ccccc2s1 ZINC000217611781 CD In-Stock Unstable PRSS3 0 41 CC(=O)N[C@H](CCO)c1nc2ccccc2s1 ZINC000217611781 CD In-Stock Unstable TPSAB1 19 42 CC(=O)N[C@H](CCO)c1nc2ccccc2s1 ZINC000217611781 CD In-Stock Unstable TMPRSS6 49 34 O=C(O)/C=C\c1cccc(CN2C(=O)CCCCC2=O)c1 ZINC000217611838 CE For-Sale Unstable PTGER2 22 41 O=C(O)/C=C\c1cccc(CN2C(=O)CCCCC2=O)c1 ZINC000217611838 CE For-Sale Unstable PTGER3 28 41 C[C@@H](NS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217611867 FG In-Stock Unstable KCNQ2 79 44 C[C@@H](NS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217611867 FG In-Stock Unstable TRY2_BOVIN 50 33 C[C@@H](NS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217611867 FG In-Stock Unstable NPY2R 57 36 C[C@@H](NS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217611867 FG In-Stock Unstable SLC6A9 18 41 C[C@@H](NS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217611867 FG In-Stock Unstable SFRP1 53 33 Cc1ccc(S(=O)(=O)N2CCN(C(=O)NCC3CCCCC3)CC2)cc1 ZINC000217611913 GF On-Demand Unstable EPHX2 45 54 Cc1ccc(S(=O)(=O)N2CCN(C(=O)NCC3CCCCC3)CC2)cc1 ZINC000217611913 GF On-Demand Unstable TGM2 87 43 Cc1ccc(S(=O)(=O)N2CCN(C(=O)NCC3CCCCC3)CC2)cc1 ZINC000217611913 GF On-Demand Unstable MMP7 42 39 Cc1ccc(S(=O)(=O)N2CCN(C(=O)NCC3CCCCC3)CC2)cc1 ZINC000217611913 GF On-Demand Unstable CACNA1I 46 33 Cc1ccc(S(=O)(=O)N2CCN(C(=O)NCC3CCCCC3)CC2)cc1 ZINC000217611913 GF On-Demand Unstable F13A1 100 43 Cc1ccc(S(=O)(=O)N2CCN(C(=O)NCC3CCCCC3)CC2)cc1 ZINC000217611913 GF On-Demand Unstable NAMPT 46 40 C[C@H](NS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217611940 FG In-Stock Unstable KCNQ2 79 44 C[C@H](NS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217611940 FG In-Stock Unstable TRY2_BOVIN 50 33 C[C@H](NS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217611940 FG In-Stock Unstable NPY2R 57 36 C[C@H](NS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217611940 FG In-Stock Unstable SLC6A9 18 41 C[C@H](NS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217611940 FG In-Stock Unstable SFRP1 53 33 Cc1cccc(S(=O)(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217611946 FF For-Sale Unstable NPY5R 27 42 O=C(c1ccccc1)N1CCN(C(=O)C(F)F)CC1 ZINC000217611994 CD On-Demand Unstable INHA 25 42 O=C(c1ccccc1)N1CCN(C(=O)C(F)F)CC1 ZINC000217611994 CD On-Demand Unstable SMO 38 41 O=C(c1ccccc1)N1CCN(C(=O)C(F)F)CC1 ZINC000217611994 CD On-Demand Unstable L3MBTL3 46 38 O=C(c1ccccc1)N1CCN(C(=O)C(F)F)CC1 ZINC000217611994 CD On-Demand Unstable SLC6A7 0 49 COc1ccc(CCOc2cc([C@H](CC(N)=O)c3c(C)[nH][nH]c3=O)ccc2OC)cc1 ZINC000217611996 IF In-Stock Unstable PDEB1 0 41 Cc1ccc(/C=C\C(=O)O)cc1N1C(=O)CCCC1=O ZINC000217612002 CE For-Sale Unstable RXRA 18 42 O=C(C(c1ccccc1)c1ccccc1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217612004 HF In-Stock Unstable AGTR2 52 36 COC(=O)N1CCN(C(=O)NCC2CCCCC2)CC1 ZINC000217612019 CD On-Demand Unstable CACNA1I 40 33 Cc1ccccc1-c1snc(Cl)c1COc1c(F)cc(CCC(=O)O)cc1F ZINC000217612021 HK Annotated Unstable THRB 16 47 Cc1ccccc1-c1snc(Cl)c1COc1c(F)cc(CCC(=O)O)cc1F ZINC000217612021 HK Annotated Unstable FFAR1 60 42 Cc1ccccc1-c1snc(Cl)c1COc1c(F)cc(CCC(=O)O)cc1F ZINC000217612021 HK Annotated Unstable FFAR4 47 37 Cc1cccc(S(=O)(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217612037 FF For-Sale Unstable NPY5R 27 42 C[C@@H](NS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217612048 GG In-Stock Unstable KCNQ2 75 43 C[C@@H](NS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217612048 GG In-Stock Unstable TRY2_BOVIN 45 34 C[C@@H](NS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217612048 GG In-Stock Unstable NPY2R 53 38 C[C@@H](NS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217612048 GG In-Stock Unstable SLC6A9 16 43 C[C@@H](NS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217612048 GG In-Stock Unstable SFRP1 50 32 C[C@@H](NS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217612048 GG In-Stock Unstable WNT3 41 32 COc1ccc(CCOc2cc([C@@H](CC(N)=O)c3c(C)[nH][nH]c3=O)ccc2OC)cc1 ZINC000217612080 IF In-Stock Unstable PDEB1 0 41 C[C@@H](NC[C@H]1CCCCN1C)[C@@H]1CCCN(C)C1 ZINC000217612092 CD For-Sale Unstable CHRNA10 48 33 CCC[C@@H](C)NC(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217612096 CF For-Sale Unstable TNFRSF1A 19 40 O=C(NCCCn1ccccc1=O)c1ccccc1N1CCOCC1 ZINC000217612098 ED In-Stock Unstable HTR1A 32 41 O=C(NCCCn1ccccc1=O)c1ccccc1N1CCOCC1 ZINC000217612098 ED In-Stock Unstable DRD2 43 42 O=C(NCCCn1ccccc1=O)c1ccccc1N1CCOCC1 ZINC000217612098 ED In-Stock Unstable DRD1 23 42 O=C(NCCCn1ccccc1=O)c1ccccc1N1CCOCC1 ZINC000217612098 ED In-Stock Unstable DRD4 21 41 O=C(NCCCn1ccccc1=O)c1ccccc1N1CCOCC1 ZINC000217612098 ED In-Stock Unstable HTR2C 36 40 O=C(NCCCn1ccccc1=O)c1ccccc1N1CCOCC1 ZINC000217612098 ED In-Stock Unstable SLC6A4 15 40 O=C(NCCCn1ccccc1=O)c1ccccc1N1CCOCC1 ZINC000217612098 ED In-Stock Unstable ADRA1A 35 41 O=C(NCCCn1ccccc1=O)c1ccccc1N1CCOCC1 ZINC000217612098 ED In-Stock Unstable ADRA1B 20 40 O=C(NCCCn1ccccc1=O)c1ccccc1N1CCOCC1 ZINC000217612098 ED In-Stock Unstable DRD3 68 40 O=C(c1ccccc1Cl)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217612109 EE In-Stock Unstable P2RX7 15 40 O=C(c1ccccc1Cl)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217612109 EE In-Stock Unstable MAPK9 34 40 O=C(c1ccccc1Cl)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217612109 EE In-Stock Unstable MAPK10 37 40 O=C(c1ccccc1Cl)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217612109 EE In-Stock Unstable AKR1C3 26 42 C[C@H](NS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217612119 GG In-Stock Unstable KCNQ2 75 43 C[C@H](NS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217612119 GG In-Stock Unstable TRY2_BOVIN 45 34 C[C@H](NS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217612119 GG In-Stock Unstable NPY2R 53 38 C[C@H](NS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217612119 GG In-Stock Unstable SLC6A9 16 43 C[C@H](NS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217612119 GG In-Stock Unstable SFRP1 50 32 C[C@H](NS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217612119 GG In-Stock Unstable WNT3 41 32 [N-]=[N+]=N[C@]1(CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)C(F)(F)[C@@H]1O ZINC000217612126 KB Annotated Unstable POLA1 43 51 [N-]=[N+]=N[C@]1(CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)C(F)(F)[C@@H]1O ZINC000217612126 KB Annotated Unstable P2RY6 94 41 [N-]=[N+]=N[C@]1(CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)C(F)(F)[C@@H]1O ZINC000217612126 KB Annotated Unstable POLB 43 51 [N-]=[N+]=N[C@]1(CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)C(F)(F)[C@@H]1O ZINC000217612126 KB Annotated Unstable P2RX1 42 35 [N-]=[N+]=N[C@]1(CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)C(F)(F)[C@@H]1O ZINC000217612126 KB Annotated Unstable P2RY4 112 41 [N-]=[N+]=N[C@]1(CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)C(F)(F)[C@@H]1O ZINC000217612126 KB Annotated Unstable P2RY2 137 43 O=C1O[C@@]2(CCCN(S(=O)(=O)c3ccccc3F)C2)c2ccccc21 ZINC000217612145 FF For-Sale Unstable NPY5R 27 45 O=C(COc1cc(C(F)(F)F)cc(C(F)(F)F)c1)Nc1ccccc1C(=O)N1CCCC1 ZINC000217612148 JJ On-Demand Unstable TACR1 40 39 O=C(COc1cc(C(F)(F)F)cc(C(F)(F)F)c1)Nc1ccccc1C(=O)N1CCCC1 ZINC000217612148 JJ On-Demand Unstable KCNQ2 29 43 O=C(COc1cc(C(F)(F)F)cc(C(F)(F)F)c1)Nc1ccccc1C(=O)N1CCCC1 ZINC000217612148 JJ On-Demand Unstable RBP4 43 37 O=C(COc1cc(C(F)(F)F)cc(C(F)(F)F)c1)Nc1ccccc1C(=O)N1CCCC1 ZINC000217612148 JJ On-Demand Unstable HCAR2 18 46 O=C(COc1cc(C(F)(F)F)cc(C(F)(F)F)c1)Nc1ccccc1C(=O)N1CCCC1 ZINC000217612148 JJ On-Demand Unstable NPSR1 15 43 O=C(COc1cc(C(F)(F)F)cc(C(F)(F)F)c1)Nc1ccccc1C(=O)N1CCCC1 ZINC000217612148 JJ On-Demand Unstable RHOA 0 41 C[C@H](NC[C@H]1CCCCN1C)[C@@H]1CCCN(C)C1 ZINC000217612172 CD For-Sale Unstable CHRNA10 48 33 CCC[C@H](C)NC(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217612173 CF For-Sale Unstable TNFRSF1A 19 40 O=C1O[C@]2(CCCN(S(=O)(=O)c3ccccc3F)C2)c2ccccc21 ZINC000217612221 FF For-Sale Unstable NPY5R 27 45 C[C@@H](NS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217612235 GE In-Stock Unstable KCNQ2 22 43 C[C@@H](NS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217612235 GE In-Stock Unstable NPY2R 46 34 C[C@@H](NS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217612235 GE In-Stock Unstable SLC6A9 26 46 Cc1ccc(Cn2nccc2NC(=O)c2sccc2S(=O)(=O)N2CCc3ccccc3C2)cc1 ZINC000217612255 JI On-Demand Unstable NOD2 41 36 C[C@H](NS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217612323 GE In-Stock Unstable KCNQ2 22 43 C[C@H](NS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217612323 GE In-Stock Unstable NPY2R 46 34 C[C@H](NS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1)c1ccccc1 ZINC000217612323 GE In-Stock Unstable SLC6A9 26 46 O=C1O[C@@]2(CCCN(S(=O)(=O)c3ccc(F)cc3)C2)c2ccccc21 ZINC000217612348 FF For-Sale Unstable NPY5R 28 44 COc1ncccc1C(=O)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217612349 EC In-Stock Unstable HSP90AB1 0 51 COc1ccc2nc(C(=O)Nc3ccnn3Cc3ccc(C)cc3)ccc2c1 ZINC000217612361 FI On-Demand Unstable NPBWR1 33 42 CN(Cc1cccc(Cl)c1)C(=O)C(F)F ZINC000217612377 BF On-Demand Unstable HSP90AB1 20 41 CN(Cc1cccc(Cl)c1)C(=O)C(F)F ZINC000217612377 BF On-Demand Unstable LIMK2 20 41 CCOCCCNc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O ZINC000217612428 HG In-Stock Unstable BDKRB1 21 42 O=C1O[C@]2(CCCN(S(=O)(=O)c3ccc(F)cc3)C2)c2ccccc21 ZINC000217612430 FF For-Sale Unstable NPY5R 28 44 COC(=O)[C@@]1(C)[C@H](N)CCN1Cc1ccccc1 ZINC000217612480 BD For-Sale Unstable DRD4 26 40 COC(=O)[C@@]1(C)[C@H](N)CCN1Cc1ccccc1 ZINC000217612480 BD For-Sale Unstable ACHE 24 40 COC(=O)[C@@]1(C)[C@H](N)CCN1Cc1ccccc1 ZINC000217612480 BD For-Sale Unstable SLC6A1 20 40 COC(=O)[C@@]1(C)[C@H](N)CCN1Cc1ccccc1 ZINC000217612480 BD For-Sale Unstable DRD3 27 40 COC(=O)[C@@]1(C)[C@H](N)CCN1Cc1ccccc1 ZINC000217612480 BD For-Sale Unstable SLC6A3 22 40 COC(=O)[C@@]1(C)[C@H](N)CCN1Cc1ccccc1 ZINC000217612480 BD For-Sale Unstable SIGMAR1 62 43 COC(=O)[C@@]1(C)[C@H](N)CCN1Cc1ccccc1 ZINC000217612480 BD For-Sale Unstable NPFFR1 49 35 COC(=O)[C@@]1(C)[C@H](N)CCN1Cc1ccccc1 ZINC000217612480 BD For-Sale Unstable SLC12A5 67 39 CN1CCN(C)[C@@H](CNC(=O)Nc2ccccc2Oc2ccccc2F)C1 ZINC000217612498 FF In-Stock Unstable ITGA4 50 37 Cc1cnc(NC(=O)c2cccc(/C=C\C(=O)O)c2)s1 ZINC000217612499 CF For-Sale Unstable HDAC8 29 44 Cc1cnc(NC(=O)c2cccc(/C=C\C(=O)O)c2)s1 ZINC000217612499 CF For-Sale Unstable HDAC6 19 44 Cc1cnc(NC(=O)c2cccc(/C=C\C(=O)O)c2)s1 ZINC000217612499 CF For-Sale Unstable KCNK3 77 38 Cc1cnc(NC(=O)c2cccc(/C=C\C(=O)O)c2)s1 ZINC000217612499 CF For-Sale Unstable KCNK9 47 38 CCOCCCNc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O ZINC000217612503 HG In-Stock Unstable BDKRB1 21 42 CN(Cc1cccnc1)C(=O)C(F)F ZINC000217612504 BD On-Demand Unstable TBXAS1 40 41 CN(Cc1cccnc1)C(=O)C(F)F ZINC000217612504 BD On-Demand Unstable KCNA5 43 38 CN(Cc1cccnc1)C(=O)C(F)F ZINC000217612504 BD On-Demand Unstable NR1D1 44 36 CC(C)(C)OC(=O)N1CCN(C(=O)NCC2CCCCC2)CC1 ZINC000217612541 EF On-Demand Unstable GPR119 38 40 CN1CCC[C@@H](CNC(=O)c2ccc(/C=C\C(=O)O)s2)C1 ZINC000217612560 DD For-Sale Unstable CACNA1I 48 35 COC(=O)[C@]1(C)[C@H](N)CCN1Cc1ccccc1 ZINC000217612575 BD For-Sale Unstable DRD4 26 40 COC(=O)[C@]1(C)[C@H](N)CCN1Cc1ccccc1 ZINC000217612575 BD For-Sale Unstable ACHE 24 40 COC(=O)[C@]1(C)[C@H](N)CCN1Cc1ccccc1 ZINC000217612575 BD For-Sale Unstable SLC6A1 20 40 COC(=O)[C@]1(C)[C@H](N)CCN1Cc1ccccc1 ZINC000217612575 BD For-Sale Unstable DRD3 27 40 COC(=O)[C@]1(C)[C@H](N)CCN1Cc1ccccc1 ZINC000217612575 BD For-Sale Unstable SLC6A3 22 40 COC(=O)[C@]1(C)[C@H](N)CCN1Cc1ccccc1 ZINC000217612575 BD For-Sale Unstable SIGMAR1 62 43 COC(=O)[C@]1(C)[C@H](N)CCN1Cc1ccccc1 ZINC000217612575 BD For-Sale Unstable NPFFR1 49 35 COC(=O)[C@]1(C)[C@H](N)CCN1Cc1ccccc1 ZINC000217612575 BD For-Sale Unstable SLC12A5 67 39 Cc1cnc(NC(=O)c2cc(/C=C\C(=O)O)ccc2F)s1 ZINC000217612579 DF For-Sale Unstable FFAR2 19 41 CC(C)OCCCNc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O ZINC000217612606 HH In-Stock Unstable BDKRB1 0 41 CN(Cc1ccc(Cl)c(Cl)c1)C(=O)C(F)F ZINC000217612620 CG On-Demand Unstable OPRK1 23 44 CN(Cc1ccc(Cl)c(Cl)c1)C(=O)C(F)F ZINC000217612620 CG On-Demand Unstable PTPRG 0 42 CN(Cc1ccc(Cl)c(Cl)c1)C(=O)C(F)F ZINC000217612620 CG On-Demand Unstable CENPE 0 42 COC(=O)[C@@]1(C)[C@@H](N)CCN1Cc1ccccc1 ZINC000217612670 BD For-Sale Unstable DRD4 26 40 COC(=O)[C@@]1(C)[C@@H](N)CCN1Cc1ccccc1 ZINC000217612670 BD For-Sale Unstable ACHE 24 40 COC(=O)[C@@]1(C)[C@@H](N)CCN1Cc1ccccc1 ZINC000217612670 BD For-Sale Unstable SLC6A1 20 40 COC(=O)[C@@]1(C)[C@@H](N)CCN1Cc1ccccc1 ZINC000217612670 BD For-Sale Unstable DRD3 27 40 COC(=O)[C@@]1(C)[C@@H](N)CCN1Cc1ccccc1 ZINC000217612670 BD For-Sale Unstable SLC6A3 22 40 COC(=O)[C@@]1(C)[C@@H](N)CCN1Cc1ccccc1 ZINC000217612670 BD For-Sale Unstable SIGMAR1 62 43 COC(=O)[C@@]1(C)[C@@H](N)CCN1Cc1ccccc1 ZINC000217612670 BD For-Sale Unstable NPFFR1 49 35 COC(=O)[C@@]1(C)[C@@H](N)CCN1Cc1ccccc1 ZINC000217612670 BD For-Sale Unstable SLC12A5 67 39 CC(C)OCCCNc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O ZINC000217612674 HH In-Stock Unstable BDKRB1 0 41 COc1ccc(NC(=O)N/C=C/c2ccccc2)cc1OC ZINC000217612677 CG For-Sale Unstable IMPDH1 0 46 COc1ccc(NC(=O)N/C=C/c2ccccc2)cc1OC ZINC000217612677 CG For-Sale Unstable CYP1B1 26 50 COc1ccc(NC(=O)N/C=C/c2ccccc2)cc1OC ZINC000217612677 CG For-Sale Unstable MTNR1B 17 43 COc1ccc(NC(=O)N/C=C/c2ccccc2)cc1OC ZINC000217612677 CG For-Sale Unstable MMP2 0 45 COc1ccc(NC(=O)N/C=C/c2ccccc2)cc1OC ZINC000217612677 CG For-Sale Unstable CYP1A1 25 50 COc1ccc(NC(=O)N/C=C/c2ccccc2)cc1OC ZINC000217612677 CG For-Sale Unstable PDGFRA 45 39 COc1ccc(NC(=O)N/C=C/c2ccccc2)cc1OC ZINC000217612677 CG For-Sale Unstable IMPDH2 0 47 COc1ccc(NC(=O)N/C=C/c2ccccc2)cc1OC ZINC000217612677 CG For-Sale Unstable ABCG2 30 42 COc1ccc(NC(=O)N/C=C/c2ccccc2)cc1OC ZINC000217612677 CG For-Sale Unstable ENPP1 74 35 O=C(c1ccc(-n2cccc2)cc1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217612689 GE In-Stock Unstable MTOR 26 41 O=C(c1ccc(-n2cccc2)cc1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217612689 GE In-Stock Unstable SLC6A7 0 52 C[C@@H]1CCc2cc(OCC(=O)O)ccc2N1 ZINC000217612700 BD In-Stock Unstable PPARG 31 40 C[C@@H]1CCc2cc(OCC(=O)O)ccc2N1 ZINC000217612700 BD In-Stock Unstable PPARD 48 40 Cc1cc(F)ccc1NC(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217612751 DH For-Sale Unstable MAPK11 28 41 COC(=O)[C@]1(C)[C@@H](N)CCN1Cc1ccccc1 ZINC000217612759 BD For-Sale Unstable DRD4 26 40 COC(=O)[C@]1(C)[C@@H](N)CCN1Cc1ccccc1 ZINC000217612759 BD For-Sale Unstable ACHE 24 40 COC(=O)[C@]1(C)[C@@H](N)CCN1Cc1ccccc1 ZINC000217612759 BD For-Sale Unstable SLC6A1 20 40 COC(=O)[C@]1(C)[C@@H](N)CCN1Cc1ccccc1 ZINC000217612759 BD For-Sale Unstable DRD3 27 40 COC(=O)[C@]1(C)[C@@H](N)CCN1Cc1ccccc1 ZINC000217612759 BD For-Sale Unstable SLC6A3 22 40 COC(=O)[C@]1(C)[C@@H](N)CCN1Cc1ccccc1 ZINC000217612759 BD For-Sale Unstable SIGMAR1 62 43 COC(=O)[C@]1(C)[C@@H](N)CCN1Cc1ccccc1 ZINC000217612759 BD For-Sale Unstable NPFFR1 49 35 COC(=O)[C@]1(C)[C@@H](N)CCN1Cc1ccccc1 ZINC000217612759 BD For-Sale Unstable SLC12A5 67 39 C[C@H]1CCc2cc(OCC(=O)O)ccc2N1 ZINC000217612775 BD In-Stock Unstable PPARG 31 40 C[C@H]1CCc2cc(OCC(=O)O)ccc2N1 ZINC000217612775 BD In-Stock Unstable PPARD 48 40 CCCCCNc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O ZINC000217612786 GI In-Stock Unstable BDKRB1 26 42 O=C(N/C=C/c1ccccc1)NCCCN1CCCC1=O ZINC000217612798 CD For-Sale Unstable TYRO3 25 43 CN(CCOc1ccc(Cl)cc1)C(=O)C(F)F ZINC000217612845 CE On-Demand Unstable UTS2 41 34 CCc1ccc(-c2nc(CC(=O)N(CCOC)[C@@H]3CCS(=O)(=O)C3)cs2)cc1 ZINC000217612866 HF On-Demand Unstable AVPR1B 17 44 CCCCCNc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O ZINC000217612870 GI In-Stock Unstable BDKRB1 26 42 [N-]=[N+]=N[C@]1(CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)[C@H](F)[C@@H]1O ZINC000217612890 KB Annotated Unstable POLA1 45 53 [N-]=[N+]=N[C@]1(CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)[C@H](F)[C@@H]1O ZINC000217612890 KB Annotated Unstable P2RY6 105 43 [N-]=[N+]=N[C@]1(CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)[C@H](F)[C@@H]1O ZINC000217612890 KB Annotated Unstable POLB 45 53 [N-]=[N+]=N[C@]1(CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)[C@H](F)[C@@H]1O ZINC000217612890 KB Annotated Unstable P2RX4 40 35 [N-]=[N+]=N[C@]1(CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)[C@H](F)[C@@H]1O ZINC000217612890 KB Annotated Unstable P2RX1 54 35 [N-]=[N+]=N[C@]1(CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)[C@H](F)[C@@H]1O ZINC000217612890 KB Annotated Unstable P2RY4 123 43 [N-]=[N+]=N[C@]1(CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)[C@H](F)[C@@H]1O ZINC000217612890 KB Annotated Unstable P2RY2 151 47 [N-]=[N+]=N[C@]1(CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)[C@H](F)[C@@H]1O ZINC000217612890 KB Annotated Unstable P2RY14 46 36 [N-]=[N+]=N[C@]1(CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)[C@H](F)[C@@H]1O ZINC000217612890 KB Annotated Unstable GPR17 42 33 O=C(N/C=C/c1ccccc1)Nc1ccc(Br)cc1 ZINC000217612915 DI For-Sale Anodyne EPHX1 0 44 O=C(N/C=C/c1ccccc1)Nc1ccc(Br)cc1 ZINC000217612915 DI For-Sale Anodyne P95276_MYCTO 0 44 Cc1cccc(C)c1NC(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217612918 DH For-Sale Unstable LCK 22 41 Cc1cccc(C)c1NC(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217612918 DH For-Sale Unstable S1PR4 25 53 CCc1ccc(-c2nc(CC(=O)N(CCOC)[C@H]3CCS(=O)(=O)C3)cs2)cc1 ZINC000217612946 HF On-Demand Unstable AVPR1B 17 44 CC[C@H](C)[C@H](C(=O)N[C@H](CO)Cc1ccccc1)N1Cc2ccccc2C1=O ZINC000217612967 GF In-Stock Unstable MME 53 37 CC[C@H](C)[C@H](C(=O)N[C@H](CO)Cc1ccccc1)N1Cc2ccccc2C1=O ZINC000217612967 GF In-Stock Unstable PAPA1_CARPA 40 31 CC[C@H](C)[C@H](C(=O)N[C@H](CO)Cc1ccccc1)N1Cc2ccccc2C1=O ZINC000217612967 GF In-Stock Unstable ACE2 55 39 CC[C@H](C)[C@H](C(=O)N[C@H](CO)Cc1ccccc1)N1Cc2ccccc2C1=O ZINC000217612967 GF In-Stock Unstable DERP1 0 44 CC(C)CCNc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O ZINC000217612987 GH In-Stock Unstable BDKRB1 17 42 C[C@@H](NC(=O)C(F)F)c1ccc(Cl)cc1Cl ZINC000217612989 CG On-Demand Unstable SDH1 0 61 C[C@@H](NC(=O)C(F)F)c1ccc(Cl)cc1Cl ZINC000217612989 CG On-Demand Unstable CPHA 0 40 O=C(N/C=C/c1ccccc1)Nc1cccc(C(=O)O)c1 ZINC000217613013 CG For-Sale Anodyne PPIA 23 43 O=C(N/C=C/c1ccccc1)Nc1cccc(C(=O)O)c1 ZINC000217613013 CG For-Sale Anodyne CCKAR 0 41 O=C(N/C=C/c1ccccc1)Nc1cccc(C(=O)O)c1 ZINC000217613013 CG For-Sale Anodyne EPHX2 17 47 O=C(N/C=C/c1ccccc1)Nc1cccc(C(=O)O)c1 ZINC000217613013 CG For-Sale Anodyne TTR 0 40 O=C(N/C=C/c1ccccc1)Nc1cccc(C(=O)O)c1 ZINC000217613013 CG For-Sale Anodyne AKR1C3 46 55 O=C(N/C=C/c1ccccc1)Nc1cccc(C(=O)O)c1 ZINC000217613013 CG For-Sale Anodyne AKR1C4 0 40 O=C(N/C=C/c1ccccc1)Nc1cccc(C(=O)O)c1 ZINC000217613013 CG For-Sale Anodyne P95276_MYCTO 0 41 O=C(N/C=C/c1ccccc1)Nc1cccc(C(=O)O)c1 ZINC000217613013 CG For-Sale Anodyne PARP14 0 40 O=C(N/C=C/c1ccccc1)Nc1cccc(C(=O)O)c1 ZINC000217613013 CG For-Sale Anodyne KCNK3 99 40 O=C(N/C=C/c1ccccc1)Nc1cccc(C(=O)O)c1 ZINC000217613013 CG For-Sale Anodyne KCNK9 54 38 O=C(N/C=C/c1ccccc1)Nc1cccc(C(=O)O)c1 ZINC000217613013 CG For-Sale Anodyne PARP10 0 40 CC(C)c1csc(NC(=O)c2sccc2S(=O)(=O)N2CCc3ccccc3C2)n1 ZINC000217613035 II On-Demand Unstable AKR1C3 41 42 CC(C)(C)NC(=O)COc1ccc(CN2C[C@@H]3CC[C@H](C2)[C@@H]3O)cc1 ZINC000217613060 EE In-Stock Unstable ADIPOR1 0 41 CC(C)(C)NC(=O)COc1ccc(CN2C[C@@H]3CC[C@H](C2)[C@@H]3O)cc1 ZINC000217613060 EE In-Stock Unstable ADIPOR2 0 41 CC(C)CCNc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O ZINC000217613062 GH In-Stock Unstable BDKRB1 16 42 COC(=O)COc1ccc2occ(-c3ccc(OC)c(OC)c3)c2c1 ZINC000217613069 EH In-Stock Unstable ALDH2 74 44 C[C@H](NC(=O)C(F)F)c1ccc(Cl)cc1Cl ZINC000217613073 CG On-Demand Unstable SDH1 0 61 C[C@H](NC(=O)C(F)F)c1ccc(Cl)cc1Cl ZINC000217613073 CG On-Demand Unstable CPHA 0 40 O=C1NC(=O)[C@H]2[C@H]1CCCN2Cc1ccccc1 ZINC000217613085 BC For-Sale Unstable SIGMAR1 51 46 O=C(c1c(F)cccc1F)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217613106 ED In-Stock Unstable HSP90AB1 15 43 O=C(N/C=C/c1ccccc1)Nc1ccccc1[N+](=O)[O-] ZINC000217613123 CG For-Sale Bother COLA 94 35 N#CCN(C(=O)c1ccc(=O)[nH]n1)C1CCCC1 ZINC000217613132 BC For-Sale Unstable ACE 40 34 O=C1NC(=O)[C@H]2[C@@H]1CCCN2Cc1ccccc1 ZINC000217613166 BC For-Sale Unstable SIGMAR1 51 46 O=C(N/C=C/c1ccccc1)Nc1cccc(O)c1 ZINC000217613218 CG For-Sale Anodyne MMP2 15 53 O=C(N/C=C/c1ccccc1)Nc1cccc(O)c1 ZINC000217613218 CG For-Sale Anodyne MMP9 15 53 O=C(N/C=C/c1ccccc1)Nc1cccc(O)c1 ZINC000217613218 CG For-Sale Anodyne MMP1 22 65 O=C(N/C=C/c1ccccc1)Nc1cccc(O)c1 ZINC000217613218 CG For-Sale Anodyne P95276_MYCTO 0 42 O=C(N/C=C/c1ccccc1)Nc1cccc(O)c1 ZINC000217613218 CG For-Sale Anodyne KCNK3 47 35 CN(C(=O)c1sccc1S(=O)(=O)N1CCc2ccccc2C1)C1CCCC1 ZINC000217613244 HH On-Demand Unstable AKR1C3 62 48 COc1ccc(CN2C[C@H]3[C@@H](C2)[C@@H]3C(=O)O)cc1Cl ZINC000217613256 CE In-Stock Unstable PDE5A 38 41 COc1ccc(CN2C[C@H]3[C@@H](C2)[C@@H]3C(=O)O)cc1Cl ZINC000217613256 CE In-Stock Unstable DRD4 23 43 COc1ccc(CN2C[C@H]3[C@@H](C2)[C@@H]3C(=O)O)cc1Cl ZINC000217613256 CE In-Stock Unstable DRD3 22 41 COc1ccc(CN2C[C@H]3[C@@H](C2)[C@@H]3C(=O)O)cc1Cl ZINC000217613256 CE In-Stock Unstable SIGMAR1 15 40 COc1ccc(CN2C[C@H]3[C@@H](C2)[C@@H]3C(=O)O)cc1Cl ZINC000217613256 CE In-Stock Unstable S1PR3 0 44 COc1ccc(CN2C[C@H]3[C@@H](C2)[C@@H]3C(=O)O)cc1Cl ZINC000217613256 CE In-Stock Unstable PDE6A 41 31 COc1ccc(CN2C[C@H]3[C@@H](C2)[C@@H]3C(=O)O)cc1Cl ZINC000217613256 CE In-Stock Unstable S1PR1 19 44 COc1ccc(CN2C[C@H]3[C@@H](C2)[C@@H]3C(=O)O)cc1Cl ZINC000217613256 CE In-Stock Unstable S1PR5 30 44 COc1ccc(CN2C[C@H]3[C@@H](C2)[C@@H]3C(=O)O)cc1Cl ZINC000217613256 CE In-Stock Unstable MCHR1 15 41 C[C@@H](Cc1nccn1Cc1ccccc1)C(=O)O ZINC000217613268 BE For-Sale Unstable MME 51 37 C[C@@H](Cc1nccn1Cc1ccccc1)C(=O)O ZINC000217613268 BE For-Sale Unstable CPA1 51 33 C[C@@H](Cc1nccn1Cc1ccccc1)C(=O)O ZINC000217613268 BE For-Sale Unstable CAPNS1 44 32 C[C@@H](Cc1nccn1Cc1ccccc1)C(=O)O ZINC000217613268 BE For-Sale Unstable ACE2 41 33 C[C@@H](Cc1nccn1Cc1ccccc1)C(=O)O ZINC000217613268 BE For-Sale Unstable FPR1 51 38 COc1cc2c(cc1OC)CN(C(=O)[C@@H](NC(=O)N1C[C@@H]3C[C@H](C1)c1cccc(=O)n1C3)C(C)C)CC2 ZINC000217613293 KF In-Stock Unstable CHRNA4 24 40 COc1cc2c(cc1OC)CN(C(=O)[C@@H](NC(=O)N1C[C@@H]3C[C@H](C1)c1cccc(=O)n1C3)C(C)C)CC2 ZINC000217613293 KF In-Stock Unstable HCRTR2 15 42 Cc1ccc(S(=O)(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1C ZINC000217613312 FG For-Sale Unstable NPY5R 25 42 O=C(O)CCNC(=O)N/C=C/c1ccccc1 ZINC000217613321 BD For-Sale Unstable MME 19 43 O=C(NCC(=O)N1Cc2cnc(N3CCOCC3)nc2C1)c1ccccc1 ZINC000217613340 FC In-Stock Unstable PIK3CA 28 41 O=C(NCC(=O)N1Cc2cnc(N3CCOCC3)nc2C1)c1ccccc1 ZINC000217613340 FC In-Stock Unstable MTOR 43 41 O=C(NCC(=O)N1Cc2cnc(N3CCOCC3)nc2C1)c1ccccc1 ZINC000217613340 FC In-Stock Unstable PIK3CG 27 41 O=C(NCC(=O)N1Cc2cnc(N3CCOCC3)nc2C1)c1ccccc1 ZINC000217613340 FC In-Stock Unstable FAP 0 40 C[C@H](Cc1nccn1Cc1ccccc1)C(=O)O ZINC000217613352 BE For-Sale Unstable MME 51 37 C[C@H](Cc1nccn1Cc1ccccc1)C(=O)O ZINC000217613352 BE For-Sale Unstable CPA1 51 33 C[C@H](Cc1nccn1Cc1ccccc1)C(=O)O ZINC000217613352 BE For-Sale Unstable CAPNS1 44 32 C[C@H](Cc1nccn1Cc1ccccc1)C(=O)O ZINC000217613352 BE For-Sale Unstable ACE2 41 33 C[C@H](Cc1nccn1Cc1ccccc1)C(=O)O ZINC000217613352 BE For-Sale Unstable FPR1 51 38 CN(C(=O)COc1cc(C(F)(F)F)cc(C(F)(F)F)c1)C1CCCC1 ZINC000217613354 FJ On-Demand Unstable TACR1 44 36 Cc1ccc(S(=O)(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1C ZINC000217613394 FG For-Sale Unstable NPY5R 25 42 Nc1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217613445 CG For-Sale Unstable EPHX1 0 44 Nc1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217613445 CG For-Sale Unstable MTCA1 29 40 Nc1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217613445 CG For-Sale Unstable P96878_MYCTU 36 40 Nc1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217613445 CG For-Sale Unstable P95276_MYCTO 0 44 C[C@@H](Cc1cncn1Cc1ccccc1)C(=O)O ZINC000217613471 BE For-Sale Unstable CYP11B1 20 43 C[C@@H](Cc1cncn1Cc1ccccc1)C(=O)O ZINC000217613471 BE For-Sale Unstable MME 45 36 C[C@@H](Cc1cncn1Cc1ccccc1)C(=O)O ZINC000217613471 BE For-Sale Unstable CPA1 52 36 C[C@@H](Cc1cncn1Cc1ccccc1)C(=O)O ZINC000217613471 BE For-Sale Unstable CYP11B2 30 57 C[C@@H](Cc1cncn1Cc1ccccc1)C(=O)O ZINC000217613471 BE For-Sale Unstable ACE2 40 33 CC[C@@H](NC(=O)c1ccc(=O)[nH]n1)c1nccs1 ZINC000217613480 CD For-Sale Unstable MAP1 41 34 COC[C@@H](C)Nc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O ZINC000217613526 GF In-Stock Unstable ADAMTS4 41 32 Cc1ccc(S(=O)(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c(C)c1 ZINC000217613529 FG For-Sale Unstable NPY5R 26 46 CC[C@H](NC(=O)c1ccc(=O)[nH]n1)c1nccs1 ZINC000217613547 CD For-Sale Unstable MAP1 41 34 C[C@H](Cc1cncn1Cc1ccccc1)C(=O)O ZINC000217613553 BE For-Sale Unstable CYP11B1 20 43 C[C@H](Cc1cncn1Cc1ccccc1)C(=O)O ZINC000217613553 BE For-Sale Unstable MME 45 36 C[C@H](Cc1cncn1Cc1ccccc1)C(=O)O ZINC000217613553 BE For-Sale Unstable CPA1 52 36 C[C@H](Cc1cncn1Cc1ccccc1)C(=O)O ZINC000217613553 BE For-Sale Unstable CYP11B2 30 57 C[C@H](Cc1cncn1Cc1ccccc1)C(=O)O ZINC000217613553 BE For-Sale Unstable ACE2 40 33 CN1c2ccccc2C(=O)N2CCc3c(n(CCC(N)=O)c4ccccc34)[C@H]21 ZINC000217613608 FF In-Stock Unstable FABI 40 32 CN1c2ccccc2C(=O)N2CCc3c(n(CCC(N)=O)c4ccccc34)[C@H]21 ZINC000217613608 FF In-Stock Unstable HDAC6 17 42 COC[C@H](C)Nc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O ZINC000217613609 GF In-Stock Unstable ADAMTS4 41 32 Cc1ccc(S(=O)(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c(C)c1 ZINC000217613616 FG For-Sale Unstable NPY5R 26 46 CN(C)C(=O)CNC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217613636 CC For-Sale Unstable HDAC8 16 44 C[C@@H](Cc1ccnn1Cc1ccccc1)C(=O)O ZINC000217613661 BE For-Sale Unstable MME 59 37 C[C@@H](Cc1ccnn1Cc1ccccc1)C(=O)O ZINC000217613661 BE For-Sale Unstable CYSP_TRYCR 44 32 C[C@@H](Cc1ccnn1Cc1ccccc1)C(=O)O ZINC000217613661 BE For-Sale Unstable CPA1 52 34 C[C@@H](Cc1ccnn1Cc1ccccc1)C(=O)O ZINC000217613661 BE For-Sale Unstable ACE2 47 34 CC(=O)Nc1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217613672 CG For-Sale Unstable EPHX1 0 45 CC(=O)Nc1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217613672 CG For-Sale Unstable MMP2 0 47 CC(=O)Nc1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217613672 CG For-Sale Unstable MMP1 0 46 CC(=O)Nc1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217613672 CG For-Sale Unstable IDO1 28 44 CC(=O)Nc1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217613672 CG For-Sale Unstable P95276_MYCTO 0 45 COC[C@@H](C)Nc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O ZINC000217613699 GF In-Stock Unstable ADAMTS4 41 32 COCc1cc(=O)c(O)c([C@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccccc2OC)o1 ZINC000217613717 JI In-Stock Unstable RORC 37 40 C[C@H](Cc1ccnn1Cc1ccccc1)C(=O)O ZINC000217613745 BE For-Sale Unstable MME 59 37 C[C@H](Cc1ccnn1Cc1ccccc1)C(=O)O ZINC000217613745 BE For-Sale Unstable CYSP_TRYCR 44 32 C[C@H](Cc1ccnn1Cc1ccccc1)C(=O)O ZINC000217613745 BE For-Sale Unstable CPA1 52 34 C[C@H](Cc1ccnn1Cc1ccccc1)C(=O)O ZINC000217613745 BE For-Sale Unstable ACE2 47 34 O=C(c1cccc(Cl)c1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217613763 EE In-Stock Unstable AKR1C3 22 43 O=C(c1cccc(Cl)c1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217613763 EE In-Stock Unstable SLC6A7 0 41 O=C(N/C=C/c1ccccc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217613772 DF For-Sale Anodyne CA2 24 48 O=C(N/C=C/c1ccccc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217613772 DF For-Sale Anodyne CA1 43 36 O=C(N/C=C/c1ccccc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217613772 DF For-Sale Anodyne CA4 15 48 O=C(N/C=C/c1ccccc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217613772 DF For-Sale Anodyne CA12 34 42 O=C(N/C=C/c1ccccc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217613772 DF For-Sale Anodyne CA9 31 42 O=C(N/C=C/c1ccccc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217613772 DF For-Sale Anodyne F13A1 56 36 O=C(N/C=C/c1ccccc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217613772 DF For-Sale Anodyne IDO1 30 40 O=C(N/C=C/c1ccccc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217613772 DF For-Sale Anodyne MTCA1 46 48 O=C(N/C=C/c1ccccc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217613772 DF For-Sale Anodyne P96878_MYCTU 58 48 O=C(N/C=C/c1ccccc1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217613772 DF For-Sale Anodyne NAMPT 26 41 COCc1cc(=O)c(O)c([C@@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccccc2OC)o1 ZINC000217613793 JI In-Stock Unstable RORC 37 40 COC[C@H](C)Nc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O ZINC000217613794 GF In-Stock Unstable ADAMTS4 41 32 CN1CCCC[C@@H]1CN[C@H](c1ccccc1)c1ccco1 ZINC000217613809 CG For-Sale Unstable CHRNA10 55 40 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1ccc(O)cc1[N+](=O)[O-] ZINC000217613828 CI For-Sale Unstable SERPINE1 42 42 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1ccc(O)cc1[N+](=O)[O-] ZINC000217613828 CI For-Sale Unstable TRPM8 16 45 O=C(N/C=C/c1ccccc1)Nc1cccc(S(=O)(=O)O)c1 ZINC000217613871 DF For-Sale Anodyne CA4 18 40 O=C(N/C=C/c1ccccc1)Nc1cccc(S(=O)(=O)O)c1 ZINC000217613871 DF For-Sale Anodyne KCNK3 42 33 CN1CCCC[C@H]1CN[C@H](c1ccccc1)c1ccco1 ZINC000217613896 CG For-Sale Unstable CHRNA10 55 40 COc1ccc(-c2cc(C(=O)NC[C@@H]3CCCN4CCCC[C@H]34)n(C)n2)cc1OC ZINC000217613903 HG In-Stock Unstable STK17B 44 38 COc1ccc(-c2cc(C(=O)NC[C@@H]3CCCN4CCCC[C@H]34)n(C)n2)cc1OC ZINC000217613903 HG In-Stock Unstable SCARB1 21 40 COC(=O)c1ccc(S)c(C#N)c1 ZINC000217613906 AD For-Sale Unstable KDM5C 0 43 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1ccc(O)cc1[N+](=O)[O-] ZINC000217613909 CI For-Sale Unstable SERPINE1 42 42 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1ccc(O)cc1[N+](=O)[O-] ZINC000217613909 CI For-Sale Unstable TRPM8 16 45 Cc1ccc(C)c(S(=O)(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217613911 FG For-Sale Unstable NPY5R 27 47 CCCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217613921 FF In-Stock Unstable TBXA2R 54 43 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1ccc(O)cc1[N+](=O)[O-] ZINC000217613980 CI For-Sale Unstable SERPINE1 42 42 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1ccc(O)cc1[N+](=O)[O-] ZINC000217613980 CI For-Sale Unstable TRPM8 16 45 O=C(c1c[nH]c2ccccc12)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217613992 ED In-Stock Unstable AVPR1A 21 43 O=C(c1c[nH]c2ccccc12)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217613992 ED In-Stock Unstable HSP90AB1 15 44 Cc1ccc(C)c(S(=O)(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217614003 FG For-Sale Unstable NPY5R 27 47 CC(C)Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614041 FF In-Stock Unstable TBXA2R 54 43 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1ccc(O)cc1[N+](=O)[O-] ZINC000217614069 CI For-Sale Unstable SERPINE1 42 42 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1ccc(O)cc1[N+](=O)[O-] ZINC000217614069 CI For-Sale Unstable TRPM8 16 45 C[C@@H]1CN(C[C@@](N)(C(=O)O)c2ccccc2)CCCO1 ZINC000217614080 CD For-Sale Unstable AMY2 43 29 C[C@@H]1CN(C[C@@](N)(C(=O)O)c2ccccc2)CCCO1 ZINC000217614080 CD For-Sale Unstable CYP2J2 45 32 Cc1cccc(CS(=O)(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217614109 FF For-Sale Unstable NPY5R 24 42 CCCCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614160 GG In-Stock Unstable CA2 17 43 CCCCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614160 GG In-Stock Unstable TBXA2R 53 42 CCCCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614160 GG In-Stock Unstable CASP3 17 40 CCCCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614160 GG In-Stock Unstable CA1 15 43 CCCCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614160 GG In-Stock Unstable ALOX15 67 41 C[C@H]1CN(C[C@@](N)(C(=O)O)c2ccccc2)CCCO1 ZINC000217614164 CD For-Sale Unstable AMY2 43 29 C[C@H]1CN(C[C@@](N)(C(=O)O)c2ccccc2)CCCO1 ZINC000217614164 CD For-Sale Unstable CYP2J2 45 32 CC(C)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217614184 CJ For-Sale Unstable CA1 25 44 CC(C)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217614184 CJ For-Sale Unstable ACAT 0 50 CC(C)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217614184 CJ For-Sale Unstable P95276_MYCTO 0 41 Cc1cccc(CS(=O)(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217614190 FF For-Sale Unstable NPY5R 24 42 O=C(c1ccccc1Br)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217614193 GE In-Stock Unstable HSP90AB1 0 47 COc1ccc(CN2C(=O)N[C@@H](CCC(=O)NCc3ccncc3)C2=O)cc1OC ZINC000217614205 HD In-Stock Unstable ENPP1 60 32 CC(C)CNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614267 GF In-Stock Unstable CA2 18 43 CC(C)CNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614267 GF In-Stock Unstable ADRB3 47 37 CC(C)CNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614267 GF In-Stock Unstable TBXA2R 53 42 CC(C)CNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614267 GF In-Stock Unstable CASP3 18 40 CC(C)CNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614267 GF In-Stock Unstable CA1 15 43 CC(C)CNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614267 GF In-Stock Unstable CA5B 29 40 CC(C)CNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614267 GF In-Stock Unstable CA5A 33 40 CC(C)CNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614267 GF In-Stock Unstable ALOX15 46 33 CC(C)CNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614267 GF In-Stock Unstable MTNN 64 35 CC(C)CNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614267 GF In-Stock Unstable SFRP1 15 49 COc1ccccc1NC(=O)N/C=C/c1ccccc1 ZINC000217614285 CG For-Sale Unstable TLR4 22 40 COc1cccc(S(=O)(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217614293 FF For-Sale Unstable NPY5R 23 45 COc1cccc(S(=O)(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217614293 FF For-Sale Unstable PKM 23 48 Cc1c(C(=O)N2Cc3cnc(N4CCOCC4)nc3C2)cnn1-c1ccccc1 ZINC000217614300 GD In-Stock Unstable HSP90AB1 0 44 COc1ccc2c(c1OC)C(=O)O[C@@H]2CC(=O)Nc1ccc(CC(=O)O)cc1 ZINC000217614314 GF In-Stock Unstable TSHR 48 32 COc1ccc2c(c1OC)C(=O)O[C@@H]2CC(=O)Nc1ccc(CC(=O)O)cc1 ZINC000217614314 GF In-Stock Unstable SELL 0 40 COC(=O)c1ccccc1CN1CC[C@H]2CC[C@@H](C1)N2C ZINC000217614337 CE For-Sale Unstable SLC6A1 66 36 COC(=O)c1ccccc1CN1CC[C@H]2CC[C@@H](C1)N2C ZINC000217614337 CE For-Sale Unstable SLC6A3 30 49 COC(=O)c1ccccc1CN1CC[C@H]2CC[C@@H](C1)N2C ZINC000217614337 CE For-Sale Unstable CCR5 20 40 COC(=O)c1ccccc1CN1CC[C@H]2CC[C@@H](C1)N2C ZINC000217614337 CE For-Sale Unstable GLRA1 44 33 CC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614376 GG In-Stock Unstable CA2 17 43 CC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614376 GG In-Stock Unstable TBXA2R 48 42 CC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614376 GG In-Stock Unstable CA1 15 43 CC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614376 GG In-Stock Unstable CA4 17 43 CC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614376 GG In-Stock Unstable ALOX15 49 35 COc1cccc(S(=O)(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217614385 FF For-Sale Unstable NPY5R 23 45 COc1cccc(S(=O)(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217614385 FF For-Sale Unstable PKM 23 48 COc1ccc2c(c1OC)C(=O)O[C@H]2CC(=O)Nc1ccc(CC(=O)O)cc1 ZINC000217614395 GF In-Stock Unstable TSHR 48 32 COc1ccc2c(c1OC)C(=O)O[C@H]2CC(=O)Nc1ccc(CC(=O)O)cc1 ZINC000217614395 GF In-Stock Unstable SELL 0 40 O=C(COc1ccc(Cl)cc1Cl)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217614399 HF In-Stock Unstable MAPK1 43 38 O=C(COc1ccc(Cl)cc1Cl)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217614399 HF In-Stock Unstable AKR1C3 0 40 CCOC(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217614403 BE On-Demand Unstable PRSS1 16 43 CCOC(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217614403 BE On-Demand Unstable CA1 16 42 CCOC(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217614403 BE On-Demand Unstable CA7 17 41 CCOC(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217614403 BE On-Demand Unstable CA14 15 41 CCOC(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217614403 BE On-Demand Unstable ACR 68 43 CCOC(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217614403 BE On-Demand Unstable CNGA1 0 44 CCOC(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217614403 BE On-Demand Unstable NOD2 17 43 CC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614442 GG In-Stock Unstable CA2 17 43 CC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614442 GG In-Stock Unstable TBXA2R 48 42 CC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614442 GG In-Stock Unstable CA1 15 43 CC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614442 GG In-Stock Unstable CA4 17 43 CC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614442 GG In-Stock Unstable ALOX15 49 35 O=C(N/C=C/c1ccccc1)Nc1ccc(Cl)c(Cl)c1 ZINC000217614478 DJ For-Sale Anodyne PYGL 25 42 O=C(N/C=C/c1ccccc1)Nc1ccc(Cl)c(Cl)c1 ZINC000217614478 DJ For-Sale Anodyne GRM4 42 38 O=C(N/C=C/c1ccccc1)Nc1ccc(Cl)c(Cl)c1 ZINC000217614478 DJ For-Sale Anodyne SMO 17 47 O=C(N/C=C/c1ccccc1)Nc1ccc(Cl)c(Cl)c1 ZINC000217614478 DJ For-Sale Anodyne BLM 0 43 O=C(N/C=C/c1ccccc1)Nc1ccc(Cl)c(Cl)c1 ZINC000217614478 DJ For-Sale Anodyne P95276_MYCTO 0 53 O=C(N/C=C/c1ccccc1)Nc1ccc(Cl)c(Cl)c1 ZINC000217614478 DJ For-Sale Anodyne WRN 0 43 O=C(N/C=C/c1ccccc1)Nc1ccc(Cl)c(Cl)c1 ZINC000217614478 DJ For-Sale Anodyne PPX1 0 44 Cc1cc(NC(=O)c2ccc(-n3cccc3)cc2)n(-c2ccc(F)cc2)n1 ZINC000217614499 FI On-Demand Unstable GRM5 15 57 Cc1cc(NC(=O)c2ccc(-n3cccc3)cc2)n(-c2ccc(F)cc2)n1 ZINC000217614499 FI On-Demand Unstable AOC2 0 44 COc1ccccc1S(=O)(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217614508 FF For-Sale Unstable NPY5R 26 48 O=C(Cn1ncccc1=O)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217614525 EB In-Stock Unstable HSP90AB1 15 44 O=C(CCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCCc1c[nH]cn1 ZINC000217614526 HE In-Stock Unstable HRH2 45 40 O=C(CCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCCc1c[nH]cn1 ZINC000217614526 HE In-Stock Unstable HRH3 42 52 O=C(CCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCCc1c[nH]cn1 ZINC000217614526 HE In-Stock Unstable HRH4 27 40 CC(C)(C)Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614553 GG In-Stock Unstable CA2 20 45 CC(C)(C)Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614553 GG In-Stock Unstable TBXA2R 54 43 CC(C)(C)Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614553 GG In-Stock Unstable CA1 16 40 CC(C)(C)Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614553 GG In-Stock Unstable CA7 16 40 CC(C)(C)Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614553 GG In-Stock Unstable PRTN3 47 34 CC(C)(C)Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614553 GG In-Stock Unstable ALOX15 47 34 CC(C)(C)Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614553 GG In-Stock Unstable TPSAB1 15 41 CC(C)(C)Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614553 GG In-Stock Unstable AKR1C3 24 59 CC(C)(C)Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614553 GG In-Stock Unstable SFRP1 26 51 CC(C)CCNC(=O)C(F)F ZINC000217614581 AD On-Demand Unstable PGA 44 40 CC(C)CCNC(=O)C(F)F ZINC000217614581 AD On-Demand Unstable DNPEP 0 50 COc1ccccc1S(=O)(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217614586 FF For-Sale Unstable NPY5R 26 48 Cc1ccc(NC(=O)N/C=C/c2ccccc2)cc1Cl ZINC000217614595 CI For-Sale Unstable PPIA 15 40 Cc1ccc(NC(=O)N/C=C/c2ccccc2)cc1Cl ZINC000217614595 CI For-Sale Unstable LPL 44 33 O=C(CCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCCc1c[nH]cn1 ZINC000217614599 HE In-Stock Unstable HRH2 45 40 O=C(CCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCCc1c[nH]cn1 ZINC000217614599 HE In-Stock Unstable HRH3 42 52 O=C(CCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCCc1c[nH]cn1 ZINC000217614599 HE In-Stock Unstable HRH4 27 40 O=C(c1ccc(S(=O)(=O)N2CCCC2)cc1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217614620 ID In-Stock Unstable NAMPT 35 40 O=C(O)/C=C\c1ccc(C(=O)NCCCn2ccnc2)s1 ZINC000217614631 DD For-Sale Unstable TBXAS1 65 67 O=C(O)/C=C\c1ccc(C(=O)NCCCn2ccnc2)s1 ZINC000217614631 DD For-Sale Unstable HMOX2 49 36 O=C(O)/C=C\c1ccc(C(=O)NCCCn2ccnc2)s1 ZINC000217614631 DD For-Sale Unstable QPCT 42 43 O=C(O)/C=C\c1ccc(C(=O)NCCCn2ccnc2)s1 ZINC000217614631 DD For-Sale Unstable NAMPT 26 45 CN1C[C@@H](CNC(=O)c2ccccc2N2CCCC2)OCC1=O ZINC000217614642 DC In-Stock Unstable KCNQ2 66 33 C=CCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614643 FF In-Stock Unstable TBXA2R 47 42 C=CCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217614643 FF In-Stock Unstable BDKRB1 0 42 O=C1O[C@@]2(CCCN(S(=O)(=O)Cc3cccc(F)c3)C2)c2ccccc21 ZINC000217614688 GF For-Sale Unstable NPY5R 26 44 Cc1cccc(C(C)C)c1NC(=O)N/C=C/c1ccccc1 ZINC000217614697 CJ For-Sale Unstable SOAT1 58 41 Cc1cccc(C(C)C)c1NC(=O)N/C=C/c1ccccc1 ZINC000217614697 CJ For-Sale Unstable ACAT 0 51 COc1ccc2c(c1)CCC[C@@H]2NC[C@@H]1CCCCN1C ZINC000217614705 CG For-Sale Unstable DRD4 41 33 COc1ccc2c(c1)CCC[C@@H]2NC[C@@H]1CCCCN1C ZINC000217614705 CG For-Sale Unstable BDKRB1 39 44 COc1ccc2c(c1)CCC[C@@H]2NC[C@@H]1CCCCN1C ZINC000217614705 CG For-Sale Unstable EBP 45 50 COc1ccc2c(c1)CCC[C@@H]2NC[C@@H]1CCCCN1C ZINC000217614705 CG For-Sale Unstable CHRNA10 68 46 COC(=O)[C@](N)(CN1CCCO[C@@H](C)C1)c1ccccc1 ZINC000217614711 CD For-Sale Unstable AMY2 46 31 O=C(c1cc(-c2ccc(F)cc2)n[nH]1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217614718 GD In-Stock Unstable TACR3 17 43 O=C(c1cc(-c2ccc(F)cc2)n[nH]1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217614718 GD In-Stock Unstable MTOR 22 42 CN1C[C@H](CNC(=O)c2ccccc2N2CCCC2)OCC1=O ZINC000217614727 DC In-Stock Unstable KCNQ2 66 33 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NC1CC1 ZINC000217614766 FE In-Stock Unstable TBXA2R 48 43 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NC1CC1 ZINC000217614766 FE In-Stock Unstable ALOX15 49 36 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NC1CC1 ZINC000217614766 FE In-Stock Unstable SFRP1 70 45 O=C1O[C@]2(CCCN(S(=O)(=O)Cc3cccc(F)c3)C2)c2ccccc21 ZINC000217614770 GF For-Sale Unstable NPY5R 26 44 COc1ccc2c(c1)CCC[C@@H]2NC[C@H]1CCCCN1C ZINC000217614785 CG For-Sale Unstable DRD4 41 33 COc1ccc2c(c1)CCC[C@@H]2NC[C@H]1CCCCN1C ZINC000217614785 CG For-Sale Unstable BDKRB1 39 44 COc1ccc2c(c1)CCC[C@@H]2NC[C@H]1CCCCN1C ZINC000217614785 CG For-Sale Unstable EBP 45 50 COc1ccc2c(c1)CCC[C@@H]2NC[C@H]1CCCCN1C ZINC000217614785 CG For-Sale Unstable CHRNA10 68 46 O=C(NCC1CCCCC1)C(F)F ZINC000217614789 AD On-Demand Unstable ADH4 0 41 O=C(N/C=C/c1ccccc1)Nc1ccccc1C(F)(F)F ZINC000217614815 DI For-Sale Anodyne RBP4 54 36 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NC1CCCC1 ZINC000217614869 GG In-Stock Unstable ADRB3 28 41 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NC1CCCC1 ZINC000217614869 GG In-Stock Unstable TBXA2R 46 41 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NC1CCCC1 ZINC000217614869 GG In-Stock Unstable CASP3 0 42 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NC1CCCC1 ZINC000217614869 GG In-Stock Unstable ALOX15 45 40 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NC1CCCC1 ZINC000217614869 GG In-Stock Unstable SFRP1 74 43 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NC1CCCC1 ZINC000217614869 GG In-Stock Unstable WNT3 50 33 Cc1cc(F)ccc1S(=O)(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217614895 GF For-Sale Unstable NPY5R 26 45 Cc1cc(NC(=O)c2sc(NC(=O)c3ccco3)cc2C)n(-c2ccc(F)cc2)n1 ZINC000217614912 HJ On-Demand Unstable KISS1R 42 32 O=C(N/C=C/c1ccccc1)Nc1ccc(C(=O)O)cc1 ZINC000217614924 CG For-Sale Anodyne EPHX1 0 44 O=C(N/C=C/c1ccccc1)Nc1ccc(C(=O)O)cc1 ZINC000217614924 CG For-Sale Anodyne EPHX2 15 44 O=C(N/C=C/c1ccccc1)Nc1ccc(C(=O)O)cc1 ZINC000217614924 CG For-Sale Anodyne P95276_MYCTO 0 44 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCCC(=O)NCc3ccccn3)[C@H]21 ZINC000217614940 JG In-Stock Unstable HTR7 24 46 Cc1nonc1CC(=O)N1CCC[C@@H](Cn2ccnc2)C1 ZINC000217614966 CD In-Stock Unstable CAMC 0 45 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NC1CCCCC1 ZINC000217614968 HH In-Stock Unstable ADRB3 30 43 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NC1CCCCC1 ZINC000217614968 HH In-Stock Unstable TBXA2R 47 43 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NC1CCCCC1 ZINC000217614968 HH In-Stock Unstable CASP3 0 41 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NC1CCCCC1 ZINC000217614968 HH In-Stock Unstable ALOX15 39 42 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NC1CCCCC1 ZINC000217614968 HH In-Stock Unstable EPHX2 21 40 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NC1CCCCC1 ZINC000217614968 HH In-Stock Unstable SFRP1 67 42 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NC1CCCCC1 ZINC000217614968 HH In-Stock Unstable WNT3 47 32 Cc1cc(F)ccc1S(=O)(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217614988 GF For-Sale Unstable NPY5R 26 45 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCCC(=O)NCc3ccccn3)[C@@H]21 ZINC000217615019 JG In-Stock Unstable HTR7 24 46 Cc1c(Cl)cccc1NC(=O)N/C=C/c1ccccc1 ZINC000217615029 CI For-Sale Unstable LPL 47 35 Cc1c(Cl)cccc1NC(=O)N/C=C/c1ccccc1 ZINC000217615029 CI For-Sale Unstable CXCL8 49 38 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCCC1=CCCCC1 ZINC000217615044 II In-Stock Unstable TBXA2R 50 40 Cc1nonc1CC(=O)N1CCC[C@H](Cn2ccnc2)C1 ZINC000217615051 CD In-Stock Unstable CAMC 0 45 Cc1cc(S(=O)(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)ccc1F ZINC000217615095 GF For-Sale Unstable NPY5R 24 40 COc1cccc(C(=O)Nc2ncc(Cc3ccc(Br)cc3)s2)c1OC(F)F ZINC000217615126 JK On-Demand Unstable SCD1 43 44 COc1cccc(C(=O)Nc2ncc(Cc3ccc(Br)cc3)s2)c1OC(F)F ZINC000217615126 JK On-Demand Unstable SCD 39 45 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCCO ZINC000217615141 FD In-Stock Unstable CA2 19 46 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCCO ZINC000217615141 FD In-Stock Unstable TBXA2R 54 44 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCCO ZINC000217615141 FD In-Stock Unstable CA1 15 46 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCCO ZINC000217615141 FD In-Stock Unstable CA7 16 40 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCCO ZINC000217615141 FD In-Stock Unstable BDKRB1 0 41 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCCO ZINC000217615141 FD In-Stock Unstable A6YCJ1_9METZ 15 40 CCOC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217615151 DH For-Sale Unstable CA1 41 43 CCOC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217615151 DH For-Sale Unstable ACR 70 41 CCOC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217615151 DH For-Sale Unstable CA12 15 51 CCOC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217615151 DH For-Sale Unstable CA9 18 51 CCOC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217615151 DH For-Sale Unstable NOD2 17 42 O=C(NCC(=O)N1Cc2cnc(N3CCOCC3)nc2C1)OCc1ccccc1 ZINC000217615170 GD In-Stock Unstable NPR 55 31 Cc1cc(S(=O)(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)ccc1F ZINC000217615174 GF For-Sale Unstable NPY5R 24 40 O=C(O)/C=C\c1cccc(NS(=O)(=O)c2ccc(Cl)s2)n1 ZINC000217615245 EF For-Sale Anodyne CCR4 54 35 O=C(O)/C=C\c1cccc(NS(=O)(=O)c2ccc(Cl)s2)n1 ZINC000217615245 EF For-Sale Anodyne NFKBIA 0 45 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCCCO ZINC000217615252 GD In-Stock Unstable TBXA2R 52 43 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCCCO ZINC000217615252 GD In-Stock Unstable BDKRB1 0 42 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCCCO ZINC000217615252 GD In-Stock Unstable ALOX15 45 33 O=C(NC(c1ccccc1)c1ccccc1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217615265 HG In-Stock Unstable PIK3CA 25 42 O=C(NC(c1ccccc1)c1ccccc1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217615265 HG In-Stock Unstable MAPK1 52 40 O=C(NC(c1ccccc1)c1ccccc1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217615265 HG In-Stock Unstable MTOR 35 42 O=C(NC(c1ccccc1)c1ccccc1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217615265 HG In-Stock Unstable PIK3CG 22 42 O=C(N/C=C/c1ccccc1)Nc1ccccc1Cl ZINC000217615266 CI For-Sale Anodyne CXCL8 56 44 O=C(N/C=C/c1ccccc1)Nc1ccccc1Cl ZINC000217615266 CI For-Sale Anodyne EPHB3 52 37 O=C1O[C@@]2(CCCN(S(=O)(=O)Cc3ccc(F)cc3)C2)c2ccccc21 ZINC000217615281 GF For-Sale Unstable NPY5R 28 45 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCc1ccccn1 ZINC000217615328 IG In-Stock Unstable TOP1 0 40 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCc1ccccn1 ZINC000217615328 IG In-Stock Unstable SCN9A 0 44 O=C1O[C@]2(CCCN(S(=O)(=O)Cc3ccc(F)cc3)C2)c2ccccc21 ZINC000217615349 GF For-Sale Unstable NPY5R 28 45 O=S(=O)(c1ccccc1)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217615375 ED In-Stock Unstable AKR1C3 42 39 CC(C)c1ccccc1NC(=O)N/C=C/c1ccccc1 ZINC000217615388 CJ For-Sale Unstable ACAT 0 46 COCCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217615391 GD In-Stock Unstable CA2 18 47 COCCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217615391 GD In-Stock Unstable TBXA2R 53 41 COCCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217615391 GD In-Stock Unstable CA1 18 43 COCCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217615391 GD In-Stock Unstable BDKRB1 0 45 COCCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217615391 GD In-Stock Unstable PRTN3 44 31 COCCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217615391 GD In-Stock Unstable ALOX15 45 35 COCCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217615391 GD In-Stock Unstable AKR1C3 17 53 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCc1ccccn1 ZINC000217615411 IG In-Stock Unstable TOP1 0 40 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCc1ccccn1 ZINC000217615411 IG In-Stock Unstable SCN9A 0 44 O=C(CCc1nc2ccccc2[nH]1)N[C@@H]1CCCN(c2cnccn2)C1 ZINC000217615415 FE In-Stock Unstable ISPE 0 41 O=C(c1ccc(NS(=O)(=O)c2cccc3ccccc23)cc1)N1CCC(O)(c2ccccc2Cl)CC1 ZINC000217615430 KK Annotated Unstable CCR1 18 44 O=C(CCc1nc2ccccc2[nH]1)N[C@H]1CCCN(c2cnccn2)C1 ZINC000217615486 FE In-Stock Unstable ISPE 0 41 COCCCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217615489 GE In-Stock Unstable CA2 15 43 COCCCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217615489 GE In-Stock Unstable TBXA2R 52 40 COCCCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217615489 GE In-Stock Unstable BDKRB1 0 46 COCCCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217615489 GE In-Stock Unstable ALOX15 50 36 COCCCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217615489 GE In-Stock Unstable AKR1C3 17 51 O=C(N/C=C/c1ccccc1)Nc1cccc(Cl)c1Cl ZINC000217615499 DJ For-Sale Anodyne CXCL8 54 38 O=C(C[C@@H]1NC(=O)N(CCc2cccc(F)c2)C1=O)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217615521 IE In-Stock Unstable CACNA1G 23 42 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCc1ccccc1 ZINC000217615588 HH In-Stock Unstable CA2 24 47 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCc1ccccc1 ZINC000217615588 HH In-Stock Unstable GNRHR 15 41 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCc1ccccc1 ZINC000217615588 HH In-Stock Unstable TBXA2R 55 45 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCc1ccccc1 ZINC000217615588 HH In-Stock Unstable TBXAS1 38 40 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCc1ccccc1 ZINC000217615588 HH In-Stock Unstable CA6 15 41 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCc1ccccc1 ZINC000217615588 HH In-Stock Unstable CA1 26 47 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCc1ccccc1 ZINC000217615588 HH In-Stock Unstable CA7 24 41 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCc1ccccc1 ZINC000217615588 HH In-Stock Unstable BDKRB1 0 42 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCc1ccccc1 ZINC000217615588 HH In-Stock Unstable CA5B 42 40 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCc1ccccc1 ZINC000217615588 HH In-Stock Unstable CA4 16 47 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCc1ccccc1 ZINC000217615588 HH In-Stock Unstable CA5A 44 40 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCc1ccccc1 ZINC000217615588 HH In-Stock Unstable ALOX15 46 36 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCc1ccccc1 ZINC000217615588 HH In-Stock Unstable CA12 17 41 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCc1ccccc1 ZINC000217615588 HH In-Stock Unstable TPSAB1 15 40 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCc1ccccc1 ZINC000217615588 HH In-Stock Unstable CA9 20 41 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCc1ccccc1 ZINC000217615588 HH In-Stock Unstable AKR1C3 15 58 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCc1ccccc1 ZINC000217615588 HH In-Stock Unstable A6YCJ1_9METZ 22 41 O=C(N/C=C/c1ccccc1)Nc1cc(Cl)ccc1Cl ZINC000217615599 DJ For-Sale Anodyne CXCL8 19 48 O=C(N/C=C/c1ccccc1)Nc1cc(Cl)ccc1Cl ZINC000217615599 DJ For-Sale Anodyne CMA1 22 45 O=C1O[C@@]2(CCCN(S(=O)(=O)c3cccc(Cl)c3)C2)c2ccccc21 ZINC000217615653 GG For-Sale Unstable NPY5R 26 43 O=C(O)/C=C\c1ccc(N2C(=O)CCCCC2=O)c(F)c1 ZINC000217615694 CE For-Sale Unstable PPOX1 17 40 C[C@@H](Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217615721 HI In-Stock Unstable ADRB1 28 40 C[C@@H](Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217615721 HI In-Stock Unstable ADRB3 49 40 C[C@@H](Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217615721 HI In-Stock Unstable TBXA2R 47 41 C[C@@H](Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217615721 HI In-Stock Unstable TBXAS1 33 40 C[C@@H](Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217615721 HI In-Stock Unstable CASP3 19 41 C[C@@H](Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217615721 HI In-Stock Unstable BDKRB1 0 43 C[C@@H](Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217615721 HI In-Stock Unstable ALOX15 40 34 COc1ccc(NC(=O)N/C=C/c2ccccc2)cc1Cl ZINC000217615731 DI For-Sale Unstable GCGR 0 41 COc1ccc(NC(=O)N/C=C/c2ccccc2)cc1Cl ZINC000217615731 DI For-Sale Unstable GRM4 24 53 COc1ccc(NC(=O)N/C=C/c2ccccc2)cc1Cl ZINC000217615731 DI For-Sale Unstable IMPDH2 0 43 COc1ccc(NC(=O)N/C=C/c2ccccc2)cc1Cl ZINC000217615731 DI For-Sale Unstable CYSP_PLAFA 40 33 O=C1O[C@]2(CCCN(S(=O)(=O)c3cccc(Cl)c3)C2)c2ccccc21 ZINC000217615733 GG For-Sale Unstable NPY5R 26 43 C[C@H](Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217615811 HI In-Stock Unstable ADRB1 28 40 C[C@H](Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217615811 HI In-Stock Unstable ADRB3 49 40 C[C@H](Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217615811 HI In-Stock Unstable TBXA2R 47 41 C[C@H](Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217615811 HI In-Stock Unstable TBXAS1 33 40 C[C@H](Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217615811 HI In-Stock Unstable CASP3 19 41 C[C@H](Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217615811 HI In-Stock Unstable BDKRB1 0 43 C[C@H](Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217615811 HI In-Stock Unstable ALOX15 40 34 O=C1O[C@@]2(CCCN(S(=O)(=O)c3ccccc3Cl)C2)c2ccccc21 ZINC000217615818 GG For-Sale Unstable NPY5R 26 45 O=S(=O)(c1c(F)cccc1F)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217615821 GD In-Stock Unstable PKM 21 45 O=C(N/C=C/c1ccccc1)Nc1cccc(C(F)(F)F)c1 ZINC000217615844 DI For-Sale Anodyne KIT 17 43 O=C(N/C=C/c1ccccc1)Nc1cccc(C(F)(F)F)c1 ZINC000217615844 DI For-Sale Anodyne UL80 22 43 O=C(N/C=C/c1ccccc1)Nc1cccc(C(F)(F)F)c1 ZINC000217615844 DI For-Sale Anodyne KDR 17 42 O=C(N/C=C/c1ccccc1)Nc1cccc(C(F)(F)F)c1 ZINC000217615844 DI For-Sale Anodyne EPHX2 19 50 O=C(N/C=C/c1ccccc1)Nc1cccc(C(F)(F)F)c1 ZINC000217615844 DI For-Sale Anodyne TEK 27 41 O=C(N/C=C/c1ccccc1)Nc1cccc(C(F)(F)F)c1 ZINC000217615844 DI For-Sale Anodyne EPHB4 26 40 O=C(N/C=C/c1ccccc1)Nc1cccc(C(F)(F)F)c1 ZINC000217615844 DI For-Sale Anodyne AKR1C3 20 51 O=C(N/C=C/c1ccccc1)Nc1cccc(C(F)(F)F)c1 ZINC000217615844 DI For-Sale Anodyne RIPK1 50 44 O=C(N/C=C/c1ccccc1)Nc1cccc(C(F)(F)F)c1 ZINC000217615844 DI For-Sale Anodyne TRPM4 0 50 O=C(N/C=C/c1ccccc1)Nc1cccc(C(F)(F)F)c1 ZINC000217615844 DI For-Sale Anodyne KCNK3 63 51 CN1CCCC[C@@H]1CNC[C@@H](O)COc1ccc(F)cc1 ZINC000217615872 CD For-Sale Unstable ADRB2 54 46 CN1CCCC[C@@H]1CNC[C@@H](O)COc1ccc(F)cc1 ZINC000217615872 CD For-Sale Unstable ADRB1 69 46 CN1CCCC[C@@H]1CNC[C@@H](O)COc1ccc(F)cc1 ZINC000217615872 CD For-Sale Unstable GRIN1 24 42 CN1CCCC[C@@H]1CNC[C@@H](O)COc1ccc(F)cc1 ZINC000217615872 CD For-Sale Unstable ADRB3 50 41 CN1CCCC[C@@H]1CNC[C@@H](O)COc1ccc(F)cc1 ZINC000217615872 CD For-Sale Unstable CHRNA10 70 40 O=C1O[C@]2(CCCN(S(=O)(=O)c3ccccc3Cl)C2)c2ccccc21 ZINC000217615897 GG For-Sale Unstable NPY5R 26 45 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCCc1ccccc1 ZINC000217615910 HH In-Stock Unstable CA2 29 49 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCCc1ccccc1 ZINC000217615910 HH In-Stock Unstable TBXA2R 57 46 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCCc1ccccc1 ZINC000217615910 HH In-Stock Unstable TBXAS1 42 42 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCCc1ccccc1 ZINC000217615910 HH In-Stock Unstable CASP3 18 40 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCCc1ccccc1 ZINC000217615910 HH In-Stock Unstable CA1 30 49 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCCc1ccccc1 ZINC000217615910 HH In-Stock Unstable CA7 25 43 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCCc1ccccc1 ZINC000217615910 HH In-Stock Unstable BDKRB1 0 43 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCCc1ccccc1 ZINC000217615910 HH In-Stock Unstable CA5B 43 42 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCCc1ccccc1 ZINC000217615910 HH In-Stock Unstable CA4 19 49 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCCc1ccccc1 ZINC000217615910 HH In-Stock Unstable CA5A 45 42 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCCc1ccccc1 ZINC000217615910 HH In-Stock Unstable CA14 16 43 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCCc1ccccc1 ZINC000217615910 HH In-Stock Unstable ALOX15 49 35 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCCc1ccccc1 ZINC000217615910 HH In-Stock Unstable CA12 19 43 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCCc1ccccc1 ZINC000217615910 HH In-Stock Unstable TPSAB1 15 41 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCCc1ccccc1 ZINC000217615910 HH In-Stock Unstable AKR1C3 17 61 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCCc1ccccc1 ZINC000217615910 HH In-Stock Unstable A6YCJ1_9METZ 22 43 CN1CCCC[C@H]1CNC[C@@H](O)COc1ccc(F)cc1 ZINC000217615960 CD For-Sale Unstable ADRB2 54 46 CN1CCCC[C@H]1CNC[C@@H](O)COc1ccc(F)cc1 ZINC000217615960 CD For-Sale Unstable ADRB1 69 46 CN1CCCC[C@H]1CNC[C@@H](O)COc1ccc(F)cc1 ZINC000217615960 CD For-Sale Unstable GRIN1 24 42 CN1CCCC[C@H]1CNC[C@@H](O)COc1ccc(F)cc1 ZINC000217615960 CD For-Sale Unstable ADRB3 50 41 CN1CCCC[C@H]1CNC[C@@H](O)COc1ccc(F)cc1 ZINC000217615960 CD For-Sale Unstable CHRNA10 70 40 O=C1O[C@@]2(CCCN(S(=O)(=O)c3ccc(F)c(F)c3)C2)c2ccccc21 ZINC000217616010 GF For-Sale Unstable NPY5R 25 42 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1 ZINC000217616018 JH In-Stock Unstable CA2 25 44 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1 ZINC000217616018 JH In-Stock Unstable TBXA2R 55 46 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1 ZINC000217616018 JH In-Stock Unstable TBXAS1 32 46 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1 ZINC000217616018 JH In-Stock Unstable HTR7 17 40 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1 ZINC000217616018 JH In-Stock Unstable BMP1 80 42 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1 ZINC000217616018 JH In-Stock Unstable CA1 26 45 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1 ZINC000217616018 JH In-Stock Unstable KCNA5 26 40 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1 ZINC000217616018 JH In-Stock Unstable MMP13 78 44 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1 ZINC000217616018 JH In-Stock Unstable BDKRB1 0 42 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1 ZINC000217616018 JH In-Stock Unstable ADAM17 55 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1 ZINC000217616018 JH In-Stock Unstable ALOX15B 0 42 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1 ZINC000217616018 JH In-Stock Unstable CA14 18 45 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1 ZINC000217616018 JH In-Stock Unstable MMP2 50 42 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1 ZINC000217616018 JH In-Stock Unstable MMP3 56 42 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1 ZINC000217616018 JH In-Stock Unstable MMP8 35 40 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1 ZINC000217616018 JH In-Stock Unstable MMP14 27 40 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1 ZINC000217616018 JH In-Stock Unstable PRTN3 47 33 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1 ZINC000217616018 JH In-Stock Unstable ALOX15 69 42 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1 ZINC000217616018 JH In-Stock Unstable MMP9 68 44 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1 ZINC000217616018 JH In-Stock Unstable MMP12 39 40 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1 ZINC000217616018 JH In-Stock Unstable CA12 19 44 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1 ZINC000217616018 JH In-Stock Unstable PTGDR 24 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1 ZINC000217616018 JH In-Stock Unstable MMP7 42 42 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1 ZINC000217616018 JH In-Stock Unstable IAP 0 46 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1 ZINC000217616018 JH In-Stock Unstable CA9 28 44 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1 ZINC000217616018 JH In-Stock Unstable MMP1 67 42 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1 ZINC000217616018 JH In-Stock Unstable AKR1C3 34 54 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1 ZINC000217616018 JH In-Stock Unstable AKR1C2 53 39 Nc1cc(C(F)(F)F)ccc1CCC(=O)O ZINC000217616019 BE In-Stock Unstable FFAR1 20 45 CCOC(=O)c1ccccc1NC(=O)N/C=C/c1ccccc1 ZINC000217616079 DH For-Sale Unstable ADORA3 16 45 O=C1O[C@]2(CCCN(S(=O)(=O)c3ccc(F)c(F)c3)C2)c2ccccc21 ZINC000217616087 GF For-Sale Unstable NPY5R 25 42 COc1ccc(C(=O)NCC(F)(F)F)cc1/C=C\C(=O)O ZINC000217616089 DE For-Sale Unstable PPARD 16 41 CS(=O)(=O)Nc1cccc2c1ccn2CC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217616100 ID In-Stock Unstable CHRNA4 28 46 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1OC ZINC000217616137 JH In-Stock Unstable CA2 15 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1OC ZINC000217616137 JH In-Stock Unstable TBXA2R 53 45 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1OC ZINC000217616137 JH In-Stock Unstable TBXAS1 28 48 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1OC ZINC000217616137 JH In-Stock Unstable CA1 15 48 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1OC ZINC000217616137 JH In-Stock Unstable CA7 17 45 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1OC ZINC000217616137 JH In-Stock Unstable BDKRB1 0 42 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1OC ZINC000217616137 JH In-Stock Unstable CA14 15 48 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1OC ZINC000217616137 JH In-Stock Unstable ALOX15 46 38 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1OC ZINC000217616137 JH In-Stock Unstable PTGDR 20 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1OC ZINC000217616137 JH In-Stock Unstable IAP 0 47 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1OC ZINC000217616137 JH In-Stock Unstable AKR1C3 18 49 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccccc3)cc2C(=O)O)cc1OC ZINC000217616137 JH In-Stock Unstable SCMU_MYCTU 0 45 O=C(N/C=C/c1ccccc1)Nc1ccc(O)cc1 ZINC000217616193 CG For-Sale Anodyne EPHX1 0 45 O=C(N/C=C/c1ccccc1)Nc1ccc(O)cc1 ZINC000217616193 CG For-Sale Anodyne F3 26 46 O=C(N/C=C/c1ccccc1)Nc1ccc(O)cc1 ZINC000217616193 CG For-Sale Anodyne MMP2 22 62 O=C(N/C=C/c1ccccc1)Nc1ccc(O)cc1 ZINC000217616193 CG For-Sale Anodyne MMP9 16 62 O=C(N/C=C/c1ccccc1)Nc1ccc(O)cc1 ZINC000217616193 CG For-Sale Anodyne MMP1 0 62 O=C(N/C=C/c1ccccc1)Nc1ccc(O)cc1 ZINC000217616193 CG For-Sale Anodyne CYP2B1 0 40 O=C(N/C=C/c1ccccc1)Nc1ccc(O)cc1 ZINC000217616193 CG For-Sale Anodyne P95276_MYCTO 0 45 O=C1O[C@@]2(CCCN(S(=O)(=O)c3cc(F)ccc3F)C2)c2ccccc21 ZINC000217616203 GF For-Sale Unstable NPY5R 27 46 COc1cc2c(cc1OC)CN(C(=O)c1cnc3c(Cl)cccc3c1O)CC2 ZINC000217616208 GH In-Stock Unstable ABCB1B 57 36 COc1cc2c(cc1OC)CN(C(=O)c1cnc3c(Cl)cccc3c1O)CC2 ZINC000217616208 GH In-Stock Unstable ABCB1 20 43 N#Cc1cccc(NC(=O)c2ccc(/C=C\C(=O)O)s2)c1 ZINC000217616254 CF For-Sale Mild KCNK3 56 36 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NCc1ccco1 ZINC000217616256 HG In-Stock Unstable TBXA2R 47 42 CN1CC[C@@H](NC(=O)Oc2ccccc2)C1=O ZINC000217616261 BD For-Sale Unstable FAAH 31 41 O=C1O[C@]2(CCCN(S(=O)(=O)c3cc(F)ccc3F)C2)c2ccccc21 ZINC000217616295 GF For-Sale Unstable NPY5R 27 46 COc1ccc(Cl)cc1NC(=O)N/C=C/c1ccccc1 ZINC000217616311 DI For-Sale Unstable CMA1 22 42 COc1ccc(Cl)cc1NC(=O)N/C=C/c1ccccc1 ZINC000217616311 DI For-Sale Unstable COLA 41 39 COc1ccc(Cl)cc1NC(=O)N/C=C/c1ccccc1 ZINC000217616311 DI For-Sale Unstable CPT1A 46 32 COc1ccc(Cl)cc1NC(=O)N/C=C/c1ccccc1 ZINC000217616311 DI For-Sale Unstable PYGL 18 45 COc1ccc(Cl)cc1NC(=O)N/C=C/c1ccccc1 ZINC000217616311 DI For-Sale Unstable RBP4 25 47 COc1ccc(Cl)cc1NC(=O)N/C=C/c1ccccc1 ZINC000217616311 DI For-Sale Unstable CYSP_PLAFA 43 35 CC(C)[C@H](NC(=O)CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)c1nc2ccccc2n1C(C)C ZINC000217616326 JI In-Stock Unstable AGAL_COFAR 0 43 CC(C)[C@H](NC(=O)CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)c1nc2ccccc2n1C(C)C ZINC000217616326 JI In-Stock Unstable HLCS 0 41 CC(C)[C@H](NC(=O)CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)c1nc2ccccc2n1C(C)C ZINC000217616326 JI In-Stock Unstable BIRA 0 42 CN1CC[C@H](NC(=O)Oc2ccccc2)C1=O ZINC000217616338 BD For-Sale Unstable FAAH 31 41 Cc1onc(-c2ccccc2Cl)c1C(=O)Nc1nc(CN2CCC[C@@H](C)C2)cs1 ZINC000217616346 IK On-Demand Unstable GHSR 15 46 Cc1onc(-c2ccccc2Cl)c1C(=O)Nc1nc(CN2CCC[C@@H](C)C2)cs1 ZINC000217616346 IK On-Demand Unstable GPBAR1 26 40 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NC[C@@H]1CCCO1 ZINC000217616360 HE In-Stock Unstable TBXA2R 43 37 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NC[C@@H]1CCCO1 ZINC000217616360 HE In-Stock Unstable SFRP1 20 43 O=C1O[C@@]2(CCCN(S(=O)(=O)c3c(F)cccc3F)C2)c2ccccc21 ZINC000217616400 GF For-Sale Unstable NPY5R 26 44 O=C1O[C@@]2(CCCN(S(=O)(=O)c3c(F)cccc3F)C2)c2ccccc21 ZINC000217616400 GF For-Sale Unstable PKM 24 46 CCCCc1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217616413 CJ For-Sale Unstable SCN2A 26 54 CCCCc1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217616413 CJ For-Sale Unstable HDAC8 21 40 CCCCc1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217616413 CJ For-Sale Unstable MMP2 24 44 CCCCc1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217616413 CJ For-Sale Unstable MMP3 28 44 CCCCc1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217616413 CJ For-Sale Unstable HDAC2 15 40 CCCCc1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217616413 CJ For-Sale Unstable HDAC6 19 40 CCCCc1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217616413 CJ For-Sale Unstable FAAH 22 41 CCCCc1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217616413 CJ For-Sale Unstable CFTR 44 34 CCCCc1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217616413 CJ For-Sale Unstable SPHK1 18 42 CCCCc1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217616413 CJ For-Sale Unstable ACAT 0 52 CCCCc1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217616413 CJ For-Sale Unstable TRPM2 0 47 CCc1cccc(NC(=O)c2ccc(/C=C\C(=O)O)s2)c1 ZINC000217616423 DH For-Sale Unstable P2RY14 43 35 CCc1cccc(NC(=O)c2ccc(/C=C\C(=O)O)s2)c1 ZINC000217616423 DH For-Sale Unstable KCNK3 87 36 CCc1cccc(NC(=O)c2ccc(/C=C\C(=O)O)s2)c1 ZINC000217616423 DH For-Sale Unstable KCNK9 55 36 Cc1onc(-c2ccccc2Cl)c1C(=O)Nc1nc(CN2CCC[C@H](C)C2)cs1 ZINC000217616424 IK On-Demand Unstable GHSR 15 46 Cc1onc(-c2ccccc2Cl)c1C(=O)Nc1nc(CN2CCC[C@H](C)C2)cs1 ZINC000217616424 IK On-Demand Unstable GPBAR1 26 40 O[C@@H]1CN(Cc2ccsc2)CCN(c2ncnc3[nH]ccc23)C1 ZINC000217616428 ED In-Stock Unstable AKT2 43 40 O[C@@H]1CN(Cc2ccsc2)CCN(c2ncnc3[nH]ccc23)C1 ZINC000217616428 ED In-Stock Unstable JAK3 15 45 O[C@@H]1CN(Cc2ccsc2)CCN(c2ncnc3[nH]ccc23)C1 ZINC000217616428 ED In-Stock Unstable AKT1 21 41 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NC[C@H]1CCCO1 ZINC000217616447 HE In-Stock Unstable TBXA2R 43 37 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1NC[C@H]1CCCO1 ZINC000217616447 HE In-Stock Unstable SFRP1 20 43 O=C1O[C@]2(CCCN(S(=O)(=O)c3c(F)cccc3F)C2)c2ccccc21 ZINC000217616489 GF For-Sale Unstable NPY5R 26 44 O=C1O[C@]2(CCCN(S(=O)(=O)c3c(F)cccc3F)C2)c2ccccc21 ZINC000217616489 GF For-Sale Unstable PKM 24 46 O=S(=O)(c1ccc2c(c1)CCCC2)N1Cc2cnc(N3CCOCC3)nc2C1 ZINC000217616495 HD In-Stock Unstable AKR1C3 51 38 COc1ccc(CCN(C)C[C@@H]2[C@H]3CNC[C@H]32)cc1OC ZINC000217616515 CD In-Stock Unstable HCN2 0 43 O=C(N/C=C/c1ccccc1)Nc1ccc(Cl)cc1Cl ZINC000217616519 DJ For-Sale Anodyne CMA1 22 45 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1N1CCCC1 ZINC000217616546 FF In-Stock Unstable TBXA2R 53 43 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1N1CCCC1 ZINC000217616546 FF In-Stock Unstable BRPF1 0 41 O=C1O[C@@]2(CCCN(S(=O)(=O)c3ccc(Cl)s3)C2)c2ccccc21 ZINC000217616604 GG For-Sale Unstable NPY5R 25 40 O=C(N/C=C/c1ccccc1)NCCc1ccc(O)cc1 ZINC000217616621 CF For-Sale Unstable F3 24 42 O=C(N/C=C/c1ccccc1)NCCc1ccc(O)cc1 ZINC000217616621 CF For-Sale Unstable MMP2 20 60 O=C(N/C=C/c1ccccc1)NCCc1ccc(O)cc1 ZINC000217616621 CF For-Sale Unstable SLC6A5 49 49 O=C(N/C=C/c1ccccc1)NCCc1ccc(O)cc1 ZINC000217616621 CF For-Sale Unstable AMP1_PLAFQ 26 41 O=C(N/C=C/c1ccccc1)NCCc1ccc(O)cc1 ZINC000217616621 CF For-Sale Unstable AKR1B10 22 45 COC(=O)C[C@H](c1ccc(OC)c(O)c1)c1oc(CN2CCCCC2)cc(=O)c1O ZINC000217616648 HF In-Stock Unstable RORC 42 33 c1ccc([C@@H](N[C@@H]2CCN3CCCC[C@@H]23)C2CC2)cc1 ZINC000217616654 CG For-Sale Unstable SLC18A3 45 37 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1N1CCCCC1 ZINC000217616662 GF In-Stock Unstable TBXA2R 54 45 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1N1CCCCC1 ZINC000217616662 GF In-Stock Unstable HTR7 20 41 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1N1CCCCC1 ZINC000217616662 GF In-Stock Unstable KCNQ2 52 43 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1N1CCCCC1 ZINC000217616662 GF In-Stock Unstable AKR1C3 18 55 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1N1CCCCC1 ZINC000217616662 GF In-Stock Unstable SFRP1 77 47 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1N1CCCCC1 ZINC000217616662 GF In-Stock Unstable WNT3 63 34 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1N1CCCCC1 ZINC000217616662 GF In-Stock Unstable BRPF1 0 42 O=C1O[C@]2(CCCN(S(=O)(=O)c3ccc(Cl)s3)C2)c2ccccc21 ZINC000217616678 GG For-Sale Unstable NPY5R 25 40 c1ccc([C@H](N[C@@H]2CCN3CCCC[C@@H]23)C2CC2)cc1 ZINC000217616730 CG For-Sale Unstable SLC18A3 45 37 COC(=O)C[C@@H](c1ccc(OC)c(O)c1)c1oc(CN2CCCCC2)cc(=O)c1O ZINC000217616748 HF In-Stock Unstable RORC 42 33 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1N1CCOCC1 ZINC000217616772 GD In-Stock Unstable TBXA2R 51 41 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1N1CCOCC1 ZINC000217616772 GD In-Stock Unstable HTR7 17 40 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1N1CCOCC1 ZINC000217616772 GD In-Stock Unstable SLC6A9 15 43 O=C(O)c1cc(S(=O)(=O)NCCc2ccccc2)ccc1N1CCOCC1 ZINC000217616772 GD In-Stock Unstable SFRP1 49 43 CCOC(=O)c1c(NC(=O)[C@@H](C)NC(=O)c2cccs2)sc2c1CCCC2 ZINC000217616808 HH On-Demand Unstable PDE4D 0 61 CCOC(=O)c1c(NC(=O)[C@@H](C)NC(=O)c2cccs2)sc2c1CCCC2 ZINC000217616808 HH On-Demand Unstable NS5B 0 52 CCOC(=O)c1c(NC(=O)[C@@H](C)NC(=O)c2cccs2)sc2c1CCCC2 ZINC000217616808 HH On-Demand Unstable FLT3 22 48 c1ccc([C@@H](N[C@H]2CCN3CCCC[C@@H]23)C2CC2)cc1 ZINC000217616811 CG For-Sale Unstable SLC18A3 45 37 CC(C)N(Cc1ccccc1)C(=O)N/C=C/c1ccccc1 ZINC000217616836 CI For-Sale Unstable MME 41 36 CC(C)N(Cc1ccccc1)C(=O)N/C=C/c1ccccc1 ZINC000217616836 CI For-Sale Unstable MMP2 18 40 CC(C)N(Cc1ccccc1)C(=O)N/C=C/c1ccccc1 ZINC000217616836 CI For-Sale Unstable MMP3 17 41 CC(C)N(Cc1ccccc1)C(=O)N/C=C/c1ccccc1 ZINC000217616836 CI For-Sale Unstable MMP9 16 41 CC(C)N(Cc1ccccc1)C(=O)N/C=C/c1ccccc1 ZINC000217616836 CI For-Sale Unstable PTGES 23 41 CN1CCCC[C@@H]1CNC[C@@H](O)COc1ccccc1Cl ZINC000217616844 DE For-Sale Unstable ADRB2 46 49 CN1CCCC[C@@H]1CNC[C@@H](O)COc1ccccc1Cl ZINC000217616844 DE For-Sale Unstable ADRB1 65 45 CN1CCCC[C@@H]1CNC[C@@H](O)COc1ccccc1Cl ZINC000217616844 DE For-Sale Unstable ADRB3 39 46 CN1CCCC[C@@H]1CNC[C@@H](O)COc1ccccc1Cl ZINC000217616844 DE For-Sale Unstable CHRNA10 63 41 CN1CCCC[C@@H]1CNC[C@@H](O)COc1ccccc1Cl ZINC000217616844 DE For-Sale Unstable ACKR3 51 32 COc1ccc(CCOc2ccc([C@@H]3CC(=O)Oc4c3c(=O)oc3ccccc43)cc2)cc1 ZINC000217616847 IJ In-Stock Unstable MAOB 34 42 CCOCCCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217616877 HF In-Stock Unstable TBXA2R 45 39 CCOCCCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217616877 HF In-Stock Unstable BDKRB1 0 43 CCOCCCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217616877 HF In-Stock Unstable ALOX15 45 35 CCOC(=O)c1c(NC(=O)[C@H](C)NC(=O)c2cccs2)sc2c1CCCC2 ZINC000217616880 HH On-Demand Unstable PDE4D 0 61 CCOC(=O)c1c(NC(=O)[C@H](C)NC(=O)c2cccs2)sc2c1CCCC2 ZINC000217616880 HH On-Demand Unstable NS5B 0 52 CCOC(=O)c1c(NC(=O)[C@H](C)NC(=O)c2cccs2)sc2c1CCCC2 ZINC000217616880 HH On-Demand Unstable FLT3 22 48 c1ccc([C@H](N[C@H]2CCN3CCCC[C@@H]23)C2CC2)cc1 ZINC000217616885 CG For-Sale Unstable SLC18A3 45 37 CN1CCCC[C@H]1CNC[C@@H](O)COc1ccccc1Cl ZINC000217616908 DE For-Sale Unstable ADRB2 46 49 CN1CCCC[C@H]1CNC[C@@H](O)COc1ccccc1Cl ZINC000217616908 DE For-Sale Unstable ADRB1 65 45 CN1CCCC[C@H]1CNC[C@@H](O)COc1ccccc1Cl ZINC000217616908 DE For-Sale Unstable ADRB3 39 46 CN1CCCC[C@H]1CNC[C@@H](O)COc1ccccc1Cl ZINC000217616908 DE For-Sale Unstable CHRNA10 63 41 CN1CCCC[C@H]1CNC[C@@H](O)COc1ccccc1Cl ZINC000217616908 DE For-Sale Unstable ACKR3 51 32 COc1ccc(CCOc2ccc([C@H]3CC(=O)Oc4c3c(=O)oc3ccccc43)cc2)cc1 ZINC000217616914 IJ In-Stock Unstable MAOB 34 42 CCCCCCCCCCCCOC(=O)C(C)(C)N(Cl)Cl ZINC000217616967 EK For-Sale Unstable AMY2 56 33 O=C(O)C[C@@H]1COc2cc(F)c(F)cc21 ZINC000217616973 BD In-Stock Unstable FFAR1 66 52 CC(=O)c1cccc(S(=O)(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217616974 GF For-Sale Unstable AKR1C3 61 40 CC(C)OCCCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217616978 HG In-Stock Unstable TBXA2R 46 39 CC(C)OCCCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217616978 HG In-Stock Unstable BDKRB1 0 43 CC(C)OCCCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217616978 HG In-Stock Unstable ALOX15 43 33 COc1ccc2c(c1OC)C(=O)O[C@@H]2CC(=O)Nc1ccc(O)cc1 ZINC000217617018 EF In-Stock Unstable TSHR 41 31 CN1CCCC[C@@H]1CNC[C@@H](O)COc1ccc(Cl)cc1 ZINC000217617036 DE For-Sale Unstable ADRB2 51 46 CN1CCCC[C@@H]1CNC[C@@H](O)COc1ccc(Cl)cc1 ZINC000217617036 DE For-Sale Unstable ADRB1 68 46 CN1CCCC[C@@H]1CNC[C@@H](O)COc1ccc(Cl)cc1 ZINC000217617036 DE For-Sale Unstable GRIN1 25 42 CN1CCCC[C@@H]1CNC[C@@H](O)COc1ccc(Cl)cc1 ZINC000217617036 DE For-Sale Unstable ADRB3 51 41 CN1CCCC[C@@H]1CNC[C@@H](O)COc1ccc(Cl)cc1 ZINC000217617036 DE For-Sale Unstable EBP 18 41 CN1CCCC[C@@H]1CNC[C@@H](O)COc1ccc(Cl)cc1 ZINC000217617036 DE For-Sale Unstable CHRNA10 69 54 O=C(O)C[C@H]1COc2cc(F)c(F)cc21 ZINC000217617059 BD In-Stock Unstable FFAR1 66 52 CC(=O)c1cccc(S(=O)(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217617066 GF For-Sale Unstable AKR1C3 61 40 CCCCCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217617092 GH In-Stock Unstable TBXA2R 52 41 CCCCCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217617092 GH In-Stock Unstable CASP3 16 42 CCCCCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217617092 GH In-Stock Unstable ALOX15 66 43 COc1ccc2c(c1OC)C(=O)O[C@H]2CC(=O)Nc1ccc(O)cc1 ZINC000217617108 EF In-Stock Unstable TSHR 41 31 CN1CCCC[C@H]1CNC[C@@H](O)COc1ccc(Cl)cc1 ZINC000217617126 DE For-Sale Unstable ADRB2 51 46 CN1CCCC[C@H]1CNC[C@@H](O)COc1ccc(Cl)cc1 ZINC000217617126 DE For-Sale Unstable ADRB1 68 46 CN1CCCC[C@H]1CNC[C@@H](O)COc1ccc(Cl)cc1 ZINC000217617126 DE For-Sale Unstable GRIN1 25 42 CN1CCCC[C@H]1CNC[C@@H](O)COc1ccc(Cl)cc1 ZINC000217617126 DE For-Sale Unstable ADRB3 51 41 CN1CCCC[C@H]1CNC[C@@H](O)COc1ccc(Cl)cc1 ZINC000217617126 DE For-Sale Unstable EBP 18 41 CN1CCCC[C@H]1CNC[C@@H](O)COc1ccc(Cl)cc1 ZINC000217617126 DE For-Sale Unstable CHRNA10 69 54 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1ccc(SC)cc1 ZINC000217617190 JI In-Stock Unstable TGFBR2 56 45 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1ccc(SC)cc1 ZINC000217617190 JI In-Stock Unstable HISG 0 43 CC(C)CCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217617213 GG In-Stock Unstable TBXA2R 52 41 CC(C)CCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217617213 GG In-Stock Unstable CASP3 18 41 CC(C)CCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217617213 GG In-Stock Unstable ALOX15 40 35 CN1CCCC[C@@H]1CNC[C@@H](O)COc1cccc(Cl)c1 ZINC000217617243 DE For-Sale Unstable ADRB2 39 50 CN1CCCC[C@@H]1CNC[C@@H](O)COc1cccc(Cl)c1 ZINC000217617243 DE For-Sale Unstable ADRB1 58 43 CN1CCCC[C@@H]1CNC[C@@H](O)COc1cccc(Cl)c1 ZINC000217617243 DE For-Sale Unstable GRIN1 0 40 CN1CCCC[C@@H]1CNC[C@@H](O)COc1cccc(Cl)c1 ZINC000217617243 DE For-Sale Unstable ADRB3 47 40 CN1CCCC[C@@H]1CNC[C@@H](O)COc1cccc(Cl)c1 ZINC000217617243 DE For-Sale Unstable CHRNA10 73 57 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217617327 GH In-Stock Unstable TBXA2R 46 40 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217617327 GH In-Stock Unstable CASP3 17 41 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217617327 GH In-Stock Unstable ALOX15 46 36 CN1CCCC[C@H]1CNC[C@@H](O)COc1cccc(Cl)c1 ZINC000217617339 DE For-Sale Unstable ADRB2 39 50 CN1CCCC[C@H]1CNC[C@@H](O)COc1cccc(Cl)c1 ZINC000217617339 DE For-Sale Unstable ADRB1 58 43 CN1CCCC[C@H]1CNC[C@@H](O)COc1cccc(Cl)c1 ZINC000217617339 DE For-Sale Unstable GRIN1 0 40 CN1CCCC[C@H]1CNC[C@@H](O)COc1cccc(Cl)c1 ZINC000217617339 DE For-Sale Unstable ADRB3 47 40 CN1CCCC[C@H]1CNC[C@@H](O)COc1cccc(Cl)c1 ZINC000217617339 DE For-Sale Unstable CHRNA10 73 57 Cc1cc(C)c(S(=O)(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c(C)c1 ZINC000217617365 GG For-Sale Unstable NPY5R 27 41 O=C(Nc1ccccc1-c1nc2ccccc2[nH]1)c1nn(-c2ccccc2)c2c1CCC2 ZINC000217617376 HK On-Demand Unstable CNR1 50 31 O=C(Nc1ccccc1-c1nc2ccccc2[nH]1)c1nn(-c2ccccc2)c2c1CCC2 ZINC000217617376 HK On-Demand Unstable SIRT1 15 51 O=C(Nc1ccccc1-c1nc2ccccc2[nH]1)c1nn(-c2ccccc2)c2c1CCC2 ZINC000217617376 HK On-Demand Unstable STK33 58 45 CCCCOC(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217617403 CF On-Demand Unstable PRSS1 16 51 CCCCOC(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217617403 CF On-Demand Unstable SCN2A 18 44 CCCCOC(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217617403 CF On-Demand Unstable ACR 80 51 CCC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217617411 GH In-Stock Unstable TBXA2R 46 40 CCC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217617411 GH In-Stock Unstable CASP3 17 41 CCC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217617411 GH In-Stock Unstable ALOX15 46 36 CCCCCCCCCCCCCCCCCCOC(=O)C(C)(C)N(Cl)Cl ZINC000217617432 HK For-Sale Unstable AMY2 56 33 O=C(N/C=C/c1ccccc1)NC1CCCCC1 ZINC000217617448 BG For-Sale Unstable FAAH 17 57 O=C(N/C=C/c1ccccc1)NC1CCCCC1 ZINC000217617448 BG For-Sale Unstable EPHX2 37 56 Cc1cc(C)c(S(=O)(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c(C)c1 ZINC000217617456 GG For-Sale Unstable NPY5R 27 41 O=C1N(Cc2ccccc2)c2ccccc2[C@@]12Oc1ccccc1[C@H]1CC(c3ccc(Cl)cc3)=NN12 ZINC000217617517 JK In-Stock Unstable HTR2B 0 59 O=C1N(Cc2ccccc2)c2ccccc2[C@@]12Oc1ccccc1[C@H]1CC(c3ccc(Cl)cc3)=NN12 ZINC000217617517 JK In-Stock Unstable SCN9A 22 42 COC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217617525 GE In-Stock Unstable TBXA2R 46 39 Cc1cc(Cl)c(Br)cc1CCN ZINC000217617534 BF For-Sale Unstable TAAR1 17 45 O=C(Nc1ccc(I)cc1)C(F)F ZINC000217617544 CE On-Demand Anodyne Q25615_ONCVO 47 42 Cc1cc(C)c(S(=O)(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1C ZINC000217617563 GG For-Sale Unstable NPY5R 28 46 O=C1C[C@@H](C2=Cc3ccccc3OC2)c2c(c3ccccc3oc2=O)O1 ZINC000217617564 EH In-Stock Unstable VKORC1 0 42 CC1CCN(C(=O)N/C=C/c2ccccc2)CC1 ZINC000217617572 BG For-Sale Unstable EPHX2 17 40 COC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217617613 GE In-Stock Unstable TBXA2R 46 39 O=C1C[C@H](C2=Cc3ccccc3OC2)c2c(c3ccccc3oc2=O)O1 ZINC000217617643 EH In-Stock Unstable VKORC1 0 42 Cc1cc(C)c(S(=O)(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1C ZINC000217617650 GG For-Sale Unstable NPY5R 28 46 O=C(c1ccco1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217617670 DD In-Stock Unstable HSP90AB1 0 44 O=C(O)C1CCN(C(=O)N/C=C/c2ccccc2)CC1 ZINC000217617686 CE For-Sale Unstable EPHX2 15 42 CCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217617688 BG On-Demand Unstable INHA 34 41 CCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217617688 BG On-Demand Unstable SCN2A 27 65 CCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217617688 BG On-Demand Unstable S1PR4 39 53 CCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217617688 BG On-Demand Unstable S1PR3 32 53 CCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217617688 BG On-Demand Unstable MMP2 19 42 CCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217617688 BG On-Demand Unstable MMP3 32 42 CCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217617688 BG On-Demand Unstable CFTR 43 35 CCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217617688 BG On-Demand Unstable S1PR2 50 53 CCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217617688 BG On-Demand Unstable S1PR1 21 52 CCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217617688 BG On-Demand Unstable SPHK1 30 58 CCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217617688 BG On-Demand Unstable S1PR5 37 53 CCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217617688 BG On-Demand Unstable NAAA 23 41 CCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217617688 BG On-Demand Unstable ENPP2 29 41 CCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217617688 BG On-Demand Unstable P96878_MYCTU 17 53 CCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217617688 BG On-Demand Unstable ACAT 0 53 COc1cccc2c1O[C@@H](c1ccc(OCc3ccc(Cl)cc3)cc1)N1N=C(c3ccccc3)C[C@@H]21 ZINC000217617702 JK In-Stock Unstable EGFR 31 42 COc1cccc2c1O[C@@H](c1ccc(OCc3ccc(Cl)cc3)cc1)N1N=C(c3ccccc3)C[C@@H]21 ZINC000217617702 JK In-Stock Unstable MAOB 26 42 O=C(Cc1cc2c(cc1Cl)OCCO2)N1CCCC[C@@H]1c1ccccn1 ZINC000217617706 FH In-Stock Unstable OPRM1 0 43 O=C(Cc1cc2c(cc1Cl)OCCO2)N1CCCC[C@@H]1c1ccccn1 ZINC000217617706 FH In-Stock Unstable OPRK1 46 43 O=C(Cc1cc2c(cc1Cl)OCCO2)N1CCCC[C@@H]1c1ccccn1 ZINC000217617706 FH In-Stock Unstable EDNRB 21 45 O=C(Cc1cc2c(cc1Cl)OCCO2)N1CCCC[C@@H]1c1ccccn1 ZINC000217617706 FH In-Stock Unstable COLA 133 44 O=C(Cc1cc2c(cc1Cl)OCCO2)N1CCCC[C@@H]1c1ccccn1 ZINC000217617706 FH In-Stock Unstable CPT1A 114 44 O=C(Cc1cc2c(cc1Cl)OCCO2)N1CCCC[C@@H]1c1ccccn1 ZINC000217617706 FH In-Stock Unstable CPT2 41 33 CCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217617730 GF In-Stock Unstable CA2 21 41 CCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217617730 GF In-Stock Unstable TBXA2R 52 46 CCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217617730 GF In-Stock Unstable TBXAS1 17 42 CCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217617730 GF In-Stock Unstable BMP1 51 37 CCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217617730 GF In-Stock Unstable CA1 17 41 CCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217617730 GF In-Stock Unstable MMP13 43 38 CCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217617730 GF In-Stock Unstable ALOX15B 0 42 CCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217617730 GF In-Stock Unstable MMP2 25 40 CCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217617730 GF In-Stock Unstable ALOX15 57 42 CCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217617730 GF In-Stock Unstable PTGDR 25 41 CCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217617730 GF In-Stock Unstable IAP 0 44 CCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217617730 GF In-Stock Unstable CA9 23 44 CCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217617730 GF In-Stock Unstable MMP1 49 39 CCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217617730 GF In-Stock Unstable AKR1C3 31 49 CCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217617730 GF In-Stock Unstable AKR1C2 51 38 CCC[C@@H](N[C@@H]1CCC[C@@H](O)C1)c1ccc(Cl)cc1 ZINC000217617743 CI For-Sale Unstable SLC6A1 0 40 C=C(C)COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)cc1OC ZINC000217617762 KK In-Stock Unstable AKR1B1 0 45 C=C(C)COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)cc1OC ZINC000217617762 KK In-Stock Unstable CYP1B1 49 36 C=C(C)COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)cc1OC ZINC000217617762 KK In-Stock Unstable CYP1A1 37 43 O=C(Cc1cc2c(cc1Cl)OCCO2)N1CCCC[C@H]1c1ccccn1 ZINC000217617776 FH In-Stock Unstable OPRM1 0 43 O=C(Cc1cc2c(cc1Cl)OCCO2)N1CCCC[C@H]1c1ccccn1 ZINC000217617776 FH In-Stock Unstable OPRK1 46 43 O=C(Cc1cc2c(cc1Cl)OCCO2)N1CCCC[C@H]1c1ccccn1 ZINC000217617776 FH In-Stock Unstable EDNRB 21 45 O=C(Cc1cc2c(cc1Cl)OCCO2)N1CCCC[C@H]1c1ccccn1 ZINC000217617776 FH In-Stock Unstable COLA 133 44 O=C(Cc1cc2c(cc1Cl)OCCO2)N1CCCC[C@H]1c1ccccn1 ZINC000217617776 FH In-Stock Unstable CPT1A 114 44 O=C(Cc1cc2c(cc1Cl)OCCO2)N1CCCC[C@H]1c1ccccn1 ZINC000217617776 FH In-Stock Unstable CPT2 41 33 O=C(c1ccno1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217617785 DC In-Stock Unstable MAPK1 41 35 O=C(c1ccno1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217617785 DC In-Stock Unstable HSP90AB1 0 44 O=C(N/C=C/c1ccccc1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217617796 GJ For-Sale Unstable NMUR2 0 51 O=C(N/C=C/c1ccccc1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217617796 GJ For-Sale Unstable NMUR1 0 51 O=C(Nc1ccccc1N1CCOCC1)C(F)F ZINC000217617799 CD For-Sale Unstable KCNQ2 107 58 O=C(Nc1ccccc1N1CCOCC1)C(F)F ZINC000217617799 CD For-Sale Unstable KCNQ4 0 48 O=C(Nc1ccccc1N1CCOCC1)C(F)F ZINC000217617799 CD For-Sale Unstable CSF1R 0 52 O=C(Nc1ccccc1N1CCOCC1)C(F)F ZINC000217617799 CD For-Sale Unstable AKR1C3 29 46 O=C(Nc1ccccc1N1CCOCC1)C(F)F ZINC000217617799 CD For-Sale Unstable DGAT1 17 40 CCC[C@H](N[C@@H]1CCC[C@@H](O)C1)c1ccc(Cl)cc1 ZINC000217617815 CI On-Demand Unstable SLC6A1 0 40 C=C(C)COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)cc1OC ZINC000217617843 KK In-Stock Unstable AKR1B1 0 45 C=C(C)COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)cc1OC ZINC000217617843 KK In-Stock Unstable CYP1B1 49 36 C=C(C)COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)cc1OC ZINC000217617843 KK In-Stock Unstable CYP1A1 37 43 Cc1cccc(C(=O)N2CCC3(CCCC3)CC2)c1I ZINC000217617847 GI On-Demand Unstable CCR5 19 43 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)C)c(C(=O)O)c2)cc1 ZINC000217617855 GF In-Stock Unstable CA2 18 48 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)C)c(C(=O)O)c2)cc1 ZINC000217617855 GF In-Stock Unstable TBXA2R 47 46 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)C)c(C(=O)O)c2)cc1 ZINC000217617855 GF In-Stock Unstable TBXAS1 19 42 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)C)c(C(=O)O)c2)cc1 ZINC000217617855 GF In-Stock Unstable BMP1 88 38 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)C)c(C(=O)O)c2)cc1 ZINC000217617855 GF In-Stock Unstable CA1 19 48 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)C)c(C(=O)O)c2)cc1 ZINC000217617855 GF In-Stock Unstable MMP13 66 42 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)C)c(C(=O)O)c2)cc1 ZINC000217617855 GF In-Stock Unstable MMP2 44 42 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)C)c(C(=O)O)c2)cc1 ZINC000217617855 GF In-Stock Unstable MMP3 47 40 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)C)c(C(=O)O)c2)cc1 ZINC000217617855 GF In-Stock Unstable MMP8 34 42 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)C)c(C(=O)O)c2)cc1 ZINC000217617855 GF In-Stock Unstable MMP14 20 40 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)C)c(C(=O)O)c2)cc1 ZINC000217617855 GF In-Stock Unstable ALOX15 41 40 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)C)c(C(=O)O)c2)cc1 ZINC000217617855 GF In-Stock Unstable MMP9 53 42 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)C)c(C(=O)O)c2)cc1 ZINC000217617855 GF In-Stock Unstable MMP12 31 40 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)C)c(C(=O)O)c2)cc1 ZINC000217617855 GF In-Stock Unstable CA12 15 44 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)C)c(C(=O)O)c2)cc1 ZINC000217617855 GF In-Stock Unstable PTGDR 0 41 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)C)c(C(=O)O)c2)cc1 ZINC000217617855 GF In-Stock Unstable IAP 0 44 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)C)c(C(=O)O)c2)cc1 ZINC000217617855 GF In-Stock Unstable CA9 23 44 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)C)c(C(=O)O)c2)cc1 ZINC000217617855 GF In-Stock Unstable MMP1 53 37 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)C)c(C(=O)O)c2)cc1 ZINC000217617855 GF In-Stock Unstable AKR1C3 32 49 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)C)c(C(=O)O)c2)cc1 ZINC000217617855 GF In-Stock Unstable AKR1C2 51 38 O=C(c1ccncc1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217617901 EC In-Stock Unstable MTOR 41 43 O=C(c1ccncc1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217617901 EC In-Stock Unstable HSP90AB1 0 46 O=C(c1ccncc1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217617901 EC In-Stock Unstable PIK3CG 24 43 CCC[C@@H](N[C@H]1CCC[C@@H](O)C1)c1ccc(Cl)cc1 ZINC000217617911 CI For-Sale Unstable SLC6A1 0 40 CC(C)CNC(=O)N/C=C/c1ccccc1 ZINC000217617916 BF For-Sale Unstable ANPEP 48 38 CC(C)CNC(=O)N/C=C/c1ccccc1 ZINC000217617916 BF For-Sale Unstable F3 17 43 O=C(Nc1ccc(N2CCOCC2)cc1)C(F)F ZINC000217617919 CD On-Demand Unstable PIK3CA 40 46 O=C(Nc1ccc(N2CCOCC2)cc1)C(F)F ZINC000217617919 CD On-Demand Unstable JAK2 15 47 O=C(Nc1ccc(N2CCOCC2)cc1)C(F)F ZINC000217617919 CD On-Demand Unstable MAPKAPK5 44 35 O=C(Nc1ccc(N2CCOCC2)cc1)C(F)F ZINC000217617919 CD On-Demand Unstable PIK3CD 17 42 O=C(Nc1ccc(N2CCOCC2)cc1)C(F)F ZINC000217617919 CD On-Demand Unstable MTOR 69 46 O=C(Nc1ccc(N2CCOCC2)cc1)C(F)F ZINC000217617919 CD On-Demand Unstable EPHX2 23 51 O=C(Nc1ccc(N2CCOCC2)cc1)C(F)F ZINC000217617919 CD On-Demand Unstable PIK3CG 37 46 O=C(Nc1ccc(N2CCOCC2)cc1)C(F)F ZINC000217617919 CD On-Demand Unstable PIK3CB 26 42 O=C(Nc1ccc(N2CCOCC2)cc1)C(F)F ZINC000217617919 CD On-Demand Unstable AKR1C3 34 51 O=C(Nc1ccc(N2CCOCC2)cc1)C(F)F ZINC000217617919 CD On-Demand Unstable STAT6 61 38 O=C(Nc1ccc(N2CCOCC2)cc1)C(F)F ZINC000217617919 CD On-Demand Unstable DGAT1 28 46 CCCC1=C(C(=O)OCC)[C@H](c2ccc(OC)c(OC)c2)C2=C(C[C@H](c3cccs3)[C@@H](C(=O)OCC)C2=O)N1 ZINC000217617933 KK In-Stock Unstable TGFBR2 25 43 O=C(c1cc(Cl)ccc1Br)N1CCC2(CCCC2)CC1 ZINC000217617948 FJ On-Demand Unstable CCKBR 74 37 CCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217617955 HG In-Stock Unstable CA2 16 44 CCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217617955 HG In-Stock Unstable TBXA2R 46 44 CCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217617955 HG In-Stock Unstable TBXAS1 21 43 CCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217617955 HG In-Stock Unstable BMP1 51 36 CCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217617955 HG In-Stock Unstable CA1 17 44 CCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217617955 HG In-Stock Unstable MMP13 49 39 CCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217617955 HG In-Stock Unstable ALOX15B 0 45 CCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217617955 HG In-Stock Unstable ALOX15 62 45 CCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217617955 HG In-Stock Unstable MMP9 44 39 CCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217617955 HG In-Stock Unstable IAP 0 45 CCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217617955 HG In-Stock Unstable CA9 23 42 CCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217617955 HG In-Stock Unstable MMP1 40 38 CCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217617955 HG In-Stock Unstable AKR1C3 31 50 CCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217617955 HG In-Stock Unstable AKR1C2 52 37 CCC[C@H](N[C@H]1CCC[C@@H](O)C1)c1ccc(Cl)cc1 ZINC000217618000 CI On-Demand Unstable SLC6A1 0 40 O=C(c1ccccn1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217618023 EC In-Stock Unstable HSP90AB1 0 48 CCCCN(CCCC)C(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217618024 DH For-Sale Unstable TSPO 20 40 COCCNC(=O)N/C=C/c1ccccc1 ZINC000217618025 BD For-Sale Unstable TLR4 18 40 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1ccc(OC)c(OC)c1 ZINC000217618038 JH In-Stock Unstable CACNA1D 62 36 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1ccc(OC)c(OC)c1 ZINC000217618038 JH In-Stock Unstable TGFBR2 52 42 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1ccc(OC)c(OC)c1 ZINC000217618038 JH In-Stock Unstable HISG 0 43 Cn1ccc(C(=O)N2CCC3(CCCC3)CC2)cc1=O ZINC000217618060 CE On-Demand Unstable CCKBR 67 36 COc1ccc(CCNS(=O)(=O)c2ccc(NCC(C)C)c(C(=O)O)c2)cc1 ZINC000217618069 HF In-Stock Unstable CA2 15 46 COc1ccc(CCNS(=O)(=O)c2ccc(NCC(C)C)c(C(=O)O)c2)cc1 ZINC000217618069 HF In-Stock Unstable ADRB3 42 38 COc1ccc(CCNS(=O)(=O)c2ccc(NCC(C)C)c(C(=O)O)c2)cc1 ZINC000217618069 HF In-Stock Unstable TBXA2R 46 44 COc1ccc(CCNS(=O)(=O)c2ccc(NCC(C)C)c(C(=O)O)c2)cc1 ZINC000217618069 HF In-Stock Unstable TBXAS1 17 41 COc1ccc(CCNS(=O)(=O)c2ccc(NCC(C)C)c(C(=O)O)c2)cc1 ZINC000217618069 HF In-Stock Unstable BMP1 95 37 COc1ccc(CCNS(=O)(=O)c2ccc(NCC(C)C)c(C(=O)O)c2)cc1 ZINC000217618069 HF In-Stock Unstable CA1 15 46 COc1ccc(CCNS(=O)(=O)c2ccc(NCC(C)C)c(C(=O)O)c2)cc1 ZINC000217618069 HF In-Stock Unstable MMP13 61 41 COc1ccc(CCNS(=O)(=O)c2ccc(NCC(C)C)c(C(=O)O)c2)cc1 ZINC000217618069 HF In-Stock Unstable BDKRB1 0 43 COc1ccc(CCNS(=O)(=O)c2ccc(NCC(C)C)c(C(=O)O)c2)cc1 ZINC000217618069 HF In-Stock Unstable MMP3 44 41 COc1ccc(CCNS(=O)(=O)c2ccc(NCC(C)C)c(C(=O)O)c2)cc1 ZINC000217618069 HF In-Stock Unstable MMP8 28 41 COc1ccc(CCNS(=O)(=O)c2ccc(NCC(C)C)c(C(=O)O)c2)cc1 ZINC000217618069 HF In-Stock Unstable ALOX15 35 41 COc1ccc(CCNS(=O)(=O)c2ccc(NCC(C)C)c(C(=O)O)c2)cc1 ZINC000217618069 HF In-Stock Unstable MMP9 51 41 COc1ccc(CCNS(=O)(=O)c2ccc(NCC(C)C)c(C(=O)O)c2)cc1 ZINC000217618069 HF In-Stock Unstable MMP7 30 40 COc1ccc(CCNS(=O)(=O)c2ccc(NCC(C)C)c(C(=O)O)c2)cc1 ZINC000217618069 HF In-Stock Unstable IAP 0 43 COc1ccc(CCNS(=O)(=O)c2ccc(NCC(C)C)c(C(=O)O)c2)cc1 ZINC000217618069 HF In-Stock Unstable CA9 20 44 COc1ccc(CCNS(=O)(=O)c2ccc(NCC(C)C)c(C(=O)O)c2)cc1 ZINC000217618069 HF In-Stock Unstable MMP1 55 38 COc1ccc(CCNS(=O)(=O)c2ccc(NCC(C)C)c(C(=O)O)c2)cc1 ZINC000217618069 HF In-Stock Unstable AKR1C3 31 48 COc1ccc(CCNS(=O)(=O)c2ccc(NCC(C)C)c(C(=O)O)c2)cc1 ZINC000217618069 HF In-Stock Unstable AKR1C2 49 37 O=C(O)/C=C\c1ccc(C(=O)Nc2cc(Cl)ccc2F)s1 ZINC000217618107 EH For-Sale Anodyne KCNMA1 18 40 COc1ccc(C[C@@H](C)N[C@@H]2CCC[C@@H](O)C2)cc1OC ZINC000217618112 CF For-Sale Unstable PDE4A 42 39 CCCCNC(=O)N/C=C/c1ccccc1 ZINC000217618124 BF For-Sale Unstable EPHX2 26 40 CCCCNC(=O)N/C=C/c1ccccc1 ZINC000217618124 BF For-Sale Unstable HDAC9 20 41 CCCCNC(=O)N/C=C/c1ccccc1 ZINC000217618124 BF For-Sale Unstable AMP1_PLAFQ 27 41 CCCCNC(=O)N/C=C/c1ccccc1 ZINC000217618124 BF For-Sale Unstable ASAH1 41 37 CCCCNC(=O)N/C=C/c1ccccc1 ZINC000217618124 BF For-Sale Unstable ACAT 0 42 O=C(c1cnccn1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217618132 EC In-Stock Unstable HSP90AB1 0 43 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1ccc(F)cc1 ZINC000217618164 JH In-Stock Unstable TGFBR2 58 46 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1ccc(F)cc1 ZINC000217618164 JH In-Stock Unstable HISG 0 44 COc1ccc(S(=O)(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1C ZINC000217618177 GF For-Sale Unstable NPY5R 22 42 CC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618195 HG In-Stock Unstable TBXA2R 46 44 CC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618195 HG In-Stock Unstable TBXAS1 17 41 CC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618195 HG In-Stock Unstable BMP1 76 37 CC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618195 HG In-Stock Unstable CA1 15 46 CC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618195 HG In-Stock Unstable MMP13 55 41 CC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618195 HG In-Stock Unstable MMP2 36 41 CC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618195 HG In-Stock Unstable MMP3 41 39 CC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618195 HG In-Stock Unstable ALOX15 44 41 CC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618195 HG In-Stock Unstable MMP9 45 41 CC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618195 HG In-Stock Unstable IAP 0 43 CC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618195 HG In-Stock Unstable CA9 18 42 CC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618195 HG In-Stock Unstable MMP1 45 37 CC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618195 HG In-Stock Unstable AKR1C3 31 48 CC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618195 HG In-Stock Unstable AKR1C2 49 37 Cc1cc(C(=O)N2CCc3cnc(N4CCOCC4)nc3C2)no1 ZINC000217618230 EC In-Stock Unstable HSP90AB1 0 41 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@H](c3cccs3)C2)[C@@H]1c1ccc(F)cc1 ZINC000217618248 JH In-Stock Unstable TGFBR2 58 46 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@H](c3cccs3)C2)[C@@H]1c1ccc(F)cc1 ZINC000217618248 JH In-Stock Unstable HISG 0 44 CC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618259 HG In-Stock Unstable TBXA2R 46 44 CC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618259 HG In-Stock Unstable TBXAS1 17 41 CC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618259 HG In-Stock Unstable BMP1 76 37 CC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618259 HG In-Stock Unstable CA1 15 46 CC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618259 HG In-Stock Unstable MMP13 55 41 CC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618259 HG In-Stock Unstable MMP2 36 41 CC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618259 HG In-Stock Unstable MMP3 41 39 CC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618259 HG In-Stock Unstable ALOX15 44 41 CC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618259 HG In-Stock Unstable MMP9 45 41 CC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618259 HG In-Stock Unstable IAP 0 43 CC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618259 HG In-Stock Unstable CA9 18 42 CC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618259 HG In-Stock Unstable MMP1 45 37 CC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618259 HG In-Stock Unstable AKR1C3 31 48 CC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618259 HG In-Stock Unstable AKR1C2 49 37 COc1ccc(S(=O)(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1C ZINC000217618264 GF For-Sale Unstable NPY5R 22 42 COc1ccc(C[C@@H](C)N[C@H]2CCC[C@@H](O)C2)cc1OC ZINC000217618282 CF For-Sale Unstable PDE4A 42 39 COc1ccc(C(=O)N2CCC3(CCCC3)CC2)c(F)c1 ZINC000217618284 CH On-Demand Unstable EPHX2 18 42 CC[C@@H](C)[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(Cc2ccc3c(c2)OCO3)C1=O ZINC000217618294 GC In-Stock Unstable NOS2 50 35 CC[C@@H](C)[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(Cc2ccc3c(c2)OCO3)C1=O ZINC000217618294 GC In-Stock Unstable SSTR3 47 31 Cc1c(N(Cc2ccc(OC(F)(F)F)cc2)S(=O)(=O)c2ccc(C(=O)O)cc2)nc(C(F)(F)F)c2ccccc12 ZINC000217618343 KK Annotated Unstable BMP1 44 37 Cc1c(N(Cc2ccc(OC(F)(F)F)cc2)S(=O)(=O)c2ccc(C(=O)O)cc2)nc(C(F)(F)F)c2ccccc12 ZINC000217618343 KK Annotated Unstable MMP13 22 43 Cc1c(N(Cc2ccc(OC(F)(F)F)cc2)S(=O)(=O)c2ccc(C(=O)O)cc2)nc(C(F)(F)F)c2ccccc12 ZINC000217618343 KK Annotated Unstable ADAM17 25 43 Cc1c(N(Cc2ccc(OC(F)(F)F)cc2)S(=O)(=O)c2ccc(C(=O)O)cc2)nc(C(F)(F)F)c2ccccc12 ZINC000217618343 KK Annotated Unstable MMP9 29 43 Cc1c(N(Cc2ccc(OC(F)(F)F)cc2)S(=O)(=O)c2ccc(C(=O)O)cc2)nc(C(F)(F)F)c2ccccc12 ZINC000217618343 KK Annotated Unstable MMP1 18 43 Cc1c(N(Cc2ccc(OC(F)(F)F)cc2)S(=O)(=O)c2ccc(C(=O)O)cc2)nc(C(F)(F)F)c2ccccc12 ZINC000217618343 KK Annotated Unstable TRPM8 67 59 O=C(c1ccsc1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217618348 ED In-Stock Unstable HSP90AB1 15 43 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)(C)C)c(C(=O)O)c2)cc1 ZINC000217618362 HG In-Stock Unstable CA2 19 41 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)(C)C)c(C(=O)O)c2)cc1 ZINC000217618362 HG In-Stock Unstable TBXA2R 47 46 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)(C)C)c(C(=O)O)c2)cc1 ZINC000217618362 HG In-Stock Unstable TBXAS1 17 42 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)(C)C)c(C(=O)O)c2)cc1 ZINC000217618362 HG In-Stock Unstable BMP1 75 37 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)(C)C)c(C(=O)O)c2)cc1 ZINC000217618362 HG In-Stock Unstable CA1 21 45 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)(C)C)c(C(=O)O)c2)cc1 ZINC000217618362 HG In-Stock Unstable MMP13 54 42 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)(C)C)c(C(=O)O)c2)cc1 ZINC000217618362 HG In-Stock Unstable MMP2 33 40 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)(C)C)c(C(=O)O)c2)cc1 ZINC000217618362 HG In-Stock Unstable MMP3 41 40 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)(C)C)c(C(=O)O)c2)cc1 ZINC000217618362 HG In-Stock Unstable MMP8 25 40 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)(C)C)c(C(=O)O)c2)cc1 ZINC000217618362 HG In-Stock Unstable MMP14 17 40 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)(C)C)c(C(=O)O)c2)cc1 ZINC000217618362 HG In-Stock Unstable PRTN3 47 33 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)(C)C)c(C(=O)O)c2)cc1 ZINC000217618362 HG In-Stock Unstable ALOX15 40 39 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)(C)C)c(C(=O)O)c2)cc1 ZINC000217618362 HG In-Stock Unstable MMP9 46 42 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)(C)C)c(C(=O)O)c2)cc1 ZINC000217618362 HG In-Stock Unstable MMP12 27 40 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)(C)C)c(C(=O)O)c2)cc1 ZINC000217618362 HG In-Stock Unstable CA12 15 44 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)(C)C)c(C(=O)O)c2)cc1 ZINC000217618362 HG In-Stock Unstable PTGDR 24 41 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)(C)C)c(C(=O)O)c2)cc1 ZINC000217618362 HG In-Stock Unstable IAP 0 44 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)(C)C)c(C(=O)O)c2)cc1 ZINC000217618362 HG In-Stock Unstable CA9 23 44 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)(C)C)c(C(=O)O)c2)cc1 ZINC000217618362 HG In-Stock Unstable MMP1 49 42 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)(C)C)c(C(=O)O)c2)cc1 ZINC000217618362 HG In-Stock Unstable AKR1C3 34 52 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)(C)C)c(C(=O)O)c2)cc1 ZINC000217618362 HG In-Stock Unstable AKR1C2 52 38 COc1ccc(S(=O)(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c(C)c1 ZINC000217618366 GF For-Sale Unstable NPY5R 25 48 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccs2)CC(=O)O4)cc1O ZINC000217618418 II In-Stock Unstable AKR1B1 0 46 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccs2)CC(=O)O4)cc1O ZINC000217618418 II In-Stock Unstable CYP1B1 57 35 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccs2)CC(=O)O4)cc1O ZINC000217618418 II In-Stock Unstable CYP1A1 44 46 COc1ccc(S(=O)(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c(C)c1 ZINC000217618449 GF For-Sale Unstable NPY5R 25 48 C=CCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618468 GF In-Stock Unstable TBXA2R 45 44 C=CCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618468 GF In-Stock Unstable TBXAS1 17 42 C=CCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618468 GF In-Stock Unstable BMP1 46 37 C=CCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618468 GF In-Stock Unstable CA1 15 43 C=CCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618468 GF In-Stock Unstable MMP13 43 38 C=CCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618468 GF In-Stock Unstable IAP 0 44 C=CCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618468 GF In-Stock Unstable CA9 22 42 C=CCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618468 GF In-Stock Unstable AKR1C3 28 47 C=CCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618468 GF In-Stock Unstable FFAR4 15 40 C=CCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217618468 GF In-Stock Unstable AKR1C2 46 36 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccs2)CC(=O)O4)cc1O ZINC000217618492 II In-Stock Unstable AKR1B1 0 46 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccs2)CC(=O)O4)cc1O ZINC000217618492 II In-Stock Unstable CYP1B1 57 35 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccs2)CC(=O)O4)cc1O ZINC000217618492 II In-Stock Unstable CYP1A1 44 46 CC(C)S(=O)(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217618509 CD For-Sale Unstable PTGER2 0 42 CC(C)S(=O)(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217618509 CD For-Sale Unstable AKR1C3 35 47 COc1cc2c(cc1OC)CN(C/C=C\CN)CC2 ZINC000217618514 CD For-Sale Unstable SLC18A2 49 34 COc1cc2c(cc1OC)CN(C/C=C\CN)CC2 ZINC000217618514 CD For-Sale Unstable ADRA2C 17 41 COc1cc2c(cc1OC)CN(C/C=C\CN)CC2 ZINC000217618514 CD For-Sale Unstable ABCB1B 63 36 COc1cc2c(cc1OC)CN(C/C=C\CN)CC2 ZINC000217618514 CD For-Sale Unstable ABCB1 26 49 O=C(N/C=C/c1ccccc1)N1CCCc2ccccc21 ZINC000217618526 CH For-Sale Unstable AVPR2 43 48 O=C(c1cc(=O)n(-c2ccccc2)[nH]1)N1CCN(c2cnccn2)CC1 ZINC000217618546 FC In-Stock Unstable SLC6A7 0 56 COc1ccc(F)cc1S(=O)(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217618557 GF For-Sale Unstable NPY5R 26 44 Cc1ccccc1C(=O)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217618559 ED In-Stock Unstable HSP90AB1 17 48 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CC3)c(C(=O)O)c2)cc1 ZINC000217618582 GE In-Stock Unstable TBXA2R 47 46 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CC3)c(C(=O)O)c2)cc1 ZINC000217618582 GE In-Stock Unstable TBXAS1 15 41 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CC3)c(C(=O)O)c2)cc1 ZINC000217618582 GE In-Stock Unstable BMP1 73 36 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CC3)c(C(=O)O)c2)cc1 ZINC000217618582 GE In-Stock Unstable MMP13 67 41 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CC3)c(C(=O)O)c2)cc1 ZINC000217618582 GE In-Stock Unstable MMP2 41 41 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CC3)c(C(=O)O)c2)cc1 ZINC000217618582 GE In-Stock Unstable MMP3 59 41 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CC3)c(C(=O)O)c2)cc1 ZINC000217618582 GE In-Stock Unstable ALOX15 58 39 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CC3)c(C(=O)O)c2)cc1 ZINC000217618582 GE In-Stock Unstable MMP9 54 41 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CC3)c(C(=O)O)c2)cc1 ZINC000217618582 GE In-Stock Unstable MMP7 48 41 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CC3)c(C(=O)O)c2)cc1 ZINC000217618582 GE In-Stock Unstable CA9 18 42 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CC3)c(C(=O)O)c2)cc1 ZINC000217618582 GE In-Stock Unstable MMP1 60 40 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CC3)c(C(=O)O)c2)cc1 ZINC000217618582 GE In-Stock Unstable AKR1C3 30 48 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CC3)c(C(=O)O)c2)cc1 ZINC000217618582 GE In-Stock Unstable AKR1C2 49 37 O=C(N/C=C/c1ccccc1)NCCc1ccccc1 ZINC000217618628 CG For-Sale Unstable SDH1 0 42 O=C(N/C=C/c1ccccc1)NCCc1ccccc1 ZINC000217618628 CG For-Sale Unstable CPA1 32 40 O=C(N/C=C/c1ccccc1)NCCc1ccccc1 ZINC000217618628 CG For-Sale Unstable HDAC8 22 51 O=C(N/C=C/c1ccccc1)NCCc1ccccc1 ZINC000217618628 CG For-Sale Unstable CA5B 15 41 O=C(N/C=C/c1ccccc1)NCCc1ccccc1 ZINC000217618628 CG For-Sale Unstable MMP2 20 65 O=C(N/C=C/c1ccccc1)NCCc1ccccc1 ZINC000217618628 CG For-Sale Unstable HDAC1 18 47 O=C(N/C=C/c1ccccc1)NCCc1ccccc1 ZINC000217618628 CG For-Sale Unstable HDAC6 19 51 O=C(N/C=C/c1ccccc1)NCCc1ccccc1 ZINC000217618628 CG For-Sale Unstable FAAH 16 40 O=C(N/C=C/c1ccccc1)NCCc1ccccc1 ZINC000217618628 CG For-Sale Unstable AMP1_PLAFQ 44 47 O=C(N/C=C/c1ccccc1)NCCc1ccccc1 ZINC000217618628 CG For-Sale Unstable 17HSDCL 0 40 O=C(N/C=C/c1ccccc1)NCCc1ccccc1 ZINC000217618628 CG For-Sale Unstable HDA106 0 41 COc1ccc(F)cc1S(=O)(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217618632 GF For-Sale Unstable NPY5R 26 44 CC(C)c1ccc(NC(=O)C(F)F)cc1 ZINC000217618654 BG On-Demand Unstable P96878_MYCTU 15 50 CC(C)c1ccc(NC(=O)C(F)F)cc1 ZINC000217618654 BG On-Demand Unstable PSBA 0 58 CN1CCCC[C@@H]1CNC[C@@H](O)c1ccc(F)cc1 ZINC000217618657 CD For-Sale Unstable CHRNA10 55 37 CC(=O)c1sc(NC(=O)c2ccc(N3CCNC3=O)cc2)nc1-c1ccccc1 ZINC000217618658 HH On-Demand Unstable PRNP 63 37 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCC3)c(C(=O)O)c2)cc1 ZINC000217618710 HG In-Stock Unstable TBXA2R 45 43 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCC3)c(C(=O)O)c2)cc1 ZINC000217618710 HG In-Stock Unstable BMP1 63 38 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCC3)c(C(=O)O)c2)cc1 ZINC000217618710 HG In-Stock Unstable MMP13 67 42 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCC3)c(C(=O)O)c2)cc1 ZINC000217618710 HG In-Stock Unstable CTSK 15 44 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCC3)c(C(=O)O)c2)cc1 ZINC000217618710 HG In-Stock Unstable MMP2 41 42 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCC3)c(C(=O)O)c2)cc1 ZINC000217618710 HG In-Stock Unstable MMP3 56 40 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCC3)c(C(=O)O)c2)cc1 ZINC000217618710 HG In-Stock Unstable MMP8 33 40 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCC3)c(C(=O)O)c2)cc1 ZINC000217618710 HG In-Stock Unstable ALOX15 50 38 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCC3)c(C(=O)O)c2)cc1 ZINC000217618710 HG In-Stock Unstable MMP9 52 40 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCC3)c(C(=O)O)c2)cc1 ZINC000217618710 HG In-Stock Unstable MMP12 22 40 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCC3)c(C(=O)O)c2)cc1 ZINC000217618710 HG In-Stock Unstable MMP7 46 40 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCC3)c(C(=O)O)c2)cc1 ZINC000217618710 HG In-Stock Unstable IAP 0 45 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCC3)c(C(=O)O)c2)cc1 ZINC000217618710 HG In-Stock Unstable CA9 17 41 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCC3)c(C(=O)O)c2)cc1 ZINC000217618710 HG In-Stock Unstable MMP1 63 39 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCC3)c(C(=O)O)c2)cc1 ZINC000217618710 HG In-Stock Unstable AKR1C3 28 46 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCC3)c(C(=O)O)c2)cc1 ZINC000217618710 HG In-Stock Unstable TYRO3 19 41 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCC3)c(C(=O)O)c2)cc1 ZINC000217618710 HG In-Stock Unstable AKR1C2 45 35 O=C(N/C=C/c1ccccc1)NC1CCCC1 ZINC000217618727 BF For-Sale Unstable EPHX2 30 54 Cc1ccc(S(=O)(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1Cl ZINC000217618736 GG For-Sale Unstable NPY5R 25 40 CN1CCCC[C@H]1CNC[C@@H](O)c1ccc(F)cc1 ZINC000217618756 CD For-Sale Unstable CHRNA10 55 37 Cc1cc(C(=O)N2CCc3cnc(N4CCOCC4)nc3C2)c(C)o1 ZINC000217618764 ED In-Stock Unstable HSP90AB1 16 45 O=C(CN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCCCCCc1nc2ccccc2[nH]1 ZINC000217618772 JI In-Stock Unstable CYSP_TRYCR 0 41 COC(=O)c1ccc(CNC(=O)C(F)F)cc1 ZINC000217618787 BD On-Demand Unstable ANPEP 23 40 Cc1ccc(S(=O)(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1Cl ZINC000217618820 GG For-Sale Unstable NPY5R 25 40 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCCC3)c(C(=O)O)c2)cc1 ZINC000217618821 IH In-Stock Unstable ADRB1 27 40 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCCC3)c(C(=O)O)c2)cc1 ZINC000217618821 IH In-Stock Unstable ADRB3 34 40 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCCC3)c(C(=O)O)c2)cc1 ZINC000217618821 IH In-Stock Unstable TBXA2R 46 42 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCCC3)c(C(=O)O)c2)cc1 ZINC000217618821 IH In-Stock Unstable BMP1 57 39 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCCC3)c(C(=O)O)c2)cc1 ZINC000217618821 IH In-Stock Unstable MMP13 64 44 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCCC3)c(C(=O)O)c2)cc1 ZINC000217618821 IH In-Stock Unstable CTSK 15 46 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCCC3)c(C(=O)O)c2)cc1 ZINC000217618821 IH In-Stock Unstable MMP2 40 44 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCCC3)c(C(=O)O)c2)cc1 ZINC000217618821 IH In-Stock Unstable MMP3 56 42 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCCC3)c(C(=O)O)c2)cc1 ZINC000217618821 IH In-Stock Unstable ALOX15 48 38 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCCC3)c(C(=O)O)c2)cc1 ZINC000217618821 IH In-Stock Unstable MMP9 49 39 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCCC3)c(C(=O)O)c2)cc1 ZINC000217618821 IH In-Stock Unstable MMP7 46 40 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCCC3)c(C(=O)O)c2)cc1 ZINC000217618821 IH In-Stock Unstable IAP 0 45 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCCC3)c(C(=O)O)c2)cc1 ZINC000217618821 IH In-Stock Unstable CA9 17 40 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCCC3)c(C(=O)O)c2)cc1 ZINC000217618821 IH In-Stock Unstable MMP1 59 38 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCCC3)c(C(=O)O)c2)cc1 ZINC000217618821 IH In-Stock Unstable AKR1C3 26 45 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCCC3)c(C(=O)O)c2)cc1 ZINC000217618821 IH In-Stock Unstable TYRO3 17 41 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCCC3)c(C(=O)O)c2)cc1 ZINC000217618821 IH In-Stock Unstable AKR1C2 44 35 O=C(N/C=C/c1ccccc1)NCc1ccccc1Cl ZINC000217618843 CH For-Sale Unstable ANPEP 17 51 O=C(N/C=C/c1ccccc1)NCc1ccccc1Cl ZINC000217618843 CH For-Sale Unstable P2RX7 36 43 O=C(N/C=C/c1ccccc1)NCc1ccccc1Cl ZINC000217618843 CH For-Sale Unstable AMP1_PLAFQ 40 35 O=C(CN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCCCCCc1nc2ccccc2[nH]1 ZINC000217618860 JI In-Stock Unstable CYSP_TRYCR 0 41 Cc1csc(C(=O)N2CCc3cnc(N4CCOCC4)nc3C2)c1 ZINC000217618872 ED In-Stock Unstable MAPK1 40 35 Cc1csc(C(=O)N2CCc3cnc(N4CCOCC4)nc3C2)c1 ZINC000217618872 ED In-Stock Unstable HSP90AB1 15 42 CN1CCCC[C@@H]1CNC[C@@H](O)c1cccc(Br)c1 ZINC000217618888 EF For-Sale Unstable SLC18A3 0 41 CN1CCCC[C@@H]1CNC[C@@H](O)c1cccc(Br)c1 ZINC000217618888 EF For-Sale Unstable CHRNA10 56 34 CN1CCCC[C@@H]1CNC[C@@H](O)c1cccc(Br)c1 ZINC000217618888 EF For-Sale Unstable PHES 0 45 COc1ccc(CCNS(=O)(=O)c2ccc(NCCC3=CCCCC3)c(C(=O)O)c2)cc1 ZINC000217618901 JI In-Stock Unstable TBXA2R 44 42 COc1ccc(CCNS(=O)(=O)c2ccc(NCCC3=CCCCC3)c(C(=O)O)c2)cc1 ZINC000217618901 JI In-Stock Unstable TBXAS1 15 41 COc1ccc(CCNS(=O)(=O)c2ccc(NCCC3=CCCCC3)c(C(=O)O)c2)cc1 ZINC000217618901 JI In-Stock Unstable IAP 0 41 COc1ccc(CCNS(=O)(=O)c2ccc(NCCC3=CCCCC3)c(C(=O)O)c2)cc1 ZINC000217618901 JI In-Stock Unstable AKR1C3 19 45 CCN(CC)S(=O)(=O)Nc1ccc(/C=C\C(=O)O)cc1C ZINC000217618917 DE For-Sale Unstable AKR1C3 30 42 Cc1ccc(Cl)cc1S(=O)(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217618933 GG For-Sale Unstable NPY5R 27 45 COc1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1OC ZINC000217618965 EG For-Sale Unstable TRPV1 0 40 COc1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1OC ZINC000217618965 EG For-Sale Unstable MTNR1A 36 43 COc1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1OC ZINC000217618965 EG For-Sale Unstable MTNR1B 41 39 COc1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1OC ZINC000217618965 EG For-Sale Unstable ABCG2 22 46 COc1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1OC ZINC000217618965 EG For-Sale Unstable CAN2 0 48 COc1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1OC ZINC000217618965 EG For-Sale Unstable ACKR3 40 36 CN1CCCC[C@H]1CNC[C@@H](O)c1cccc(Br)c1 ZINC000217618969 EF For-Sale Unstable SLC18A3 0 41 CN1CCCC[C@H]1CNC[C@@H](O)c1cccc(Br)c1 ZINC000217618969 EF For-Sale Unstable CHRNA10 56 34 CN1CCCC[C@H]1CNC[C@@H](O)c1cccc(Br)c1 ZINC000217618969 EF For-Sale Unstable PHES 0 45 N#Cc1cccc(C(=O)N2CCc3cnc(N4CCOCC4)nc3C2)c1 ZINC000217618971 ED In-Stock Unstable HSP90AB1 15 42 NC/C=C\CN1CCN(c2ccccc2F)CC1 ZINC000217618973 BD For-Sale Unstable DRD3 24 46 COc1ccc(CCNS(=O)(=O)c2ccc(NCCO)c(C(=O)O)c2)cc1 ZINC000217618997 GD In-Stock Unstable CA2 19 43 COc1ccc(CCNS(=O)(=O)c2ccc(NCCO)c(C(=O)O)c2)cc1 ZINC000217618997 GD In-Stock Unstable TBXA2R 52 46 COc1ccc(CCNS(=O)(=O)c2ccc(NCCO)c(C(=O)O)c2)cc1 ZINC000217618997 GD In-Stock Unstable TBXAS1 16 42 COc1ccc(CCNS(=O)(=O)c2ccc(NCCO)c(C(=O)O)c2)cc1 ZINC000217618997 GD In-Stock Unstable BMP1 51 37 COc1ccc(CCNS(=O)(=O)c2ccc(NCCO)c(C(=O)O)c2)cc1 ZINC000217618997 GD In-Stock Unstable CA1 17 45 COc1ccc(CCNS(=O)(=O)c2ccc(NCCO)c(C(=O)O)c2)cc1 ZINC000217618997 GD In-Stock Unstable MMP13 44 38 COc1ccc(CCNS(=O)(=O)c2ccc(NCCO)c(C(=O)O)c2)cc1 ZINC000217618997 GD In-Stock Unstable MMP2 25 43 COc1ccc(CCNS(=O)(=O)c2ccc(NCCO)c(C(=O)O)c2)cc1 ZINC000217618997 GD In-Stock Unstable MMP14 15 43 COc1ccc(CCNS(=O)(=O)c2ccc(NCCO)c(C(=O)O)c2)cc1 ZINC000217618997 GD In-Stock Unstable PTGDR 24 41 COc1ccc(CCNS(=O)(=O)c2ccc(NCCO)c(C(=O)O)c2)cc1 ZINC000217618997 GD In-Stock Unstable IAP 0 44 COc1ccc(CCNS(=O)(=O)c2ccc(NCCO)c(C(=O)O)c2)cc1 ZINC000217618997 GD In-Stock Unstable CA9 23 44 COc1ccc(CCNS(=O)(=O)c2ccc(NCCO)c(C(=O)O)c2)cc1 ZINC000217618997 GD In-Stock Unstable MMP1 51 37 COc1ccc(CCNS(=O)(=O)c2ccc(NCCO)c(C(=O)O)c2)cc1 ZINC000217618997 GD In-Stock Unstable AKR1C3 31 49 COc1ccc(CCNS(=O)(=O)c2ccc(NCCO)c(C(=O)O)c2)cc1 ZINC000217618997 GD In-Stock Unstable AKR1C2 51 38 CC(=O)N1c2ccc(S(=O)(=O)Nc3cc([N+](=O)[O-])c(C)cc3C)cc2C[C@@H]1C ZINC000217619011 HG On-Demand Unstable NOD2 18 41 Cc1ccc(Cl)cc1S(=O)(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217619014 GG For-Sale Unstable NPY5R 27 45 CC(=O)N1c2ccc(S(=O)(=O)Nc3cc([N+](=O)[O-])c(C)cc3C)cc2C[C@H]1C ZINC000217619092 HG On-Demand Unstable NOD2 18 41 CN1CCCC[C@@H]1CNC[C@@H](O)c1ccccc1F ZINC000217619098 CD For-Sale Unstable CHRNA10 58 43 COc1ccc(CCNS(=O)(=O)c2ccc(NCCCO)c(C(=O)O)c2)cc1 ZINC000217619118 HD In-Stock Unstable CA2 16 41 COc1ccc(CCNS(=O)(=O)c2ccc(NCCCO)c(C(=O)O)c2)cc1 ZINC000217619118 HD In-Stock Unstable TBXA2R 46 44 COc1ccc(CCNS(=O)(=O)c2ccc(NCCCO)c(C(=O)O)c2)cc1 ZINC000217619118 HD In-Stock Unstable TBXAS1 21 43 COc1ccc(CCNS(=O)(=O)c2ccc(NCCCO)c(C(=O)O)c2)cc1 ZINC000217619118 HD In-Stock Unstable BMP1 50 36 COc1ccc(CCNS(=O)(=O)c2ccc(NCCCO)c(C(=O)O)c2)cc1 ZINC000217619118 HD In-Stock Unstable CA1 16 44 COc1ccc(CCNS(=O)(=O)c2ccc(NCCCO)c(C(=O)O)c2)cc1 ZINC000217619118 HD In-Stock Unstable MMP13 48 41 COc1ccc(CCNS(=O)(=O)c2ccc(NCCCO)c(C(=O)O)c2)cc1 ZINC000217619118 HD In-Stock Unstable MMP2 27 41 COc1ccc(CCNS(=O)(=O)c2ccc(NCCCO)c(C(=O)O)c2)cc1 ZINC000217619118 HD In-Stock Unstable MMP8 20 41 COc1ccc(CCNS(=O)(=O)c2ccc(NCCCO)c(C(=O)O)c2)cc1 ZINC000217619118 HD In-Stock Unstable ALOX15 46 40 COc1ccc(CCNS(=O)(=O)c2ccc(NCCCO)c(C(=O)O)c2)cc1 ZINC000217619118 HD In-Stock Unstable MMP9 43 41 COc1ccc(CCNS(=O)(=O)c2ccc(NCCCO)c(C(=O)O)c2)cc1 ZINC000217619118 HD In-Stock Unstable MMP12 24 41 COc1ccc(CCNS(=O)(=O)c2ccc(NCCCO)c(C(=O)O)c2)cc1 ZINC000217619118 HD In-Stock Unstable IAP 0 45 COc1ccc(CCNS(=O)(=O)c2ccc(NCCCO)c(C(=O)O)c2)cc1 ZINC000217619118 HD In-Stock Unstable CA9 20 42 COc1ccc(CCNS(=O)(=O)c2ccc(NCCCO)c(C(=O)O)c2)cc1 ZINC000217619118 HD In-Stock Unstable MMP1 43 36 COc1ccc(CCNS(=O)(=O)c2ccc(NCCCO)c(C(=O)O)c2)cc1 ZINC000217619118 HD In-Stock Unstable AKR1C3 31 50 COc1ccc(CCNS(=O)(=O)c2ccc(NCCCO)c(C(=O)O)c2)cc1 ZINC000217619118 HD In-Stock Unstable AKR1C2 52 37 O=C1O[C@@]2(CCCN(S(=O)(=O)Cc3ccccc3Cl)C2)c2ccccc21 ZINC000217619139 GG In-Stock Unstable NPY5R 26 44 O=C(O)/C=C\c1cccc(CN2CCCCC2=O)c1 ZINC000217619168 CE For-Sale Unstable PTGER2 16 52 CN1CCCC[C@H]1CNC[C@@H](O)c1ccccc1F ZINC000217619196 CD For-Sale Unstable CHRNA10 58 43 COCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217619234 HD In-Stock Unstable CA2 20 40 COCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217619234 HD In-Stock Unstable TBXA2R 52 45 COCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217619234 HD In-Stock Unstable TBXAS1 17 42 COCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217619234 HD In-Stock Unstable BMP1 53 36 COCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217619234 HD In-Stock Unstable CA1 20 45 COCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217619234 HD In-Stock Unstable MMP13 51 40 COCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217619234 HD In-Stock Unstable MMP2 31 40 COCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217619234 HD In-Stock Unstable MMP8 25 40 COCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217619234 HD In-Stock Unstable MMP14 16 40 COCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217619234 HD In-Stock Unstable MMP9 46 40 COCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217619234 HD In-Stock Unstable MMP12 24 40 COCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217619234 HD In-Stock Unstable PTGDR 16 40 COCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217619234 HD In-Stock Unstable IAP 0 43 COCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217619234 HD In-Stock Unstable CA9 25 45 COCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217619234 HD In-Stock Unstable MMP1 47 37 COCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217619234 HD In-Stock Unstable AKR1C3 30 48 COCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217619234 HD In-Stock Unstable AKR1C2 50 37 O=C1O[C@]2(CCCN(S(=O)(=O)Cc3ccccc3Cl)C2)c2ccccc21 ZINC000217619242 GG In-Stock Unstable NPY5R 26 44 CN1CCCC[C@@H]1CNC[C@@H](O)c1ccc(Cl)cc1 ZINC000217619307 CE For-Sale Unstable HRH1 18 40 CN1CCCC[C@@H]1CNC[C@@H](O)c1ccc(Cl)cc1 ZINC000217619307 CE For-Sale Unstable SLC6A3 18 40 CN1CCCC[C@@H]1CNC[C@@H](O)c1ccc(Cl)cc1 ZINC000217619307 CE For-Sale Unstable CHRNA10 48 44 O=C(N/C=C/c1ccccc1)NCc1cccnc1 ZINC000217619309 CF For-Sale Unstable TBXAS1 55 48 O=C(N/C=C/c1ccccc1)NCc1cccnc1 ZINC000217619309 CF For-Sale Unstable PTAFR 35 44 O=C(N/C=C/c1ccccc1)NCc1cccnc1 ZINC000217619309 CF For-Sale Unstable KCNA5 15 40 O=C(N/C=C/c1ccccc1)NCc1cccnc1 ZINC000217619309 CF For-Sale Unstable CHRNA7 22 42 O=C(N/C=C/c1ccccc1)NCc1cccnc1 ZINC000217619309 CF For-Sale Unstable NAMPT 92 56 O=C1O[C@@]2(CCCN(S(=O)(=O)Cc3cccc(Cl)c3)C2)c2ccccc21 ZINC000217619361 GG For-Sale Unstable NPY5R 23 42 COCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217619362 HE In-Stock Unstable CA2 16 44 COCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217619362 HE In-Stock Unstable TBXA2R 45 44 COCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217619362 HE In-Stock Unstable TBXAS1 17 42 COCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217619362 HE In-Stock Unstable BMP1 55 35 COCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217619362 HE In-Stock Unstable CA1 17 44 COCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217619362 HE In-Stock Unstable MMP13 46 38 COCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217619362 HE In-Stock Unstable ALOX15 40 39 COCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217619362 HE In-Stock Unstable IAP 0 44 COCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217619362 HE In-Stock Unstable CA9 20 44 COCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217619362 HE In-Stock Unstable MMP1 40 36 COCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217619362 HE In-Stock Unstable AKR1C3 29 49 COCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217619362 HE In-Stock Unstable AKR1C2 51 37 CN1CCCC[C@H]1CNC[C@@H](O)c1ccc(Cl)cc1 ZINC000217619393 CE For-Sale Unstable HRH1 18 40 CN1CCCC[C@H]1CNC[C@@H](O)c1ccc(Cl)cc1 ZINC000217619393 CE For-Sale Unstable SLC6A3 18 40 CN1CCCC[C@H]1CNC[C@@H](O)c1ccc(Cl)cc1 ZINC000217619393 CE For-Sale Unstable CHRNA10 48 44 CC[C@@H](N[C@@H]1CCC[C@@H](O)C1)c1ccc(OC)c(OC)c1 ZINC000217619419 CG For-Sale Unstable PDE4A 39 41 CC[C@@H](N[C@@H]1CCC[C@@H](O)C1)c1ccc(OC)c(OC)c1 ZINC000217619419 CG For-Sale Unstable PDE4B 21 40 C[C@@H](O)c1cc(Br)ccc1N1CC[C@@H](c2ccccc2)C1 ZINC000217619436 EI For-Sale Unstable VACHT_TETCF 0 44 C[C@@H](O)c1cc(Br)ccc1N1CC[C@@H](c2ccccc2)C1 ZINC000217619436 EI For-Sale Unstable SLC18A3 31 45 O=C1O[C@]2(CCCN(S(=O)(=O)Cc3cccc(Cl)c3)C2)c2ccccc21 ZINC000217619442 GG For-Sale Unstable NPY5R 23 42 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619486 IH In-Stock Unstable CA2 26 44 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619486 IH In-Stock Unstable GNRHR 16 49 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619486 IH In-Stock Unstable TBXA2R 53 44 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619486 IH In-Stock Unstable TBXAS1 28 43 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619486 IH In-Stock Unstable BMP1 72 41 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619486 IH In-Stock Unstable CA1 27 44 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619486 IH In-Stock Unstable MMP13 71 45 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619486 IH In-Stock Unstable BDKRB1 0 41 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619486 IH In-Stock Unstable ADAM17 51 43 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619486 IH In-Stock Unstable ALOX15B 0 41 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619486 IH In-Stock Unstable CA14 20 44 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619486 IH In-Stock Unstable MMP2 40 41 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619486 IH In-Stock Unstable MMP3 49 41 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619486 IH In-Stock Unstable PRTN3 46 32 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619486 IH In-Stock Unstable ALOX15 69 41 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619486 IH In-Stock Unstable MMP9 60 45 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619486 IH In-Stock Unstable CA12 18 44 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619486 IH In-Stock Unstable PTGDR 22 41 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619486 IH In-Stock Unstable MMP7 33 41 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619486 IH In-Stock Unstable IAP 0 43 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619486 IH In-Stock Unstable CA9 32 42 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619486 IH In-Stock Unstable MMP1 58 42 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619486 IH In-Stock Unstable AKR1C3 33 52 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619486 IH In-Stock Unstable AKR1C2 51 37 CC[C@H](N[C@@H]1CCC[C@@H](O)C1)c1ccc(OC)c(OC)c1 ZINC000217619510 CG On-Demand Unstable PDE4A 39 41 CC[C@H](N[C@@H]1CCC[C@@H](O)C1)c1ccc(OC)c(OC)c1 ZINC000217619510 CG On-Demand Unstable PDE4B 21 40 O=C(N/C=C/c1ccccc1)N1CCC(Cc2ccccc2)CC1 ZINC000217619511 DI For-Sale Unstable GRIN2B 95 58 O=C(N/C=C/c1ccccc1)N1CCC(Cc2ccccc2)CC1 ZINC000217619511 DI For-Sale Unstable SIGMAR1 35 47 O=C(N/C=C/c1ccccc1)N1CCC(Cc2ccccc2)CC1 ZINC000217619511 DI For-Sale Unstable CCR3 55 44 O=C(N/C=C/c1ccccc1)N1CCC(Cc2ccccc2)CC1 ZINC000217619511 DI For-Sale Unstable AMP1_PLAFQ 26 53 C[C@H](O)c1cc(Br)ccc1N1CC[C@@H](c2ccccc2)C1 ZINC000217619529 EI For-Sale Unstable VACHT_TETCF 0 44 C[C@H](O)c1cc(Br)ccc1N1CC[C@@H](c2ccccc2)C1 ZINC000217619529 EI For-Sale Unstable SLC18A3 31 45 O=C(Nc1ccc(N2CCCCC2)cc1)C(F)F ZINC000217619531 CF On-Demand Unstable KCNQ2 64 56 O=C1O[C@@]2(CCCN(S(=O)(=O)c3cccc4ccccc34)C2)c2ccccc21 ZINC000217619550 GH For-Sale Unstable NPY5R 27 40 CCn1c(C)cc(C)c(C(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)c1=O ZINC000217619580 FD In-Stock Unstable CHRNA4 29 47 CC[C@@H](N[C@H]1CCC[C@@H](O)C1)c1ccc(OC)c(OC)c1 ZINC000217619597 CG For-Sale Unstable PDE4A 39 41 CC[C@@H](N[C@H]1CCC[C@@H](O)C1)c1ccc(OC)c(OC)c1 ZINC000217619597 CG For-Sale Unstable PDE4B 21 40 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619599 JI In-Stock Unstable ADRB1 43 38 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619599 JI In-Stock Unstable ADRB3 57 38 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619599 JI In-Stock Unstable TBXA2R 46 42 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619599 JI In-Stock Unstable TBXAS1 19 41 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619599 JI In-Stock Unstable BMP1 76 41 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619599 JI In-Stock Unstable KCNA5 24 41 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619599 JI In-Stock Unstable MMP13 56 40 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619599 JI In-Stock Unstable BDKRB1 0 41 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619599 JI In-Stock Unstable ADAM17 29 40 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619599 JI In-Stock Unstable ALOX15B 0 40 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619599 JI In-Stock Unstable MMP2 41 41 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619599 JI In-Stock Unstable MMP3 39 41 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619599 JI In-Stock Unstable ALOX15 54 40 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619599 JI In-Stock Unstable MMP9 48 40 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619599 JI In-Stock Unstable IAP 0 41 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619599 JI In-Stock Unstable ADAMTS4 41 35 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619599 JI In-Stock Unstable CA9 19 40 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619599 JI In-Stock Unstable MMP1 43 38 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619599 JI In-Stock Unstable AKR1C3 31 48 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619599 JI In-Stock Unstable AKR1C2 49 35 CN1CCC(N(C)C(=O)N/C=C/c2ccccc2)CC1 ZINC000217619613 CE For-Sale Unstable NPY2R 15 42 C[C@@H](O)c1ccc(Br)cc1N1CC[C@@H](c2ccccc2)C1 ZINC000217619621 EI For-Sale Unstable VACHT_TETCF 0 44 C[C@@H](O)c1ccc(Br)cc1N1CC[C@@H](c2ccccc2)C1 ZINC000217619621 EI For-Sale Unstable SLC18A3 32 45 O=C1O[C@]2(CCCN(S(=O)(=O)c3cccc4ccccc34)C2)c2ccccc21 ZINC000217619631 GH For-Sale Unstable NPY5R 27 40 O=C(COc1ccc(Cl)cc1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217619648 GD In-Stock Unstable MAPK1 45 38 CC(C)c1nc(N(Cc2ccc(OC(F)(F)F)cc2)S(=O)(=O)c2ccc(C(=O)O)cc2)c(C(F)(F)F)c2ccccc12 ZINC000217619650 KK Annotated Unstable BMP1 46 37 CC(C)c1nc(N(Cc2ccc(OC(F)(F)F)cc2)S(=O)(=O)c2ccc(C(=O)O)cc2)c(C(F)(F)F)c2ccccc12 ZINC000217619650 KK Annotated Unstable MMP13 23 42 CC(C)c1nc(N(Cc2ccc(OC(F)(F)F)cc2)S(=O)(=O)c2ccc(C(=O)O)cc2)c(C(F)(F)F)c2ccccc12 ZINC000217619650 KK Annotated Unstable ADAM17 21 42 CC(C)c1nc(N(Cc2ccc(OC(F)(F)F)cc2)S(=O)(=O)c2ccc(C(=O)O)cc2)c(C(F)(F)F)c2ccccc12 ZINC000217619650 KK Annotated Unstable MMP9 31 42 CC(C)c1nc(N(Cc2ccc(OC(F)(F)F)cc2)S(=O)(=O)c2ccc(C(=O)O)cc2)c(C(F)(F)F)c2ccccc12 ZINC000217619650 KK Annotated Unstable MMP1 18 42 CC(C)c1nc(N(Cc2ccc(OC(F)(F)F)cc2)S(=O)(=O)c2ccc(C(=O)O)cc2)c(C(F)(F)F)c2ccccc12 ZINC000217619650 KK Annotated Unstable TRPM8 63 55 CC[C@H](N[C@H]1CCC[C@@H](O)C1)c1ccc(OC)c(OC)c1 ZINC000217619673 CG On-Demand Unstable PDE4A 39 41 CC[C@H](N[C@H]1CCC[C@@H](O)C1)c1ccc(OC)c(OC)c1 ZINC000217619673 CG On-Demand Unstable PDE4B 21 40 CN1CCCC[C@@H]1CNC[C@@H](O)c1cccs1 ZINC000217619685 CD For-Sale Unstable CHRNA10 49 35 CN1CCCC[C@@H]1CNC[C@@H](O)c1cccs1 ZINC000217619685 CD For-Sale Unstable NAMPT 0 40 COc1cccc2c(O)c(C(=O)NCCc3c[nH]cn3)cnc12 ZINC000217619689 DD In-Stock Unstable HRH2 46 34 COc1cccc2c(O)c(C(=O)NCCc3c[nH]cn3)cnc12 ZINC000217619689 DD In-Stock Unstable HRH3 56 44 BrCc1ccc(-n2nnc(-c3ccccc3)n2)cc1 ZINC000217619694 DG For-Sale Unstable GRM5 18 42 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619697 JI In-Stock Unstable ADRB1 43 38 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619697 JI In-Stock Unstable ADRB3 57 38 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619697 JI In-Stock Unstable TBXA2R 46 42 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619697 JI In-Stock Unstable TBXAS1 19 41 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619697 JI In-Stock Unstable BMP1 76 41 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619697 JI In-Stock Unstable KCNA5 24 41 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619697 JI In-Stock Unstable MMP13 56 40 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619697 JI In-Stock Unstable BDKRB1 0 41 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619697 JI In-Stock Unstable ADAM17 29 40 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619697 JI In-Stock Unstable ALOX15B 0 40 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619697 JI In-Stock Unstable MMP2 41 41 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619697 JI In-Stock Unstable MMP3 39 41 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619697 JI In-Stock Unstable ALOX15 54 40 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619697 JI In-Stock Unstable MMP9 48 40 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619697 JI In-Stock Unstable IAP 0 41 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619697 JI In-Stock Unstable ADAMTS4 41 35 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619697 JI In-Stock Unstable CA9 19 40 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619697 JI In-Stock Unstable MMP1 43 38 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619697 JI In-Stock Unstable AKR1C3 31 48 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@H](C)c3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619697 JI In-Stock Unstable AKR1C2 49 35 C[C@H](O)c1ccc(Br)cc1N1CC[C@@H](c2ccccc2)C1 ZINC000217619702 EI For-Sale Unstable VACHT_TETCF 0 44 C[C@H](O)c1ccc(Br)cc1N1CC[C@@H](c2ccccc2)C1 ZINC000217619702 EI For-Sale Unstable SLC18A3 32 45 O=C(Nc1ccc(N2CCOCC2)cc1N1CCOCC1)c1nn(-c2ccccc2)c2c1CCC2 ZINC000217619707 JG On-Demand Unstable CNR1 51 31 O=C(Nc1ccc(N2CCOCC2)cc1N1CCOCC1)c1nn(-c2ccccc2)c2c1CCC2 ZINC000217619707 JG On-Demand Unstable CSF1R 26 43 COc1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217619717 CG For-Sale Unstable BMP1 46 45 COc1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217619717 CG For-Sale Unstable NQO2 25 40 COc1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217619717 CG For-Sale Unstable MMP13 26 41 COc1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217619717 CG For-Sale Unstable HDAC8 26 40 COc1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217619717 CG For-Sale Unstable MMP16 0 40 COc1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217619717 CG For-Sale Unstable MTNR1A 93 42 COc1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217619717 CG For-Sale Unstable MTNR1B 81 41 COc1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217619717 CG For-Sale Unstable MMP2 30 50 COc1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217619717 CG For-Sale Unstable MMP3 38 45 COc1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217619717 CG For-Sale Unstable MMP8 20 40 COc1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217619717 CG For-Sale Unstable HDAC6 17 40 COc1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217619717 CG For-Sale Unstable MMP9 33 50 COc1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217619717 CG For-Sale Unstable MMP12 25 40 COc1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217619717 CG For-Sale Unstable CA9 18 45 COc1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217619717 CG For-Sale Unstable MMP1 35 42 COc1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217619717 CG For-Sale Unstable GPR183 0 41 COc1ccc(Cl)cc1C(=O)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217619754 GE In-Stock Unstable MAPK1 44 40 COc1ccc(Cl)cc1C(=O)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217619754 GE In-Stock Unstable HSP90AB1 0 50 COC(=O)/C(O)=C\c1ccc(O)cc1 ZINC000217619758 AD For-Sale Unstable CA7 0 50 COC(=O)/C(O)=C\c1ccc(O)cc1 ZINC000217619758 AD For-Sale Unstable CA14 0 50 COC(=O)/C(O)=C\c1ccc(O)cc1 ZINC000217619758 AD For-Sale Unstable LSDA 0 43 COC(=O)/C(O)=C\c1ccc(O)cc1 ZINC000217619758 AD For-Sale Unstable TLR4 38 53 CN1CCCC[C@H]1CNC[C@@H](O)c1cccs1 ZINC000217619764 CD For-Sale Unstable CHRNA10 49 35 CN1CCCC[C@H]1CNC[C@@H](O)c1cccs1 ZINC000217619764 CD For-Sale Unstable NAMPT 0 40 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619777 JH In-Stock Unstable CA2 25 44 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619777 JH In-Stock Unstable TBXA2R 55 46 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619777 JH In-Stock Unstable TBXAS1 32 46 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619777 JH In-Stock Unstable HTR7 17 40 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619777 JH In-Stock Unstable BMP1 80 42 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619777 JH In-Stock Unstable CA1 26 45 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619777 JH In-Stock Unstable KCNA5 26 40 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619777 JH In-Stock Unstable MMP13 78 44 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619777 JH In-Stock Unstable BDKRB1 0 42 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619777 JH In-Stock Unstable ADAM17 55 43 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619777 JH In-Stock Unstable ALOX15B 0 42 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619777 JH In-Stock Unstable CA14 18 45 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619777 JH In-Stock Unstable MMP2 50 42 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619777 JH In-Stock Unstable MMP3 56 42 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619777 JH In-Stock Unstable MMP8 35 40 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619777 JH In-Stock Unstable MMP14 27 40 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619777 JH In-Stock Unstable PRTN3 47 33 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619777 JH In-Stock Unstable ALOX15 69 42 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619777 JH In-Stock Unstable MMP9 68 44 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619777 JH In-Stock Unstable MMP12 39 40 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619777 JH In-Stock Unstable CA12 19 44 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619777 JH In-Stock Unstable PTGDR 24 43 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619777 JH In-Stock Unstable MMP7 42 42 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619777 JH In-Stock Unstable IAP 0 46 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619777 JH In-Stock Unstable CA9 28 44 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619777 JH In-Stock Unstable MMP1 67 42 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619777 JH In-Stock Unstable AKR1C3 34 54 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1 ZINC000217619777 JH In-Stock Unstable AKR1C2 53 39 COC[C@H](C)NC(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217619778 CD For-Sale Unstable TNFRSF1A 19 40 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)Nc3cccc4[nH]ccc34)[C@H]21 ZINC000217619796 JH In-Stock Unstable TSHR 41 32 CN(CCOc1ccc(Br)cc1)C(=O)C(F)F ZINC000217619827 DF On-Demand Unstable LSS 60 43 O=C(N/C=C/c1ccccc1)NC[C@@H]1CCCO1 ZINC000217619836 BE For-Sale Unstable OXTR 27 44 O=C(N/C=C/c1ccccc1)NC[C@@H]1CCCO1 ZINC000217619836 BE For-Sale Unstable AVPR1A 0 41 O=C(N/C=C/c1ccccc1)NC[C@@H]1CCCO1 ZINC000217619836 BE For-Sale Unstable PDE8B 17 41 O=C(c1cccc(C(F)(F)F)c1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217619848 GF In-Stock Unstable MAP3K12 16 41 O=C(c1cccc(C(F)(F)F)c1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217619848 GF In-Stock Unstable SLC6A7 0 42 COC(=O)/C(O)=C/c1ccc(O)cc1 ZINC000217619849 AD For-Sale Unstable CA7 0 50 COC(=O)/C(O)=C/c1ccc(O)cc1 ZINC000217619849 AD For-Sale Unstable CA14 0 50 COC(=O)/C(O)=C/c1ccc(O)cc1 ZINC000217619849 AD For-Sale Unstable LSDA 0 43 COC(=O)/C(O)=C/c1ccc(O)cc1 ZINC000217619849 AD For-Sale Unstable TLR4 38 53 COC[C@@H](C)NC(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217619864 CD For-Sale Unstable TNFRSF1A 19 40 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)Nc3cccc4[nH]ccc34)[C@@H]21 ZINC000217619872 JH In-Stock Unstable TSHR 41 32 CN1CCCC[C@@H]1CNC[C@@H](O)c1ccccc1Cl ZINC000217619881 CE For-Sale Unstable OPRL1 46 47 CN1CCCC[C@@H]1CNC[C@@H](O)c1ccccc1Cl ZINC000217619881 CE For-Sale Unstable CHRNA10 57 42 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)cc3)cc2C(=O)O)cc1 ZINC000217619882 JH In-Stock Unstable CA2 25 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)cc3)cc2C(=O)O)cc1 ZINC000217619882 JH In-Stock Unstable TBXA2R 55 48 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)cc3)cc2C(=O)O)cc1 ZINC000217619882 JH In-Stock Unstable TBXAS1 25 46 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)cc3)cc2C(=O)O)cc1 ZINC000217619882 JH In-Stock Unstable BMP1 79 39 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)cc3)cc2C(=O)O)cc1 ZINC000217619882 JH In-Stock Unstable CA1 28 48 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)cc3)cc2C(=O)O)cc1 ZINC000217619882 JH In-Stock Unstable MMP13 63 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)cc3)cc2C(=O)O)cc1 ZINC000217619882 JH In-Stock Unstable BDKRB1 0 40 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)cc3)cc2C(=O)O)cc1 ZINC000217619882 JH In-Stock Unstable ADAM17 40 38 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)cc3)cc2C(=O)O)cc1 ZINC000217619882 JH In-Stock Unstable ALOX15B 0 40 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)cc3)cc2C(=O)O)cc1 ZINC000217619882 JH In-Stock Unstable CA14 15 48 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)cc3)cc2C(=O)O)cc1 ZINC000217619882 JH In-Stock Unstable MMP2 38 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)cc3)cc2C(=O)O)cc1 ZINC000217619882 JH In-Stock Unstable MMP3 52 38 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)cc3)cc2C(=O)O)cc1 ZINC000217619882 JH In-Stock Unstable MMP8 30 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)cc3)cc2C(=O)O)cc1 ZINC000217619882 JH In-Stock Unstable MMP14 18 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)cc3)cc2C(=O)O)cc1 ZINC000217619882 JH In-Stock Unstable ALOX15 51 40 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)cc3)cc2C(=O)O)cc1 ZINC000217619882 JH In-Stock Unstable MMP9 55 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)cc3)cc2C(=O)O)cc1 ZINC000217619882 JH In-Stock Unstable MMP12 27 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)cc3)cc2C(=O)O)cc1 ZINC000217619882 JH In-Stock Unstable CA12 20 46 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)cc3)cc2C(=O)O)cc1 ZINC000217619882 JH In-Stock Unstable PTGDR 26 45 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)cc3)cc2C(=O)O)cc1 ZINC000217619882 JH In-Stock Unstable MMP7 40 38 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)cc3)cc2C(=O)O)cc1 ZINC000217619882 JH In-Stock Unstable IAP 0 48 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)cc3)cc2C(=O)O)cc1 ZINC000217619882 JH In-Stock Unstable CA9 27 46 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)cc3)cc2C(=O)O)cc1 ZINC000217619882 JH In-Stock Unstable MMP1 57 39 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)cc3)cc2C(=O)O)cc1 ZINC000217619882 JH In-Stock Unstable AKR1C3 32 52 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)cc3)cc2C(=O)O)cc1 ZINC000217619882 JH In-Stock Unstable AKR1C2 54 40 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)cc3)cc2C(=O)O)cc1 ZINC000217619882 JH In-Stock Unstable A6YCJ1_9METZ 15 41 CN1[C@@H]2CC[C@@H]1CC(N[C@@H](c1ccccc1)C(C)(C)C)C2 ZINC000217619923 CH For-Sale Unstable CHRM1 22 58 CN1[C@@H]2CC[C@@H]1CC(N[C@@H](c1ccccc1)C(C)(C)C)C2 ZINC000217619923 CH For-Sale Unstable SLC6A1 0 58 CN1[C@@H]2CC[C@@H]1CC(N[C@@H](c1ccccc1)C(C)(C)C)C2 ZINC000217619923 CH For-Sale Unstable SLC6A3 28 58 CN1[C@@H]2CC[C@@H]1CC(N[C@@H](c1ccccc1)C(C)(C)C)C2 ZINC000217619923 CH For-Sale Unstable CHRM4 18 48 CN1[C@@H]2CC[C@@H]1CC(N[C@@H](c1ccccc1)C(C)(C)C)C2 ZINC000217619923 CH For-Sale Unstable GLRA1 42 31 O=C(N/C=C/c1ccccc1)NC[C@H]1CCCO1 ZINC000217619928 BE For-Sale Unstable OXTR 27 44 O=C(N/C=C/c1ccccc1)NC[C@H]1CCCO1 ZINC000217619928 BE For-Sale Unstable AVPR1A 0 41 O=C(N/C=C/c1ccccc1)NC[C@H]1CCCO1 ZINC000217619928 BE For-Sale Unstable PDE8B 17 41 CC(C)(C)c1ccc(S(=O)(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217619958 GH For-Sale Unstable NPY5R 24 42 CN1CCCC[C@H]1CNC[C@@H](O)c1ccccc1Cl ZINC000217619975 CE For-Sale Unstable OPRL1 46 47 CN1CCCC[C@H]1CNC[C@@H](O)c1ccccc1Cl ZINC000217619975 CE For-Sale Unstable CHRNA10 57 42 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccc(OC)c(OC)c3)c(C(=O)O)c2)cc1 ZINC000217619994 KH In-Stock Unstable TBXA2R 51 43 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccc(OC)c(OC)c3)c(C(=O)O)c2)cc1 ZINC000217619994 KH In-Stock Unstable TBXAS1 19 46 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccc(OC)c(OC)c3)c(C(=O)O)c2)cc1 ZINC000217619994 KH In-Stock Unstable PTGDR 35 40 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccc(OC)c(OC)c3)c(C(=O)O)c2)cc1 ZINC000217619994 KH In-Stock Unstable IAP 0 46 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccc(OC)c(OC)c3)c(C(=O)O)c2)cc1 ZINC000217619994 KH In-Stock Unstable CA9 22 41 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccc(OC)c(OC)c3)c(C(=O)O)c2)cc1 ZINC000217619994 KH In-Stock Unstable AKR1C3 28 48 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccc(OC)c(OC)c3)c(C(=O)O)c2)cc1 ZINC000217619994 KH In-Stock Unstable AKR1C2 46 38 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccc(OC)c(OC)c3)c(C(=O)O)c2)cc1 ZINC000217619994 KH In-Stock Unstable SCMU_MYCTU 0 44 C[C@@H](NC(=O)N/C=C/c1ccccc1)c1ccccc1 ZINC000217620036 CH For-Sale Unstable ACACA 32 41 CC(C)(C)c1ccc(S(=O)(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217620043 GH For-Sale Unstable NPY5R 24 42 CN1CCCC[C@@H]1CNC[C@@H](O)c1cc(Cl)ccc1Cl ZINC000217620081 DG For-Sale Unstable CHRNA10 52 44 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccco3)c(C(=O)O)c2)cc1 ZINC000217620093 IG In-Stock Unstable TBXA2R 46 43 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccco3)c(C(=O)O)c2)cc1 ZINC000217620093 IG In-Stock Unstable TBXAS1 15 40 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccco3)c(C(=O)O)c2)cc1 ZINC000217620093 IG In-Stock Unstable BMP1 37 41 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccco3)c(C(=O)O)c2)cc1 ZINC000217620093 IG In-Stock Unstable IAP 0 41 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccco3)c(C(=O)O)c2)cc1 ZINC000217620093 IG In-Stock Unstable AKR1C3 26 46 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccco3)c(C(=O)O)c2)cc1 ZINC000217620093 IG In-Stock Unstable AKR1C2 40 33 O=C(O)/C=C\c1cccc(C(=O)Nc2ccc(F)cc2)c1 ZINC000217620117 CG For-Sale Anodyne MAOB 0 41 O=C(O)/C=C\c1cccc(C(=O)Nc2ccc(F)cc2)c1 ZINC000217620117 CG For-Sale Anodyne UL80 22 41 O=C(O)/C=C\c1cccc(C(=O)Nc2ccc(F)cc2)c1 ZINC000217620117 CG For-Sale Anodyne CXCR2 0 45 O=C(O)/C=C\c1cccc(C(=O)Nc2ccc(F)cc2)c1 ZINC000217620117 CG For-Sale Anodyne PRNP 17 42 O=C(O)/C=C\c1cccc(C(=O)Nc2ccc(F)cc2)c1 ZINC000217620117 CG For-Sale Anodyne MMP2 0 57 O=C(O)/C=C\c1cccc(C(=O)Nc2ccc(F)cc2)c1 ZINC000217620117 CG For-Sale Anodyne TDO2 0 41 O=C(O)/C=C\c1cccc(C(=O)Nc2ccc(F)cc2)c1 ZINC000217620117 CG For-Sale Anodyne MMP9 0 57 O=C(O)/C=C\c1cccc(C(=O)Nc2ccc(F)cc2)c1 ZINC000217620117 CG For-Sale Anodyne MMP1 22 57 O=C(O)/C=C\c1cccc(C(=O)Nc2ccc(F)cc2)c1 ZINC000217620117 CG For-Sale Anodyne AKR1C3 44 37 O=C(O)/C=C\c1cccc(C(=O)Nc2ccc(F)cc2)c1 ZINC000217620117 CG For-Sale Anodyne RHOA 0 41 O=C(O)/C=C\c1cccc(C(=O)Nc2ccc(F)cc2)c1 ZINC000217620117 CG For-Sale Anodyne SENP1 0 40 O=C(O)/C=C\c1cccc(C(=O)Nc2ccc(F)cc2)c1 ZINC000217620117 CG For-Sale Anodyne KCNK3 109 53 O=C(O)/C=C\c1cccc(C(=O)Nc2ccc(F)cc2)c1 ZINC000217620117 CG For-Sale Anodyne KCNK9 58 46 C[C@H](NC(=O)N/C=C/c1ccccc1)c1ccccc1 ZINC000217620125 CH For-Sale Unstable ACACA 32 41 CN1CCCC[C@H]1CNC[C@@H](O)c1cc(Cl)ccc1Cl ZINC000217620163 DG For-Sale Unstable CHRNA10 52 44 Cc1cc(C)c(C)c(S(=O)(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1C ZINC000217620174 GH For-Sale Unstable NPY5R 26 41 CNS(=O)(=O)c1ccc(CCC(=O)NCCc2scnc2C)cc1 ZINC000217620197 FD In-Stock Unstable CA2 17 44 CNS(=O)(=O)c1ccc(CCC(=O)NCCc2scnc2C)cc1 ZINC000217620197 FD In-Stock Unstable CA4 15 42 O=C(O)/C=C\c1ccc(C(=O)Nc2ccccc2Cl)s1 ZINC000217620199 DH For-Sale Anodyne EPHB3 63 42 COc1ccc(CCNS(=O)(=O)c2ccc(NC[C@@H]3CCCO3)c(C(=O)O)c2)cc1 ZINC000217620217 IF In-Stock Unstable TBXA2R 32 41 COc1ccc(CCNS(=O)(=O)c2ccc(NC[C@@H]3CCCO3)c(C(=O)O)c2)cc1 ZINC000217620217 IF In-Stock Unstable BMP1 50 33 COc1ccc(CCNS(=O)(=O)c2ccc(NC[C@@H]3CCCO3)c(C(=O)O)c2)cc1 ZINC000217620217 IF In-Stock Unstable MMP13 40 36 COc1ccc(CCNS(=O)(=O)c2ccc(NC[C@@H]3CCCO3)c(C(=O)O)c2)cc1 ZINC000217620217 IF In-Stock Unstable IAP 0 41 COc1ccc(CCNS(=O)(=O)c2ccc(NC[C@@H]3CCCO3)c(C(=O)O)c2)cc1 ZINC000217620217 IF In-Stock Unstable AKR1C3 25 44 Cc1cc(C)c(C)c(S(=O)(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1C ZINC000217620268 GH For-Sale Unstable NPY5R 26 41 CCOCCCNC(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217620280 CD For-Sale Unstable KCNQ1 0 40 CCOCCCNC(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217620280 CD For-Sale Unstable HDA106 0 42 NCCCC[C@@H]1NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](CC(=O)O)NC(=O)CNC(=O)[C@H](CCCN=C(N)N)NC1=O ZINC000217620283 KA For-Sale Mild BDKRB2 18 45 NCCCC[C@@H]1NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](CC(=O)O)NC(=O)CNC(=O)[C@H](CCCN=C(N)N)NC1=O ZINC000217620283 KA For-Sale Mild SSTR4 21 41 NCCCC[C@@H]1NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](CC(=O)O)NC(=O)CNC(=O)[C@H](CCCN=C(N)N)NC1=O ZINC000217620283 KA For-Sale Mild GALR1 45 32 NCCCC[C@@H]1NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](CC(=O)O)NC(=O)CNC(=O)[C@H](CCCN=C(N)N)NC1=O ZINC000217620283 KA For-Sale Mild CXCR4 81 63 NCCCC[C@@H]1NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](CC(=O)O)NC(=O)CNC(=O)[C@H](CCCN=C(N)N)NC1=O ZINC000217620283 KA For-Sale Mild UTS2R 24 48 NCCCC[C@@H]1NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](CC(=O)O)NC(=O)CNC(=O)[C@H](CCCN=C(N)N)NC1=O ZINC000217620283 KA For-Sale Mild MC3R 36 45 NCCCC[C@@H]1NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](CC(=O)O)NC(=O)CNC(=O)[C@H](CCCN=C(N)N)NC1=O ZINC000217620283 KA For-Sale Mild MC5R 30 41 NCCCC[C@@H]1NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](CC(=O)O)NC(=O)CNC(=O)[C@H](CCCN=C(N)N)NC1=O ZINC000217620283 KA For-Sale Mild HDAC3 15 40 NCCCC[C@@H]1NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](CC(=O)O)NC(=O)CNC(=O)[C@H](CCCN=C(N)N)NC1=O ZINC000217620283 KA For-Sale Mild ITGA3 62 39 NCCCC[C@@H]1NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](CC(=O)O)NC(=O)CNC(=O)[C@H](CCCN=C(N)N)NC1=O ZINC000217620283 KA For-Sale Mild SSTR3 22 41 NCCCC[C@@H]1NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](CC(=O)O)NC(=O)CNC(=O)[C@H](CCCN=C(N)N)NC1=O ZINC000217620283 KA For-Sale Mild MC1R 19 50 NCCCC[C@@H]1NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](CC(=O)O)NC(=O)CNC(=O)[C@H](CCCN=C(N)N)NC1=O ZINC000217620283 KA For-Sale Mild ITGAV 26 53 CN1CCCC[C@@H]1CNC[C@@H](O)c1ccc(F)cc1F ZINC000217620290 CE For-Sale Unstable CHRNA10 56 39 CN1CCCC[C@@H]1CNC[C@@H](O)c1ccc(F)cc1F ZINC000217620290 CE For-Sale Unstable ACKR3 40 34 CN1CCCC[C@@H]1CCNC[C@@H](O)c1ccccc1 ZINC000217620291 CE For-Sale Unstable ADRB2 25 42 CN1CCCC[C@@H]1CCNC[C@@H](O)c1ccccc1 ZINC000217620291 CE For-Sale Unstable ADRB1 34 40 CN1CCCC[C@@H]1CCNC[C@@H](O)c1ccccc1 ZINC000217620291 CE For-Sale Unstable HRH1 15 40 CN1CCCC[C@@H]1CCNC[C@@H](O)c1ccccc1 ZINC000217620291 CE For-Sale Unstable SLC6A3 18 45 CN1CCCC[C@@H]1CCNC[C@@H](O)c1ccccc1 ZINC000217620291 CE For-Sale Unstable SLC18A2 55 44 CN1CCCC[C@@H]1CCNC[C@@H](O)c1ccccc1 ZINC000217620291 CE For-Sale Unstable CHRM5 20 40 CN1CCCC[C@@H]1CCNC[C@@H](O)c1ccccc1 ZINC000217620291 CE For-Sale Unstable ADRB3 58 40 CN1CCCC[C@@H]1CCNC[C@@H](O)c1ccccc1 ZINC000217620291 CE For-Sale Unstable CHRNA10 52 41 CN1CCCC[C@@H]1CCNC[C@@H](O)c1ccccc1 ZINC000217620291 CE For-Sale Unstable Q8WSF8_APLCA 18 44 COc1ccc(CCNS(=O)(=O)c2ccc(NC[C@H]3CCCO3)c(C(=O)O)c2)cc1 ZINC000217620304 IF In-Stock Unstable TBXA2R 32 41 COc1ccc(CCNS(=O)(=O)c2ccc(NC[C@H]3CCCO3)c(C(=O)O)c2)cc1 ZINC000217620304 IF In-Stock Unstable BMP1 50 33 COc1ccc(CCNS(=O)(=O)c2ccc(NC[C@H]3CCCO3)c(C(=O)O)c2)cc1 ZINC000217620304 IF In-Stock Unstable MMP13 40 36 COc1ccc(CCNS(=O)(=O)c2ccc(NC[C@H]3CCCO3)c(C(=O)O)c2)cc1 ZINC000217620304 IF In-Stock Unstable IAP 0 41 COc1ccc(CCNS(=O)(=O)c2ccc(NC[C@H]3CCCO3)c(C(=O)O)c2)cc1 ZINC000217620304 IF In-Stock Unstable AKR1C3 25 44 COc1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620358 CG For-Sale Unstable ANPEP 37 50 COc1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620358 CG For-Sale Unstable PTGER4 0 43 COc1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620358 CG For-Sale Unstable BMP1 45 42 COc1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620358 CG For-Sale Unstable MMP13 47 45 COc1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620358 CG For-Sale Unstable HDAC8 19 40 COc1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620358 CG For-Sale Unstable MTNR1A 39 44 COc1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620358 CG For-Sale Unstable MTNR1B 36 44 COc1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620358 CG For-Sale Unstable MMP2 28 49 COc1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620358 CG For-Sale Unstable MMP3 38 40 COc1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620358 CG For-Sale Unstable HDAC1 16 43 COc1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620358 CG For-Sale Unstable MMP9 48 49 COc1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620358 CG For-Sale Unstable MMP7 19 40 COc1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620358 CG For-Sale Unstable CA9 18 43 COc1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620358 CG For-Sale Unstable MMP1 47 45 COc1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620358 CG For-Sale Unstable U38 0 41 COc1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620358 CG For-Sale Unstable AMP1_PLAFQ 51 40 COc1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620358 CG For-Sale Unstable KCNJ2 0 42 COc1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620358 CG For-Sale Unstable PDS 49 38 COc1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620358 CG For-Sale Unstable GPR183 0 43 CCOCCCNC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217620363 CD For-Sale Unstable DRD4 40 30 CN1CCCC[C@H]1CCNC[C@@H](O)c1ccccc1 ZINC000217620371 CE For-Sale Unstable ADRB2 25 42 CN1CCCC[C@H]1CCNC[C@@H](O)c1ccccc1 ZINC000217620371 CE For-Sale Unstable ADRB1 34 40 CN1CCCC[C@H]1CCNC[C@@H](O)c1ccccc1 ZINC000217620371 CE For-Sale Unstable HRH1 15 40 CN1CCCC[C@H]1CCNC[C@@H](O)c1ccccc1 ZINC000217620371 CE For-Sale Unstable SLC6A3 18 45 CN1CCCC[C@H]1CCNC[C@@H](O)c1ccccc1 ZINC000217620371 CE For-Sale Unstable SLC18A2 55 44 CN1CCCC[C@H]1CCNC[C@@H](O)c1ccccc1 ZINC000217620371 CE For-Sale Unstable CHRM5 20 40 CN1CCCC[C@H]1CCNC[C@@H](O)c1ccccc1 ZINC000217620371 CE For-Sale Unstable ADRB3 58 40 CN1CCCC[C@H]1CCNC[C@@H](O)c1ccccc1 ZINC000217620371 CE For-Sale Unstable CHRNA10 52 41 CN1CCCC[C@H]1CCNC[C@@H](O)c1ccccc1 ZINC000217620371 CE For-Sale Unstable Q8WSF8_APLCA 18 44 CN1CCCC[C@H]1CNC[C@@H](O)c1ccc(F)cc1F ZINC000217620373 CE For-Sale Unstable CHRNA10 56 39 CN1CCCC[C@H]1CNC[C@@H](O)c1ccc(F)cc1F ZINC000217620373 CE For-Sale Unstable ACKR3 40 34 CC(=O)Nc1ccc(S(=O)(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217620380 HE For-Sale Unstable LPL 41 33 CC(=O)Nc1ccc(S(=O)(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217620380 HE For-Sale Unstable NPY5R 35 40 CC(=O)Nc1ccc(S(=O)(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217620380 HE For-Sale Unstable TGM2 58 36 CC(=O)Nc1ccc(S(=O)(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217620380 HE For-Sale Unstable F13A1 86 40 CC(=O)Nc1ccc(S(=O)(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217620380 HE For-Sale Unstable NAMPT 24 40 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCC3)c(C(=O)O)c2)cc1 ZINC000217620423 HF In-Stock Unstable CA2 15 40 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCC3)c(C(=O)O)c2)cc1 ZINC000217620423 HF In-Stock Unstable TBXA2R 52 45 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCC3)c(C(=O)O)c2)cc1 ZINC000217620423 HF In-Stock Unstable TBXAS1 18 42 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCC3)c(C(=O)O)c2)cc1 ZINC000217620423 HF In-Stock Unstable HTR7 26 44 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCC3)c(C(=O)O)c2)cc1 ZINC000217620423 HF In-Stock Unstable BMP1 74 36 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCC3)c(C(=O)O)c2)cc1 ZINC000217620423 HF In-Stock Unstable CA1 15 44 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCC3)c(C(=O)O)c2)cc1 ZINC000217620423 HF In-Stock Unstable MMP13 74 40 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCC3)c(C(=O)O)c2)cc1 ZINC000217620423 HF In-Stock Unstable HTR6 25 42 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCC3)c(C(=O)O)c2)cc1 ZINC000217620423 HF In-Stock Unstable ADAM17 44 40 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCC3)c(C(=O)O)c2)cc1 ZINC000217620423 HF In-Stock Unstable MMP2 43 40 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCC3)c(C(=O)O)c2)cc1 ZINC000217620423 HF In-Stock Unstable MMP3 62 40 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCC3)c(C(=O)O)c2)cc1 ZINC000217620423 HF In-Stock Unstable MMP8 39 40 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCC3)c(C(=O)O)c2)cc1 ZINC000217620423 HF In-Stock Unstable MMP14 17 40 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCC3)c(C(=O)O)c2)cc1 ZINC000217620423 HF In-Stock Unstable ALOX15 41 38 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCC3)c(C(=O)O)c2)cc1 ZINC000217620423 HF In-Stock Unstable MMP9 63 40 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCC3)c(C(=O)O)c2)cc1 ZINC000217620423 HF In-Stock Unstable MMP12 30 40 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCC3)c(C(=O)O)c2)cc1 ZINC000217620423 HF In-Stock Unstable MMP7 50 40 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCC3)c(C(=O)O)c2)cc1 ZINC000217620423 HF In-Stock Unstable IAP 0 43 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCC3)c(C(=O)O)c2)cc1 ZINC000217620423 HF In-Stock Unstable CA9 24 43 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCC3)c(C(=O)O)c2)cc1 ZINC000217620423 HF In-Stock Unstable MMP1 68 40 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCC3)c(C(=O)O)c2)cc1 ZINC000217620423 HF In-Stock Unstable AKR1C3 27 48 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCC3)c(C(=O)O)c2)cc1 ZINC000217620423 HF In-Stock Unstable AKR1C2 40 33 COc1ccc(Br)c(C(=O)N2CCc3cnc(N4CCOCC4)nc3C2)c1 ZINC000217620445 IE In-Stock Unstable MAPK1 44 34 COc1ccc(Br)c(C(=O)N2CCc3cnc(N4CCOCC4)nc3C2)c1 ZINC000217620445 IE In-Stock Unstable HSP90AB1 0 54 C=CCn1c(COc2ccc(Cl)cc2)nnc1S[C@@H]1CCN(c2ccc(C#N)cc2)C1=O ZINC000217620452 JI On-Demand Unstable VCP 46 39 CN1CCCC[C@@H]1CNC[C@@H](O)c1cc(F)ccc1F ZINC000217620469 CE For-Sale Unstable CHRNA10 57 39 CN1CCCC[C@@H]1CNC[C@@H](O)c1cc(F)ccc1F ZINC000217620469 CE For-Sale Unstable ACKR3 40 33 CC(=O)Nc1ccc(S(=O)(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217620487 HE For-Sale Unstable LPL 41 33 CC(=O)Nc1ccc(S(=O)(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217620487 HE For-Sale Unstable NPY5R 35 40 CC(=O)Nc1ccc(S(=O)(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217620487 HE For-Sale Unstable TGM2 58 36 CC(=O)Nc1ccc(S(=O)(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217620487 HE For-Sale Unstable F13A1 86 40 CC(=O)Nc1ccc(S(=O)(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217620487 HE For-Sale Unstable NAMPT 24 40 C=CCn1c(COc2ccc(Cl)cc2)nnc1S[C@H]1CCN(c2ccc(C#N)cc2)C1=O ZINC000217620530 JI On-Demand Unstable VCP 46 39 O=C(NCCOc1ccccc1)C(F)F ZINC000217620534 BD On-Demand Unstable DRD4 21 45 O=C(NCCOc1ccccc1)C(F)F ZINC000217620534 BD On-Demand Unstable ADRB3 19 45 O=C(NCCOc1ccccc1)C(F)F ZINC000217620534 BD On-Demand Unstable LTA4H 37 43 O=C(NCCOc1ccccc1)C(F)F ZINC000217620534 BD On-Demand Unstable SDH1 0 53 O=C(NCCOc1ccccc1)C(F)F ZINC000217620534 BD On-Demand Unstable MTNR1B 26 48 O=C(NCCOc1ccccc1)C(F)F ZINC000217620534 BD On-Demand Unstable PLA2G4B 46 34 O=C(NCCOc1ccccc1)C(F)F ZINC000217620534 BD On-Demand Unstable FAAH 22 40 O=C(NCCOc1ccccc1)C(F)F ZINC000217620534 BD On-Demand Unstable ACE2 41 32 O=C(NCCOc1ccccc1)C(F)F ZINC000217620534 BD On-Demand Unstable AMP1_PLAFQ 43 35 O=C(NCCOc1ccccc1)C(F)F ZINC000217620534 BD On-Demand Unstable PDS 64 40 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCCC3)c(C(=O)O)c2)cc1 ZINC000217620542 HF In-Stock Unstable TBXA2R 52 44 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCCC3)c(C(=O)O)c2)cc1 ZINC000217620542 HF In-Stock Unstable TBXAS1 17 41 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCCC3)c(C(=O)O)c2)cc1 ZINC000217620542 HF In-Stock Unstable HTR7 25 43 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCCC3)c(C(=O)O)c2)cc1 ZINC000217620542 HF In-Stock Unstable CASP3 23 40 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCCC3)c(C(=O)O)c2)cc1 ZINC000217620542 HF In-Stock Unstable BMP1 71 36 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCCC3)c(C(=O)O)c2)cc1 ZINC000217620542 HF In-Stock Unstable MMP13 69 40 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCCC3)c(C(=O)O)c2)cc1 ZINC000217620542 HF In-Stock Unstable HTR6 23 41 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCCC3)c(C(=O)O)c2)cc1 ZINC000217620542 HF In-Stock Unstable ADAM17 42 39 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCCC3)c(C(=O)O)c2)cc1 ZINC000217620542 HF In-Stock Unstable MMP3 59 40 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCCC3)c(C(=O)O)c2)cc1 ZINC000217620542 HF In-Stock Unstable ALOX15 42 38 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCCC3)c(C(=O)O)c2)cc1 ZINC000217620542 HF In-Stock Unstable MMP9 60 40 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCCC3)c(C(=O)O)c2)cc1 ZINC000217620542 HF In-Stock Unstable MMP7 50 40 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCCC3)c(C(=O)O)c2)cc1 ZINC000217620542 HF In-Stock Unstable IAP 0 43 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCCC3)c(C(=O)O)c2)cc1 ZINC000217620542 HF In-Stock Unstable CA9 17 42 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCCC3)c(C(=O)O)c2)cc1 ZINC000217620542 HF In-Stock Unstable MMP1 65 40 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCCC3)c(C(=O)O)c2)cc1 ZINC000217620542 HF In-Stock Unstable AKR1C3 25 48 Cn1c(CO)nnc1C1CCN(C(=O)CCc2nc3ccccc3[nH]2)CC1 ZINC000217620560 FD In-Stock Unstable ETHR 52 34 O=C(c1ccc(OC(F)(F)F)cc1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217620563 HE In-Stock Unstable SLC6A7 0 41 CN1CCCC[C@H]1CNC[C@@H](O)c1cc(F)ccc1F ZINC000217620564 CE For-Sale Unstable CHRNA10 57 39 CN1CCCC[C@H]1CNC[C@@H](O)c1cc(F)ccc1F ZINC000217620564 CE For-Sale Unstable ACKR3 40 33 O=C(N/C=C/c1ccccc1)NCc1ccc2c(c1)OCO2 ZINC000217620600 CF For-Sale Unstable PDE5A 30 43 O=C(N/C=C/c1ccccc1)NCc1ccc2c(c1)OCO2 ZINC000217620600 CF For-Sale Unstable EDNRB 25 41 O=C(N/C=C/c1ccccc1)NCc1ccc2c(c1)OCO2 ZINC000217620600 CF For-Sale Unstable EDNRA 32 41 O=C(N/C=C/c1ccccc1)NCc1ccc2c(c1)OCO2 ZINC000217620600 CF For-Sale Unstable BMP1 57 40 O=C(N/C=C/c1ccccc1)NCc1ccc2c(c1)OCO2 ZINC000217620600 CF For-Sale Unstable SCN9A 27 45 O=C(N/C=C/c1ccccc1)NCc1ccc2c(c1)OCO2 ZINC000217620600 CF For-Sale Unstable NOS2 93 36 O=C(N/C=C/c1ccccc1)NCc1ccc2c(c1)OCO2 ZINC000217620600 CF For-Sale Unstable MCHR1 17 45 O=C1O[C@@]2(CCCN(S(=O)(=O)c3ccc4c(c3)OCCO4)C2)c2ccccc21 ZINC000217620617 HE For-Sale Unstable PKM 47 53 COc1ccc(N(Cc2cccs2)C(=O)[C@@H](C)NC(=O)c2cccs2)cc1 ZINC000217620629 HI On-Demand Unstable BMP1 39 42 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCOCC3)c(C(=O)O)c2)cc1 ZINC000217620641 HD In-Stock Unstable TBXA2R 50 43 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCOCC3)c(C(=O)O)c2)cc1 ZINC000217620641 HD In-Stock Unstable HTR7 20 42 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCOCC3)c(C(=O)O)c2)cc1 ZINC000217620641 HD In-Stock Unstable BMP1 66 38 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCOCC3)c(C(=O)O)c2)cc1 ZINC000217620641 HD In-Stock Unstable MMP13 66 43 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCOCC3)c(C(=O)O)c2)cc1 ZINC000217620641 HD In-Stock Unstable MMP2 35 43 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCOCC3)c(C(=O)O)c2)cc1 ZINC000217620641 HD In-Stock Unstable MMP3 52 41 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCOCC3)c(C(=O)O)c2)cc1 ZINC000217620641 HD In-Stock Unstable MMP8 35 41 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCOCC3)c(C(=O)O)c2)cc1 ZINC000217620641 HD In-Stock Unstable ALOX15 45 38 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCOCC3)c(C(=O)O)c2)cc1 ZINC000217620641 HD In-Stock Unstable MMP9 53 41 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCOCC3)c(C(=O)O)c2)cc1 ZINC000217620641 HD In-Stock Unstable MMP7 48 39 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCOCC3)c(C(=O)O)c2)cc1 ZINC000217620641 HD In-Stock Unstable IAP 0 45 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCOCC3)c(C(=O)O)c2)cc1 ZINC000217620641 HD In-Stock Unstable CA9 17 41 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCOCC3)c(C(=O)O)c2)cc1 ZINC000217620641 HD In-Stock Unstable MMP1 58 41 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCOCC3)c(C(=O)O)c2)cc1 ZINC000217620641 HD In-Stock Unstable AKR1C3 17 46 C[C@@H](NC(=O)C(F)F)c1ccc(S(N)(=O)=O)cc1 ZINC000217620660 CC On-Demand Unstable CA2 102 49 C[C@@H](NC(=O)C(F)F)c1ccc(S(N)(=O)=O)cc1 ZINC000217620660 CC On-Demand Unstable CA1 79 49 C[C@@H](NC(=O)C(F)F)c1ccc(S(N)(=O)=O)cc1 ZINC000217620660 CC On-Demand Unstable CA7 57 38 C[C@@H](NC(=O)C(F)F)c1ccc(S(N)(=O)=O)cc1 ZINC000217620660 CC On-Demand Unstable CA5B 46 34 C[C@@H](NC(=O)C(F)F)c1ccc(S(N)(=O)=O)cc1 ZINC000217620660 CC On-Demand Unstable CA4 81 45 C[C@@H](NC(=O)C(F)F)c1ccc(S(N)(=O)=O)cc1 ZINC000217620660 CC On-Demand Unstable CA5A 49 34 C[C@@H](NC(=O)C(F)F)c1ccc(S(N)(=O)=O)cc1 ZINC000217620660 CC On-Demand Unstable CA14 39 45 C[C@@H](NC(=O)C(F)F)c1ccc(S(N)(=O)=O)cc1 ZINC000217620660 CC On-Demand Unstable CA12 49 43 C[C@@H](NC(=O)C(F)F)c1ccc(S(N)(=O)=O)cc1 ZINC000217620660 CC On-Demand Unstable CA9 58 41 C[C@@H](NC(=O)C(F)F)c1ccc(S(N)(=O)=O)cc1 ZINC000217620660 CC On-Demand Unstable CYNT 41 36 C[C@@H](NC(=O)C(F)F)c1ccc(S(N)(=O)=O)cc1 ZINC000217620660 CC On-Demand Unstable P96878_MYCTU 54 50 COCC(=O)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217620675 CB In-Stock Unstable MAPK1 51 38 CN1CCCC[C@@H]1CNC[C@@H](O)c1cccc(F)c1 ZINC000217620678 CD For-Sale Unstable CHRNA10 66 47 CN1CCCC[C@@H]1CNC[C@@H](O)c1cccc(F)c1 ZINC000217620678 CD For-Sale Unstable ACKR3 51 35 O=C(NCCc1noc(CO)n1)[C@@H]1CCCCN1Cc1ccccc1 ZINC000217620683 ED In-Stock Unstable FKBP1A 39 43 O=C(NCCc1noc(CO)n1)[C@@H]1CCCCN1Cc1ccccc1 ZINC000217620683 ED In-Stock Unstable TRY1_BOVIN 41 32 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620700 DE For-Sale Unstable CA2 142 66 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620700 DE For-Sale Unstable CA6 26 40 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620700 DE For-Sale Unstable CA1 129 66 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620700 DE For-Sale Unstable CA7 56 52 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620700 DE For-Sale Unstable CA13 21 41 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620700 DE For-Sale Unstable CA5B 70 52 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620700 DE For-Sale Unstable CA4 111 66 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620700 DE For-Sale Unstable CA5A 76 52 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620700 DE For-Sale Unstable CA14 42 52 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620700 DE For-Sale Unstable CA12 100 66 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620700 DE For-Sale Unstable CA9 103 55 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620700 DE For-Sale Unstable CAH_METTE 22 40 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620700 DE For-Sale Unstable IDO1 26 40 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620700 DE For-Sale Unstable CYNT 40 42 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620700 DE For-Sale Unstable NCE103 66 53 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620700 DE For-Sale Unstable MTCA1 68 66 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620700 DE For-Sale Unstable P96878_MYCTU 85 66 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217620700 DE For-Sale Unstable NAMPT 22 40 O=C1O[C@]2(CCCN(S(=O)(=O)c3ccc4c(c3)OCCO4)C2)c2ccccc21 ZINC000217620711 HE For-Sale Unstable PKM 47 53 COc1ccc(N(Cc2cccs2)C(=O)[C@H](C)NC(=O)c2cccs2)cc1 ZINC000217620718 HI On-Demand Unstable BMP1 39 42 C[C@H](NC(=O)C(F)F)c1ccc(S(N)(=O)=O)cc1 ZINC000217620736 CC On-Demand Unstable CA2 102 49 C[C@H](NC(=O)C(F)F)c1ccc(S(N)(=O)=O)cc1 ZINC000217620736 CC On-Demand Unstable CA1 79 49 C[C@H](NC(=O)C(F)F)c1ccc(S(N)(=O)=O)cc1 ZINC000217620736 CC On-Demand Unstable CA7 57 38 C[C@H](NC(=O)C(F)F)c1ccc(S(N)(=O)=O)cc1 ZINC000217620736 CC On-Demand Unstable CA5B 46 34 C[C@H](NC(=O)C(F)F)c1ccc(S(N)(=O)=O)cc1 ZINC000217620736 CC On-Demand Unstable CA4 81 45 C[C@H](NC(=O)C(F)F)c1ccc(S(N)(=O)=O)cc1 ZINC000217620736 CC On-Demand Unstable CA5A 49 34 C[C@H](NC(=O)C(F)F)c1ccc(S(N)(=O)=O)cc1 ZINC000217620736 CC On-Demand Unstable CA14 39 45 C[C@H](NC(=O)C(F)F)c1ccc(S(N)(=O)=O)cc1 ZINC000217620736 CC On-Demand Unstable CA12 49 43 C[C@H](NC(=O)C(F)F)c1ccc(S(N)(=O)=O)cc1 ZINC000217620736 CC On-Demand Unstable CA9 58 41 C[C@H](NC(=O)C(F)F)c1ccc(S(N)(=O)=O)cc1 ZINC000217620736 CC On-Demand Unstable CYNT 41 36 C[C@H](NC(=O)C(F)F)c1ccc(S(N)(=O)=O)cc1 ZINC000217620736 CC On-Demand Unstable P96878_MYCTU 54 50 CCOCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217620762 IF In-Stock Unstable TBXA2R 44 42 CCOCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217620762 IF In-Stock Unstable TBXAS1 15 41 CCOCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217620762 IF In-Stock Unstable BMP1 45 34 CCOCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217620762 IF In-Stock Unstable ALOX15 43 40 CCOCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217620762 IF In-Stock Unstable IAP 0 42 CCOCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217620762 IF In-Stock Unstable CA9 17 40 CCOCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217620762 IF In-Stock Unstable AKR1C3 28 47 CCOCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217620762 IF In-Stock Unstable AKR1C2 49 35 O=C(NCCc1noc(CO)n1)[C@H]1CCCCN1Cc1ccccc1 ZINC000217620770 ED In-Stock Unstable FKBP1A 39 43 O=C(NCCc1noc(CO)n1)[C@H]1CCCCN1Cc1ccccc1 ZINC000217620770 ED In-Stock Unstable TRY1_BOVIN 41 32 CN1CCCC[C@H]1CNC[C@@H](O)c1cccc(F)c1 ZINC000217620771 CD For-Sale Unstable CHRNA10 66 47 CN1CCCC[C@H]1CNC[C@@H](O)c1cccc(F)c1 ZINC000217620771 CD For-Sale Unstable ACKR3 51 35 O=C(N/C=C/c1ccccc1)NCc1ccccc1 ZINC000217620821 CG For-Sale Unstable MME 24 40 O=C(N/C=C/c1ccccc1)NCc1ccccc1 ZINC000217620821 CG For-Sale Unstable ANPEP 43 48 O=C(N/C=C/c1ccccc1)NCc1ccccc1 ZINC000217620821 CG For-Sale Unstable HDAC8 21 44 O=C(N/C=C/c1ccccc1)NCc1ccccc1 ZINC000217620821 CG For-Sale Unstable HDAC1 18 42 O=C(N/C=C/c1ccccc1)NCc1ccccc1 ZINC000217620821 CG For-Sale Unstable HDAC6 18 47 O=C(N/C=C/c1ccccc1)NCc1ccccc1 ZINC000217620821 CG For-Sale Unstable AMP1_PLAFQ 52 44 O=C(N/C=C/c1ccccc1)NCc1ccccc1 ZINC000217620821 CG For-Sale Unstable 17HSDCL 0 43 O=C(N/C=C/c1ccccc1)NCc1ccccc1 ZINC000217620821 CG For-Sale Unstable NAMPT 15 40 O=C(N/C=C/c1ccccc1)NCc1ccccc1 ZINC000217620821 CG For-Sale Unstable PDS 51 35 COc1cc(C)c(C)cc1S(=O)(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217620824 HG For-Sale Unstable NPY5R 24 43 COc1ccc(CCNS(=O)(=O)c2ccc(NCCCOC(C)C)c(C(=O)O)c2)cc1 ZINC000217620837 JG In-Stock Unstable TBXA2R 44 44 COc1ccc(CCNS(=O)(=O)c2ccc(NCCCOC(C)C)c(C(=O)O)c2)cc1 ZINC000217620837 JG In-Stock Unstable TBXAS1 20 43 COc1ccc(CCNS(=O)(=O)c2ccc(NCCCOC(C)C)c(C(=O)O)c2)cc1 ZINC000217620837 JG In-Stock Unstable BMP1 70 35 COc1ccc(CCNS(=O)(=O)c2ccc(NCCCOC(C)C)c(C(=O)O)c2)cc1 ZINC000217620837 JG In-Stock Unstable IAP 0 42 COc1ccc(CCNS(=O)(=O)c2ccc(NCCCOC(C)C)c(C(=O)O)c2)cc1 ZINC000217620837 JG In-Stock Unstable CA9 17 40 COc1ccc(CCNS(=O)(=O)c2ccc(NCCCOC(C)C)c(C(=O)O)c2)cc1 ZINC000217620837 JG In-Stock Unstable AKR1C3 29 47 COc1ccc(CCNS(=O)(=O)c2ccc(NCCCOC(C)C)c(C(=O)O)c2)cc1 ZINC000217620837 JG In-Stock Unstable AKR1C2 50 36 COc1ccc([C@H](O)CNC[C@@H]2CCCCN2C)cc1 ZINC000217620883 CD For-Sale Unstable CHRNA10 63 41 COc1cc(C)c(C)cc1S(=O)(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217620917 HG For-Sale Unstable NPY5R 24 43 C[C@@H](NC(=O)N/C=C/c1ccccc1)C12CC3CC(CC(C3)C1)C2 ZINC000217620933 DJ For-Sale Unstable EPHX2 21 56 CN(C/C=C\CN)CCc1ccccc1 ZINC000217620944 BD For-Sale Unstable AOC3 22 52 CCCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217620966 HH In-Stock Unstable CA2 15 43 CCCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217620966 HH In-Stock Unstable TBXA2R 45 44 CCCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217620966 HH In-Stock Unstable TBXAS1 22 42 CCCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217620966 HH In-Stock Unstable BMP1 44 35 CCCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217620966 HH In-Stock Unstable CA1 16 43 CCCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217620966 HH In-Stock Unstable MMP13 46 39 CCCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217620966 HH In-Stock Unstable ALOX15B 0 47 CCCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217620966 HH In-Stock Unstable ALOX15 65 47 CCCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217620966 HH In-Stock Unstable IAP 0 44 CCCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217620966 HH In-Stock Unstable CA9 22 42 CCCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217620966 HH In-Stock Unstable AKR1C3 29 49 CCCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217620966 HH In-Stock Unstable AKR1C2 52 37 COc1ccc([C@H](O)CNC[C@H]2CCCCN2C)cc1 ZINC000217620972 CD For-Sale Unstable CHRNA10 63 41 O=C(CCc1ccc(C(F)(F)F)cc1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217620997 HF In-Stock Unstable MAPK1 41 35 O=C(CCc1ccc(C(F)(F)F)cc1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217620997 HF In-Stock Unstable GPBAR1 21 42 C[C@H](NC(=O)N/C=C/c1ccccc1)C12CC3CC(CC(C3)C1)C2 ZINC000217621012 DJ For-Sale Unstable EPHX2 21 56 NC1(C(=O)O)C[C@H]2CCC[C@H](C2)C1 ZINC000217621037 AD In-Stock Unstable GRM1 0 44 CCOc1ccc(C)cc1S(=O)(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217621039 HG For-Sale Unstable NPY5R 24 42 CN1CCCC[C@@H]1CNC[C@@H](O)c1ccc(F)c(F)c1 ZINC000217621079 CE For-Sale Unstable CHRNA10 52 44 COc1ccc(CCNS(=O)(=O)c2ccc(NCCC(C)C)c(C(=O)O)c2)cc1 ZINC000217621090 HG In-Stock Unstable TBXA2R 45 44 COc1ccc(CCNS(=O)(=O)c2ccc(NCCC(C)C)c(C(=O)O)c2)cc1 ZINC000217621090 HG In-Stock Unstable TBXAS1 20 41 COc1ccc(CCNS(=O)(=O)c2ccc(NCCC(C)C)c(C(=O)O)c2)cc1 ZINC000217621090 HG In-Stock Unstable BMP1 80 37 COc1ccc(CCNS(=O)(=O)c2ccc(NCCC(C)C)c(C(=O)O)c2)cc1 ZINC000217621090 HG In-Stock Unstable MMP13 58 40 COc1ccc(CCNS(=O)(=O)c2ccc(NCCC(C)C)c(C(=O)O)c2)cc1 ZINC000217621090 HG In-Stock Unstable MMP2 39 40 COc1ccc(CCNS(=O)(=O)c2ccc(NCCC(C)C)c(C(=O)O)c2)cc1 ZINC000217621090 HG In-Stock Unstable MMP3 48 43 COc1ccc(CCNS(=O)(=O)c2ccc(NCCC(C)C)c(C(=O)O)c2)cc1 ZINC000217621090 HG In-Stock Unstable MMP8 26 40 COc1ccc(CCNS(=O)(=O)c2ccc(NCCC(C)C)c(C(=O)O)c2)cc1 ZINC000217621090 HG In-Stock Unstable ALOX15 33 40 COc1ccc(CCNS(=O)(=O)c2ccc(NCCC(C)C)c(C(=O)O)c2)cc1 ZINC000217621090 HG In-Stock Unstable MMP9 47 40 COc1ccc(CCNS(=O)(=O)c2ccc(NCCC(C)C)c(C(=O)O)c2)cc1 ZINC000217621090 HG In-Stock Unstable IAP 0 42 COc1ccc(CCNS(=O)(=O)c2ccc(NCCC(C)C)c(C(=O)O)c2)cc1 ZINC000217621090 HG In-Stock Unstable CA9 20 42 COc1ccc(CCNS(=O)(=O)c2ccc(NCCC(C)C)c(C(=O)O)c2)cc1 ZINC000217621090 HG In-Stock Unstable MMP1 49 37 COc1ccc(CCNS(=O)(=O)c2ccc(NCCC(C)C)c(C(=O)O)c2)cc1 ZINC000217621090 HG In-Stock Unstable AKR1C3 29 47 COc1ccc(CCNS(=O)(=O)c2ccc(NCCC(C)C)c(C(=O)O)c2)cc1 ZINC000217621090 HG In-Stock Unstable AKR1C2 46 36 O=C(N/C=C/c1ccccc1)Nc1cccc2c(O)cccc12 ZINC000217621109 DI For-Sale Anodyne MMP2 16 47 Cc1cc(CCC(=O)N2CCc3cnc(N4CCOCC4)nc3C2)ccc1F ZINC000217621113 GE In-Stock Unstable MAPK1 44 37 COc1ccc(S(C)(=O)=O)cc1C(C)(C)O ZINC000217621118 BD For-Sale Unstable PTGS2 21 45 COc1ccc(S(C)(=O)=O)cc1C(C)(C)O ZINC000217621118 BD For-Sale Unstable LOX1.1 17 41 NC1(C(=O)O)C[C@H]2CCC[C@@H](C2)C1 ZINC000217621133 AD In-Stock Unstable GRM1 0 44 CCOc1ccc(C)cc1S(=O)(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217621143 HG For-Sale Unstable NPY5R 24 42 CN1CCCC[C@H]1CNC[C@@H](O)c1ccc(F)c(F)c1 ZINC000217621156 CE For-Sale Unstable CHRNA10 52 44 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621207 HH In-Stock Unstable TBXA2R 44 42 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621207 HH In-Stock Unstable BMP1 73 36 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621207 HH In-Stock Unstable MMP13 53 39 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621207 HH In-Stock Unstable ALOX15B 0 40 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621207 HH In-Stock Unstable MMP3 47 40 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621207 HH In-Stock Unstable ALOX15 48 41 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621207 HH In-Stock Unstable MMP9 42 39 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621207 HH In-Stock Unstable IAP 0 41 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621207 HH In-Stock Unstable CA9 17 40 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621207 HH In-Stock Unstable MMP1 45 36 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621207 HH In-Stock Unstable AKR1C3 27 45 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621207 HH In-Stock Unstable AKR1C2 44 35 NC1(C(=O)O)C[C@@H]2CCC[C@H](C2)C1 ZINC000217621220 AD In-Stock Unstable GRM1 0 44 CC(=O)Nc1ccc(CC(=O)N2CCc3cnc(N4CCOCC4)nc3C2)cc1 ZINC000217621222 GD In-Stock Unstable PIK3CA 34 43 CC(=O)Nc1ccc(CC(=O)N2CCc3cnc(N4CCOCC4)nc3C2)cc1 ZINC000217621222 GD In-Stock Unstable MAPK1 40 34 CC(=O)Nc1ccc(CC(=O)N2CCc3cnc(N4CCOCC4)nc3C2)cc1 ZINC000217621222 GD In-Stock Unstable MTOR 77 43 CC(=O)Nc1ccc(CC(=O)N2CCc3cnc(N4CCOCC4)nc3C2)cc1 ZINC000217621222 GD In-Stock Unstable PIK3CG 36 43 CC(=O)Nc1ccc(CC(=O)N2CCc3cnc(N4CCOCC4)nc3C2)cc1 ZINC000217621222 GD In-Stock Unstable STAT6 42 31 Cc1cc(O)ccc1NC(=O)N/C=C/c1ccccc1 ZINC000217621224 CG For-Sale Unstable LPL 49 35 Cc1cc(O)ccc1NC(=O)N/C=C/c1ccccc1 ZINC000217621224 CG For-Sale Unstable MMP2 15 46 Cc1cc(O)ccc1NC(=O)N/C=C/c1ccccc1 ZINC000217621224 CG For-Sale Unstable MMP9 0 46 Cc1cc(O)ccc1NC(=O)N/C=C/c1ccccc1 ZINC000217621224 CG For-Sale Unstable MMP1 0 46 CNC(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217621238 BD On-Demand Unstable PPO2 16 40 CN1CCCC[C@@H]1CNC[C@@H](O)c1c(F)cccc1F ZINC000217621279 CE For-Sale Unstable CHRNA10 59 43 CCC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621311 HH In-Stock Unstable TBXA2R 44 42 CCC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621311 HH In-Stock Unstable BMP1 73 36 CCC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621311 HH In-Stock Unstable MMP13 53 39 CCC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621311 HH In-Stock Unstable ALOX15B 0 40 CCC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621311 HH In-Stock Unstable MMP3 47 40 CCC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621311 HH In-Stock Unstable ALOX15 48 41 CCC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621311 HH In-Stock Unstable MMP9 42 39 CCC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621311 HH In-Stock Unstable IAP 0 41 CCC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621311 HH In-Stock Unstable CA9 17 40 CCC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621311 HH In-Stock Unstable MMP1 45 36 CCC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621311 HH In-Stock Unstable AKR1C3 27 45 CCC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621311 HH In-Stock Unstable AKR1C2 44 35 O=C(N/C=C/c1ccccc1)N1CCOCC1 ZINC000217621331 BD For-Sale Unstable AKR1C3 31 45 O=C(c1ccc(-c2cccs2)cc1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217621344 HG In-Stock Unstable PIK3CA 32 43 O=C(c1ccc(-c2cccs2)cc1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217621344 HG In-Stock Unstable MTOR 43 43 O=C(c1ccc(-c2cccs2)cc1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217621344 HG In-Stock Unstable PIK3CG 28 43 CN1CCCC[C@H]1CNC[C@@H](O)c1c(F)cccc1F ZINC000217621362 CE For-Sale Unstable CHRNA10 59 43 COc1ccc([C@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c(OC)c1OC ZINC000217621376 KH In-Stock Unstable PRKDC 39 40 COc1ccc([C@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c(OC)c1OC ZINC000217621376 KH In-Stock Unstable CYP1B1 61 40 COc1ccc([C@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c(OC)c1OC ZINC000217621376 KH In-Stock Unstable CYP1A1 46 40 COc1ccc([C@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c(OC)c1OC ZINC000217621376 KH In-Stock Unstable CYP1A2 39 40 COc1ccc([C@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c(OC)c1OC ZINC000217621376 KH In-Stock Unstable RORC 46 36 COC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621426 HE In-Stock Unstable TBXA2R 45 43 COC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621426 HE In-Stock Unstable TBXAS1 15 40 COC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621426 HE In-Stock Unstable BMP1 55 36 COC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621426 HE In-Stock Unstable MMP13 49 42 COC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621426 HE In-Stock Unstable MMP8 24 42 COC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621426 HE In-Stock Unstable MMP9 40 42 COC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621426 HE In-Stock Unstable IAP 0 42 COC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621426 HE In-Stock Unstable CA9 17 41 COC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621426 HE In-Stock Unstable AKR1C3 29 46 COC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621426 HE In-Stock Unstable AKR1C2 45 35 O=C(CSc1ccncc1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217621460 FD In-Stock Unstable MAPK1 40 36 COc1ccc([C@@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c(OC)c1OC ZINC000217621462 KH In-Stock Unstable PRKDC 39 40 COc1ccc([C@@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c(OC)c1OC ZINC000217621462 KH In-Stock Unstable CYP1B1 61 40 COc1ccc([C@@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c(OC)c1OC ZINC000217621462 KH In-Stock Unstable CYP1A1 46 40 COc1ccc([C@@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c(OC)c1OC ZINC000217621462 KH In-Stock Unstable CYP1A2 39 40 COc1ccc([C@@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c(OC)c1OC ZINC000217621462 KH In-Stock Unstable RORC 46 36 O=C(O)CNC(=O)N/C=C/c1ccccc1 ZINC000217621470 BD For-Sale Unstable MME 15 48 CN1CCCC[C@@H]1CNC[C@@H](O)c1ccc2c(c1)OCO2 ZINC000217621483 CD For-Sale Unstable CHRNA10 31 47 COC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621512 HE In-Stock Unstable TBXA2R 45 43 COC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621512 HE In-Stock Unstable TBXAS1 15 40 COC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621512 HE In-Stock Unstable BMP1 55 36 COC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621512 HE In-Stock Unstable MMP13 49 42 COC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621512 HE In-Stock Unstable MMP8 24 42 COC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621512 HE In-Stock Unstable MMP9 40 42 COC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621512 HE In-Stock Unstable IAP 0 42 COC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621512 HE In-Stock Unstable CA9 17 41 COC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621512 HE In-Stock Unstable AKR1C3 29 46 COC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217621512 HE In-Stock Unstable AKR1C2 45 35 COc1ccc(-c2nnc(S[C@@H]3CCN(c4ccc(C#N)cc4)C3=O)n2Cc2ccco2)cc1 ZINC000217621559 JI On-Demand Unstable HCRTR2 15 40 CN1CCCC[C@H]1CNC[C@@H](O)c1ccc2c(c1)OCO2 ZINC000217621560 CD For-Sale Unstable CHRNA10 31 47 COc1ccc(-c2cc(C(=O)NC[C@@H]3CCCN4CCCC[C@H]34)[nH]n2)c(OC)c1 ZINC000217621572 GG In-Stock Unstable GRIN2B 0 40 COc1ccc(-c2cc(C(=O)NC[C@@H]3CCCN4CCCC[C@H]34)[nH]n2)c(OC)c1 ZINC000217621572 GG In-Stock Unstable ALPL 53 37 O=C(c1cc(-c2ccccc2)n[nH]1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217621579 GD In-Stock Unstable TACR3 18 43 O=C(c1cc(-c2ccccc2)n[nH]1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217621579 GD In-Stock Unstable HSP90AB1 0 44 O=C(O)/C=C\c1ccc(C(=O)NCC2CCCCC2)cc1 ZINC000217621603 CG For-Sale Unstable GRIN2B 17 44 O=C(O)/C=C\c1ccc(C(=O)NCC2CCCCC2)cc1 ZINC000217621603 CG For-Sale Unstable KCNQ1 0 40 O=C(O)/C=C\c1ccc(C(=O)NCC2CCCCC2)cc1 ZINC000217621603 CG For-Sale Unstable CACNA1I 63 37 CCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217621612 HF In-Stock Unstable TBXA2R 50 40 CCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217621612 HF In-Stock Unstable TBXAS1 15 43 CCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217621612 HF In-Stock Unstable IAP 0 45 CCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217621612 HF In-Stock Unstable AKR1C3 15 45 CCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217621612 HF In-Stock Unstable SCMU_MYCTU 0 44 COc1ccc(-c2nnc(S[C@H]3CCN(c4ccc(C#N)cc4)C3=O)n2Cc2ccco2)cc1 ZINC000217621640 JI On-Demand Unstable HCRTR2 15 40 CCc1ccc(OC)c(S(=O)(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217621666 HG For-Sale Unstable NPY5R 20 41 C[C@@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217621682 BD For-Sale Unstable MME 27 43 C[C@@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217621682 BD For-Sale Unstable ANPEP 26 43 C[C@@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217621682 BD For-Sale Unstable SLC15A1 0 41 O=C(c1cnn(-c2ccccc2)n1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217621692 GD In-Stock Unstable HSP90AB1 0 42 O=C(O)/C=C\c1cccc(C(=O)NCC2CCCCC2)c1 ZINC000217621698 CG For-Sale Unstable HDAC8 24 43 O=C(O)/C=C\c1cccc(C(=O)NCC2CCCCC2)c1 ZINC000217621698 CG For-Sale Unstable CACNA1I 64 43 C[C@@H]1C(=O)NN=C2COc3cc(-c4ccccc4F)c(C4CCN(C)CC4)cc3N21 ZINC000217621705 HG Annotated Unstable PRKCA 17 79 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)C)c(C(=O)O)c2)cc1OC ZINC000217621719 HF In-Stock Unstable TBXA2R 50 40 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)C)c(C(=O)O)c2)cc1OC ZINC000217621719 HF In-Stock Unstable TBXAS1 15 43 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)C)c(C(=O)O)c2)cc1OC ZINC000217621719 HF In-Stock Unstable IAP 0 45 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)C)c(C(=O)O)c2)cc1OC ZINC000217621719 HF In-Stock Unstable AKR1C3 15 45 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)C)c(C(=O)O)c2)cc1OC ZINC000217621719 HF In-Stock Unstable SCMU_MYCTU 0 42 CN(C)CCCNC(=O)c1ccc2[nH]c3ccccc3c(=O)c2c1 ZINC000217621723 DE On-Demand Unstable MAPKAPK2 17 47 CN(C)CCCNC(=O)c1ccc2[nH]c3ccccc3c(=O)c2c1 ZINC000217621723 DE On-Demand Unstable MAP2K1 15 42 CN(C)CCCNC(=O)c1ccc2[nH]c3ccccc3c(=O)c2c1 ZINC000217621723 DE On-Demand Unstable METG 21 48 CN(C)CCCNC(=O)c1ccc2[nH]c3ccccc3c(=O)c2c1 ZINC000217621723 DE On-Demand Unstable TERT 25 47 CN(C)CCCNC(=O)c1ccc2[nH]c3ccccc3c(=O)c2c1 ZINC000217621723 DE On-Demand Unstable POLR1A 20 40 CCc1ccc(OC)c(S(=O)(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217621744 HG For-Sale Unstable NPY5R 20 41 NC/C=C\CSc1ccc(O)cc1 ZINC000217621769 AD For-Sale Unstable H9TVJ1_CHISP 50 36 C[C@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217621771 BD For-Sale Unstable MME 27 43 C[C@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217621771 BD For-Sale Unstable ANPEP 26 43 C[C@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217621771 BD For-Sale Unstable SLC15A1 0 41 CC[C@@H](C)[C@@H](CO)NC(=O)CC[C@@H]1NC(=O)N(Cc2ccc3c(c2)OCO3)C1=O ZINC000217621789 HD In-Stock Unstable MCHR1 21 40 CCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217621834 IG In-Stock Unstable TBXA2R 49 39 CCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217621834 IG In-Stock Unstable TBXAS1 17 44 CCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217621834 IG In-Stock Unstable BDKRB1 0 40 CCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217621834 IG In-Stock Unstable ALOX15 46 41 CCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217621834 IG In-Stock Unstable PTGDR 25 43 CCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217621834 IG In-Stock Unstable IAP 0 46 CCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217621834 IG In-Stock Unstable PTGDR2 17 43 CCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217621834 IG In-Stock Unstable AKR1C3 15 46 CCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217621834 IG In-Stock Unstable SCMU_MYCTU 0 42 COc1ccc(CCS(=O)(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217621857 HF For-Sale Unstable NPY5R 22 43 CC(C)CCn1c(COc2ccccc2)nnc1S[C@@H]1CCN(c2ccc(C#N)cc2)C1=O ZINC000217621871 JJ On-Demand Unstable VCP 57 41 CC1(C)CN(C(=O)c2ccc(/C=C\C(=O)O)cc2)CCO1 ZINC000217621879 CE For-Sale Unstable RARA 28 40 CC1(C)CN(C(=O)c2ccc(/C=C\C(=O)O)cc2)CCO1 ZINC000217621879 CE For-Sale Unstable RARG 32 40 CC1(C)CN(C(=O)c2ccc(/C=C\C(=O)O)cc2)CCO1 ZINC000217621879 CE For-Sale Unstable RARB 28 40 O=C(O)CCCCCNC(=O)N/C=C/c1ccccc1 ZINC000217621886 CF For-Sale Unstable HDAC10 22 50 O=C(O)CCCCCNC(=O)N/C=C/c1ccccc1 ZINC000217621886 CF For-Sale Unstable HDAC1 26 50 O=C(O)CCCCCNC(=O)N/C=C/c1ccccc1 ZINC000217621886 CF For-Sale Unstable HDAC2 22 50 O=C(O)CCCCCNC(=O)N/C=C/c1ccccc1 ZINC000217621886 CF For-Sale Unstable HDAC3 23 50 O=C(O)CCCCCNC(=O)N/C=C/c1ccccc1 ZINC000217621886 CF For-Sale Unstable HDAC4 15 48 O=C(O)CCCCCNC(=O)N/C=C/c1ccccc1 ZINC000217621886 CF For-Sale Unstable HDAC5 15 50 O=C(O)CCCCCNC(=O)N/C=C/c1ccccc1 ZINC000217621886 CF For-Sale Unstable HDAC6 20 50 O=C(O)CCCCCNC(=O)N/C=C/c1ccccc1 ZINC000217621886 CF For-Sale Unstable EPHX2 26 44 O=C(O)CCCCCNC(=O)N/C=C/c1ccccc1 ZINC000217621886 CF For-Sale Unstable HDAC9 39 48 O=C(O)CCCCCNC(=O)N/C=C/c1ccccc1 ZINC000217621886 CF For-Sale Unstable HDAC11 16 50 O=C(O)CCCCCNC(=O)N/C=C/c1ccccc1 ZINC000217621886 CF For-Sale Unstable HDAC7 34 48 O=C(O)CCCCCNC(=O)N/C=C/c1ccccc1 ZINC000217621886 CF For-Sale Unstable AMP1_PLAFQ 17 42 O=C(c1ccc(-n2cccc2)cc1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217621928 GE In-Stock Unstable HSP90AB1 0 42 O=C(c1ccc(-n2cccc2)cc1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217621928 GE In-Stock Unstable SLC6A7 0 50 COc1ccc(CCS(=O)(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217621935 HF For-Sale Unstable NPY5R 22 43 CN1CCCC[C@@H]1CNC[C@@H](O)COc1ccccc1 ZINC000217621936 CD For-Sale Unstable ADRB2 71 58 CN1CCCC[C@@H]1CNC[C@@H](O)COc1ccccc1 ZINC000217621936 CD For-Sale Unstable ADRB1 91 46 CN1CCCC[C@@H]1CNC[C@@H](O)COc1ccccc1 ZINC000217621936 CD For-Sale Unstable SLC18A2 47 33 CN1CCCC[C@@H]1CNC[C@@H](O)COc1ccccc1 ZINC000217621936 CD For-Sale Unstable ADRB3 73 46 CN1CCCC[C@@H]1CNC[C@@H](O)COc1ccccc1 ZINC000217621936 CD For-Sale Unstable COLA 59 34 CN1CCCC[C@@H]1CNC[C@@H](O)COc1ccccc1 ZINC000217621936 CD For-Sale Unstable CPT1A 57 34 CN1CCCC[C@@H]1CNC[C@@H](O)COc1ccccc1 ZINC000217621936 CD For-Sale Unstable ABCB1 36 45 CN1CCCC[C@@H]1CNC[C@@H](O)COc1ccccc1 ZINC000217621936 CD For-Sale Unstable CHRNA10 82 51 CC(C)CCn1c(COc2ccccc2)nnc1S[C@H]1CCN(c2ccc(C#N)cc2)C1=O ZINC000217621950 JJ On-Demand Unstable VCP 57 41 COc1ccc(CCNS(=O)(=O)c2ccc(NCC(C)C)c(C(=O)O)c2)cc1OC ZINC000217621954 IF In-Stock Unstable TBXA2R 49 39 COc1ccc(CCNS(=O)(=O)c2ccc(NCC(C)C)c(C(=O)O)c2)cc1OC ZINC000217621954 IF In-Stock Unstable BDKRB1 0 43 COc1ccc(CCNS(=O)(=O)c2ccc(NCC(C)C)c(C(=O)O)c2)cc1OC ZINC000217621954 IF In-Stock Unstable IAP 0 44 COc1ccc(CCNS(=O)(=O)c2ccc(NCC(C)C)c(C(=O)O)c2)cc1OC ZINC000217621954 IF In-Stock Unstable SCMU_MYCTU 0 42 C=CCN1C(=O)/C(=C/c2ccc(OCc3ccc(Cl)cc3)c(OC)c2)C(=O)NC1=S ZINC000217621993 IH In-Stock Unstable ENPP2 16 50 CN1CCCC[C@H]1CNC[C@@H](O)COc1ccccc1 ZINC000217622014 CD For-Sale Unstable ADRB2 71 58 CN1CCCC[C@H]1CNC[C@@H](O)COc1ccccc1 ZINC000217622014 CD For-Sale Unstable ADRB1 91 46 CN1CCCC[C@H]1CNC[C@@H](O)COc1ccccc1 ZINC000217622014 CD For-Sale Unstable SLC18A2 47 33 CN1CCCC[C@H]1CNC[C@@H](O)COc1ccccc1 ZINC000217622014 CD For-Sale Unstable ADRB3 73 46 CN1CCCC[C@H]1CNC[C@@H](O)COc1ccccc1 ZINC000217622014 CD For-Sale Unstable COLA 59 34 CN1CCCC[C@H]1CNC[C@@H](O)COc1ccccc1 ZINC000217622014 CD For-Sale Unstable CPT1A 57 34 CN1CCCC[C@H]1CNC[C@@H](O)COc1ccccc1 ZINC000217622014 CD For-Sale Unstable ABCB1 36 45 CN1CCCC[C@H]1CNC[C@@H](O)COc1ccccc1 ZINC000217622014 CD For-Sale Unstable CHRNA10 82 51 COc1ccc(OC)c(S(=O)(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217622041 HF For-Sale Unstable NPY5R 25 48 Cc1noc(C)c1C(=O)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217622043 ED In-Stock Unstable MAPK1 30 40 CC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217622055 IG In-Stock Unstable TBXA2R 49 39 CC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217622055 IG In-Stock Unstable IAP 0 44 CC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217622055 IG In-Stock Unstable SCMU_MYCTU 0 41 Cc1nc(C(=O)N2CCC(O)(c3ccccc3Cl)CC2)ccc1NS(=O)(=O)c1cccc2cccnc12 ZINC000217622068 KJ Annotated Unstable C0L093_TOBAC 58 35 C[C@@H](O)c1cc(Br)ccc1N1CC[C@@H](N2CCCC2)C1 ZINC000217622072 EG For-Sale Unstable L3MBTL3 73 38 C[C@@H](O)c1cc(Br)ccc1N1CC[C@@H](N2CCCC2)C1 ZINC000217622072 EG For-Sale Unstable MBTD1 0 43 COc1ccc(OC)c(S(=O)(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)c1 ZINC000217622121 HF For-Sale Unstable NPY5R 25 48 CN1CCCC[C@@H]1CNC[C@@H](O)COc1ccccc1F ZINC000217622124 CD For-Sale Unstable ADRB2 40 44 CN1CCCC[C@@H]1CNC[C@@H](O)COc1ccccc1F ZINC000217622124 CD For-Sale Unstable ADRB1 53 44 CN1CCCC[C@@H]1CNC[C@@H](O)COc1ccccc1F ZINC000217622124 CD For-Sale Unstable ADRB3 31 44 CN1CCCC[C@@H]1CNC[C@@H](O)COc1ccccc1F ZINC000217622124 CD For-Sale Unstable CHRNA10 65 56 CN1CCCC[C@@H]1CNC[C@@H](O)COc1ccccc1F ZINC000217622124 CD For-Sale Unstable ACKR3 66 35 CC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217622129 IG In-Stock Unstable TBXA2R 49 39 CC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217622129 IG In-Stock Unstable IAP 0 44 CC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217622129 IG In-Stock Unstable SCMU_MYCTU 0 41 C[C@H](O)c1cc(Br)ccc1N1CC[C@@H](N2CCCC2)C1 ZINC000217622146 EG For-Sale Unstable L3MBTL3 73 38 C[C@H](O)c1cc(Br)ccc1N1CC[C@@H](N2CCCC2)C1 ZINC000217622146 EG For-Sale Unstable MBTD1 0 43 O=C(/C=C/c1ccccc1Cl)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217622157 GF In-Stock Unstable ITGAL 54 35 O=C(O)CCCNC(=O)N/C=C/c1ccccc1 ZINC000217622182 BD For-Sale Unstable HDAC9 27 41 O=C(O)CCCNC(=O)N/C=C/c1ccccc1 ZINC000217622182 BD For-Sale Unstable HDA106 0 40 CN1CCCC[C@H]1CNC[C@@H](O)COc1ccccc1F ZINC000217622199 CD For-Sale Unstable ADRB2 40 44 CN1CCCC[C@H]1CNC[C@@H](O)COc1ccccc1F ZINC000217622199 CD For-Sale Unstable ADRB1 53 44 CN1CCCC[C@H]1CNC[C@@H](O)COc1ccccc1F ZINC000217622199 CD For-Sale Unstable ADRB3 31 44 CN1CCCC[C@H]1CNC[C@@H](O)COc1ccccc1F ZINC000217622199 CD For-Sale Unstable CHRNA10 65 56 CN1CCCC[C@H]1CNC[C@@H](O)COc1ccccc1F ZINC000217622199 CD For-Sale Unstable ACKR3 66 35 COc1ccc(S(=O)(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1OC ZINC000217622221 HF For-Sale Unstable NPY5R 23 41 CC(=O)NCCNC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217622233 CC For-Sale Unstable DRD4 42 32 CC(=O)NCCNC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217622233 CC For-Sale Unstable HDAC8 30 47 CC(=O)NCCNC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217622233 CC For-Sale Unstable HDAC6 15 47 CC(=O)NCCNC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217622233 CC For-Sale Unstable TTR 0 40 CC(=O)NCCNC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217622233 CC For-Sale Unstable KCNK3 43 35 C[C@@H](O)c1ccc(Br)cc1N1CC[C@@H](N2CCCC2)C1 ZINC000217622240 EG For-Sale Unstable L3MBTL1 0 41 C[C@@H](O)c1ccc(Br)cc1N1CC[C@@H](N2CCCC2)C1 ZINC000217622240 EG For-Sale Unstable L3MBTL3 90 38 C[C@@H](O)c1ccc(Br)cc1N1CC[C@@H](N2CCCC2)C1 ZINC000217622240 EG For-Sale Unstable MBTD1 0 43 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)(C)C)c(C(=O)O)c2)cc1OC ZINC000217622263 IG In-Stock Unstable TBXA2R 50 40 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)(C)C)c(C(=O)O)c2)cc1OC ZINC000217622263 IG In-Stock Unstable TBXAS1 15 43 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)(C)C)c(C(=O)O)c2)cc1OC ZINC000217622263 IG In-Stock Unstable IAP 0 45 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)(C)C)c(C(=O)O)c2)cc1OC ZINC000217622263 IG In-Stock Unstable AKR1C3 18 48 COc1ccc(CCNS(=O)(=O)c2ccc(NC(C)(C)C)c(C(=O)O)c2)cc1OC ZINC000217622263 IG In-Stock Unstable SCMU_MYCTU 0 46 O=C(Cc1c(F)cccc1Cl)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217622265 GE In-Stock Unstable MAPK1 45 38 CSc1ncccc1C(=O)NC1CCN(C(=O)N2CCOCC2)CC1 ZINC000217622266 FD In-Stock Unstable CNR1 16 43 CSc1ncccc1C(=O)NC1CCN(C(=O)N2CCOCC2)CC1 ZINC000217622266 FD In-Stock Unstable CNR2 17 46 CSc1ncccc1C(=O)NC1CCN(C(=O)N2CCOCC2)CC1 ZINC000217622266 FD In-Stock Unstable FAAH 0 40 CSc1ncccc1C(=O)NC1CCN(C(=O)N2CCOCC2)CC1 ZINC000217622266 FD In-Stock Unstable CCR8 26 43 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622297 CE For-Sale Unstable ACE 30 49 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622297 CE For-Sale Unstable FOLH1 26 49 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622297 CE For-Sale Unstable MME 80 51 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622297 CE For-Sale Unstable ANPEP 61 49 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622297 CE For-Sale Unstable FCER2 46 37 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622297 CE For-Sale Unstable RNPEP 36 46 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622297 CE For-Sale Unstable CTSB 27 41 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622297 CE For-Sale Unstable RIR1_HHV11 41 35 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622297 CE For-Sale Unstable CTSK 31 43 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622297 CE For-Sale Unstable CTSL 18 43 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622297 CE For-Sale Unstable NAALAD2 48 47 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622297 CE For-Sale Unstable CAPNS1 59 37 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622297 CE For-Sale Unstable ECE1 17 40 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622297 CE For-Sale Unstable CAPN1 81 46 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622297 CE For-Sale Unstable CAPN2 82 37 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622297 CE For-Sale Unstable ACE2 57 40 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622297 CE For-Sale Unstable LAP3 22 46 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622297 CE For-Sale Unstable FPR1 89 48 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622297 CE For-Sale Unstable NPR 85 40 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622297 CE For-Sale Unstable AMP1_PLAFQ 31 46 COc1ccc(S(=O)(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1OC ZINC000217622313 HF For-Sale Unstable NPY5R 23 41 C[C@H](O)c1ccc(Br)cc1N1CC[C@@H](N2CCCC2)C1 ZINC000217622327 EG For-Sale Unstable L3MBTL1 0 41 C[C@H](O)c1ccc(Br)cc1N1CC[C@@H](N2CCCC2)C1 ZINC000217622327 EG For-Sale Unstable L3MBTL3 90 38 C[C@H](O)c1ccc(Br)cc1N1CC[C@@H](N2CCCC2)C1 ZINC000217622327 EG For-Sale Unstable MBTD1 0 43 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622377 CE For-Sale Unstable ACE 30 49 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622377 CE For-Sale Unstable FOLH1 26 49 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622377 CE For-Sale Unstable MME 80 51 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622377 CE For-Sale Unstable ANPEP 61 49 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622377 CE For-Sale Unstable FCER2 46 37 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622377 CE For-Sale Unstable RNPEP 36 46 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622377 CE For-Sale Unstable CTSB 27 41 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622377 CE For-Sale Unstable RIR1_HHV11 41 35 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622377 CE For-Sale Unstable CTSK 31 43 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622377 CE For-Sale Unstable CTSL 18 43 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622377 CE For-Sale Unstable NAALAD2 48 47 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622377 CE For-Sale Unstable CAPNS1 59 37 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622377 CE For-Sale Unstable ECE1 17 40 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622377 CE For-Sale Unstable CAPN1 81 46 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622377 CE For-Sale Unstable CAPN2 82 37 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622377 CE For-Sale Unstable ACE2 57 40 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622377 CE For-Sale Unstable LAP3 22 46 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622377 CE For-Sale Unstable FPR1 89 48 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622377 CE For-Sale Unstable NPR 85 40 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1)C(=O)O ZINC000217622377 CE For-Sale Unstable AMP1_PLAFQ 31 46 C=CCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217622382 HF In-Stock Unstable TBXA2R 48 38 C=CCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217622382 HF In-Stock Unstable IAP 0 45 C=CCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217622382 HF In-Stock Unstable SCMU_MYCTU 0 42 C[C@@H](O)c1cc(Br)ccc1N1CC[C@@H](N2CCCCC2)C1 ZINC000217622413 FH For-Sale Unstable L3MBTL3 47 32 C[C@@H](O)c1cc(Br)ccc1N1CC[C@@H](N2CCCCC2)C1 ZINC000217622413 FH For-Sale Unstable MBTD1 0 43 C[C@@H](NC(=O)C(F)F)c1ccccc1Cl ZINC000217622472 BF On-Demand Unstable CXCL8 47 42 C[C@@H](NC(=O)C(F)F)c1ccccc1Cl ZINC000217622472 BF On-Demand Unstable SDH1 0 41 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](CC(C)C)C(=O)Nc3cccnc3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217622476 KJ In-Stock Unstable TUBA1A 18 62 C[C@H](O)c1cc(Br)ccc1N1CC[C@@H](N2CCCCC2)C1 ZINC000217622478 FH For-Sale Unstable L3MBTL3 47 32 C[C@H](O)c1cc(Br)ccc1N1CC[C@@H](N2CCCCC2)C1 ZINC000217622478 FH For-Sale Unstable MBTD1 0 43 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CC3)c(C(=O)O)c2)cc1OC ZINC000217622489 HE In-Stock Unstable TBXA2R 50 39 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CC3)c(C(=O)O)c2)cc1OC ZINC000217622489 HE In-Stock Unstable IAP 0 48 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CC3)c(C(=O)O)c2)cc1OC ZINC000217622489 HE In-Stock Unstable SCMU_MYCTU 0 41 COc1ccc([C@@H](C)NC(=O)N/C=C/c2ccccc2)cc1OC ZINC000217622494 EH For-Sale Unstable CYP1B1 19 46 COc1ccc([C@@H](C)NC(=O)N/C=C/c2ccccc2)cc1OC ZINC000217622494 EH For-Sale Unstable CYP1A1 19 46 C[C@H](NC(=O)C(F)F)c1ccccc1Cl ZINC000217622556 BF On-Demand Unstable CXCL8 47 42 C[C@H](NC(=O)C(F)F)c1ccccc1Cl ZINC000217622556 BF On-Demand Unstable SDH1 0 41 C[C@@H](O)c1ccc(Br)cc1N1CC[C@@H](N2CCCCC2)C1 ZINC000217622559 FH For-Sale Unstable L3MBTL1 0 40 C[C@@H](O)c1ccc(Br)cc1N1CC[C@@H](N2CCCCC2)C1 ZINC000217622559 FH For-Sale Unstable L3MBTL3 72 37 C[C@@H](O)c1ccc(Br)cc1N1CC[C@@H](N2CCCCC2)C1 ZINC000217622559 FH For-Sale Unstable MBTD1 0 43 COc1ccc([C@H](C)NC(=O)N/C=C/c2ccccc2)cc1OC ZINC000217622588 EH For-Sale Unstable CYP1B1 19 46 COc1ccc([C@H](C)NC(=O)N/C=C/c2ccccc2)cc1OC ZINC000217622588 EH For-Sale Unstable CYP1A1 19 46 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc(OC)c2OC)CC(=O)O4)cc1O ZINC000217622594 JI In-Stock Unstable ALOX5 0 50 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc(OC)c2OC)CC(=O)O4)cc1O ZINC000217622594 JI In-Stock Unstable AKR1B1 0 50 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc(OC)c2OC)CC(=O)O4)cc1O ZINC000217622594 JI In-Stock Unstable CYP1B1 69 39 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc(OC)c2OC)CC(=O)O4)cc1O ZINC000217622594 JI In-Stock Unstable CYP1A1 50 46 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc(OC)c2OC)CC(=O)O4)cc1O ZINC000217622594 JI In-Stock Unstable CYP1A2 41 40 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCC3)c(C(=O)O)c2)cc1OC ZINC000217622608 IG In-Stock Unstable FKBP1A 41 42 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCC3)c(C(=O)O)c2)cc1OC ZINC000217622608 IG In-Stock Unstable ABCC8 19 44 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCC3)c(C(=O)O)c2)cc1OC ZINC000217622608 IG In-Stock Unstable TBXA2R 43 38 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCC3)c(C(=O)O)c2)cc1OC ZINC000217622608 IG In-Stock Unstable PTGDR 15 40 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCC3)c(C(=O)O)c2)cc1OC ZINC000217622608 IG In-Stock Unstable IAP 0 47 O=C(c1cccc(F)c1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217622612 ED In-Stock Unstable MAPK1 41 36 COC(=O)c1sccc1S(=O)(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217622625 HE For-Sale Unstable NPY5R 24 43 C[C@H](O)c1ccc(Br)cc1N1CC[C@@H](N2CCCCC2)C1 ZINC000217622648 FH For-Sale Unstable L3MBTL1 0 40 C[C@H](O)c1ccc(Br)cc1N1CC[C@@H](N2CCCCC2)C1 ZINC000217622648 FH For-Sale Unstable L3MBTL3 72 37 C[C@H](O)c1ccc(Br)cc1N1CC[C@@H](N2CCCCC2)C1 ZINC000217622648 FH For-Sale Unstable MBTD1 0 43 Cc1cc(/C=C\C(=O)O)ccc1NS(=O)(=O)N1CCCC1 ZINC000217622662 DD For-Sale Unstable LPL 44 35 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc(OC)c2OC)CC(=O)O4)cc1O ZINC000217622666 JI In-Stock Unstable ALOX5 0 50 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc(OC)c2OC)CC(=O)O4)cc1O ZINC000217622666 JI In-Stock Unstable AKR1B1 0 50 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc(OC)c2OC)CC(=O)O4)cc1O ZINC000217622666 JI In-Stock Unstable CYP1B1 69 39 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc(OC)c2OC)CC(=O)O4)cc1O ZINC000217622666 JI In-Stock Unstable CYP1A1 50 46 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc(OC)c2OC)CC(=O)O4)cc1O ZINC000217622666 JI In-Stock Unstable CYP1A2 41 40 C[C@@H](NC(=O)C(F)F)c1cccc(Cl)c1 ZINC000217622686 BF On-Demand Unstable CASR 0 40 CN1CCCC[C@@H]1CNC[C@@H](O)COc1ccc(Br)cc1 ZINC000217622695 FE For-Sale Unstable ADRB2 50 46 CN1CCCC[C@@H]1CNC[C@@H](O)COc1ccc(Br)cc1 ZINC000217622695 FE For-Sale Unstable ADRB1 63 46 CN1CCCC[C@@H]1CNC[C@@H](O)COc1ccc(Br)cc1 ZINC000217622695 FE For-Sale Unstable ADRB3 44 42 CN1CCCC[C@@H]1CNC[C@@H](O)COc1ccc(Br)cc1 ZINC000217622695 FE For-Sale Unstable CHRNA10 65 40 COc1ccc([C@@H](C)NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217622703 CH For-Sale Unstable ACACA 24 47 COc1ccc([C@@H](C)NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217622703 CH For-Sale Unstable ACACB 28 44 COc1ccc([C@@H](C)NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217622703 CH For-Sale Unstable MMP2 19 47 COc1ccc([C@@H](C)NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217622703 CH For-Sale Unstable MMP9 19 47 COC(=O)c1sccc1S(=O)(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217622710 HE For-Sale Unstable NPY5R 24 43 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCCC3)c(C(=O)O)c2)cc1OC ZINC000217622727 JH In-Stock Unstable FKBP1A 40 42 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCCC3)c(C(=O)O)c2)cc1OC ZINC000217622727 JH In-Stock Unstable ABCC8 20 46 COc1ccc(CCNS(=O)(=O)c2ccc(NC3CCCCC3)c(C(=O)O)c2)cc1OC ZINC000217622727 JH In-Stock Unstable IAP 0 46 CC(C)n1ncc2c(C(=O)Nc3ccc(CN4CCOCC4)cc3)cc(-c3cccs3)nc21 ZINC000217622740 JJ On-Demand Unstable PIK3CA 19 40 C[C@H](NC(=O)C(F)F)c1cccc(Cl)c1 ZINC000217622766 BF On-Demand Unstable CASR 0 40 COc1ccc([C@H](C)NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217622777 CH For-Sale Unstable ACACA 24 47 COc1ccc([C@H](C)NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217622777 CH For-Sale Unstable ACACB 28 44 COc1ccc([C@H](C)NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217622777 CH For-Sale Unstable MMP2 19 47 COc1ccc([C@H](C)NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217622777 CH For-Sale Unstable MMP9 19 47 CN1CCCC[C@H]1CNC[C@@H](O)COc1ccc(Br)cc1 ZINC000217622784 FE For-Sale Unstable ADRB2 50 46 CN1CCCC[C@H]1CNC[C@@H](O)COc1ccc(Br)cc1 ZINC000217622784 FE For-Sale Unstable ADRB1 63 46 CN1CCCC[C@H]1CNC[C@@H](O)COc1ccc(Br)cc1 ZINC000217622784 FE For-Sale Unstable ADRB3 44 42 CN1CCCC[C@H]1CNC[C@@H](O)COc1ccc(Br)cc1 ZINC000217622784 FE For-Sale Unstable CHRNA10 65 40 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)Nc3nc4c(s3)CCC4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217622787 KH In-Stock Unstable TUBA1A 17 62 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)Nc3nc4c(s3)CCC4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217622787 KH In-Stock Unstable TPPP 0 58 COc1ncccc1C(=O)N1CCC2(CC1)CN(C)C(=O)CO2 ZINC000217622799 DC In-Stock Unstable ACACA 33 42 COc1ccc(CCNS(=O)(=O)c2ccc(NCCC3=CCCCC3)c(C(=O)O)c2)cc1OC ZINC000217622819 JI In-Stock Unstable TBXA2R 43 39 COc1ccc(CCNS(=O)(=O)c2ccc(NCCC3=CCCCC3)c(C(=O)O)c2)cc1OC ZINC000217622819 JI In-Stock Unstable IAP 0 42 COc1ccc(CCNS(=O)(=O)c2ccc(NCCC3=CCCCC3)c(C(=O)O)c2)cc1OC ZINC000217622819 JI In-Stock Unstable SCMU_MYCTU 0 41 O=C(NCC(=O)N1CCc2cnc(N3CCOCC3)nc2C1)c1ccccc1 ZINC000217622827 GC In-Stock Unstable MAPK1 41 35 O=C(NCC(=O)N1CCc2cnc(N3CCOCC3)nc2C1)c1ccccc1 ZINC000217622827 GC In-Stock Unstable MTOR 44 40 COc1ccc(Cl)cc1S(=O)(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217622834 HG For-Sale Unstable CPT1A 68 39 COc1ccc(Cl)cc1S(=O)(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217622834 HG For-Sale Unstable CPT2 47 37 COc1ccc(Cl)cc1S(=O)(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217622834 HG For-Sale Unstable NPY5R 23 43 COc1ccc(Cl)cc1S(=O)(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217622834 HG For-Sale Unstable CPT1B 58 37 O=C1C[C@@H](c2ccc3c(c2)OCCO3)c2c(ccc3c(=O)c(-c4ccc(O)cc4)coc23)O1 ZINC000217622903 II In-Stock Unstable ALDH2 94 39 CCOC(=O)N1CCN(C(=O)C(F)F)CC1 ZINC000217622923 BC On-Demand Unstable P2RY12 43 36 CCOC(=O)N1CCN(C(=O)C(F)F)CC1 ZINC000217622923 BC On-Demand Unstable CHRNA3 20 40 CN1CCCC[C@@H]1CNC[C@@H](O)COc1cccc(Br)c1 ZINC000217622924 FE For-Sale Unstable ADRB2 38 44 CN1CCCC[C@@H]1CNC[C@@H](O)COc1cccc(Br)c1 ZINC000217622924 FE For-Sale Unstable ADRB1 45 43 CN1CCCC[C@@H]1CNC[C@@H](O)COc1cccc(Br)c1 ZINC000217622924 FE For-Sale Unstable CHRNA10 70 41 COc1ccc(Cl)cc1S(=O)(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217622932 HG For-Sale Unstable CPT1A 68 39 COc1ccc(Cl)cc1S(=O)(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217622932 HG For-Sale Unstable CPT2 47 37 COc1ccc(Cl)cc1S(=O)(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217622932 HG For-Sale Unstable NPY5R 23 43 COc1ccc(Cl)cc1S(=O)(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217622932 HG For-Sale Unstable CPT1B 58 37 COc1ccc(CCNS(=O)(=O)c2ccc(NCCO)c(C(=O)O)c2)cc1OC ZINC000217622941 HD In-Stock Unstable TBXA2R 50 40 COc1ccc(CCNS(=O)(=O)c2ccc(NCCO)c(C(=O)O)c2)cc1OC ZINC000217622941 HD In-Stock Unstable TBXAS1 15 43 COc1ccc(CCNS(=O)(=O)c2ccc(NCCO)c(C(=O)O)c2)cc1OC ZINC000217622941 HD In-Stock Unstable IAP 0 45 COc1ccc(CCNS(=O)(=O)c2ccc(NCCO)c(C(=O)O)c2)cc1OC ZINC000217622941 HD In-Stock Unstable AKR1C3 15 45 COc1ccc(CCNS(=O)(=O)c2ccc(NCCO)c(C(=O)O)c2)cc1OC ZINC000217622941 HD In-Stock Unstable SCMU_MYCTU 0 44 O=C(c1ccc(Cl)cc1Cl)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217622942 GF In-Stock Unstable P2RX7 16 44 O=C(c1ccc(Cl)cc1Cl)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217622942 GF In-Stock Unstable MAPK1 46 40 O=C(c1ccc(Cl)cc1Cl)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217622942 GF In-Stock Unstable AKR1C3 0 42 O=C1C[C@H](c2ccc3c(c2)OCCO3)c2c(ccc3c(=O)c(-c4ccc(O)cc4)coc23)O1 ZINC000217622986 II In-Stock Unstable ALDH2 94 39 CN1CCCC[C@H]1CNC[C@@H](O)COc1cccc(Br)c1 ZINC000217623001 FE For-Sale Unstable ADRB2 38 44 CN1CCCC[C@H]1CNC[C@@H](O)COc1cccc(Br)c1 ZINC000217623001 FE For-Sale Unstable ADRB1 45 43 CN1CCCC[C@H]1CNC[C@@H](O)COc1cccc(Br)c1 ZINC000217623001 FE For-Sale Unstable CHRNA10 70 41 CSC[C@@](C)(O)CNC(=O)c1cnc2cc(C)nn2c1C ZINC000217623018 DD On-Demand Unstable DPP8 16 51 CSC[C@@](C)(O)CNC(=O)c1cnc2cc(C)nn2c1C ZINC000217623018 DD On-Demand Unstable DPP9 27 51 O=C(Nc1ccnn1Cc1cccc(Cl)c1Cl)c1ccc(N2CCNC2=O)cc1 ZINC000217623028 II On-Demand Unstable MRGPRX1 44 39 O=C1O[C@@]2(CCCN(S(=O)(=O)c3ccc(C(F)(F)F)cc3)C2)c2ccccc21 ZINC000217623042 HH For-Sale Unstable NPY5R 22 44 COc1ccc(CCNS(=O)(=O)c2ccc(NCCCO)c(C(=O)O)c2)cc1OC ZINC000217623053 ID In-Stock Unstable TBXA2R 49 39 COc1ccc(CCNS(=O)(=O)c2ccc(NCCCO)c(C(=O)O)c2)cc1OC ZINC000217623053 ID In-Stock Unstable TBXAS1 17 44 COc1ccc(CCNS(=O)(=O)c2ccc(NCCCO)c(C(=O)O)c2)cc1OC ZINC000217623053 ID In-Stock Unstable IAP 0 46 COc1ccc(CCNS(=O)(=O)c2ccc(NCCCO)c(C(=O)O)c2)cc1OC ZINC000217623053 ID In-Stock Unstable AKR1C3 16 46 COc1ccc(CCNS(=O)(=O)c2ccc(NCCCO)c(C(=O)O)c2)cc1OC ZINC000217623053 ID In-Stock Unstable SCMU_MYCTU 0 42 O=C(C(F)F)N1CCN(c2ccc(F)cc2)CC1 ZINC000217623093 CD On-Demand Unstable AKR1C3 26 59 COc1ccc2cc([C@@H]3CC(=O)Oc4ccc5c(c43)OC(=C(C)C)C5=O)c(=O)[nH]c2c1 ZINC000217623094 HH In-Stock Unstable MT-ND4 40 32 C[C@@H](CNCc1cncn1C1CC1)N(C)C1CC1 ZINC000217623097 BD For-Sale Unstable CAMC 0 44 CSC[C@](C)(O)CNC(=O)c1cnc2cc(C)nn2c1C ZINC000217623113 DD On-Demand Unstable DPP8 16 51 CSC[C@](C)(O)CNC(=O)c1cnc2cc(C)nn2c1C ZINC000217623113 DD On-Demand Unstable DPP9 27 51 O=C1O[C@]2(CCCN(S(=O)(=O)c3ccc(C(F)(F)F)cc3)C2)c2ccccc21 ZINC000217623123 HH For-Sale Unstable NPY5R 22 44 CN1CCCC[C@@H]1CNC[C@@H](O)COCc1ccccc1 ZINC000217623138 CD For-Sale Unstable ADRB2 17 44 CN1CCCC[C@@H]1CNC[C@@H](O)COCc1ccccc1 ZINC000217623138 CD For-Sale Unstable SLC18A2 54 35 CN1CCCC[C@@H]1CNC[C@@H](O)COCc1ccccc1 ZINC000217623138 CD For-Sale Unstable CHRNA10 52 40 COCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217623160 ID In-Stock Unstable TBXA2R 50 39 COCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217623160 ID In-Stock Unstable IAP 0 45 COCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217623160 ID In-Stock Unstable SCMU_MYCTU 0 43 CC(C)C(=O)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217623166 CC In-Stock Unstable MAPK1 43 39 COc1ccc2cc([C@H]3CC(=O)Oc4ccc5c(c43)OC(=C(C)C)C5=O)c(=O)[nH]c2c1 ZINC000217623176 HH In-Stock Unstable MT-ND4 40 32 C[C@H](CNCc1cncn1C1CC1)N(C)C1CC1 ZINC000217623185 BD For-Sale Unstable CAMC 0 44 CN1CCCC[C@H]1CNC[C@@H](O)COCc1ccccc1 ZINC000217623215 CD For-Sale Unstable ADRB2 17 44 CN1CCCC[C@H]1CNC[C@@H](O)COCc1ccccc1 ZINC000217623215 CD For-Sale Unstable SLC18A2 54 35 CN1CCCC[C@H]1CNC[C@@H](O)COCc1ccccc1 ZINC000217623215 CD For-Sale Unstable CHRNA10 52 40 O=C(C(F)F)N1CCc2ccccc21 ZINC000217623217 AD On-Demand Unstable AVPR2 29 42 O=C1O[C@@]2(CCCN(S(=O)(=O)c3cccc(C(F)(F)F)c3)C2)c2ccccc21 ZINC000217623252 HH For-Sale Unstable CACNA1B 33 41 O=C1O[C@@]2(CCCN(S(=O)(=O)c3cccc(C(F)(F)F)c3)C2)c2ccccc21 ZINC000217623252 HH For-Sale Unstable NPY5R 21 44 O=C1O[C@@]2(CCCN(S(=O)(=O)c3cccc(C(F)(F)F)c3)C2)c2ccccc21 ZINC000217623252 HH For-Sale Unstable PKM 17 48 COCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217623258 JE In-Stock Unstable TBXA2R 48 38 CCc1ccc([C@@H](C)NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217623271 CI For-Sale Unstable ACACA 19 42 CCc1ccc([C@@H](C)NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217623271 CI For-Sale Unstable ACACB 16 42 CCc1ccc([C@@H](C)NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217623271 CI For-Sale Unstable ACE2 41 33 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCCc1ccccc1 ZINC000217623282 IH In-Stock Unstable TOP1 0 44 COc1ccc(S(N)(=O)=O)cc1C(=O)N1CCC[C@@H]1c1ccccn1 ZINC000217623303 FD In-Stock Unstable CA7 19 48 O=C1O[C@]2(CCCN(S(=O)(=O)c3cccc(C(F)(F)F)c3)C2)c2ccccc21 ZINC000217623338 HH For-Sale Unstable CACNA1B 33 41 O=C1O[C@]2(CCCN(S(=O)(=O)c3cccc(C(F)(F)F)c3)C2)c2ccccc21 ZINC000217623338 HH For-Sale Unstable NPY5R 21 44 O=C1O[C@]2(CCCN(S(=O)(=O)c3cccc(C(F)(F)F)c3)C2)c2ccccc21 ZINC000217623338 HH For-Sale Unstable PKM 17 48 COc1ccc(CCNC(=O)C(F)F)cc1 ZINC000217623339 BD On-Demand Unstable CA2 15 44 COc1ccc(CCNC(=O)C(F)F)cc1 ZINC000217623339 BD On-Demand Unstable ADRB2 17 45 COc1ccc(CCNC(=O)C(F)F)cc1 ZINC000217623339 BD On-Demand Unstable ADRB1 17 40 COc1ccc(CCNC(=O)C(F)F)cc1 ZINC000217623339 BD On-Demand Unstable PTGS2 0 40 COc1ccc(CCNC(=O)C(F)F)cc1 ZINC000217623339 BD On-Demand Unstable SLC18A2 26 41 COc1ccc(CCNC(=O)C(F)F)cc1 ZINC000217623339 BD On-Demand Unstable ADRB3 24 44 COc1ccc(CCNC(=O)C(F)F)cc1 ZINC000217623339 BD On-Demand Unstable ANPEP 16 44 COc1ccc(CCNC(=O)C(F)F)cc1 ZINC000217623339 BD On-Demand Unstable BMP1 66 38 COc1ccc(CCNC(=O)C(F)F)cc1 ZINC000217623339 BD On-Demand Unstable NQO2 34 48 COc1ccc(CCNC(=O)C(F)F)cc1 ZINC000217623339 BD On-Demand Unstable TRPV1 0 48 COc1ccc(CCNC(=O)C(F)F)cc1 ZINC000217623339 BD On-Demand Unstable MMP13 26 43 COc1ccc(CCNC(=O)C(F)F)cc1 ZINC000217623339 BD On-Demand Unstable CTSL 24 42 COc1ccc(CCNC(=O)C(F)F)cc1 ZINC000217623339 BD On-Demand Unstable ADAM17 0 42 COc1ccc(CCNC(=O)C(F)F)cc1 ZINC000217623339 BD On-Demand Unstable MMP16 0 44 COc1ccc(CCNC(=O)C(F)F)cc1 ZINC000217623339 BD On-Demand Unstable MTNR1A 87 48 COc1ccc(CCNC(=O)C(F)F)cc1 ZINC000217623339 BD On-Demand Unstable MTNR1B 65 41 COc1ccc(CCNC(=O)C(F)F)cc1 ZINC000217623339 BD On-Demand Unstable MMP2 22 44 COc1ccc(CCNC(=O)C(F)F)cc1 ZINC000217623339 BD On-Demand Unstable MMP8 23 44 COc1ccc(CCNC(=O)C(F)F)cc1 ZINC000217623339 BD On-Demand Unstable MMP12 27 43 COc1ccc(CCNC(=O)C(F)F)cc1 ZINC000217623339 BD On-Demand Unstable CA12 15 53 COc1ccc(CCNC(=O)C(F)F)cc1 ZINC000217623339 BD On-Demand Unstable PTGDR 31 43 COc1ccc(CCNC(=O)C(F)F)cc1 ZINC000217623339 BD On-Demand Unstable CA9 26 53 COc1ccc(CCNC(=O)C(F)F)cc1 ZINC000217623339 BD On-Demand Unstable MMP1 37 44 COc1ccc(CCNC(=O)C(F)F)cc1 ZINC000217623339 BD On-Demand Unstable AMP1_PLAFQ 23 40 COc1ccc(CCNC(=O)C(F)F)cc1 ZINC000217623339 BD On-Demand Unstable LEF 54 39 COc1ccc(CCNC(=O)C(F)F)cc1 ZINC000217623339 BD On-Demand Unstable NCE103 21 40 COc1ccc(CCNC(=O)C(F)F)cc1 ZINC000217623339 BD On-Demand Unstable PROKR1 54 35 COc1ccc(CCNC(=O)C(F)F)cc1 ZINC000217623339 BD On-Demand Unstable CAN2 0 40 CCc1ccc([C@H](C)NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217623351 CI For-Sale Unstable ACACA 19 42 CCc1ccc([C@H](C)NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217623351 CI For-Sale Unstable ACACB 16 42 CCc1ccc([C@H](C)NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217623351 CI For-Sale Unstable ACE2 41 33 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccccc3)c(C(=O)O)c2)cc1OC ZINC000217623370 JH In-Stock Unstable TBXA2R 52 42 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccccc3)c(C(=O)O)c2)cc1OC ZINC000217623370 JH In-Stock Unstable TBXAS1 25 44 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccccc3)c(C(=O)O)c2)cc1OC ZINC000217623370 JH In-Stock Unstable BDKRB1 0 42 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccccc3)c(C(=O)O)c2)cc1OC ZINC000217623370 JH In-Stock Unstable PTGDR 15 40 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccccc3)c(C(=O)O)c2)cc1OC ZINC000217623370 JH In-Stock Unstable IAP 0 44 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccccc3)c(C(=O)O)c2)cc1OC ZINC000217623370 JH In-Stock Unstable AKR1C3 17 48 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccccc3)c(C(=O)O)c2)cc1OC ZINC000217623370 JH In-Stock Unstable SCMU_MYCTU 0 42 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCCc1ccccc1 ZINC000217623376 IH In-Stock Unstable TOP1 0 44 COc1ccc(S(N)(=O)=O)cc1C(=O)N1CCC[C@H]1c1ccccn1 ZINC000217623390 FD In-Stock Unstable CA7 19 48 COC[C@H](C)NC(=O)c1cc(/C=C\C(=O)O)ccc1F ZINC000217623407 CD For-Sale Unstable AKR1C3 40 39 O=C1O[C@@]2(CCCN(S(=O)(=O)c3cc(Cl)ccc3Cl)C2)c2ccccc21 ZINC000217623449 HH For-Sale Unstable NPY5R 26 46 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable ACE 64 39 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable FOLH1 17 41 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable MME 91 44 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable LTA4H 16 42 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable ANPEP 91 38 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable SDH1 0 59 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable CASP3 23 41 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable KLK3 57 36 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable CTSB 53 38 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable PAPA1_CARPA 53 35 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable CYSP_TRYCR 64 36 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable CTSG 22 43 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable CTSK 34 42 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable CTSL 46 38 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable CPA1 42 38 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable SLC15A1 0 43 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable ACACB 15 43 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable CTRB1 33 43 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable CAPNS1 56 34 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable MMP2 33 43 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable MMP3 68 42 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable MMP8 25 44 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable MMP14 15 40 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable CELA2A 26 43 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable PAM 0 42 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable CTSS 20 44 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable CAPN1 80 43 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable MMP9 20 40 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable CAPN2 92 38 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable ACE2 65 38 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable MMP12 16 41 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable LAP3 55 41 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable CTSC 19 43 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable MMP1 31 42 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable FPR1 46 38 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable POL 0 48 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable NPR 66 36 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable AMP1_PLAFQ 63 43 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable HDA106 0 40 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable SLC15A2 0 41 C[C@@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623454 BE On-Demand Unstable POLG_WNV 45 32 COC[C@@H](C)NC(=O)c1cc(/C=C\C(=O)O)ccc1F ZINC000217623492 CD For-Sale Unstable SDH1 0 40 COC[C@@H](C)NC(=O)c1cc(/C=C\C(=O)O)ccc1F ZINC000217623492 CD For-Sale Unstable AKR1C3 40 39 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@@H](C)c3ccccc3)c(C(=O)O)c2)cc1OC ZINC000217623494 JI In-Stock Unstable ADRB3 45 37 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@@H](C)c3ccccc3)c(C(=O)O)c2)cc1OC ZINC000217623494 JI In-Stock Unstable TBXA2R 39 41 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@@H](C)c3ccccc3)c(C(=O)O)c2)cc1OC ZINC000217623494 JI In-Stock Unstable TBXAS1 15 42 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@@H](C)c3ccccc3)c(C(=O)O)c2)cc1OC ZINC000217623494 JI In-Stock Unstable BDKRB1 0 42 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@@H](C)c3ccccc3)c(C(=O)O)c2)cc1OC ZINC000217623494 JI In-Stock Unstable IAP 0 43 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@@H](C)c3ccccc3)c(C(=O)O)c2)cc1OC ZINC000217623494 JI In-Stock Unstable AKR1C3 15 44 COc1cc(OC)cc(OC/C=C\CN)c1 ZINC000217623528 BD For-Sale Unstable CYP1A1 18 40 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable ACE 64 39 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable FOLH1 17 41 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable MME 91 44 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable LTA4H 16 42 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable ANPEP 91 38 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable SDH1 0 59 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable CASP3 23 41 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable KLK3 57 36 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable CTSB 53 38 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable PAPA1_CARPA 53 35 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable CYSP_TRYCR 64 36 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable CTSG 22 43 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable CTSK 34 42 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable CTSL 46 38 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable CPA1 42 38 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable SLC15A1 0 43 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable ACACB 15 43 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable CTRB1 33 43 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable CAPNS1 56 34 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable MMP2 33 43 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable MMP3 68 42 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable MMP8 25 44 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable MMP14 15 40 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable CELA2A 26 43 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable PAM 0 42 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable CTSS 20 44 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable CAPN1 80 43 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable MMP9 20 40 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable CAPN2 92 38 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable ACE2 65 38 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable MMP12 16 41 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable LAP3 55 41 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable CTSC 19 43 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable MMP1 31 42 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable FPR1 46 38 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable POL 0 48 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable NPR 66 36 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable AMP1_PLAFQ 63 43 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable HDA106 0 40 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable SLC15A2 0 41 C[C@H](CCc1ccccc1)NC(=O)C(F)F ZINC000217623529 BE On-Demand Unstable POLG_WNV 45 32 C[C@H](O)c1cc(Br)ccc1N1CCN(C)[C@@H](C)C1 ZINC000217623537 DF For-Sale Unstable SORD 51 35 O=C1O[C@]2(CCCN(S(=O)(=O)c3cc(Cl)ccc3Cl)C2)c2ccccc21 ZINC000217623538 HH For-Sale Unstable NPY5R 26 46 Cc1cc(NC(=O)c2nn(-c3ccccc3)c3c2CCC3)n(-c2ccc(F)cc2)n1 ZINC000217623556 HI On-Demand Unstable GRM5 15 50 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@H](C)c3ccccc3)c(C(=O)O)c2)cc1OC ZINC000217623574 JI In-Stock Unstable ADRB3 45 37 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@H](C)c3ccccc3)c(C(=O)O)c2)cc1OC ZINC000217623574 JI In-Stock Unstable TBXA2R 39 41 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@H](C)c3ccccc3)c(C(=O)O)c2)cc1OC ZINC000217623574 JI In-Stock Unstable TBXAS1 15 42 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@H](C)c3ccccc3)c(C(=O)O)c2)cc1OC ZINC000217623574 JI In-Stock Unstable BDKRB1 0 42 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@H](C)c3ccccc3)c(C(=O)O)c2)cc1OC ZINC000217623574 JI In-Stock Unstable IAP 0 43 COc1ccc(CCNS(=O)(=O)c2ccc(N[C@H](C)c3ccccc3)c(C(=O)O)c2)cc1OC ZINC000217623574 JI In-Stock Unstable AKR1C3 15 44 C[C@H](O)c1ccc(Br)cc1N1CCN(C)[C@@H](C)C1 ZINC000217623618 DF For-Sale Unstable SORD 51 35 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1OC ZINC000217623651 JH In-Stock Unstable CA2 15 41 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1OC ZINC000217623651 JH In-Stock Unstable TBXA2R 53 45 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1OC ZINC000217623651 JH In-Stock Unstable TBXAS1 28 48 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1OC ZINC000217623651 JH In-Stock Unstable CA1 15 48 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1OC ZINC000217623651 JH In-Stock Unstable CA7 17 45 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1OC ZINC000217623651 JH In-Stock Unstable BDKRB1 0 42 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1OC ZINC000217623651 JH In-Stock Unstable CA14 15 48 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1OC ZINC000217623651 JH In-Stock Unstable ALOX15 46 38 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1OC ZINC000217623651 JH In-Stock Unstable PTGDR 20 41 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1OC ZINC000217623651 JH In-Stock Unstable IAP 0 47 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1OC ZINC000217623651 JH In-Stock Unstable AKR1C3 18 49 COc1ccc(CCNS(=O)(=O)c2ccc(NCCc3ccccc3)c(C(=O)O)c2)cc1OC ZINC000217623651 JH In-Stock Unstable SCMU_MYCTU 0 45 COC[C@@H](C)NC(=O)c1ccc(/C=C\C(=O)O)cc1F ZINC000217623654 CD For-Sale Unstable SDH1 0 40 O=C(Nc1nc(-c2ccc3c(c2)CCO3)cs1)c1ccc(N2CCNC2=O)cc1 ZINC000217623662 HH On-Demand Unstable MPL 49 42 CCc1cccc(CC)c1NC(=O)N/C=C/c1ccccc1 ZINC000217623680 CJ For-Sale Unstable ACAT 0 47 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)c(OC)c3)cc2C(=O)O)cc1 ZINC000217623725 KH In-Stock Unstable TBXA2R 51 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)c(OC)c3)cc2C(=O)O)cc1 ZINC000217623725 KH In-Stock Unstable TBXAS1 19 46 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)c(OC)c3)cc2C(=O)O)cc1 ZINC000217623725 KH In-Stock Unstable PTGDR 35 40 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)c(OC)c3)cc2C(=O)O)cc1 ZINC000217623725 KH In-Stock Unstable IAP 0 46 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)c(OC)c3)cc2C(=O)O)cc1 ZINC000217623725 KH In-Stock Unstable CA9 22 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)c(OC)c3)cc2C(=O)O)cc1 ZINC000217623725 KH In-Stock Unstable AKR1C3 28 48 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)c(OC)c3)cc2C(=O)O)cc1 ZINC000217623725 KH In-Stock Unstable AKR1C2 46 38 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)c(OC)c3)cc2C(=O)O)cc1 ZINC000217623725 KH In-Stock Unstable SCMU_MYCTU 0 44 CCOc1ccc(C(=O)N2CCC(NC(=O)c3nn(-c4ccccc4)c4c3CCC4)CC2)cc1 ZINC000217623781 JH On-Demand Unstable AVPR1A 23 45 CCOc1ccc(C(=O)N2CCC(NC(=O)c3nn(-c4ccccc4)c4c3CCC4)CC2)cc1 ZINC000217623781 JH On-Demand Unstable SSTR5 50 40 CCOc1ccc(C(=O)N2CCC(NC(=O)c3nn(-c4ccccc4)c4c3CCC4)CC2)cc1 ZINC000217623781 JH On-Demand Unstable L3MBTL3 47 33 O=C(N/C=C/c1ccccc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217623790 EK For-Sale Anodyne LTA4H 42 43 O=C(N/C=C/c1ccccc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217623790 EK For-Sale Anodyne CA1 49 52 O=C(N/C=C/c1ccccc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217623790 EK For-Sale Anodyne RAF1 24 44 O=C(N/C=C/c1ccccc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217623790 EK For-Sale Anodyne MMP2 16 49 O=C(N/C=C/c1ccccc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217623790 EK For-Sale Anodyne NPY5R 26 40 O=C(N/C=C/c1ccccc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217623790 EK For-Sale Anodyne CA12 23 52 O=C(N/C=C/c1ccccc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217623790 EK For-Sale Anodyne CA9 24 52 O=C(N/C=C/c1ccccc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217623790 EK For-Sale Anodyne Q8MMZ8_EIMTE 40 44 O=C(N/C=C/c1ccccc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217623790 EK For-Sale Anodyne F13A1 22 44 O=C(N/C=C/c1ccccc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217623790 EK For-Sale Anodyne NCE103 19 42 O=C(N/C=C/c1ccccc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217623790 EK For-Sale Anodyne P96878_MYCTU 15 52 O=C(N/C=C/c1ccccc1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217623790 EK For-Sale Anodyne P95276_MYCTO 0 42 NC(=O)[C@H]1CCCN(C(=O)c2ccc(/C=C\C(=O)O)s2)C1 ZINC000217623811 DD For-Sale Unstable L3MBTL1 0 40 O=C(c1ccoc1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217623836 DD In-Stock Unstable HSP90AB1 0 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)c(OC)c3)cc2C(=O)O)cc1OC ZINC000217623838 KH In-Stock Unstable TBXA2R 53 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)c(OC)c3)cc2C(=O)O)cc1OC ZINC000217623838 KH In-Stock Unstable TBXAS1 21 47 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)c(OC)c3)cc2C(=O)O)cc1OC ZINC000217623838 KH In-Stock Unstable BDKRB1 0 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)c(OC)c3)cc2C(=O)O)cc1OC ZINC000217623838 KH In-Stock Unstable PTGDR 20 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)c(OC)c3)cc2C(=O)O)cc1OC ZINC000217623838 KH In-Stock Unstable IAP 0 49 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)c(OC)c3)cc2C(=O)O)cc1OC ZINC000217623838 KH In-Stock Unstable AKR1C3 19 48 COc1ccc(CCNc2ccc(S(=O)(=O)NCCc3ccc(OC)c(OC)c3)cc2C(=O)O)cc1OC ZINC000217623838 KH In-Stock Unstable SCMU_MYCTU 0 48 CCCOc1ccc(S(=O)(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1C ZINC000217623851 HH For-Sale Unstable PDE5A 35 40 Cc1ccc(Cl)cc1NC(=O)N/C=C/c1ccccc1 ZINC000217623889 CI For-Sale Unstable LPL 41 32 Cc1ccc(Cl)cc1NC(=O)N/C=C/c1ccccc1 ZINC000217623889 CI For-Sale Unstable CMA1 22 44 NC(=O)[C@@H]1CCCN(C(=O)c2ccc(/C=C\C(=O)O)s2)C1 ZINC000217623891 DD For-Sale Unstable L3MBTL1 0 40 Cc1c(N[C@H]2C[C@H](C)CC[C@H]2C(C)C)cccc1C(N)=O ZINC000217623893 CH For-Sale Unstable TRPM8 17 46 CC(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217623918 BE On-Demand Unstable CCR3 21 41 CC(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217623918 BE On-Demand Unstable GUAB 0 40 CC(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217623918 BE On-Demand Unstable TAAR1 29 42 CC(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217623918 BE On-Demand Unstable AKR1C3 35 56 CC(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217623918 BE On-Demand Unstable IMDH_CRYPV 55 40 CC(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217623918 BE On-Demand Unstable GRB7 0 40 CC(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217623918 BE On-Demand Unstable PARP14 0 40 CC(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217623918 BE On-Demand Unstable PARP15 0 43 CC(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217623918 BE On-Demand Unstable PSBA 0 43 CC(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217623918 BE On-Demand Unstable KCNK3 125 45 CC(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217623918 BE On-Demand Unstable KCNK9 85 44 CC(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217623918 BE On-Demand Unstable PARP10 0 46 COc1ccc2cc(C(=O)N3CCc4cnc(N5CCOCC5)nc4C3)[nH]c2c1 ZINC000217623936 GE In-Stock Unstable HSP90AB1 0 50 CCCOc1ccc(S(=O)(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1C ZINC000217623940 HH For-Sale Unstable PDE5A 35 40 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccco3)c(C(=O)O)c2)cc1OC ZINC000217623952 JG In-Stock Unstable TBXA2R 44 39 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccco3)c(C(=O)O)c2)cc1OC ZINC000217623952 JG In-Stock Unstable IAP 0 43 COc1ccc(CCNS(=O)(=O)c2ccc(NCc3ccco3)c(C(=O)O)c2)cc1OC ZINC000217623952 JG In-Stock Unstable SCMU_MYCTU 0 41 Cc1c(N[C@H]2C[C@@H](C)CC[C@H]2C(C)C)cccc1C(N)=O ZINC000217623982 CH For-Sale Unstable TRPM8 17 46 COc1ccc(OC)c(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217624007 CG For-Sale Unstable CYP1B1 69 47 COc1ccc(OC)c(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217624007 CG For-Sale Unstable MTNR1A 34 48 COc1ccc(OC)c(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217624007 CG For-Sale Unstable MTNR1B 38 48 COc1ccc(OC)c(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217624007 CG For-Sale Unstable CYP1A1 43 47 COc1ccc(OC)c(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217624007 CG For-Sale Unstable AKR1C3 23 40 COc1ccc(OC)c(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217624007 CG For-Sale Unstable ABCG2 22 41 COc1ccc(OC)c(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217624007 CG For-Sale Unstable AKR1C2 54 38 C=C(C)Cn1nc(C)c(CCC(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)c1C ZINC000217624014 GF In-Stock Unstable CHRNA4 36 48 CC[C@@H]1CCCN(c2ccccc2CBr)CC1 ZINC000217624016 CJ For-Sale Unstable KCNQ2 47 33 O=C(Nc1ccccc1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217624042 ED In-Stock Unstable PIK3CA 37 44 O=C(Nc1ccccc1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217624042 ED In-Stock Unstable MAPK1 44 39 O=C(Nc1ccccc1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217624042 ED In-Stock Unstable MTOR 67 39 O=C(Nc1ccccc1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217624042 ED In-Stock Unstable PIK3CG 34 50 O=C(Nc1ccccc1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217624042 ED In-Stock Unstable P2RY14 40 34 O=C(Nc1ccccc1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217624042 ED In-Stock Unstable DGAT1 23 41 O=C1O[C@@]2(CCCN(S(=O)(=O)c3ccccc3Br)C2)c2ccccc21 ZINC000217624045 HG For-Sale Unstable NPY5R 23 40 O=C(NC1CCN(Cc2ccccc2)CC1)C(F)F ZINC000217624057 CE On-Demand Unstable CHRM2 35 52 O=C(NC1CCN(Cc2ccccc2)CC1)C(F)F ZINC000217624057 CE On-Demand Unstable CHRM1 26 44 O=C(NC1CCN(Cc2ccccc2)CC1)C(F)F ZINC000217624057 CE On-Demand Unstable ACE 49 34 O=C(NC1CCN(Cc2ccccc2)CC1)C(F)F ZINC000217624057 CE On-Demand Unstable DRD2 34 61 O=C(NC1CCN(Cc2ccccc2)CC1)C(F)F ZINC000217624057 CE On-Demand Unstable DRD4 66 55 O=C(NC1CCN(Cc2ccccc2)CC1)C(F)F ZINC000217624057 CE On-Demand Unstable ACHE 47 52 O=C(NC1CCN(Cc2ccccc2)CC1)C(F)F ZINC000217624057 CE On-Demand Unstable HRH1 29 42 O=C(NC1CCN(Cc2ccccc2)CC1)C(F)F ZINC000217624057 CE On-Demand Unstable DRD3 29 65 O=C(NC1CCN(Cc2ccccc2)CC1)C(F)F ZINC000217624057 CE On-Demand Unstable SLC6A3 30 48 O=C(NC1CCN(Cc2ccccc2)CC1)C(F)F ZINC000217624057 CE On-Demand Unstable CHRM3 50 46 O=C(NC1CCN(Cc2ccccc2)CC1)C(F)F ZINC000217624057 CE On-Demand Unstable GRIN2B 48 36 O=C(NC1CCN(Cc2ccccc2)CC1)C(F)F ZINC000217624057 CE On-Demand Unstable LTA4H 28 47 O=C(NC1CCN(Cc2ccccc2)CC1)C(F)F ZINC000217624057 CE On-Demand Unstable SIGMAR1 100 72 O=C(NC1CCN(Cc2ccccc2)CC1)C(F)F ZINC000217624057 CE On-Demand Unstable SSTR5 52 38 O=C(NC1CCN(Cc2ccccc2)CC1)C(F)F ZINC000217624057 CE On-Demand Unstable BCHE 23 41 O=C(NC1CCN(Cc2ccccc2)CC1)C(F)F ZINC000217624057 CE On-Demand Unstable CCR1 22 43 O=C(NC1CCN(Cc2ccccc2)CC1)C(F)F ZINC000217624057 CE On-Demand Unstable CCR3 77 59 O=C(NC1CCN(Cc2ccccc2)CC1)C(F)F ZINC000217624057 CE On-Demand Unstable C3AR1 44 39 O=C(NC1CCN(Cc2ccccc2)CC1)C(F)F ZINC000217624057 CE On-Demand Unstable SLC18A3 23 42 O=C(NC1CCN(Cc2ccccc2)CC1)C(F)F ZINC000217624057 CE On-Demand Unstable MLNR 44 35 O=C(NC1CCN(Cc2ccccc2)CC1)C(F)F ZINC000217624057 CE On-Demand Unstable CCR2 23 44 O=C(NC1CCN(Cc2ccccc2)CC1)C(F)F ZINC000217624057 CE On-Demand Unstable SLC6A5 26 51 O=C(NC1CCN(Cc2ccccc2)CC1)C(F)F ZINC000217624057 CE On-Demand Unstable BACE1 23 44 O=C(NC1CCN(Cc2ccccc2)CC1)C(F)F ZINC000217624057 CE On-Demand Unstable CXCR3 44 39 O=C(NC1CCN(Cc2ccccc2)CC1)C(F)F ZINC000217624057 CE On-Demand Unstable MCHR1 65 55 O=C(NC1CCN(Cc2ccccc2)CC1)C(F)F ZINC000217624057 CE On-Demand Unstable CACNA1G 43 57 O=C(NC1CCN(Cc2ccccc2)CC1)C(F)F ZINC000217624057 CE On-Demand Unstable MGLL 0 40 O=C(NC1CCN(Cc2ccccc2)CC1)C(F)F ZINC000217624057 CE On-Demand Unstable CCR8 25 47 O=C(NC1CCN(Cc2ccccc2)CC1)C(F)F ZINC000217624057 CE On-Demand Unstable BIRC2 40 46 O=C(NC1CCN(Cc2ccccc2)CC1)C(F)F ZINC000217624057 CE On-Demand Unstable NPFFR1 58 36 O=C(NC1CCN(Cc2ccccc2)CC1)C(F)F ZINC000217624057 CE On-Demand Unstable ADIPOR1 0 54 O=C(NC1CCN(Cc2ccccc2)CC1)C(F)F ZINC000217624057 CE On-Demand Unstable ADIPOR2 0 54 COc1ccc(CCNS(=O)(=O)c2ccc(NC[C@@H]3CCCO3)c(C(=O)O)c2)cc1OC ZINC000217624062 JF In-Stock Unstable IAP 0 43 COc1ccc(CCNS(=O)(=O)c2ccc(NC[C@@H]3CCCO3)c(C(=O)O)c2)cc1OC ZINC000217624062 JF In-Stock Unstable SCMU_MYCTU 0 40 CC[C@H]1CCCN(c2ccccc2CBr)CC1 ZINC000217624096 CJ For-Sale Unstable KCNQ2 47 33 C[C@@H](C(=O)NC1CC1)N1CCN(C(=O)c2ccccc2Nc2cccc(C(F)(F)F)c2)CC1 ZINC000217624103 JH On-Demand Unstable ITGAL 41 33 C[C@@H](C(=O)NC1CC1)N1CCN(C(=O)c2ccccc2Nc2cccc(C(F)(F)F)c2)CC1 ZINC000217624103 JH On-Demand Unstable CACNA1B 44 37 C[C@@H](C(=O)NC1CC1)N1CCN(C(=O)c2ccccc2Nc2cccc(C(F)(F)F)c2)CC1 ZINC000217624103 JH On-Demand Unstable CCR2 39 42 C[C@@H](C(=O)NC1CC1)N1CCN(C(=O)c2ccccc2Nc2cccc(C(F)(F)F)c2)CC1 ZINC000217624103 JH On-Demand Unstable EPHX2 18 49 C[C@@H](C(=O)NC1CC1)N1CCN(C(=O)c2ccccc2Nc2cccc(C(F)(F)F)c2)CC1 ZINC000217624103 JH On-Demand Unstable AKR1C3 23 53 C[C@@H](C(=O)NC1CC1)N1CCN(C(=O)c2ccccc2Nc2cccc(C(F)(F)F)c2)CC1 ZINC000217624103 JH On-Demand Unstable AKR1C2 32 53 CCc1cccc(C)c1NC(=O)N/C=C/c1ccccc1 ZINC000217624104 CI For-Sale Unstable ACAT 0 41 O=C1O[C@]2(CCCN(S(=O)(=O)c3ccccc3Br)C2)c2ccccc21 ZINC000217624107 HG For-Sale Unstable NPY5R 23 40 COc1cc([C@H](CC(=O)O)c2c(O)cc(C)n(CC(=O)O)c2=O)ccc1O ZINC000217624121 GD In-Stock Unstable FOLH1 0 40 COc1cc([C@H](CC(=O)O)c2c(O)cc(C)n(CC(=O)O)c2=O)ccc1O ZINC000217624121 GD In-Stock Unstable RORC 48 37 COc1ccc(CCNS(=O)(=O)c2ccc(NC[C@H]3CCCO3)c(C(=O)O)c2)cc1OC ZINC000217624132 JF In-Stock Unstable IAP 0 43 COc1ccc(CCNS(=O)(=O)c2ccc(NC[C@H]3CCCO3)c(C(=O)O)c2)cc1OC ZINC000217624132 JF In-Stock Unstable SCMU_MYCTU 0 40 CCNC(=O)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217624160 CC In-Stock Unstable MAPK1 46 42 CCNC(=O)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217624160 CC In-Stock Unstable MTOR 47 46 C[C@H](C(=O)NC1CC1)N1CCN(C(=O)c2ccccc2Nc2cccc(C(F)(F)F)c2)CC1 ZINC000217624180 JH On-Demand Unstable ITGAL 41 33 C[C@H](C(=O)NC1CC1)N1CCN(C(=O)c2ccccc2Nc2cccc(C(F)(F)F)c2)CC1 ZINC000217624180 JH On-Demand Unstable CACNA1B 44 37 C[C@H](C(=O)NC1CC1)N1CCN(C(=O)c2ccccc2Nc2cccc(C(F)(F)F)c2)CC1 ZINC000217624180 JH On-Demand Unstable CCR2 39 42 C[C@H](C(=O)NC1CC1)N1CCN(C(=O)c2ccccc2Nc2cccc(C(F)(F)F)c2)CC1 ZINC000217624180 JH On-Demand Unstable EPHX2 18 49 C[C@H](C(=O)NC1CC1)N1CCN(C(=O)c2ccccc2Nc2cccc(C(F)(F)F)c2)CC1 ZINC000217624180 JH On-Demand Unstable AKR1C3 23 53 C[C@H](C(=O)NC1CC1)N1CCN(C(=O)c2ccccc2Nc2cccc(C(F)(F)F)c2)CC1 ZINC000217624180 JH On-Demand Unstable AKR1C2 32 53 Cc1cc(C)c(NC(=O)N/C=C/c2ccccc2)c(C)c1 ZINC000217624203 CI For-Sale Unstable PYGL 22 40 COc1cc([C@@H](CC(=O)O)c2c(O)cc(C)n(CC(=O)O)c2=O)ccc1O ZINC000217624220 GD In-Stock Unstable FOLH1 0 40 COc1cc([C@@H](CC(=O)O)c2c(O)cc(C)n(CC(=O)O)c2=O)ccc1O ZINC000217624220 GD In-Stock Unstable RORC 48 37 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCC3)c(C(=O)O)c2)cc1OC ZINC000217624243 IF In-Stock Unstable DRD2 18 42 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCC3)c(C(=O)O)c2)cc1OC ZINC000217624243 IF In-Stock Unstable FKBP1A 32 42 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCC3)c(C(=O)O)c2)cc1OC ZINC000217624243 IF In-Stock Unstable DRD3 20 42 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCC3)c(C(=O)O)c2)cc1OC ZINC000217624243 IF In-Stock Unstable ABCC8 30 40 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCC3)c(C(=O)O)c2)cc1OC ZINC000217624243 IF In-Stock Unstable TBXA2R 50 39 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCC3)c(C(=O)O)c2)cc1OC ZINC000217624243 IF In-Stock Unstable HTR7 15 41 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCC3)c(C(=O)O)c2)cc1OC ZINC000217624243 IF In-Stock Unstable HTR6 22 42 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCC3)c(C(=O)O)c2)cc1OC ZINC000217624243 IF In-Stock Unstable IAP 0 45 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCC3)c(C(=O)O)c2)cc1OC ZINC000217624243 IF In-Stock Unstable SCMU_MYCTU 0 41 O=C(Nc1ccc(C(F)(F)F)cc1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217624285 HF In-Stock Unstable TRPV1 22 44 O=C(Nc1ccc(C(F)(F)F)cc1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217624285 HF In-Stock Unstable PIK3CA 41 41 O=C(Nc1ccc(C(F)(F)F)cc1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217624285 HF In-Stock Unstable MAPK1 53 38 O=C(Nc1ccc(C(F)(F)F)cc1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217624285 HF In-Stock Unstable MTOR 82 41 O=C(Nc1ccc(C(F)(F)F)cc1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217624285 HF In-Stock Unstable EPHX2 38 47 O=C(Nc1ccc(C(F)(F)F)cc1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217624285 HF In-Stock Unstable PIK3CG 32 41 O=C(Nc1ccc(C(F)(F)F)cc1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217624285 HF In-Stock Unstable TRPM8 56 42 O=C(Nc1ccc(C(F)(F)F)cc1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217624285 HF In-Stock Unstable DGAT1 25 40 COC(=O)c1ccccc1NC(=O)N/C=C/c1ccccc1 ZINC000217624303 CG For-Sale Unstable MMP2 15 44 COC(=O)c1ccccc1NC(=O)N/C=C/c1ccccc1 ZINC000217624303 CG For-Sale Unstable FAS 21 48 Cc1noc(C)c1COc1ccc(CC(=O)N2CCN([C@@H](C)C(=O)NC3CC3)CC2)cc1 ZINC000217624319 IE On-Demand Unstable ADAM17 41 34 O=C(CCCCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCc1ccc2c(c1)OCO2 ZINC000217624333 JI In-Stock Unstable NOS2 83 34 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCCC3)c(C(=O)O)c2)cc1OC ZINC000217624337 IF In-Stock Unstable DRD2 16 41 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCCC3)c(C(=O)O)c2)cc1OC ZINC000217624337 IF In-Stock Unstable FKBP1A 30 41 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCCC3)c(C(=O)O)c2)cc1OC ZINC000217624337 IF In-Stock Unstable DRD3 18 41 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCCC3)c(C(=O)O)c2)cc1OC ZINC000217624337 IF In-Stock Unstable ABCC8 31 41 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCCC3)c(C(=O)O)c2)cc1OC ZINC000217624337 IF In-Stock Unstable TBXA2R 51 41 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCCC3)c(C(=O)O)c2)cc1OC ZINC000217624337 IF In-Stock Unstable HTR6 0 41 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCCC3)c(C(=O)O)c2)cc1OC ZINC000217624337 IF In-Stock Unstable IAP 0 44 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCCCC3)c(C(=O)O)c2)cc1OC ZINC000217624337 IF In-Stock Unstable SCMU_MYCTU 0 41 CN1CCCC[C@@H]1CNC[C@@H](O)c1ccc(C#N)cc1 ZINC000217624393 CD For-Sale Unstable CHRNA10 53 40 Cc1noc(C)c1COc1ccc(CC(=O)N2CCN([C@H](C)C(=O)NC3CC3)CC2)cc1 ZINC000217624398 IE On-Demand Unstable ADAM17 41 34 COc1ccc(CNC(=O)N2CCc3cnc(N4CCOCC4)nc3C2)cc1 ZINC000217624399 GD In-Stock Unstable MAPK1 43 38 COc1ccc(CNC(=O)N2CCc3cnc(N4CCOCC4)nc3C2)cc1 ZINC000217624399 GD In-Stock Unstable NAMPT 36 40 O=C(N/C=C/c1ccccc1)Nc1ccc(F)cc1 ZINC000217624422 CH For-Sale Anodyne MMP2 16 63 O=C(N/C=C/c1ccccc1)Nc1ccc(F)cc1 ZINC000217624422 CH For-Sale Anodyne P96878_MYCTU 17 43 O=C(CCCCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCc1ccc2c(c1)OCO2 ZINC000217624427 JI In-Stock Unstable NOS2 83 34 NC/C=C\CN1CCc2ccccc2C1 ZINC000217624428 BD For-Sale Unstable CHRNA6 0 51 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCOCC3)c(C(=O)O)c2)cc1OC ZINC000217624449 JD In-Stock Unstable TBXA2R 48 38 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCOCC3)c(C(=O)O)c2)cc1OC ZINC000217624449 JD In-Stock Unstable IAP 0 47 COc1ccc(CCNS(=O)(=O)c2ccc(N3CCOCC3)c(C(=O)O)c2)cc1OC ZINC000217624449 JD In-Stock Unstable SCMU_MYCTU 0 41 CN1CCCC[C@H]1CNC[C@@H](O)c1ccc(C#N)cc1 ZINC000217624472 CD For-Sale Unstable CHRNA10 53 40 O=C(NCc1ccccc1Cl)C(F)F ZINC000217624500 BE On-Demand Unstable SLC6A11 0 43 O=C(NCc1ccccc1Cl)C(F)F ZINC000217624500 BE On-Demand Unstable SLC6A12 0 44 O=C(NCc1ccccc1Cl)C(F)F ZINC000217624500 BE On-Demand Unstable SLC6A13 0 42 O=C(NCc1cccs1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217624508 FD In-Stock Unstable MAPK1 43 36 O=C(O)/C=C\c1ccc(C(=O)N2CCCC[C@@H]2CCO)s1 ZINC000217624526 DE For-Sale Unstable HCRTR1 15 41 O=C(N/C=C/c1ccccc1)Nc1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217624529 DI For-Sale Bother IMDH_CRYPV 25 45 O=C(N/C=C/c1ccccc1)Nc1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217624529 DI For-Sale Bother BLM 0 49 CCOCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217624561 JF In-Stock Unstable TBXA2R 42 37 CCOCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217624561 JF In-Stock Unstable BDKRB1 0 40 CCOCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217624561 JF In-Stock Unstable IAP 0 44 CCOCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217624561 JF In-Stock Unstable SCMU_MYCTU 0 40 COC(=O)c1ccc(S(=O)(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217624583 HE For-Sale Unstable NPY5R 25 48 O=C(O)/C=C\c1ccc(C(=O)N2CCCC[C@H]2CCO)s1 ZINC000217624607 DE For-Sale Unstable HCRTR1 15 41 O=S(=O)(c1cccnc1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217624617 FC In-Stock Unstable AKR1C3 50 39 COc1cc([N+](=O)[O-])ccc1NC(=O)N/C=C/c1ccccc1 ZINC000217624635 DG For-Sale Unstable EPHX1 0 57 COc1cc([N+](=O)[O-])ccc1NC(=O)N/C=C/c1ccccc1 ZINC000217624635 DG For-Sale Unstable CACNA1C 48 40 COc1cc([N+](=O)[O-])ccc1NC(=O)N/C=C/c1ccccc1 ZINC000217624635 DG For-Sale Unstable CACNA1D 76 40 COc1cc([N+](=O)[O-])ccc1NC(=O)N/C=C/c1ccccc1 ZINC000217624635 DG For-Sale Unstable KCNMA1 25 57 COc1cc([N+](=O)[O-])ccc1NC(=O)N/C=C/c1ccccc1 ZINC000217624635 DG For-Sale Unstable TRPM8 0 53 O=C(NCc1cccc(Cl)c1)C(F)F ZINC000217624638 BE On-Demand Unstable MAOB 20 40 O=C(NCc1cccc(Cl)c1)C(F)F ZINC000217624638 BE On-Demand Unstable GRIN2B 0 56 O=C(NCc1cccc(Cl)c1)C(F)F ZINC000217624638 BE On-Demand Unstable CTSL 15 42 O=C(NCc1cccc(Cl)c1)C(F)F ZINC000217624638 BE On-Demand Unstable GUAB 0 41 O=C(NCc1cccc(Cl)c1)C(F)F ZINC000217624638 BE On-Demand Unstable FBP1 23 43 O=C(NCc1cccc(Cl)c1)C(F)F ZINC000217624638 BE On-Demand Unstable CTSV 30 42 O=C(NCc1cccc(Cl)c1)C(F)F ZINC000217624638 BE On-Demand Unstable AMP1_PLAFQ 45 43 O=C(NCc1cccc(Cl)c1)C(F)F ZINC000217624638 BE On-Demand Unstable PTGES 15 40 O=C(NCc1cccc(Cl)c1)C(F)F ZINC000217624638 BE On-Demand Unstable PDS 78 45 O=C(NCc1cccc(Cl)c1)C(F)F ZINC000217624638 BE On-Demand Unstable LMGT2 0 46 COC(=O)c1ccc(S(=O)(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217624663 HE For-Sale Unstable NPY5R 25 48 COc1ccc(CCNS(=O)(=O)c2ccc(NCCCOC(C)C)c(C(=O)O)c2)cc1OC ZINC000217624676 JG In-Stock Unstable TBXA2R 47 37 COc1ccc(CCNS(=O)(=O)c2ccc(NCCCOC(C)C)c(C(=O)O)c2)cc1OC ZINC000217624676 JG In-Stock Unstable BDKRB1 0 40 COc1ccc(CCNS(=O)(=O)c2ccc(NCCCOC(C)C)c(C(=O)O)c2)cc1OC ZINC000217624676 JG In-Stock Unstable IAP 0 44 COc1ccc(CCNS(=O)(=O)c2ccc(NCCCOC(C)C)c(C(=O)O)c2)cc1OC ZINC000217624676 JG In-Stock Unstable SCMU_MYCTU 0 40 O=C(N/C=C/c1ccccc1)Nc1ccc([N+](=O)[O-])cc1 ZINC000217624746 CG For-Sale Bother NADE 0 43 O=C(N/C=C/c1ccccc1)Nc1ccc([N+](=O)[O-])cc1 ZINC000217624746 CG For-Sale Bother MMP2 22 42 O=C(N/C=C/c1ccccc1)Nc1ccc([N+](=O)[O-])cc1 ZINC000217624746 CG For-Sale Bother MMP8 24 43 O=C(N/C=C/c1ccccc1)Nc1ccc([N+](=O)[O-])cc1 ZINC000217624746 CG For-Sale Bother MMP9 19 43 O=C(N/C=C/c1ccccc1)Nc1ccc([N+](=O)[O-])cc1 ZINC000217624746 CG For-Sale Bother MMP1 22 43 O=C(N/C=C/c1ccccc1)Nc1ccc([N+](=O)[O-])cc1 ZINC000217624746 CG For-Sale Bother NCE103 22 45 O=C(N/C=C/c1ccccc1)Nc1ccc([N+](=O)[O-])cc1 ZINC000217624746 CG For-Sale Bother P96878_MYCTU 17 40 O=C(N/C=C/c1ccccc1)Nc1ccc([N+](=O)[O-])cc1 ZINC000217624746 CG For-Sale Bother H9B8T9_CAPHI 19 44 C[C@@H](CNCc1cn(CCO)nn1)N(C)C1CC1 ZINC000217624756 CB For-Sale Unstable GBA 15 40 O=C(Nc1ccc(F)cc1Cl)C(F)F ZINC000217624772 BF On-Demand Anodyne PYGL 30 51 O=C1O[C@@]2(CCCN(S(=O)(=O)Cc3cc(F)ccc3F)C2)c2ccccc21 ZINC000217624777 GF For-Sale Unstable NPY5R 24 41 CCCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217624797 JH In-Stock Unstable INHA 44 37 CCCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217624797 JH In-Stock Unstable TBXA2R 48 38 CCCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217624797 JH In-Stock Unstable TBXAS1 15 43 CCCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217624797 JH In-Stock Unstable ALOX15 49 42 CCCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217624797 JH In-Stock Unstable PTGDR 25 40 CCCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217624797 JH In-Stock Unstable IAP 0 45 CCCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217624797 JH In-Stock Unstable PTGDR2 15 40 CCCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217624797 JH In-Stock Unstable AKR1C3 15 45 CCCCCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217624797 JH In-Stock Unstable SCMU_MYCTU 0 42 CN1C(=O)C[C@@H](CNC(=O)CCc2nc3ccccc3[nH]2)c2ccccc21 ZINC000217624807 FF In-Stock Unstable ISPE 0 47 C[C@H](CNCc1cn(CCO)nn1)N(C)C1CC1 ZINC000217624842 CB For-Sale Unstable GBA 15 40 Cc1ccc(CN(C)C(=O)c2ccc(/C=C\C(=O)O)s2)o1 ZINC000217624870 DG For-Sale Unstable HSD17B2 32 40 O=C1O[C@]2(CCCN(S(=O)(=O)Cc3cc(F)ccc3F)C2)c2ccccc21 ZINC000217624874 GF For-Sale Unstable NPY5R 24 41 CN1C(=O)C[C@H](CNC(=O)CCc2nc3ccccc3[nH]2)c2ccccc21 ZINC000217624889 FF In-Stock Unstable ISPE 0 47 O=C(C(F)F)N1CCN(c2ccccc2Cl)CC1 ZINC000217624898 CE On-Demand Unstable DRD2 24 47 O=C(C(F)F)N1CCN(c2ccccc2Cl)CC1 ZINC000217624898 CE On-Demand Unstable DRD3 36 42 O=C(C(F)F)N1CCN(c2ccccc2Cl)CC1 ZINC000217624898 CE On-Demand Unstable MC4R 72 40 O=C(C(F)F)N1CCN(c2ccccc2Cl)CC1 ZINC000217624898 CE On-Demand Unstable KCNQ2 70 40 COc1ccc(CCNS(=O)(=O)c2ccc(NCCC(C)C)c(C(=O)O)c2)cc1OC ZINC000217624900 JG In-Stock Unstable TBXA2R 48 38 COc1ccc(CCNS(=O)(=O)c2ccc(NCCC(C)C)c(C(=O)O)c2)cc1OC ZINC000217624900 JG In-Stock Unstable IAP 0 44 COc1ccc(CCNS(=O)(=O)c2ccc(NCCC(C)C)c(C(=O)O)c2)cc1OC ZINC000217624900 JG In-Stock Unstable SCMU_MYCTU 0 42 C[C@@H](C(=O)NC1CC1)N1CCN(C(=O)CNC(=O)c2ccc(C(C)(C)C)cc2)CC1 ZINC000217624923 HD On-Demand Unstable CCR2 27 42 C[C@@H](C(=O)NC1CC1)N1CCN(C(=O)CNC(=O)c2ccc(C(C)(C)C)cc2)CC1 ZINC000217624923 HD On-Demand Unstable EPHX2 22 42 CN(Cc1ccco1)C(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217624956 CF For-Sale Unstable HSD17B2 29 43 O=C(N/C=C/c1ccccc1)NCCCCl ZINC000217624959 BF For-Sale Unstable AMP1_PLAFQ 20 41 Cc1ccc(S(=O)(=O)N2CCc3cnc(N4CCOCC4)nc3C2)cc1C ZINC000217624967 GD In-Stock Unstable AKR1C3 57 42 O=C1O[C@@]2(CCCN(S(=O)(=O)Cc3ccc(C(F)(F)F)cc3)C2)c2ccccc21 ZINC000217624983 IH For-Sale Unstable NPY5R 21 44 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217625000 JH In-Stock Unstable IAP 0 43 C[C@H](C(=O)NC1CC1)N1CCN(C(=O)CNC(=O)c2ccc(C(C)(C)C)cc2)CC1 ZINC000217625001 HD On-Demand Unstable CCR2 27 42 C[C@H](C(=O)NC1CC1)N1CCN(C(=O)CNC(=O)c2ccc(C(C)(C)C)cc2)CC1 ZINC000217625001 HD On-Demand Unstable EPHX2 22 42 O=C1O[C@]2(CCCN(S(=O)(=O)Cc3ccc(C(F)(F)F)cc3)C2)c2ccccc21 ZINC000217625051 IH For-Sale Unstable NPY5R 21 44 CN1CCCC[C@@H]1CNC(=O)c1cc(C(C)(C)C)nc(=O)[nH]1 ZINC000217625070 DD In-Stock Unstable CACNA1I 41 35 O=C(N/C=C/c1ccccc1)N1CCN(c2ccc(F)cc2)CC1 ZINC000217625078 EG For-Sale Unstable SSTR1 18 41 O=C(N/C=C/c1ccccc1)N1CCN(c2ccc(F)cc2)CC1 ZINC000217625078 EG For-Sale Unstable FAAH 23 42 O=C(N/C=C/c1ccccc1)N1CCN(c2ccc(F)cc2)CC1 ZINC000217625078 EG For-Sale Unstable AKR1C3 0 47 CCC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217625087 JH In-Stock Unstable IAP 0 43 Fc1ccc([C@H]2Oc3c(Br)cc(Br)cc3[C@H]3CC(c4ccc(Cl)cc4)=NN32)cc1 ZINC000217625116 KK In-Stock Unstable MAOB 0 44 Fc1ccc([C@H]2Oc3c(Br)cc(Br)cc3[C@H]3CC(c4ccc(Cl)cc4)=NN32)cc1 ZINC000217625116 KK In-Stock Unstable GRIN2D 71 34 CN1CCCC[C@H]1CNC(=O)c1cc(C(C)(C)C)nc(=O)[nH]1 ZINC000217625149 DD In-Stock Unstable CACNA1I 41 35 O=C(N/C=C/c1ccccc1)Nc1ccccc1O ZINC000217625186 CG For-Sale Anodyne F3 17 40 O=C(N/C=C/c1ccccc1)Nc1ccccc1O ZINC000217625186 CG For-Sale Anodyne MMP2 16 61 COC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217625188 JE In-Stock Unstable TBXA2R 43 38 COC[C@@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217625188 JE In-Stock Unstable IAP 0 43 Clc1ccc(C2=NN3[C@H](C2)c2cc(Br)cc(Br)c2O[C@@H]3c2ccc(OCc3ccccc3)cc2)cc1 ZINC000217625194 KK In-Stock Unstable GRIN2D 69 33 CC(C)Cc1ccc(-c2cc(C(=O)N3CCc4c([nH]c5ccccc45)C3)[nH]n2)cc1 ZINC000217625204 GJ In-Stock Unstable FABI 53 33 CC(C)Cc1ccc(-c2cc(C(=O)N3CCc4c([nH]c5ccccc45)C3)[nH]n2)cc1 ZINC000217625204 GJ In-Stock Unstable TACR3 18 41 COC[C@H](C)Nc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217625270 JE In-Stock Unstable TBXA2R 43 38 CCOc1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217625309 CH For-Sale Unstable LTA4H 33 40 CCOc1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217625309 CH For-Sale Unstable CA1 52 43 CCOc1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217625309 CH For-Sale Unstable SCN2A 37 41 CCOc1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217625309 CH For-Sale Unstable PRNP 19 47 CCOc1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217625309 CH For-Sale Unstable FAAH 21 46 CCOc1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217625309 CH For-Sale Unstable EPHX2 15 42 CCOc1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217625309 CH For-Sale Unstable CA12 22 43 CCOc1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217625309 CH For-Sale Unstable CA9 23 43 CCOc1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217625309 CH For-Sale Unstable NCE103 30 40 O=C(O)[C@H]1CN(Cc2cc3ccccc3o2)CCN(CC2CC2)C1 ZINC000217625402 EF In-Stock Unstable SLC6A1 87 35 O=C(O)[C@H]1CN(Cc2cc3ccccc3o2)CCN(CC2CC2)C1 ZINC000217625402 EF In-Stock Unstable HTR2B 16 55 O=C(O)[C@H]1CN(Cc2cc3ccccc3o2)CCN(CC2CC2)C1 ZINC000217625402 EF In-Stock Unstable SIGMAR1 23 55 CCCCOC(=O)c1ccccc1NC(=O)N/C=C/c1ccccc1 ZINC000217625421 EI For-Sale Unstable TRPM2 0 45 COC(=O)[C@H](CC(C)C)NC(=O)CC/C(C)=C/Cc1c(OC)c(C)c2c(c1OC)C(=O)OC2 ZINC000217625444 JH In-Stock Unstable IMPDH1 0 74 COC(=O)[C@H](CC(C)C)NC(=O)CC/C(C)=C/Cc1c(OC)c(C)c2c(c1OC)C(=O)OC2 ZINC000217625444 JH In-Stock Unstable IMPDH2 0 74 O=S(=O)(c1c(F)cccc1F)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217625523 GD In-Stock Unstable PKM 18 43 CCCN1C[C@H](O)[C@H](O)[C@H](O)[C@@H]1C ZINC000217625536 AB For-Sale Unstable MGAM 29 41 CCCN1C[C@H](O)[C@H](O)[C@H](O)[C@@H]1C ZINC000217625536 AB For-Sale Unstable UGCG 23 44 CCCN1C[C@H](O)[C@H](O)[C@H](O)[C@@H]1C ZINC000217625536 AB For-Sale Unstable GAA 15 49 CCCN1C[C@H](O)[C@H](O)[C@H](O)[C@@H]1C ZINC000217625536 AB For-Sale Unstable GBA2 68 46 CCCN1C[C@H](O)[C@H](O)[C@H](O)[C@@H]1C ZINC000217625536 AB For-Sale Unstable SI 35 49 CC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217625538 CH For-Sale Unstable CA1 24 43 CC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217625538 CH For-Sale Unstable PRNP 28 50 CC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217625538 CH For-Sale Unstable AKR1C3 16 42 CC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217625538 CH For-Sale Unstable P96878_MYCTU 15 45 CC[C@@H]1CCCN(c2ccc(CBr)cc2)CC1 ZINC000217625611 CJ For-Sale Unstable L3MBTL3 33 41 O=C(NCc1cnc2cnccn12)c1cccc(-c2ccccc2)c1 ZINC000217625612 EG In-Stock Unstable E1 0 42 O=C(Nc1cccc(Cl)c1Cl)C(F)F ZINC000217625619 BG On-Demand Anodyne CXCL8 51 39 O=C(Nc1cccc(Cl)c1Cl)C(F)F ZINC000217625619 BG On-Demand Anodyne KCNQ2 42 36 CC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217625660 CH For-Sale Unstable CCR3 18 42 CC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217625660 CH For-Sale Unstable HDAC8 15 47 CC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217625660 CH For-Sale Unstable MMP1 0 45 CC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217625660 CH For-Sale Unstable AKR1C3 43 54 CC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217625660 CH For-Sale Unstable IMDH_CRYPV 46 35 CC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217625660 CH For-Sale Unstable KCNK3 107 40 CC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217625660 CH For-Sale Unstable KCNK9 60 40 O=C(O)Cc1cc(O)c(F)c(Br)c1 ZINC000217625667 BD For-Sale Unstable NR3C1 17 41 O=C(O)Cc1cc(O)c(F)c(Br)c1 ZINC000217625667 BD For-Sale Unstable THRA 51 46 O=C(O)Cc1cc(O)c(F)c(Br)c1 ZINC000217625667 BD For-Sale Unstable THRB 44 46 CC[C@H]1CCCN(c2ccc(CBr)cc2)CC1 ZINC000217625682 CJ For-Sale Unstable L3MBTL3 33 41 O=S(=O)(c1ccc(F)c(Cl)c1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217625725 HD In-Stock Unstable MAPK1 39 40 O=S(=O)(c1ccc(F)c(Cl)c1)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217625725 HD In-Stock Unstable AKR1C3 51 38 O=C(Nc1ccc(F)c(F)c1)C(F)F ZINC000217625730 BE On-Demand Anodyne ENV 40 31 CC(C)CNc1ccc(S(=O)(=O)NCc2ccco2)cc1C(=O)O ZINC000217625740 FF In-Stock Unstable MTNN 40 32 O=C1O[C@@]2(CCCN(S(=O)(=O)c3ccc(F)cc3F)C2)c2ccccc21 ZINC000217625744 GF For-Sale Unstable NPY5R 26 42 O=C(O)Cc1cc(O)c(Br)c(F)c1 ZINC000217625769 BD For-Sale Unstable THRA 35 40 O=C(O)Cc1cc(O)c(Br)c(F)c1 ZINC000217625769 BD For-Sale Unstable THRB 36 40 O=C1[C@@H]2[C@@H](ON(c3ccccc3)[C@H]2c2cccc(Br)c2)C(=O)N1c1cc(Cl)cc(Cl)c1 ZINC000217625815 KK In-Stock Anodyne ACHE 16 63 O=S(=O)(c1ccc2c(c1)OCCO2)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217625835 HC In-Stock Unstable PKM 45 49 O=S(=O)(c1ccc2c(c1)OCCO2)N1CCc2cnc(N3CCOCC3)nc2C1 ZINC000217625835 HC In-Stock Unstable AKR1C3 52 41 O=C1O[C@]2(CCCN(S(=O)(=O)c3ccc(F)cc3F)C2)c2ccccc21 ZINC000217625841 GF For-Sale Unstable NPY5R 26 42 CN1CCCC[C@@H]1CN1CC[C@@H](N)C1=O ZINC000217625932 BC For-Sale Unstable CHRNA10 42 33 COc1ccc(S(=O)(=O)N2CCc3cnc(N4CCOCC4)nc3C2)cc1Cl ZINC000217625938 HD In-Stock Unstable PDE5A 19 43 O=C1O[C@@]2(CCCN(S(=O)(=O)Cc3ccccc3)C2)c2ccccc21 ZINC000217625968 FF For-Sale Unstable SIGMAR1 17 56 O=C1O[C@@]2(CCCN(S(=O)(=O)Cc3ccccc3)C2)c2ccccc21 ZINC000217625968 FF For-Sale Unstable NPY5R 24 40 NS(=O)(=O)c1ccc(CCNC(=O)C(F)F)cc1 ZINC000217625977 CC On-Demand Unstable CA2 175 72 NS(=O)(=O)c1ccc(CCNC(=O)C(F)F)cc1 ZINC000217625977 CC On-Demand Unstable CA6 31 49 NS(=O)(=O)c1ccc(CCNC(=O)C(F)F)cc1 ZINC000217625977 CC On-Demand Unstable CA1 140 72 NS(=O)(=O)c1ccc(CCNC(=O)C(F)F)cc1 ZINC000217625977 CC On-Demand Unstable CA7 86 60 NS(=O)(=O)c1ccc(CCNC(=O)C(F)F)cc1 ZINC000217625977 CC On-Demand Unstable CA13 47 49 NS(=O)(=O)c1ccc(CCNC(=O)C(F)F)cc1 ZINC000217625977 CC On-Demand Unstable CA5B 69 60 NS(=O)(=O)c1ccc(CCNC(=O)C(F)F)cc1 ZINC000217625977 CC On-Demand Unstable CA4 131 68 NS(=O)(=O)c1ccc(CCNC(=O)C(F)F)cc1 ZINC000217625977 CC On-Demand Unstable CA5A 72 60 NS(=O)(=O)c1ccc(CCNC(=O)C(F)F)cc1 ZINC000217625977 CC On-Demand Unstable CA14 69 50 NS(=O)(=O)c1ccc(CCNC(=O)C(F)F)cc1 ZINC000217625977 CC On-Demand Unstable CA12 97 66 NS(=O)(=O)c1ccc(CCNC(=O)C(F)F)cc1 ZINC000217625977 CC On-Demand Unstable CA9 107 66 NS(=O)(=O)c1ccc(CCNC(=O)C(F)F)cc1 ZINC000217625977 CC On-Demand Unstable CAH_METTE 36 49 NS(=O)(=O)c1ccc(CCNC(=O)C(F)F)cc1 ZINC000217625977 CC On-Demand Unstable CYNT 53 59 NS(=O)(=O)c1ccc(CCNC(=O)C(F)F)cc1 ZINC000217625977 CC On-Demand Unstable NCE103 49 53 NS(=O)(=O)c1ccc(CCNC(=O)C(F)F)cc1 ZINC000217625977 CC On-Demand Unstable MTCA1 40 49 NS(=O)(=O)c1ccc(CCNC(=O)C(F)F)cc1 ZINC000217625977 CC On-Demand Unstable P96878_MYCTU 60 53 NS(=O)(=O)c1ccc(CCNC(=O)C(F)F)cc1 ZINC000217625977 CC On-Demand Unstable A6YCJ1_9METZ 32 64 Cc1cc(Cl)ccc1NC(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217626010 DI For-Sale Unstable MAPK11 29 41 Cc1cc(Cl)ccc1NC(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217626010 DI For-Sale Unstable H9CNL0_SPOEX 0 41 CN1CCCC[C@H]1CN1CC[C@@H](N)C1=O ZINC000217626019 BC For-Sale Unstable CHRNA10 42 33 O=C1O[C@]2(CCCN(S(=O)(=O)Cc3ccccc3)C2)c2ccccc21 ZINC000217626066 FF For-Sale Unstable SIGMAR1 17 56 O=C1O[C@]2(CCCN(S(=O)(=O)Cc3ccccc3)C2)c2ccccc21 ZINC000217626066 FF For-Sale Unstable NPY5R 24 40 O=C1O[C@@]2(CCCN(S(=O)(=O)c3cc(F)cc(F)c3)C2)c2ccccc21 ZINC000217626166 GF For-Sale Unstable NPY5R 26 41 CCN(C(=O)c1ccc(/C=C\C(=O)O)s1)C1CCCC1 ZINC000217626191 CG For-Sale Unstable ACE 47 36 COc1cc(F)c(Br)c(C(=O)O)c1 ZINC000217626222 BE For-Sale Unstable AKR1C3 24 40 COc1cc(F)c(Br)c(C(=O)O)c1 ZINC000217626222 BE For-Sale Unstable AKR1C2 58 40 Cc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217626232 CH For-Sale Unstable KIT 22 40 Cc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217626232 CH For-Sale Unstable CCKAR 28 53 Cc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217626232 CH For-Sale Unstable HDAC8 35 42 Cc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217626232 CH For-Sale Unstable KDR 20 41 Cc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217626232 CH For-Sale Unstable MMP2 0 53 Cc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217626232 CH For-Sale Unstable HDAC6 23 48 Cc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217626232 CH For-Sale Unstable CCKBR 40 39 Cc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217626232 CH For-Sale Unstable MMP9 0 53 Cc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217626232 CH For-Sale Unstable IMPDH2 0 45 Cc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217626232 CH For-Sale Unstable MMP1 0 53 Cc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217626232 CH For-Sale Unstable AKR1C3 23 47 Cc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217626232 CH For-Sale Unstable TRPM8 0 47 Cc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217626232 CH For-Sale Unstable KCNK3 113 48 Cc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217626232 CH For-Sale Unstable KCNK9 72 48 O=C1O[C@]2(CCCN(S(=O)(=O)c3cc(F)cc(F)c3)C2)c2ccccc21 ZINC000217626260 GF For-Sale Unstable NPY5R 26 41 CCN(C(=O)c1ccc(/C=C\C(=O)O)cc1)C1CCCC1 ZINC000217626292 CG For-Sale Unstable ACE 61 47 CCN(C(=O)c1ccc(/C=C\C(=O)O)cc1)C1CCCC1 ZINC000217626292 CG For-Sale Unstable LGB 0 40 CCN(C(=O)c1ccc(/C=C\C(=O)O)cc1)C1CCCC1 ZINC000217626292 CG For-Sale Unstable MBTPS1 49 33 CC[C@@H](C)[C@@H](CO)NC(=O)CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217626310 HD In-Stock Unstable CCKAR 48 36 CC[C@@H](C)[C@@H](CO)NC(=O)CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217626310 HD In-Stock Unstable CCKBR 44 36 CC[C@@H](C)[C@@H](CO)NC(=O)CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217626310 HD In-Stock Unstable GHSR 57 38 CC[C@@H](C)[C@@H](CO)NC(=O)CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217626310 HD In-Stock Unstable Q7YY76_CRYPV 0 40 CC[C@@H](C)[C@@H](CO)NC(=O)CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217626310 HD In-Stock Unstable Q7YY07_CRYPV 43 35 O=C(N/C=C/c1ccccc1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217626322 EK For-Sale Anodyne GUAB 0 46 O=C(N/C=C/c1ccccc1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217626322 EK For-Sale Anodyne RAF1 33 45 O=C(N/C=C/c1ccccc1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217626322 EK For-Sale Anodyne Q8MMZ8_EIMTE 54 46 O=C(N/C=C/c1ccccc1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217626322 EK For-Sale Anodyne BRAF 16 42 O=C(N/C=C/c1ccccc1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217626322 EK For-Sale Anodyne PTPA 0 48 O=C(N/C=C/c1ccccc1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217626322 EK For-Sale Anodyne RIPK1 15 44 O=C(N/C=C/c1ccccc1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217626322 EK For-Sale Anodyne IMDH_CRYPV 31 48 O=C(N/C=C/c1ccccc1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217626322 EK For-Sale Anodyne BLM 0 48 CC1(C)[C@H]2CCC(=O)[C@@]1(C)OC2=O ZINC000217626436 AD In-Stock Unstable PPP2R1A 40 29 Cc1cc(Br)c(O)c(C(=O)O)c1F ZINC000217626453 BE For-Sale Unstable AKR1C2 22 40 Cc1cc(Br)c(O)c(C(=O)O)c1F ZINC000217626453 BE For-Sale Unstable AKR1C1 23 40 CC1(C)[C@@H]2CCC(=O)[C@]1(C)OC2=O ZINC000217626514 AD In-Stock Unstable PPP2R1A 40 29 CSC[C@@](C)(O)CNC(=O)Cn1ccc(=O)[nH]c1=O ZINC000217626544 CA For-Sale Unstable DUT 52 33 CSC[C@@](C)(O)CNC(=O)Cn1ccc(=O)[nH]c1=O ZINC000217626544 CA For-Sale Unstable Q8II92_PLAF7 54 36 Cc1cc(/C=C\C(=O)O)ccc1NS(=O)(=O)c1cccs1 ZINC000217626546 DF For-Sale Unstable PTGER3 17 41 O=C1O[C@@]2(CCCN(S(=O)(=O)c3cccc(F)c3)C2)c2ccccc21 ZINC000217626572 FF For-Sale Unstable NPY5R 25 43 O=C1O[C@@]2(CCCN(S(=O)(=O)c3cccc(F)c3)C2)c2ccccc21 ZINC000217626572 FF For-Sale Unstable PKM 28 45 CC1(C)[C@H]2CCC(=O)[C@]1(C)OC2=O ZINC000217626592 AD In-Stock Unstable PPP2R1A 40 29 Cc1cc(NC(=O)C2CCN(C(=O)Cc3c(C)nc4ccccc4c3-c3ccccc3)CC2)no1 ZINC000217626597 JJ On-Demand Unstable ADAM17 46 36 CSC[C@](C)(O)CNC(=O)Cn1ccc(=O)[nH]c1=O ZINC000217626633 CA For-Sale Unstable DUT 52 33 CSC[C@](C)(O)CNC(=O)Cn1ccc(=O)[nH]c1=O ZINC000217626633 CA For-Sale Unstable Q8II92_PLAF7 54 36 O=C1O[C@]2(CCCN(S(=O)(=O)c3cccc(F)c3)C2)c2ccccc21 ZINC000217626651 FF For-Sale Unstable NPY5R 25 43 O=C1O[C@]2(CCCN(S(=O)(=O)c3cccc(F)c3)C2)c2ccccc21 ZINC000217626651 FF For-Sale Unstable PKM 28 45 O=C(N/C=C/c1ccccc1)Nc1cccc(Cl)c1 ZINC000217626749 CI For-Sale Anodyne PPIA 26 43 O=C(N/C=C/c1ccccc1)Nc1cccc(Cl)c1 ZINC000217626749 CI For-Sale Anodyne CMA1 0 41 O=C(N/C=C/c1ccccc1)Nc1cccc(Cl)c1 ZINC000217626749 CI For-Sale Anodyne MMP1 0 66 O=C(N/C=C/c1ccccc1)Nc1cccc(Cl)c1 ZINC000217626749 CI For-Sale Anodyne P95276_MYCTO 0 41 O=C(N/C=C/c1ccccc1)Nc1cccc(Cl)c1 ZINC000217626749 CI For-Sale Anodyne PSBA 0 47 O=C(N/C=C/c1ccccc1)Nc1cccc(Cl)c1 ZINC000217626749 CI For-Sale Anodyne KCNK3 55 48 COc1ccc(CNC(=O)C(F)F)cc1 ZINC000217626750 BD On-Demand Unstable ANPEP 30 55 COc1ccc(CNC(=O)C(F)F)cc1 ZINC000217626750 BD On-Demand Unstable BMP1 59 38 COc1ccc(CNC(=O)C(F)F)cc1 ZINC000217626750 BD On-Demand Unstable TRPV1 30 45 COc1ccc(CNC(=O)C(F)F)cc1 ZINC000217626750 BD On-Demand Unstable MMP13 38 40 COc1ccc(CNC(=O)C(F)F)cc1 ZINC000217626750 BD On-Demand Unstable CTSL 20 40 COc1ccc(CNC(=O)C(F)F)cc1 ZINC000217626750 BD On-Demand Unstable MTNR1A 49 40 COc1ccc(CNC(=O)C(F)F)cc1 ZINC000217626750 BD On-Demand Unstable CA9 23 50 COc1ccc(CNC(=O)C(F)F)cc1 ZINC000217626750 BD On-Demand Unstable U38 0 44 COc1ccc(CNC(=O)C(F)F)cc1 ZINC000217626750 BD On-Demand Unstable PROKR1 56 36 COc1ccc(CNC(=O)C(F)F)cc1 ZINC000217626750 BD On-Demand Unstable KCNJ2 0 45 COc1ccc(CNC(=O)C(F)F)cc1 ZINC000217626750 BD On-Demand Unstable Q76353_9HIV1 0 45 O=C1O[C@@]2(CCCN(S(=O)(=O)c3ccc4ccccc4c3)C2)c2ccccc21 ZINC000217626759 GH For-Sale Unstable NPY5R 27 42 O=C1O[C@@]2(CCCN(S(=O)(=O)c3ccc4ccccc4c3)C2)c2ccccc21 ZINC000217626759 GH For-Sale Unstable PKM 24 42 O=C1O[C@@]2(CCCN(S(=O)(=O)c3ccc4ccccc4c3)C2)c2ccccc21 ZINC000217626759 GH For-Sale Unstable AKR1C3 15 43 CC(=O)Nc1cccc([C@@H](C)N[C@@H]2CCC[C@@H](O)C2)c1 ZINC000217626839 CF For-Sale Unstable PTGIR 15 41 Cc1cccc(S(=O)(=O)NCC(=O)N2CCc3ncncc3C2)c1 ZINC000217626840 EC In-Stock Unstable HTR7 15 40 O=C1O[C@]2(CCCN(S(=O)(=O)c3ccc4ccccc4c3)C2)c2ccccc21 ZINC000217626854 GH For-Sale Unstable NPY5R 27 42 O=C1O[C@]2(CCCN(S(=O)(=O)c3ccc4ccccc4c3)C2)c2ccccc21 ZINC000217626854 GH For-Sale Unstable PKM 24 42 O=C1O[C@]2(CCCN(S(=O)(=O)c3ccc4ccccc4c3)C2)c2ccccc21 ZINC000217626854 GH For-Sale Unstable AKR1C3 15 43 O=C(Nc1ccc(F)c(Cl)c1)C(F)F ZINC000217626884 BF On-Demand Anodyne MAOB 17 45 O=C(Nc1ccc(F)c(Cl)c1)C(F)F ZINC000217626884 BF On-Demand Anodyne SLC1A1 32 41 O=C(Nc1ccc(F)c(Cl)c1)C(F)F ZINC000217626884 BF On-Demand Anodyne SLC1A2 34 41 O=C(Nc1ccc(F)c(Cl)c1)C(F)F ZINC000217626884 BF On-Demand Anodyne ERBB4 46 38 O=C(Nc1ccc(F)c(Cl)c1)C(F)F ZINC000217626884 BF On-Demand Anodyne ENV 44 34 O=C(Nc1ccc(F)c(Cl)c1)C(F)F ZINC000217626884 BF On-Demand Anodyne P95276_MYCTO 0 49 O=C(Nc1ccc(F)c(Cl)c1)C(F)F ZINC000217626884 BF On-Demand Anodyne PSBA 0 40 O=C(Nc1ccc(F)c(Cl)c1)C(F)F ZINC000217626884 BF On-Demand Anodyne PPX1 0 40 CC(=O)Nc1cccc([C@H](C)N[C@@H]2CCC[C@@H](O)C2)c1 ZINC000217626934 CF On-Demand Unstable PTGIR 15 41 COCCNc1ccc(S(=O)(=O)NCc2ccco2)cc1C(=O)O ZINC000217626952 FD In-Stock Unstable BDKRB1 0 41 O=C(N/C=C/c1ccccc1)N1CCN(Cc2ccccc2)CC1 ZINC000217626955 DG For-Sale Unstable DRD2 24 42 O=C(N/C=C/c1ccccc1)N1CCN(Cc2ccccc2)CC1 ZINC000217626955 DG For-Sale Unstable DRD4 54 42 O=C(N/C=C/c1ccccc1)N1CCN(Cc2ccccc2)CC1 ZINC000217626955 DG For-Sale Unstable DRD3 0 40 O=C(N/C=C/c1ccccc1)N1CCN(Cc2ccccc2)CC1 ZINC000217626955 DG For-Sale Unstable CHRM3 15 42 O=C(N/C=C/c1ccccc1)N1CCN(Cc2ccccc2)CC1 ZINC000217626955 DG For-Sale Unstable SIGMAR1 68 52 O=C(N/C=C/c1ccccc1)N1CCN(Cc2ccccc2)CC1 ZINC000217626955 DG For-Sale Unstable FAAH 35 54 O=C(N/C=C/c1ccccc1)N1CCN(Cc2ccccc2)CC1 ZINC000217626955 DG For-Sale Unstable MGLL 0 48 O=C(N/C=C/c1ccccc1)N1CCN(Cc2ccccc2)CC1 ZINC000217626955 DG For-Sale Unstable ABHD6 0 42 O=C(N/C=C/c1ccccc1)N1CCN(Cc2ccccc2)CC1 ZINC000217626955 DG For-Sale Unstable NPFFR1 51 35 O=C(N/C=C/c1ccccc1)N1CCN(Cc2ccccc2)CC1 ZINC000217626955 DG For-Sale Unstable GPR183 0 40 Cc1ccc(S(=O)(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217626960 FF For-Sale Unstable NPY5R 26 42 O=C(C(F)F)N1CCN(c2ccccc2O)CC1 ZINC000217626996 CD On-Demand Unstable KCNQ2 44 38 CC(=O)Nc1cccc([C@@H](C)N[C@H]2CCC[C@@H](O)C2)c1 ZINC000217626998 CF For-Sale Unstable PTGIR 15 41 Cc1ccc(S(=O)(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217627036 FF For-Sale Unstable NPY5R 26 42 COCCCNc1ccc(S(=O)(=O)NCc2ccco2)cc1C(=O)O ZINC000217627051 FD In-Stock Unstable BDKRB1 0 42 Cn1c([C@@H]2CCCN(C(=O)CN3CCCC3)C2)nc2ccccc21 ZINC000217627070 EE In-Stock Unstable SLC6A1 67 33 CCC[C@@H](N[C@@H]1CCN2CCCC[C@@H]12)c1ccc(Cl)cc1 ZINC000217627080 DI For-Sale Unstable SLC6A1 0 43 CC(=O)Nc1cccc([C@H](C)N[C@H]2CCC[C@@H](O)C2)c1 ZINC000217627090 CF On-Demand Unstable PTGIR 15 41 O=C(C(F)F)N1CCN(c2cccc(Cl)c2)CC1 ZINC000217627110 CE On-Demand Unstable HTR1A 24 54 O=C(C(F)F)N1CCN(c2cccc(Cl)c2)CC1 ZINC000217627110 CE On-Demand Unstable SLC6A7 0 40 O=C1O[C@@]2(CCCN(S(=O)(=O)c3ccc(Cl)cc3)C2)c2ccccc21 ZINC000217627142 GG For-Sale Unstable NPY5R 24 42 Cn1c([C@H]2CCCN(C(=O)CN3CCCC3)C2)nc2ccccc21 ZINC000217627150 EE In-Stock Unstable SLC6A1 67 33 CCC[C@H](N[C@@H]1CCN2CCCC[C@@H]12)c1ccc(Cl)cc1 ZINC000217627157 DI For-Sale Unstable SLC6A1 0 43 O=C1O[C@]2(CCCN(S(=O)(=O)c3ccc(Cl)cc3)C2)c2ccccc21 ZINC000217627211 GG For-Sale Unstable NPY5R 24 42 CCC[C@@H](N[C@H]1CCN2CCCC[C@@H]12)c1ccc(Cl)cc1 ZINC000217627237 DI For-Sale Unstable SLC6A1 0 43 Cc1cc(C)cc(NC(=O)C(F)F)c1 ZINC000217627245 AF On-Demand Unstable SCN10A 35 41 COC(=O)c1ccc(S(=O)(=O)N2CCc3ncncc3C2)cc1 ZINC000217627251 ED In-Stock Unstable TGM2 40 32 COC(=O)c1ccc(S(=O)(=O)N2CCc3ncncc3C2)cc1 ZINC000217627251 ED In-Stock Unstable F13A1 49 34 COC(=O)c1ccc(S(=O)(=O)N2CCc3ncncc3C2)cc1 ZINC000217627251 ED In-Stock Unstable AKR1C3 61 43 O=C(N/C=C/c1ccccc1)NC1CCCCCCCCCCC1 ZINC000217627258 EK For-Sale Unstable FAAH 17 57 O=C(N/C=C/c1ccccc1)NC1CCCCCCCCCCC1 ZINC000217627258 EK For-Sale Unstable EPHX2 33 56 CN1CCN(CCC(=O)NCCc2noc(C3CCCC3)n2)CC1 ZINC000217627262 ED In-Stock Unstable ETHR 47 37 C[C@@H](Nc1ccc(S(=O)(=O)NCc2ccco2)cc1C(=O)O)c1ccccc1 ZINC000217627264 HH In-Stock Unstable CASP3 19 41 CSC[C@@](C)(O)CNC(=O)c1c[nH]c2ccccc12 ZINC000217627299 CE For-Sale Unstable CFTR 37 44 CSC[C@@](C)(O)CNC(=O)c1c[nH]c2ccccc12 ZINC000217627299 CE For-Sale Unstable MMP7 23 40 CCC[C@H](N[C@H]1CCN2CCCC[C@@H]12)c1ccc(Cl)cc1 ZINC000217627320 DI For-Sale Unstable SLC6A1 0 43 COc1ccc(S(=O)(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217627327 FF For-Sale Unstable NPY5R 27 46 COc1ccc(S(=O)(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217627327 FF For-Sale Unstable PKM 15 47 C[C@H](Nc1ccc(S(=O)(=O)NCc2ccco2)cc1C(=O)O)c1ccccc1 ZINC000217627343 HH In-Stock Unstable CASP3 19 41 O=C(N/C=C/c1ccccc1)NCCN1CCOCC1 ZINC000217627367 CD For-Sale Unstable CNR1 0 41 O=C(N/C=C/c1ccccc1)NCCN1CCOCC1 ZINC000217627367 CD For-Sale Unstable CASR 49 37 O=C(N/C=C/c1ccccc1)NCCN1CCOCC1 ZINC000217627367 CD For-Sale Unstable ADCY5 17 40 O=C(N/C=C/c1ccccc1)NCCN1CCOCC1 ZINC000217627367 CD For-Sale Unstable PTGDS 38 40 O=C(N/C=C/c1ccccc1)NCCN1CCOCC1 ZINC000217627367 CD For-Sale Unstable EPHX2 23 54 O=C(N/C=C/c1ccccc1)NCCN1CCOCC1 ZINC000217627367 CD For-Sale Unstable PLD2 45 32 O=C(N/C=C/c1ccccc1)NCCN1CCOCC1 ZINC000217627367 CD For-Sale Unstable HPGDS 24 43 CSC[C@](C)(O)CNC(=O)c1c[nH]c2ccccc12 ZINC000217627383 CE For-Sale Unstable CFTR 37 44 CSC[C@](C)(O)CNC(=O)c1c[nH]c2ccccc12 ZINC000217627383 CE For-Sale Unstable MMP7 23 40 O=C(C[C@H](c1ccc2c(c1)OCO2)c1c(O)c(O)c(O)c2c(=O)cc(-c3ccccc3)oc12)N1CCOCC1 ZINC000217627394 KH In-Stock Unstable RORC 36 45 COc1ccc(S(=O)(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217627407 FF For-Sale Unstable NPY5R 27 46 COc1ccc(S(=O)(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217627407 FF For-Sale Unstable PKM 15 47 O=C(O)c1cc(S(=O)(=O)NCc2ccco2)ccc1NCCc1ccccc1 ZINC000217627460 HG In-Stock Unstable TBXA2R 42 37 O=C(C[C@@H](c1ccc2c(c1)OCO2)c1c(O)c(O)c(O)c2c(=O)cc(-c3ccccc3)oc12)N1CCOCC1 ZINC000217627465 KH In-Stock Unstable RORC 0 45 O=C1O[C@@]2(CCCN(S(=O)(=O)Cc3ccc(Cl)cc3)C2)c2ccccc21 ZINC000217627522 GG For-Sale Unstable NPY5R 23 42 O=C(Nc1ccc(Cl)cc1F)C(F)F ZINC000217627535 BF On-Demand Anodyne ACPS 0 40 O=C(CCc1ccc(=O)n(Cc2ccccc2)n1)Nc1nc(-c2cccnc2)cs1 ZINC000217627560 HG In-Stock Unstable PDE5A 19 42 O=C(CCc1ccc(=O)n(Cc2ccccc2)n1)Nc1nc(-c2cccnc2)cs1 ZINC000217627560 HG In-Stock Unstable ROCK1 22 44 O=C(CCc1ccc(=O)n(Cc2ccccc2)n1)Nc1nc(-c2cccnc2)cs1 ZINC000217627560 HG In-Stock Unstable ROCK2 16 43 O=C(CCc1ccc(=O)n(Cc2ccccc2)n1)Nc1nc(-c2cccnc2)cs1 ZINC000217627560 HG In-Stock Unstable HDAC9 15 45 O=C(CCc1ccc(=O)n(Cc2ccccc2)n1)Nc1nc(-c2cccnc2)cs1 ZINC000217627560 HG In-Stock Unstable TRPA1 20 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccco3)cc2C(=O)O)cc1 ZINC000217627573 IG In-Stock Unstable BMP1 45 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccco3)cc2C(=O)O)cc1 ZINC000217627573 IG In-Stock Unstable IAP 0 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccco3)cc2C(=O)O)cc1 ZINC000217627573 IG In-Stock Unstable AKR1C3 25 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccco3)cc2C(=O)O)cc1 ZINC000217627573 IG In-Stock Unstable AKR1C2 40 33 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(C(C)C)cc2)CC(=O)O4)cc1O ZINC000217627583 JK In-Stock Unstable AKR1B1 0 47 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(C(C)C)cc2)CC(=O)O4)cc1O ZINC000217627583 JK In-Stock Unstable CYP1B1 57 37 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(C(C)C)cc2)CC(=O)O4)cc1O ZINC000217627583 JK In-Stock Unstable CYP1A1 40 47 O=C(O)COc1cc2c(cc1Cl)OCCO2 ZINC000217627587 BD For-Sale Unstable PTGDR2 35 40 O=C1O[C@]2(CCCN(S(=O)(=O)Cc3ccc(Cl)cc3)C2)c2ccccc21 ZINC000217627608 GG For-Sale Unstable NPY5R 23 42 CCCCCN[C@@H]1CCN2CCCC[C@@H]12 ZINC000217627611 BE For-Sale Unstable GLB1 25 40 CC1CCC(NC(=O)c2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217627628 CG For-Sale Unstable HDAC8 15 43 Cc1ccc(F)cc1NC(=O)C(F)F ZINC000217627653 BE On-Demand Unstable LEF 62 34 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(C(C)C)cc2)CC(=O)O4)cc1O ZINC000217627662 JK In-Stock Unstable AKR1B1 0 47 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(C(C)C)cc2)CC(=O)O4)cc1O ZINC000217627662 JK In-Stock Unstable CYP1B1 57 37 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(C(C)C)cc2)CC(=O)O4)cc1O ZINC000217627662 JK In-Stock Unstable CYP1A1 40 47 COc1ccc(CC(=O)NC[C@@](C)(O)CSC)cc1F ZINC000217627667 DD On-Demand Unstable TRPV1 29 43 CCCCCN[C@H]1CCN2CCCC[C@@H]12 ZINC000217627684 BE For-Sale Unstable GLB1 25 40 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccco3)cc2C(=O)O)cc1OC ZINC000217627690 JG In-Stock Unstable IAP 0 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCc3ccco3)cc2C(=O)O)cc1OC ZINC000217627690 JG In-Stock Unstable SCMU_MYCTU 0 43 O=C(N/C=C/c1ccccc1)NCCN1CCNCC1 ZINC000217627700 CC For-Sale Unstable PLD2 62 34 O=C1O[C@@]2(CCCN(S(=O)(=O)Cc3cc(F)cc(F)c3)C2)c2ccccc21 ZINC000217627727 GF In-Stock Unstable NPY5R 25 40 COc1ccc(CC(=O)NC[C@](C)(O)CSC)cc1F ZINC000217627753 DD On-Demand Unstable TRPV1 29 43 O=C(Nc1cc([N+](=O)[O-])ccc1F)C(F)F ZINC000217627780 BD On-Demand Bother WDR5 35 41 COc1ccc(O)c(CN[C@@H]2CCN3CCCC[C@@H]23)c1 ZINC000217627785 CE On-Demand Unstable SIGMAR1 0 43 Cc1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217627805 CG For-Sale Unstable ANPEP 37 47 Cc1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217627805 CG For-Sale Unstable AMP1_PLAFQ 45 42 COc1ccc([C@H]2SCCN2C(=O)c2ccco2)cc1 ZINC000217627810 CG In-Stock Unstable MMP7 17 45 O=C1O[C@]2(CCCN(S(=O)(=O)Cc3cc(F)cc(F)c3)C2)c2ccccc21 ZINC000217627813 GF In-Stock Unstable NPY5R 25 40 Cc1ccc(CC(=O)Nc2ccc(-c3ccccc3)cn2)cc1 ZINC000217627856 DI On-Demand Unstable MME 43 38 Cc1ccc(CC(=O)Nc2ccc(-c3ccccc3)cn2)cc1 ZINC000217627856 DI On-Demand Unstable GSK3A 17 40 Cc1ccc(CC(=O)Nc2ccc(-c3ccccc3)cn2)cc1 ZINC000217627856 DI On-Demand Unstable CA5A 40 35 Cc1ccc(CC(=O)Nc2ccc(-c3ccccc3)cn2)cc1 ZINC000217627856 DI On-Demand Unstable MAPK8 15 40 Cc1ccc(CC(=O)Nc2ccc(-c3ccccc3)cn2)cc1 ZINC000217627856 DI On-Demand Unstable CDK5 24 42 Cc1ccc(CC(=O)Nc2ccc(-c3ccccc3)cn2)cc1 ZINC000217627856 DI On-Demand Unstable LUCI_LUCLA 55 59 Cc1ccc(CC(=O)Nc2ccc(-c3ccccc3)cn2)cc1 ZINC000217627856 DI On-Demand Unstable RORC 35 40 COc1ccc(O)c(CN[C@H]2CCN3CCCC[C@@H]23)c1 ZINC000217627874 CE On-Demand Unstable SIGMAR1 0 43 COc1ccc([C@@H]2SCCN2C(=O)c2ccco2)cc1 ZINC000217627893 CG In-Stock Unstable MMP7 17 45 COC(=O)c1ccc([N+](=O)[O-])cc1OC(F)F ZINC000217627914 BD For-Sale Unstable CACNA1C 43 35 COC(=O)c1ccc([N+](=O)[O-])cc1OC(F)F ZINC000217627914 BD For-Sale Unstable CACNA1D 71 35 COC(=O)c1ccc([N+](=O)[O-])cc1OC(F)F ZINC000217627914 BD For-Sale Unstable KCNMA1 21 43 O=C(N/C=C/c1ccccc1)NCc1ccncc1 ZINC000217627916 CF For-Sale Unstable ANPEP 15 40 O=C(N/C=C/c1ccccc1)NCc1ccncc1 ZINC000217627916 CF For-Sale Unstable NAMPT 41 41 O=C(O)c1cc(S(=O)(=O)NCc2ccco2)ccc1NC[C@@H]1CCCO1 ZINC000217627918 GE In-Stock Unstable BDKRB1 0 40 O=C(O)/C=C\c1cccc(C(=O)NC[C@@H]2CCCO2)c1 ZINC000217627946 CD For-Sale Unstable HDAC8 19 40 O=C(Nc1ccc(F)c([N+](=O)[O-])c1)C(F)F ZINC000217627977 BD On-Demand Bother AADAC 0 49 O=C(O)c1cc(S(=O)(=O)NCc2ccco2)ccc1NC[C@H]1CCCO1 ZINC000217628009 GE In-Stock Unstable BDKRB1 0 40 O=C(O)/C=C\c1cccc(C(=O)NC[C@H]2CCCO2)c1 ZINC000217628037 CD For-Sale Unstable HDAC8 19 40 CCOC(=O)COc1cccc(CCCO)c1 ZINC000217628058 BD For-Sale Unstable UPP1 48 35 CCOC(=O)COc1cccc(CCCO)c1 ZINC000217628058 BD For-Sale Unstable MTNR1A 16 43 CCOC(=O)COc1cccc(CCCO)c1 ZINC000217628058 BD For-Sale Unstable PLA2G4B 54 42 CCOC(=O)COc1cccc(CCCO)c1 ZINC000217628058 BD For-Sale Unstable CRTM 68 39 CCOC(=O)COc1cccc(CCCO)c1 ZINC000217628058 BD For-Sale Unstable PDS 48 33 O=C(O)c1cc(S(=O)(=O)NCc2ccco2)ccc1N1CCCC1 ZINC000217628109 FE In-Stock Unstable SFRP1 53 32 O=C(O)c1cc(S(=O)(=O)NCc2ccco2)ccc1N1CCCC1 ZINC000217628109 FE In-Stock Unstable WNT3 45 32 O=C(N/C=C/c1ccccc1)NCCCN1CCOCC1 ZINC000217628141 CD For-Sale Unstable HTR1A 23 43 O=C(N/C=C/c1ccccc1)NCCCN1CCOCC1 ZINC000217628141 CD For-Sale Unstable DRD2 28 47 O=C(N/C=C/c1ccccc1)NCCCN1CCOCC1 ZINC000217628141 CD For-Sale Unstable ADRA1D 15 40 O=C(N/C=C/c1ccccc1)NCCCN1CCOCC1 ZINC000217628141 CD For-Sale Unstable ADRA1A 30 40 O=C(N/C=C/c1ccccc1)NCCCN1CCOCC1 ZINC000217628141 CD For-Sale Unstable ADRA1B 18 40 O=C(N/C=C/c1ccccc1)NCCCN1CCOCC1 ZINC000217628141 CD For-Sale Unstable DRD3 51 47 O=C(N/C=C/c1ccccc1)NCCCN1CCOCC1 ZINC000217628141 CD For-Sale Unstable CASR 49 36 O=C(N/C=C/c1ccccc1)NCCCN1CCOCC1 ZINC000217628141 CD For-Sale Unstable HTR7 16 41 O=C(N/C=C/c1ccccc1)NCCCN1CCOCC1 ZINC000217628141 CD For-Sale Unstable TACR2 30 45 O=C(N/C=C/c1ccccc1)NCCCN1CCOCC1 ZINC000217628141 CD For-Sale Unstable SIGMAR1 18 40 O=C(N/C=C/c1ccccc1)NCCCN1CCOCC1 ZINC000217628141 CD For-Sale Unstable CCR3 24 40 O=C(N/C=C/c1ccccc1)NCCCN1CCOCC1 ZINC000217628141 CD For-Sale Unstable EPHX2 25 50 CCc1ccc(NC(=O)C(F)F)cc1 ZINC000217628193 AE On-Demand Unstable SCN2A 22 41 O=C(O)c1cc(S(=O)(=O)NCc2ccco2)ccc1N1CCCCC1 ZINC000217628231 FE In-Stock Unstable WNT3 43 31 N#Cc1cc2c(nc1NCCc1c[nH]c3ccccc13)CCCC2 ZINC000217628347 DH On-Demand Unstable ACHE 41 43 N#Cc1cc2c(nc1NCCc1c[nH]c3ccccc13)CCCC2 ZINC000217628347 DH On-Demand Unstable BCHE 35 44 CN(Cc1ccccc1)C(=O)N/C=C/c1ccccc1 ZINC000217628365 CG For-Sale Unstable LIMK2 41 39 COc1ccc(SCC(=O)NC[C@@](C)(O)CSC)cc1 ZINC000217628475 DE On-Demand Unstable FAS 50 45 NCc1cccc(CNC(=O)N/C=C/c2ccccc2)c1 ZINC000217628488 CF For-Sale Unstable TPSAB1 41 40 NCc1cccc(CNC(=O)N/C=C/c2ccccc2)c1 ZINC000217628488 CF For-Sale Unstable AMP1_PLAFQ 43 35 Cn1nnc(Br)c1C[C@H](N)C(=O)O ZINC000217628509 BB In-Stock Unstable GRIA3 61 38 Cn1nnc(Br)c1C[C@H](N)C(=O)O ZINC000217628509 BB In-Stock Unstable GRIA2 50 38 Cn1nnc(Br)c1C[C@H](N)C(=O)O ZINC000217628509 BB In-Stock Unstable GRIA4 59 38 COc1ccc(SCC(=O)NC[C@](C)(O)CSC)cc1 ZINC000217628571 DE On-Demand Unstable FAS 50 45 Cn1nnc(Br)c1C[C@@H](N)C(=O)O ZINC000217628592 BB In-Stock Unstable GRIA3 61 38 Cn1nnc(Br)c1C[C@@H](N)C(=O)O ZINC000217628592 BB In-Stock Unstable GRIA2 50 38 Cn1nnc(Br)c1C[C@@H](N)C(=O)O ZINC000217628592 BB In-Stock Unstable GRIA4 59 38 COc1ccc([C@H]2SCCN2C(=O)c2ccccc2C(F)(F)F)cc1 ZINC000217628600 FJ In-Stock Unstable RBP4 40 35 Cc1csc(NC(=O)N/C=C/c2ccccc2)n1 ZINC000217628603 CG For-Sale Unstable GCK 18 46 Cc1csc(NC(=O)N/C=C/c2ccccc2)n1 ZINC000217628603 CG For-Sale Unstable SLC12A5 15 43 COc1ccc([C@@H]2SCCN2C(=O)c2ccccc2C(F)(F)F)cc1 ZINC000217628684 FJ In-Stock Unstable RBP4 48 35 O=C1O[C@@]2(CCCN(S(=O)(=O)c3ccc4oc(=O)[nH]c4c3)C2)c2ccccc21 ZINC000217628707 HD For-Sale Unstable NPY5R 25 42 N#Cc1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217628718 CG For-Sale Mild DHODH 0 41 N#Cc1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217628718 CG For-Sale Mild P95276_MYCTO 0 41 O=C1O[C@]2(CCCN(S(=O)(=O)c3ccc4oc(=O)[nH]c4c3)C2)c2ccccc21 ZINC000217628793 HD For-Sale Unstable NPY5R 25 42 CN(C)C1CCN(C(=O)c2ccc(/C=C\C(=O)O)s2)CC1 ZINC000217628795 DE For-Sale Unstable L3MBTL1 0 44 CN(C)C1CCN(C(=O)c2ccc(/C=C\C(=O)O)s2)CC1 ZINC000217628795 DE For-Sale Unstable L3MBTL3 18 44 CCc1cc(OC)c(OC)c(C(=O)O)c1Cl ZINC000217628804 BF For-Sale Unstable DRD2 23 40 CCc1cc(OC)c(OC)c(C(=O)O)c1Cl ZINC000217628804 BF For-Sale Unstable ALS 46 35 O=C(NC1CCCCCCC1)C(F)F ZINC000217628822 BE On-Demand Unstable EPHX2 25 40 O=C(NC1CCCCCCC1)C(F)F ZINC000217628822 BE On-Demand Unstable P95276_MYCTO 0 40 COc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217628840 CG For-Sale Unstable LPL 41 32 COc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217628840 CG For-Sale Unstable CYP1B1 36 40 COc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217628840 CG For-Sale Unstable CA1 15 41 COc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217628840 CG For-Sale Unstable CCKAR 0 43 COc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217628840 CG For-Sale Unstable MTNR1A 35 50 COc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217628840 CG For-Sale Unstable MTNR1B 40 50 COc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217628840 CG For-Sale Unstable CYP1A1 17 40 COc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217628840 CG For-Sale Unstable EPHX2 18 48 COc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217628840 CG For-Sale Unstable IMPDH2 0 41 COc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217628840 CG For-Sale Unstable TAAR1 35 45 COc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217628840 CG For-Sale Unstable AKR1C3 35 50 COc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217628840 CG For-Sale Unstable AKR1C2 54 39 COc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217628840 CG For-Sale Unstable PSBA 0 51 COc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217628840 CG For-Sale Unstable KCNK3 85 51 COc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217628840 CG For-Sale Unstable KCNK9 65 42 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NCc2ccco2)cc1C(=O)O ZINC000217628887 FG In-Stock Unstable CASP3 15 40 CCOC(=O)CN1C(=O)[C@]2(N[C@H](C)[C@@H]3C(=O)N(Cc4ccccc4)C(=O)[C@@H]32)c2ccccc21 ZINC000217628894 ID In-Stock Unstable EDNRB 42 38 COc1ccccc1Oc1ccc(S(=O)(=O)N2CCC[C@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217628905 JI For-Sale Unstable NPY5R 17 41 COc1ccc2[nH]c3c(c2c1)CCC[C@@H]3NC(=O)Cc1c(C)[nH]c2ccccc12 ZINC000217628944 GJ In-Stock Unstable MAPKAPK2 23 46 COc1ccc2[nH]c3c(c2c1)CCC[C@@H]3NC(=O)Cc1c(C)[nH]c2ccccc12 ZINC000217628944 GJ In-Stock Unstable MTNR1A 54 38 COc1ccc2[nH]c3c(c2c1)CCC[C@@H]3NC(=O)Cc1c(C)[nH]c2ccccc12 ZINC000217628944 GJ In-Stock Unstable MTNR1B 45 38 O=C(N/C=C/c1ccccc1)Nc1cc(Cl)ccc1O ZINC000217628954 CH For-Sale Anodyne CMA1 0 44 O=C(N/C=C/c1ccccc1)Nc1cc(Cl)ccc1O ZINC000217628954 CH For-Sale Anodyne KCNMA1 33 52 O=C(N/C=C/c1ccccc1)Nc1cc(Cl)ccc1O ZINC000217628954 CH For-Sale Anodyne MMP1 0 44 COc1ccc([C@H]2SCCN2S(=O)(=O)c2ccc(Br)s2)cc1 ZINC000217628962 HH In-Stock Unstable MMP13 26 40 COc1ccc([C@H]2SCCN2S(=O)(=O)c2ccc(Br)s2)cc1 ZINC000217628962 HH In-Stock Unstable MMP3 28 40 COc1ccc([C@H]2SCCN2S(=O)(=O)c2ccc(Br)s2)cc1 ZINC000217628962 HH In-Stock Unstable MMP9 19 40 COc1ccc([C@H]2SCCN2S(=O)(=O)c2ccc(Br)s2)cc1 ZINC000217628962 HH In-Stock Unstable MMP7 33 40 COc1ccc([C@H]2SCCN2S(=O)(=O)c2ccc(Br)s2)cc1 ZINC000217628962 HH In-Stock Unstable MMP1 29 40 NS(=O)(=O)c1ccc(CNC(=O)C(F)F)cc1 ZINC000217628973 CC On-Demand Unstable CA2 188 68 NS(=O)(=O)c1ccc(CNC(=O)C(F)F)cc1 ZINC000217628973 CC On-Demand Unstable CA6 37 46 NS(=O)(=O)c1ccc(CNC(=O)C(F)F)cc1 ZINC000217628973 CC On-Demand Unstable CA1 158 68 NS(=O)(=O)c1ccc(CNC(=O)C(F)F)cc1 ZINC000217628973 CC On-Demand Unstable CA7 97 68 NS(=O)(=O)c1ccc(CNC(=O)C(F)F)cc1 ZINC000217628973 CC On-Demand Unstable CA13 52 46 NS(=O)(=O)c1ccc(CNC(=O)C(F)F)cc1 ZINC000217628973 CC On-Demand Unstable CA5B 72 57 NS(=O)(=O)c1ccc(CNC(=O)C(F)F)cc1 ZINC000217628973 CC On-Demand Unstable CA4 134 65 NS(=O)(=O)c1ccc(CNC(=O)C(F)F)cc1 ZINC000217628973 CC On-Demand Unstable CA5A 77 57 NS(=O)(=O)c1ccc(CNC(=O)C(F)F)cc1 ZINC000217628973 CC On-Demand Unstable CA14 72 68 NS(=O)(=O)c1ccc(CNC(=O)C(F)F)cc1 ZINC000217628973 CC On-Demand Unstable CA12 116 64 NS(=O)(=O)c1ccc(CNC(=O)C(F)F)cc1 ZINC000217628973 CC On-Demand Unstable ALPL 15 63 NS(=O)(=O)c1ccc(CNC(=O)C(F)F)cc1 ZINC000217628973 CC On-Demand Unstable CA9 127 64 NS(=O)(=O)c1ccc(CNC(=O)C(F)F)cc1 ZINC000217628973 CC On-Demand Unstable AMP1_PLAFQ 27 40 NS(=O)(=O)c1ccc(CNC(=O)C(F)F)cc1 ZINC000217628973 CC On-Demand Unstable CAH_METTE 46 46 NS(=O)(=O)c1ccc(CNC(=O)C(F)F)cc1 ZINC000217628973 CC On-Demand Unstable CYNT 54 53 NS(=O)(=O)c1ccc(CNC(=O)C(F)F)cc1 ZINC000217628973 CC On-Demand Unstable NCE103 44 49 NS(=O)(=O)c1ccc(CNC(=O)C(F)F)cc1 ZINC000217628973 CC On-Demand Unstable CA15 33 46 NS(=O)(=O)c1ccc(CNC(=O)C(F)F)cc1 ZINC000217628973 CC On-Demand Unstable MTCA1 57 51 NS(=O)(=O)c1ccc(CNC(=O)C(F)F)cc1 ZINC000217628973 CC On-Demand Unstable P96878_MYCTU 72 51 NS(=O)(=O)c1ccc(CNC(=O)C(F)F)cc1 ZINC000217628973 CC On-Demand Unstable CA 0 49 NS(=O)(=O)c1ccc(CNC(=O)C(F)F)cc1 ZINC000217628973 CC On-Demand Unstable NAMPT 58 39 NS(=O)(=O)c1ccc(CNC(=O)C(F)F)cc1 ZINC000217628973 CC On-Demand Unstable A6YCJ1_9METZ 35 48 NS(=O)(=O)c1ccc(CNC(=O)C(F)F)cc1 ZINC000217628973 CC On-Demand Unstable Q5TU56_ANOGA 0 46 COc1ccccc1Oc1ccc(S(=O)(=O)N2CCC[C@@]3(C2)OC(=O)c2ccccc23)cc1 ZINC000217628978 JI For-Sale Unstable NPY5R 17 41 CCC[C@H](C)Nc1ccc(S(=O)(=O)NCc2ccco2)cc1C(=O)O ZINC000217628984 FG In-Stock Unstable CASP3 15 40 COc1ccc2[nH]c3c(c2c1)CCC[C@H]3NC(=O)Cc1c(C)[nH]c2ccccc12 ZINC000217629027 GJ In-Stock Unstable MAPKAPK2 23 46 COc1ccc2[nH]c3c(c2c1)CCC[C@H]3NC(=O)Cc1c(C)[nH]c2ccccc12 ZINC000217629027 GJ In-Stock Unstable MTNR1A 54 38 COc1ccc2[nH]c3c(c2c1)CCC[C@H]3NC(=O)Cc1c(C)[nH]c2ccccc12 ZINC000217629027 GJ In-Stock Unstable MTNR1B 45 38 COc1ccc([C@@H]2SCCN2S(=O)(=O)c2ccc(Br)s2)cc1 ZINC000217629038 HH In-Stock Unstable MMP13 26 40 COc1ccc([C@@H]2SCCN2S(=O)(=O)c2ccc(Br)s2)cc1 ZINC000217629038 HH In-Stock Unstable MMP3 28 40 COc1ccc([C@@H]2SCCN2S(=O)(=O)c2ccc(Br)s2)cc1 ZINC000217629038 HH In-Stock Unstable MMP9 19 40 COc1ccc([C@@H]2SCCN2S(=O)(=O)c2ccc(Br)s2)cc1 ZINC000217629038 HH In-Stock Unstable MMP7 33 40 COc1ccc([C@@H]2SCCN2S(=O)(=O)c2ccc(Br)s2)cc1 ZINC000217629038 HH In-Stock Unstable MMP1 29 40 C[C@@H](Cc1cccnc1)NC(=O)c1ccc(=O)[nH]c1 ZINC000217629084 CD In-Stock Unstable TBXAS1 17 40 C[C@@H](Cc1cccnc1)NC(=O)c1ccc(=O)[nH]c1 ZINC000217629084 CD In-Stock Unstable PTAFR 28 41 COc1ccc(C)cc1NC(=O)C(F)F ZINC000217629102 BE On-Demand Unstable KCNMA1 18 46 COc1ccc(C)cc1NC(=O)C(F)F ZINC000217629102 BE On-Demand Unstable KCNK9 42 39 O=C(O)/C=C\c1cccc(C(=O)Nc2ncccn2)c1 ZINC000217629150 CD For-Sale Anodyne HDAC8 21 50 O=C(O)/C=C\c1cccc(C(=O)Nc2ncccn2)c1 ZINC000217629150 CD For-Sale Anodyne MMP1 0 40 O=C(O)/C=C\c1cccc(C(=O)Nc2ncccn2)c1 ZINC000217629150 CD For-Sale Anodyne KCNK3 90 42 O=C(O)/C=C\c1cccc(C(=O)Nc2ncccn2)c1 ZINC000217629150 CD For-Sale Anodyne KCNK9 42 38 C[C@H](Cc1cccnc1)NC(=O)c1ccc(=O)[nH]c1 ZINC000217629162 CD In-Stock Unstable TBXAS1 17 40 C[C@H](Cc1cccnc1)NC(=O)c1ccc(=O)[nH]c1 ZINC000217629162 CD In-Stock Unstable PTAFR 28 41 O=C(N/C=C/c1ccccc1)Nc1nccs1 ZINC000217629172 BF For-Sale Anodyne MAP 0 50 O=C(N/C=C/c1ccccc1)Nc1nccs1 ZINC000217629172 BF For-Sale Anodyne MAP1 129 43 CCN(C(=O)c1cccc(/C=C\C(=O)O)c1)C1CCCC1 ZINC000217629224 CG For-Sale Unstable ACE 63 49 O=C(C[C@@H]1NC(=O)N(Cc2ccc3c(c2)OCO3)C1=O)N[C@H](CO)c1ccccc1 ZINC000217629235 HD In-Stock Unstable NOS2 77 33 O=C(C[C@@H]1NC(=O)N(Cc2ccc3c(c2)OCO3)C1=O)N[C@H](CO)c1ccccc1 ZINC000217629235 HD In-Stock Unstable MCHR1 21 45 CCOC(=O)CN1C(=O)[C@]2(N[C@H](CCSC)[C@@H]3C(=O)N(Cc4ccccc4)C(=O)[C@@H]32)c2ccccc21 ZINC000217629241 KE In-Stock Unstable EDNRB 40 37 CSc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217629266 CI For-Sale Unstable KCNK3 52 33 CCCNc1ccc(S(=O)(=O)NC[C@@H]2CCCO2)cc1C(=O)O ZINC000217629287 ED In-Stock Unstable BDKRB1 27 41 CC[C@@H](C)[C@@H](CO)NC(=O)Cc1ccc2c(c1)CCC(C)(C)O2 ZINC000217629351 DF In-Stock Unstable NDUFA4 0 42 CC[C@@H](C)[C@@H](CO)NC(=O)Cc1ccc2c(c1)CCC(C)(C)O2 ZINC000217629351 DF In-Stock Unstable DAGLA 22 40 CCc1cc(Br)c(O)c(F)c1OC ZINC000217629354 BF For-Sale Unstable SLC22A12 78 39 COc1cc(/C=C/c2ccccc2)c(C(=O)O)c(OC)c1 ZINC000217629356 CH Annotated Unstable PTGS2 0 55 COc1cc(/C=C/c2ccccc2)c(C(=O)O)c(OC)c1 ZINC000217629356 CH Annotated Unstable CYP1B1 93 60 COc1cc(/C=C/c2ccccc2)c(C(=O)O)c(OC)c1 ZINC000217629356 CH Annotated Unstable P2RX1 0 40 COc1cc(/C=C/c2ccccc2)c(C(=O)O)c(OC)c1 ZINC000217629356 CH Annotated Unstable APP 34 42 COc1cc(/C=C/c2ccccc2)c(C(=O)O)c(OC)c1 ZINC000217629356 CH Annotated Unstable CYP1A1 63 60 COc1cc(/C=C/c2ccccc2)c(C(=O)O)c(OC)c1 ZINC000217629356 CH Annotated Unstable CYP1A2 22 60 COc1cc(/C=C/c2ccccc2)c(C(=O)O)c(OC)c1 ZINC000217629356 CH Annotated Unstable ALS 70 37 COc1cc(/C=C/c2ccccc2)c(C(=O)O)c(OC)c1 ZINC000217629356 CH Annotated Unstable TLR4 19 40 COc1cc(/C=C/c2ccccc2)c(C(=O)O)c(OC)c1 ZINC000217629356 CH Annotated Unstable AKR1C3 15 40 COc1cc(/C=C/c2ccccc2)c(C(=O)O)c(OC)c1 ZINC000217629356 CH Annotated Unstable ABCG2 22 48 COc1cc(/C=C/c2ccccc2)c(C(=O)O)c(OC)c1 ZINC000217629356 CH Annotated Unstable CYSP_PLAFA 49 36 CCCNc1ccc(S(=O)(=O)NC[C@H]2CCCO2)cc1C(=O)O ZINC000217629380 ED In-Stock Unstable BDKRB1 27 41 CS(=O)(=O)NCCNC(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217629381 DC For-Sale Unstable CA2 15 41 O=C(N/C=C/c1ccccc1)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217629386 HG For-Sale Unstable LPL 57 47 O=C(N/C=C/c1ccccc1)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217629386 HG For-Sale Unstable F13A1 50 36 O=C(N/C=C/c1ccccc1)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217629386 HG For-Sale Unstable LIPG 23 47 CCOC(=O)[C@@H]1CCCN(C(=O)C(F)F)C1 ZINC000217629391 BD On-Demand Unstable RHODESAIN 0 46 CCOC(=O)[C@H]1CCCN(C(=O)C(F)F)C1 ZINC000217629463 BD On-Demand Unstable RHODESAIN 0 46 COc1cc2c(c(OC)c1OC)-c1ccc(NCCCCCC(=O)NCc3ccncc3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217629473 KJ In-Stock Unstable TUBA1A 18 64 CC(C)Nc1ccc(S(=O)(=O)NC[C@@H]2CCCO2)cc1C(=O)O ZINC000217629490 ED In-Stock Unstable BDKRB1 22 42 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217629495 ED For-Sale Unstable CA2 149 64 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217629495 ED For-Sale Unstable CA6 24 40 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217629495 ED For-Sale Unstable CA1 123 64 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217629495 ED For-Sale Unstable CA7 68 59 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217629495 ED For-Sale Unstable CA13 32 40 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217629495 ED For-Sale Unstable CA5B 64 59 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217629495 ED For-Sale Unstable CA4 106 64 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217629495 ED For-Sale Unstable CA5A 68 59 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217629495 ED For-Sale Unstable CA14 53 59 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217629495 ED For-Sale Unstable CA12 90 60 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217629495 ED For-Sale Unstable CA9 103 60 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217629495 ED For-Sale Unstable CAH_METTE 28 40 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217629495 ED For-Sale Unstable CYNT 31 46 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217629495 ED For-Sale Unstable NCE103 46 45 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217629495 ED For-Sale Unstable CA15 18 40 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217629495 ED For-Sale Unstable MTCA1 49 60 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217629495 ED For-Sale Unstable P96878_MYCTU 64 60 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217629495 ED For-Sale Unstable CA 0 42 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217629495 ED For-Sale Unstable NAMPT 52 43 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217629495 ED For-Sale Unstable A6YCJ1_9METZ 24 41 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217629495 ED For-Sale Unstable Q5TU56_ANOGA 0 40 O=C1O[C@@]2(CCCN(S(=O)(=O)c3c(Cl)cccc3Cl)C2)c2ccccc21 ZINC000217629505 HH For-Sale Unstable NPY5R 24 40 CCCCS(=O)(=O)Nc1ccc(/C=C\C(=O)O)cc1C ZINC000217629568 CF For-Sale Unstable AKR1C3 0 41 CC(C)Nc1ccc(S(=O)(=O)NC[C@H]2CCCO2)cc1C(=O)O ZINC000217629569 ED In-Stock Unstable BDKRB1 22 42 COC(=O)C[C@H](c1ccccc1OCc1ccccn1)c1c(O)c2ccccc2oc1=O ZINC000217629587 II In-Stock Unstable NQO1 29 46 COC(=O)[C@@]1(N)C[C@@H]1Br ZINC000217629593 AC For-Sale Unstable CPT1 54 29 O=C1O[C@]2(CCCN(S(=O)(=O)c3c(Cl)cccc3Cl)C2)c2ccccc21 ZINC000217629595 HH For-Sale Unstable NPY5R 24 40 N#Cc1cc2c(nc1N1CCN(S(=O)(=O)c3cc(Cl)ccc3Cl)CC1)CCCC2 ZINC000217629597 JH On-Demand Unstable TRPV4 47 38 O=C(N/C=C/c1ccccc1)Nc1cccnc1Cl ZINC000217629606 CH For-Sale Anodyne G2YM83_BOTF4 67 34 COC(=O)C[C@@H](c1ccccc1OCc1ccccn1)c1c(O)c2ccccc2oc1=O ZINC000217629666 II In-Stock Unstable NQO1 29 46 COC(=O)[C@@]1(N)C[C@H]1Br ZINC000217629669 AC For-Sale Unstable CPT1 54 29 CCCCNc1ccc(S(=O)(=O)NC[C@@H]2CCCO2)cc1C(=O)O ZINC000217629673 FE In-Stock Unstable BDKRB1 27 40 Cc1cc(N2CCN(Cc3cccc(C#N)c3)C[C@@H](O)C2)nc(N)n1 ZINC000217629688 EC In-Stock Unstable HRH4 22 40 Cc1ccc(-c2ccc(S(=O)(=O)N3CCC[C@]4(C3)OC(=O)c3ccccc34)cc2)cc1 ZINC000217629705 IJ For-Sale Unstable NPY5R 25 40 C[C@@H]1C[C@@H](C)CN(C(=O)N/C=C/c2ccccc2)C1 ZINC000217629713 CG For-Sale Unstable RBP4 41 31 N#Cc1cc2c(nc1N1CCN(S(=O)(=O)c3ccc(Cl)c(C(F)(F)F)c3)CC1)CCCC2 ZINC000217629722 JI On-Demand Unstable GCK 45 37 CCCCNc1ccc(S(=O)(=O)NC[C@H]2CCCO2)cc1C(=O)O ZINC000217629771 FE In-Stock Unstable BDKRB1 27 40 Cc1ccc(-c2ccc(S(=O)(=O)N3CCC[C@@]4(C3)OC(=O)c3ccccc34)cc2)cc1 ZINC000217629788 IJ For-Sale Unstable NPY5R 25 40 C[C@H]1C[C@@H](C)CN(C(=O)N/C=C/c2ccccc2)C1 ZINC000217629802 CG For-Sale Unstable RBP4 41 31 COC(=O)c1ccnc(C2CCCCC2)c1 ZINC000217629808 BF In-Stock Unstable KDM4C 0 55 COC(=O)c1ccnc(C2CCCCC2)c1 ZINC000217629808 BF In-Stock Unstable KDM3A 0 55 COC(=O)c1ccnc(C2CCCCC2)c1 ZINC000217629808 BF In-Stock Unstable KDM5C 0 55 C[C@H]1C[C@H](C)CN(C(=O)N/C=C/c2ccccc2)C1 ZINC000217629895 CG For-Sale Unstable RBP4 41 31 O=C1O[C@@]2(CCCN(S(=O)(=O)c3ccc(-c4ccc(F)cc4)cc3)C2)c2ccccc21 ZINC000217629901 II For-Sale Unstable NPY5R 29 46 CC(C)CNc1ccc(S(=O)(=O)NC[C@@H]2CCCO2)cc1C(=O)O ZINC000217629905 FD In-Stock Unstable BDKRB1 0 41 O=C1O[C@]2(CCCN(S(=O)(=O)c3ccc(-c4ccc(F)cc4)cc3)C2)c2ccccc21 ZINC000217629980 II For-Sale Unstable NPY5R 29 46 CC(C)CNc1ccc(S(=O)(=O)NC[C@H]2CCCO2)cc1C(=O)O ZINC000217629989 FD In-Stock Unstable BDKRB1 0 41 CS(=O)(=O)c1ccc(OC/C=C\CN)cc1 ZINC000217630069 BC For-Sale Unstable CA7 17 47 CS(=O)(=O)c1ccc(OC/C=C\CN)cc1 ZINC000217630069 BC For-Sale Unstable LOX1.1 46 33 CS(=O)(=O)c1ccc(OC/C=C\CN)cc1 ZINC000217630069 BC For-Sale Unstable O49150_SOLTU 50 34 Cc1ccc(NC(=O)C(F)F)cc1F ZINC000217630101 BE On-Demand Unstable FPR2 21 45 Cc1ccc(NC(=O)C(F)F)cc1F ZINC000217630101 BE On-Demand Unstable LEF 78 37 COc1ccc(-c2ccc(S(=O)(=O)N3CCC[C@]4(C3)OC(=O)c3ccccc34)cc2)cc1 ZINC000217630113 II For-Sale Unstable NPY5R 27 49 CC[C@@H](C)Nc1ccc(S(=O)(=O)NC[C@@H]2CCCO2)cc1C(=O)O ZINC000217630121 FE In-Stock Unstable BDKRB1 21 41 FC(F)(F)Oc1ccccc1-c1cccc(C(F)(F)F)c1Cl ZINC000217630129 EK For-Sale Anodyne TRPA1 15 41 O=[N+]([O-])c1cccc(CN[C@@H]2CCN3CCCC[C@@H]23)c1 ZINC000217630138 CE On-Demand Unstable CACNA1D 52 36 CCc1c(C(=O)O)cc(Cl)c(OC)c1OC ZINC000217630153 BF For-Sale Unstable AKR1C2 45 33 CCc1c(C(=O)O)cc(Cl)c(OC)c1OC ZINC000217630153 BF For-Sale Unstable AKR1C1 41 33 CS(=O)(=O)c1cccc(OC/C=C\CN)c1 ZINC000217630188 BC For-Sale Unstable NR1H3 42 36 CS(=O)(=O)c1cccc(OC/C=C\CN)c1 ZINC000217630188 BC For-Sale Unstable AO-ACHE 0 40 COc1ccc(-c2ccc(S(=O)(=O)N3CCC[C@@]4(C3)OC(=O)c3ccccc34)cc2)cc1 ZINC000217630206 II For-Sale Unstable NPY5R 27 49 CC[C@H](C)Nc1ccc(S(=O)(=O)NC[C@@H]2CCCO2)cc1C(=O)O ZINC000217630209 FE In-Stock Unstable BDKRB1 21 41 O=[N+]([O-])c1cccc(CN[C@H]2CCN3CCCC[C@@H]23)c1 ZINC000217630218 CE On-Demand Unstable CACNA1D 52 36 CSC[C@@](C)(O)CNC(=O)c1ccc(C(C)C)cc1 ZINC000217630247 CF On-Demand Unstable ECR 33 42 COc1ccc(/C=C\C(=O)O)cc1N1C(=O)[C@H]2C[C@H]2C1=O ZINC000217630249 CD For-Sale Unstable TUBB1 42 38 COc1ccc(/C=C\C(=O)O)cc1N1C(=O)[C@H]2C[C@H]2C1=O ZINC000217630249 CD For-Sale Unstable ABCG2 15 43 O=C(N[C@@H]1CCCc2ccccc21)C(F)F ZINC000217630259 BE On-Demand Unstable BDKRB1 43 39 O=C(N[C@@H]1CCCc2ccccc21)C(F)F ZINC000217630259 BE On-Demand Unstable KCNN3 18 41 O=C(N[C@@H]1CCCc2ccccc21)C(F)F ZINC000217630259 BE On-Demand Unstable TSPAN17 0 40 O=C(N[C@@H]1CCCc2ccccc21)C(F)F ZINC000217630259 BE On-Demand Unstable XIAP 24 44 O=C(N[C@@H]1CCCc2ccccc21)C(F)F ZINC000217630259 BE On-Demand Unstable BIRC3 43 48 O=C(N[C@@H]1CCCc2ccccc21)C(F)F ZINC000217630259 BE On-Demand Unstable BIRC2 54 48 CC[C@@H](C)Nc1ccc(S(=O)(=O)NC[C@H]2CCCO2)cc1C(=O)O ZINC000217630292 FE In-Stock Unstable BDKRB1 21 41 O=C(Nc1ccc2c(c1)OCO2)N1CCS[C@@H]1c1ccccc1F ZINC000217630326 EH In-Stock Unstable TRPC6 41 39 O=C(Nc1ccc2c(c1)OCO2)N1CCS[C@@H]1c1ccccc1F ZINC000217630326 EH In-Stock Unstable TRPC3 41 39 CSC[C@](C)(O)CNC(=O)c1ccc(C(C)C)cc1 ZINC000217630327 CF On-Demand Unstable ECR 33 42 COc1ccc(/C=C\C(=O)O)cc1N1C(=O)[C@H]2C[C@@H]2C1=O ZINC000217630330 CD For-Sale Unstable TUBB1 42 38 COc1ccc(/C=C\C(=O)O)cc1N1C(=O)[C@H]2C[C@@H]2C1=O ZINC000217630330 CD For-Sale Unstable ABCG2 15 43 O=C(O)c1ccnc([C@@H]2CCCC23SCCS3)c1 ZINC000217630335 CG In-Stock Unstable FTO 0 40 O=C(N[C@H]1CCCc2ccccc21)C(F)F ZINC000217630337 BE On-Demand Unstable BDKRB1 43 39 O=C(N[C@H]1CCCc2ccccc21)C(F)F ZINC000217630337 BE On-Demand Unstable KCNN3 18 41 O=C(N[C@H]1CCCc2ccccc21)C(F)F ZINC000217630337 BE On-Demand Unstable TSPAN17 0 40 O=C(N[C@H]1CCCc2ccccc21)C(F)F ZINC000217630337 BE On-Demand Unstable XIAP 24 44 O=C(N[C@H]1CCCc2ccccc21)C(F)F ZINC000217630337 BE On-Demand Unstable BIRC3 43 48 O=C(N[C@H]1CCCc2ccccc21)C(F)F ZINC000217630337 BE On-Demand Unstable BIRC2 54 48 CC[C@H](C)Nc1ccc(S(=O)(=O)NC[C@H]2CCCO2)cc1C(=O)O ZINC000217630370 FE In-Stock Unstable BDKRB1 21 41 O=C(Nc1ccc2c(c1)OCO2)N1CCS[C@H]1c1ccccc1F ZINC000217630414 EH In-Stock Unstable TRPC6 41 39 O=C(Nc1ccc2c(c1)OCO2)N1CCS[C@H]1c1ccccc1F ZINC000217630414 EH In-Stock Unstable TRPC3 41 39 O=C(O)c1ccnc([C@H]2CCCC23SCCS3)c1 ZINC000217630422 CG In-Stock Unstable FTO 0 40 CCc1c(OC)c(OC)cc(Cl)c1C(=O)O ZINC000217630473 BF For-Sale Unstable ALS 42 36 CC(C)(C)Nc1ccc(S(=O)(=O)NC[C@@H]2CCCO2)cc1C(=O)O ZINC000217630493 FE In-Stock Unstable BDKRB1 22 42 O=C1O[C@@]2(CCCN(S(=O)(=O)c3ccc(Br)cc3)C2)c2ccccc21 ZINC000217630507 HG For-Sale Unstable NPY5R 22 42 O=C(CC[C@@H]1NC(=O)N(Cc2ccccc2)C1=O)NCCc1ccc(O)cc1 ZINC000217630513 GD In-Stock Unstable NCE103 21 44 O=C(CC[C@@H]1NC(=O)N(Cc2ccccc2)C1=O)NCCc1ccc(O)cc1 ZINC000217630513 GD In-Stock Unstable P96878_MYCTU 16 44 O=C(CC[C@@H]1NC(=O)N(Cc2ccccc2)C1=O)NCCc1ccc(O)cc1 ZINC000217630513 GD In-Stock Unstable CAN2 0 44 NC/C=C\COc1cc([N+](=O)[O-])ccc1Cl ZINC000217630544 BE For-Sale Unstable SNCA 46 39 O=[N+]([O-])c1ccccc1CN[C@@H]1CCN2CCCC[C@@H]12 ZINC000217630557 CE For-Sale Unstable COLA 91 33 O=C1O[C@]2(CCCN(S(=O)(=O)c3ccc(Br)cc3)C2)c2ccccc21 ZINC000217630571 HG For-Sale Unstable NPY5R 22 42 CC(C)(C)Nc1ccc(S(=O)(=O)NC[C@H]2CCCO2)cc1C(=O)O ZINC000217630584 FE In-Stock Unstable BDKRB1 22 42 COc1cc(Cl)c(OC)c(C(C)=O)c1OC ZINC000217630586 BF For-Sale Unstable TUBB1 48 37 O=[N+]([O-])c1ccccc1CN[C@H]1CCN2CCCC[C@@H]12 ZINC000217630636 CE For-Sale Unstable COLA 91 33 O=C1O[C@@]2(CCCN(S(=O)(=O)c3ccccc3C(F)(F)F)C2)c2ccccc21 ZINC000217630680 HH For-Sale Unstable NPY5R 26 48 C=CCNc1ccc(S(=O)(=O)NC[C@@H]2CCCO2)cc1C(=O)O ZINC000217630684 ED In-Stock Unstable BDKRB1 22 42 COc1cc(Cl)c(C(C)=O)c(OC)c1OC ZINC000217630697 BF For-Sale Unstable TUBB1 43 34 N#Cc1cccc(C(=O)N2CCS[C@@H]2c2ccc(C(F)(F)F)cc2)c1 ZINC000217630709 FI In-Stock Unstable TRPM8 39 45 CCNC(=O)N/C=C/c1ccccc1 ZINC000217630742 AD For-Sale Unstable 17HSDCL 44 37 O=C(O)/C=C\c1cccc(C(=O)NC2CCC(O)CC2)c1 ZINC000217630749 CD For-Sale Unstable HDAC8 34 44 O=C(O)/C=C\c1cccc(C(=O)NC2CCC(O)CC2)c1 ZINC000217630749 CD For-Sale Unstable HDAC6 21 44 C=CCNc1ccc(S(=O)(=O)NC[C@H]2CCCO2)cc1C(=O)O ZINC000217630762 ED In-Stock Unstable BDKRB1 22 42 O=C1O[C@]2(CCCN(S(=O)(=O)c3ccccc3C(F)(F)F)C2)c2ccccc21 ZINC000217630773 HH For-Sale Unstable NPY5R 26 48 N#Cc1cccc(C(=O)N2CCS[C@H]2c2ccc(C(F)(F)F)cc2)c1 ZINC000217630788 FI In-Stock Unstable TRPM8 39 45 COc1cc(C(C)=O)c(OC)c(Cl)c1OC ZINC000217630804 BF For-Sale Unstable TUBB1 42 34 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccc2F)c1 ZINC000217630826 CG For-Sale Anodyne HDAC8 16 51 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccc2F)c1 ZINC000217630826 CG For-Sale Anodyne MMP2 0 58 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccc2F)c1 ZINC000217630826 CG For-Sale Anodyne NR1H4 0 40 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccc2F)c1 ZINC000217630826 CG For-Sale Anodyne HDAC1 0 43 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccc2F)c1 ZINC000217630826 CG For-Sale Anodyne MMP9 0 58 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccc2F)c1 ZINC000217630826 CG For-Sale Anodyne MMP1 0 58 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccc2F)c1 ZINC000217630826 CG For-Sale Anodyne FABH 0 48 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccc2F)c1 ZINC000217630826 CG For-Sale Anodyne RHOA 0 40 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccc2F)c1 ZINC000217630826 CG For-Sale Anodyne KCNK3 94 42 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccc2F)c1 ZINC000217630826 CG For-Sale Anodyne KCNK9 47 39 CCCCN(CCC)C(=O)N/C=C/c1ccccc1 ZINC000217630847 CH For-Sale Unstable TSPO 43 39 NNC(=O)c1ccnc(C2CCCC2)c1 ZINC000217630854 BD In-Stock Unstable KDM4E 33 40 O=C(O)c1cc(S(=O)(=O)NC[C@@H]2CCCO2)ccc1NC1CC1 ZINC000217630871 ED In-Stock Unstable BDKRB1 22 45 N#Cc1ccccc1S(=O)(=O)N1CCC[C@]2(C1)OC(=O)c1ccccc12 ZINC000217630892 FE For-Sale Unstable NPY5R 23 41 O=C(c1cc2ccccc2o1)N1CCS[C@@H]1c1ccc(C(F)(F)F)cc1 ZINC000217630899 GK In-Stock Unstable TRPM8 40 35 Cc1sc(CCC(=O)O)cc1Br ZINC000217630900 BF For-Sale Unstable THRB 18 40 COc1cc(OC)c(C(C)=O)c(Cl)c1OC ZINC000217630914 BF For-Sale Unstable TUBB1 43 35 O=C(O)c1cc(S(=O)(=O)NC[C@H]2CCCO2)ccc1NC1CC1 ZINC000217630947 ED In-Stock Unstable BDKRB1 22 45 CCCCCNC(=O)N/C=C/c1ccccc1 ZINC000217630950 BG For-Sale Unstable EPHX2 19 48 CCCCCNC(=O)N/C=C/c1ccccc1 ZINC000217630950 BG For-Sale Unstable HDAC9 27 43 CCCCCNC(=O)N/C=C/c1ccccc1 ZINC000217630950 BG For-Sale Unstable HDAC7 21 43 CCCCCNC(=O)N/C=C/c1ccccc1 ZINC000217630950 BG For-Sale Unstable AMP1_PLAFQ 28 43 CCCCCNC(=O)N/C=C/c1ccccc1 ZINC000217630950 BG For-Sale Unstable ASAH1 88 39 CCCCCNC(=O)N/C=C/c1ccccc1 ZINC000217630950 BG For-Sale Unstable ACAT 0 48 CCCCCNC(=O)N/C=C/c1ccccc1 ZINC000217630950 BG For-Sale Unstable TRPM2 0 41 CN1CCCC[C@@H]1CNC(=O)[C@@H](Cl)c1ccccc1 ZINC000217630953 CF For-Sale Unstable DRD2 36 40 CN1CCCC[C@@H]1CNC(=O)[C@@H](Cl)c1ccccc1 ZINC000217630953 CF For-Sale Unstable SLC6A1 82 39 CN1CCCC[C@@H]1CNC(=O)[C@@H](Cl)c1ccccc1 ZINC000217630953 CF For-Sale Unstable DRD3 22 40 CN1CCCC[C@@H]1CNC(=O)[C@@H](Cl)c1ccccc1 ZINC000217630953 CF For-Sale Unstable SLC6A3 21 48 CN1CCCC[C@@H]1CNC(=O)[C@@H](Cl)c1ccccc1 ZINC000217630953 CF For-Sale Unstable SLC18A2 49 38 CN1CCCC[C@@H]1CNC(=O)[C@@H](Cl)c1ccccc1 ZINC000217630953 CF For-Sale Unstable HCRTR1 19 41 CN1CCCC[C@@H]1CNC(=O)[C@@H](Cl)c1ccccc1 ZINC000217630953 CF For-Sale Unstable KCNQ2 47 36 CN1CCCC[C@@H]1CNC(=O)[C@@H](Cl)c1ccccc1 ZINC000217630953 CF For-Sale Unstable CHRNA10 52 40 CN1CCCC[C@@H]1CNC(=O)[C@@H](Cl)c1ccccc1 ZINC000217630953 CF For-Sale Unstable HCRTR2 0 41 CN1CCCC[C@@H]1CNC(=O)[C@@H](Cl)c1ccccc1 ZINC000217630953 CF For-Sale Unstable XIAP 42 35 CN1CCCC[C@@H]1CNC(=O)[C@@H](Cl)c1ccccc1 ZINC000217630953 CF For-Sale Unstable ACKR3 64 35 N#Cc1ccccc1S(=O)(=O)N1CCC[C@@]2(C1)OC(=O)c1ccccc12 ZINC000217630980 FE For-Sale Unstable NPY5R 23 41 O=C(c1cc2ccccc2o1)N1CCS[C@H]1c1ccc(C(F)(F)F)cc1 ZINC000217630989 GK In-Stock Unstable TRPM8 40 35 COc1c(OCC(=O)O)cc(C)c(Cl)c1C ZINC000217631021 BE For-Sale Unstable PPARD 40 37 CN1CCCC[C@H]1CNC(=O)[C@@H](Cl)c1ccccc1 ZINC000217631037 CF For-Sale Unstable DRD2 36 40 CN1CCCC[C@H]1CNC(=O)[C@@H](Cl)c1ccccc1 ZINC000217631037 CF For-Sale Unstable SLC6A1 82 39 CN1CCCC[C@H]1CNC(=O)[C@@H](Cl)c1ccccc1 ZINC000217631037 CF For-Sale Unstable DRD3 22 40 CN1CCCC[C@H]1CNC(=O)[C@@H](Cl)c1ccccc1 ZINC000217631037 CF For-Sale Unstable SLC6A3 21 48 CN1CCCC[C@H]1CNC(=O)[C@@H](Cl)c1ccccc1 ZINC000217631037 CF For-Sale Unstable SLC18A2 49 38 CN1CCCC[C@H]1CNC(=O)[C@@H](Cl)c1ccccc1 ZINC000217631037 CF For-Sale Unstable HCRTR1 19 41 CN1CCCC[C@H]1CNC(=O)[C@@H](Cl)c1ccccc1 ZINC000217631037 CF For-Sale Unstable KCNQ2 47 36 CN1CCCC[C@H]1CNC(=O)[C@@H](Cl)c1ccccc1 ZINC000217631037 CF For-Sale Unstable CHRNA10 52 40 CN1CCCC[C@H]1CNC(=O)[C@@H](Cl)c1ccccc1 ZINC000217631037 CF For-Sale Unstable HCRTR2 0 41 CN1CCCC[C@H]1CNC(=O)[C@@H](Cl)c1ccccc1 ZINC000217631037 CF For-Sale Unstable XIAP 42 35 CN1CCCC[C@H]1CNC(=O)[C@@H](Cl)c1ccccc1 ZINC000217631037 CF For-Sale Unstable ACKR3 64 35 O=C(O)c1cc(S(=O)(=O)NC[C@@H]2CCCO2)ccc1NC1CCCC1 ZINC000217631062 FE In-Stock Unstable BDKRB1 21 42 C[C@@H]1CCCC[C@@H]1NC(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217631064 CG For-Sale Unstable SSTR3 26 43 O=C(N/C=C/c1ccccc1)Nc1ccccc1 ZINC000217631074 BG For-Sale Anodyne EPHX1 0 57 O=C(N/C=C/c1ccccc1)Nc1ccccc1 ZINC000217631074 BG For-Sale Anodyne PFHDAC1 0 42 O=C(N/C=C/c1ccccc1)Nc1ccccc1 ZINC000217631074 BG For-Sale Anodyne P95276_MYCTO 0 57 CSC[C@@](C)(O)CNC(=O)c1cn2ccccc2n1 ZINC000217631079 CD On-Demand Unstable MAP3K5 52 34 C[C@@H](N[C@@H]1CCC[C@@H](O)C1)c1ccc(OC(F)(F)F)cc1 ZINC000217631109 DH For-Sale Unstable EPHX2 24 42 O=C(O)c1cc(S(=O)(=O)NC[C@H]2CCCO2)ccc1NC1CCCC1 ZINC000217631144 FE In-Stock Unstable BDKRB1 21 42 C[C@H]1CCCC[C@@H]1NC(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217631149 CG For-Sale Unstable SSTR3 26 43 CSC[C@](C)(O)CNC(=O)c1cn2ccccc2n1 ZINC000217631164 CD On-Demand Unstable MAP3K5 52 34 CCOC(=O)[C@@H]1CCCN(C(=O)N/C=C/c2ccccc2)C1 ZINC000217631174 DF For-Sale Unstable CHRM1 15 42 CCOC(=O)[C@@H]1CCCN(C(=O)N/C=C/c2ccccc2)C1 ZINC000217631174 DF For-Sale Unstable SLC6A1 112 37 CCOC(=O)[C@@H]1CCCN(C(=O)N/C=C/c2ccccc2)C1 ZINC000217631174 DF For-Sale Unstable FDFT1 33 41 CCOC(=O)[C@@H]1CCCN(C(=O)N/C=C/c2ccccc2)C1 ZINC000217631174 DF For-Sale Unstable PREP 43 37 C[C@H](N[C@@H]1CCC[C@@H](O)C1)c1ccc(OC(F)(F)F)cc1 ZINC000217631192 DH On-Demand Unstable EPHX2 24 42 O=C(c1ccc(Cl)s1)N1CCS[C@H]1c1ccc(C(F)(F)F)cc1 ZINC000217631194 GK In-Stock Unstable TRPM8 42 34 COc1cccc(N2CCN(C/C=C\CN)CC2)c1 ZINC000217631206 CD For-Sale Unstable HTR1A 31 60 COc1cccc(N2CCN(C/C=C\CN)CC2)c1 ZINC000217631206 CD For-Sale Unstable DRD2 22 60 COc1cccc(N2CCN(C/C=C\CN)CC2)c1 ZINC000217631206 CD For-Sale Unstable DRD4 50 40 COc1cccc(N2CCN(C/C=C\CN)CC2)c1 ZINC000217631206 CD For-Sale Unstable DRD3 25 44 COc1cccc(N2CCN(C/C=C\CN)CC2)c1 ZINC000217631206 CD For-Sale Unstable HTR7 26 46 CCOC(=O)[C@H]1CCCN(C(=O)N/C=C/c2ccccc2)C1 ZINC000217631247 DF For-Sale Unstable CHRM1 15 42 CCOC(=O)[C@H]1CCCN(C(=O)N/C=C/c2ccccc2)C1 ZINC000217631247 DF For-Sale Unstable SLC6A1 112 37 CCOC(=O)[C@H]1CCCN(C(=O)N/C=C/c2ccccc2)C1 ZINC000217631247 DF For-Sale Unstable FDFT1 33 41 CCOC(=O)[C@H]1CCCN(C(=O)N/C=C/c2ccccc2)C1 ZINC000217631247 DF For-Sale Unstable PREP 43 37 O=C(O)c1cc(S(=O)(=O)NC[C@@H]2CCCO2)ccc1NC1CCCCC1 ZINC000217631254 GF In-Stock Unstable BDKRB1 21 42 C[C@@H](N[C@H]1CCC[C@@H](O)C1)c1ccc(OC(F)(F)F)cc1 ZINC000217631276 DH For-Sale Unstable EPHX2 24 42 O=C1O[C@@]2(CCCN(S(=O)(=O)Cc3cccc(C(F)(F)F)c3)C2)c2ccccc21 ZINC000217631293 IH For-Sale Unstable NPY5R 21 45 O=C1C[C@@H](c2ccc(O)c(Cl)c2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217631326 JJ In-Stock Unstable AKR1B1 0 43 O=C1C[C@@H](c2ccc(O)c(Cl)c2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217631326 JJ In-Stock Unstable CYP1B1 19 41 O=C1C[C@@H](c2ccc(O)c(Cl)c2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217631326 JJ In-Stock Unstable CYP1A1 18 41 O=C(O)c1cc(S(=O)(=O)NC[C@H]2CCCO2)ccc1NC1CCCCC1 ZINC000217631328 GF In-Stock Unstable BDKRB1 21 42 c1ccc(CCCN[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217631357 CF For-Sale Unstable FKBP1A 31 43 c1ccc(CCCN[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217631357 CF For-Sale Unstable SIGMAR1 35 52 c1ccc(CCCN[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217631357 CF For-Sale Unstable SLC18A3 37 51 C[C@H](N[C@H]1CCC[C@@H](O)C1)c1ccc(OC(F)(F)F)cc1 ZINC000217631358 DH On-Demand Unstable EPHX2 24 42 CC(C)(C)OC(=O)N1CCC(O)(Cc2cccnc2)CC1 ZINC000217631365 CE For-Sale Unstable GPR119 45 44 O=C(O)Cc1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217631367 CG For-Sale Unstable P95276_MYCTO 0 41 O=C1O[C@]2(CCCN(S(=O)(=O)Cc3cccc(C(F)(F)F)c3)C2)c2ccccc21 ZINC000217631373 IH For-Sale Unstable NPY5R 21 45 O=C(CCN1CCN(Cc2cc(=O)n3ccsc3n2)CC1)Nc1ccccc1Cl ZINC000217631384 IF On-Demand Unstable HTR7 19 40 O=C(CCN1CCN(Cc2cc(=O)n3ccsc3n2)CC1)Nc1ccccc1Cl ZINC000217631384 IF On-Demand Unstable EPHB3 41 32 O=C1C[C@H](c2ccc(O)c(Cl)c2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217631407 JJ In-Stock Unstable AKR1B1 0 43 O=C1C[C@H](c2ccc(O)c(Cl)c2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217631407 JJ In-Stock Unstable CYP1B1 19 41 O=C1C[C@H](c2ccc(O)c(Cl)c2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217631407 JJ In-Stock Unstable CYP1A1 18 41 Cc1c(NN)nc(C2CC2)nc1N[C@@H]1CCN2CCC[C@@H]12 ZINC000217631426 CD For-Sale Unstable CHRM3 19 43 c1ccc(CCCN[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217631450 CF For-Sale Unstable FKBP1A 31 43 c1ccc(CCCN[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217631450 CF For-Sale Unstable SIGMAR1 35 52 c1ccc(CCCN[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217631450 CF For-Sale Unstable SLC18A3 37 51 CSC[C@@](C)(O)CNC(=O)CCn1ccnc1 ZINC000217631469 CC On-Demand Unstable TBXAS1 28 42 CC(C)c1nccn1CCCNC(=O)[C@@H]1CC[C@H](O)CC1 ZINC000217631484 CE In-Stock Unstable TBK1 42 32 CN[C@@H]1CC[C@@H](C)C[C@@H]1CCCc1ccccc1 ZINC000217631485 BI For-Sale Unstable SLC18A2 43 44 CN[C@@H]1CC[C@@H](C)C[C@@H]1CCCc1ccccc1 ZINC000217631485 BI For-Sale Unstable SIGMAR1 15 40 O=C(N/C=C/c1ccccc1)NCc1ccc(C(=O)O)cc1 ZINC000217631503 CF For-Sale Unstable AMP1_PLAFQ 33 42 Cc1c(NN)nc(C2CC2)nc1N[C@H]1CCN2CCC[C@@H]12 ZINC000217631516 CD For-Sale Unstable CHRM3 19 43 NC/C=C\CN1CCC(N2CCCCC2)CC1 ZINC000217631540 BD For-Sale Unstable L3MBTL3 52 35 CSC[C@](C)(O)CNC(=O)CCn1ccnc1 ZINC000217631546 CC On-Demand Unstable TBXAS1 28 42 CN[C@H]1CC[C@@H](C)C[C@@H]1CCCc1ccccc1 ZINC000217631566 BI For-Sale Unstable SLC18A2 43 44 CN[C@H]1CC[C@@H](C)C[C@@H]1CCCc1ccccc1 ZINC000217631566 BI For-Sale Unstable SIGMAR1 15 40 O=C(c1ccc2nsnc2c1)N1CCS[C@H]1c1ccc(C(F)(F)F)cc1 ZINC000217631595 GJ In-Stock Unstable TRPM8 40 36 C[C@H]1C(=O)NN=C2COc3ccc(N)cc3N21 ZINC000217631596 BC For-Sale Unstable PRKCQ 24 57 O=C(O)c1cc(S(=O)(=O)NC[C@@H]2CCCO2)ccc1NCCO ZINC000217631617 EC In-Stock Unstable BDKRB1 0 42 C[C@H]1CN(C[C@H](C)C(=O)c2ccccc2)CCCO1 ZINC000217631641 CF For-Sale Unstable SLC6A1 43 34 C[C@H]1CN(C[C@H](C)C(=O)c2ccccc2)CCCO1 ZINC000217631641 CF For-Sale Unstable FABP4 44 36 CN[C@@H]1CC[C@H](C)C[C@@H]1CCCc1ccccc1 ZINC000217631654 BI For-Sale Unstable SLC18A2 43 44 CN[C@@H]1CC[C@H](C)C[C@@H]1CCCc1ccccc1 ZINC000217631654 BI For-Sale Unstable SIGMAR1 15 40 O=C1O[C@@]2(CCCN(S(=O)(=O)c3cccc(-c4ccccc4)c3)C2)c2ccccc21 ZINC000217631686 HI For-Sale Unstable NPY5R 31 43 Cn1nc(-c2ccc(F)cc2)cc1C(=O)N1CCS[C@@H]1c1ccc(C(F)(F)F)cc1 ZINC000217631697 IK In-Stock Unstable TACR1 40 35 Cn1nc(-c2ccc(F)cc2)cc1C(=O)N1CCS[C@@H]1c1ccc(C(F)(F)F)cc1 ZINC000217631697 IK In-Stock Unstable TRPM8 42 40 O=C(O)c1cc(S(=O)(=O)NC[C@H]2CCCO2)ccc1NCCO ZINC000217631700 EC In-Stock Unstable BDKRB1 0 42 CN[C@H]1CC[C@H](C)C[C@@H]1CCCc1ccccc1 ZINC000217631729 BI For-Sale Unstable SLC18A2 43 44 CN[C@H]1CC[C@H](C)C[C@@H]1CCCc1ccccc1 ZINC000217631729 BI For-Sale Unstable SIGMAR1 15 40 Cn1cc(NC(=O)c2ccc(/C=C\C(=O)O)cc2)cn1 ZINC000217631730 CD For-Sale Unstable PRNP 45 35 O=C1O[C@]2(CCCN(S(=O)(=O)c3cccc(-c4ccccc4)c3)C2)c2ccccc21 ZINC000217631764 HI For-Sale Unstable NPY5R 31 43 Cn1nc(-c2ccc(F)cc2)cc1C(=O)N1CCS[C@H]1c1ccc(C(F)(F)F)cc1 ZINC000217631787 IK In-Stock Unstable TACR1 40 35 Cn1nc(-c2ccc(F)cc2)cc1C(=O)N1CCS[C@H]1c1ccc(C(F)(F)F)cc1 ZINC000217631787 IK In-Stock Unstable TRPM8 42 40 O=C(O)c1cc(S(=O)(=O)NC[C@@H]2CCCO2)ccc1NCCCO ZINC000217631800 FC In-Stock Unstable BDKRB1 0 41 Cn1cc(NC(=O)c2cccc(/C=C\C(=O)O)c2)cn1 ZINC000217631818 CD For-Sale Unstable HDAC8 56 49 Cn1cc(NC(=O)c2cccc(/C=C\C(=O)O)c2)cn1 ZINC000217631818 CD For-Sale Unstable HDAC6 45 49 Cn1cc(NC(=O)c2cccc(/C=C\C(=O)O)c2)cn1 ZINC000217631818 CD For-Sale Unstable MAPK10 21 48 Cn1cc(NC(=O)c2cccc(/C=C\C(=O)O)c2)cn1 ZINC000217631818 CD For-Sale Unstable RPS6KA3 17 42 Cn1cc(NC(=O)c2cccc(/C=C\C(=O)O)c2)cn1 ZINC000217631818 CD For-Sale Unstable DDR1 51 35 Cn1cc(NC(=O)c2cccc(/C=C\C(=O)O)c2)cn1 ZINC000217631818 CD For-Sale Unstable RHOA 0 41 Cn1cc(NC(=O)c2cccc(/C=C\C(=O)O)c2)cn1 ZINC000217631818 CD For-Sale Unstable KCNK3 98 40 Cn1cc(NC(=O)c2cccc(/C=C\C(=O)O)c2)cn1 ZINC000217631818 CD For-Sale Unstable KCNK9 49 40 O=C(NCCc1ccc(Cl)cc1)C(F)F ZINC000217631830 BE On-Demand Unstable AMP1_PLAFQ 32 42 O=C(NCCc1ccc(Cl)cc1)C(F)F ZINC000217631830 BE On-Demand Unstable LEF 60 37 CCc1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217631843 CI For-Sale Unstable P95276_MYCTO 0 41 O=C(c1ccoc1)N1CCS[C@@H]1c1ccc(C(F)(F)F)cc1 ZINC000217631893 EI In-Stock Unstable TRPM8 41 35 O=C(O)c1cc(S(=O)(=O)NC[C@H]2CCCO2)ccc1NCCCO ZINC000217631896 FC In-Stock Unstable BDKRB1 0 41 O=C(NC1CCCCCC1)C(F)F ZINC000217631949 AE On-Demand Unstable EPHX2 25 40 O=C(NC1CCCCCC1)C(F)F ZINC000217631949 AE On-Demand Unstable P95276_MYCTO 0 40 O=C(c1ccoc1)N1CCS[C@H]1c1ccc(C(F)(F)F)cc1 ZINC000217631971 EI In-Stock Unstable TRPM8 41 35 CC1(C)CC(NC(=O)N/C=C/c2ccccc2)CC(C)(C)N1 ZINC000217632088 DG For-Sale Unstable EZH2 54 39 CC1(C)CC(NC(=O)N/C=C/c2ccccc2)CC(C)(C)N1 ZINC000217632088 DG For-Sale Unstable HIV1_ENV 0 42 CCCN(CC)CCNCc1c[nH]c2ccccc12 ZINC000217632149 CF For-Sale Unstable MPO 35 40 CC(C)[C@@H]1CCCN(c2ccccc2CBr)CC1 ZINC000217632179 DJ For-Sale Unstable KCNQ2 61 35 O=C(NC[C@@H]1CCCN2CCCC[C@H]12)c1cc2cc(F)ccc2[nH]1 ZINC000217632228 EG In-Stock Unstable PYGL 77 43 O=C(NC[C@@H]1CCCN2CCCC[C@H]12)c1cc2cc(F)ccc2[nH]1 ZINC000217632228 EG In-Stock Unstable PLD1 35 47 O=C(NC[C@@H]1CCCN2CCCC[C@H]12)c1cc2cc(F)ccc2[nH]1 ZINC000217632228 EG In-Stock Unstable PYGM 25 41 O=C(NC[C@@H]1CCCN2CCCC[C@H]12)c1cc2cc(F)ccc2[nH]1 ZINC000217632228 EG In-Stock Unstable PLD2 51 47 Cc1cc(C)n(CCCNC(=O)c2cn3c4c(cccc4c2=O)CC3)n1 ZINC000217632229 FE In-Stock Unstable MTNR1C 0 43 COC(CNC(=O)[C@@H](C)c1ccccc1)OC ZINC000217632233 BD For-Sale Unstable CAPN2 24 41 COC(CNC(=O)[C@@H](C)c1ccccc1)OC ZINC000217632233 BD For-Sale Unstable GPR88 0 48 CN1CCCC[C@@H]1CNC(=O)C[C@@H](N)c1ccccc1 ZINC000217632239 CD For-Sale Unstable SLC6A3 21 52 CN1CCCC[C@@H]1CNC(=O)C[C@@H](N)c1ccccc1 ZINC000217632239 CD For-Sale Unstable DPP4 18 41 CN1CCCC[C@@H]1CNC(=O)C[C@@H](N)c1ccccc1 ZINC000217632239 CD For-Sale Unstable CHRNA10 44 38 CN1CCCC[C@@H]1CNC(=O)C[C@@H](N)c1ccccc1 ZINC000217632239 CD For-Sale Unstable ACKR3 69 35 CC(C)[C@H]1CCCN(c2ccccc2CBr)CC1 ZINC000217632265 DJ For-Sale Unstable KCNQ2 61 35 CCC(CC)N(C)C(=O)c1cc(/C=C\C(=O)O)ccc1F ZINC000217632302 CG For-Sale Unstable APP 40 31 COC(CNC(=O)[C@H](C)c1ccccc1)OC ZINC000217632314 BD For-Sale Unstable CAPN2 24 41 COC(CNC(=O)[C@H](C)c1ccccc1)OC ZINC000217632314 BD For-Sale Unstable GPR88 0 48 CN1CCCC[C@H]1CNC(=O)C[C@@H](N)c1ccccc1 ZINC000217632319 CD For-Sale Unstable SLC6A3 21 52 CN1CCCC[C@H]1CNC(=O)C[C@@H](N)c1ccccc1 ZINC000217632319 CD For-Sale Unstable DPP4 18 41 CN1CCCC[C@H]1CNC(=O)C[C@@H](N)c1ccccc1 ZINC000217632319 CD For-Sale Unstable CHRNA10 44 38 CN1CCCC[C@H]1CNC(=O)C[C@@H](N)c1ccccc1 ZINC000217632319 CD For-Sale Unstable ACKR3 69 35 O=C(C[C@@H]1NC(=O)N(CCc2ccc(F)cc2)C1=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217632358 JD In-Stock Unstable CHRNA4 31 57 O=C(O)c1cc(S(=O)(=O)NC[C@@H]2CCCO2)ccc1NCc1ccccc1 ZINC000217632374 GE In-Stock Unstable BDKRB1 0 44 O=C(O)c1cc(S(=O)(=O)NC[C@@H]2CCCO2)ccc1NCc1ccccc1 ZINC000217632374 GE In-Stock Unstable TNK2 41 38 O=C(O)c1cc(S(=O)(=O)NC[C@@H]2CCCO2)ccc1NCc1ccccc1 ZINC000217632374 GE In-Stock Unstable SFRP1 40 31 C=CCOc1ccc(CN[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217632409 CF On-Demand Unstable HRH3 15 44 CCN(CC)C(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217632412 CE For-Sale Unstable OPRD1 36 46 CCN(CC)C(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217632412 CE For-Sale Unstable KCNK3 104 39 CCN(CC)C(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217632412 CE For-Sale Unstable KCNK9 72 38 C[C@@H]1CCCN(C(=O)N/C=C/c2ccccc2)C1 ZINC000217632414 BG For-Sale Unstable PREP 43 35 O=C(O)c1cc(S(=O)(=O)NC[C@H]2CCCO2)ccc1NCc1ccccc1 ZINC000217632465 GE In-Stock Unstable BDKRB1 0 44 O=C(O)c1cc(S(=O)(=O)NC[C@H]2CCCO2)ccc1NCc1ccccc1 ZINC000217632465 GE In-Stock Unstable TNK2 41 38 O=C(O)c1cc(S(=O)(=O)NC[C@H]2CCCO2)ccc1NCc1ccccc1 ZINC000217632465 GE In-Stock Unstable SFRP1 40 31 N#Cc1cc2c(nc1N1CCN(S(=O)(=O)c3cccc(Br)c3)CC1)CCCC2 ZINC000217632474 JG On-Demand Unstable AKR1C3 45 37 COc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)N1CCN(C(c3ccccc3)c3ccccc3)CC1)C(=O)OC2 ZINC000217632475 KK In-Stock Unstable IMPDH2 84 56 COC(=O)c1ccc(S(=O)(=O)N2CCS[C@@H]2c2ccc(C(F)(F)F)cc2)cc1 ZINC000217632492 IH In-Stock Unstable HSD11B1 15 41 COC(=O)c1ccc(S(=O)(=O)N2CCS[C@@H]2c2ccc(C(F)(F)F)cc2)cc1 ZINC000217632492 IH In-Stock Unstable MMP13 35 43 COC(=O)c1ccc(S(=O)(=O)N2CCS[C@@H]2c2ccc(C(F)(F)F)cc2)cc1 ZINC000217632492 IH In-Stock Unstable ADAM17 17 40 COC(=O)c1ccc(S(=O)(=O)N2CCS[C@@H]2c2ccc(C(F)(F)F)cc2)cc1 ZINC000217632492 IH In-Stock Unstable MMP2 22 43 COC(=O)c1ccc(S(=O)(=O)N2CCS[C@@H]2c2ccc(C(F)(F)F)cc2)cc1 ZINC000217632492 IH In-Stock Unstable MMP3 37 43 COC(=O)c1ccc(S(=O)(=O)N2CCS[C@@H]2c2ccc(C(F)(F)F)cc2)cc1 ZINC000217632492 IH In-Stock Unstable MMP9 24 43 COC(=O)c1ccc(S(=O)(=O)N2CCS[C@@H]2c2ccc(C(F)(F)F)cc2)cc1 ZINC000217632492 IH In-Stock Unstable MMP7 44 43 COC(=O)c1ccc(S(=O)(=O)N2CCS[C@@H]2c2ccc(C(F)(F)F)cc2)cc1 ZINC000217632492 IH In-Stock Unstable MMP1 39 43 C=CCOc1ccc(CN[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217632500 CF On-Demand Unstable HRH3 15 44 C[C@H]1CCCN(C(=O)N/C=C/c2ccccc2)C1 ZINC000217632503 BG For-Sale Unstable PREP 43 35 O=C(Cc1cnccn1)N1CCC[C@@H]1c1nc2cc(F)ccc2[nH]1 ZINC000217632518 EE In-Stock Unstable PRCP 67 53 O=C(Cc1cnccn1)N1CCC[C@@H]1c1nc2cc(F)ccc2[nH]1 ZINC000217632518 EE In-Stock Unstable COLA 58 40 O=C(Cc1cnccn1)N1CCC[C@@H]1c1nc2cc(F)ccc2[nH]1 ZINC000217632518 EE In-Stock Unstable CPT1A 58 37 C[C@@H](Nc1ccc(S(=O)(=O)NC[C@@H]2CCCO2)cc1C(=O)O)c1ccccc1 ZINC000217632579 HG In-Stock Unstable BDKRB1 0 43 COC(=O)c1ccc(S(=O)(=O)N2CCS[C@H]2c2ccc(C(F)(F)F)cc2)cc1 ZINC000217632584 IH In-Stock Unstable HSD11B1 15 41 COC(=O)c1ccc(S(=O)(=O)N2CCS[C@H]2c2ccc(C(F)(F)F)cc2)cc1 ZINC000217632584 IH In-Stock Unstable MMP13 35 43 COC(=O)c1ccc(S(=O)(=O)N2CCS[C@H]2c2ccc(C(F)(F)F)cc2)cc1 ZINC000217632584 IH In-Stock Unstable ADAM17 17 40 COC(=O)c1ccc(S(=O)(=O)N2CCS[C@H]2c2ccc(C(F)(F)F)cc2)cc1 ZINC000217632584 IH In-Stock Unstable MMP2 22 43 COC(=O)c1ccc(S(=O)(=O)N2CCS[C@H]2c2ccc(C(F)(F)F)cc2)cc1 ZINC000217632584 IH In-Stock Unstable MMP3 37 43 COC(=O)c1ccc(S(=O)(=O)N2CCS[C@H]2c2ccc(C(F)(F)F)cc2)cc1 ZINC000217632584 IH In-Stock Unstable MMP9 24 43 COC(=O)c1ccc(S(=O)(=O)N2CCS[C@H]2c2ccc(C(F)(F)F)cc2)cc1 ZINC000217632584 IH In-Stock Unstable MMP7 44 43 COC(=O)c1ccc(S(=O)(=O)N2CCS[C@H]2c2ccc(C(F)(F)F)cc2)cc1 ZINC000217632584 IH In-Stock Unstable MMP1 39 43 O=C(Cc1cnccn1)N1CCC[C@H]1c1nc2cc(F)ccc2[nH]1 ZINC000217632597 EE In-Stock Unstable PRCP 67 53 O=C(Cc1cnccn1)N1CCC[C@H]1c1nc2cc(F)ccc2[nH]1 ZINC000217632597 EE In-Stock Unstable COLA 58 40 O=C(Cc1cnccn1)N1CCC[C@H]1c1nc2cc(F)ccc2[nH]1 ZINC000217632597 EE In-Stock Unstable CPT1A 58 37 CCCOc1ccc(CN[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217632607 CG On-Demand Unstable LTA4H 35 40 CCCOc1ccc(CN[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217632607 CG On-Demand Unstable HRH3 33 50 C[C@H](Nc1ccc(S(=O)(=O)NC[C@@H]2CCCO2)cc1C(=O)O)c1ccccc1 ZINC000217632665 HG In-Stock Unstable BDKRB1 0 43 CCCOc1ccc(CN[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217632679 CG On-Demand Unstable LTA4H 35 40 CCCOc1ccc(CN[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217632679 CG On-Demand Unstable HRH3 33 50 O=S(=O)(c1ccc2c(c1)OCCCO2)N1CCS[C@@H]1c1ccc(C(F)(F)F)cc1 ZINC000217632687 II In-Stock Unstable PKM 40 49 CCN(Cc1ccccc1)C(=O)N/C=C/c1ccccc1 ZINC000217632723 CH For-Sale Unstable TSPO 23 40 CCN(Cc1ccccc1)C(=O)N/C=C/c1ccccc1 ZINC000217632723 CH For-Sale Unstable HDAC6 16 40 CCN(Cc1ccccc1)C(=O)N/C=C/c1ccccc1 ZINC000217632723 CH For-Sale Unstable PTGES 20 40 CCN(Cc1ccccc1)C(=O)N/C=C/c1ccccc1 ZINC000217632723 CH For-Sale Unstable LIMK2 20 43 C[C@@H](Nc1ccc(S(=O)(=O)NC[C@H]2CCCO2)cc1C(=O)O)c1ccccc1 ZINC000217632741 HG In-Stock Unstable BDKRB1 0 43 O=C(O)/C=C\c1ccc(F)c(C(=O)Nc2ncccn2)c1 ZINC000217632747 CD For-Sale Anodyne MMP1 16 40 O=C(Cn1c(=O)[nH]c2ccccc2c1=O)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217632750 FD In-Stock Unstable Q7YY07_CRYPV 41 32 O=S(=O)(c1ccc2c(c1)OCCCO2)N1CCS[C@H]1c1ccc(C(F)(F)F)cc1 ZINC000217632765 II In-Stock Unstable PKM 40 49 C[C@@H](NC(=O)C(F)F)c1ccc(Cl)cc1 ZINC000217632776 BF On-Demand Unstable PTGER4 15 43 C[C@@H](NC(=O)C(F)F)c1ccc(Cl)cc1 ZINC000217632776 BF On-Demand Unstable SDH1 0 51 C[C@@H](NC(=O)C(F)F)c1ccc(Cl)cc1 ZINC000217632776 BF On-Demand Unstable ACACA 42 38 C[C@@H](NC(=O)C(F)F)c1ccc(Cl)cc1 ZINC000217632776 BF On-Demand Unstable PRCP 19 40 C[C@@H](NC(=O)C(F)F)c1ccc(Cl)cc1 ZINC000217632776 BF On-Demand Unstable FFAR2 30 40 C[C@@H](NC(=O)C(F)F)c1ccc(Cl)cc1 ZINC000217632776 BF On-Demand Unstable UTS2 42 35 C[C@H](Nc1ccc(S(=O)(=O)NC[C@H]2CCCO2)cc1C(=O)O)c1ccccc1 ZINC000217632817 HG In-Stock Unstable BDKRB1 0 43 O=C(O)/C=C\c1ccc(C(=O)Nc2ncccn2)c(F)c1 ZINC000217632826 CD For-Sale Anodyne MMP1 0 40 C[C@@H]1CCCCN1C(=O)N/C=C/c1ccccc1 ZINC000217632841 BG For-Sale Unstable CPT1A 42 34 C[C@@H]1CCCCN1C(=O)N/C=C/c1ccccc1 ZINC000217632841 BG For-Sale Unstable PREP 45 35 C[C@H](NC(=O)C(F)F)c1ccc(Cl)cc1 ZINC000217632866 BF On-Demand Unstable PTGER4 15 43 C[C@H](NC(=O)C(F)F)c1ccc(Cl)cc1 ZINC000217632866 BF On-Demand Unstable SDH1 0 51 C[C@H](NC(=O)C(F)F)c1ccc(Cl)cc1 ZINC000217632866 BF On-Demand Unstable ACACA 42 38 C[C@H](NC(=O)C(F)F)c1ccc(Cl)cc1 ZINC000217632866 BF On-Demand Unstable PRCP 19 40 C[C@H](NC(=O)C(F)F)c1ccc(Cl)cc1 ZINC000217632866 BF On-Demand Unstable FFAR2 30 40 C[C@H](NC(=O)C(F)F)c1ccc(Cl)cc1 ZINC000217632866 BF On-Demand Unstable UTS2 42 35 O=S(=O)(c1ccc2c(c1)CCO2)N1CCS[C@@H]1c1ccc(C(F)(F)F)cc1 ZINC000217632878 HI In-Stock Unstable PKM 35 43 O=C(O)c1cc(S(=O)(=O)NC[C@@H]2CCCO2)ccc1NCCc1ccccc1 ZINC000217632918 HE In-Stock Unstable BDKRB1 28 43 CCC[C@@H](COC)NC(=O)N[C@H](CC(=O)OC)C(=O)O ZINC000217632920 CC For-Sale Unstable FOLH1 16 40 C[C@H]1CCCCN1C(=O)N/C=C/c1ccccc1 ZINC000217632931 BG For-Sale Unstable CPT1A 42 34 C[C@H]1CCCCN1C(=O)N/C=C/c1ccccc1 ZINC000217632931 BG For-Sale Unstable PREP 45 35 O=S(=O)(c1ccc2c(c1)CCO2)N1CCS[C@H]1c1ccc(C(F)(F)F)cc1 ZINC000217632964 HI In-Stock Unstable PKM 35 43 O=C([C@H]1CCCN(Cc2cncs2)C1)N1CCCC1 ZINC000217632980 CD On-Demand Unstable SLC6A1 78 35 CCC[C@H](COC)NC(=O)N[C@H](CC(=O)OC)C(=O)O ZINC000217632998 CC For-Sale Unstable FOLH1 16 40 O=C(O)c1cc(S(=O)(=O)NC[C@H]2CCCO2)ccc1NCCc1ccccc1 ZINC000217633001 HE In-Stock Unstable BDKRB1 28 43 O=C(NCc1ccc(C(=O)O)cc1)OCc1ccc(F)cc1 ZINC000217633032 DF For-Sale Unstable TPSAB1 34 50 O=C(NCc1ccc(C(=O)O)cc1)OCc1ccc(F)cc1 ZINC000217633032 DF For-Sale Unstable NPR 52 32 O=C(NCc1ccc(C(=O)O)cc1)OCc1ccc(F)cc1 ZINC000217633032 DF For-Sale Unstable NAAA 28 42 O=C(NCc1ccc(C(=O)O)cc1)OCc1ccc(F)cc1 ZINC000217633032 DF For-Sale Unstable PDS 42 38 CC[C@@H]1CCCCN1C(=O)N/C=C/c1ccccc1 ZINC000217633033 CH For-Sale Unstable COLA 53 35 CC[C@@H]1CCCCN1C(=O)N/C=C/c1ccccc1 ZINC000217633033 CH For-Sale Unstable CPT1A 51 34 CC[C@@H]1CCCCN1C(=O)N/C=C/c1ccccc1 ZINC000217633033 CH For-Sale Unstable PREP 50 36 O=C([C@@H]1CCCN(Cc2cncs2)C1)N1CCCC1 ZINC000217633062 CD On-Demand Unstable SLC6A1 78 35 O=C(Nc1cccs1)N1CCS[C@@H]1c1ccc(C(F)(F)F)cc1 ZINC000217633081 FK In-Stock Unstable TRPM8 64 49 COc1ccc(CCNc2ccc(S(=O)(=O)NC[C@@H]3CCCO3)cc2C(=O)O)cc1 ZINC000217633110 IF In-Stock Unstable IAP 0 41 COc1ccc(CCNc2ccc(S(=O)(=O)NC[C@@H]3CCCO3)cc2C(=O)O)cc1 ZINC000217633110 IF In-Stock Unstable AKR1C3 16 40 CC[C@H]1CCCCN1C(=O)N/C=C/c1ccccc1 ZINC000217633118 CH For-Sale Unstable COLA 53 35 CC[C@H]1CCCCN1C(=O)N/C=C/c1ccccc1 ZINC000217633118 CH For-Sale Unstable CPT1A 51 34 CC[C@H]1CCCCN1C(=O)N/C=C/c1ccccc1 ZINC000217633118 CH For-Sale Unstable PREP 50 36 O=C(Nc1cccs1)N1CCS[C@H]1c1ccc(C(F)(F)F)cc1 ZINC000217633148 FK In-Stock Unstable TRPM8 70 49 Cc1ccc(S(=O)(=O)Nc2onc(C)c2C)s1 ZINC000217633150 CE On-Demand Unstable EDNRA 80 60 C[C@@H](NC(=O)C(F)F)c1ccc(Br)cc1 ZINC000217633156 CF On-Demand Unstable SDH1 0 55 COc1ccc(CCNc2ccc(S(=O)(=O)NC[C@H]3CCCO3)cc2C(=O)O)cc1 ZINC000217633189 IF In-Stock Unstable IAP 0 41 COc1ccc(CCNc2ccc(S(=O)(=O)NC[C@H]3CCCO3)cc2C(=O)O)cc1 ZINC000217633189 IF In-Stock Unstable AKR1C3 16 40 O=C(c1ccc(NS(=O)(=O)c2cccc3cccnc23)cc1)N1CCC(O)(Cc2cccnc2)CC1 ZINC000217633197 KH Annotated Unstable NAMPT 36 44 O=C(N/C=C/c1ccccc1)N(Cc1ccccc1)Cc1ccccc1 ZINC000217633222 EK For-Sale Unstable HDAC6 18 41 O=C(N/C=C/c1ccccc1)N(Cc1ccccc1)Cc1ccccc1 ZINC000217633222 EK For-Sale Unstable 17HSDCL 0 41 O=C(N/C=C/c1ccccc1)N(Cc1ccccc1)Cc1ccccc1 ZINC000217633222 EK For-Sale Unstable PTGES 24 43 C[C@H](NC(=O)C(F)F)c1ccc(Br)cc1 ZINC000217633227 CF On-Demand Unstable SDH1 0 55 CSCC[C@@H](CO)NC(=O)[C@@H]1CC(=O)N(Cc2ccc3c(c2)OCO3)C1 ZINC000217633229 GC In-Stock Unstable NOS2 47 33 O=C(Nc1ccccc1Cl)N1CCS[C@@H]1c1ccc(C(F)(F)F)cc1 ZINC000217633253 GK In-Stock Unstable TRPM8 75 47 COc1ccc(CCNc2ccc(S(=O)(=O)NC[C@@H]3CCCO3)cc2C(=O)O)cc1OC ZINC000217633310 JF In-Stock Unstable IAP 0 43 COc1ccc(CCNc2ccc(S(=O)(=O)NC[C@@H]3CCCO3)cc2C(=O)O)cc1OC ZINC000217633310 JF In-Stock Unstable SCMU_MYCTU 0 41 CSCC[C@@H](CO)NC(=O)[C@H]1CC(=O)N(Cc2ccc3c(c2)OCO3)C1 ZINC000217633320 GC In-Stock Unstable NOS2 47 33 O=C(Nc1ccccc1Cl)N1CCS[C@H]1c1ccc(C(F)(F)F)cc1 ZINC000217633338 GK In-Stock Unstable TRPM8 66 47 O=C(N/C=C/c1ccccc1)N(CCO)Cc1ccccc1 ZINC000217633339 CF For-Sale Unstable LIMK2 21 44 CC(C)NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217633372 CD On-Demand Unstable CA2 27 43 CC(C)NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217633372 CD On-Demand Unstable CA1 37 43 CC(C)NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217633372 CD On-Demand Unstable MMP13 36 40 CC(C)NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217633372 CD On-Demand Unstable CA4 37 47 CC(C)NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217633372 CD On-Demand Unstable MMP2 30 48 CC(C)NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217633372 CD On-Demand Unstable MMP14 0 40 CC(C)NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217633372 CD On-Demand Unstable MMP9 23 42 CC(C)NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217633372 CD On-Demand Unstable MMP12 45 40 CC(C)NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217633372 CD On-Demand Unstable CA12 23 41 CC(C)NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217633372 CD On-Demand Unstable MMP7 23 40 CC(C)NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217633372 CD On-Demand Unstable CA9 22 41 CC(C)NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217633372 CD On-Demand Unstable LEF 53 35 CC(C)NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217633372 CD On-Demand Unstable IDO1 37 42 CC(C)NS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217633372 CD On-Demand Unstable P96878_MYCTU 47 41 COc1ccc(CCNc2ccc(S(=O)(=O)NC[C@H]3CCCO3)cc2C(=O)O)cc1OC ZINC000217633391 JF In-Stock Unstable IAP 0 43 COc1ccc(CCNc2ccc(S(=O)(=O)NC[C@H]3CCCO3)cc2C(=O)O)cc1OC ZINC000217633391 JF In-Stock Unstable SCMU_MYCTU 0 41 COc1ccc(NC(=O)N/C=C/c2ccccc2)c(OC)c1 ZINC000217633432 CG For-Sale Unstable CYP1B1 64 50 COc1ccc(NC(=O)N/C=C/c2ccccc2)c(OC)c1 ZINC000217633432 CG For-Sale Unstable MTNR1A 33 45 COc1ccc(NC(=O)N/C=C/c2ccccc2)c(OC)c1 ZINC000217633432 CG For-Sale Unstable MTNR1B 35 45 COc1ccc(NC(=O)N/C=C/c2ccccc2)c(OC)c1 ZINC000217633432 CG For-Sale Unstable CYP1A1 38 50 COc1ccc(NC(=O)N/C=C/c2ccccc2)c(OC)c1 ZINC000217633432 CG For-Sale Unstable ABCG2 20 44 COc1ccc(NC(=O)N/C=C/c2ccccc2)c(OC)c1 ZINC000217633432 CG For-Sale Unstable AKR1C2 51 36 COc1cc2c(cc1OC)CN(Cc1oc(CN3CCCCCC3)cc(=O)c1O)CC2 ZINC000217633437 IG In-Stock Unstable ABCB1B 61 35 COc1cc2c(cc1OC)CN(Cc1oc(CN3CCCCCC3)cc(=O)c1O)CC2 ZINC000217633437 IG In-Stock Unstable ABCB1 23 47 CN(C)S(=O)(=O)NCc1cc(/C=C\C(=O)O)ccc1F ZINC000217633443 DC For-Sale Unstable AKR1C3 29 45 CNS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217633505 CC On-Demand Unstable CA2 35 53 CNS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217633505 CC On-Demand Unstable CA1 40 43 CNS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217633505 CC On-Demand Unstable CA7 17 45 CNS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217633505 CC On-Demand Unstable MMP13 32 40 CNS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217633505 CC On-Demand Unstable CA4 35 49 CNS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217633505 CC On-Demand Unstable CA14 21 50 CNS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217633505 CC On-Demand Unstable MMP2 26 43 CNS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217633505 CC On-Demand Unstable CA12 28 42 CNS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217633505 CC On-Demand Unstable CA9 30 53 CNS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217633505 CC On-Demand Unstable LEF 29 43 CNS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217633505 CC On-Demand Unstable IDO1 44 48 CNS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217633505 CC On-Demand Unstable MTCA1 42 41 CNS(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217633505 CC On-Demand Unstable P96878_MYCTU 52 41 O=C(O)c1cc(S(=O)(=O)NC[C@@H]2CCCO2)ccc1NCc1ccco1 ZINC000217633508 GE In-Stock Unstable BDKRB1 0 40 NC(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000217633515 AD On-Demand Unstable MDM2 45 33 CC(C)[C@@H]1CCCN(c2ccc(CBr)cc2)CC1 ZINC000217633560 DJ For-Sale Unstable L3MBTL3 40 41 O=C(O)c1cc(S(=O)(=O)NC[C@H]2CCCO2)ccc1NCc1ccco1 ZINC000217633594 GE In-Stock Unstable BDKRB1 0 40 CC(C)[C@H]1CCCN(c2ccc(CBr)cc2)CC1 ZINC000217633634 DJ For-Sale Unstable L3MBTL3 40 41 Cc1cc(Cl)ccc1NC(=O)N/C=C/c1ccccc1 ZINC000217633656 CI For-Sale Unstable LPL 41 32 Cc1cc(Cl)ccc1NC(=O)N/C=C/c1ccccc1 ZINC000217633656 CI For-Sale Unstable CMA1 22 44 O=C(O)c1cc(S(=O)(=O)NC[C@@H]2CCCO2)ccc1NC[C@@H]1CCCO1 ZINC000217633705 GD In-Stock Unstable BDKRB1 0 44 C[C@H](c1ccc(Br)cc1F)N1CCC[C@@H]([C@@H]2CCCN2)C1 ZINC000217633743 FI For-Sale Unstable MBTD1 0 41 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1ccc(O)c(OC)c1 ZINC000217633747 JG In-Stock Unstable CACNA1D 46 35 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1ccc(O)c(OC)c1 ZINC000217633747 JG In-Stock Unstable TGFBR2 51 41 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1ccc(O)c(OC)c1 ZINC000217633747 JG In-Stock Unstable HISG 0 42 O=C(N/C=C/c1ccccc1)NCCCO ZINC000217633758 BD For-Sale Unstable HDAC9 21 42 O=C(O)c1cc(S(=O)(=O)NC[C@H]2CCCO2)ccc1NC[C@@H]1CCCO1 ZINC000217633780 GD In-Stock Unstable BDKRB1 0 44 O=C(O)c1cc(S(=O)(=O)NC[C@H]2CCCO2)ccc1NC[C@@H]1CCCO1 ZINC000217633780 GD In-Stock Unstable TNK2 40 37 COc1ccc(/C=C\C(=O)O)cc1NS(=O)(=O)N(C)C ZINC000217633810 DD For-Sale Unstable TUBB1 53 39 COc1ccc(/C=C\C(=O)O)cc1NS(=O)(=O)N(C)C ZINC000217633810 DD For-Sale Unstable ABCG2 18 41 COc1ccc(/C=C\C(=O)O)cc1NS(=O)(=O)N(C)C ZINC000217633810 DD For-Sale Unstable NFE2L2 0 41 N#Cc1ccc(C(=O)N2CCS[C@@H]2c2cccc(F)c2)cc1 ZINC000217633820 DH In-Stock Unstable NR3C2 0 53 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@H](c3cccs3)C2)[C@@H]1c1ccc(O)c(OC)c1 ZINC000217633841 JG In-Stock Unstable CACNA1D 46 35 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@H](c3cccs3)C2)[C@@H]1c1ccc(O)c(OC)c1 ZINC000217633841 JG In-Stock Unstable TGFBR2 51 41 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@H](c3cccs3)C2)[C@@H]1c1ccc(O)c(OC)c1 ZINC000217633841 JG In-Stock Unstable HISG 0 42 O=C(O)c1cc(S(=O)(=O)NC[C@@H]2CCCO2)ccc1NC[C@H]1CCCO1 ZINC000217633870 GD In-Stock Unstable BDKRB1 0 44 O=C(O)c1cc(S(=O)(=O)NC[C@@H]2CCCO2)ccc1NC[C@H]1CCCO1 ZINC000217633870 GD In-Stock Unstable TNK2 40 37 C[C@H](c1cc(Br)ccc1F)N1CCC[C@@H]([C@@H]2CCCN2)C1 ZINC000217633921 FI For-Sale Unstable MBTD1 0 40 N#Cc1ccc(C(=O)N2CCS[C@H]2c2cccc(F)c2)cc1 ZINC000217633923 DH In-Stock Unstable NR3C2 0 53 O=C(O)c1cc(S(=O)(=O)NC[C@H]2CCCO2)ccc1NC[C@H]1CCCO1 ZINC000217633950 GD In-Stock Unstable BDKRB1 0 44 O=C(O)c1cc(S(=O)(=O)NC[C@H]2CCCO2)ccc1NC[C@H]1CCCO1 ZINC000217633950 GD In-Stock Unstable TNK2 40 37 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1ccc2c(c1)OCO2 ZINC000217633955 JG In-Stock Unstable CACNA1C 23 41 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1ccc2c(c1)OCO2 ZINC000217633955 JG In-Stock Unstable CACNA1D 44 41 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1ccc2c(c1)OCO2 ZINC000217633955 JG In-Stock Unstable TGFBR2 50 40 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@@H](c3cccs3)C2)[C@@H]1c1ccc2c(c1)OCO2 ZINC000217633955 JG In-Stock Unstable HISG 0 40 CN1CCC(c2noc(C(=O)O)c2Cl)CC1 ZINC000217633982 BD For-Sale Unstable HTR1F 20 40 CCCCCCCNCCN(CC)CCC ZINC000217634001 BG For-Sale Unstable PAOX 18 44 CCCCCCCNCCN(CC)CCC ZINC000217634001 BG For-Sale Unstable S1PR2 29 41 C[C@@]12CC[C@@H](CC#N)[C@@]1(C)CC(=O)O2 ZINC000217634024 AE In-Stock Unstable PPP2R1A 40 29 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@H](c3cccs3)C2)[C@@H]1c1ccc2c(c1)OCO2 ZINC000217634046 JG In-Stock Unstable CACNA1C 23 41 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@H](c3cccs3)C2)[C@@H]1c1ccc2c(c1)OCO2 ZINC000217634046 JG In-Stock Unstable CACNA1D 44 41 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@H](c3cccs3)C2)[C@@H]1c1ccc2c(c1)OCO2 ZINC000217634046 JG In-Stock Unstable TGFBR2 50 40 COC(=O)C1=C(C)NC2=C(C(=O)[C@H](C(=O)OC)[C@H](c3cccs3)C2)[C@@H]1c1ccc2c(c1)OCO2 ZINC000217634046 JG In-Stock Unstable HISG 0 40 CNC[C@@H]1CCCN([C@@H](C)c2ccc(Br)cc2F)C1 ZINC000217634052 EH For-Sale Unstable GHSR 21 40 O=C(O)c1cc(S(=O)(=O)NC[C@@H]2CCCO2)ccc1N1CCCC1 ZINC000217634070 FD In-Stock Unstable BDKRB1 0 41 O=C(O)c1cc(S(=O)(=O)NC[C@@H]2CCCO2)ccc1N1CCCC1 ZINC000217634070 FD In-Stock Unstable SFRP1 79 33 O=C(O)c1cc(S(=O)(=O)NC[C@@H]2CCCO2)ccc1N1CCCC1 ZINC000217634070 FD In-Stock Unstable WNT3 53 33 CC(C)OC(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217634088 CE For-Sale Unstable ACR 61 39 N#Cc1c(OCc2ccccc2)ccnc1Cl ZINC000217634102 BG For-Sale Unstable PTGER1 41 38 CCCCN(CCCC)C(=O)N/C=C/c1ccccc1 ZINC000217634107 CI For-Sale Unstable TSPO 37 41 C[C@]12CC[C@@H](CC#N)[C@@]1(C)CC(=O)O2 ZINC000217634122 AE In-Stock Unstable PPP2R1A 40 29 O=C(O)c1cc(S(=O)(=O)NC[C@H]2CCCO2)ccc1N1CCCC1 ZINC000217634167 FD In-Stock Unstable BDKRB1 0 41 O=C(O)c1cc(S(=O)(=O)NC[C@H]2CCCO2)ccc1N1CCCC1 ZINC000217634167 FD In-Stock Unstable SFRP1 79 33 O=C(O)c1cc(S(=O)(=O)NC[C@H]2CCCO2)ccc1N1CCCC1 ZINC000217634167 FD In-Stock Unstable WNT3 53 33 CCc1ccc([C@@H](C)NC(=O)C(F)F)cc1 ZINC000217634206 BF On-Demand Unstable SDH1 0 43 CCc1ccc([C@@H](C)NC(=O)C(F)F)cc1 ZINC000217634206 BF On-Demand Unstable ACACA 63 42 CCc1ccc([C@@H](C)NC(=O)C(F)F)cc1 ZINC000217634206 BF On-Demand Unstable ACACB 30 42 CCc1ccc([C@@H](C)NC(=O)C(F)F)cc1 ZINC000217634206 BF On-Demand Unstable ACE2 45 33 C[C@@]12CC[C@H](CC#N)[C@@]1(C)CC(=O)O2 ZINC000217634212 AE In-Stock Unstable PPP2R1A 40 29 N#Cc1cc2c(nc1NCCN1CCN(Cc3ccccc3)CC1)CCCC2 ZINC000217634241 GG On-Demand Unstable ACHE 41 52 N#Cc1cc2c(nc1NCCN1CCN(Cc3ccccc3)CC1)CCCC2 ZINC000217634241 GG On-Demand Unstable SIGMAR1 27 40 N#Cc1cc2c(nc1NCCN1CCN(Cc3ccccc3)CC1)CCCC2 ZINC000217634241 GG On-Demand Unstable BCHE 40 52 N#Cc1cc2c(nc1NCCN1CCN(Cc3ccccc3)CC1)CCCC2 ZINC000217634241 GG On-Demand Unstable HNMT 35 42 CCc1ccc([C@H](C)NC(=O)C(F)F)cc1 ZINC000217634284 BF On-Demand Unstable SDH1 0 43 CCc1ccc([C@H](C)NC(=O)C(F)F)cc1 ZINC000217634284 BF On-Demand Unstable ACACA 63 42 CCc1ccc([C@H](C)NC(=O)C(F)F)cc1 ZINC000217634284 BF On-Demand Unstable ACACB 30 42 CCc1ccc([C@H](C)NC(=O)C(F)F)cc1 ZINC000217634284 BF On-Demand Unstable ACE2 45 33 CC(C)[C@H](NC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)C(=O)N1CCc2c([nH]c3ccccc23)C1 ZINC000217634288 JG In-Stock Unstable SSTR4 49 33 CC(C)[C@H](NC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)C(=O)N1CCc2c([nH]c3ccccc23)C1 ZINC000217634288 JG In-Stock Unstable SSTR5 40 33 O=C(O)c1cc(S(=O)(=O)NC[C@@H]2CCCO2)ccc1N1CCCCC1 ZINC000217634289 FD In-Stock Unstable BDKRB1 0 40 O=C(O)c1cc(S(=O)(=O)NC[C@@H]2CCCO2)ccc1N1CCCCC1 ZINC000217634289 FD In-Stock Unstable SFRP1 70 32 O=C(O)c1cc(S(=O)(=O)NC[C@@H]2CCCO2)ccc1N1CCCCC1 ZINC000217634289 FD In-Stock Unstable WNT3 53 33 C[C@]12CC[C@H](CC#N)[C@@]1(C)CC(=O)O2 ZINC000217634290 AE In-Stock Unstable PPP2R1A 40 29 COC(=O)[C@@H](NC[C@H]1CCCO1)[C@@H](C)c1ccccc1 ZINC000217634314 CE For-Sale Unstable TNK2 49 40 COC(=O)c1ccc(OS(=O)(=O)C(F)(F)F)c(C(=O)N2CCc3ccccc3C2)c1 ZINC000217634320 IF For-Sale Unstable SLC6A9 26 41 COC(=O)c1ccc(OS(=O)(=O)C(F)(F)F)c(C(=O)N2CCc3ccccc3C2)c1 ZINC000217634320 IF For-Sale Unstable BCL2L1 26 40 COC(=O)c1ccc(OS(=O)(=O)C(F)(F)F)c(C(=O)N2CCc3ccccc3C2)c1 ZINC000217634320 IF For-Sale Unstable AKR1C3 48 38 COC(=O)c1ccc(OS(=O)(=O)C(F)(F)F)c(C(=O)N2CCc3ccccc3C2)c1 ZINC000217634320 IF For-Sale Unstable NOD2 40 36 CN(C)CCCNC(=O)N/C=C/c1ccccc1 ZINC000217634346 BD For-Sale Unstable NPY2R 0 40 CN(C)CCCNC(=O)N/C=C/c1ccccc1 ZINC000217634346 BD For-Sale Unstable DNM1 0 40 O=C(O)c1cc(S(=O)(=O)NC[C@H]2CCCO2)ccc1N1CCCCC1 ZINC000217634361 FD In-Stock Unstable BDKRB1 0 40 O=C(O)c1cc(S(=O)(=O)NC[C@H]2CCCO2)ccc1N1CCCCC1 ZINC000217634361 FD In-Stock Unstable SFRP1 70 32 O=C(O)c1cc(S(=O)(=O)NC[C@H]2CCCO2)ccc1N1CCCCC1 ZINC000217634361 FD In-Stock Unstable WNT3 53 33 COC(=O)[C@H](NC[C@H]1CCCO1)[C@@H](C)c1ccccc1 ZINC000217634385 CE For-Sale Unstable TNK2 49 40 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1N[C@@H]1CCC[C@@H](O)C1 ZINC000217634403 CG For-Sale Unstable TRPM8 15 42 COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc2c1OCCO2 ZINC000217634413 JI In-Stock Unstable AKR1B1 0 45 COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc2c1OCCO2 ZINC000217634413 JI In-Stock Unstable CYP1B1 48 35 COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc2c1OCCO2 ZINC000217634413 JI In-Stock Unstable CYP1A2 30 45 CN(CCCNc1nc2c(cc1C#N)CCCC2)c1ccccc1 ZINC000217634415 DH On-Demand Unstable BCHE 40 38 C[C@@H]1CCC[C@@H](C)N1C(=O)N/C=C/c1ccccc1 ZINC000217634452 CH For-Sale Unstable EDNRB 45 36 O=C(O)c1cc(S(=O)(=O)NC[C@@H]2CCCO2)ccc1N1CCOCC1 ZINC000217634467 FC In-Stock Unstable BDKRB1 0 40 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1N[C@@H]1CCC[C@@H](O)C1 ZINC000217634483 CG On-Demand Unstable TRPM8 15 42 COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc2c1OCCO2 ZINC000217634487 JI In-Stock Unstable AKR1B1 0 45 COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc2c1OCCO2 ZINC000217634487 JI In-Stock Unstable CYP1B1 48 35 COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc2c1OCCO2 ZINC000217634487 JI In-Stock Unstable CYP1A2 30 45 COc1ccc(/C=C\C(=O)O)cc1N1C(=O)CCC1=O ZINC000217634500 CD For-Sale Unstable TUBB1 52 40 COc1ccc(/C=C\C(=O)O)cc1N1C(=O)CCC1=O ZINC000217634500 CD For-Sale Unstable ABCG2 17 43 CCOC(=O)[C@@H](NC[C@H]1CCCO1)[C@@H](C)c1ccccc1 ZINC000217634523 CE For-Sale Unstable TNK2 45 39 C[C@H]1CCC[C@@H](C)N1C(=O)N/C=C/c1ccccc1 ZINC000217634541 CH For-Sale Unstable EDNRB 45 36 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1N[C@@H]1CCC[C@@H](O)C1 ZINC000217634550 CG For-Sale Unstable TRPM8 15 42 O=C(O)c1cc(S(=O)(=O)NC[C@H]2CCCO2)ccc1N1CCOCC1 ZINC000217634557 FC In-Stock Unstable BDKRB1 0 40 COc1ccc(/C=C\C(=O)O)cc1N1C(=O)CCCC1=O ZINC000217634589 CD For-Sale Unstable TUBB1 47 39 COc1ccc(/C=C\C(=O)O)cc1N1C(=O)CCCC1=O ZINC000217634589 CD For-Sale Unstable ABCG2 16 41 CCOC(=O)[C@H](NC[C@H]1CCCO1)[C@@H](C)c1ccccc1 ZINC000217634599 CE For-Sale Unstable TNK2 45 39 Cc1ccccc1[C@@H](C)NC(=O)C(F)F ZINC000217634631 BE On-Demand Unstable CTSA 60 38 C[C@H]1CCC[C@H](C)N1C(=O)N/C=C/c1ccccc1 ZINC000217634633 CH For-Sale Unstable EDNRB 45 36 CC(C)[C@H]1CC[C@H](C)C[C@@H]1N[C@@H]1CCC[C@@H](O)C1 ZINC000217634646 CG For-Sale Unstable TRPM8 15 42 Cc1ccccc1[C@H](C)NC(=O)C(F)F ZINC000217634709 BE On-Demand Unstable CTSA 60 38 CCCCNC(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217634754 CE For-Sale Unstable DRD4 41 31 CCCCNC(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217634754 CE For-Sale Unstable DRD3 28 40 CCCCNC(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217634754 CE For-Sale Unstable PTGDR 21 44 COc1ccc(NC(=O)C[C@@H]2OC(=O)c3c2ccc(OC)c3OC)cc1 ZINC000217634797 FF In-Stock Unstable TSHR 41 30 COc1ccc(NC(=O)C[C@@H]2OC(=O)c3c2ccc(OC)c3OC)cc1 ZINC000217634797 FF In-Stock Unstable MTNR1B 27 41 C[C@@H](c1ccc(Br)cc1F)N1CCC[C@@H](CN)C1 ZINC000217634799 DG For-Sale Unstable GHSR 21 41 CC(C)c1ccc([C@@H](C)NC(=O)C(F)F)cc1 ZINC000217634836 BG On-Demand Unstable SDH1 0 40 CC(C)c1ccc([C@@H](C)NC(=O)C(F)F)cc1 ZINC000217634836 BG On-Demand Unstable ACACA 51 40 C[C@H](c1ccc(Br)cc1F)N1CCC[C@@H](CN)C1 ZINC000217634879 DG For-Sale Unstable GHSR 21 41 COc1ccc(NC(=O)C[C@H]2OC(=O)c3c2ccc(OC)c3OC)cc1 ZINC000217634892 FF In-Stock Unstable TSHR 41 30 COc1ccc(NC(=O)C[C@H]2OC(=O)c3c2ccc(OC)c3OC)cc1 ZINC000217634892 FF In-Stock Unstable MTNR1B 27 41 CC(C)c1ccc([C@H](C)NC(=O)C(F)F)cc1 ZINC000217634917 BG On-Demand Unstable SDH1 0 40 CC(C)c1ccc([C@H](C)NC(=O)C(F)F)cc1 ZINC000217634917 BG On-Demand Unstable ACACA 51 40 COc1ccc(CNC(=O)N2CCS[C@@H]2c2cccc(F)c2)cc1OC ZINC000217634934 GH In-Stock Unstable GRIN2B 22 44 COc1ccc(CNC(=O)N2CCS[C@@H]2c2cccc(F)c2)cc1OC ZINC000217634934 GH In-Stock Unstable HCRTR1 25 41 COc1ccc(CNC(=O)N2CCS[C@@H]2c2cccc(F)c2)cc1OC ZINC000217634934 GH In-Stock Unstable CCR4 40 34 COc1ccc(CNC(=O)N2CCS[C@@H]2c2cccc(F)c2)cc1OC ZINC000217634934 GH In-Stock Unstable HCRTR2 24 40 C[C@@H](c1cc(Br)ccc1F)N1CCC[C@@H](CN)C1 ZINC000217634978 DG For-Sale Unstable GHSR 21 41 Cc1c(NN)nc(C2CC2)nc1N1CCN(C)[C@@H](C)C1 ZINC000217634979 CD For-Sale Unstable CHRM3 21 49 CCN(CC)CCNC(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217635001 CD For-Sale Unstable KCNQ1 0 52 CC(C)CNC(=O)CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12 ZINC000217635009 GG In-Stock Unstable TOP1 21 42 COc1ccc(CNC(=O)N2CCS[C@H]2c2cccc(F)c2)cc1OC ZINC000217635012 GH In-Stock Unstable GRIN2B 22 44 COc1ccc(CNC(=O)N2CCS[C@H]2c2cccc(F)c2)cc1OC ZINC000217635012 GH In-Stock Unstable HCRTR1 25 41 COc1ccc(CNC(=O)N2CCS[C@H]2c2cccc(F)c2)cc1OC ZINC000217635012 GH In-Stock Unstable CCR4 40 34 COc1ccc(CNC(=O)N2CCS[C@H]2c2cccc(F)c2)cc1OC ZINC000217635012 GH In-Stock Unstable HCRTR2 24 40 C[C@H](c1cc(Br)ccc1F)N1CCC[C@@H](CN)C1 ZINC000217635084 DG For-Sale Unstable GHSR 21 41 CC(C)CNC(=O)CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12 ZINC000217635090 GG In-Stock Unstable TOP1 21 42 CCN(CC)CCNC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217635133 CD For-Sale Unstable DRD4 41 31 CCN(CC)CCNC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217635133 CD For-Sale Unstable HDAC8 15 43 O=C(Nc1c(F)cccc1F)N1CCS[C@@H]1c1ccc(F)cc1 ZINC000217635140 EI In-Stock Unstable TRPM8 33 43 C[C@@H]1CCCC[C@@H]1NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217635221 CG For-Sale Unstable HDAC8 19 43 O=C(Nc1c(F)cccc1F)N1CCS[C@H]1c1ccc(F)cc1 ZINC000217635226 EI In-Stock Unstable TRPM8 33 43 CC(C)CCNc1ccc(S(=O)(=O)NC[C@@H]2CCCO2)cc1C(=O)O ZINC000217635234 FE In-Stock Unstable BDKRB1 27 40 C[C@H]1CCCC[C@@H]1NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217635318 CG For-Sale Unstable HDAC8 19 43 CC(C)CCNc1ccc(S(=O)(=O)NC[C@H]2CCCO2)cc1C(=O)O ZINC000217635327 FE In-Stock Unstable BDKRB1 27 40 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)c1ccccc1 ZINC000217635370 IE In-Stock Unstable HTR1D 26 42 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)c1ccccc1 ZINC000217635370 IE In-Stock Unstable HTR1B 20 42 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)c1ccccc1 ZINC000217635370 IE In-Stock Unstable CCKAR 41 39 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)c1ccccc1 ZINC000217635370 IE In-Stock Unstable SSTR3 42 35 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)c1ccccc1 ZINC000217635370 IE In-Stock Unstable CCKBR 37 41 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)c1ccccc1 ZINC000217635370 IE In-Stock Unstable GHSR 52 38 COC(=O)C1(c2ccccc2)CCC(O)CC1 ZINC000217635389 BE In-Stock Unstable ADRA1D 22 42 COC(=O)C1(c2ccccc2)CCC(O)CC1 ZINC000217635389 BE In-Stock Unstable ADRA1A 21 42 COC(=O)C1(c2ccccc2)CCC(O)CC1 ZINC000217635389 BE In-Stock Unstable ADRA1B 18 42 COC(=O)C1(c2ccccc2)CCC(O)CC1 ZINC000217635389 BE In-Stock Unstable KCNA3 44 39 O=C(N/C=C/c1ccccc1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217635433 EK For-Sale Anodyne EPHX1 0 50 O=C(N/C=C/c1ccccc1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217635433 EK For-Sale Anodyne AKR1C3 22 41 O=C(N/C=C/c1ccccc1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217635433 EK For-Sale Anodyne P96878_MYCTU 22 41 O=C(N/C=C/c1ccccc1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217635433 EK For-Sale Anodyne P95276_MYCTO 0 50 O=C(O)/C=C\c1ccc(C(=O)N[C@@H]2CN3CCC2CC3)s1 ZINC000217635458 DD For-Sale Unstable HTR3A 20 54 O=C(O)/C=C\c1ccc(C(=O)N[C@@H]2CN3CCC2CC3)s1 ZINC000217635458 DD For-Sale Unstable CHRNA7 27 66 COC(=O)C[C@@H](c1ccccc1OC)c1oc(CN2CCCCC2)cc(=O)c1O ZINC000217635476 HG In-Stock Unstable DRD2 17 42 CC(=O)c1c(C)nn(CC(=O)N2CCN(C)[C@@H](c3ccccc3)C2)c1C ZINC000217635491 FE In-Stock Unstable P2RX7 0 40 O=C(O)/C=C\c1ccc(C(=O)N[C@H]2CN3CCC2CC3)s1 ZINC000217635537 DD For-Sale Unstable HTR3A 20 54 O=C(O)/C=C\c1ccc(C(=O)N[C@H]2CN3CCC2CC3)s1 ZINC000217635537 DD For-Sale Unstable CHRNA7 27 66 O=C(N/C=C/c1ccccc1)N1CCc2ccccc2C1 ZINC000217635555 CG For-Sale Unstable HDAC6 37 47 O=C(N/C=C/c1ccccc1)N1CCc2ccccc2C1 ZINC000217635555 CG For-Sale Unstable DPP8 17 45 COC(=O)C[C@H](c1ccccc1OC)c1oc(CN2CCCCC2)cc(=O)c1O ZINC000217635561 HG In-Stock Unstable DRD2 17 42 CC(=O)c1c(C)nn(CC(=O)N2CCN(C)[C@H](c3ccccc3)C2)c1C ZINC000217635574 FE In-Stock Unstable P2RX7 0 40 O=C(O)/C=C\c1ccc(C(=O)NCCc2cccs2)s1 ZINC000217635629 DF For-Sale Unstable ADAM17 18 42 Cc1cccc(NC(=O)N/C=C/c2ccccc2)n1 ZINC000217635668 CG For-Sale Unstable GRM5 19 49 Cc1cccc(NC(=O)N/C=C/c2ccccc2)n1 ZINC000217635668 CG For-Sale Unstable SORT1 18 44 C[C@@H](N[C@@H]1CCC[C@@H](O)C1)c1ccc(Br)cc1 ZINC000217635686 CG For-Sale Unstable SDH1 0 50 CCN1CCN(C(=O)c2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217635730 CD For-Sale Unstable PARP1 15 43 CCN1CCN(C(=O)c2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217635730 CD For-Sale Unstable GPR183 0 46 C[C@H](N[C@@H]1CCC[C@@H](O)C1)c1ccc(Br)cc1 ZINC000217635767 CG On-Demand Unstable SDH1 0 50 O=C(N/C=C/c1ccccc1)NCCCCCO ZINC000217635795 BE For-Sale Unstable HDAC2 16 43 O=C(N/C=C/c1ccccc1)NCCCCCO ZINC000217635795 BE For-Sale Unstable HDAC9 35 43 O=C(N/C=C/c1ccccc1)NCCCCCO ZINC000217635795 BE For-Sale Unstable HDAC7 31 43 O=C(N/C=C/c1ccccc1)NCCCCCO ZINC000217635795 BE For-Sale Unstable AMP1_PLAFQ 20 43 O=C(N/C=C/c1ccccc1)NCCCCCO ZINC000217635795 BE For-Sale Unstable HDA106 0 42 COc1cccc(NC(=O)c2ccc(/C=C\C(=O)O)s2)c1 ZINC000217635809 DG For-Sale Unstable MTNR1A 17 42 COc1cccc(NC(=O)c2ccc(/C=C\C(=O)O)s2)c1 ZINC000217635809 DG For-Sale Unstable MTNR1B 24 42 COc1cccc(NC(=O)c2ccc(/C=C\C(=O)O)s2)c1 ZINC000217635809 DG For-Sale Unstable TAAR1 44 46 COc1cccc(NC(=O)c2ccc(/C=C\C(=O)O)s2)c1 ZINC000217635809 DG For-Sale Unstable KCNK3 112 49 COc1cccc(NC(=O)c2ccc(/C=C\C(=O)O)s2)c1 ZINC000217635809 DG For-Sale Unstable KCNK9 82 40 COc1cccc(NC(=O)c2ccc(/C=C\C(=O)O)s2)c1 ZINC000217635809 DG For-Sale Unstable BRPF1 0 41 C[C@@H](N[C@H]1CCC[C@@H](O)C1)c1ccc(Br)cc1 ZINC000217635861 CG For-Sale Unstable SDH1 0 50 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)NCc1ccncc1)C(=O)OC2 ZINC000217635864 HH In-Stock Unstable IMPDH1 0 63 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)NCc1ccncc1)C(=O)OC2 ZINC000217635864 HH In-Stock Unstable IMPDH2 0 63 COc1ncccc1-c1c(C(N)=O)sc2cnc(Nc3cccc(N4CCN(C)CC4)c3OC(C)C)nc12 ZINC000217635869 KI Annotated Unstable MAPK7 52 37 C[C@H](N[C@H]1CCC[C@@H](O)C1)c1ccc(Br)cc1 ZINC000217635945 CG On-Demand Unstable SDH1 0 50 Cn1cnnc1SCCNC(=O)c1ccc2c(c1)CCO2 ZINC000217636008 DD In-Stock Unstable MTNR1A 41 34 O=C(N/C=C/c1ccccc1)Nc1cccnc1 ZINC000217636011 BF For-Sale Anodyne NAMPT 38 50 O=C(N/C=C/c1ccccc1)Nc1cccnc1 ZINC000217636011 BF For-Sale Anodyne P95276_MYCTO 0 41 C[C@@H](N[C@@H]1CCC[C@@H](O)C1)c1ccc(Cl)cc1 ZINC000217636065 CG For-Sale Unstable SLC6A1 24 44 CC(C)(Oc1ccc(Cl)cc1)C(=O)N1CCS[C@@H]1c1ccsc1 ZINC000217636128 FJ In-Stock Unstable NPBWR1 44 34 CNC(=O)N/C=C/c1ccccc1 ZINC000217636133 AD For-Sale Unstable 17HSDCL 42 35 CNC(=O)N/C=C/c1ccccc1 ZINC000217636133 AD For-Sale Unstable TLR4 16 40 O=C(OCc1ccccc1)[C@@H]1CNCCC[C@@H]1O ZINC000217636144 BD For-Sale Unstable SLC12A5 53 36 C[C@H](N[C@@H]1CCC[C@@H](O)C1)c1ccc(Cl)cc1 ZINC000217636145 CG On-Demand Unstable SLC6A1 24 44 O=C(Cn1c(=O)[nH]c2ccccc2c1=O)NC[C@@H]1CC[C@@H](C(=O)N[C@@H](Cc2ccccc2)C(=O)O)CC1 ZINC000217636160 KD In-Stock Unstable AVPR1B 34 42 O=C(Cn1c(=O)[nH]c2ccccc2c1=O)NC[C@@H]1CC[C@@H](C(=O)N[C@@H](Cc2ccccc2)C(=O)O)CC1 ZINC000217636160 KD In-Stock Unstable MME 43 35 O=C(Cn1c(=O)[nH]c2ccccc2c1=O)NC[C@@H]1CC[C@@H](C(=O)N[C@@H](Cc2ccccc2)C(=O)O)CC1 ZINC000217636160 KD In-Stock Unstable EDNRA 44 34 O=C(Cn1c(=O)[nH]c2ccccc2c1=O)NC[C@@H]1CC[C@@H](C(=O)N[C@@H](Cc2ccccc2)C(=O)O)CC1 ZINC000217636160 KD In-Stock Unstable CMA1 48 33 O=C(Cn1c(=O)[nH]c2ccccc2c1=O)NC[C@@H]1CC[C@@H](C(=O)N[C@@H](Cc2ccccc2)C(=O)O)CC1 ZINC000217636160 KD In-Stock Unstable CTRA_BOVIN 47 33 O=C(Cn1c(=O)[nH]c2ccccc2c1=O)NC[C@@H]1CC[C@@H](C(=O)N[C@@H](Cc2ccccc2)C(=O)O)CC1 ZINC000217636160 KD In-Stock Unstable CCKAR 17 40 O=C(Cn1c(=O)[nH]c2ccccc2c1=O)NC[C@@H]1CC[C@@H](C(=O)N[C@@H](Cc2ccccc2)C(=O)O)CC1 ZINC000217636160 KD In-Stock Unstable ITGA4 58 37 O=C(Cn1c(=O)[nH]c2ccccc2c1=O)NC[C@@H]1CC[C@@H](C(=O)N[C@@H](Cc2ccccc2)C(=O)O)CC1 ZINC000217636160 KD In-Stock Unstable F11 49 38 O=C(Cn1c(=O)[nH]c2ccccc2c1=O)NC[C@@H]1CC[C@@H](C(=O)N[C@@H](Cc2ccccc2)C(=O)O)CC1 ZINC000217636160 KD In-Stock Unstable ACE2 48 33 O=C(Cn1c(=O)[nH]c2ccccc2c1=O)NC[C@@H]1CC[C@@H](C(=O)N[C@@H](Cc2ccccc2)C(=O)O)CC1 ZINC000217636160 KD In-Stock Unstable FPR1 53 35 COC(=O)C[C@H](c1ccc(OCCc2ccccc2)c(OC)c1)c1c(O)c2ccccc2oc1=O ZINC000217636181 JJ In-Stock Unstable NQO1 49 46 COC(=O)C[C@H](c1ccc(OCCc2ccccc2)c(OC)c1)c1c(O)c2ccccc2oc1=O ZINC000217636181 JJ In-Stock Unstable ABCG2 15 41 CCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636196 EG In-Stock Unstable ADRB2 15 47 CCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636196 EG In-Stock Unstable ADRB1 0 47 CCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636196 EG In-Stock Unstable ADRB3 21 47 CCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636196 EG In-Stock Unstable CA1 20 44 CCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636196 EG In-Stock Unstable PRTN3 56 37 CCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636196 EG In-Stock Unstable AKR1C2 47 34 CCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636196 EG In-Stock Unstable LIMK2 54 42 CCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636196 EG In-Stock Unstable MGAT1 46 39 O=C(OCc1ccccc1)[C@H]1CNCCC[C@@H]1O ZINC000217636209 BD For-Sale Unstable SLC12A5 53 36 CC(C)(Oc1ccc(Cl)cc1)C(=O)N1CCS[C@H]1c1ccsc1 ZINC000217636212 FJ In-Stock Unstable NPBWR1 44 34 C[C@@H](N[C@H]1CCC[C@@H](O)C1)c1ccc(Cl)cc1 ZINC000217636223 CG For-Sale Unstable SLC6A1 24 44 C=CC[C@@H](C#Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000217636250 CH For-Sale Unstable PAPA1_CARPA 39 42 C=CC[C@@H](C#Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000217636250 CH For-Sale Unstable CTSK 24 47 C=CC[C@@H](C#Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000217636250 CH For-Sale Unstable FPR1 47 37 COC(=O)C[C@@H](c1ccc(OCCc2ccccc2)c(OC)c1)c1c(O)c2ccccc2oc1=O ZINC000217636251 JJ In-Stock Unstable NQO1 49 46 COC(=O)C[C@@H](c1ccc(OCCc2ccccc2)c(OC)c1)c1c(O)c2ccccc2oc1=O ZINC000217636251 JJ In-Stock Unstable ABCG2 15 41 O=C(OCc1ccccc1)[C@@H]1CNCCC[C@H]1O ZINC000217636290 BD For-Sale Unstable SLC12A5 53 36 CC(C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636298 EG In-Stock Unstable CA2 17 40 CC(C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636298 EG In-Stock Unstable LPL 38 42 CC(C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636298 EG In-Stock Unstable CA4 30 40 CC(C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636298 EG In-Stock Unstable PRTN3 52 35 CC(C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636298 EG In-Stock Unstable MTNN 41 35 CC(C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636298 EG In-Stock Unstable AKR1C3 43 40 CC(C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636298 EG In-Stock Unstable LIPG 15 42 CC(C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636298 EG In-Stock Unstable AKR1C2 60 36 CC(C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636298 EG In-Stock Unstable LIMK2 53 42 CC(C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636298 EG In-Stock Unstable UQCRB 0 40 C[C@H](N[C@H]1CCC[C@@H](O)C1)c1ccc(Cl)cc1 ZINC000217636318 CG On-Demand Unstable SLC6A1 24 44 C=CC[C@H](C#Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000217636347 CH For-Sale Unstable PAPA1_CARPA 39 42 C=CC[C@H](C#Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000217636347 CH For-Sale Unstable CTSK 24 47 C=CC[C@H](C#Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000217636347 CH For-Sale Unstable FPR1 47 37 COC(=O)C[C@H](c1ccc(O)c(OC)c1)c1c(O)c2ccccc2oc1=O ZINC000217636352 FF In-Stock Unstable NQO1 51 40 CC[C@@H](CO)NC(=O)N/C=C/c1ccccc1 ZINC000217636358 BD For-Sale Unstable CTSC 15 41 O=C(OCc1ccccc1)[C@H]1CNCCC[C@H]1O ZINC000217636373 BD For-Sale Unstable SLC12A5 53 36 CCCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636398 EG In-Stock Unstable ADRB2 21 50 CCCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636398 EG In-Stock Unstable ADRB1 0 50 CCCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636398 EG In-Stock Unstable ADRB3 27 50 CCCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636398 EG In-Stock Unstable PRTN3 55 36 CCCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636398 EG In-Stock Unstable AKR1C2 43 33 CCCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636398 EG In-Stock Unstable LIMK2 52 40 CCCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636398 EG In-Stock Unstable MGAT1 45 38 CCC[C@@H](Nc1ccc(C(=O)NC(C)C)cc1[N+](=O)[O-])c1ccccc1 ZINC000217636427 FJ On-Demand Unstable BCL2L1 64 32 CCC[C@@H](Nc1ccc(C(=O)NC(C)C)cc1[N+](=O)[O-])c1ccccc1 ZINC000217636427 FJ On-Demand Unstable BCL2 50 31 CCC[C@@H](Nc1ccc(C(=O)NC(C)C)cc1[N+](=O)[O-])c1ccccc1 ZINC000217636427 FJ On-Demand Unstable TAAR1 20 48 CCC[C@@H](Nc1ccc(C(=O)NC(C)C)cc1[N+](=O)[O-])c1ccccc1 ZINC000217636427 FJ On-Demand Unstable UTS2 59 33 CC[C@H](CO)NC(=O)N/C=C/c1ccccc1 ZINC000217636440 BD For-Sale Unstable CTSC 15 41 COC(=O)C[C@@H](c1ccc(O)c(OC)c1)c1c(O)c2ccccc2oc1=O ZINC000217636444 FF In-Stock Unstable NQO1 51 40 O=C(O)[C@@H]1CC[C@@H](CNC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](Cc2ccccc2)n2c(=O)[nH]c3ccccc3c2=O)CC1 ZINC000217636469 KG In-Stock Unstable EDNRA 49 34 O=C(O)[C@@H]1CC[C@@H](CNC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](Cc2ccccc2)n2c(=O)[nH]c3ccccc3c2=O)CC1 ZINC000217636469 KG In-Stock Unstable PGC 41 33 O=C(O)[C@@H]1CC[C@@H](CNC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](Cc2ccccc2)n2c(=O)[nH]c3ccccc3c2=O)CC1 ZINC000217636469 KG In-Stock Unstable SSTR4 44 31 O=C(O)[C@@H]1CC[C@@H](CNC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](Cc2ccccc2)n2c(=O)[nH]c3ccccc3c2=O)CC1 ZINC000217636469 KG In-Stock Unstable TIMP3 61 36 O=C(O)[C@@H]1CC[C@@H](CNC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](Cc2ccccc2)n2c(=O)[nH]c3ccccc3c2=O)CC1 ZINC000217636469 KG In-Stock Unstable REN 43 34 O=C(O)[C@@H]1CC[C@@H](CNC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](Cc2ccccc2)n2c(=O)[nH]c3ccccc3c2=O)CC1 ZINC000217636469 KG In-Stock Unstable FPR1 51 35 CC(C)CNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636514 EG In-Stock Unstable ADRB2 21 40 CC(C)CNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636514 EG In-Stock Unstable ADRB1 16 40 CC(C)CNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636514 EG In-Stock Unstable ADRB3 29 40 CC(C)CNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636514 EG In-Stock Unstable BDKRB1 0 42 CC(C)CNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636514 EG In-Stock Unstable F3 41 32 CC(C)CNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636514 EG In-Stock Unstable PRTN3 53 35 CC(C)CNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636514 EG In-Stock Unstable MTNN 91 44 CC(C)CNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636514 EG In-Stock Unstable LIMK2 54 41 O=S(=O)(c1ccc2c(c1)OCCO2)N1CCS[C@@H]1c1ccsc1 ZINC000217636515 FF In-Stock Unstable PKM 29 44 CCC[C@H](Nc1ccc(C(=O)NC(C)C)cc1[N+](=O)[O-])c1ccccc1 ZINC000217636520 FJ On-Demand Unstable BCL2L1 64 32 CCC[C@H](Nc1ccc(C(=O)NC(C)C)cc1[N+](=O)[O-])c1ccccc1 ZINC000217636520 FJ On-Demand Unstable BCL2 50 31 CCC[C@H](Nc1ccc(C(=O)NC(C)C)cc1[N+](=O)[O-])c1ccccc1 ZINC000217636520 FJ On-Demand Unstable TAAR1 20 48 CCC[C@H](Nc1ccc(C(=O)NC(C)C)cc1[N+](=O)[O-])c1ccccc1 ZINC000217636520 FJ On-Demand Unstable UTS2 59 33 COc1cc2c(c(OC)c1OC)-c1ccc(NCCCCCC(=O)NCc3nc4ccccc4n3C(C)C)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217636565 KK In-Stock Unstable TUBA1A 16 55 O=S(=O)(c1ccc2c(c1)OCCO2)N1CCS[C@H]1c1ccsc1 ZINC000217636602 FF In-Stock Unstable PKM 29 44 CC[C@@H](C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636629 EG In-Stock Unstable ADRB2 15 42 CC[C@@H](C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636629 EG In-Stock Unstable ADRB1 0 44 CC[C@@H](C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636629 EG In-Stock Unstable ADRB3 17 42 CC[C@@H](C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636629 EG In-Stock Unstable MTNN 56 34 CC[C@@H](C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636629 EG In-Stock Unstable LIMK2 53 41 CC[C@@H](C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636629 EG In-Stock Unstable MGAT1 55 39 C[C@@H](NC(=O)C(F)F)c1ccc(F)cc1F ZINC000217636637 BE On-Demand Unstable SDH1 0 40 C[C@@H](NC(=O)C(F)F)c1ccc(F)cc1F ZINC000217636637 BE On-Demand Unstable BDKRB1 17 42 C[C@@H](NC(=O)C(F)F)c1ccc(F)cc1F ZINC000217636637 BE On-Demand Unstable CES2 20 46 CC(C)C[C@@H](NC(=O)[C@@H]1CC[C@@H](CNC(=O)Cn2c(=O)[nH]c3ccccc3c2=O)CC1)C(=O)O ZINC000217636710 JD In-Stock Unstable AVPR1B 37 42 CC(C)C[C@@H](NC(=O)[C@@H]1CC[C@@H](CNC(=O)Cn2c(=O)[nH]c3ccccc3c2=O)CC1)C(=O)O ZINC000217636710 JD In-Stock Unstable EDNRB 29 40 CC(C)C[C@@H](NC(=O)[C@@H]1CC[C@@H](CNC(=O)Cn2c(=O)[nH]c3ccccc3c2=O)CC1)C(=O)O ZINC000217636710 JD In-Stock Unstable EDNRA 25 40 CC(C)C[C@@H](NC(=O)[C@@H]1CC[C@@H](CNC(=O)Cn2c(=O)[nH]c3ccccc3c2=O)CC1)C(=O)O ZINC000217636710 JD In-Stock Unstable FPR1 46 34 CC(C)C[C@@H](NC(=O)[C@@H]1CC[C@@H](CNC(=O)Cn2c(=O)[nH]c3ccccc3c2=O)CC1)C(=O)O ZINC000217636710 JD In-Stock Unstable NPR 45 33 CC[C@H](C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636716 EG In-Stock Unstable ADRB2 15 42 CC[C@H](C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636716 EG In-Stock Unstable ADRB1 0 44 CC[C@H](C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636716 EG In-Stock Unstable ADRB3 17 42 CC[C@H](C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636716 EG In-Stock Unstable MTNN 56 34 CC[C@H](C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636716 EG In-Stock Unstable LIMK2 53 41 CC[C@H](C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636716 EG In-Stock Unstable MGAT1 55 39 C[C@H](NC(=O)C(F)F)c1ccc(F)cc1F ZINC000217636729 BE On-Demand Unstable SDH1 0 40 C[C@H](NC(=O)C(F)F)c1ccc(F)cc1F ZINC000217636729 BE On-Demand Unstable BDKRB1 17 42 C[C@H](NC(=O)C(F)F)c1ccc(F)cc1F ZINC000217636729 BE On-Demand Unstable CES2 20 46 O=C1CCCN1c1ccc(CN[C@@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217636763 CF For-Sale Unstable AKR1C3 22 40 CC(=O)Nc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217636765 CG For-Sale Unstable HDAC8 23 43 CC(=O)Nc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217636765 CG For-Sale Unstable HDAC6 15 43 CC(=O)Nc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217636765 CG For-Sale Unstable MMP1 0 47 CC(=O)Nc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217636765 CG For-Sale Unstable P95276_MYCTO 0 42 CC(=O)Nc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217636765 CG For-Sale Unstable KCNK3 113 39 CC(=O)Nc1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217636765 CG For-Sale Unstable KCNK9 78 39 CC(C)(C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636829 EG In-Stock Unstable LPL 31 42 CC(C)(C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636829 EG In-Stock Unstable PRTN3 62 42 CC(C)(C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636829 EG In-Stock Unstable AKR1C3 50 45 CC(C)(C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636829 EG In-Stock Unstable LIPG 15 42 CC(C)(C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636829 EG In-Stock Unstable AKR1C2 66 36 CC(C)(C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636829 EG In-Stock Unstable LIMK2 53 41 CC(C)(C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636829 EG In-Stock Unstable UQCRB 0 42 CC(C)(C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636829 EG In-Stock Unstable MGAT2 0 41 O=C(O)/C=C\c1cccc(C(=O)NC2CCCCCC2)c1 ZINC000217636837 CG For-Sale Unstable CNR1 17 40 O=C(O)/C=C\c1cccc(C(=O)NC2CCCCCC2)c1 ZINC000217636837 CG For-Sale Unstable CNR2 22 42 O=C(O)/C=C\c1cccc(C(=O)NC2CCCCCC2)c1 ZINC000217636837 CG For-Sale Unstable HDAC8 16 45 O=C(O)/C=C\c1cccc(C(=O)NC2CCCCCC2)c1 ZINC000217636837 CG For-Sale Unstable FAAH 17 45 O=C(O)/C=C\c1cccc(C(=O)NC2CCCCCC2)c1 ZINC000217636837 CG For-Sale Unstable EPHX2 23 41 O=C1CCCN1c1ccc(CN[C@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217636849 CF For-Sale Unstable AKR1C3 22 40 C[C@@H](NC(=O)C(F)F)c1cccc(C(F)(F)F)c1 ZINC000217636859 CG On-Demand Unstable PHES 0 43 Cc1c(NN)nc(C2CC2)nc1N[C@@H]1CC[C@@H](C)[C@@H](C)C1 ZINC000217636868 CG For-Sale Unstable CHRM3 0 56 COc1cc2c(c(OC)c1OC)-c1ccc(NCCCCCC(=O)NCCc3nc4ccccc4n3C(C)C)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217636889 KK In-Stock Unstable TUBA1A 15 53 COc1cccc([C@H]2SCCN2C(=O)c2ccsc2)c1 ZINC000217636891 DH In-Stock Unstable NPBWR1 52 30 O=C1CCCN1c1ccc(CN[C@@H]2C[C@H]3CC=C[C@H]32)cc1 ZINC000217636925 CF For-Sale Unstable AKR1C3 22 40 CC(C)CN(CC(C)C)C(=O)c1csc2ccccc12 ZINC000217636926 CJ On-Demand Unstable C5AR1 35 50 Cc1n[nH]c(C)c1NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217636929 CE For-Sale Unstable HDAC8 27 44 Cc1n[nH]c(C)c1NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217636929 CE For-Sale Unstable KCNK3 75 38 Cc1n[nH]c(C)c1NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217636929 CE For-Sale Unstable KCNK9 42 38 C[C@H](NC(=O)C(F)F)c1cccc(C(F)(F)F)c1 ZINC000217636938 CG On-Demand Unstable PHES 0 43 C=CCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636947 EF In-Stock Unstable PRTN3 44 33 C=CCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636947 EF In-Stock Unstable F13A1 46 32 C=CCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217636947 EF In-Stock Unstable LIMK2 51 40 Cc1c(NN)nc(C2CC2)nc1N[C@H]1CC[C@@H](C)[C@@H](C)C1 ZINC000217636972 CG For-Sale Unstable CHRM3 0 56 COc1cccc([C@@H]2SCCN2C(=O)c2ccsc2)c1 ZINC000217636973 DH In-Stock Unstable NPBWR1 52 30 COc1cccc(-c2cc3c(cc2[C@@H]2CCN(C)C[C@@H]2C)N2C(=NNC(=O)[C@H]2C)CO3)c1 ZINC000217636985 IG Annotated Unstable PRKCA 15 77 COc1cccc(-c2cc3c(cc2[C@@H]2CCN(C)C[C@@H]2C)N2C(=NNC(=O)[C@H]2C)CO3)c1 ZINC000217636985 IG Annotated Unstable PRKCQ 68 84 O=C1CCCN1c1ccc(CN[C@H]2C[C@H]3CC=C[C@@H]23)cc1 ZINC000217637019 CF For-Sale Unstable AKR1C3 22 40 O=[N+]([O-])c1cccc(S(=O)(=O)NCC2(c3ccccc3)CCC2)c1 ZINC000217637047 EF On-Demand Unstable ACAT 0 44 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NC1CC1 ZINC000217637058 EF In-Stock Unstable GRM4 15 42 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NC1CC1 ZINC000217637058 EF In-Stock Unstable SFRP1 74 34 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NC1CC1 ZINC000217637058 EF In-Stock Unstable LIMK2 50 38 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NC1CC1 ZINC000217637058 EF In-Stock Unstable WNT3 66 33 Cc1c(NN)nc(C2CC2)nc1N[C@@H]1CC[C@H](C)[C@@H](C)C1 ZINC000217637062 CG For-Sale Unstable CHRM3 0 56 CC[C@H](C)[C@@H](c1ccccc1)[C@@H](NN)C1CCCCCC1 ZINC000217637100 CJ For-Sale Unstable AMY2 47 34 Cc1c(NN)nc(C2CC2)nc1N[C@H]1CC[C@H](C)[C@@H](C)C1 ZINC000217637153 CG For-Sale Unstable CHRM3 0 56 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NC1CCCC1 ZINC000217637173 FH In-Stock Unstable GRM4 16 43 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NC1CCCC1 ZINC000217637173 FH In-Stock Unstable SFRP1 76 33 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NC1CCCC1 ZINC000217637173 FH In-Stock Unstable LIMK2 47 37 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NC1CCCC1 ZINC000217637173 FH In-Stock Unstable WNT3 63 33 COC(=O)c1ccccc1S(=O)(=O)NCC1(c2ccccc2)CCC1 ZINC000217637176 FF On-Demand Unstable KCNA3 44 45 COC(=O)c1ccccc1S(=O)(=O)NCC1(c2ccccc2)CCC1 ZINC000217637176 FF On-Demand Unstable ACAT 0 45 CC(C)(C)[C@@H]1CCCN(c2ccc(CBr)cc2)CC1 ZINC000217637194 DK For-Sale Unstable L3MBTL3 40 40 CCCN([C@@H]1CCNC1)[C@H](C)c1ccc(Br)cc1F ZINC000217637204 EH For-Sale Unstable SLC6A2 26 41 CSC1C[C@@H]2CC[C@H](C1)N2C(=O)c1ccco1 ZINC000217637247 CF In-Stock Unstable GLRA1 16 47 CC(C)(C)[C@H]1CCCN(c2ccc(CBr)cc2)CC1 ZINC000217637268 DK For-Sale Unstable L3MBTL3 40 40 CC[C@H](C)[C@H](c1ccccc1)[C@@H](NN)C1CCCCCC1 ZINC000217637282 CJ For-Sale Unstable AMY2 47 34 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NC1CCCCC1 ZINC000217637287 FH In-Stock Unstable GRM4 16 43 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NC1CCCCC1 ZINC000217637287 FH In-Stock Unstable EPHX2 22 41 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NC1CCCCC1 ZINC000217637287 FH In-Stock Unstable SFRP1 76 33 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NC1CCCCC1 ZINC000217637287 FH In-Stock Unstable LIMK2 46 36 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NC1CCCCC1 ZINC000217637287 FH In-Stock Unstable WNT3 62 33 CCCN([C@@H]1CCNC1)[C@H](C)c1cc(Br)ccc1F ZINC000217637291 EH For-Sale Unstable SLC6A2 26 41 C[C@@H](NC(=O)C(F)F)c1ccc(F)c(F)c1 ZINC000217637306 BE On-Demand Unstable SDH1 0 40 C[C@@H](NC(=O)C(F)F)c1ccc(F)c(F)c1 ZINC000217637306 BE On-Demand Unstable KCNQ2 46 35 C[C@H](NC(=O)C(F)F)c1ccc(F)c(F)c1 ZINC000217637390 BE On-Demand Unstable SDH1 0 40 C[C@H](NC(=O)C(F)F)c1ccc(F)c(F)c1 ZINC000217637390 BE On-Demand Unstable KCNQ2 46 35 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NCCC1=CCCCC1 ZINC000217637403 HI In-Stock Unstable LIMK2 49 39 COc1cc2c(cc1OC)CN(C(=O)Cn1c(C)nc3cc(OC)c(OC)cc3c1=O)CC2 ZINC000217637416 JE In-Stock Unstable ADRA1B 26 44 COc1cc2c(cc1OC)CN(C(=O)Cn1c(C)nc3cc(OC)c(OC)cc3c1=O)CC2 ZINC000217637416 JE In-Stock Unstable ABCC1 15 46 COc1cc2c(cc1OC)CN(C(=O)Cn1c(C)nc3cc(OC)c(OC)cc3c1=O)CC2 ZINC000217637416 JE In-Stock Unstable ABCB1B 70 45 COc1cc2c(cc1OC)CN(C(=O)Cn1c(C)nc3cc(OC)c(OC)cc3c1=O)CC2 ZINC000217637416 JE In-Stock Unstable ABCB1 15 48 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NCCO ZINC000217637503 ED In-Stock Unstable ADRB2 15 41 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NCCO ZINC000217637503 ED In-Stock Unstable PRTN3 49 39 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NCCO ZINC000217637503 ED In-Stock Unstable LIMK2 53 44 COc1cccc([C@H]2SCCN2C(=O)c2ccc3nsnc3c2)c1 ZINC000217637507 FH In-Stock Unstable DRD4 40 30 O=C(CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)N[C@H](CO)Cc1ccccc1 ZINC000217637515 GD In-Stock Unstable PLCD1 0 41 O=C(CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)N[C@H](CO)Cc1ccccc1 ZINC000217637515 GD In-Stock Unstable AGAL_COFAR 0 49 O=C(CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)N[C@H](CO)Cc1ccccc1 ZINC000217637515 GD In-Stock Unstable CYTH3 0 41 O=C(CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)N[C@H](CO)Cc1ccccc1 ZINC000217637515 GD In-Stock Unstable HLCS 0 50 O=C(CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)N[C@H](CO)Cc1ccccc1 ZINC000217637515 GD In-Stock Unstable BIRA 0 40 O=C(Nc1cccc(I)c1)C(F)F ZINC000217637524 CE On-Demand Anodyne KCNK3 82 39 O=C(Nc1cccc(I)c1)C(F)F ZINC000217637524 CE On-Demand Anodyne KCNK9 54 36 COc1cccc([C@@H]2SCCN2C(=O)c2ccc3nsnc3c2)c1 ZINC000217637591 FH In-Stock Unstable DRD4 40 30 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NCCCO ZINC000217637600 FD In-Stock Unstable PRTN3 47 35 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NCCCO ZINC000217637600 FD In-Stock Unstable LIMK2 52 42 CCCS(=O)(=O)NCc1cc(/C=C\C(=O)O)ccc1F ZINC000217637644 DD For-Sale Unstable AKR1C3 25 41 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable HRH2 23 40 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable SCNN1A 20 40 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable MME 66 45 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable ANPEP 55 59 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable SDH1 0 59 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable SIGMAR1 21 46 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable CTSB 23 43 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable CPA1 37 41 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable SCN2A 33 42 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable SLC15A1 0 40 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable NPFFR2 40 35 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable S1PR3 17 40 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable LIPC 0 48 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable MTNR1A 40 48 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable MTNR1B 63 48 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable MMP2 27 41 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable MMP3 51 41 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable MMP8 22 63 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable GRIA1 25 42 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable FAAH 54 43 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable PAM 0 47 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable FURIN 40 35 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable CAPN1 36 43 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable CES1 49 34 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable CAPN2 59 43 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable LAP3 45 38 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable POL 0 40 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable NPR 47 36 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable AMP1_PLAFQ 71 62 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable HDA106 0 51 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable POLG_WNV 48 34 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable CRTM 54 46 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable NPFFR1 55 35 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable PDS 38 42 O=C(NCCCc1ccccc1)C(F)F ZINC000217637653 BE On-Demand Unstable CES1D 43 31 N[C@@H]1CC[C@@H](NC(=O)c2cc(C(F)(F)F)ccc2Cl)C1 ZINC000217637668 DF In-Stock Unstable LIPC 0 41 N[C@@H]1CC[C@@H](NC(=O)c2cc(C(F)(F)F)ccc2Cl)C1 ZINC000217637668 DF In-Stock Unstable CCR2 26 41 N[C@@H]1CC[C@@H](NC(=O)c2cc(C(F)(F)F)ccc2Cl)C1 ZINC000217637668 DF In-Stock Unstable LIPG 35 41 COCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217637711 FE In-Stock Unstable ADRB3 17 40 COCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217637711 FE In-Stock Unstable GRM4 19 41 COCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217637711 FE In-Stock Unstable PRTN3 58 36 COCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217637711 FE In-Stock Unstable AKR1C3 40 36 COCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217637711 FE In-Stock Unstable AKR1C2 61 32 COCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217637711 FE In-Stock Unstable LIMK2 53 44 COc1ccc(/C=C\C(=O)O)cc1NS(=O)(=O)C(F)F ZINC000217637734 DD For-Sale Unstable TUBB1 49 38 COc1ccc(CNC(=O)C(F)F)cc1OC ZINC000217637769 BD On-Demand Unstable TRPV1 51 45 COc1ccc(CNC(=O)C(F)F)cc1OC ZINC000217637769 BD On-Demand Unstable MT-ND1 30 51 COc1ccc(CNC(=O)C(F)F)cc1OC ZINC000217637769 BD On-Demand Unstable LEF 40 33 COc1ccc(CNC(=O)C(F)F)cc1OC ZINC000217637769 BD On-Demand Unstable DRTS_TRYCR 52 36 COc1ccc(CNC(=O)C(F)F)cc1OC ZINC000217637769 BD On-Demand Unstable CAN2 0 42 COC(=O)COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OC ZINC000217637803 KG In-Stock Unstable ALOX5 0 42 COC(=O)COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OC ZINC000217637803 KG In-Stock Unstable CYP1B1 46 39 COC(=O)COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OC ZINC000217637803 KG In-Stock Unstable CYP1A1 46 39 COC(=O)COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OC ZINC000217637803 KG In-Stock Unstable ABCB1A 22 41 CCCS(=O)(=O)Nc1cc(/C=C\C(=O)O)ccc1OC ZINC000217637813 CD For-Sale Unstable TUBB1 52 38 CCCS(=O)(=O)Nc1cc(/C=C\C(=O)O)ccc1OC ZINC000217637813 CD For-Sale Unstable AKR1C3 29 40 COCCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217637828 FF In-Stock Unstable ADRB2 15 41 COCCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217637828 FF In-Stock Unstable BDKRB1 21 42 COCCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217637828 FF In-Stock Unstable GRM4 17 40 COCCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217637828 FF In-Stock Unstable PRTN3 56 35 COCCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217637828 FF In-Stock Unstable AKR1C2 61 33 COCCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217637828 FF In-Stock Unstable LIMK2 51 42 COC(=O)COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OC ZINC000217637893 KG In-Stock Unstable ALOX5 0 42 COC(=O)COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OC ZINC000217637893 KG In-Stock Unstable CYP1B1 46 39 COC(=O)COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OC ZINC000217637893 KG In-Stock Unstable CYP1A1 46 39 COC(=O)COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OC ZINC000217637893 KG In-Stock Unstable ABCB1A 22 41 O=C(C(F)F)N1CCN(c2ncccn2)CC1 ZINC000217637894 BC On-Demand Unstable SLC6A7 0 51 COc1cccc([C@H]2SCCN2C(=O)c2cccc(C(F)(F)F)c2)c1 ZINC000217637913 FJ In-Stock Unstable CACNA1B 47 33 COc1cccc([C@H]2SCCN2C(=O)c2cccc(C(F)(F)F)c2)c1 ZINC000217637913 FJ In-Stock Unstable CCR2 49 46 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NCc1ccccc1 ZINC000217637941 GH In-Stock Unstable CA2 23 43 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NCc1ccccc1 ZINC000217637941 GH In-Stock Unstable CA1 24 43 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NCc1ccccc1 ZINC000217637941 GH In-Stock Unstable GRM4 15 42 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NCc1ccccc1 ZINC000217637941 GH In-Stock Unstable PRTN3 46 34 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NCc1ccccc1 ZINC000217637941 GH In-Stock Unstable MTNN 42 34 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NCc1ccccc1 ZINC000217637941 GH In-Stock Unstable CA9 15 45 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NCc1ccccc1 ZINC000217637941 GH In-Stock Unstable LIMK2 58 45 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NCc1ccccc1 ZINC000217637941 GH In-Stock Unstable NAMPT 27 43 COc1cccc([C@@H]2SCCN2C(=O)c2cccc(C(F)(F)F)c2)c1 ZINC000217637986 FJ In-Stock Unstable CACNA1B 47 33 COc1cccc([C@@H]2SCCN2C(=O)c2cccc(C(F)(F)F)c2)c1 ZINC000217637986 FJ In-Stock Unstable CCR2 49 46 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1OC(=O)Cc1ccccc1N ZINC000217637990 CH For-Sale Unstable TRPM8 16 42 CC(=O)Nc1cccc2c1ccn2CC(=O)N1CCc2[nH]c3ccccc3c2C1 ZINC000217638019 GH In-Stock Unstable FABI 44 30 C[C@@H](Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217638040 GI In-Stock Unstable ADRB1 0 44 C[C@@H](Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217638040 GI In-Stock Unstable LIMK2 50 39 CC(C)(F)c1ccc(CCC(=O)O)c(Cl)c1 ZINC000217638059 BH For-Sale Unstable FFAR1 40 36 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1OC(=O)Cc1ccccc1N ZINC000217638063 CH For-Sale Unstable TRPM8 16 42 C[C@@H](OCCCNc1nc2c(cc1C#N)CCCC2)c1ccccc1 ZINC000217638112 EI On-Demand Unstable BCHE 45 33 C[C@H](Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217638115 GI In-Stock Unstable ADRB1 0 44 C[C@H](Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O)c1ccccc1 ZINC000217638115 GI In-Stock Unstable LIMK2 50 39 O=C(N/C=C/c1ccccc1)Nc1ccccc1N1CCOCC1 ZINC000217638125 DG For-Sale Unstable KCNQ2 86 45 O=C(N/C=C/c1ccccc1)Nc1ccccc1N1CCOCC1 ZINC000217638125 DG For-Sale Unstable KCNQ4 0 40 O=C(N/C=C/c1ccccc1)Nc1ccccc1N1CCOCC1 ZINC000217638125 DG For-Sale Unstable CSF1R 0 49 O=C(N/C=C/c1ccccc1)Nc1ccccc1N1CCOCC1 ZINC000217638125 DG For-Sale Unstable AKR1C3 26 43 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1OC(=O)Cc1ccccc1N ZINC000217638142 CH For-Sale Unstable TRPM8 16 42 COc1ccc(/C=C2\Oc3c(ccc4c3[C@H](c3ccc(O)c(OC)c3)CC(=O)O4)C2=O)cc1 ZINC000217638158 II In-Stock Unstable HSD17B3 15 42 CC(C)(F)c1c(Cl)cccc1CCC(=O)O ZINC000217638169 BH For-Sale Unstable CXCL8 44 36 CC(C)(F)c1c(Cl)cccc1CCC(=O)O ZINC000217638169 BH For-Sale Unstable FFAR1 45 38 CC(C)(F)c1c(Cl)cccc1CCC(=O)O ZINC000217638169 BH For-Sale Unstable FFAR4 45 33 Clc1cccc(N2CCc3ccccc3CC2)c1CBr ZINC000217638200 FJ For-Sale Unstable DRD3 17 41 C[C@H](OCCCNc1nc2c(cc1C#N)CCCC2)c1ccccc1 ZINC000217638207 EI On-Demand Unstable BCHE 45 33 CS(=O)(=O)CCCNC(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217638216 DC For-Sale Unstable HDA106 0 41 CC(C)[C@H]1CC[C@H](C)C[C@@H]1OC(=O)Cc1ccccc1N ZINC000217638219 CH For-Sale Unstable TRPM8 16 42 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NCCc1ccccc1 ZINC000217638222 GH In-Stock Unstable CA2 28 40 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NCCc1ccccc1 ZINC000217638222 GH In-Stock Unstable ADRB2 47 39 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NCCc1ccccc1 ZINC000217638222 GH In-Stock Unstable ADRB1 34 43 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NCCc1ccccc1 ZINC000217638222 GH In-Stock Unstable ADRB3 59 46 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NCCc1ccccc1 ZINC000217638222 GH In-Stock Unstable CA1 30 40 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NCCc1ccccc1 ZINC000217638222 GH In-Stock Unstable CA4 24 40 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NCCc1ccccc1 ZINC000217638222 GH In-Stock Unstable PRTN3 46 33 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NCCc1ccccc1 ZINC000217638222 GH In-Stock Unstable CA12 17 43 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NCCc1ccccc1 ZINC000217638222 GH In-Stock Unstable CA9 22 43 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NCCc1ccccc1 ZINC000217638222 GH In-Stock Unstable AKR1C3 27 46 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NCCc1ccccc1 ZINC000217638222 GH In-Stock Unstable NCE103 19 40 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NCCc1ccccc1 ZINC000217638222 GH In-Stock Unstable LIMK2 59 46 CN1CCN(c2ccc(NC(=O)N/C=C/c3ccccc3)cc2)CC1 ZINC000217638236 EG For-Sale Unstable ERBB2 0 40 CN1CCN(c2ccc(NC(=O)N/C=C/c3ccccc3)cc2)CC1 ZINC000217638236 EG For-Sale Unstable LCK 19 40 CN1CCN(c2ccc(NC(=O)N/C=C/c3ccccc3)cc2)CC1 ZINC000217638236 EG For-Sale Unstable PRNP 44 55 CN1CCN(c2ccc(NC(=O)N/C=C/c3ccccc3)cc2)CC1 ZINC000217638236 EG For-Sale Unstable MTOR 29 45 CN1CCN(c2ccc(NC(=O)N/C=C/c3ccccc3)cc2)CC1 ZINC000217638236 EG For-Sale Unstable HCK 24 41 CN1CCN(c2ccc(NC(=O)N/C=C/c3ccccc3)cc2)CC1 ZINC000217638236 EG For-Sale Unstable FLT3 19 50 CN1CCN(c2ccc(NC(=O)N/C=C/c3ccccc3)cc2)CC1 ZINC000217638236 EG For-Sale Unstable AURKA 17 50 CN1CCN(c2ccc(NC(=O)N/C=C/c3ccccc3)cc2)CC1 ZINC000217638236 EG For-Sale Unstable ADAM10 25 40 C[C@@H](NC(=O)C(F)F)C12CC3CC(CC(C3)C1)C2 ZINC000217638237 CF On-Demand Unstable EPHX2 0 57 COc1ccc(/C=C2\Oc3c(ccc4c3[C@@H](c3ccc(O)c(OC)c3)CC(=O)O4)C2=O)cc1 ZINC000217638249 II In-Stock Unstable HSD17B3 15 42 C[C@@H](CC(=O)O)c1cccc(Cl)c1[C@@H](C)F ZINC000217638284 BH For-Sale Unstable CXCL8 44 35 COc1cccc([C@H]2SCCN2C(=O)c2csc(-c3ccccc3)n2)c1 ZINC000217638300 GJ In-Stock Unstable PTGER1 15 41 C[C@H](NC(=O)C(F)F)C12CC3CC(CC(C3)C1)C2 ZINC000217638317 CF On-Demand Unstable EPHX2 0 57 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1 ZINC000217638319 IH In-Stock Unstable CA2 24 40 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1 ZINC000217638319 IH In-Stock Unstable ADRB2 60 45 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1 ZINC000217638319 IH In-Stock Unstable ADRB1 52 45 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1 ZINC000217638319 IH In-Stock Unstable ADRB3 89 45 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1 ZINC000217638319 IH In-Stock Unstable BMP1 84 48 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1 ZINC000217638319 IH In-Stock Unstable CA1 26 43 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1 ZINC000217638319 IH In-Stock Unstable KCNA5 26 41 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1 ZINC000217638319 IH In-Stock Unstable MMP13 66 41 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1 ZINC000217638319 IH In-Stock Unstable HTR6 0 42 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1 ZINC000217638319 IH In-Stock Unstable ADAM17 46 40 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1 ZINC000217638319 IH In-Stock Unstable MMP2 43 39 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1 ZINC000217638319 IH In-Stock Unstable MMP3 50 40 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1 ZINC000217638319 IH In-Stock Unstable PRTN3 58 37 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1 ZINC000217638319 IH In-Stock Unstable PTPRB 50 39 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1 ZINC000217638319 IH In-Stock Unstable MMP9 58 41 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1 ZINC000217638319 IH In-Stock Unstable CA12 17 43 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1 ZINC000217638319 IH In-Stock Unstable PTGDR 26 42 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1 ZINC000217638319 IH In-Stock Unstable MMP7 33 40 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1 ZINC000217638319 IH In-Stock Unstable IAP 0 41 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1 ZINC000217638319 IH In-Stock Unstable CA9 28 43 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1 ZINC000217638319 IH In-Stock Unstable MMP1 59 41 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1 ZINC000217638319 IH In-Stock Unstable AKR1C3 38 42 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1 ZINC000217638319 IH In-Stock Unstable AKR1C2 62 40 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1 ZINC000217638319 IH In-Stock Unstable LIMK2 54 44 CS(=O)(=O)CCCNC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217638339 DC For-Sale Unstable HDAC8 16 42 O=C(N/C=C/c1ccccc1)Nc1ccc(N2CCCCC2)cc1 ZINC000217638361 DI For-Sale Unstable LPL 43 37 O=C(N/C=C/c1ccccc1)Nc1ccc(N2CCCCC2)cc1 ZINC000217638361 DI For-Sale Unstable KCNQ2 32 47 O=C(N/C=C/c1ccccc1)Nc1ccc(N2CCCCC2)cc1 ZINC000217638361 DI For-Sale Unstable PRNP 39 40 C[C@@H](F)c1c(Cl)cccc1[C@H](C)CC(=O)O ZINC000217638372 BH For-Sale Unstable CXCL8 44 35 COc1cccc([C@@H]2SCCN2C(=O)c2csc(-c3ccccc3)n2)c1 ZINC000217638382 GJ In-Stock Unstable PTGER1 15 41 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1OC ZINC000217638432 JH In-Stock Unstable ADRB2 21 40 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1OC ZINC000217638432 JH In-Stock Unstable FKBP1A 18 40 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1OC ZINC000217638432 JH In-Stock Unstable ADRB3 51 38 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1OC ZINC000217638432 JH In-Stock Unstable HTR6 0 43 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1OC ZINC000217638432 JH In-Stock Unstable CPT1A 44 30 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1OC ZINC000217638432 JH In-Stock Unstable PRTN3 45 32 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1OC ZINC000217638432 JH In-Stock Unstable PTGDR 24 41 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1OC ZINC000217638432 JH In-Stock Unstable IAP 0 43 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1OC ZINC000217638432 JH In-Stock Unstable LIMK2 50 38 COc1ccc(CCNc2ccc(S(=O)(=O)Nc3ccccc3)cc2C(=O)O)cc1OC ZINC000217638432 JH In-Stock Unstable SCMU_MYCTU 0 45 CC(C)CCNS(=O)(=O)c1ccc(CCO)cc1 ZINC000217638444 CD For-Sale Unstable CA2 26 49 CC(C)CCNS(=O)(=O)c1ccc(CCO)cc1 ZINC000217638444 CD For-Sale Unstable TBXA2R 48 36 CC(C)CCNS(=O)(=O)c1ccc(CCO)cc1 ZINC000217638444 CD For-Sale Unstable CA1 23 49 CC(C)CCNS(=O)(=O)c1ccc(CCO)cc1 ZINC000217638444 CD For-Sale Unstable CHUK 15 40 CC(C)CCNS(=O)(=O)c1ccc(CCO)cc1 ZINC000217638444 CD For-Sale Unstable CA4 16 49 CC(C)CCNS(=O)(=O)c1ccc(CCO)cc1 ZINC000217638444 CD For-Sale Unstable ALOX15 51 40 CC(C)CCNS(=O)(=O)c1ccc(CCO)cc1 ZINC000217638444 CD For-Sale Unstable CA12 16 49 CC(C)CCNS(=O)(=O)c1ccc(CCO)cc1 ZINC000217638444 CD For-Sale Unstable CA9 20 49 CC(C)CCNS(=O)(=O)c1ccc(CCO)cc1 ZINC000217638444 CD For-Sale Unstable CA 0 49 CC(C)CCNS(=O)(=O)c1ccc(CCO)cc1 ZINC000217638444 CD For-Sale Unstable A6YCJ1_9METZ 25 49 CC(C)CCNS(=O)(=O)c1ccc(CCO)cc1 ZINC000217638444 CD For-Sale Unstable Q5TU56_ANOGA 0 49 C[C@H](F)c1c(Cl)cccc1[C@@H](C)CC(=O)O ZINC000217638463 BH For-Sale Unstable CXCL8 44 35 COc1cccc([C@H]2SCCN2C(=O)c2cc(-c3ccc(F)cc3)nn2C)c1 ZINC000217638491 GI In-Stock Unstable TACR3 17 44 COc1cccc([C@H]2SCCN2C(=O)c2cc(-c3ccc(F)cc3)nn2C)c1 ZINC000217638491 GI In-Stock Unstable NR1H2 0 42 C[C@@H](c1ccc(Br)cc1F)N1CCC[C@@H](CCN)C1 ZINC000217638500 EH For-Sale Unstable GHSR 21 41 Cc1nnc(CNC(=O)c2ccccc2N2CCOCC2)o1 ZINC000217638529 DD In-Stock Unstable STAT6 53 34 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NCc1ccco1 ZINC000217638547 FG In-Stock Unstable LIMK2 45 36 C[C@H](F)c1c(Cl)cccc1[C@H](C)CC(=O)O ZINC000217638548 BH For-Sale Unstable CXCL8 44 35 Clc1cccc(CN[C@@H]2CCN3CCCC[C@@H]23)c1Cl ZINC000217638553 CH On-Demand Unstable P2RX7 18 42 COc1cccc([C@@H]2SCCN2C(=O)c2cc(-c3ccc(F)cc3)nn2C)c1 ZINC000217638572 GI In-Stock Unstable TACR3 17 44 COc1cccc([C@@H]2SCCN2C(=O)c2cc(-c3ccc(F)cc3)nn2C)c1 ZINC000217638572 GI In-Stock Unstable NR1H2 0 42 C[C@H](c1ccc(Br)cc1F)N1CCC[C@@H](CCN)C1 ZINC000217638575 EH For-Sale Unstable GHSR 21 41 CN(C)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217638576 CH For-Sale Unstable CA1 18 44 N#Cc1cccc(NC(=O)C(F)F)c1 ZINC000217638597 AD On-Demand Mild MCHR1 25 40 N#Cc1cccc(NC(=O)C(F)F)c1 ZINC000217638597 AD On-Demand Mild PARP10 45 33 COc1cccc(O)c1/C=C/C(C)=O ZINC000217638618 AE For-Sale Unstable CYP1B1 19 44 COc1cccc(O)c1/C=C/C(C)=O ZINC000217638618 AE For-Sale Unstable CYP1A1 16 44 COc1cccc(O)c1/C=C/C(C)=O ZINC000217638618 AE For-Sale Unstable TUBB1 36 40 COc1cccc(O)c1/C=C/C(C)=O ZINC000217638618 AE For-Sale Unstable ABCG2 23 53 COc1cccc(O)c1/C=C/C(C)=O ZINC000217638618 AE For-Sale Unstable CYSP_PLAFA 21 51 Clc1cccc(CN[C@H]2CCN3CCCC[C@@H]23)c1Cl ZINC000217638644 CH On-Demand Unstable P2RX7 18 42 C[C@@H](Cc1cccc(Cl)c1[C@@H](C)F)C(=O)O ZINC000217638657 BH For-Sale Unstable CXCL8 53 33 C[C@@H](c1cc(Br)ccc1F)N1CCC[C@@H](CCN)C1 ZINC000217638662 EH For-Sale Unstable GHSR 21 40 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NC[C@@H]1CCCO1 ZINC000217638666 GF In-Stock Unstable POL 0 40 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NC[C@@H]1CCCO1 ZINC000217638666 GF In-Stock Unstable TNK2 55 40 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NC[C@@H]1CCCO1 ZINC000217638666 GF In-Stock Unstable LIMK2 49 37 N#Cc1cc2c(nc1NC1CCN(Cc3ccc(Cl)cc3)CC1)CCCC2 ZINC000217638706 GJ On-Demand Unstable DRD4 24 42 N#Cc1cc2c(nc1NC1CCN(Cc3ccc(Cl)cc3)CC1)CCCC2 ZINC000217638706 GJ On-Demand Unstable SIGMAR1 15 40 N#Cc1cc2c(nc1NC1CCN(Cc3ccc(Cl)cc3)CC1)CCCC2 ZINC000217638706 GJ On-Demand Unstable SSTR5 61 40 N#Cc1cc2c(nc1NC1CCN(Cc3ccc(Cl)cc3)CC1)CCCC2 ZINC000217638706 GJ On-Demand Unstable CXCR3 25 40 N#Cc1cc2c(nc1NC1CCN(Cc3ccc(Cl)cc3)CC1)CCCC2 ZINC000217638706 GJ On-Demand Unstable MCHR1 26 52 Cn1cccc(C(=O)NC[C@@H]2CCCN2c2nc3ccccc3o2)c1=O ZINC000217638727 FD In-Stock Unstable HTR3A 30 40 Cn1cccc(C(=O)NC[C@@H]2CCCN2c2nc3ccccc3o2)c1=O ZINC000217638727 FD In-Stock Unstable HCRTR1 39 40 Cn1cccc(C(=O)NC[C@@H]2CCCN2c2nc3ccccc3o2)c1=O ZINC000217638727 FD In-Stock Unstable HCRTR2 15 40 Cn1cccc(C(=O)NC[C@@H]2CCCN2c2nc3ccccc3o2)c1=O ZINC000217638727 FD In-Stock Unstable POLR1A 69 36 C[C@H](Cc1cccc(Cl)c1[C@@H](C)F)C(=O)O ZINC000217638737 BH For-Sale Unstable CXCL8 53 33 CCCCCCCCN[C@@H]1CCN2CCCC[C@@H]12 ZINC000217638744 CH For-Sale Unstable GLB1 33 42 COc1ccc(CCNC(=O)C(F)F)cc1OC ZINC000217638746 CD On-Demand Unstable NQO2 45 32 COc1ccc(CCNC(=O)C(F)F)cc1OC ZINC000217638746 CD On-Demand Unstable TRPV1 22 43 COc1ccc(CCNC(=O)C(F)F)cc1OC ZINC000217638746 CD On-Demand Unstable RAF1 24 40 COc1ccc(CCNC(=O)C(F)F)cc1OC ZINC000217638746 CD On-Demand Unstable MTNR1A 41 37 COc1ccc(CCNC(=O)C(F)F)cc1OC ZINC000217638746 CD On-Demand Unstable ABCB1 0 43 COc1ccc(CCNC(=O)C(F)F)cc1OC ZINC000217638746 CD On-Demand Unstable MT-ND1 26 42 COc1ccc(CCNC(=O)C(F)F)cc1OC ZINC000217638746 CD On-Demand Unstable Q8MMZ8_EIMTE 0 40 COc1ccc(CCNC(=O)C(F)F)cc1OC ZINC000217638746 CD On-Demand Unstable LEF 49 37 COc1ccc(CCNC(=O)C(F)F)cc1OC ZINC000217638746 CD On-Demand Unstable SCMU_MYCTU 0 41 COc1ccc(CCNC(=O)C(F)F)cc1OC ZINC000217638746 CD On-Demand Unstable CAN2 0 56 C[C@H](c1cc(Br)ccc1F)N1CCC[C@@H](CCN)C1 ZINC000217638749 EH For-Sale Unstable GHSR 21 40 CC[C@@H](C)[C@@H](CO)NC(=O)CN1C=Cc2cc(OC)c(OC)cc2CC1=O ZINC000217638759 GD In-Stock Unstable HCN2 0 44 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NC[C@H]1CCCO1 ZINC000217638767 GF In-Stock Unstable POL 0 40 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NC[C@H]1CCCO1 ZINC000217638767 GF In-Stock Unstable TNK2 55 40 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1NC[C@H]1CCCO1 ZINC000217638767 GF In-Stock Unstable LIMK2 49 37 BrCc1ccc(N2CCc3ccccc3CC2)nc1 ZINC000217638792 DH For-Sale Unstable SMO 28 40 Cn1cccc(C(=O)NC[C@H]2CCCN2c2nc3ccccc3o2)c1=O ZINC000217638802 FD In-Stock Unstable HTR3A 30 40 Cn1cccc(C(=O)NC[C@H]2CCCN2c2nc3ccccc3o2)c1=O ZINC000217638802 FD In-Stock Unstable HCRTR1 39 40 Cn1cccc(C(=O)NC[C@H]2CCCN2c2nc3ccccc3o2)c1=O ZINC000217638802 FD In-Stock Unstable HCRTR2 15 40 Cn1cccc(C(=O)NC[C@H]2CCCN2c2nc3ccccc3o2)c1=O ZINC000217638802 FD In-Stock Unstable POLR1A 69 36 O=C(N/C=C/c1ccccc1)Nc1cccc2ccccc12 ZINC000217638807 CJ For-Sale Anodyne CHAT 45 35 O=C(N/C=C/c1ccccc1)Nc1cccc2ccccc12 ZINC000217638807 CJ For-Sale Anodyne TRPV1 48 49 O=C(N/C=C/c1ccccc1)Nc1cccc2ccccc12 ZINC000217638807 CJ For-Sale Anodyne CASP9 15 40 O=C(N/C=C/c1ccccc1)Nc1cccc2ccccc12 ZINC000217638807 CJ For-Sale Anodyne 17HSDCL 0 43 O=C(N/C=C/c1ccccc1)Nc1cccc2ccccc12 ZINC000217638807 CJ For-Sale Anodyne HDAH 18 40 C[C@@H](Cc1cccc(Cl)c1[C@H](C)F)C(=O)O ZINC000217638816 BH For-Sale Unstable CXCL8 53 33 CCCCCCCCN[C@H]1CCN2CCCC[C@@H]12 ZINC000217638817 CH For-Sale Unstable GLB1 33 42 COc1ccc2c(c1OC)C(=O)O[C@@H]2CC(=O)Nc1ccc2oc(=O)ccc2c1 ZINC000217638866 GG In-Stock Unstable CA7 0 40 COc1ccc2c(c1OC)C(=O)O[C@@H]2CC(=O)Nc1ccc2oc(=O)ccc2c1 ZINC000217638866 GG In-Stock Unstable ENPP1 60 31 CCOc1ccc([C@@H](C)N[C@@H]2CCC[C@@H](O)C2)cc1 ZINC000217638867 CG For-Sale Unstable ACACA 35 42 COc1ccccc1CNC(=O)C(F)F ZINC000217638872 BD On-Demand Unstable GRIN2B 24 50 COc1ccccc1CNC(=O)C(F)F ZINC000217638872 BD On-Demand Unstable ANPEP 29 56 COc1ccccc1CNC(=O)C(F)F ZINC000217638872 BD On-Demand Unstable TACR1 24 45 COc1ccccc1CNC(=O)C(F)F ZINC000217638872 BD On-Demand Unstable P2RX7 18 47 COc1ccccc1CNC(=O)C(F)F ZINC000217638872 BD On-Demand Unstable AMP1_PLAFQ 45 36 COc1ccccc1CNC(=O)C(F)F ZINC000217638872 BD On-Demand Unstable PHES 0 43 COc1ccccc1CNC(=O)C(F)F ZINC000217638872 BD On-Demand Unstable GPM3 0 50 COc1ccccc1CNC(=O)C(F)F ZINC000217638872 BD On-Demand Unstable CARM1 24 42 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1N1CCCC1 ZINC000217638874 EF In-Stock Unstable ADRB2 0 54 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1N1CCCC1 ZINC000217638874 EF In-Stock Unstable ADRB1 0 53 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1N1CCCC1 ZINC000217638874 EF In-Stock Unstable KCNQ2 74 38 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1N1CCCC1 ZINC000217638874 EF In-Stock Unstable HTR6 23 42 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1N1CCCC1 ZINC000217638874 EF In-Stock Unstable CA4 18 40 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1N1CCCC1 ZINC000217638874 EF In-Stock Unstable SLC6A9 15 43 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1N1CCCC1 ZINC000217638874 EF In-Stock Unstable AKR1C3 19 40 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1N1CCCC1 ZINC000217638874 EF In-Stock Unstable SFRP1 91 35 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1N1CCCC1 ZINC000217638874 EF In-Stock Unstable LIMK2 49 39 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1N1CCCC1 ZINC000217638874 EF In-Stock Unstable WNT3 77 34 C[C@H](F)c1c(Cl)cccc1C[C@@H](C)C(=O)O ZINC000217638903 BH For-Sale Unstable CXCL8 53 33 CCCCCCN[C@@H]1CCN2CCCC[C@@H]12 ZINC000217638916 BF For-Sale Unstable GLB1 33 42 COC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217638942 CG For-Sale Unstable ACR 67 39 COc1ccc2c(c1OC)C(=O)O[C@H]2CC(=O)Nc1ccc2oc(=O)ccc2c1 ZINC000217638952 GG In-Stock Unstable CA7 0 40 COc1ccc2c(c1OC)C(=O)O[C@H]2CC(=O)Nc1ccc2oc(=O)ccc2c1 ZINC000217638952 GG In-Stock Unstable ENPP1 60 31 CCOc1ccc([C@H](C)N[C@@H]2CCC[C@@H](O)C2)cc1 ZINC000217638968 CG On-Demand Unstable ACACA 35 42 CCCCCCN[C@H]1CCN2CCCC[C@@H]12 ZINC000217638988 BF For-Sale Unstable GLB1 33 42 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1N1CCCCC1 ZINC000217638992 FG In-Stock Unstable ADRB2 0 53 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1N1CCCCC1 ZINC000217638992 FG In-Stock Unstable ADRB1 0 52 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1N1CCCCC1 ZINC000217638992 FG In-Stock Unstable KCNQ2 67 37 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1N1CCCCC1 ZINC000217638992 FG In-Stock Unstable HTR6 22 41 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1N1CCCCC1 ZINC000217638992 FG In-Stock Unstable AKR1C3 17 40 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1N1CCCCC1 ZINC000217638992 FG In-Stock Unstable SFRP1 88 34 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1N1CCCCC1 ZINC000217638992 FG In-Stock Unstable LIMK2 48 38 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1N1CCCCC1 ZINC000217638992 FG In-Stock Unstable WNT3 77 34 CC(C)CCNS(=O)(=O)c1ccc(F)c(CO)c1 ZINC000217639002 CD For-Sale Unstable LEF 59 38 O=C(Nc1ccc(Cl)c(C(F)(F)F)c1)C(F)F ZINC000217639003 CH On-Demand Anodyne RAF1 34 45 O=C(Nc1ccc(Cl)c(C(F)(F)F)c1)C(F)F ZINC000217639003 CH On-Demand Anodyne ENV 42 32 O=C(Nc1ccc(Cl)c(C(F)(F)F)c1)C(F)F ZINC000217639003 CH On-Demand Anodyne Q8MMZ8_EIMTE 55 45 O=C(Nc1ccc(Cl)c(C(F)(F)F)c1)C(F)F ZINC000217639003 CH On-Demand Anodyne BRAF 16 43 O=C(Nc1ccc(Cl)c(C(F)(F)F)c1)C(F)F ZINC000217639003 CH On-Demand Anodyne IMDH_CRYPV 34 51 O=C(N/C=C/c1ccccc1)N(Cc1ccccc1)c1ccccc1 ZINC000217639050 EK For-Sale Unstable NR1H4 42 39 CCOc1ccc([C@@H](C)N[C@H]2CCC[C@@H](O)C2)cc1 ZINC000217639051 CG For-Sale Unstable ACACA 35 42 NC/C=C\CN1CCCc2ccccc2C1 ZINC000217639076 BD For-Sale Unstable CHRNA6 0 41 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1N1CCOCC1 ZINC000217639099 FE In-Stock Unstable ADRB1 0 49 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1N1CCOCC1 ZINC000217639099 FE In-Stock Unstable HTR6 0 42 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1N1CCOCC1 ZINC000217639099 FE In-Stock Unstable SLC6A9 0 47 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1N1CCOCC1 ZINC000217639099 FE In-Stock Unstable SFRP1 42 37 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1N1CCOCC1 ZINC000217639099 FE In-Stock Unstable LIMK2 46 36 O=C(O)c1cc(S(=O)(=O)Nc2ccccc2)ccc1N1CCOCC1 ZINC000217639099 FE In-Stock Unstable WNT3 48 37 CCOc1ccc([C@H](C)N[C@H]2CCC[C@@H](O)C2)cc1 ZINC000217639145 CG On-Demand Unstable ACACA 35 42 O=C(NCCc1ccc(Cl)cc1Cl)C(F)F ZINC000217639146 CF On-Demand Unstable CNR1 32 48 O=C(NCCc1ccc(Cl)cc1Cl)C(F)F ZINC000217639146 CF On-Demand Unstable P2RX7 67 44 O=C(NCCc1ccc(Cl)cc1Cl)C(F)F ZINC000217639146 CF On-Demand Unstable MC3R 36 40 O=C(NCCc1ccc(Cl)cc1Cl)C(F)F ZINC000217639146 CF On-Demand Unstable MC5R 64 42 O=C(NCCc1ccc(Cl)cc1Cl)C(F)F ZINC000217639146 CF On-Demand Unstable EPHX2 16 41 O=C(NCCc1ccc(Cl)cc1Cl)C(F)F ZINC000217639146 CF On-Demand Unstable PTGDR 21 41 O=C(NCCc1ccc(Cl)cc1Cl)C(F)F ZINC000217639146 CF On-Demand Unstable ALPL 44 36 CN(C(=O)c1cccc(/C=C\C(=O)O)c1)C1CCCCC1 ZINC000217639152 CG For-Sale Unstable ACE 38 42 CC[C@@H](COC)NC(=O)/C=C\C(=O)O ZINC000217639155 BC For-Sale Unstable HCAR2 32 41 O=C(N/C=C/c1ccccc1)Nc1ccc2ccccc2c1 ZINC000217639168 CJ For-Sale Anodyne CA1 22 47 O=C(N/C=C/c1ccccc1)Nc1ccc2ccccc2c1 ZINC000217639168 CJ For-Sale Anodyne IMDH_CRYPV 24 41 CCOCCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217639202 GG In-Stock Unstable PRTN3 54 34 CCOCCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217639202 GG In-Stock Unstable LIMK2 49 37 O=C(O)/C=C\c1cccc(C(=O)NCCc2cccs2)c1 ZINC000217639243 DF For-Sale Unstable ADAM17 17 41 CC[C@H](COC)NC(=O)/C=C\C(=O)O ZINC000217639255 BC For-Sale Unstable HCAR2 32 41 CN(C(=O)N/C=C/c1ccccc1)c1ccc(O)cc1 ZINC000217639283 CG For-Sale Unstable F3 24 43 COc1cccc([C@H]2SCCN2S(=O)(=O)c2cc3c4c(c2)CCN4C(=O)CC3)c1 ZINC000217639306 IF In-Stock Unstable CYP11B1 34 46 COc1cccc([C@H]2SCCN2S(=O)(=O)c2cc3c4c(c2)CCN4C(=O)CC3)c1 ZINC000217639306 IF In-Stock Unstable CYP11B2 36 51 Oc1ccc(Cl)c(F)c1CN1CCNCC1 ZINC000217639325 BD On-Demand Unstable CXCR4 20 40 CC(C)OCCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217639331 GG In-Stock Unstable ADRB2 26 40 CC(C)OCCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217639331 GG In-Stock Unstable ADRB1 19 40 CC(C)OCCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217639331 GG In-Stock Unstable ADRB3 25 40 CC(C)OCCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217639331 GG In-Stock Unstable PRTN3 54 34 CC(C)OCCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217639331 GG In-Stock Unstable MTNN 41 34 CC(C)OCCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217639331 GG In-Stock Unstable LIMK2 52 39 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1OC(=O)c1cc(N)cc(N)c1 ZINC000217639362 CG For-Sale Unstable TRPM8 0 40 CCCCN(C)C(=O)N/C=C/c1ccccc1 ZINC000217639400 BG For-Sale Unstable TSPO 29 40 COc1cccc([C@@H]2SCCN2S(=O)(=O)c2cc3c4c(c2)CCN4C(=O)CC3)c1 ZINC000217639402 IF In-Stock Unstable CYP11B1 34 46 COc1cccc([C@@H]2SCCN2S(=O)(=O)c2cc3c4c(c2)CCN4C(=O)CC3)c1 ZINC000217639402 IF In-Stock Unstable CYP11B2 36 51 Oc1c(Cl)ccc(F)c1CN1CCNCC1 ZINC000217639432 BD For-Sale Unstable CXCR4 20 40 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1OC(=O)c1cc(N)cc(N)c1 ZINC000217639441 CG For-Sale Unstable TRPM8 0 40 O=C(C(F)F)N1CCN(c2ccccn2)CC1 ZINC000217639458 BC On-Demand Unstable DRD4 30 42 O=C(C(F)F)N1CCN(c2ccccn2)CC1 ZINC000217639458 BC On-Demand Unstable EBP 27 42 O=C(C(F)F)N1CCN(c2ccccn2)CC1 ZINC000217639458 BC On-Demand Unstable SMO 0 40 O=C(C(F)F)N1CCN(c2ccccn2)CC1 ZINC000217639458 BC On-Demand Unstable SLC6A7 0 57 CCCCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217639463 FH In-Stock Unstable ADRB2 23 54 CCCCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217639463 FH In-Stock Unstable ADRB1 22 54 CCCCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217639463 FH In-Stock Unstable ADRB3 26 54 CCCCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217639463 FH In-Stock Unstable PRTN3 48 35 CCCCCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217639463 FH In-Stock Unstable LIMK2 52 40 CN1C[C@@]2(CCCN(C(=O)CCc3cccnc3)C2)OC1=O ZINC000217639479 DD In-Stock Unstable C3AR1 50 45 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1OC(=O)c1cc(N)cc(N)c1 ZINC000217639532 CG For-Sale Unstable TRPM8 0 40 CN1C[C@]2(CCCN(C(=O)CCc3cccnc3)C2)OC1=O ZINC000217639561 DD In-Stock Unstable C3AR1 50 45 CC(C)CCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217639573 FH In-Stock Unstable ADRB2 18 40 CC(C)CCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217639573 FH In-Stock Unstable ADRB1 0 45 CC(C)CCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217639573 FH In-Stock Unstable ADRB3 19 40 CC(C)CCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217639573 FH In-Stock Unstable PRTN3 48 34 CC(C)CCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217639573 FH In-Stock Unstable MTNN 72 35 CC(C)CCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217639573 FH In-Stock Unstable LIMK2 52 40 CCNC(=O)N1CCN(c2ccc(C(=O)NC(C)C)cc2[N+](=O)[O-])CC1 ZINC000217639582 FD On-Demand Unstable CXCR3 19 43 CCNC(=O)N1CCN(c2ccc(C(=O)NC(C)C)cc2[N+](=O)[O-])CC1 ZINC000217639582 FD On-Demand Unstable TAAR1 28 48 Nc1nc(C(F)F)c2nc[nH]c2n1 ZINC000217639593 AC In-Stock Unstable GDA 0 59 Nc1nc(C(F)F)c2nc[nH]c2n1 ZINC000217639593 AC In-Stock Unstable MGMT 33 43 COc1ccc(C(=O)Nc2cn[nH]c2)cc1/C=C\C(=O)O ZINC000217639596 CD For-Sale Unstable CPT1A 52 46 COc1ccc(C(=O)Nc2cn[nH]c2)cc1/C=C\C(=O)O ZINC000217639596 CD For-Sale Unstable KCNK3 78 38 COc1ccc(C(=O)Nc2cn[nH]c2)cc1/C=C\C(=O)O ZINC000217639596 CD For-Sale Unstable KCNK9 53 38 CC[C@@H]1CC[C@@H](N)[C@@H](CCCc2ccccc2)C1 ZINC000217639599 BI For-Sale Unstable SLC18A2 44 45 CC[C@@H]1CC[C@@H](N)[C@@H](CCCc2ccccc2)C1 ZINC000217639599 BI For-Sale Unstable SIGMAR1 20 40 CC(C)[C@H]1CC[C@H](C)C[C@@H]1OC(=O)c1cc(N)cc(N)c1 ZINC000217639615 CG For-Sale Unstable TRPM8 0 40 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc(O)c2)CC(=O)O4)cc1O ZINC000217639627 II In-Stock Unstable AKR1B1 0 47 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc(O)c2)CC(=O)O4)cc1O ZINC000217639627 II In-Stock Unstable CYP1B1 66 38 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc(O)c2)CC(=O)O4)cc1O ZINC000217639627 II In-Stock Unstable CYP1A1 49 49 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc(O)c2)CC(=O)O4)cc1O ZINC000217639627 II In-Stock Unstable CYP1A2 41 41 Cc1nc2ccccc2n1C/C=C\CN ZINC000217639646 BD For-Sale Unstable PDE6D 17 41 Cc1cccc(C(=O)c2ccccc2C(=O)O)n1 ZINC000217639671 BE For-Sale Unstable SORT1 22 44 Cc1cccc(C(=O)c2ccccc2C(=O)O)n1 ZINC000217639671 BE For-Sale Unstable ALS 73 35 Cc1cccc(C(=O)c2ccccc2C(=O)O)n1 ZINC000217639671 BE For-Sale Unstable MT-CO2 46 33 CCC[C@@H](C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217639684 FH In-Stock Unstable ADRB1 0 43 CCC[C@@H](C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217639684 FH In-Stock Unstable LIMK2 51 39 CC[C@H](C)[C@H](NC(=O)[C@@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217639687 KG In-Stock Unstable EDNRA 59 38 CC[C@H](C)[C@H](NC(=O)[C@@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217639687 KG In-Stock Unstable BMP1 57 35 CC[C@H](C)[C@H](NC(=O)[C@@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217639687 KG In-Stock Unstable POL 0 42 CC[C@H]1CC[C@@H](N)[C@@H](CCCc2ccccc2)C1 ZINC000217639689 BI For-Sale Unstable SLC18A2 44 45 CC[C@H]1CC[C@@H](N)[C@@H](CCCc2ccccc2)C1 ZINC000217639689 BI For-Sale Unstable SIGMAR1 20 40 CCNC(=O)N1CCN(c2ccc(C(=O)NC3CC3)cc2[N+](=O)[O-])CC1 ZINC000217639704 FD On-Demand Unstable CXCR3 20 42 CCNC(=O)N1CCN(c2ccc(C(=O)NC3CC3)cc2[N+](=O)[O-])CC1 ZINC000217639704 FD On-Demand Unstable TAAR1 15 43 COc1cccc([C@H]2SCCN2C(=O)Nc2ccccc2C)c1 ZINC000217639708 EI In-Stock Unstable P2RX7 28 43 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc(O)c2)CC(=O)O4)cc1O ZINC000217639720 II In-Stock Unstable AKR1B1 0 47 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc(O)c2)CC(=O)O4)cc1O ZINC000217639720 II In-Stock Unstable CYP1B1 66 38 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc(O)c2)CC(=O)O4)cc1O ZINC000217639720 II In-Stock Unstable CYP1A1 49 49 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc(O)c2)CC(=O)O4)cc1O ZINC000217639720 II In-Stock Unstable CYP1A2 41 41 CCC[C@H](C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217639751 FH In-Stock Unstable ADRB1 0 43 CCC[C@H](C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217639751 FH In-Stock Unstable LIMK2 51 39 NC/C=C\CN1c2ccccc2Sc2ccccc21 ZINC000217639758 CH For-Sale Unstable BCHE 0 41 CC[C@@H]1CC[C@H](N)[C@@H](CCCc2ccccc2)C1 ZINC000217639766 BI For-Sale Unstable SLC18A2 44 45 CC[C@@H]1CC[C@H](N)[C@@H](CCCc2ccccc2)C1 ZINC000217639766 BI For-Sale Unstable SIGMAR1 20 40 CCCCCN(C)C(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217639767 CG For-Sale Unstable THRA 44 38 CCCCCN(C)C(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217639767 CG For-Sale Unstable PLM2_PLAFA 24 40 COc1cccc([C@@H]2SCCN2C(=O)Nc2ccccc2C)c1 ZINC000217639777 EI In-Stock Unstable P2RX7 28 43 CCNc1nc(Cl)nc(C(F)F)c1N ZINC000217639814 BE In-Stock Unstable PPX1 0 40 N#Cc1cc2c(nc1NCCCOc1ccccc1)CCCC2 ZINC000217639815 DH On-Demand Unstable ACHE 45 41 N#Cc1cc2c(nc1NCCCOc1ccccc1)CCCC2 ZINC000217639815 DH On-Demand Unstable BCHE 69 38 O=CNCCCNC(=O)N/C=C/c1ccccc1 ZINC000217639845 BD For-Sale Unstable HDAC9 27 40 COC[C@@H](C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217639849 FF In-Stock Unstable AKR1C2 40 31 CC[C@H]1CC[C@H](N)[C@@H](CCCc2ccccc2)C1 ZINC000217639861 BI For-Sale Unstable SLC18A2 44 45 CC[C@H]1CC[C@H](N)[C@@H](CCCc2ccccc2)C1 ZINC000217639861 BI For-Sale Unstable SIGMAR1 20 40 CCCCCN(C)C(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217639866 CG For-Sale Unstable LTB4R 15 53 CCCCCN(C)C(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217639866 CG For-Sale Unstable TTR 0 43 CCCCCN(C)C(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217639866 CG For-Sale Unstable AKR1C3 25 41 O=C(O)[C@@H]1CC[C@@H](CNC(=O)[C@@H](Cc2ccccc2)n2c(=O)[nH]c3ccccc3c2=O)CC1 ZINC000217639895 IE In-Stock Unstable SSTR4 51 35 O=C(O)[C@@H]1CC[C@@H](CNC(=O)[C@@H](Cc2ccccc2)n2c(=O)[nH]c3ccccc3c2=O)CC1 ZINC000217639895 IE In-Stock Unstable SSTR5 41 35 Cc1cccc(-c2ccccc2C(=O)N2CCC[C@@H](c3nc(C)n[nH]3)C2)c1 ZINC000217639901 FI In-Stock Unstable MAP3K12 36 42 COC[C@H](C)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217639915 FF In-Stock Unstable AKR1C2 40 31 COc1cccc([C@H]2SCCN2C(=O)Nc2ccccc2F)c1 ZINC000217639917 EI In-Stock Unstable DRD4 40 31 Cc1cccc(-c2ccccc2C(=O)N2CCC[C@H](c3nc(C)n[nH]3)C2)c1 ZINC000217639980 FI In-Stock Unstable MAP3K12 36 42 CNCCNc1ccnc(N)n1 ZINC000217639988 AB For-Sale Unstable HRH4 0 82 COc1cccc([C@@H]2SCCN2C(=O)Nc2ccccc2F)c1 ZINC000217639997 EI In-Stock Unstable DRD4 40 31 CC(C)c1cccc(NC(=O)C(F)F)c1 ZINC000217640022 BG On-Demand Unstable PSBA 0 41 CC(C)c1cccc(NC(=O)C(F)F)c1 ZINC000217640022 BG On-Demand Unstable KCNK3 77 38 CC(C)c1cccc(NC(=O)C(F)F)c1 ZINC000217640022 BG On-Demand Unstable KCNK9 69 38 CCCNc1ccc(S(=O)(=O)NCCCOCC)cc1C(=O)O ZINC000217640025 ED In-Stock Unstable CASP3 15 44 Nc1c(NCc2ccccc2)nc(Cl)nc1C(F)F ZINC000217640049 CG In-Stock Unstable PETD 0 42 Nc1c(NCc2ccccc2)nc(Cl)nc1C(F)F ZINC000217640049 CG In-Stock Unstable Q31945_CHEAL 0 42 COc1cccc([C@H]2SCCN2C(=O)Nc2ccc3c(c2)OCO3)c1 ZINC000217640103 FH In-Stock Unstable EDNRB 54 40 COc1cccc([C@H]2SCCN2C(=O)Nc2ccc3c(c2)OCO3)c1 ZINC000217640103 FH In-Stock Unstable EDNRA 45 39 CC1(C)C[C@H]2C[C@@](C)(CN2C(=O)N/C=C/c2ccccc2)C1 ZINC000217640128 CI For-Sale Unstable AVPR2 17 47 CC1(C)C[C@H]2C[C@@](C)(CN2C(=O)N/C=C/c2ccccc2)C1 ZINC000217640128 CI For-Sale Unstable AVPR1A 39 47 CCOCCCNS(=O)(=O)c1ccc(NC(C)C)c(C(=O)O)c1 ZINC000217640135 ED In-Stock Unstable CASP3 16 42 CCOC(=O)N1CCC(NC(=O)C(F)F)CC1 ZINC000217640157 CC On-Demand Unstable EPHX2 25 41 COc1cccc([C@@H]2SCCN2C(=O)Nc2ccc3c(c2)OCO3)c1 ZINC000217640187 FH In-Stock Unstable EDNRB 54 40 COc1cccc([C@@H]2SCCN2C(=O)Nc2ccc3c(c2)OCO3)c1 ZINC000217640187 FH In-Stock Unstable EDNRA 45 39 CCCCNc1ccc(S(=O)(=O)NCCCOCC)cc1C(=O)O ZINC000217640225 FE In-Stock Unstable CASP3 22 44 CC[S@@](=O)CCn1c(=O)cc(O)[nH]c1=O ZINC000217640233 BB For-Sale Unstable POLC 65 34 O=C1N[C@@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)C(=O)Nc2ccccc21 ZINC000217640279 GE In-Stock Unstable SSTR4 49 32 O=C1N[C@@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)C(=O)Nc2ccccc21 ZINC000217640279 GE In-Stock Unstable SSTR5 40 33 COCCNc1nc2cc(C(=O)NC[C@@H]3CCCCO3)ccc2n1C ZINC000217640294 ED In-Stock Unstable ITK 43 40 CCCCOc1ccc(NC(=O)N2CCS[C@@H]2c2cccc(OC)c2)cc1 ZINC000217640312 GK In-Stock Unstable HRH2 19 41 CCCCOc1ccc(NC(=O)N2CCS[C@@H]2c2cccc(OC)c2)cc1 ZINC000217640312 GK In-Stock Unstable PDGFRB 56 41 CCCCOc1ccc(NC(=O)N2CCS[C@@H]2c2cccc(OC)c2)cc1 ZINC000217640312 GK In-Stock Unstable MMP13 19 42 CCCCOc1ccc(NC(=O)N2CCS[C@@H]2c2cccc(OC)c2)cc1 ZINC000217640312 GK In-Stock Unstable MTNR1A 34 44 CCCCOc1ccc(NC(=O)N2CCS[C@@H]2c2cccc(OC)c2)cc1 ZINC000217640312 GK In-Stock Unstable MTNR1B 39 44 CCCCOc1ccc(NC(=O)N2CCS[C@@H]2c2cccc(OC)c2)cc1 ZINC000217640312 GK In-Stock Unstable PLA2G4B 53 36 CCCCOc1ccc(NC(=O)N2CCS[C@@H]2c2cccc(OC)c2)cc1 ZINC000217640312 GK In-Stock Unstable FAAH 26 41 CCCCOc1ccc(NC(=O)N2CCS[C@@H]2c2cccc(OC)c2)cc1 ZINC000217640312 GK In-Stock Unstable CFTR 47 33 CC[S@](=O)CCn1c(=O)cc(O)[nH]c1=O ZINC000217640313 BB For-Sale Unstable POLC 65 34 CN(C)c1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217640324 CH For-Sale Unstable KCNK3 53 46 CCCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217640326 BH On-Demand Unstable THRA 0 47 CCCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217640326 BH On-Demand Unstable INHA 85 46 CCCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217640326 BH On-Demand Unstable BDKRB2 26 46 CCCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217640326 BH On-Demand Unstable SCN2A 27 64 CCCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217640326 BH On-Demand Unstable S1PR4 53 58 CCCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217640326 BH On-Demand Unstable S1PR3 37 58 CCCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217640326 BH On-Demand Unstable MMP2 18 41 CCCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217640326 BH On-Demand Unstable MMP3 30 41 CCCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217640326 BH On-Demand Unstable FAAH 20 43 CCCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217640326 BH On-Demand Unstable CFTR 48 39 CCCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217640326 BH On-Demand Unstable S1PR2 61 58 CCCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217640326 BH On-Demand Unstable S1PR1 25 58 CCCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217640326 BH On-Demand Unstable SPHK1 33 64 CCCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217640326 BH On-Demand Unstable S1PR5 53 58 CCCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217640326 BH On-Demand Unstable PLM2_PLAFA 70 39 CCCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217640326 BH On-Demand Unstable ENPP2 31 43 CCCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217640326 BH On-Demand Unstable LIPG 19 44 CCCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217640326 BH On-Demand Unstable ACAT 0 54 CCCCCc1ccc(NC(=O)C(F)F)cc1 ZINC000217640326 BH On-Demand Unstable UNG 0 41 CCOCCCNS(=O)(=O)c1ccc(NCC(C)C)c(C(=O)O)c1 ZINC000217640330 FE In-Stock Unstable CASP3 0 43 COCCNc1nc2cc(C(=O)NC[C@H]3CCCCO3)ccc2n1C ZINC000217640390 ED In-Stock Unstable ITK 43 40 CCCCOc1ccc(NC(=O)N2CCS[C@H]2c2cccc(OC)c2)cc1 ZINC000217640391 GK In-Stock Unstable HRH2 19 41 CCCCOc1ccc(NC(=O)N2CCS[C@H]2c2cccc(OC)c2)cc1 ZINC000217640391 GK In-Stock Unstable PDGFRB 56 41 CCCCOc1ccc(NC(=O)N2CCS[C@H]2c2cccc(OC)c2)cc1 ZINC000217640391 GK In-Stock Unstable MMP13 19 42 CCCCOc1ccc(NC(=O)N2CCS[C@H]2c2cccc(OC)c2)cc1 ZINC000217640391 GK In-Stock Unstable MTNR1A 34 44 CCCCOc1ccc(NC(=O)N2CCS[C@H]2c2cccc(OC)c2)cc1 ZINC000217640391 GK In-Stock Unstable MTNR1B 39 44 CCCCOc1ccc(NC(=O)N2CCS[C@H]2c2cccc(OC)c2)cc1 ZINC000217640391 GK In-Stock Unstable PLA2G4B 53 36 CCCCOc1ccc(NC(=O)N2CCS[C@H]2c2cccc(OC)c2)cc1 ZINC000217640391 GK In-Stock Unstable FAAH 26 41 CCCCOc1ccc(NC(=O)N2CCS[C@H]2c2cccc(OC)c2)cc1 ZINC000217640391 GK In-Stock Unstable CFTR 47 33 FC(F)c1nc(Cl)nc2c1ncn2Cc1ccccc1 ZINC000217640397 CG In-Stock Unstable Q6R7Z5_9TRYP 0 44 CCOCCCNS(=O)(=O)c1ccc(N[C@@H](C)CC)c(C(=O)O)c1 ZINC000217640421 FE In-Stock Unstable CASP3 0 44 CN1CCc2nc(NC(=O)N/C=C/c3ccccc3)sc2C1 ZINC000217640444 DF For-Sale Unstable F10 26 48 CCOCCCNS(=O)(=O)c1ccc(N[C@H](C)CC)c(C(=O)O)c1 ZINC000217640497 FE In-Stock Unstable CASP3 0 44 Cc1cc(C(=O)N2CCS[C@@H]2c2ccc(Cl)c(Cl)c2)no1 ZINC000217640504 EI In-Stock Unstable KCNA5 27 41 CC(C)(O)[C@@H]1CCN(C(=O)c2ccc(N)nc2)C1 ZINC000217640521 BC In-Stock Unstable L3MBTL1 0 42 CC(C)(O)[C@@H]1CCN(C(=O)c2ccc(N)nc2)C1 ZINC000217640521 BC In-Stock Unstable L3MBTL3 50 37 Cc1cccc(NC(=O)c2ccc(/C=C\C(=O)O)s2)n1 ZINC000217640558 CF For-Sale Unstable GRM5 21 50 Cc1cccc(NC(=O)c2ccc(/C=C\C(=O)O)s2)n1 ZINC000217640558 CF For-Sale Unstable SORT1 23 45 Cc1cc(C(=O)N2CCS[C@H]2c2ccc(Cl)c(Cl)c2)no1 ZINC000217640588 EI In-Stock Unstable KCNA5 26 43 N#Cc1cc2c(nc1NCCCc1nc3ccccc3[nH]1)CCCC2 ZINC000217640597 EH On-Demand Unstable ACHE 46 37 N#Cc1cc2c(nc1NCCCc1nc3ccccc3[nH]1)CCCC2 ZINC000217640597 EH On-Demand Unstable BCHE 55 37 CC(C)(O)[C@H]1CCN(C(=O)c2ccc(N)nc2)C1 ZINC000217640600 BC In-Stock Unstable L3MBTL1 0 42 CC(C)(O)[C@H]1CCN(C(=O)c2ccc(N)nc2)C1 ZINC000217640600 BC In-Stock Unstable L3MBTL3 50 37 CCOCCCNS(=O)(=O)c1ccc(NC(C)(C)C)c(C(=O)O)c1 ZINC000217640624 FE In-Stock Unstable CASP3 0 42 Cc1cccc(NC(=O)c2ccc(/C=C\C(=O)O)cc2)n1 ZINC000217640641 CF For-Sale Unstable GRM5 25 54 Cc1cccc(NC(=O)c2ccc(/C=C\C(=O)O)cc2)n1 ZINC000217640641 CF For-Sale Unstable SORT1 28 48 Cc1cccc(NC(=O)c2ccc(/C=C\C(=O)O)cc2)n1 ZINC000217640641 CF For-Sale Unstable MAP3K5 51 36 Cc1cccc(NC(=O)c2ccc(/C=C\C(=O)O)cc2)n1 ZINC000217640641 CF For-Sale Unstable KCNK3 48 36 O=C(Cn1c(=O)[nH]c2ccccc2c1=O)NC[C@@H]1CC[C@@H](C(=O)N[C@H](Cc2ccccc2)C(=O)O)CC1 ZINC000217640689 KD In-Stock Unstable AVPR1B 34 42 O=C(Cn1c(=O)[nH]c2ccccc2c1=O)NC[C@@H]1CC[C@@H](C(=O)N[C@H](Cc2ccccc2)C(=O)O)CC1 ZINC000217640689 KD In-Stock Unstable MME 43 35 O=C(Cn1c(=O)[nH]c2ccccc2c1=O)NC[C@@H]1CC[C@@H](C(=O)N[C@H](Cc2ccccc2)C(=O)O)CC1 ZINC000217640689 KD In-Stock Unstable EDNRB 60 37 O=C(Cn1c(=O)[nH]c2ccccc2c1=O)NC[C@@H]1CC[C@@H](C(=O)N[C@H](Cc2ccccc2)C(=O)O)CC1 ZINC000217640689 KD In-Stock Unstable EDNRA 44 34 O=C(Cn1c(=O)[nH]c2ccccc2c1=O)NC[C@@H]1CC[C@@H](C(=O)N[C@H](Cc2ccccc2)C(=O)O)CC1 ZINC000217640689 KD In-Stock Unstable CMA1 48 33 O=C(Cn1c(=O)[nH]c2ccccc2c1=O)NC[C@@H]1CC[C@@H](C(=O)N[C@H](Cc2ccccc2)C(=O)O)CC1 ZINC000217640689 KD In-Stock Unstable CTRA_BOVIN 47 33 O=C(Cn1c(=O)[nH]c2ccccc2c1=O)NC[C@@H]1CC[C@@H](C(=O)N[C@H](Cc2ccccc2)C(=O)O)CC1 ZINC000217640689 KD In-Stock Unstable CCKAR 17 40 O=C(Cn1c(=O)[nH]c2ccccc2c1=O)NC[C@@H]1CC[C@@H](C(=O)N[C@H](Cc2ccccc2)C(=O)O)CC1 ZINC000217640689 KD In-Stock Unstable ITGA4 58 37 O=C(Cn1c(=O)[nH]c2ccccc2c1=O)NC[C@@H]1CC[C@@H](C(=O)N[C@H](Cc2ccccc2)C(=O)O)CC1 ZINC000217640689 KD In-Stock Unstable F11 49 38 O=C(Cn1c(=O)[nH]c2ccccc2c1=O)NC[C@@H]1CC[C@@H](C(=O)N[C@H](Cc2ccccc2)C(=O)O)CC1 ZINC000217640689 KD In-Stock Unstable ACE2 48 33 O=C(Cn1c(=O)[nH]c2ccccc2c1=O)NC[C@@H]1CC[C@@H](C(=O)N[C@H](Cc2ccccc2)C(=O)O)CC1 ZINC000217640689 KD In-Stock Unstable FPR1 53 35 O=S(=O)(Cl)CCc1ccc2occc2c1 ZINC000217640716 BF For-Sale Unstable CYP2A6 15 42 Nc1nc(C(F)F)c2ncn(Cc3ccccc3)c2n1 ZINC000217640720 CE In-Stock Unstable ADORA2A 25 49 Nc1nc(C(F)F)c2ncn(Cc3ccccc3)c2n1 ZINC000217640720 CE In-Stock Unstable Q6R7Z5_9TRYP 0 43 Nc1nc(C(F)F)c2ncn(Cc3ccccc3)c2n1 ZINC000217640720 CE In-Stock Unstable TAG 0 40 Cc1cccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)n1 ZINC000217640724 CF For-Sale Unstable HDAC8 43 46 Cc1cccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)n1 ZINC000217640724 CF For-Sale Unstable HDAC6 27 46 Cc1cccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)n1 ZINC000217640724 CF For-Sale Unstable GRM5 27 61 Cc1cccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)n1 ZINC000217640724 CF For-Sale Unstable SORT1 28 49 Cc1cccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)n1 ZINC000217640724 CF For-Sale Unstable KCNK3 91 40 Cc1cccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)n1 ZINC000217640724 CF For-Sale Unstable KCNK9 48 40 O=C(COc1ccc2nncn2n1)N1CCC[C@@H]1c1ccccn1 ZINC000217640732 DD In-Stock Unstable CPT1A 116 44 C=CCNc1ccc(S(=O)(=O)NCCCOCC)cc1C(=O)O ZINC000217640734 ED In-Stock Unstable CASP3 0 42 CSC1C[C@@H]2CC[C@H](C1)N2C(=O)COc1ccccc1 ZINC000217640775 CF In-Stock Unstable CPT1A 117 42 CSC1C[C@@H]2CC[C@H](C1)N2C(=O)COc1ccccc1 ZINC000217640775 CF In-Stock Unstable CPT2 47 37 CSC1C[C@@H]2CC[C@H](C1)N2C(=O)COc1ccccc1 ZINC000217640775 CF In-Stock Unstable GLRA1 42 31 Clc1ccccc1CN[C@@H]1CCN2CCCC[C@@H]12 ZINC000217640801 CG On-Demand Unstable SLC18A3 52 38 O=C(COc1ccc2nncn2n1)N1CCC[C@H]1c1ccccn1 ZINC000217640811 DD In-Stock Unstable CPT1A 116 44 O=C(O)/C=C\c1ccc(C(=O)NCc2cccs2)cc1 ZINC000217640814 CF For-Sale Unstable PYGM 32 44 COc1ccccc1[C@@H](CNC(=O)c1csc2ccccc12)N1CCCC1 ZINC000217640818 GI On-Demand Unstable DRD2 20 46 COc1ccccc1[C@@H](CNC(=O)c1csc2ccccc12)N1CCCC1 ZINC000217640818 GI On-Demand Unstable DRD3 26 41 COc1ccccc1[C@@H](CNC(=O)c1csc2ccccc12)N1CCCC1 ZINC000217640818 GI On-Demand Unstable HCN1 71 40 COc1ccccc1[C@@H](CNC(=O)c1csc2ccccc12)N1CCCC1 ZINC000217640818 GI On-Demand Unstable HCN4 54 40 CSC[C@@](C)(O)CNC(=O)c1cccc2cccnc12 ZINC000217640820 CE On-Demand Unstable EGLN1 0 44 CCOCCCNS(=O)(=O)c1ccc(NC2CC2)c(C(=O)O)c1 ZINC000217640835 ED In-Stock Unstable CASP3 0 43 FC(F)c1nc(Cl)nc2[nH]cnc12 ZINC000217640837 BD In-Stock Anodyne PRIM_HHV11 40 35 FC(F)c1nc(Cl)nc2[nH]cnc12 ZINC000217640837 BD In-Stock Anodyne AHK4 0 44 FC(F)c1nc(Cl)nc2[nH]cnc12 ZINC000217640837 BD In-Stock Anodyne AHK3 0 43 FC(F)c1nc(Cl)nc2[nH]cnc12 ZINC000217640837 BD In-Stock Anodyne CKX2 0 43 CCC[C@@H](COC)NC(=O)/C=C\C(=O)O ZINC000217640843 BC For-Sale Unstable HCAR2 31 42 Clc1ccccc1CN[C@H]1CCN2CCCC[C@@H]12 ZINC000217640880 CG On-Demand Unstable SLC18A3 52 38 COc1ccccc1[C@H](CNC(=O)c1csc2ccccc12)N1CCCC1 ZINC000217640886 GI On-Demand Unstable DRD2 20 46 COc1ccccc1[C@H](CNC(=O)c1csc2ccccc12)N1CCCC1 ZINC000217640886 GI On-Demand Unstable DRD3 26 41 COc1ccccc1[C@H](CNC(=O)c1csc2ccccc12)N1CCCC1 ZINC000217640886 GI On-Demand Unstable HCN1 71 40 COc1ccccc1[C@H](CNC(=O)c1csc2ccccc12)N1CCCC1 ZINC000217640886 GI On-Demand Unstable HCN4 54 40 CSC[C@](C)(O)CNC(=O)c1cccc2cccnc12 ZINC000217640900 CE On-Demand Unstable EGLN1 0 44 O=C(c1ccccc1F)N1CCS[C@@H]1c1ccc(Cl)c(Cl)c1 ZINC000217640903 FK In-Stock Unstable KCNA5 27 40 CCC[C@H](COC)NC(=O)/C=C\C(=O)O ZINC000217640925 BC For-Sale Unstable HCAR2 31 42 CCOCCCNS(=O)(=O)c1ccc(NC2CCCC2)c(C(=O)O)c1 ZINC000217640941 FE In-Stock Unstable CASP3 0 46 O=C(c1ccccc1F)N1CCS[C@H]1c1ccc(Cl)c(Cl)c1 ZINC000217640956 FK In-Stock Unstable KCNA5 27 40 O=C(N/C=C/c1ccccc1)Nc1cccc(Br)c1 ZINC000217640992 DI For-Sale Anodyne EGFR 40 42 O=C(N/C=C/c1ccccc1)Nc1cccc(Br)c1 ZINC000217640992 DI For-Sale Anodyne P95276_MYCTO 0 41 O=C(N/C=C/c1ccccc1)Nc1cccc(Br)c1 ZINC000217640992 DI For-Sale Anodyne KCNK3 46 34 Cc1cc(C(=O)N2CCS[C@@H]2c2ccc(Cl)c(Cl)c2)c(C)o1 ZINC000217641054 FK In-Stock Unstable KCNA5 30 41 CCOCCCNS(=O)(=O)c1ccc(NC2CCCCC2)c(C(=O)O)c1 ZINC000217641070 GF In-Stock Unstable CASP3 0 45 Cc1cc(C(=O)N2CCS[C@H]2c2ccc(Cl)c(Cl)c2)c(C)o1 ZINC000217641138 FK In-Stock Unstable KCNA5 26 41 COC(=O)c1ccc(Cl)c(NC(=O)C(F)F)c1 ZINC000217641174 CE On-Demand Unstable DYRK1A 18 44 COC(=O)c1ccc(Cl)c(NC(=O)C(F)F)c1 ZINC000217641174 CE On-Demand Unstable DYRK1B 21 44 CCOc1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1OCC ZINC000217641213 FH For-Sale Unstable AKR1C3 28 43 Cn1ccc(NC(=O)c2ccc(/C=C\C(=O)O)cc2)n1 ZINC000217641254 CD For-Sale Unstable GCK 20 47 Cn1ccc(NC(=O)c2ccc(/C=C\C(=O)O)cc2)n1 ZINC000217641254 CD For-Sale Unstable MAP3K5 52 32 Cc1nnsc1C(=O)N1CCS[C@@H]1c1ccc(Cl)c(Cl)c1 ZINC000217641259 FI In-Stock Unstable KCNA5 30 43 CN(C)CCCNS(=O)(=O)c1ccc(N2CCCN(Cc3ccc(F)cc3)CC2)c([N+](=O)[O-])c1 ZINC000217641270 JF On-Demand Unstable HTR7 27 41 CN(C)CCCNS(=O)(=O)c1ccc(N2CCCN(Cc3ccc(F)cc3)CC2)c([N+](=O)[O-])c1 ZINC000217641270 JF On-Demand Unstable BCL2L1 62 36 CN(C)CCCNS(=O)(=O)c1ccc(N2CCCN(Cc3ccc(F)cc3)CC2)c([N+](=O)[O-])c1 ZINC000217641270 JF On-Demand Unstable BCL2 60 36 CCOCCCNS(=O)(=O)c1ccc(NCCO)c(C(=O)O)c1 ZINC000217641307 EC In-Stock Unstable CASP3 15 42 CCOCCCNS(=O)(=O)c1ccc(NCCO)c(C(=O)O)c1 ZINC000217641307 EC In-Stock Unstable BDKRB1 0 41 CC(C)(C)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217641313 CJ For-Sale Unstable EPHX1 0 42 CC(C)(C)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217641313 CJ For-Sale Unstable TRPV1 26 57 CC(C)(C)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217641313 CJ For-Sale Unstable P95276_MYCTO 0 42 Cc1nnsc1C(=O)N1CCS[C@H]1c1ccc(Cl)c(Cl)c1 ZINC000217641340 FI In-Stock Unstable KCNA5 25 43 CCOCCCNS(=O)(=O)c1ccc(NCCCO)c(C(=O)O)c1 ZINC000217641377 FC In-Stock Unstable CASP3 15 43 CCOCCCNS(=O)(=O)c1ccc(NCCCO)c(C(=O)O)c1 ZINC000217641377 FC In-Stock Unstable BDKRB1 0 41 N#Cc1cc2c(nc1N1CCc3[nH]c4ccccc4c3C1)CCCC2 ZINC000217641379 EH On-Demand Unstable DRD5 20 41 CC[C@@H](C)[C@@H](CO)NC(=O)CCn1cnc2ccccc2c1=O ZINC000217641382 DD In-Stock Unstable HTR7 16 41 CC[C@@H](C)[C@@H](CO)NC(=O)CCn1cnc2ccccc2c1=O ZINC000217641382 DD In-Stock Unstable PSMB5 16 51 CC[C@@H](C)[C@@H](CO)NC(=O)CCn1cnc2ccccc2c1=O ZINC000217641382 DD In-Stock Unstable PSMB1 18 51 Brc1ccc(CN[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217641389 DG On-Demand Unstable VACHT_TETCF 0 42 COc1cccc(C(=O)N2[C@H]3CC[C@H]2CC(SC)C3)c1 ZINC000217641434 CG In-Stock Unstable DRD4 44 34 COc1cccc(C(=O)N2[C@H]3CC[C@H]2CC(SC)C3)c1 ZINC000217641434 CG In-Stock Unstable KCNH2 40 37 N#Cc1cccc(C(=O)N2CCS[C@@H]2c2ccc(Cl)c(Cl)c2)c1 ZINC000217641454 FJ In-Stock Unstable HCRTR1 15 54 CCOC(=O)CCNC(=O)/C=C\c1cc(Cl)cc(Cl)c1 ZINC000217641458 DG For-Sale Unstable PYGL 24 47 Brc1ccc(CN[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217641461 DG On-Demand Unstable VACHT_TETCF 0 42 COc1ccc(CN2C(=O)N[C@@H](CC(=O)N3CCCC3)C2=O)cc1OC ZINC000217641501 FD In-Stock Unstable FKBP1A 29 40 CCOCCCNS(=O)(=O)c1ccc(NCCOC)c(C(=O)O)c1 ZINC000217641502 FD In-Stock Unstable CASP3 22 42 CCOCCCNS(=O)(=O)c1ccc(NCCOC)c(C(=O)O)c1 ZINC000217641502 FD In-Stock Unstable BDKRB1 0 44 N#Cc1cccc(C(=O)N2CCS[C@H]2c2ccc(Cl)c(Cl)c2)c1 ZINC000217641531 FJ In-Stock Unstable HCRTR1 15 54 Clc1ccc(CN[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217641576 CG On-Demand Unstable SLC18A3 19 40 CCOC(=O)CCNC(=O)/C=C\c1ccccc1OCC ZINC000217641589 CE On-Demand Unstable HCN1 41 32 CCOC(=O)CCNC(=O)/C=C\c1ccccc1OCC ZINC000217641589 CE On-Demand Unstable HCN4 40 32 CCOCCCNS(=O)(=O)c1ccc(NCCCOC)c(C(=O)O)c1 ZINC000217641597 FD In-Stock Unstable CASP3 23 42 CCOCCCNS(=O)(=O)c1ccc(NCCCOC)c(C(=O)O)c1 ZINC000217641597 FD In-Stock Unstable BDKRB1 0 44 COc1ccccc1CNC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641621 HE In-Stock Unstable TSHR 41 31 COc1ccccc1CNC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641621 HE In-Stock Unstable TACR1 30 46 COc1ccccc1CNC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641621 HE In-Stock Unstable BRS3 25 41 COc1ccccc1CNC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641621 HE In-Stock Unstable CCKBR 43 36 COc1ccccc1CNC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641621 HE In-Stock Unstable GHSR 54 39 CSCC[C@H](NC(=O)[C@@H]1CC[C@@H](CNC(=O)Cn2c(=O)[nH]c3ccccc3c2=O)CC1)C(=O)O ZINC000217641622 JC In-Stock Unstable EDNRB 29 41 COC(=O)c1ccc(C(=O)N2CCS[C@@H]2c2ccc(Cl)c(Cl)c2)cc1 ZINC000217641646 GJ In-Stock Unstable KCNA5 25 41 Clc1ccc(CN[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217641664 CG On-Demand Unstable SLC18A3 19 40 CCOC(=O)CCNC(=O)/C=C\c1ccc(OCC)cc1 ZINC000217641668 CE On-Demand Unstable HDAC7 40 37 CC(C)S(=O)(=O)NCc1cc(/C=C\C(=O)O)ccc1F ZINC000217641691 DD For-Sale Unstable AKR1C3 29 41 CCOCCCNS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217641708 GF In-Stock Unstable CASP3 16 40 COC(=O)c1ccc(C(=O)N2CCS[C@H]2c2ccc(Cl)c(Cl)c2)cc1 ZINC000217641733 GJ In-Stock Unstable SLC6A3 15 41 COC(=O)c1ccc(C(=O)N2CCS[C@H]2c2ccc(Cl)c(Cl)c2)cc1 ZINC000217641733 GJ In-Stock Unstable KCNA5 29 41 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable ACE 45 41 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable HTR1D 33 40 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable HTR1B 27 40 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable SSTR2 91 38 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable GNRHR 0 40 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable OPRM1 16 41 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable OPRD1 0 40 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable MME 30 42 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable EDNRA 45 41 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable TACR1 39 45 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable MC4R 48 37 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable SSTR4 48 36 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable TACR2 70 45 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable CCKAR 120 42 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable CTSL 29 40 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable BRS3 31 49 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable NMBR 38 40 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable MC3R 72 38 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable MC5R 69 38 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable MMP2 29 42 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable MMP8 36 40 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable MMP14 28 42 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable GRPR 64 33 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable ECE1 59 40 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable LNPEP 17 40 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable SSTR3 64 38 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable MMP11 101 40 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable CCKBR 104 41 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable GHSR 82 43 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable MMP9 29 42 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable MC1R 96 38 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable C5AR1 42 36 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable MMP1 23 42 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable SLC15A2 0 41 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable KISS1R 75 35 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable BIRC2 20 41 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable ERAP2 40 40 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable ERAP1 0 40 C[C@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641740 IG In-Stock Unstable NRDE 0 40 CCCCS(=O)(=O)Nc1cc(/C=C\C(=O)O)ccc1OC ZINC000217641771 DE For-Sale Unstable TUBB1 42 36 CCCCS(=O)(=O)Nc1cc(/C=C\C(=O)O)ccc1OC ZINC000217641771 DE For-Sale Unstable AKR1C3 28 42 CCCCS(=O)(=O)Nc1cc(/C=C\C(=O)O)ccc1OC ZINC000217641771 DE For-Sale Unstable ACAT 0 42 Cc1ccccc1N1CCN(C(=O)C(F)F)CC1 ZINC000217641773 CD On-Demand Unstable KCNQ2 48 36 Cc1ccccc1N1CCN(C(=O)C(F)F)CC1 ZINC000217641773 CD On-Demand Unstable ABCB1 40 37 Cc1cncnc1C1CCN(C(=O)c2csc(-c3cccs3)n2)CC1 ZINC000217641790 FH In-Stock Unstable ETHR 47 39 Cc1cncnc1C1CCN(C(=O)c2csc(-c3cccs3)n2)CC1 ZINC000217641790 FH In-Stock Unstable TRPC6 49 37 O=C(N/C=C/c1ccccc1)Nc1ccc2cn[nH]c2c1 ZINC000217641796 CG For-Sale Anodyne PHLPP2 0 51 COc1cccc(OC/C=C\CN)c1 ZINC000217641811 AD For-Sale Unstable MTNR1A 15 42 COc1cccc(OC/C=C\CN)c1 ZINC000217641811 AD For-Sale Unstable MTNR1B 19 42 CCOCCCNS(=O)(=O)c1ccc(N[C@@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217641817 HG In-Stock Unstable CASP3 16 40 CCOCCCNS(=O)(=O)c1ccc(N[C@@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217641817 HG In-Stock Unstable BDKRB1 0 44 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable ACE 45 41 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable HTR1D 33 40 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable HTR1B 27 40 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable SSTR2 91 38 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable GNRHR 0 40 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable OPRM1 16 41 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable OPRD1 0 40 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable MME 30 42 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable EDNRA 45 41 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable TACR1 39 45 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable MC4R 48 37 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable SSTR4 48 36 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable TACR2 70 45 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable CCKAR 120 42 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable CTSL 29 40 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable BRS3 31 49 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable NMBR 38 40 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable MC3R 72 38 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable MC5R 69 38 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable MMP2 29 42 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable MMP8 36 40 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable MMP14 28 42 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable GRPR 64 33 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable ECE1 59 40 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable LNPEP 17 40 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable SSTR3 64 38 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable MMP11 101 40 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable CCKBR 104 41 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable GHSR 82 43 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable MMP9 29 42 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable MC1R 96 38 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable C5AR1 42 36 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable MMP1 23 42 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable SLC15A2 0 41 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable KISS1R 75 35 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable BIRC2 20 41 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable ERAP2 40 40 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable ERAP1 0 40 C[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217641822 IG In-Stock Unstable NRDE 0 40 O=C(c1ccoc1)N1CCS[C@@H]1c1ccc(Cl)c(Cl)c1 ZINC000217641848 EI In-Stock Unstable KCNA5 26 40 COc1ccc(/C=C\C(=O)O)cc1NS(=O)(=O)C(C)C ZINC000217641872 CD For-Sale Unstable TUBB1 52 38 COc1ccc(/C=C\C(=O)O)cc1NS(=O)(=O)C(C)C ZINC000217641872 CD For-Sale Unstable ABCG2 16 40 CCOCCCNS(=O)(=O)c1ccc(N[C@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217641905 HG In-Stock Unstable CASP3 16 40 CCOCCCNS(=O)(=O)c1ccc(N[C@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217641905 HG In-Stock Unstable BDKRB1 0 44 CC(C)(C)c1ccccc1NC(=O)N/C=C/c1ccccc1 ZINC000217641908 CJ For-Sale Unstable P2RY1 15 40 COc1ccccc1CCNC(=O)C(F)F ZINC000217641925 BD On-Demand Unstable GRIN2B 0 40 COc1ccccc1CCNC(=O)C(F)F ZINC000217641925 BD On-Demand Unstable NQO2 47 44 COc1ccccc1CCNC(=O)C(F)F ZINC000217641925 BD On-Demand Unstable MTNR1A 73 44 COc1ccccc1CCNC(=O)C(F)F ZINC000217641925 BD On-Demand Unstable MTNR1B 58 44 COc1ccccc1CCNC(=O)C(F)F ZINC000217641925 BD On-Demand Unstable MBTPS1 41 33 Cn1nc(C(C)(C)C)cc1C(=O)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217641933 EF In-Stock Unstable CTSV 51 35 Cn1nc(C(C)(C)C)cc1C(=O)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217641933 EF In-Stock Unstable CACNA1I 42 32 O=C(c1ccoc1)N1CCS[C@H]1c1ccc(Cl)c(Cl)c1 ZINC000217641940 EI In-Stock Unstable KCNA5 26 40 O=C(c1ccnnc1)N1CCC[C@@]2(CCCN(Cc3ccccc3)C2)C1 ZINC000217641957 FF In-Stock Unstable CCR8 24 41 O=C(c1ccnnc1)N1CCC[C@@]2(CCCN(Cc3ccccc3)C2)C1 ZINC000217641957 FF In-Stock Unstable NPFFR1 44 38 Fc1ccc(CN[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217641969 BF On-Demand Unstable VACHT_TETCF 0 42 Fc1ccc(CN[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217641969 BF On-Demand Unstable SSTR3 20 40 Cc1cc(Cl)c(Br)cc1C(=O)O ZINC000217641995 BG For-Sale Unstable PRS 39 41 Cc1cc(Cl)c(Br)cc1C(=O)O ZINC000217641995 BG For-Sale Unstable AKR1C2 58 38 Cc1cc(Cl)c(Br)cc1C(=O)O ZINC000217641995 BG For-Sale Unstable AKR1C1 63 38 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217642019 ED For-Sale Unstable CA2 142 67 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217642019 ED For-Sale Unstable CA6 22 42 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217642019 ED For-Sale Unstable CA1 118 67 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217642019 ED For-Sale Unstable CA7 71 61 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217642019 ED For-Sale Unstable CA13 33 42 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217642019 ED For-Sale Unstable CA5B 65 61 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217642019 ED For-Sale Unstable CA4 97 65 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217642019 ED For-Sale Unstable CA5A 67 61 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217642019 ED For-Sale Unstable CA14 51 60 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217642019 ED For-Sale Unstable MMP2 20 40 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217642019 ED For-Sale Unstable MMP3 15 46 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217642019 ED For-Sale Unstable CA12 88 67 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217642019 ED For-Sale Unstable CA9 99 67 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217642019 ED For-Sale Unstable CAH_METTE 27 41 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217642019 ED For-Sale Unstable CYNT 33 48 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217642019 ED For-Sale Unstable NCE103 47 62 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217642019 ED For-Sale Unstable LIG1 0 48 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217642019 ED For-Sale Unstable CA15 17 42 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217642019 ED For-Sale Unstable MTCA1 48 45 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217642019 ED For-Sale Unstable P96878_MYCTU 61 46 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217642019 ED For-Sale Unstable CA 0 47 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217642019 ED For-Sale Unstable A6YCJ1_9METZ 27 54 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217642019 ED For-Sale Unstable Q5TU56_ANOGA 0 42 CCOCCCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217642021 HF In-Stock Unstable CASP3 15 41 CCOCCCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217642021 HF In-Stock Unstable BDKRB1 0 43 O=C(c1ccnnc1)N1CCC[C@]2(CCCN(Cc3ccccc3)C2)C1 ZINC000217642039 FF In-Stock Unstable CCR8 24 41 O=C(c1ccnnc1)N1CCC[C@]2(CCCN(Cc3ccccc3)C2)C1 ZINC000217642039 FF In-Stock Unstable NPFFR1 44 38 Fc1ccc(CN[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217642052 BF On-Demand Unstable VACHT_TETCF 0 42 Fc1ccc(CN[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217642052 BF On-Demand Unstable SSTR3 20 40 COCC(=O)NCCc1ccccc1OC ZINC000217642053 BD On-Demand Unstable NQO2 50 41 COCC(=O)NCCc1ccccc1OC ZINC000217642053 BD On-Demand Unstable MTNR1A 87 45 COCC(=O)NCCc1ccccc1OC ZINC000217642053 BD On-Demand Unstable MTNR1B 75 44 COCC(=O)NCCc1ccccc1OC ZINC000217642053 BD On-Demand Unstable MBTPS1 43 36 COCC(=O)NCCc1ccccc1OC ZINC000217642053 BD On-Demand Unstable CAN2 0 40 Cn1cc(-c2nc3ccccc3s2)c2ccccc21 ZINC000217642055 CI In-Stock Unstable PRKCG 56 45 Cn1cc(-c2nc3ccccc3s2)c2ccccc21 ZINC000217642055 CI In-Stock Unstable IMPDH2 21 43 Cn1cc(-c2nc3ccccc3s2)c2ccccc21 ZINC000217642055 CI In-Stock Unstable LUCI_PHOPY 15 43 Cn1cc(-c2nc3ccccc3s2)c2ccccc21 ZINC000217642055 CI In-Stock Unstable LUCI_PHOPE 16 43 CN(C)CCCNS(=O)(=O)c1ccc(N[C@@H](c2ccccc2)C2CC2)c([N+](=O)[O-])c1 ZINC000217642058 IG On-Demand Unstable BDKRB1 45 58 CN(C)CCCNS(=O)(=O)c1ccc(N[C@@H](c2ccccc2)C2CC2)c([N+](=O)[O-])c1 ZINC000217642058 IG On-Demand Unstable BCL2L1 128 42 CN(C)CCCNS(=O)(=O)c1ccc(N[C@@H](c2ccccc2)C2CC2)c([N+](=O)[O-])c1 ZINC000217642058 IG On-Demand Unstable BCL2 107 37 CN(C)CCCNS(=O)(=O)c1ccc(N[C@@H](c2ccccc2)C2CC2)c([N+](=O)[O-])c1 ZINC000217642058 IG On-Demand Unstable BCL2L2 56 40 CCOCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217642118 IF In-Stock Unstable TBXA2R 28 40 CCOCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217642118 IF In-Stock Unstable TBXAS1 19 41 CCOCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217642118 IF In-Stock Unstable BMP1 45 34 CCOCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217642118 IF In-Stock Unstable IAP 0 46 CCOCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217642118 IF In-Stock Unstable CA9 19 40 CCOCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217642118 IF In-Stock Unstable AKR1C3 24 43 CCOCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217642118 IF In-Stock Unstable AKR1C2 40 34 O=C(N/C=C/c1ccccc1)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217642123 FK For-Sale Anodyne JUN 21 41 O=C(N/C=C/c1ccccc1)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217642123 FK For-Sale Anodyne PTPA 0 49 O=C(N/C=C/c1ccccc1)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217642123 FK For-Sale Anodyne TRPM4 0 40 CN(C)CCCNS(=O)(=O)c1ccc(N[C@H](c2ccccc2)C2CC2)c([N+](=O)[O-])c1 ZINC000217642138 IG On-Demand Unstable BDKRB1 45 58 CN(C)CCCNS(=O)(=O)c1ccc(N[C@H](c2ccccc2)C2CC2)c([N+](=O)[O-])c1 ZINC000217642138 IG On-Demand Unstable BCL2L1 128 42 CN(C)CCCNS(=O)(=O)c1ccc(N[C@H](c2ccccc2)C2CC2)c([N+](=O)[O-])c1 ZINC000217642138 IG On-Demand Unstable BCL2 107 37 CN(C)CCCNS(=O)(=O)c1ccc(N[C@H](c2ccccc2)C2CC2)c([N+](=O)[O-])c1 ZINC000217642138 IG On-Demand Unstable BCL2L2 56 40 NC(=O)NCCC[C@H](NC(=O)[C@@H]1CC[C@@H](CNC(=O)Cn2c(=O)[nH]c3ccccc3c2=O)CC1)C(=O)O ZINC000217642147 KB In-Stock Unstable F2 22 40 NC(=O)NCCC[C@H](NC(=O)[C@@H]1CC[C@@H](CNC(=O)Cn2c(=O)[nH]c3ccccc3c2=O)CC1)C(=O)O ZINC000217642147 KB In-Stock Unstable SSTR4 43 31 NC(=O)NCCC[C@H](NC(=O)[C@@H]1CC[C@@H](CNC(=O)Cn2c(=O)[nH]c3ccccc3c2=O)CC1)C(=O)O ZINC000217642147 KB In-Stock Unstable C3AR1 80 35 NC(=O)NCCC[C@H](NC(=O)[C@@H]1CC[C@@H](CNC(=O)Cn2c(=O)[nH]c3ccccc3c2=O)CC1)C(=O)O ZINC000217642147 KB In-Stock Unstable MC3R 19 40 NC(=O)NCCC[C@H](NC(=O)[C@@H]1CC[C@@H](CNC(=O)Cn2c(=O)[nH]c3ccccc3c2=O)CC1)C(=O)O ZINC000217642147 KB In-Stock Unstable MC1R 19 40 Brc1cccc(CN[C@@H]2CCN3CCCC[C@@H]23)c1 ZINC000217642172 DG On-Demand Unstable VACHT_TETCF 0 43 Cc1nc2cc(CNC(=O)CN(C)Cc3cccnc3)ccc2n1C ZINC000217642190 EE In-Stock Unstable NAMPT 45 42 O=C(Nc1cccc(CO)c1)C(F)F ZINC000217642194 BD On-Demand Unstable NAMPT 0 57 O=C(Nc1cccc(CO)c1)C(F)F ZINC000217642194 BD On-Demand Unstable KCNK3 72 37 O=C(Nc1cccc(CO)c1)C(F)F ZINC000217642194 BD On-Demand Unstable KCNK9 70 37 COc1cc(NC(=O)CCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@H]23)cc(OC)c1OC ZINC000217642226 JH In-Stock Unstable MAPK7 41 31 COc1cc(NC(=O)CCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@H]23)cc(OC)c1OC ZINC000217642226 JH In-Stock Unstable ENPP1 59 32 Brc1cccc(CN[C@H]2CCN3CCCC[C@@H]23)c1 ZINC000217642250 DG On-Demand Unstable VACHT_TETCF 0 43 CCOCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217642254 JF In-Stock Unstable BDKRB1 0 40 CCOCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217642254 JF In-Stock Unstable IAP 0 47 CCOCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217642254 JF In-Stock Unstable SCMU_MYCTU 0 42 CN(C)CCNS(=O)(=O)c1ccc(N[C@@H](c2ccccc2)C2CC2)c([N+](=O)[O-])c1 ZINC000217642265 HF On-Demand Unstable BDKRB1 0 56 CN(C)CCNS(=O)(=O)c1ccc(N[C@@H](c2ccccc2)C2CC2)c([N+](=O)[O-])c1 ZINC000217642265 HF On-Demand Unstable BCL2L1 129 41 CN(C)CCNS(=O)(=O)c1ccc(N[C@@H](c2ccccc2)C2CC2)c([N+](=O)[O-])c1 ZINC000217642265 HF On-Demand Unstable BCL2 110 38 CN(C)CCNS(=O)(=O)c1ccc(N[C@@H](c2ccccc2)C2CC2)c([N+](=O)[O-])c1 ZINC000217642265 HF On-Demand Unstable BCL2L2 57 41 COc1cc(NC(=O)CCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@@H]23)cc(OC)c1OC ZINC000217642311 JH In-Stock Unstable MAPK7 41 31 COc1cc(NC(=O)CCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@@H]23)cc(OC)c1OC ZINC000217642311 JH In-Stock Unstable ENPP1 59 32 CC[C@@H]1CC[C@@H](N)[C@@H](Cc2cccc(C(F)(F)F)c2)C1 ZINC000217642333 CI For-Sale Unstable PDS 15 43 CN(C)CCNS(=O)(=O)c1ccc(N[C@H](c2ccccc2)C2CC2)c([N+](=O)[O-])c1 ZINC000217642351 HF On-Demand Unstable BDKRB1 0 56 CN(C)CCNS(=O)(=O)c1ccc(N[C@H](c2ccccc2)C2CC2)c([N+](=O)[O-])c1 ZINC000217642351 HF On-Demand Unstable BCL2L1 129 41 CN(C)CCNS(=O)(=O)c1ccc(N[C@H](c2ccccc2)C2CC2)c([N+](=O)[O-])c1 ZINC000217642351 HF On-Demand Unstable BCL2 110 38 CN(C)CCNS(=O)(=O)c1ccc(N[C@H](c2ccccc2)C2CC2)c([N+](=O)[O-])c1 ZINC000217642351 HF On-Demand Unstable BCL2L2 57 41 COc1ccc(-c2coc3ccc(OCC(=O)N[C@@H]4CCS(=O)(=O)C4)cc23)cc1 ZINC000217642416 HF In-Stock Unstable ALDH2 81 36 CC[C@H]1CC[C@@H](N)[C@@H](Cc2cccc(C(F)(F)F)c2)C1 ZINC000217642422 CI For-Sale Unstable PDS 15 43 O=C(CN1CCOc2ccccc2C1)NCc1cnc2cnccn12 ZINC000217642447 ED In-Stock Unstable NOS2 61 32 COc1ccc(NC(=O)c2ccc(=O)[nH]n2)cc1O ZINC000217642478 CC For-Sale Unstable GRM4 29 45 COc1ccc(NC(=O)c2ccc(=O)[nH]n2)cc1O ZINC000217642478 CC For-Sale Unstable ENPP1 73 35 NC/C=C\COc1ccc2ccccc2c1Br ZINC000217642482 CG For-Sale Unstable NCEH1 23 40 COc1ccc(-c2coc3ccc(OCC(=O)N[C@H]4CCS(=O)(=O)C4)cc23)cc1 ZINC000217642485 HF In-Stock Unstable ALDH2 81 36 CCOC(=O)CCNC(=O)/C=C\c1ccc(OC)c(F)c1 ZINC000217642487 CD For-Sale Unstable HPSE 16 42 CCOC(=O)CCNC(=O)/C=C\c1ccc(OC)c(F)c1 ZINC000217642487 CD For-Sale Unstable TUBB1 58 49 CCOC(=O)CCNC(=O)/C=C\c1ccc(OC)c(F)c1 ZINC000217642487 CD For-Sale Unstable NFE2L2 0 43 NC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217642494 CF For-Sale Unstable MTCA1 23 42 NC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217642494 CF For-Sale Unstable P96878_MYCTU 26 42 CC[C@@H]1CC[C@H](N)[C@@H](Cc2cccc(C(F)(F)F)c2)C1 ZINC000217642499 CI For-Sale Unstable PDS 15 43 CS(=O)(=O)c1ccccc1N1CCC(CCc2ccccc2)CC1 ZINC000217642511 EH On-Demand Unstable SLC18A2 46 40 CS(=O)(=O)c1ccccc1N1CCC(CCc2ccccc2)CC1 ZINC000217642511 EH On-Demand Unstable SIGMAR1 15 42 COc1ccc(/C=C\C(=O)O)cc1N1C(=O)COCC1=O ZINC000217642557 CC For-Sale Unstable TUBB1 42 38 COc1ccc(/C=C\C(=O)O)cc1N1C(=O)COCC1=O ZINC000217642557 CC For-Sale Unstable ABCG2 15 40 COc1ccc(CN[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217642572 CE On-Demand Unstable SIGMAR1 18 50 CN[C@@H]1CCN([C@@H](C)c2cc(Br)ccc2F)C1 ZINC000217642584 DF For-Sale Unstable HRH4 44 37 CC[C@H]1CC[C@H](N)[C@@H](Cc2cccc(C(F)(F)F)c2)C1 ZINC000217642585 CI For-Sale Unstable PDS 15 43 NC/C=C\COc1ccc([N+](=O)[O-])cc1 ZINC000217642591 BD For-Sale Unstable ACR 22 47 NC/C=C\COc1ccc([N+](=O)[O-])cc1 ZINC000217642591 BD For-Sale Unstable SNCA 26 43 COc1ccc(NC(=O)c2cc(Br)ccc2I)cc1O ZINC000217642596 II For-Sale Unstable PYK 61 38 COc1ccc(NC(=O)c2cc(Br)ccc2I)cc1O ZINC000217642596 II For-Sale Unstable ENPP1 57 36 COc1ccc(NC(=O)c2cc(Br)ccc2I)cc1O ZINC000217642596 II For-Sale Unstable Q25615_ONCVO 72 46 COc1ccc(NC(=O)c2cc(Br)ccc2I)cc1O ZINC000217642596 II For-Sale Unstable KCNK3 52 43 COc1ccc(NC(=O)c2cc(Br)ccc2I)cc1O ZINC000217642596 II For-Sale Unstable KCNK9 44 43 O=C(N/C=C/c1ccccc1)Nc1ccc(F)c(Cl)c1 ZINC000217642603 CI For-Sale Anodyne MMP1 0 48 O=C(N/C=C/c1ccccc1)Nc1ccc(F)c(Cl)c1 ZINC000217642603 CI For-Sale Anodyne P95276_MYCTO 0 45 CCOC(=O)CCNC(=O)/C=C\c1ccc(CC)cc1 ZINC000217642640 CE For-Sale Unstable HDAC8 17 40 CCOC(=O)CCNC(=O)/C=C\c1ccc(CC)cc1 ZINC000217642640 CE For-Sale Unstable HDAC7 41 37 CS(=O)(=O)CCNC(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217642641 CC For-Sale Unstable CA2 17 43 CCOCCCNS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217642650 FD In-Stock Unstable CASP3 28 40 CCOCCCNS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217642650 FD In-Stock Unstable LIPG 30 41 CCOCCCNS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217642650 FD In-Stock Unstable SFRP1 61 32 COc1ccc(CN[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217642651 CE On-Demand Unstable SIGMAR1 18 50 O=C1C[C@@H](c2cc(F)c(F)c(F)c2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217642703 JJ In-Stock Unstable CYP1B1 19 41 O=C1C[C@@H](c2cc(F)c(F)c(F)c2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217642703 JJ In-Stock Unstable CYP1A1 18 41 NC/C=C\COc1cccc([N+](=O)[O-])c1 ZINC000217642705 BD For-Sale Unstable CACNA1C 46 37 NC/C=C\COc1cccc([N+](=O)[O-])c1 ZINC000217642705 BD For-Sale Unstable CACNA1D 40 33 NC/C=C\COc1cccc([N+](=O)[O-])c1 ZINC000217642705 BD For-Sale Unstable ACR 25 50 NC/C=C\COc1cccc([N+](=O)[O-])c1 ZINC000217642705 BD For-Sale Unstable ATSA 0 50 O=C(O)/C=C\c1ccc(C(=O)NCc2ccccc2Cl)s1 ZINC000217642720 DG For-Sale Unstable P2RX7 21 40 CCN(CC)c1ccc(NC(=O)N/C=C/c2ccccc2)cc1 ZINC000217642724 DI For-Sale Unstable GHSR 0 45 COc1ccc(CN[C@@H]2CCN3CCCC[C@@H]23)c(OC)c1 ZINC000217642762 CE On-Demand Unstable TACR1 23 43 CCOCCCNS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217642764 FE In-Stock Unstable LIPG 27 41 CCOCCCNS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217642764 FE In-Stock Unstable SFRP1 50 31 O=C1C[C@H](c2cc(F)c(F)c(F)c2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217642788 JJ In-Stock Unstable CYP1B1 19 41 O=C1C[C@H](c2cc(F)c(F)c(F)c2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217642788 JJ In-Stock Unstable CYP1A1 18 41 CCCOc1ccc([C@@H](C)N[C@@H]2CCC[C@@H](O)C2)cc1 ZINC000217642806 CG For-Sale Unstable ACACA 44 48 CCCOc1ccc([C@@H](C)N[C@@H]2CCC[C@@H](O)C2)cc1 ZINC000217642806 CG For-Sale Unstable ACACB 24 48 COc1ccc(CN[C@H]2CCN3CCCC[C@@H]23)c(OC)c1 ZINC000217642840 CE On-Demand Unstable TACR1 23 43 O=C(N/C=C/c1ccccc1)NCc1ccc(F)cc1 ZINC000217642856 CG For-Sale Unstable AMP1_PLAFQ 34 58 O=C(N/C=C/c1ccccc1)NCc1ccc(F)cc1 ZINC000217642856 CG For-Sale Unstable Q76353_9HIV1 0 40 Cc1ccccc1NC(=O)N1CCS[C@@H]1c1ccc(Cl)c(Cl)c1 ZINC000217642869 FK In-Stock Unstable KCNA5 27 45 Cc1ccccc1NC(=O)N1CCS[C@@H]1c1ccc(Cl)c(Cl)c1 ZINC000217642869 FK In-Stock Unstable P2RX7 26 48 CCOCCCNS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1 ZINC000217642872 FC In-Stock Unstable SLC6A9 19 45 CCCOc1ccc([C@H](C)N[C@@H]2CCC[C@@H](O)C2)cc1 ZINC000217642900 CG On-Demand Unstable ACACA 44 48 CCCOc1ccc([C@H](C)N[C@@H]2CCC[C@@H](O)C2)cc1 ZINC000217642900 CG On-Demand Unstable ACACB 24 48 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)c(OC)c1 ZINC000217642911 JI In-Stock Unstable AKR1B1 0 44 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)c(OC)c1 ZINC000217642911 JI In-Stock Unstable CYP1B1 52 45 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)c(OC)c1 ZINC000217642911 JI In-Stock Unstable CYP1A1 41 45 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)c(OC)c1 ZINC000217642911 JI In-Stock Unstable CYP1A2 32 45 CSC[C@@](C)(O)CNC(=O)c1ccc2c(c1)OCCO2 ZINC000217642945 CD On-Demand Unstable PLK1 18 43 Cc1ccccc1NC(=O)N1CCS[C@H]1c1ccc(Cl)c(Cl)c1 ZINC000217642946 FK In-Stock Unstable KCNA5 30 45 Cc1ccccc1NC(=O)N1CCS[C@H]1c1ccc(Cl)c(Cl)c1 ZINC000217642946 FK In-Stock Unstable P2RX7 26 48 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2)CC1 ZINC000217642962 EG For-Sale Unstable HTR1A 97 54 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2)CC1 ZINC000217642962 EG For-Sale Unstable DRD2 73 54 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2)CC1 ZINC000217642962 EG For-Sale Unstable DRD1 28 43 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2)CC1 ZINC000217642962 EG For-Sale Unstable DRD4 39 49 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2)CC1 ZINC000217642962 EG For-Sale Unstable ADRA1D 77 43 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2)CC1 ZINC000217642962 EG For-Sale Unstable HTR1D 22 47 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2)CC1 ZINC000217642962 EG For-Sale Unstable HTR1B 19 54 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2)CC1 ZINC000217642962 EG For-Sale Unstable HTR2A 36 47 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2)CC1 ZINC000217642962 EG For-Sale Unstable ADRA1A 69 43 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2)CC1 ZINC000217642962 EG For-Sale Unstable ADRA1B 63 43 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2)CC1 ZINC000217642962 EG For-Sale Unstable DRD3 75 54 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2)CC1 ZINC000217642962 EG For-Sale Unstable PDGFRB 26 41 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2)CC1 ZINC000217642962 EG For-Sale Unstable HTR7 63 48 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2)CC1 ZINC000217642962 EG For-Sale Unstable TACR3 24 48 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2)CC1 ZINC000217642962 EG For-Sale Unstable RBP4 15 46 CCCOc1ccc([C@@H](C)N[C@H]2CCC[C@@H](O)C2)cc1 ZINC000217642976 CG For-Sale Unstable ACACA 44 48 CCCOc1ccc([C@@H](C)N[C@H]2CCC[C@@H](O)C2)cc1 ZINC000217642976 CG For-Sale Unstable ACACB 24 48 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)c(OC)c1 ZINC000217642980 JI In-Stock Unstable AKR1B1 0 44 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)c(OC)c1 ZINC000217642980 JI In-Stock Unstable CYP1B1 52 45 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)c(OC)c1 ZINC000217642980 JI In-Stock Unstable CYP1A1 41 45 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)c(OC)c1 ZINC000217642980 JI In-Stock Unstable CYP1A2 32 45 CCOCCCNc1ccc(S(=O)(=O)NCCCOCC)cc1C(=O)O ZINC000217642995 GD In-Stock Unstable CASP3 16 43 CCOCCCNc1ccc(S(=O)(=O)NCCCOCC)cc1C(=O)O ZINC000217642995 GD In-Stock Unstable BDKRB1 0 43 CN1CCC(N(C)C(=O)c2ccc(/C=C\C(=O)O)s2)CC1 ZINC000217643023 DE For-Sale Unstable MCHR1 0 47 CSC[C@](C)(O)CNC(=O)c1ccc2c(c1)OCCO2 ZINC000217643032 CD On-Demand Unstable PLK1 18 43 C[C@H](NC(=O)[C@@H]1CC[C@@H](CNC(=O)Cn2c(=O)[nH]c3ccccc3c2=O)CC1)C(=O)O ZINC000217643033 IC In-Stock Unstable AVPR1B 33 41 O=C(Nc1ccccc1F)N1CCS[C@@H]1c1ccc(Cl)c(Cl)c1 ZINC000217643056 FK In-Stock Unstable TRPM8 24 43 CCCOc1ccc([C@H](C)N[C@H]2CCC[C@@H](O)C2)cc1 ZINC000217643060 CG On-Demand Unstable ACACA 44 48 CCCOc1ccc([C@H](C)N[C@H]2CCC[C@@H](O)C2)cc1 ZINC000217643060 CG On-Demand Unstable ACACB 24 48 CCOCCCNS(=O)(=O)c1ccc(NCCCOC(C)C)c(C(=O)O)c1 ZINC000217643097 HE In-Stock Unstable CASP3 15 42 CCOCCCNS(=O)(=O)c1ccc(NCCCOC(C)C)c(C(=O)O)c1 ZINC000217643097 HE In-Stock Unstable BDKRB1 16 41 O=C(O)/C=C\c1ccc(C(=O)NCCc2ccccc2)s1 ZINC000217643115 DF For-Sale Unstable HDAC1 20 57 O=C(Nc1ccccc1F)N1CCS[C@H]1c1ccc(Cl)c(Cl)c1 ZINC000217643136 FK In-Stock Unstable TRPM8 24 43 CC[S@@](=O)CCn1c(=O)cc(Cl)[nH]c1=O ZINC000217643156 CB For-Sale Unstable POLC 78 35 Clc1ccc(CN[C@@H]2CCN3CCCC[C@@H]23)cc1Cl ZINC000217643158 CH On-Demand Unstable OPRK1 16 47 Clc1ccc(CN[C@@H]2CCN3CCCC[C@@H]23)cc1Cl ZINC000217643158 CH On-Demand Unstable SIGMAR1 15 70 Clc1ccc(CN[C@@H]2CCN3CCCC[C@@H]23)cc1Cl ZINC000217643158 CH On-Demand Unstable SSTR3 20 50 Clc1ccc(CN[C@@H]2CCN3CCCC[C@@H]23)cc1Cl ZINC000217643158 CH On-Demand Unstable KCNB1 0 44 CSC[C@@](C)(O)CNC(=O)COc1cccc(F)c1 ZINC000217643160 CD On-Demand Unstable PDS 57 43 CC(C)CN(CC(C)C)C(=O)N/C=C/c1ccccc1 ZINC000217643180 CH For-Sale Unstable MME 17 42 COCCn1c(C)cc(C)c(C(=O)N2CCc3cc(OC)c(OC)cc3C2)c1=O ZINC000217643214 HE In-Stock Unstable ABCB1B 62 35 COCCn1c(C)cc(C)c(C(=O)N2CCc3cc(OC)c(OC)cc3C2)c1=O ZINC000217643214 HE In-Stock Unstable ABCB1 18 45 CCCCCNc1ccc(S(=O)(=O)NCCCOCC)cc1C(=O)O ZINC000217643216 FF In-Stock Unstable CASP3 15 45 CCCCCNc1ccc(S(=O)(=O)NCCCOCC)cc1C(=O)O ZINC000217643216 FF In-Stock Unstable BDKRB1 16 41 Cc1cc(N2CCC(N3CCCC3)CC2)ccc1N ZINC000217643244 CF For-Sale Unstable HRH3 22 42 Cc1cc(N2CCC(N3CCCC3)CC2)ccc1N ZINC000217643244 CF For-Sale Unstable L3MBTL3 127 62 CC[S@](=O)CCn1c(=O)cc(Cl)[nH]c1=O ZINC000217643246 CB For-Sale Unstable POLC 78 35 Clc1ccc(CN[C@H]2CCN3CCCC[C@@H]23)cc1Cl ZINC000217643248 CH On-Demand Unstable OPRK1 16 47 Clc1ccc(CN[C@H]2CCN3CCCC[C@@H]23)cc1Cl ZINC000217643248 CH On-Demand Unstable SIGMAR1 15 70 Clc1ccc(CN[C@H]2CCN3CCCC[C@@H]23)cc1Cl ZINC000217643248 CH On-Demand Unstable SSTR3 20 50 Clc1ccc(CN[C@H]2CCN3CCCC[C@@H]23)cc1Cl ZINC000217643248 CH On-Demand Unstable KCNB1 0 44 CSC[C@](C)(O)CNC(=O)COc1cccc(F)c1 ZINC000217643251 CD On-Demand Unstable PDS 57 43 COc1cccc(NC(=O)N2CCS[C@@H]2c2ccc(Cl)c(Cl)c2)c1OC ZINC000217643257 HK In-Stock Unstable KCNA5 24 41 FC(F)(F)Oc1ccc(CNc2ncccc2Cl)cc1 ZINC000217643306 DI On-Demand Unstable GRIN2B 27 40 FC(F)(F)Oc1ccc(CNc2ncccc2Cl)cc1 ZINC000217643306 DI On-Demand Unstable SCN10A 18 41 FC(F)(F)Oc1ccc(CNc2ncccc2Cl)cc1 ZINC000217643306 DI On-Demand Unstable GPR39 0 51 CCOC(=O)CCNC(=O)/C=C\c1cccc(F)c1 ZINC000217643307 CD On-Demand Unstable HDAC8 44 33 Nc1nc2c(c(C(=O)N3CCN(c4ccc(Cl)cn4)CC3)n1)CCCC2 ZINC000217643318 FD In-Stock Unstable NPBWR1 46 33 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1N[C@@H]1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217643324 CK For-Sale Unstable TRPM8 0 41 C[C@@H](CNC(=O)C(F)F)c1ccccc1 ZINC000217643337 BE On-Demand Unstable MME 35 41 C[C@@H](CNC(=O)C(F)F)c1ccccc1 ZINC000217643337 BE On-Demand Unstable GRIA4 15 40 C[C@@H](CNC(=O)C(F)F)c1ccccc1 ZINC000217643337 BE On-Demand Unstable AOC3 18 50 CCOCCCNS(=O)(=O)c1ccc(NCCC(C)C)c(C(=O)O)c1 ZINC000217643339 FF In-Stock Unstable CASP3 15 45 CCOCCCNS(=O)(=O)c1ccc(NCCC(C)C)c(C(=O)O)c1 ZINC000217643339 FF In-Stock Unstable BDKRB1 16 41 COc1cccc(NC(=O)N2CCS[C@H]2c2ccc(Cl)c(Cl)c2)c1OC ZINC000217643343 HK In-Stock Unstable KCNA5 24 41 O=C(O)/C=C\c1ccc(C(=O)N2CCc3ccccc32)s1 ZINC000217643377 CG For-Sale Unstable AVPR2 33 40 O=C(N/C=C/c1ccccc1)NC1CCCCCC1 ZINC000217643386 CH For-Sale Unstable FAAH 17 57 O=C(N/C=C/c1ccccc1)NC1CCCCCC1 ZINC000217643386 CH For-Sale Unstable EPHX2 37 56 CC[C@@H]1CC[C@@H](N)[C@@H](Cc2cccc(Cl)c2)C1 ZINC000217643391 CI For-Sale Unstable CACNA1D 31 44 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1N[C@@H]1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217643401 CK For-Sale Unstable TRPM8 0 41 CCOC(=O)CCNC(=O)/C=C\c1ccccc1[N+](=O)[O-] ZINC000217643425 CD On-Demand Unstable TLR4 23 47 C[C@H](CNC(=O)C(F)F)c1ccccc1 ZINC000217643427 BE On-Demand Unstable MME 35 41 C[C@H](CNC(=O)C(F)F)c1ccccc1 ZINC000217643427 BE On-Demand Unstable GRIA4 15 40 C[C@H](CNC(=O)C(F)F)c1ccccc1 ZINC000217643427 BE On-Demand Unstable AOC3 18 50 O=C(c1cccs1)N1CCS[C@@H]1c1ccc(OC(F)(F)F)cc1 ZINC000217643456 FJ In-Stock Unstable EPHX2 41 35 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NCCCOCC)cc1C(=O)O ZINC000217643459 FF In-Stock Unstable CASP3 0 45 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1N[C@@H]1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217643483 CK For-Sale Unstable TRPM8 0 41 CC[C@H]1CC[C@@H](N)[C@@H](Cc2cccc(Cl)c2)C1 ZINC000217643485 CI For-Sale Unstable CACNA1D 31 44 CCC[C@H](C)Nc1ccc(S(=O)(=O)NCCCOCC)cc1C(=O)O ZINC000217643545 FF In-Stock Unstable CASP3 15 45 O=C(c1cccs1)N1CCS[C@H]1c1ccc(OC(F)(F)F)cc1 ZINC000217643547 FJ In-Stock Unstable EPHX2 41 35 COc1ccc2[nH]c(=O)c([C@H](CC(N)=O)c3oc(C)cc(=O)c3O)cc2c1 ZINC000217643554 FD In-Stock Unstable TUBB2B 40 38 Cc1ccc(C)c(NC(=O)c2ccc(/C=C\C(=O)O)s2)c1 ZINC000217643555 DH For-Sale Unstable MAPK11 35 43 CC(C)[C@H]1CC[C@H](C)C[C@@H]1N[C@@H]1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217643560 CK For-Sale Unstable TRPM8 0 41 CC[C@@H]1CC[C@H](N)[C@@H](Cc2cccc(Cl)c2)C1 ZINC000217643568 CI For-Sale Unstable CACNA1D 31 44 CCOC(=O)CCNC(=O)/C=C\c1ccc([N+](=O)[O-])cc1 ZINC000217643624 CD On-Demand Unstable CACNA1D 42 37 O=C(N/C=C/c1ccccc1)Nc1cc(Cl)cc(Cl)c1 ZINC000217643627 DJ For-Sale Anodyne PPIA 19 45 COc1ccc2[nH]c(=O)c([C@@H](CC(N)=O)c3oc(C)cc(=O)c3O)cc2c1 ZINC000217643653 FD In-Stock Unstable TUBB2B 40 38 CC[C@H]1CC[C@H](N)[C@@H](Cc2cccc(Cl)c2)C1 ZINC000217643662 CI For-Sale Unstable CACNA1D 31 44 CCOCCCNS(=O)(=O)c1ccc(N[C@@H](C)COC)c(C(=O)O)c1 ZINC000217643680 FD In-Stock Unstable CASP3 0 40 NC/C=C\CN1CCN(c2ccccc2Cl)CC1 ZINC000217643699 CD For-Sale Unstable HTR1A 27 48 NC/C=C\CN1CCN(c2ccccc2Cl)CC1 ZINC000217643699 CD For-Sale Unstable DRD2 36 52 NC/C=C\CN1CCN(c2ccccc2Cl)CC1 ZINC000217643699 CD For-Sale Unstable DRD1 16 43 NC/C=C\CN1CCN(c2ccccc2Cl)CC1 ZINC000217643699 CD For-Sale Unstable DRD4 27 48 NC/C=C\CN1CCN(c2ccccc2Cl)CC1 ZINC000217643699 CD For-Sale Unstable ADRA1D 15 48 NC/C=C\CN1CCN(c2ccccc2Cl)CC1 ZINC000217643699 CD For-Sale Unstable HTR2A 18 41 NC/C=C\CN1CCN(c2ccccc2Cl)CC1 ZINC000217643699 CD For-Sale Unstable ADRA1B 15 48 NC/C=C\CN1CCN(c2ccccc2Cl)CC1 ZINC000217643699 CD For-Sale Unstable DRD3 54 51 COc1cccc(CN[C@@H]2CCN3CCCC[C@@H]23)c1 ZINC000217643742 CE On-Demand Unstable SIGMAR1 18 43 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)Nc1ccccn1 ZINC000217643767 HH In-Stock Unstable TOP1 0 42 CCOCCCNS(=O)(=O)c1ccc(N[C@H](C)COC)c(C(=O)O)c1 ZINC000217643773 FD In-Stock Unstable CASP3 0 40 CNC(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217643796 BD On-Demand Unstable TAAR1 41 38 CNC(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217643796 BD On-Demand Unstable AKR1C3 26 40 CNC(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217643796 BD On-Demand Unstable PSBA 0 40 CNC(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217643796 BD On-Demand Unstable KCNK3 102 48 CNC(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217643796 BD On-Demand Unstable KCNK9 90 48 CNC(=O)c1cccc(NC(=O)C(F)F)c1 ZINC000217643796 BD On-Demand Unstable PARP10 0 45 CCOC(=O)CCNC(=O)/C=C\c1cccc(Br)c1 ZINC000217643806 EF On-Demand Unstable PYGL 0 43 CCOC(=O)CCNC(=O)/C=C\c1cccc(Br)c1 ZINC000217643806 EF On-Demand Unstable HDAC8 60 35 CCOC(=O)CCNC(=O)/C=C\c1cccc(Br)c1 ZINC000217643806 EF On-Demand Unstable MMP2 0 43 CCOC(=O)CCNC(=O)/C=C\c1cccc(Br)c1 ZINC000217643806 EF On-Demand Unstable HDAC9 33 40 CCOC(=O)CCNC(=O)/C=C\c1cccc(Br)c1 ZINC000217643806 EF On-Demand Unstable HDAC7 41 40 CCOC(=O)CCNC(=O)/C=C\c1cccc(Br)c1 ZINC000217643806 EF On-Demand Unstable MMP1 0 43 CCOC(=O)CCNC(=O)/C=C\c1cccc(Br)c1 ZINC000217643806 EF On-Demand Unstable HDA106 0 42 CCOC(=O)CCNC(=O)/C=C\c1cccc(Br)c1 ZINC000217643806 EF On-Demand Unstable HD1B 0 42 COc1cccc(CN[C@H]2CCN3CCCC[C@@H]23)c1 ZINC000217643813 CE On-Demand Unstable SIGMAR1 18 43 O=C(O)/C=C\c1ccc(C(=O)NCc2ccc(Cl)cc2)s1 ZINC000217643823 DG For-Sale Unstable UL54 88 38 O=C(O)/C=C\c1ccc(C(=O)NCc2ccc(Cl)cc2)s1 ZINC000217643823 DG For-Sale Unstable DPOL_VZVD 42 38 O=C(c1ccoc1)N1CCS[C@@H]1c1ccc(OC(F)(F)F)cc1 ZINC000217643840 EI In-Stock Unstable EPHX2 43 35 C/C=C/C=C/C(=O)NC[C@@](C)(O)CSC ZINC000217643842 BD On-Demand Unstable CNR2 0 56 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)Nc1ccccn1 ZINC000217643859 HH In-Stock Unstable TOP1 0 42 CCCNc1ccc(S(=O)(=O)NCCCOC(C)C)cc1C(=O)O ZINC000217643876 FE In-Stock Unstable CASP3 0 44 CCOC(=O)CCNC(=O)/C=C\c1cccc([N+](=O)[O-])c1 ZINC000217643922 CD On-Demand Unstable CACNA1C 61 41 CCOC(=O)CCNC(=O)/C=C\c1cccc([N+](=O)[O-])c1 ZINC000217643922 CD On-Demand Unstable CACNA1D 90 41 CCOC(=O)CCNC(=O)/C=C\c1cccc([N+](=O)[O-])c1 ZINC000217643922 CD On-Demand Unstable TRPM8 0 57 O=C(c1ccoc1)N1CCS[C@H]1c1ccc(OC(F)(F)F)cc1 ZINC000217643926 EI In-Stock Unstable EPHX2 43 35 C/C=C/C=C/C(=O)NC[C@](C)(O)CSC ZINC000217643932 BD On-Demand Unstable CNR2 0 56 FC(F)(F)c1cccc(CN[C@@H]2CCN3CCCC[C@@H]23)c1 ZINC000217643934 CG On-Demand Unstable TACR1 22 41 FC(F)(F)c1cccc(CN[C@@H]2CCN3CCCC[C@@H]23)c1 ZINC000217643934 CG On-Demand Unstable CCR2 27 42 COc1ccc(OCCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217643963 DG For-Sale Unstable HRH2 21 40 COc1ccc(OCCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217643963 DG For-Sale Unstable PPARG 15 43 COc1ccc(OCCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217643963 DG For-Sale Unstable LTA4H 21 41 COc1ccc(OCCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217643963 DG For-Sale Unstable MMP13 19 41 COc1ccc(OCCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217643963 DG For-Sale Unstable MTNR1A 58 45 COc1ccc(OCCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217643963 DG For-Sale Unstable MTNR1B 50 45 COc1ccc(OCCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217643963 DG For-Sale Unstable MMP2 17 47 COc1ccc(OCCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217643963 DG For-Sale Unstable MMP9 23 47 COc1ccc(OCCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217643963 DG For-Sale Unstable MMP1 21 41 CC(C)Nc1ccc(S(=O)(=O)NCCCOC(C)C)cc1C(=O)O ZINC000217643988 FE In-Stock Unstable CASP3 0 42 FC(F)(F)c1cccc(CN[C@H]2CCN3CCCC[C@@H]23)c1 ZINC000217644019 CG On-Demand Unstable TACR1 22 41 FC(F)(F)c1cccc(CN[C@H]2CCN3CCCC[C@@H]23)c1 ZINC000217644019 CG On-Demand Unstable CCR2 27 42 O=S(=O)(c1ccc2c(c1)OCCO2)N1CCS[C@@H]1c1ccc(OC(F)(F)F)cc1 ZINC000217644034 IH In-Stock Unstable PKM 41 46 CCOC(=O)CCNC(=O)/C=C\c1ccc(F)cc1 ZINC000217644066 CD On-Demand Unstable PYGL 0 41 CCOC(=O)CCNC(=O)/C=C\c1ccc(F)cc1 ZINC000217644066 CD On-Demand Unstable HDAC7 41 36 CCCCNc1ccc(S(=O)(=O)NCCCOC(C)C)cc1C(=O)O ZINC000217644076 FF In-Stock Unstable CASP3 15 43 CCCCNc1ccc(S(=O)(=O)NCCCOC(C)C)cc1C(=O)O ZINC000217644076 FF In-Stock Unstable BDKRB1 16 41 O=C(C(F)F)N1CCC[C@@H]1c1cccs1 ZINC000217644088 BF On-Demand Unstable ADAM17 47 45 O=S(=O)(c1ccc2c(c1)OCCO2)N1CCS[C@H]1c1ccc(OC(F)(F)F)cc1 ZINC000217644122 IH In-Stock Unstable PKM 41 46 CCOc1ccccc1CN[C@@H]1CCN2CCCC[C@@H]12 ZINC000217644147 CF For-Sale Unstable HCN1 47 37 CCOc1ccccc1CN[C@@H]1CCN2CCCC[C@@H]12 ZINC000217644147 CF For-Sale Unstable HCN4 45 37 CCOC(=O)CCNC(=O)/C=C\c1ccc2c(c1)OCO2 ZINC000217644151 CD On-Demand Unstable PLK1 16 41 CCOC(=O)CCNC(=O)/C=C\c1ccc2c(c1)OCO2 ZINC000217644151 CD On-Demand Unstable DYRK2 66 39 O=C(C(F)F)N1CCC[C@H]1c1cccs1 ZINC000217644173 BF On-Demand Unstable ADAM17 47 45 CC(C)CNc1ccc(S(=O)(=O)NCCCOC(C)C)cc1C(=O)O ZINC000217644181 FF In-Stock Unstable CASP3 15 43 CC(C)CNc1ccc(S(=O)(=O)NCCCOC(C)C)cc1C(=O)O ZINC000217644181 FF In-Stock Unstable BDKRB1 22 45 CC(=O)NCCNC(=O)N/C=C/c1ccccc1 ZINC000217644184 BD For-Sale Unstable MTNR1B 30 40 CCOc1ccccc1CN[C@H]1CCN2CCCC[C@@H]12 ZINC000217644234 CF For-Sale Unstable HCN1 47 37 CCOc1ccccc1CN[C@H]1CCN2CCCC[C@@H]12 ZINC000217644234 CF For-Sale Unstable HCN4 45 37 O=C(Nc1cccs1)N1CCS[C@@H]1c1ccc(OC(F)(F)F)cc1 ZINC000217644242 FJ In-Stock Unstable EPHX2 52 38 O=C(Nc1cccs1)N1CCS[C@@H]1c1ccc(OC(F)(F)F)cc1 ZINC000217644242 FJ In-Stock Unstable TRPM8 44 38 C[C@@H](N[C@@H]1CCC[C@@H](O)C1)c1cccc2ccccc12 ZINC000217644276 CH For-Sale Unstable CASR 0 47 CC[C@@H](C)Nc1ccc(S(=O)(=O)NCCCOC(C)C)cc1C(=O)O ZINC000217644327 FF In-Stock Unstable CASP3 15 40 CCOc1ccc(CN[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217644338 CF On-Demand Unstable HRH3 23 46 C[C@H](N[C@@H]1CCC[C@@H](O)C1)c1cccc2ccccc12 ZINC000217644356 CH On-Demand Unstable CASR 0 47 O=C(Nc1cccs1)N1CCS[C@H]1c1ccc(OC(F)(F)F)cc1 ZINC000217644360 FJ In-Stock Unstable P2RY1 44 39 O=C(Nc1cccs1)N1CCS[C@H]1c1ccc(OC(F)(F)F)cc1 ZINC000217644360 FJ In-Stock Unstable EPHX2 52 38 O=C(Nc1cccs1)N1CCS[C@H]1c1ccc(OC(F)(F)F)cc1 ZINC000217644360 FJ In-Stock Unstable TRPM8 50 38 CN(Cc1ccccn1)C(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217644403 DF For-Sale Unstable HSD17B2 27 45 CC[C@H](C)Nc1ccc(S(=O)(=O)NCCCOC(C)C)cc1C(=O)O ZINC000217644407 FF In-Stock Unstable CASP3 15 40 CCOc1ccc(CN[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217644413 CF On-Demand Unstable HRH3 23 46 COc1ccc(Cn2[nH]c(=O)c(Br)cc2=O)cc1 ZINC000217644429 DD For-Sale Unstable PROKR1 45 32 C[C@@H](N[C@H]1CCC[C@@H](O)C1)c1cccc2ccccc12 ZINC000217644433 CH For-Sale Unstable CASR 0 47 CCOC(=O)c1coc(C(F)F)c1C(=O)OCC ZINC000217644437 CF In-Stock Unstable CA14 0 48 O=C(N/C=C/c1ccccc1)NC12CC3CC(CC(C3)C1)C2 ZINC000217644449 CH For-Sale Unstable CNR2 17 46 O=C(N/C=C/c1ccccc1)NC12CC3CC(CC(C3)C1)C2 ZINC000217644449 CH For-Sale Unstable EPHX2 114 59 O=C(NCCc1cccs1)C(F)F ZINC000217644458 BD On-Demand Unstable ADAM17 26 62 O=C(NCCc1cccs1)C(F)F ZINC000217644458 BD On-Demand Unstable CA5B 30 42 O=C(NCCc1cccs1)C(F)F ZINC000217644458 BD On-Demand Unstable CTSC 35 46 Cc1ccccc1NC(=O)N1CCS[C@@H]1c1ccc(OC(F)(F)F)cc1 ZINC000217644482 GK In-Stock Unstable P2RX7 0 41 Cc1ccccc1NC(=O)N1CCS[C@@H]1c1ccc(OC(F)(F)F)cc1 ZINC000217644482 GK In-Stock Unstable P2RY1 65 44 Cc1ccccc1NC(=O)N1CCS[C@@H]1c1ccc(OC(F)(F)F)cc1 ZINC000217644482 GK In-Stock Unstable EPHX2 53 39 Cc1ccccc1NC(=O)N1CCS[C@@H]1c1ccc(OC(F)(F)F)cc1 ZINC000217644482 GK In-Stock Unstable SHH 40 39 CCOC(=O)CCNC(=O)/C=C\c1ccc(F)c(Cl)c1 ZINC000217644502 CF On-Demand Unstable HDAC4 23 42 CCOC(=O)CCNC(=O)/C=C\c1ccc(F)c(Cl)c1 ZINC000217644502 CF On-Demand Unstable HDAC9 39 42 CCOC(=O)CCNC(=O)/C=C\c1ccc(F)c(Cl)c1 ZINC000217644502 CF On-Demand Unstable HDAC7 40 42 CCOC(=O)CCNC(=O)/C=C\c1ccc(F)c(Cl)c1 ZINC000217644502 CF On-Demand Unstable HD1B 0 43 C[C@H](N[C@H]1CCC[C@@H](O)C1)c1cccc2ccccc12 ZINC000217644503 CH On-Demand Unstable CASR 0 47 Fc1cccc(CN[C@@H]2CCN3CCCC[C@@H]23)c1 ZINC000217644515 BF On-Demand Unstable VACHT_TETCF 0 43 Fc1cccc(CN[C@@H]2CCN3CCCC[C@@H]23)c1 ZINC000217644515 BF On-Demand Unstable SSTR3 18 41 CC(C)OCCCNS(=O)(=O)c1ccc(NC(C)(C)C)c(C(=O)O)c1 ZINC000217644526 FF In-Stock Unstable CASP3 17 41 O=C(Cn1c(=O)[nH]c2ccccc2c1=O)NC[C@@H]1CC[C@@H](C(=O)NC[C@@H]2CC[C@@H](C(=O)O)CC2)CC1 ZINC000217644562 JD In-Stock Unstable AVPR1B 31 42 Cc1ccccc1NC(=O)N1CCS[C@H]1c1ccc(OC(F)(F)F)cc1 ZINC000217644565 GK In-Stock Unstable P2RX7 0 41 Cc1ccccc1NC(=O)N1CCS[C@H]1c1ccc(OC(F)(F)F)cc1 ZINC000217644565 GK In-Stock Unstable P2RY1 65 44 Cc1ccccc1NC(=O)N1CCS[C@H]1c1ccc(OC(F)(F)F)cc1 ZINC000217644565 GK In-Stock Unstable EPHX2 53 39 Cc1ccccc1NC(=O)N1CCS[C@H]1c1ccc(OC(F)(F)F)cc1 ZINC000217644565 GK In-Stock Unstable SHH 40 39 O=C(N/C=C/c1ccccc1)Nc1cccc2cccnc12 ZINC000217644570 CI For-Sale Anodyne PFHDAC1 0 51 CCCNC(=O)CNC(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217644576 CD For-Sale Unstable CA2 23 41 Fc1cccc(CN[C@H]2CCN3CCCC[C@@H]23)c1 ZINC000217644593 BF On-Demand Unstable VACHT_TETCF 0 43 Fc1cccc(CN[C@H]2CCN3CCCC[C@@H]23)c1 ZINC000217644593 BF On-Demand Unstable SSTR3 18 41 CSCC[C@@H](CO)NC(=O)CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217644621 ID In-Stock Unstable EDNRA 18 40 C=CCNc1ccc(S(=O)(=O)NCCCOC(C)C)cc1C(=O)O ZINC000217644632 FE In-Stock Unstable CASP3 0 41 C[C@H](N[C@@H]1CCCC[C@@H]1C)C(=O)Nc1nc2ccccc2s1 ZINC000217644657 DH On-Demand Unstable CSNK1D 27 44 C[C@H](N[C@@H]1CCCC[C@@H]1C)C(=O)Nc1nc2ccccc2s1 ZINC000217644657 DH On-Demand Unstable TMPRSS6 46 34 COc1ccc(C(=O)Nc2nncs2)cc1/C=C\C(=O)O ZINC000217644659 DD For-Sale Unstable COLA 26 42 COc1ccc(C(=O)Nc2nncs2)cc1/C=C\C(=O)O ZINC000217644659 DD For-Sale Unstable CPT1A 32 42 COc1cccc(NC(=O)N2CCS[C@@H]2c2ccc(OC(F)(F)F)cc2)c1OC ZINC000217644677 IJ In-Stock Unstable HCRTR1 24 41 COc1cccc(NC(=O)N2CCS[C@@H]2c2ccc(OC(F)(F)F)cc2)c1OC ZINC000217644677 IJ In-Stock Unstable P2RY1 60 41 COc1cccc(NC(=O)N2CCS[C@@H]2c2ccc(OC(F)(F)F)cc2)c1OC ZINC000217644677 IJ In-Stock Unstable EPHX2 46 39 COc1cccc(NC(=O)N2CCS[C@@H]2c2ccc(OC(F)(F)F)cc2)c1OC ZINC000217644677 IJ In-Stock Unstable HCRTR2 16 41 CCOC(=O)CCNC(=O)/C=C\c1ccc(C(C)C)cc1 ZINC000217644684 CF For-Sale Unstable PYGL 0 42 COc1ccccc1CN[C@@H]1CCN2CCCC[C@@H]12 ZINC000217644716 CE On-Demand Unstable TACR1 35 41 Cc1ncn(CCNC(=O)Cc2ccc(O)c(F)c2)c1C ZINC000217644744 CD In-Stock Unstable P2RX7 39 40 CC(C)OCCCNS(=O)(=O)c1ccc(NC2CC2)c(C(=O)O)c1 ZINC000217644749 FE In-Stock Unstable CASP3 0 43 COc1cccc(NC(=O)N2CCS[C@H]2c2ccc(OC(F)(F)F)cc2)c1OC ZINC000217644768 IJ In-Stock Unstable HCRTR1 24 41 COc1cccc(NC(=O)N2CCS[C@H]2c2ccc(OC(F)(F)F)cc2)c1OC ZINC000217644768 IJ In-Stock Unstable P2RY1 60 41 COc1cccc(NC(=O)N2CCS[C@H]2c2ccc(OC(F)(F)F)cc2)c1OC ZINC000217644768 IJ In-Stock Unstable EPHX2 46 39 COc1cccc(NC(=O)N2CCS[C@H]2c2ccc(OC(F)(F)F)cc2)c1OC ZINC000217644768 IJ In-Stock Unstable HCRTR2 16 41 NS(=O)(=O)c1ccc(CNC(=O)C(F)F)s1 ZINC000217644787 CC On-Demand Unstable CA2 16 40 COc1ccccc1CN[C@H]1CCN2CCCC[C@@H]12 ZINC000217644795 CE On-Demand Unstable TACR1 35 41 C[C@@H]1Cc2ccccc2N1C(=O)N/C=C/c1ccccc1 ZINC000217644808 CH For-Sale Unstable ACE 17 43 C[C@@H]1Cc2ccccc2N1C(=O)N/C=C/c1ccccc1 ZINC000217644808 CH For-Sale Unstable DRD4 28 44 C[C@@H]1Cc2ccccc2N1C(=O)N/C=C/c1ccccc1 ZINC000217644808 CH For-Sale Unstable TPP2 56 35 C[C@H](N[C@H]1CCCC[C@@H]1C)C(=O)Nc1nc2ccccc2s1 ZINC000217644825 DH On-Demand Unstable CSNK1D 27 44 C[C@H](N[C@H]1CCCC[C@@H]1C)C(=O)Nc1nc2ccccc2s1 ZINC000217644825 DH On-Demand Unstable TMPRSS6 46 34 CCOC(=O)CCNC(=O)/C=C\c1ccccc1F ZINC000217644845 CD On-Demand Unstable KCNQ2 41 38 CCOC(=O)CCNC(=O)/C=C\c1ccccc1F ZINC000217644845 CD On-Demand Unstable HDAC9 20 41 CCOC(=O)CCNC(=O)/C=C\c1ccccc1F ZINC000217644845 CD On-Demand Unstable HDAC7 31 41 Cn1ccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)n1 ZINC000217644850 CD For-Sale Unstable HDAC8 33 44 Cn1ccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)n1 ZINC000217644850 CD For-Sale Unstable HDAC6 15 44 Cn1ccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)n1 ZINC000217644850 CD For-Sale Unstable GCK 24 48 Cn1ccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)n1 ZINC000217644850 CD For-Sale Unstable RHOA 0 40 Cn1ccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)n1 ZINC000217644850 CD For-Sale Unstable KCNK3 70 36 CC(C)OCCCNS(=O)(=O)c1ccc(NC2CCCC2)c(C(=O)O)c1 ZINC000217644871 GF In-Stock Unstable CASP3 0 45 C[C@H]1Cc2ccccc2N1C(=O)N/C=C/c1ccccc1 ZINC000217644899 CH For-Sale Unstable ACE 17 43 C[C@H]1Cc2ccccc2N1C(=O)N/C=C/c1ccccc1 ZINC000217644899 CH For-Sale Unstable DRD4 28 44 C[C@H]1Cc2ccccc2N1C(=O)N/C=C/c1ccccc1 ZINC000217644899 CH For-Sale Unstable TPP2 56 35 Cn1ccc(NC(=O)c2cc(/C=C\C(=O)O)ccc2F)n1 ZINC000217644957 CD For-Sale Unstable GCK 18 43 C=CCn1c(SCCC(=O)Nc2sc3c(c2C#N)CCCC3)nnc1-c1ccccc1F ZINC000217644962 JK On-Demand Unstable MAPK10 18 48 C=CCn1c(SCCC(=O)Nc2sc3c(c2C#N)CCCC3)nnc1-c1ccccc1F ZINC000217644962 JK On-Demand Unstable VIPR1 29 49 CC(C)OCCCNS(=O)(=O)c1ccc(NC2CCCCC2)c(C(=O)O)c1 ZINC000217644975 GG In-Stock Unstable CASP3 0 45 CN1CCN(C(=O)[C@@H]2CC[C@H](O)CC2)C[C@@H]1c1ccccc1 ZINC000217644998 DE In-Stock Unstable VACHT_TETCF 0 44 Cn1ccc(NC(=O)c2ccc(/C=C\C(=O)O)cc2F)n1 ZINC000217645039 CD For-Sale Unstable GCK 19 43 CN1CCN(C(=O)[C@@H]2CC[C@H](O)CC2)C[C@H]1c1ccccc1 ZINC000217645068 DE In-Stock Unstable VACHT_TETCF 0 44 COC(=O)CS(=O)(=O)Nc1cccc(/C=C\C(=O)O)c1 ZINC000217645123 CC For-Sale Unstable HDAC8 17 42 Cc1ccccc1CN[C@@H]1CCN2CCCC[C@@H]12 ZINC000217645124 BF On-Demand Unstable VACHT_TETCF 0 44 Cc1ccccc1CN[C@@H]1CCN2CCCC[C@@H]12 ZINC000217645124 BF On-Demand Unstable SLC18A3 48 39 COc1ccc(-c2coc3ccc(OCC(C)=O)cc23)cc1 ZINC000217645127 CI In-Stock Unstable ALDH2 110 47 COc1ccc(-c2coc3ccc(OCC(C)=O)cc23)cc1 ZINC000217645127 CI In-Stock Unstable IL2 25 42 COc1ccc(-c2coc3ccc(OCC(C)=O)cc23)cc1 ZINC000217645127 CI In-Stock Unstable NQO2 21 46 COc1ccc(-c2coc3ccc(OCC(C)=O)cc23)cc1 ZINC000217645127 CI In-Stock Unstable GSK3B 0 54 COc1ccc(-c2coc3ccc(OCC(C)=O)cc23)cc1 ZINC000217645127 CI In-Stock Unstable MTNR1A 63 46 COc1ccc(-c2coc3ccc(OCC(C)=O)cc23)cc1 ZINC000217645127 CI In-Stock Unstable MTNR1B 47 46 COc1ccccc1CNC(=O)N/C=C/c1ccccc1 ZINC000217645129 CG For-Sale Unstable ANPEP 25 55 COc1ccccc1CNC(=O)N/C=C/c1ccccc1 ZINC000217645129 CG For-Sale Unstable TACR1 0 43 COc1ccccc1CNC(=O)N/C=C/c1ccccc1 ZINC000217645129 CG For-Sale Unstable KCNA3 40 38 COc1ccccc1CNC(=O)N/C=C/c1ccccc1 ZINC000217645129 CG For-Sale Unstable AMP1_PLAFQ 44 33 COc1ccccc1CNC(=O)N/C=C/c1ccccc1 ZINC000217645129 CG For-Sale Unstable GPM3 0 47 CC(C)OCCCNS(=O)(=O)c1ccc(NCCO)c(C(=O)O)c1 ZINC000217645188 FC In-Stock Unstable CASP3 16 41 CC(C)OCCCNS(=O)(=O)c1ccc(NCCO)c(C(=O)O)c1 ZINC000217645188 FC In-Stock Unstable BDKRB1 0 41 N#Cc1cccnc1N1CCN(c2ccc(C(=O)O)cn2)C[C@@H](O)C1 ZINC000217645201 EC In-Stock Unstable SMO 27 43 Cc1ccccc1CN[C@H]1CCN2CCCC[C@@H]12 ZINC000217645206 BF On-Demand Unstable VACHT_TETCF 0 44 Cc1ccccc1CN[C@H]1CCN2CCCC[C@@H]12 ZINC000217645206 BF On-Demand Unstable SLC18A3 48 39 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](C)C(=O)Nc3ccc4ccn(C)c4c3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217645228 KJ In-Stock Unstable TUBA1A 17 62 O=C(N/C=C/c1ccccc1)N1CCN(c2ncccn2)CC1 ZINC000217645268 DD For-Sale Unstable FAAH 25 41 O=C(N/C=C/c1ccccc1)N1CCN(c2ncccn2)CC1 ZINC000217645268 DD For-Sale Unstable SLC6A7 0 50 CC(C)OCCCNS(=O)(=O)c1ccc(NCCCO)c(C(=O)O)c1 ZINC000217645278 FD In-Stock Unstable CASP3 16 41 CC(C)OCCCNS(=O)(=O)c1ccc(NCCCO)c(C(=O)O)c1 ZINC000217645278 FD In-Stock Unstable BDKRB1 0 41 Cc1ccc(CN[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217645318 BF On-Demand Unstable SLC18A3 19 45 N#Cc1c(NC(=O)CCN2CCN([C@@H](C#N)c3ccccc3)CC2)sc2c1CCCCC2 ZINC000217645341 II On-Demand Unstable PTAFR 34 45 N#Cc1c(NC(=O)CCN2CCN([C@@H](C#N)c3ccccc3)CC2)sc2c1CCCCC2 ZINC000217645341 II On-Demand Unstable MAPK10 0 56 N#Cc1c(NC(=O)CCN2CCN([C@@H](C#N)c3ccccc3)CC2)sc2c1CCCCC2 ZINC000217645341 II On-Demand Unstable FLT3 0 43 N#Cc1c(NC(=O)CCN2CCN([C@@H](C#N)c3ccccc3)CC2)sc2c1CCCCC2 ZINC000217645341 II On-Demand Unstable MURF 0 42 N#Cc1c(NC(=O)CCN2CCN([C@@H](C#N)c3ccccc3)CC2)sc2c1CCCCC2 ZINC000217645341 II On-Demand Unstable VIPR1 34 60 O=C1COc2ccc(NC(=O)C(F)F)cc2N1 ZINC000217645357 BD On-Demand Unstable NR3C2 24 46 O=C1COc2ccc(NC(=O)C(F)F)cc2N1 ZINC000217645357 BD On-Demand Unstable TRPV1 0 52 Cc1cccc(N2CCN(C(=O)N/C=C/c3ccccc3)CC2)c1 ZINC000217645380 DG For-Sale Unstable MMP2 0 42 Cc1cccc(N2CCN(C(=O)N/C=C/c3ccccc3)CC2)c1 ZINC000217645380 DG For-Sale Unstable FAAH 0 42 Cc1cccc(N2CCN(C(=O)N/C=C/c3ccccc3)CC2)c1 ZINC000217645380 DG For-Sale Unstable ADAM10 32 42 Cc1cccc(N2CCN(C(=O)N/C=C/c3ccccc3)CC2)c1 ZINC000217645380 DG For-Sale Unstable GPR183 0 41 COCCNc1ccc(S(=O)(=O)NCCCOC(C)C)cc1C(=O)O ZINC000217645383 FD In-Stock Unstable CASP3 16 41 COCCNc1ccc(S(=O)(=O)NCCCOC(C)C)cc1C(=O)O ZINC000217645383 FD In-Stock Unstable BDKRB1 0 44 Cc1ccc(CN[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217645394 BF On-Demand Unstable SLC18A3 19 45 N#Cc1c(NC(=O)CCN2CCN([C@H](C#N)c3ccccc3)CC2)sc2c1CCCCC2 ZINC000217645413 II On-Demand Unstable PTAFR 34 45 N#Cc1c(NC(=O)CCN2CCN([C@H](C#N)c3ccccc3)CC2)sc2c1CCCCC2 ZINC000217645413 II On-Demand Unstable MAPK10 0 56 N#Cc1c(NC(=O)CCN2CCN([C@H](C#N)c3ccccc3)CC2)sc2c1CCCCC2 ZINC000217645413 II On-Demand Unstable FLT3 0 43 N#Cc1c(NC(=O)CCN2CCN([C@H](C#N)c3ccccc3)CC2)sc2c1CCCCC2 ZINC000217645413 II On-Demand Unstable MURF 0 42 N#Cc1c(NC(=O)CCN2CCN([C@H](C#N)c3ccccc3)CC2)sc2c1CCCCC2 ZINC000217645413 II On-Demand Unstable VIPR1 34 60 CC(C)C[C@H](NC(=O)Cn1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217645458 JD In-Stock Unstable AVPR1B 61 42 CC(C)C[C@H](NC(=O)Cn1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217645458 JD In-Stock Unstable ELANE 20 42 CC(C)C[C@H](NC(=O)Cn1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217645458 JD In-Stock Unstable BRS3 18 41 CC(C)C[C@H](NC(=O)Cn1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217645458 JD In-Stock Unstable NMBR 18 40 CC(C)C[C@H](NC(=O)Cn1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217645458 JD In-Stock Unstable CAPN1 52 37 CC(C)C[C@H](NC(=O)Cn1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217645458 JD In-Stock Unstable CAPN2 80 37 CC(C)C[C@H](NC(=O)Cn1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217645458 JD In-Stock Unstable NPR 58 32 CC(C)C[C@H](NC(=O)Cn1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217645458 JD In-Stock Unstable KISS1R 49 31 COCCCNc1ccc(S(=O)(=O)NCCCOC(C)C)cc1C(=O)O ZINC000217645480 GD In-Stock Unstable CASP3 17 41 COCCCNc1ccc(S(=O)(=O)NCCCOC(C)C)cc1C(=O)O ZINC000217645480 GD In-Stock Unstable BDKRB1 0 44 CCOC(=O)N1CCC(NC(=O)N/C=C/c2ccccc2)CC1 ZINC000217645498 DF For-Sale Unstable CHRM1 18 52 CCOC(=O)N1CCC(NC(=O)N/C=C/c2ccccc2)CC1 ZINC000217645498 DF For-Sale Unstable P2RY12 56 37 CCOC(=O)N1CCC(NC(=O)N/C=C/c2ccccc2)CC1 ZINC000217645498 DF For-Sale Unstable SIGMAR1 16 43 CCOC(=O)N1CCC(NC(=O)N/C=C/c2ccccc2)CC1 ZINC000217645498 DF For-Sale Unstable EPHX2 44 50 CCOC(=O)N1CCC(NC(=O)N/C=C/c2ccccc2)CC1 ZINC000217645498 DF For-Sale Unstable CCR8 65 45 C=C(NC(=O)c1ccccc1)C(=O)OCC ZINC000217645505 BD For-Sale Unstable CTSG 31 40 C=C(NC(=O)c1ccccc1)C(=O)OCC ZINC000217645505 BD For-Sale Unstable CTRB1 36 40 C=C(NC(=O)c1ccccc1)C(=O)OCC ZINC000217645505 BD For-Sale Unstable CELA2A 22 40 C=C(NC(=O)c1ccccc1)C(=O)OCC ZINC000217645505 BD For-Sale Unstable CASP1 15 42 C=C(NC(=O)c1ccccc1)C(=O)OCC ZINC000217645505 BD For-Sale Unstable CTRB_BOVIN 45 33 C=C(NC(=O)c1ccccc1)C(=O)OCC ZINC000217645505 BD For-Sale Unstable KCNK3 69 40 C=C(NC(=O)c1ccccc1)C(=O)OCC ZINC000217645505 BD For-Sale Unstable KCNK9 49 40 N#Cc1c(NC(=O)CCN2CCN([C@@H](C#N)c3ccccc3)CC2)sc2c1CCCC2 ZINC000217645516 IH On-Demand Unstable PTAFR 36 45 N#Cc1c(NC(=O)CCN2CCN([C@@H](C#N)c3ccccc3)CC2)sc2c1CCCC2 ZINC000217645516 IH On-Demand Unstable GRM1 0 41 N#Cc1c(NC(=O)CCN2CCN([C@@H](C#N)c3ccccc3)CC2)sc2c1CCCC2 ZINC000217645516 IH On-Demand Unstable MAPK10 0 57 N#Cc1c(NC(=O)CCN2CCN([C@@H](C#N)c3ccccc3)CC2)sc2c1CCCC2 ZINC000217645516 IH On-Demand Unstable FLT3 0 44 N#Cc1c(NC(=O)CCN2CCN([C@@H](C#N)c3ccccc3)CC2)sc2c1CCCC2 ZINC000217645516 IH On-Demand Unstable VIPR1 35 61 CCOc1cc(CN[C@@H]2CCN3CCCC[C@@H]23)ccc1O ZINC000217645522 CF For-Sale Unstable SSTR5 61 43 CC(C)OCCCNS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217645593 HG In-Stock Unstable BDKRB1 0 43 CCOc1cc(CN[C@H]2CCN3CCCC[C@@H]23)ccc1O ZINC000217645603 CF For-Sale Unstable SSTR5 61 43 N#Cc1c(NC(=O)CCN2CCN([C@H](C#N)c3ccccc3)CC2)sc2c1CCCC2 ZINC000217645605 IH On-Demand Unstable PTAFR 36 45 N#Cc1c(NC(=O)CCN2CCN([C@H](C#N)c3ccccc3)CC2)sc2c1CCCC2 ZINC000217645605 IH On-Demand Unstable GRM1 0 41 N#Cc1c(NC(=O)CCN2CCN([C@H](C#N)c3ccccc3)CC2)sc2c1CCCC2 ZINC000217645605 IH On-Demand Unstable MAPK10 0 57 N#Cc1c(NC(=O)CCN2CCN([C@H](C#N)c3ccccc3)CC2)sc2c1CCCC2 ZINC000217645605 IH On-Demand Unstable FLT3 0 44 N#Cc1c(NC(=O)CCN2CCN([C@H](C#N)c3ccccc3)CC2)sc2c1CCCC2 ZINC000217645605 IH On-Demand Unstable VIPR1 35 61 O=C(N/C=C/c1ccccc1)N1CCN(c2cccc(Cl)c2)CC1 ZINC000217645606 EH For-Sale Unstable HTR1A 20 47 O=C(N/C=C/c1ccccc1)N1CCN(c2cccc(Cl)c2)CC1 ZINC000217645606 EH For-Sale Unstable HTR2A 16 47 O=C(N/C=C/c1ccccc1)N1CCN(c2cccc(Cl)c2)CC1 ZINC000217645606 EH For-Sale Unstable HTR7 17 43 O=C(N/C=C/c1ccccc1)N1CCN(c2cccc(Cl)c2)CC1 ZINC000217645606 EH For-Sale Unstable FAAH 16 45 O=C(N/C=C/c1ccccc1)N1CCN(c2cccc(Cl)c2)CC1 ZINC000217645606 EH For-Sale Unstable ADAM10 29 42 CCc1cccc(NC(=O)C(F)F)c1 ZINC000217645644 AE On-Demand Unstable SIGMAR1 16 56 CCc1cccc(NC(=O)C(F)F)c1 ZINC000217645644 AE On-Demand Unstable PTGER3 20 46 CCc1cccc(NC(=O)C(F)F)c1 ZINC000217645644 AE On-Demand Unstable NAMPT 22 44 CCc1cccc(NC(=O)C(F)F)c1 ZINC000217645644 AE On-Demand Unstable PSBA 0 40 CCc1cccc(NC(=O)C(F)F)c1 ZINC000217645644 AE On-Demand Unstable KCNK3 68 36 CCc1cccc(NC(=O)C(F)F)c1 ZINC000217645644 AE On-Demand Unstable KCNK9 64 36 CCc1cccc(NC(=O)C(F)F)c1 ZINC000217645644 AE On-Demand Unstable PARP10 50 38 CC(C)OCCCNS(=O)(=O)c1ccc(N[C@@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217645704 HH In-Stock Unstable CASP3 18 42 CC(C)OCCCNS(=O)(=O)c1ccc(N[C@@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217645704 HH In-Stock Unstable BDKRB1 0 44 Cc1ccc2nc(-c3ccc(NC(=O)N/C=C/c4ccccc4)cc3)sc2c1 ZINC000217645706 GK For-Sale Unstable APP 26 54 Cc1cccc(CN[C@@H]2CCN3CCCC[C@@H]23)c1 ZINC000217645725 BF On-Demand Unstable VACHT_TETCF 0 43 O=C(NCCc1ccc(Cl)cc1Cl)NCc1coc(-c2cccs2)n1 ZINC000217645729 GJ On-Demand Unstable MC5R 41 36 O=C(Cc1ccsc1)Nc1ccccc1Cc1nc(-c2cnccn2)no1 ZINC000217645768 GG In-Stock Unstable HCAR2 25 42 O=C(NCCc1ccc(F)cc1)C(F)F ZINC000217645780 BD On-Demand Unstable CA12 15 51 O=C(NCCc1ccc(F)cc1)C(F)F ZINC000217645780 BD On-Demand Unstable AMP1_PLAFQ 31 44 O=C(NCCc1ccc(F)cc1)C(F)F ZINC000217645780 BD On-Demand Unstable LEF 78 44 O=C(NCCc1ccc(F)cc1)C(F)F ZINC000217645780 BD On-Demand Unstable Q76353_9HIV1 0 44 CC(C)OCCCNS(=O)(=O)c1ccc(N[C@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217645797 HH In-Stock Unstable CASP3 18 42 CC(C)OCCCNS(=O)(=O)c1ccc(N[C@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217645797 HH In-Stock Unstable BDKRB1 0 44 Cc1cccc(CN[C@H]2CCN3CCCC[C@@H]23)c1 ZINC000217645808 BF On-Demand Unstable VACHT_TETCF 0 43 O=C(N/C=C/c1ccccc1)Nc1ccc2c(c1)OCO2 ZINC000217645812 CG For-Sale Unstable DYRK2 52 38 Cc1nc2ccccc2n1CCNC(=O)NCCc1ccc(Cl)cc1Cl ZINC000217645822 GI On-Demand Unstable CNR1 41 45 Cc1nc2ccccc2n1CCNC(=O)NCCc1ccc(Cl)cc1Cl ZINC000217645822 GI On-Demand Unstable CNR2 20 42 Cc1nc2ccccc2n1CCNC(=O)NCCc1ccc(Cl)cc1Cl ZINC000217645822 GI On-Demand Unstable P2RX7 37 41 Cc1nc2ccccc2n1CCNC(=O)NCCc1ccc(Cl)cc1Cl ZINC000217645822 GI On-Demand Unstable MC5R 41 35 Cc1nc2ccccc2n1CCNC(=O)NCCc1ccc(Cl)cc1Cl ZINC000217645822 GI On-Demand Unstable PTGDR2 18 43 Cc1nc2ccccc2n1CCNC(=O)NCCc1ccc(Cl)cc1Cl ZINC000217645822 GI On-Demand Unstable IMDH_CRYPV 32 41 CSCC[C@@H](NC(=O)[C@@H]1CC[C@@H](CNC(=O)Cn2c(=O)[nH]c3ccccc3c2=O)CC1)C(=O)O ZINC000217645869 JC In-Stock Unstable EDNRB 29 41 CC(C)OCCCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217645921 HG In-Stock Unstable TBXA2R 44 37 CC(C)OCCCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217645921 HG In-Stock Unstable CASP3 17 41 CC(C)OCCCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217645921 HG In-Stock Unstable BDKRB1 0 43 COc1cc(N)c(Br)cc1Cc1ccccc1 ZINC000217645923 CH For-Sale Unstable DRTS_PLAFK 39 40 C[C@@H](C(=O)NC1CC1)N1CCN(C(=O)NCCOc2ccc3ccccc3c2)CC1 ZINC000217645944 HE On-Demand Unstable HRH3 15 41 CC(C)C[C@H](NC(=O)[C@@H]1CC[C@@H](CNC(=O)Cn2c(=O)[nH]c3ccccc3c2=O)CC1)C(=O)O ZINC000217645969 JD In-Stock Unstable AVPR1B 37 42 CC(C)C[C@H](NC(=O)[C@@H]1CC[C@@H](CNC(=O)Cn2c(=O)[nH]c3ccccc3c2=O)CC1)C(=O)O ZINC000217645969 JD In-Stock Unstable EDNRB 29 40 CC(C)C[C@H](NC(=O)[C@@H]1CC[C@@H](CNC(=O)Cn2c(=O)[nH]c3ccccc3c2=O)CC1)C(=O)O ZINC000217645969 JD In-Stock Unstable EDNRA 25 40 CC(C)C[C@H](NC(=O)[C@@H]1CC[C@@H](CNC(=O)Cn2c(=O)[nH]c3ccccc3c2=O)CC1)C(=O)O ZINC000217645969 JD In-Stock Unstable FPR1 46 34 CC(C)C[C@H](NC(=O)[C@@H]1CC[C@@H](CNC(=O)Cn2c(=O)[nH]c3ccccc3c2=O)CC1)C(=O)O ZINC000217645969 JD In-Stock Unstable NPR 45 33 C[C@@H]1O[C@H](c2cc(Br)ccc2F)CN[C@@H]1C(=O)O ZINC000217646002 DE For-Sale Unstable GRIK2 79 41 CSC[C@@](C)(O)CNC(=O)CCOc1cccc(F)c1 ZINC000217646004 DD On-Demand Unstable PDS 41 41 O=C(N/C=C/c1ccccc1)Nc1cccc(F)c1 ZINC000217646018 CH For-Sale Anodyne MMP1 0 66 O=C(N/C=C/c1ccccc1)Nc1cccc(F)c1 ZINC000217646018 CH For-Sale Anodyne KCNK3 53 48 C[C@H](C(=O)NC1CC1)N1CCN(C(=O)NCCOc2ccc3ccccc3c2)CC1 ZINC000217646036 HE On-Demand Unstable HRH3 15 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCCCOC(C)C)cc2C(=O)O)cc1 ZINC000217646037 JG In-Stock Unstable TBXA2R 38 42 COc1ccc(CCNc2ccc(S(=O)(=O)NCCCOC(C)C)cc2C(=O)O)cc1 ZINC000217646037 JG In-Stock Unstable TBXAS1 27 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCCCOC(C)C)cc2C(=O)O)cc1 ZINC000217646037 JG In-Stock Unstable BMP1 74 35 COc1ccc(CCNc2ccc(S(=O)(=O)NCCCOC(C)C)cc2C(=O)O)cc1 ZINC000217646037 JG In-Stock Unstable IAP 0 46 COc1ccc(CCNc2ccc(S(=O)(=O)NCCCOC(C)C)cc2C(=O)O)cc1 ZINC000217646037 JG In-Stock Unstable CA9 19 40 COc1ccc(CCNc2ccc(S(=O)(=O)NCCCOC(C)C)cc2C(=O)O)cc1 ZINC000217646037 JG In-Stock Unstable AKR1C3 25 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCCCOC(C)C)cc2C(=O)O)cc1 ZINC000217646037 JG In-Stock Unstable AKR1C2 41 36 Clc1nccc2c1CN(Cc1ccccc1)C2 ZINC000217646070 BG For-Sale Unstable SIGMAR1 30 44 CSC[C@](C)(O)CNC(=O)CCOc1cccc(F)c1 ZINC000217646085 DD On-Demand Unstable PDS 41 41 Cc1ccc([C@@H](NC(=O)CCCN2CCOCC2)c2ccncc2)cc1 ZINC000217646107 FF In-Stock Unstable CASR 41 35 Cc1ccc([C@@H](NC(=O)CCCN2CCOCC2)c2ccncc2)cc1 ZINC000217646107 FF In-Stock Unstable PRCP 33 48 O=C(N/C=C/c1ccccc1)NCCc1ccc(F)cc1 ZINC000217646144 CG For-Sale Unstable MMP2 15 53 O=C(N/C=C/c1ccccc1)NCCc1ccc(F)cc1 ZINC000217646144 CG For-Sale Unstable AMP1_PLAFQ 31 46 CCOC(=O)CCCNC(=O)C(F)F ZINC000217646147 BC On-Demand Unstable EPHX2 25 44 CCOC(=O)CCCNC(=O)C(F)F ZINC000217646147 BC On-Demand Unstable MLYCD 0 42 COc1ccc(CCNc2ccc(S(=O)(=O)NCCCOC(C)C)cc2C(=O)O)cc1OC ZINC000217646149 JG In-Stock Unstable TBXAS1 18 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCCCOC(C)C)cc2C(=O)O)cc1OC ZINC000217646149 JG In-Stock Unstable BDKRB1 0 40 COc1ccc(CCNc2ccc(S(=O)(=O)NCCCOC(C)C)cc2C(=O)O)cc1OC ZINC000217646149 JG In-Stock Unstable IAP 0 47 COc1ccc(CCNc2ccc(S(=O)(=O)NCCCOC(C)C)cc2C(=O)O)cc1OC ZINC000217646149 JG In-Stock Unstable SCMU_MYCTU 0 42 COCCNC(=O)NC[C@H](c1ccc(Cl)cc1Cl)c1c[nH]c2ccccc12 ZINC000217646161 HJ On-Demand Unstable ALPL 37 43 COC(=O)C[C@H](c1cc2cc(OC)ccc2[nH]c1=O)c1c(O)c2ccccc2oc1=O ZINC000217646162 HG In-Stock Unstable TUBB2B 37 40 COC(=O)C[C@H](c1cc2cc(OC)ccc2[nH]c1=O)c1c(O)c2ccccc2oc1=O ZINC000217646162 HG In-Stock Unstable NQO1 37 52 Cc1ccc([C@H](NC(=O)CCCN2CCOCC2)c2ccncc2)cc1 ZINC000217646178 FF In-Stock Unstable CASR 41 35 Cc1ccc([C@H](NC(=O)CCCN2CCOCC2)c2ccncc2)cc1 ZINC000217646178 FF In-Stock Unstable PRCP 33 48 C[C@@H]1O[C@H](c2ccc(Br)cc2F)CN[C@@H]1C(=O)O ZINC000217646184 DE For-Sale Unstable GRIK2 80 41 NC[C@@H](O)c1cc(O)c(Br)c(F)c1 ZINC000217646237 CD For-Sale Unstable ADRB1 18 71 COC(=O)C[C@@H](c1cc2cc(OC)ccc2[nH]c1=O)c1c(O)c2ccccc2oc1=O ZINC000217646249 HG In-Stock Unstable TUBB2B 37 40 COC(=O)C[C@@H](c1cc2cc(OC)ccc2[nH]c1=O)c1c(O)c2ccccc2oc1=O ZINC000217646249 HG In-Stock Unstable NQO1 37 52 COCCNC(=O)NC[C@@H](c1ccc(Cl)cc1Cl)c1c[nH]c2ccccc12 ZINC000217646254 HJ On-Demand Unstable ALPL 37 43 NC[C@H](O)c1cc(O)c(Br)c(F)c1 ZINC000217646323 CD For-Sale Unstable ADRB1 18 71 O=C(N/C=C/c1ccccc1)Nc1ccc(I)cc1 ZINC000217646368 FI For-Sale Anodyne EPHX1 0 44 O=C(N/C=C/c1ccccc1)Nc1ccc(I)cc1 ZINC000217646368 FI For-Sale Anodyne P95276_MYCTO 0 44 c1ccc2cc([C@H]3CC[C@H]3c3ccc4ccccc4c3)ccc2c1 ZINC000217646378 DK For-Sale Unstable SLC6A3 22 42 c1ccc2cc([C@H]3CC[C@H]3c3ccc4ccccc4c3)ccc2c1 ZINC000217646378 DK For-Sale Unstable ERBB2 17 40 c1ccc2cc([C@H]3CC[C@H]3c3ccc4ccccc4c3)ccc2c1 ZINC000217646378 DK For-Sale Unstable TRYP_PIG 19 43 c1ccc2cc([C@H]3CC[C@@H]3c3ccc4ccccc4c3)ccc2c1 ZINC000217646460 DK For-Sale Unstable SLC6A3 22 42 c1ccc2cc([C@H]3CC[C@@H]3c3ccc4ccccc4c3)ccc2c1 ZINC000217646460 DK For-Sale Unstable ERBB2 17 40 c1ccc2cc([C@H]3CC[C@@H]3c3ccc4ccccc4c3)ccc2c1 ZINC000217646460 DK For-Sale Unstable TRYP_PIG 19 43 O=C(N/C=C/c1ccccc1)NCCc1c[nH]c2ccccc12 ZINC000217646468 DH For-Sale Unstable TACR1 18 45 O=C(N/C=C/c1ccccc1)NCCc1c[nH]c2ccccc12 ZINC000217646468 DH For-Sale Unstable CCKAR 70 47 O=C(N/C=C/c1ccccc1)NCCc1c[nH]c2ccccc12 ZINC000217646468 DH For-Sale Unstable MPO 36 43 O=C(N/C=C/c1ccccc1)NCCc1c[nH]c2ccccc12 ZINC000217646468 DH For-Sale Unstable BRS3 29 46 O=C(N/C=C/c1ccccc1)NCCc1c[nH]c2ccccc12 ZINC000217646468 DH For-Sale Unstable NMBR 47 47 O=C(N/C=C/c1ccccc1)NCCc1c[nH]c2ccccc12 ZINC000217646468 DH For-Sale Unstable MC5R 33 41 O=C(N/C=C/c1ccccc1)NCCc1c[nH]c2ccccc12 ZINC000217646468 DH For-Sale Unstable ECE1 40 39 O=C(N/C=C/c1ccccc1)NCCc1c[nH]c2ccccc12 ZINC000217646468 DH For-Sale Unstable HDAC3 17 44 O=C(N/C=C/c1ccccc1)NCCc1c[nH]c2ccccc12 ZINC000217646468 DH For-Sale Unstable MMP11 54 33 O=C(N/C=C/c1ccccc1)NCCc1c[nH]c2ccccc12 ZINC000217646468 DH For-Sale Unstable CCKBR 53 38 O=C(N/C=C/c1ccccc1)NCCc1c[nH]c2ccccc12 ZINC000217646468 DH For-Sale Unstable ALOX15 23 41 O=C(N/C=C/c1ccccc1)NCCc1c[nH]c2ccccc12 ZINC000217646468 DH For-Sale Unstable MMP9 24 41 O=C(N/C=C/c1ccccc1)NCCc1c[nH]c2ccccc12 ZINC000217646468 DH For-Sale Unstable HDAC9 26 44 O=C(N/C=C/c1ccccc1)NCCc1c[nH]c2ccccc12 ZINC000217646468 DH For-Sale Unstable MC1R 42 42 O=C(N/C=C/c1ccccc1)NCCc1c[nH]c2ccccc12 ZINC000217646468 DH For-Sale Unstable HDAC7 31 44 O=C(N/C=C/c1ccccc1)NCCc1c[nH]c2ccccc12 ZINC000217646468 DH For-Sale Unstable SSSIM 27 40 CS(=O)(=O)CCNC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217646491 CC For-Sale Unstable HDAC8 17 43 c1ccc2cc([C@@H]3CC[C@H]3c3ccc4ccccc4c3)ccc2c1 ZINC000217646543 DK For-Sale Unstable SLC6A3 22 42 c1ccc2cc([C@@H]3CC[C@H]3c3ccc4ccccc4c3)ccc2c1 ZINC000217646543 DK For-Sale Unstable ERBB2 17 40 c1ccc2cc([C@@H]3CC[C@H]3c3ccc4ccccc4c3)ccc2c1 ZINC000217646543 DK For-Sale Unstable TRYP_PIG 19 43 CC(C)OCCCNS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217646561 FE In-Stock Unstable CASP3 15 40 CCCCSCC(=O)NC[C@@](C)(O)CSC ZINC000217646574 CD On-Demand Unstable CES1 23 43 CCCCSCC(=O)NC[C@@](C)(O)CSC ZINC000217646574 CD On-Demand Unstable EST1_PIG 49 43 CCCCSCC(=O)NC[C@@](C)(O)CSC ZINC000217646574 CD On-Demand Unstable Q9GPG0_MANSE 0 40 CCCCSCC(=O)NC[C@@](C)(O)CSC ZINC000217646574 CD On-Demand Unstable EST5_RAT 0 40 CC[C@@H](N[C@@H]1CCC[C@@H](O)C1)c1cccc([N+](=O)[O-])c1 ZINC000217646650 CF For-Sale Unstable CACNA1D 49 33 CCCCSCC(=O)NC[C@](C)(O)CSC ZINC000217646665 CD On-Demand Unstable CES1 23 43 CCCCSCC(=O)NC[C@](C)(O)CSC ZINC000217646665 CD On-Demand Unstable EST1_PIG 49 43 CCCCSCC(=O)NC[C@](C)(O)CSC ZINC000217646665 CD On-Demand Unstable Q9GPG0_MANSE 0 40 CCCCSCC(=O)NC[C@](C)(O)CSC ZINC000217646665 CD On-Demand Unstable EST5_RAT 0 40 COc1ccc(C(=O)NCCC(C)C)cc1/C=C\C(=O)O ZINC000217646739 CF For-Sale Unstable DRD4 40 30 CC(C)OCCCNS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1 ZINC000217646787 GD In-Stock Unstable SLC6A9 20 44 CSC[C@@](C)(O)CNC(=O)COc1cccc([N+](=O)[O-])c1 ZINC000217646788 DD On-Demand Unstable CACNA1D 67 33 CSC[C@@](C)(O)CNC(=O)COc1cccc([N+](=O)[O-])c1 ZINC000217646788 DD On-Demand Unstable ACR 18 42 CSC[C@@](C)(O)CNC(=O)COc1cccc([N+](=O)[O-])c1 ZINC000217646788 DD On-Demand Unstable PDS 30 46 CCOC(=O)[C@@H]1C[C@@H]1c1ccc(C)nc1 ZINC000217646793 BE In-Stock Unstable SLC6A1 57 36 CCOC(=O)[C@@H]1C[C@@H]1c1ccc(C)nc1 ZINC000217646793 BE In-Stock Unstable SLC6A3 33 40 C=C(CC)COc1c(C)cc(/C=C\C(=O)O)cc1C ZINC000217646802 CH For-Sale Unstable AKR1C3 20 40 Cc1ccc(NC(=O)N/C=C/c2ccccc2)c(O)c1 ZINC000217646822 CG For-Sale Unstable LPL 41 32 CC[C@@H](N[C@H]1CCC[C@@H](O)C1)c1cccc([N+](=O)[O-])c1 ZINC000217646825 CF For-Sale Unstable CACNA1D 49 33 CCOC(=O)[C@H]1C[C@@H]1c1ccc(C)nc1 ZINC000217646873 BE In-Stock Unstable SLC6A1 57 36 CCOC(=O)[C@H]1C[C@@H]1c1ccc(C)nc1 ZINC000217646873 BE In-Stock Unstable SLC6A3 33 40 CCOCCCNc1ccc(S(=O)(=O)NCCCOC(C)C)cc1C(=O)O ZINC000217646876 HE In-Stock Unstable CASP3 15 42 CCOCCCNc1ccc(S(=O)(=O)NCCCOC(C)C)cc1C(=O)O ZINC000217646876 HE In-Stock Unstable BDKRB1 16 41 CSC[C@](C)(O)CNC(=O)COc1cccc([N+](=O)[O-])c1 ZINC000217646880 DD On-Demand Unstable CACNA1D 67 33 CSC[C@](C)(O)CNC(=O)COc1cccc([N+](=O)[O-])c1 ZINC000217646880 DD On-Demand Unstable ACR 18 42 CSC[C@](C)(O)CNC(=O)COc1cccc([N+](=O)[O-])c1 ZINC000217646880 DD On-Demand Unstable PDS 30 46 C=C(CC)COc1ccc(/C=C\C(=O)O)cc1 ZINC000217646919 BG For-Sale Unstable PLA2G4B 63 34 C=C(CC)COc1ccc(/C=C\C(=O)O)cc1 ZINC000217646919 BG For-Sale Unstable AKR1C3 32 40 O=C(N/C=C/c1ccccc1)Nc1ccc(Cl)cc1C(F)(F)F ZINC000217646927 EK For-Sale Anodyne CMA1 0 41 CSc1ccc(Cl)cc1[C@@H](C)CC(=O)O ZINC000217646959 BH For-Sale Unstable OXER1 40 34 CCOC(=O)[C@@H]1C[C@H]1c1ccc(C)nc1 ZINC000217646962 BE In-Stock Unstable SLC6A1 57 36 CCOC(=O)[C@@H]1C[C@H]1c1ccc(C)nc1 ZINC000217646962 BE In-Stock Unstable SLC6A3 33 40 CC(C)OCCCNc1ccc(S(=O)(=O)NCCCOC(C)C)cc1C(=O)O ZINC000217646979 HF In-Stock Unstable CASP3 16 43 CC(C)OCCCNc1ccc(S(=O)(=O)NCCCOC(C)C)cc1C(=O)O ZINC000217646979 HF In-Stock Unstable BDKRB1 0 43 COCc1cc(=O)c(O)c([C@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccc3c(c2)OCO3)o1 ZINC000217646988 KH In-Stock Unstable PDE11A 56 34 COCc1cc(=O)c(O)c([C@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccc3c(c2)OCO3)o1 ZINC000217646988 KH In-Stock Unstable RORC 34 40 O[C@@H]1CCC[C@H](N[C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217647008 CE For-Sale Unstable DRD2 17 52 O[C@@H]1CCC[C@H](N[C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217647008 CE For-Sale Unstable DRD4 47 52 O[C@@H]1CCC[C@H](N[C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217647008 CE For-Sale Unstable ACHE 34 42 O[C@@H]1CCC[C@H](N[C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217647008 CE For-Sale Unstable CHRM3 16 41 O[C@@H]1CCC[C@H](N[C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217647008 CE For-Sale Unstable LTA4H 25 40 O[C@@H]1CCC[C@H](N[C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217647008 CE For-Sale Unstable SIGMAR1 58 48 O[C@@H]1CCC[C@H](N[C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217647008 CE For-Sale Unstable CCR3 22 42 O[C@@H]1CCC[C@H](N[C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217647008 CE For-Sale Unstable SLC18A3 30 43 O[C@@H]1CCC[C@H](N[C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217647008 CE For-Sale Unstable MCHR1 18 46 O[C@@H]1CCC[C@H](N[C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217647008 CE For-Sale Unstable BIRC2 30 43 CSc1ccc(Cl)cc1[C@H](C)CC(=O)O ZINC000217647041 BH For-Sale Unstable OXER1 40 34 C1CCN2CC[C@@H](N[C@H]3C[C@@H]4CC[C@@H]3C4)[C@@H]2C1 ZINC000217647053 BE For-Sale Unstable CYP2D26 0 42 C=C(CC)COc1ccccc1/C=C\C(=O)O ZINC000217647057 BG For-Sale Unstable PTGER2 58 57 C=C(CC)COc1ccccc1/C=C\C(=O)O ZINC000217647057 BG For-Sale Unstable PTGER4 30 57 C=C(CC)COc1ccccc1/C=C\C(=O)O ZINC000217647057 BG For-Sale Unstable PTGER3 24 45 C=C(CC)COc1ccccc1/C=C\C(=O)O ZINC000217647057 BG For-Sale Unstable AKR1C3 15 41 CCOC(=O)[C@H]1C[C@H]1c1ccc(C)nc1 ZINC000217647061 BE In-Stock Unstable SLC6A1 57 36 CCOC(=O)[C@H]1C[C@H]1c1ccc(C)nc1 ZINC000217647061 BE In-Stock Unstable SLC6A3 33 40 COCc1cc(=O)c(O)c([C@@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccc3c(c2)OCO3)o1 ZINC000217647077 KH In-Stock Unstable PDE11A 56 34 COCc1cc(=O)c(O)c([C@@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccc3c(c2)OCO3)o1 ZINC000217647077 KH In-Stock Unstable RORC 34 40 O[C@H]1CCC[C@H](N[C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217647085 CE For-Sale Unstable DRD2 17 52 O[C@H]1CCC[C@H](N[C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217647085 CE For-Sale Unstable DRD4 47 52 O[C@H]1CCC[C@H](N[C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217647085 CE For-Sale Unstable ACHE 34 42 O[C@H]1CCC[C@H](N[C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217647085 CE For-Sale Unstable CHRM3 16 41 O[C@H]1CCC[C@H](N[C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217647085 CE For-Sale Unstable LTA4H 25 40 O[C@H]1CCC[C@H](N[C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217647085 CE For-Sale Unstable SIGMAR1 58 48 O[C@H]1CCC[C@H](N[C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217647085 CE For-Sale Unstable CCR3 22 42 O[C@H]1CCC[C@H](N[C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217647085 CE For-Sale Unstable SLC18A3 30 43 O[C@H]1CCC[C@H](N[C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217647085 CE For-Sale Unstable MCHR1 18 46 O[C@H]1CCC[C@H](N[C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217647085 CE For-Sale Unstable BIRC2 30 43 CCCCCNc1ccc(S(=O)(=O)NCCCOC(C)C)cc1C(=O)O ZINC000217647098 GG In-Stock Unstable CASP3 15 44 C1CCN2CC[C@@H](N[C@H]3C[C@@H]4CC[C@H]3C4)[C@@H]2C1 ZINC000217647149 BE For-Sale Unstable CYP2D26 0 42 O[C@@H]1CCC[C@@H](N[C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217647161 CE For-Sale Unstable DRD2 17 52 O[C@@H]1CCC[C@@H](N[C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217647161 CE For-Sale Unstable DRD4 47 52 O[C@@H]1CCC[C@@H](N[C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217647161 CE For-Sale Unstable ACHE 34 42 O[C@@H]1CCC[C@@H](N[C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217647161 CE For-Sale Unstable CHRM3 16 41 O[C@@H]1CCC[C@@H](N[C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217647161 CE For-Sale Unstable LTA4H 25 40 O[C@@H]1CCC[C@@H](N[C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217647161 CE For-Sale Unstable SIGMAR1 58 48 O[C@@H]1CCC[C@@H](N[C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217647161 CE For-Sale Unstable CCR3 22 42 O[C@@H]1CCC[C@@H](N[C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217647161 CE For-Sale Unstable SLC18A3 30 43 O[C@@H]1CCC[C@@H](N[C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217647161 CE For-Sale Unstable MCHR1 18 46 O[C@@H]1CCC[C@@H](N[C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000217647161 CE For-Sale Unstable BIRC2 30 43 Cc1ccc(F)cc1NC(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217647174 DH For-Sale Unstable MAPK11 33 48 NC/C=C\CSc1nc2ccccc2s1 ZINC000217647184 BF For-Sale Unstable HMOX2 17 42 COC(=O)[C@H](C)NC(=O)CCn1cc(C(C)=O)c2ccccc21 ZINC000217647200 DD In-Stock Unstable CNR1 17 44 COC(=O)[C@H](C)NC(=O)CCn1cc(C(C)=O)c2ccccc21 ZINC000217647200 DD In-Stock Unstable CNR2 26 51 O=C(NCCn1ccnc1)c1cc(=O)[nH]c2ccc(F)cc12 ZINC000217647203 DD In-Stock Unstable TBXAS1 43 43 O=C(NCCn1ccnc1)c1cc(=O)[nH]c2ccc(F)cc12 ZINC000217647203 DD In-Stock Unstable PLD2 49 35 O=C(NCCn1ccnc1)c1cc(=O)[nH]c2ccc(F)cc12 ZINC000217647203 DD In-Stock Unstable POLR1A 19 46 CC(C)CCNc1ccc(S(=O)(=O)NCCCOC(C)C)cc1C(=O)O ZINC000217647215 GF In-Stock Unstable CASP3 16 44 C1CCN2CC[C@@H](N[C@H]3C[C@H]4CC[C@@H]3C4)[C@@H]2C1 ZINC000217647230 BE For-Sale Unstable CYP2D26 0 42 CCCCCCC[C@@H](C)N[C@@H]1CCC[C@@H](O)C1 ZINC000217647238 BH For-Sale Unstable ADH1B 0 40 CCCCCCC[C@@H](C)N[C@@H]1CCC[C@@H](O)C1 ZINC000217647238 BH For-Sale Unstable ADH1C 0 40 O=C(O)/C=C\c1ccc(C(=O)NCCN2CCOCC2)s1 ZINC000217647252 DC For-Sale Unstable DRD4 41 31 O=C(O)/C=C\c1ccc(C(=O)NCCN2CCOCC2)s1 ZINC000217647252 DC For-Sale Unstable HPGDS 23 41 CCOc1ccc2nc(SC/C=C\CN)[nH]c2c1 ZINC000217647287 CF For-Sale Unstable CYP2C8 31 45 CCOc1ccc2nc(SC/C=C\CN)[nH]c2c1 ZINC000217647287 CF For-Sale Unstable CYP1A2 15 53 CCOc1ccc2nc(SC/C=C\CN)[nH]c2c1 ZINC000217647287 CF For-Sale Unstable CYP2C19 42 52 O=C(N/C=C/c1ccccc1)Nc1c(Cl)cccc1Cl ZINC000217647294 DJ For-Sale Anodyne CXCL8 50 31 C1CCN2CC[C@@H](N[C@H]3C[C@H]4CC[C@H]3C4)[C@@H]2C1 ZINC000217647314 BE For-Sale Unstable CYP2D26 0 42 CCCCCCC[C@H](C)N[C@@H]1CCC[C@@H](O)C1 ZINC000217647316 BH For-Sale Unstable ADH1B 0 40 CCCCCCC[C@H](C)N[C@@H]1CCC[C@@H](O)C1 ZINC000217647316 BH For-Sale Unstable ADH1C 0 40 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NCCCOC(C)C)cc1C(=O)O ZINC000217647328 GG In-Stock Unstable CASP3 15 44 COc1ccc(C(=O)N2CCSCC2)cc1/C=C\C(=O)O ZINC000217647345 DD For-Sale Unstable GPR183 0 42 COc1cc(I)c(Cl)cc1C(=O)NC[C@@](C)(O)CSC ZINC000217647361 IF On-Demand Unstable HTR4 30 42 CCCCCCC[C@@H](C)N[C@H]1CCC[C@@H](O)C1 ZINC000217647387 BH For-Sale Unstable ADH1B 0 40 CCCCCCC[C@@H](C)N[C@H]1CCC[C@@H](O)C1 ZINC000217647387 BH For-Sale Unstable ADH1C 0 40 CCC[C@H](C)Nc1ccc(S(=O)(=O)NCCCOC(C)C)cc1C(=O)O ZINC000217647398 GG In-Stock Unstable CASP3 15 44 Cc1cccc(N2CCN(C(=O)N/C=C/c3ccccc3)CC2)c1C ZINC000217647420 EH For-Sale Unstable HTR2A 15 40 Cc1cccc(N2CCN(C(=O)N/C=C/c3ccccc3)CC2)c1C ZINC000217647420 EH For-Sale Unstable HTR2C 15 40 Cc1cccc(N2CCN(C(=O)N/C=C/c3ccccc3)CC2)c1C ZINC000217647420 EH For-Sale Unstable ABCB1 23 41 C[C@@H]1CCC[C@H](NC(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217647432 CG For-Sale Unstable HDAC8 18 40 COc1cc(I)c(Cl)cc1C(=O)NC[C@](C)(O)CSC ZINC000217647454 IF On-Demand Unstable HTR4 30 42 CCCCCCC[C@H](C)N[C@H]1CCC[C@@H](O)C1 ZINC000217647482 BH For-Sale Unstable ADH1B 0 40 CCCCCCC[C@H](C)N[C@H]1CCC[C@@H](O)C1 ZINC000217647482 BH For-Sale Unstable ADH1C 0 40 Cc1cc(=O)c(O)c([C@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccc(C(C)C)cc2)o1 ZINC000217647492 JK In-Stock Unstable SSTR4 46 33 O=C(O)[C@@H]1CC[C@@H]1N1CCc2ccccc21 ZINC000217647493 BD For-Sale Unstable ACE 22 45 C[C@H]1CCC[C@H](NC(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217647498 CG For-Sale Unstable HDAC8 18 40 O=C(N/C=C/c1ccccc1)N1CCN(c2ccccc2)CC1 ZINC000217647515 DG For-Sale Unstable ERBB2 0 45 O=C(N/C=C/c1ccccc1)N1CCN(c2ccccc2)CC1 ZINC000217647515 DG For-Sale Unstable MMP2 0 45 O=C(N/C=C/c1ccccc1)N1CCN(c2ccccc2)CC1 ZINC000217647515 DG For-Sale Unstable FAAH 0 43 O=C(N/C=C/c1ccccc1)N1CCN(c2ccccc2)CC1 ZINC000217647515 DG For-Sale Unstable ADAM10 38 40 O=C(N/C=C/c1ccccc1)N1CCN(c2ccccc2)CC1 ZINC000217647515 DG For-Sale Unstable AKR1C3 22 48 O=C(N/C=C/c1ccccc1)N1CCN(c2ccccc2)CC1 ZINC000217647515 DG For-Sale Unstable SLC6A7 0 45 O=C(O)[C@@H]1CC[C@H]1N1CCc2ccccc21 ZINC000217647561 BD For-Sale Unstable ACE 22 45 O=C(O)/C=C\c1ccc(C(=O)NCC2CCCC2)cc1 ZINC000217647573 CF For-Sale Unstable GRIN2B 18 45 O=C(O)/C=C\c1ccc(C(=O)NCC2CCCC2)cc1 ZINC000217647573 CF For-Sale Unstable CACNA1I 64 37 Cc1cc(=O)c(O)c([C@@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccc(C(C)C)cc2)o1 ZINC000217647576 JK In-Stock Unstable SSTR4 46 33 Cc1cc(=O)c(O)c([C@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccc3c(c2)OCO3)o1 ZINC000217647705 JH In-Stock Unstable PDE11A 51 33 Cc1cc(=O)c(O)c([C@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccc3c(c2)OCO3)o1 ZINC000217647705 JH In-Stock Unstable RORC 32 40 CCCCCNS(=O)(=O)c1ccc(NCCC)c(C(=O)O)c1 ZINC000217647717 EF In-Stock Unstable CASP3 22 48 CC(C)n1nc(-c2cccnc2)cc1N ZINC000217647728 BE In-Stock Unstable PRKDC 0 50 CC(C)n1nc(-c2cccnc2)cc1N ZINC000217647728 BE In-Stock Unstable CYP2E1 46 40 CC(C)n1nc(-c2cccnc2)cc1N ZINC000217647728 BE In-Stock Unstable CYP2A6 52 49 Cc1cccc(C)c1NC(=O)N/C=C/c1ccccc1 ZINC000217647731 CI For-Sale Unstable S1PR4 0 41 Cc1cccc(C)c1NC(=O)N/C=C/c1ccccc1 ZINC000217647731 CI For-Sale Unstable ACAT 0 44 COc1ccccc1N1C[C@@H](C(=O)NCCSc2nncn2C)CC1=O ZINC000217647732 GD In-Stock Unstable HTR1A 38 40 COc1ccccc1N1C[C@@H](C(=O)NCCSc2nncn2C)CC1=O ZINC000217647732 GD In-Stock Unstable DRD2 29 43 Cc1cc(=O)c(O)c([C@@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccc3c(c2)OCO3)o1 ZINC000217647785 JH In-Stock Unstable PDE11A 51 33 Cc1cc(=O)c(O)c([C@@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccc3c(c2)OCO3)o1 ZINC000217647785 JH In-Stock Unstable RORC 32 40 O=C(NC[C@@H]1CCCN1c1nc2ccccc2o1)c1ccccc1C(F)(F)F ZINC000217647803 GI In-Stock Unstable HTR3A 26 41 O=C(NC[C@@H]1CCCN1c1nc2ccccc2o1)c1ccccc1C(F)(F)F ZINC000217647803 GI In-Stock Unstable HCRTR1 37 40 O=C(NC[C@@H]1CCCN1c1nc2ccccc2o1)c1ccccc1C(F)(F)F ZINC000217647803 GI In-Stock Unstable HCRTR2 17 40 O=C(NC[C@@H]1CCCN1c1nc2ccccc2o1)c1ccccc1C(F)(F)F ZINC000217647803 GI In-Stock Unstable RBP4 45 32 O=C(O)/C=C\c1ccc(C(=O)NCC(=O)NC2CC2)cc1 ZINC000217647813 CC For-Sale Unstable CCR2 50 42 COc1ccccc1N1C[C@H](C(=O)NCCSc2nncn2C)CC1=O ZINC000217647819 GD In-Stock Unstable HTR1A 49 44 COc1ccccc1N1C[C@H](C(=O)NCCSc2nncn2C)CC1=O ZINC000217647819 GD In-Stock Unstable DRD2 32 43 COc1ccccc1N1C[C@H](C(=O)NCCSc2nncn2C)CC1=O ZINC000217647819 GD In-Stock Unstable DRD3 45 40 CCCCCNS(=O)(=O)c1ccc(NC(C)C)c(C(=O)O)c1 ZINC000217647837 EF In-Stock Unstable CASP3 22 46 COc1ccc([N+](=O)[O-])cc1NC(=O)N/C=C/c1ccccc1 ZINC000217647848 DG For-Sale Unstable CACNA1D 51 38 COc1ccc([N+](=O)[O-])cc1NC(=O)N/C=C/c1ccccc1 ZINC000217647848 DG For-Sale Unstable KCNMA1 24 57 COc1ccc([N+](=O)[O-])cc1NC(=O)N/C=C/c1ccccc1 ZINC000217647848 DG For-Sale Unstable TLR4 16 42 COc1ccc([N+](=O)[O-])cc1NC(=O)N/C=C/c1ccccc1 ZINC000217647848 DG For-Sale Unstable TRPM8 0 53 O=C(NC[C@H]1CCCN1c1nc2ccccc2o1)c1ccccc1C(F)(F)F ZINC000217647882 GI In-Stock Unstable HTR3A 26 41 O=C(NC[C@H]1CCCN1c1nc2ccccc2o1)c1ccccc1C(F)(F)F ZINC000217647882 GI In-Stock Unstable HCRTR1 37 40 O=C(NC[C@H]1CCCN1c1nc2ccccc2o1)c1ccccc1C(F)(F)F ZINC000217647882 GI In-Stock Unstable HCRTR2 17 40 O=C(NC[C@H]1CCCN1c1nc2ccccc2o1)c1ccccc1C(F)(F)F ZINC000217647882 GI In-Stock Unstable RBP4 45 32 CC(C)[C@@H](NC(=O)[C@@H]1CC[C@@H](CNC(=O)Cn2c(=O)[nH]c3ccccc3c2=O)CC1)C(=O)O ZINC000217647896 JC In-Stock Unstable AVPR1B 33 42 CC(C)[C@@H](NC(=O)[C@@H]1CC[C@@H](CNC(=O)Cn2c(=O)[nH]c3ccccc3c2=O)CC1)C(=O)O ZINC000217647896 JC In-Stock Unstable ELANE 50 43 O=C(NCc1ccc(F)cc1)C(F)F ZINC000217647903 BD On-Demand Unstable SLC6A11 0 42 O=C(NCc1ccc(F)cc1)C(F)F ZINC000217647903 BD On-Demand Unstable SLC6A12 0 42 O=C(NCc1ccc(F)cc1)C(F)F ZINC000217647903 BD On-Demand Unstable AMP1_PLAFQ 25 56 O=C(NCc1ccc(F)cc1)C(F)F ZINC000217647903 BD On-Demand Unstable LEF 40 37 O=C(NCc1ccc(F)cc1)C(F)F ZINC000217647903 BD On-Demand Unstable Q76353_9HIV1 0 41 CCCCCNS(=O)(=O)c1ccc(NCCCC)c(C(=O)O)c1 ZINC000217647924 EG In-Stock Unstable CASP3 22 48 CCCCCNS(=O)(=O)c1ccc(NCCCC)c(C(=O)O)c1 ZINC000217647924 EG In-Stock Unstable BDKRB1 0 43 Cc1noc2nc(C(C)C)cc(C(=O)NC34CC5CC(CC(C5)C3)C4)c12 ZINC000217647945 FI On-Demand Unstable CNR2 28 50 Cc1noc2nc(C(C)C)cc(C(=O)NC34CC5CC(CC(C5)C3)C4)c12 ZINC000217647945 FI On-Demand Unstable EPHX2 31 46 COc1cc(Cl)c(C)cc1NC(=O)N/C=C/c1ccccc1 ZINC000217647963 DI For-Sale Unstable PYGL 16 44 Cc1noc(-c2ccsc2NC(=O)c2cccc(Cl)c2)n1 ZINC000217647992 DI In-Stock Unstable KCNK3 64 45 Cc1noc(-c2ccsc2NC(=O)c2cccc(Cl)c2)n1 ZINC000217647992 DI In-Stock Unstable KCNK9 38 45 CCCCCNS(=O)(=O)c1ccc(NCC(C)C)c(C(=O)O)c1 ZINC000217648040 EF In-Stock Unstable CASP3 17 47 COc1cccc([C@@H](CNC(=O)N2CCN(c3ncccc3C#N)CC2)N2CCCC2)c1 ZINC000217648083 IF On-Demand Unstable DRD4 46 35 COc1cccc([C@@H](CNC(=O)N2CCN(c3ncccc3C#N)CC2)N2CCCC2)c1 ZINC000217648083 IF On-Demand Unstable P2RY12 41 44 COc1cccc([C@@H](CNC(=O)N2CCN(c3ncccc3C#N)CC2)N2CCCC2)c1 ZINC000217648083 IF On-Demand Unstable PDGFRB 42 37 COc1cccc([C@@H](CNC(=O)N2CCN(c3ncccc3C#N)CC2)N2CCCC2)c1 ZINC000217648083 IF On-Demand Unstable PTAFR 41 40 COc1ccc(C(=O)NCCC(N)=O)cc1/C=C\C(=O)O ZINC000217648091 CC For-Sale Unstable DRD4 40 30 COC(=O)c1nc(NC(=O)[C@H](C)Nc2ccc3c(cc2=O)[C@@H](NC(C)=O)CCc2cc(OC)c(OC)c(OC)c2-3)sc1C ZINC000217648099 KH In-Stock Unstable TUBA1A 17 62 COC(=O)c1nc(NC(=O)[C@H](C)Nc2ccc3c(cc2=O)[C@@H](NC(C)=O)CCc2cc(OC)c(OC)c(OC)c2-3)sc1C ZINC000217648099 KH In-Stock Unstable TPPP 0 61 Cc1ccc(S(=O)(=O)NCCC(C)C)cc1CO ZINC000217648129 CD For-Sale Unstable LEF 40 34 CC[C@@H](C)c1ccc(NC(=O)C(F)F)cc1 ZINC000217648146 BG For-Sale Unstable SCN2A 33 67 CC[C@@H](C)c1ccc(NC(=O)C(F)F)cc1 ZINC000217648146 BG For-Sale Unstable PSBA 0 40 COc1cccc([C@H](CNC(=O)N2CCN(c3ncccc3C#N)CC2)N2CCCC2)c1 ZINC000217648154 IF On-Demand Unstable DRD4 46 35 COc1cccc([C@H](CNC(=O)N2CCN(c3ncccc3C#N)CC2)N2CCCC2)c1 ZINC000217648154 IF On-Demand Unstable P2RY12 41 44 COc1cccc([C@H](CNC(=O)N2CCN(c3ncccc3C#N)CC2)N2CCCC2)c1 ZINC000217648154 IF On-Demand Unstable PDGFRB 42 37 COc1cccc([C@H](CNC(=O)N2CCN(c3ncccc3C#N)CC2)N2CCCC2)c1 ZINC000217648154 IF On-Demand Unstable PTAFR 41 40 CCCCCNS(=O)(=O)c1ccc(N[C@@H](C)CC)c(C(=O)O)c1 ZINC000217648157 EG In-Stock Unstable CASP3 22 46 O=C(O)[C@@H]1CC[C@@H]1N1CCc2ccccc2C1 ZINC000217648186 BD For-Sale Unstable AGTR2 48 40 O=C(O)[C@@H]1CC[C@@H]1N1CCc2ccccc2C1 ZINC000217648186 BD For-Sale Unstable CHRNA6 0 40 CCN(C(=O)N/C=C/c1ccccc1)c1cccc(C)c1 ZINC000217648191 CI For-Sale Unstable NR1H4 43 38 COC(=O)C[C@H](c1ccc2c(c1)OCCO2)c1c(O)c2ccccc2oc1=O ZINC000217648215 GF In-Stock Unstable NQO1 56 48 CCCCCNS(=O)(=O)c1ccc(N[C@H](C)CC)c(C(=O)O)c1 ZINC000217648225 EG In-Stock Unstable CASP3 22 46 CC[C@H](C)c1ccc(NC(=O)C(F)F)cc1 ZINC000217648237 BG For-Sale Unstable SCN2A 33 67 CC[C@H](C)c1ccc(NC(=O)C(F)F)cc1 ZINC000217648237 BG For-Sale Unstable PSBA 0 40 NCCc1cc(F)c(O)c(Br)c1O ZINC000217648260 CD For-Sale Unstable TAAR1 17 42 Cc1ccc(Cl)cc1NC(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217648277 DI For-Sale Unstable MAPK11 35 48 O=C(O)[C@@H]1CC[C@H]1N1CCc2ccccc2C1 ZINC000217648279 BD For-Sale Unstable AGTR2 48 40 O=C(O)[C@@H]1CC[C@H]1N1CCc2ccccc2C1 ZINC000217648279 BD For-Sale Unstable CHRNA6 0 40 COc1cccc([C@@H](CNC(=O)NCCn2c(C)nc3ccccc32)N2CCCC2)c1 ZINC000217648281 HG On-Demand Unstable DRD4 45 35 COc1cccc([C@@H](CNC(=O)NCCn2c(C)nc3ccccc32)N2CCCC2)c1 ZINC000217648281 HG On-Demand Unstable PDE6D 25 40 COC(=O)C[C@@H](c1ccc2c(c1)OCCO2)c1c(O)c2ccccc2oc1=O ZINC000217648293 GF In-Stock Unstable NQO1 53 37 CC(C)CCNC(=O)N/C=C/c1ccccc1 ZINC000217648297 BG For-Sale Unstable MME 27 44 CC(C)CCNC(=O)N/C=C/c1ccccc1 ZINC000217648297 BG For-Sale Unstable ANPEP 40 38 CC(C)CCNC(=O)N/C=C/c1ccccc1 ZINC000217648297 BG For-Sale Unstable DNPEP 0 45 Cc1noc(-c2ccsc2NC(=O)COc2ccc(Cl)cc2Cl)n1 ZINC000217648331 GI In-Stock Unstable AGPAT2 44 32 Cc1noc(-c2ccsc2NC(=O)COc2ccc(Cl)cc2Cl)n1 ZINC000217648331 GI In-Stock Unstable MCHR2 23 42 Cc1nc(N2CCCn3nc(CO)cc3C2)c2ccccc2n1 ZINC000217648351 DE In-Stock Unstable NPY5R 0 42 CCCCCNS(=O)(=O)c1ccc(NC(C)(C)C)c(C(=O)O)c1 ZINC000217648355 EG In-Stock Unstable CASP3 17 46 Cc1ccc(NC(=O)c2ccc(/C=C\C(=O)O)s2)nc1 ZINC000217648366 CF For-Sale Unstable LUCI_LUCLA 38 41 O=C(O)[C@@H]1CC[C@@H]1N1CCCc2ccccc21 ZINC000217648369 BE For-Sale Unstable ACE 21 40 O=C(O)[C@@H]1CC[C@@H]1N1CCCc2ccccc21 ZINC000217648369 BE For-Sale Unstable AVPR2 22 40 COc1cccc([C@H](CNC(=O)NCCn2c(C)nc3ccccc32)N2CCCC2)c1 ZINC000217648379 HG On-Demand Unstable DRD4 45 35 COc1cccc([C@H](CNC(=O)NCCn2c(C)nc3ccccc32)N2CCCC2)c1 ZINC000217648379 HG On-Demand Unstable PDE6D 25 40 NCCc1cc(Br)c(O)c(F)c1O ZINC000217648388 CD For-Sale Unstable TAAR1 20 41 O=C(C(F)F)N1CCN(c2cccc(C(F)(F)F)c2)CC1 ZINC000217648432 DF On-Demand Unstable CACNA1B 40 34 O=C(C(F)F)N1CCN(c2cccc(C(F)(F)F)c2)CC1 ZINC000217648432 DF On-Demand Unstable SERPINE1 28 44 O=C(C(F)F)N1CCN(c2cccc(C(F)(F)F)c2)CC1 ZINC000217648432 DF On-Demand Unstable SLC6A9 0 48 O=C(C(F)F)N1CCN(c2cccc(C(F)(F)F)c2)CC1 ZINC000217648432 DF On-Demand Unstable AKR1C3 0 47 NC/C=C\COc1ccccc1F ZINC000217648435 AD For-Sale Unstable TAAR1 18 44 Cc1ccc(NC(=O)c2ccc(/C=C\C(=O)O)cc2)nc1 ZINC000217648437 CF For-Sale Unstable F10 29 46 Cc1ccc(NC(=O)c2ccc(/C=C\C(=O)O)cc2)nc1 ZINC000217648437 CF For-Sale Unstable GCK 34 40 Cc1ccc(NC(=O)c2ccc(/C=C\C(=O)O)cc2)nc1 ZINC000217648437 CF For-Sale Unstable MAP3K5 40 36 Cc1ccc(NC(=O)c2ccc(/C=C\C(=O)O)cc2)nc1 ZINC000217648437 CF For-Sale Unstable LUCI_LUCLA 47 45 O=C(O)[C@@H]1CC[C@H]1N1CCCc2ccccc21 ZINC000217648461 BE For-Sale Unstable ACE 21 40 O=C(O)[C@@H]1CC[C@H]1N1CCCc2ccccc21 ZINC000217648461 BE For-Sale Unstable AVPR2 22 40 C=CCNc1ccc(S(=O)(=O)NCCCCC)cc1C(=O)O ZINC000217648481 EE In-Stock Unstable CASP3 0 46 O=C(O)/C=C\c1ccc(NC(=O)c2ccon2)cc1 ZINC000217648520 CE For-Sale Anodyne SMO 15 43 CCN(CC)S(=O)(=O)Nc1ccc(/C=C\C(=O)O)cc1F ZINC000217648530 DD For-Sale Unstable NFE2L2 0 40 COc1ccc(C(C)(C)C)cc1NC(=O)C(F)F ZINC000217648561 CG On-Demand Unstable TRPV1 22 41 COc1ccc(C(C)(C)C)cc1NC(=O)C(F)F ZINC000217648561 CG On-Demand Unstable Q8MMZ8_EIMTE 24 40 CCCCCNS(=O)(=O)c1ccc(NC2CC2)c(C(=O)O)c1 ZINC000217648594 EE In-Stock Unstable TBXA2R 15 44 CCCCCNS(=O)(=O)c1ccc(NC2CC2)c(C(=O)O)c1 ZINC000217648594 EE In-Stock Unstable CASP3 15 43 O=C(N/C=C/c1ccccc1)N1CCN(c2ccccc2F)CC1 ZINC000217648599 EG For-Sale Unstable NPY2R 55 36 O=C(N/C=C/c1ccccc1)N1CCN(c2ccccc2F)CC1 ZINC000217648599 EG For-Sale Unstable FAAH 0 46 O[C@@H]1CCC[C@H](N[C@@H]2CCCN(Cc3ccccc3)C2)C1 ZINC000217648604 CF On-Demand Unstable DRD2 0 42 O[C@@H]1CCC[C@H](N[C@@H]2CCCN(Cc3ccccc3)C2)C1 ZINC000217648604 CF On-Demand Unstable DRD3 24 44 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)N3CCc4ccccc4C3)[C@H]21 ZINC000217648605 JH In-Stock Unstable HTR7 17 47 COC(=O)Cc1cccc(OC)n1 ZINC000217648625 AC For-Sale Unstable ALS 78 36 O[C@H]1CCC[C@H](N[C@@H]2CCCN(Cc3ccccc3)C2)C1 ZINC000217648676 CF For-Sale Unstable DRD2 0 42 O[C@H]1CCC[C@H](N[C@@H]2CCCN(Cc3ccccc3)C2)C1 ZINC000217648676 CF For-Sale Unstable DRD4 36 46 O[C@H]1CCC[C@H](N[C@@H]2CCCN(Cc3ccccc3)C2)C1 ZINC000217648676 CF For-Sale Unstable DRD3 24 44 O[C@H]1CCC[C@H](N[C@@H]2CCCN(Cc3ccccc3)C2)C1 ZINC000217648676 CF For-Sale Unstable SIGMAR1 53 45 O[C@H]1CCC[C@H](N[C@@H]2CCCN(Cc3ccccc3)C2)C1 ZINC000217648676 CF For-Sale Unstable BIRC2 28 45 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)N3CCc4ccccc4C3)[C@@H]21 ZINC000217648682 JH In-Stock Unstable HTR7 17 47 CCCCCNS(=O)(=O)c1ccc(NC2CCCC2)c(C(=O)O)c1 ZINC000217648716 FG In-Stock Unstable ADRB2 0 41 CCCCCNS(=O)(=O)c1ccc(NC2CCCC2)c(C(=O)O)c1 ZINC000217648716 FG In-Stock Unstable CASP3 15 42 CNC(=O)CNC(=O)NC[C@H](c1ccc(Cl)cc1Cl)c1c[nH]c2ccccc12 ZINC000217648720 HH On-Demand Unstable GRPR 49 34 O[C@@H]1CCC[C@@H](N[C@@H]2CCCN(Cc3ccccc3)C2)C1 ZINC000217648767 CF On-Demand Unstable DRD2 0 42 O[C@@H]1CCC[C@@H](N[C@@H]2CCCN(Cc3ccccc3)C2)C1 ZINC000217648767 CF On-Demand Unstable DRD3 24 44 CNC(=O)CNC(=O)NC[C@@H](c1ccc(Cl)cc1Cl)c1c[nH]c2ccccc12 ZINC000217648801 HH On-Demand Unstable GRPR 49 34 CCCCCNS(=O)(=O)c1ccc(NC2CCCCC2)c(C(=O)O)c1 ZINC000217648824 FH In-Stock Unstable ADRB1 0 40 CCCCCNS(=O)(=O)c1ccc(NC2CCCCC2)c(C(=O)O)c1 ZINC000217648824 FH In-Stock Unstable CASP3 0 47 NC/C=C\COc1cccc(C(F)(F)F)c1 ZINC000217648908 BF For-Sale Unstable PDS 44 42 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable HTR1A 60 47 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable DRD2 64 47 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable FKBP1A 30 43 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable DRD1 24 45 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable DRD4 37 42 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable ACHE 19 50 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable HRH2 42 45 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable ADRA1D 49 41 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable HTR2A 60 53 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable HTR2C 48 47 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable SLC6A4 27 42 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable ADRA1A 63 44 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable HRH1 19 43 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable ADRA1B 48 41 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable OPRM1 18 47 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable DRD3 81 47 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable OPRD1 15 45 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable SLC6A3 20 40 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable KCNH2 16 43 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable HTR4 28 44 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable LTA4H 26 49 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable HTR7 52 42 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable HRH3 67 54 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable SIGMAR1 83 59 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable BCHE 25 45 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable CCR3 26 47 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable SCN2A 23 50 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable CHRNA7 34 52 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable PYGL 15 43 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable EBP 18 59 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable FAAH 18 49 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable HNMT 94 39 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable ABCB1 26 47 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable DPP7 35 43 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable TPSAB1 16 41 O=C(NCCCN1CCCCC1)N1CCN(CCc2ccccc2)CC1 ZINC000217648923 FE On-Demand Unstable BIRC2 22 40 O=C(c1ccccc1N1CCCC1)N1CCC(n2cnnc2)CC1 ZINC000217648925 EE In-Stock Unstable KCNQ2 47 34 O=C(c1ccccc1N1CCCC1)N1CCC(n2cnnc2)CC1 ZINC000217648925 EE In-Stock Unstable L3MBTL1 0 55 O=C(c1ccccc1N1CCCC1)N1CCC(n2cnnc2)CC1 ZINC000217648925 EE In-Stock Unstable L3MBTL3 78 55 O=C(c1ccccc1N1CCCC1)N1CCC(n2cnnc2)CC1 ZINC000217648925 EE In-Stock Unstable L3MBTL4 0 41 O=C(c1ccccc1N1CCCC1)N1CCC(n2cnnc2)CC1 ZINC000217648925 EE In-Stock Unstable MBTD1 0 48 O=C(c1ccccc1N1CCCC1)N1CCC(n2cnnc2)CC1 ZINC000217648925 EE In-Stock Unstable TP53BP1 0 55 O[C@@H]1CCC[C@H](N[C@@H]2CCCc3ccccc32)C1 ZINC000217648954 BF On-Demand Unstable KCNN3 18 40 O[C@@H]1CCC[C@H](N[C@@H]2CCCc3ccccc32)C1 ZINC000217648954 BF On-Demand Unstable TSPAN17 0 40 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCC1CCOCC1 ZINC000217648978 GD In-Stock Unstable NMBR 36 40 Cc1noc(-c2ccsc2NC(=O)Cc2ccccc2)n1 ZINC000217648993 CG In-Stock Unstable MAPK10 26 43 Cc1noc(-c2ccsc2NC(=O)Cc2ccccc2)n1 ZINC000217648993 CG In-Stock Unstable MAPK8 26 41 O=C(NCCCN1CCCCC1)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000217649031 HF On-Demand Unstable HTR1A 67 41 O=C(NCCCN1CCCCC1)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000217649031 HF On-Demand Unstable DRD2 69 42 O=C(NCCCN1CCCCC1)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000217649031 HF On-Demand Unstable DRD1 33 41 O=C(NCCCN1CCCCC1)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000217649031 HF On-Demand Unstable DRD4 36 41 O=C(NCCCN1CCCCC1)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000217649031 HF On-Demand Unstable ACHE 15 42 O=C(NCCCN1CCCCC1)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000217649031 HF On-Demand Unstable ADRA1D 45 38 O=C(NCCCN1CCCCC1)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000217649031 HF On-Demand Unstable HTR2A 60 41 O=C(NCCCN1CCCCC1)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000217649031 HF On-Demand Unstable HTR2C 46 41 O=C(NCCCN1CCCCC1)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000217649031 HF On-Demand Unstable ADRA1A 55 39 O=C(NCCCN1CCCCC1)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000217649031 HF On-Demand Unstable DRD3 89 42 O=C(NCCCN1CCCCC1)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000217649031 HF On-Demand Unstable HTR4 50 43 O=C(NCCCN1CCCCC1)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000217649031 HF On-Demand Unstable DRD5 27 41 O=C(NCCCN1CCCCC1)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000217649031 HF On-Demand Unstable LTA4H 38 40 O=C(NCCCN1CCCCC1)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000217649031 HF On-Demand Unstable HTR7 63 39 O=C(NCCCN1CCCCC1)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000217649031 HF On-Demand Unstable HRH3 68 45 O=C(NCCCN1CCCCC1)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000217649031 HF On-Demand Unstable BCHE 17 42 O=C(NCCCN1CCCCC1)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000217649031 HF On-Demand Unstable CHRNA7 32 43 O=C(NCCCN1CCCCC1)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000217649031 HF On-Demand Unstable PYGL 18 43 O=C(NCCCN1CCCCC1)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000217649031 HF On-Demand Unstable HNMT 88 36 O=C(NCCCN1CCCCC1)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000217649031 HF On-Demand Unstable PSMB2 49 35 O=C(NCCCN1CCCCC1)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000217649031 HF On-Demand Unstable PSMB1 42 39 O[C@@H]1CCC[C@@H](N[C@@H]2CCCc3ccccc32)C1 ZINC000217649044 BF On-Demand Unstable KCNN3 18 40 O[C@@H]1CCC[C@@H](N[C@@H]2CCCc3ccccc32)C1 ZINC000217649044 BF On-Demand Unstable TSPAN17 0 40 CCCCCNS(=O)(=O)c1ccc(NCCO)c(C(=O)O)c1 ZINC000217649056 ED In-Stock Unstable CASP3 17 46 C=CCOC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C ZINC000217649060 CF On-Demand Unstable CELA1 26 48 C=CCOC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C ZINC000217649060 CF On-Demand Unstable ELANE 45 51 C=CCOC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C ZINC000217649060 CF On-Demand Unstable MME 54 48 C=CCOC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C ZINC000217649060 CF On-Demand Unstable CTSD 18 48 C=CCOC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C ZINC000217649060 CF On-Demand Unstable CTRA_BOVIN 19 55 C=CCOC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C ZINC000217649060 CF On-Demand Unstable HRAS 51 36 C=CCOC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C ZINC000217649060 CF On-Demand Unstable CASP3 33 55 C=CCOC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C ZINC000217649060 CF On-Demand Unstable BMP1 22 48 C=CCOC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C ZINC000217649060 CF On-Demand Unstable KLK3 92 45 C=CCOC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C ZINC000217649060 CF On-Demand Unstable CTSB 86 60 C=CCOC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C ZINC000217649060 CF On-Demand Unstable PAPA1_CARPA 101 55 C=CCOC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C ZINC000217649060 CF On-Demand Unstable CYSP_TRYCR 66 44 C=CCOC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C ZINC000217649060 CF On-Demand Unstable CTSK 55 58 C=CCOC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C ZINC000217649060 CF On-Demand Unstable CTSL 56 58 C=CCOC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C ZINC000217649060 CF On-Demand Unstable PGA 39 54 C=CCOC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C ZINC000217649060 CF On-Demand Unstable CAPNS1 76 42 C=CCOC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C ZINC000217649060 CF On-Demand Unstable HLA-DRB1 63 39 C=CCOC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C ZINC000217649060 CF On-Demand Unstable MMP11 59 34 C=CCOC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C ZINC000217649060 CF On-Demand Unstable CTSS 27 58 C=CCOC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C ZINC000217649060 CF On-Demand Unstable CAPN1 112 60 C=CCOC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C ZINC000217649060 CF On-Demand Unstable CASP1 43 56 C=CCOC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C ZINC000217649060 CF On-Demand Unstable CTRC 16 49 C=CCOC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C ZINC000217649060 CF On-Demand Unstable CAPN2 158 60 C=CCOC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C ZINC000217649060 CF On-Demand Unstable PLAU 15 42 C=CCOC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C ZINC000217649060 CF On-Demand Unstable CASP6 39 55 C=CCOC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C ZINC000217649060 CF On-Demand Unstable CASP9 52 55 C=CCOC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C ZINC000217649060 CF On-Demand Unstable TGM2 39 41 C=CCOC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C ZINC000217649060 CF On-Demand Unstable TPSAB1 41 40 C=CCOC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C ZINC000217649060 CF On-Demand Unstable ADAMTS4 51 35 C=CCOC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C ZINC000217649060 CF On-Demand Unstable NPR 86 44 C=CCOC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C ZINC000217649060 CF On-Demand Unstable CASP10 38 41 C=CCOC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C ZINC000217649060 CF On-Demand Unstable PSMB5 52 44 C=CCOC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C ZINC000217649060 CF On-Demand Unstable Q6PRC7_IXORI 44 39 CCC(=O)C[C@@H]1CCCN1C ZINC000217649087 AD For-Sale Unstable CHRNA10 59 38 CCCCCNS(=O)(=O)c1ccc(NCCCO)c(C(=O)O)c1 ZINC000217649139 ED In-Stock Unstable CASP3 17 48 N#Cc1cccnc1N1CCN(C(=O)NCc2ccc(C(=O)N3CCCCC3)cc2)CC1 ZINC000217649154 IF On-Demand Unstable P2RY12 36 44 N#Cc1cccnc1N1CCN(C(=O)NCc2ccc(C(=O)N3CCCCC3)cc2)CC1 ZINC000217649154 IF On-Demand Unstable NAMPT 32 45 Cc1noc(-c2ccsc2NC(=O)c2ccco2)n1 ZINC000217649199 CF In-Stock Unstable KISS1R 43 33 CN1CCCN(C(=O)c2ccc(=O)[nH]n2)CC1 ZINC000217649226 BB For-Sale Unstable HRH4 28 43 NC/C=C\COc1ccc([N+](=O)[O-])cc1Cl ZINC000217649237 BE For-Sale Unstable SNCA 46 39 NC/C=C\COc1ccc([N+](=O)[O-])cc1Cl ZINC000217649237 BE For-Sale Unstable ENR 0 46 CNCCc1cc(Br)c(F)cc1F ZINC000217649242 CE For-Sale Unstable TAAR1 15 50 CCCCCNS(=O)(=O)c1ccc(NCCOC)c(C(=O)O)c1 ZINC000217649254 ED In-Stock Unstable CASP3 17 44 CCCCCNS(=O)(=O)c1ccc(NCCOC)c(C(=O)O)c1 ZINC000217649254 ED In-Stock Unstable BDKRB1 0 44 COCCCNC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217649295 FD In-Stock Unstable EDNRA 22 40 COCCCNC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217649295 FD In-Stock Unstable MC4R 49 37 COCCCNC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217649295 FD In-Stock Unstable MC5R 32 40 COCCCNC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217649295 FD In-Stock Unstable GRIA1 17 42 COCCCNC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217649295 FD In-Stock Unstable KISS1R 42 31 COc1ccc(CCC(=O)Nc2sccc2-c2nc(C)no2)cc1 ZINC000217649304 EH In-Stock Unstable VIPR1 23 44 CCCCCNS(=O)(=O)c1ccc(NCCCOC)c(C(=O)O)c1 ZINC000217649341 FE In-Stock Unstable CASP3 0 44 Cc1cccc(N2CCN(C(=O)C(F)F)CC2)c1C ZINC000217649372 CE On-Demand Unstable ABCB1 22 41 CNCCc1cc(F)c(Br)cc1F ZINC000217649375 CE For-Sale Unstable TAAR1 15 50 CCCCCNS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217649453 GG In-Stock Unstable HTR7 17 40 CCCCCNS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217649453 GG In-Stock Unstable CASP3 19 44 CCCCCNS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217649453 GG In-Stock Unstable ALOX15 46 39 CC[C@@H]1CCCN1C(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217649461 CF For-Sale Unstable PREP 31 40 CC[C@@H]1CCCN1C(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217649461 CF For-Sale Unstable L3MBTL3 46 35 CNCCc1ccc(F)c(Br)c1F ZINC000217649486 CE For-Sale Unstable TAAR1 15 55 CSC[C@@](C)(O)CNC(=O)CCn1cncn1 ZINC000217649488 CB On-Demand Unstable HIS3 47 33 CC[C@@H](C)c1ccccc1NC(=O)N/C=C/c1ccccc1 ZINC000217649489 CJ For-Sale Unstable AO-ACHE 0 42 CC[C@H]1CCCN1C(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217649545 CF For-Sale Unstable PREP 31 40 CC[C@H]1CCCN1C(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217649545 CF For-Sale Unstable L3MBTL3 46 35 CCCCCNS(=O)(=O)c1ccc(N[C@@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217649556 GI In-Stock Unstable TBXA2R 15 40 CCCCCNS(=O)(=O)c1ccc(N[C@@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217649556 GI In-Stock Unstable CASP3 18 44 CC[C@H](C)c1ccccc1NC(=O)N/C=C/c1ccccc1 ZINC000217649561 CJ For-Sale Unstable AO-ACHE 0 42 CC[C@@H](CCO)NC(=O)c1cccc(N)c1 ZINC000217649571 BD For-Sale Unstable ABAT 20 40 CSC[C@](C)(O)CNC(=O)CCn1cncn1 ZINC000217649574 CB On-Demand Unstable HIS3 47 33 CC(C)Oc1ccc([C@@H]2CC(=O)Oc3cc4c(cc32)OCO4)cc1 ZINC000217649589 EH In-Stock Unstable EDNRB 20 41 CC(C)Oc1ccc([C@@H]2CC(=O)Oc3cc4c(cc32)OCO4)cc1 ZINC000217649589 EH In-Stock Unstable EDNRA 27 41 Cc1noc(-c2ccsc2NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)n1 ZINC000217649612 HC In-Stock Unstable TRPA1 17 55 CC[C@@H]1CCCN1C(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217649635 CF For-Sale Unstable PREP 47 43 CC[C@@H]1CCCN1C(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217649635 CF For-Sale Unstable ACKR3 45 33 C[C@@H](NC(=O)N1CCN(c2ncccc2C#N)CC1)c1ccc(-c2ccccc2)cc1 ZINC000217649647 HI On-Demand Unstable P2RY12 46 51 C[C@@H](NC(=O)N1CCN(c2ncccc2C#N)CC1)c1ccc(-c2ccccc2)cc1 ZINC000217649647 HI On-Demand Unstable PTAFR 48 40 C[C@@H](NC(=O)N1CCN(c2ncccc2C#N)CC1)c1ccc(-c2ccccc2)cc1 ZINC000217649647 HI On-Demand Unstable ACACA 43 36 C[C@@H](NC(=O)N1CCN(c2ncccc2C#N)CC1)c1ccc(-c2ccccc2)cc1 ZINC000217649647 HI On-Demand Unstable PRNP 53 36 C[C@@H](NC(=O)N1CCN(c2ncccc2C#N)CC1)c1ccc(-c2ccccc2)cc1 ZINC000217649647 HI On-Demand Unstable FAAH 0 41 C[C@@H](NC(=O)N1CCN(c2ncccc2C#N)CC1)c1ccc(-c2ccccc2)cc1 ZINC000217649647 HI On-Demand Unstable SLC6A7 0 42 CCCCCNS(=O)(=O)c1ccc(N[C@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217649649 GI In-Stock Unstable TBXA2R 15 40 CCCCCNS(=O)(=O)c1ccc(N[C@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217649649 GI In-Stock Unstable CASP3 18 44 C/C(=N\O)c1cccc(NC(=O)c2cc(C)no2)c1 ZINC000217649655 CE For-Sale Unstable GUAB 0 41 C/C(=N\O)c1cccc(NC(=O)c2cc(C)no2)c1 ZINC000217649655 CE For-Sale Unstable KCNK3 120 42 C/C(=N\O)c1cccc(NC(=O)c2cc(C)no2)c1 ZINC000217649655 CE For-Sale Unstable KCNK9 78 42 CC[C@H](CCO)NC(=O)c1cccc(N)c1 ZINC000217649659 BD For-Sale Unstable ABAT 20 40 CC(C)Oc1ccc([C@H]2CC(=O)Oc3cc4c(cc32)OCO4)cc1 ZINC000217649678 EH In-Stock Unstable EDNRB 20 41 CC(C)Oc1ccc([C@H]2CC(=O)Oc3cc4c(cc32)OCO4)cc1 ZINC000217649678 EH In-Stock Unstable EDNRA 27 41 O=C(N/C=C/c1ccccc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217649686 EH For-Sale Unstable CHRM2 27 44 O=C(N/C=C/c1ccccc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217649686 EH For-Sale Unstable CHRM1 18 50 O=C(N/C=C/c1ccccc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217649686 EH For-Sale Unstable DRD2 28 64 O=C(N/C=C/c1ccccc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217649686 EH For-Sale Unstable DRD4 63 64 O=C(N/C=C/c1ccccc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217649686 EH For-Sale Unstable ACHE 47 49 O=C(N/C=C/c1ccccc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217649686 EH For-Sale Unstable HRH2 16 41 O=C(N/C=C/c1ccccc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217649686 EH For-Sale Unstable DRD3 29 64 O=C(N/C=C/c1ccccc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217649686 EH For-Sale Unstable KCNH2 17 44 O=C(N/C=C/c1ccccc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217649686 EH For-Sale Unstable CHRM3 30 50 O=C(N/C=C/c1ccccc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217649686 EH For-Sale Unstable LTA4H 23 42 O=C(N/C=C/c1ccccc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217649686 EH For-Sale Unstable SIGMAR1 75 70 O=C(N/C=C/c1ccccc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217649686 EH For-Sale Unstable SSTR5 54 38 O=C(N/C=C/c1ccccc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217649686 EH For-Sale Unstable BCHE 0 43 O=C(N/C=C/c1ccccc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217649686 EH For-Sale Unstable CCR3 51 50 O=C(N/C=C/c1ccccc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217649686 EH For-Sale Unstable SLC6A5 31 46 O=C(N/C=C/c1ccccc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217649686 EH For-Sale Unstable EPHX2 30 57 O=C(N/C=C/c1ccccc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217649686 EH For-Sale Unstable MCHR1 57 50 O=C(N/C=C/c1ccccc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217649686 EH For-Sale Unstable CACNA1G 30 46 O=C(N/C=C/c1ccccc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217649686 EH For-Sale Unstable CCR8 15 45 O=C(N/C=C/c1ccccc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217649686 EH For-Sale Unstable NPFFR1 50 35 O=C(N/C=C/c1ccccc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217649686 EH For-Sale Unstable ADIPOR1 0 48 O=C(N/C=C/c1ccccc1)NC1CCN(Cc2ccccc2)CC1 ZINC000217649686 EH For-Sale Unstable ADIPOR2 0 48 Cc1noc(-c2ccsc2NC(=O)CSc2ccc(F)cc2)n1 ZINC000217649723 EH In-Stock Unstable FAS 48 42 C[C@H](NC(=O)N1CCN(c2ncccc2C#N)CC1)c1ccc(-c2ccccc2)cc1 ZINC000217649733 HI On-Demand Unstable P2RY12 46 51 C[C@H](NC(=O)N1CCN(c2ncccc2C#N)CC1)c1ccc(-c2ccccc2)cc1 ZINC000217649733 HI On-Demand Unstable PTAFR 48 40 C[C@H](NC(=O)N1CCN(c2ncccc2C#N)CC1)c1ccc(-c2ccccc2)cc1 ZINC000217649733 HI On-Demand Unstable ACACA 43 36 C[C@H](NC(=O)N1CCN(c2ncccc2C#N)CC1)c1ccc(-c2ccccc2)cc1 ZINC000217649733 HI On-Demand Unstable PRNP 53 36 C[C@H](NC(=O)N1CCN(c2ncccc2C#N)CC1)c1ccc(-c2ccccc2)cc1 ZINC000217649733 HI On-Demand Unstable FAAH 0 41 C[C@H](NC(=O)N1CCN(c2ncccc2C#N)CC1)c1ccc(-c2ccccc2)cc1 ZINC000217649733 HI On-Demand Unstable SLC6A7 0 42 CC[C@H]1CCCN1C(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217649736 CF For-Sale Unstable PREP 47 43 CC[C@H]1CCCN1C(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217649736 CF For-Sale Unstable ACKR3 45 33 C/C(=N\O)c1cccc(NC(=O)c2ccon2)c1 ZINC000217649744 BE For-Sale Unstable GUAB 0 44 C/C(=N\O)c1cccc(NC(=O)c2ccon2)c1 ZINC000217649744 BE For-Sale Unstable IMDH_CRYPV 42 41 C/C(=N\O)c1cccc(NC(=O)c2ccon2)c1 ZINC000217649744 BE For-Sale Unstable PARP15 0 40 C/C(=N\O)c1cccc(NC(=O)c2ccon2)c1 ZINC000217649744 BE For-Sale Unstable KCNK3 121 41 C/C(=N\O)c1cccc(NC(=O)c2ccon2)c1 ZINC000217649744 BE For-Sale Unstable KCNK9 81 40 C/C(=N\O)c1cccc(NC(=O)c2ccon2)c1 ZINC000217649744 BE For-Sale Unstable PARP10 0 40 CCCCCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217649757 GH In-Stock Unstable CA2 16 40 CCCCCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217649757 GH In-Stock Unstable TBXA2R 50 39 CCCCCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217649757 GH In-Stock Unstable HTR7 16 40 CCCCCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217649757 GH In-Stock Unstable CASP3 15 44 CCCCCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217649757 GH In-Stock Unstable ALOX15 53 42 CC[C@@H](CCO)NC(=O)c1cc(N)n[nH]1 ZINC000217649776 BB For-Sale Unstable ALPL 58 38 Cn1nccc1[C@@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc3c21 ZINC000217649786 HG In-Stock Unstable AKR1B1 0 43 Cn1nccc1[C@@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc3c21 ZINC000217649786 HG In-Stock Unstable CYP1B1 25 40 Cn1nccc1[C@@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc3c21 ZINC000217649786 HG In-Stock Unstable CYP1A1 23 40 C[C@@H](C(=O)NC1CC1)N1CCN(C(=O)N[C@H](C)c2ccc(-c3ccccc3)cc2)CC1 ZINC000217649840 HG On-Demand Unstable ACACA 47 40 C[C@@H](C(=O)NC1CC1)N1CCN(C(=O)N[C@H](C)c2ccc(-c3ccccc3)cc2)CC1 ZINC000217649840 HG On-Demand Unstable PRCP 22 41 C[C@@H](C(=O)NC1CC1)N1CCN(C(=O)N[C@H](C)c2ccc(-c3ccccc3)cc2)CC1 ZINC000217649840 HG On-Demand Unstable ACACB 18 40 C[C@@H](C(=O)NC1CC1)N1CCN(C(=O)N[C@H](C)c2ccc(-c3ccccc3)cc2)CC1 ZINC000217649840 HG On-Demand Unstable BIRC3 42 34 C[C@@H](C(=O)NC1CC1)N1CCN(C(=O)N[C@H](C)c2ccc(-c3ccccc3)cc2)CC1 ZINC000217649840 HG On-Demand Unstable BIRC2 41 34 C[C@@H](C(=O)NC1CC1)N1CCN(C(=O)N[C@H](C)c2ccc(-c3ccccc3)cc2)CC1 ZINC000217649840 HG On-Demand Unstable BIRC8 47 33 NCCCc1cc(Br)c(F)cc1F ZINC000217649851 CF For-Sale Unstable MPO 20 41 CC[C@H](CCO)NC(=O)c1cc(N)n[nH]1 ZINC000217649874 BB For-Sale Unstable ALPL 58 38 Cn1nccc1[C@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc3c21 ZINC000217649875 HG In-Stock Unstable AKR1B1 0 43 Cn1nccc1[C@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc3c21 ZINC000217649875 HG In-Stock Unstable CYP1B1 25 40 Cn1nccc1[C@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc3c21 ZINC000217649875 HG In-Stock Unstable CYP1A1 23 40 CCCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217649887 HH In-Stock Unstable CA2 15 42 CCCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217649887 HH In-Stock Unstable TBXA2R 38 42 CCCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217649887 HH In-Stock Unstable TBXAS1 30 42 CCCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217649887 HH In-Stock Unstable CASP3 0 41 CCCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217649887 HH In-Stock Unstable BMP1 46 35 CCCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217649887 HH In-Stock Unstable CA1 16 42 CCCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217649887 HH In-Stock Unstable MMP13 45 39 CCCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217649887 HH In-Stock Unstable ALOX15B 0 45 CCCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217649887 HH In-Stock Unstable ALOX15 60 46 CCCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217649887 HH In-Stock Unstable MMP9 40 39 CCCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217649887 HH In-Stock Unstable PTGDR 30 41 CCCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217649887 HH In-Stock Unstable IAP 0 48 CCCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217649887 HH In-Stock Unstable CA9 25 42 CCCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217649887 HH In-Stock Unstable AKR1C3 28 45 CCCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217649887 HH In-Stock Unstable AKR1C2 46 36 CCCCCC[C@@H](C)N[C@@H]1CCC[C@@H](O)C1 ZINC000217649914 BG For-Sale Unstable ADH1B 0 40 CCCCCC[C@@H](C)N[C@@H]1CCC[C@@H](O)C1 ZINC000217649914 BG For-Sale Unstable ADH1C 0 40 C[C@H](NC(=O)N1CCN([C@@H](C)C(=O)NC2CC2)CC1)c1ccc(-c2ccccc2)cc1 ZINC000217649926 HG On-Demand Unstable ACACA 47 40 C[C@H](NC(=O)N1CCN([C@@H](C)C(=O)NC2CC2)CC1)c1ccc(-c2ccccc2)cc1 ZINC000217649926 HG On-Demand Unstable PRCP 22 41 C[C@H](NC(=O)N1CCN([C@@H](C)C(=O)NC2CC2)CC1)c1ccc(-c2ccccc2)cc1 ZINC000217649926 HG On-Demand Unstable ACACB 18 40 C[C@H](NC(=O)N1CCN([C@@H](C)C(=O)NC2CC2)CC1)c1ccc(-c2ccccc2)cc1 ZINC000217649926 HG On-Demand Unstable BIRC3 42 34 C[C@H](NC(=O)N1CCN([C@@H](C)C(=O)NC2CC2)CC1)c1ccc(-c2ccccc2)cc1 ZINC000217649926 HG On-Demand Unstable BIRC2 41 34 C[C@H](NC(=O)N1CCN([C@@H](C)C(=O)NC2CC2)CC1)c1ccc(-c2ccccc2)cc1 ZINC000217649926 HG On-Demand Unstable BIRC8 47 33 Cc1c(C(=O)Nc2ccccc2-c2cn3ccsc3n2)cnn1-c1ccccc1 ZINC000217649956 GJ In-Stock Unstable SLC9A2 0 40 NCCCc1cc(F)c(Br)cc1F ZINC000217649964 CF For-Sale Unstable MPO 20 41 O=C(O)[C@@H]1CC[C@@H]1N1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217649983 BE For-Sale Unstable CYP2D26 0 40 CCCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217649991 JH In-Stock Unstable INHA 41 35 CCCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217649991 JH In-Stock Unstable TBXAS1 20 43 CCCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217649991 JH In-Stock Unstable ALOX15 45 38 CCCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217649991 JH In-Stock Unstable PTGDR 25 40 CCCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217649991 JH In-Stock Unstable IAP 0 49 CCCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217649991 JH In-Stock Unstable PTGDR2 15 40 CCCCCNS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217649991 JH In-Stock Unstable SCMU_MYCTU 0 44 Cc1cc(NC(=O)c2cccc(/C=C\C(=O)O)c2)n(C)n1 ZINC000217649994 CE For-Sale Unstable HDAC8 41 44 Cc1cc(NC(=O)c2cccc(/C=C\C(=O)O)c2)n(C)n1 ZINC000217649994 CE For-Sale Unstable HDAC6 29 44 Cc1cc(NC(=O)c2cccc(/C=C\C(=O)O)c2)n(C)n1 ZINC000217649994 CE For-Sale Unstable KCNK3 80 38 Cc1cc(NC(=O)c2cccc(/C=C\C(=O)O)c2)n(C)n1 ZINC000217649994 CE For-Sale Unstable KCNK9 42 38 CCCCCC[C@H](C)N[C@@H]1CCC[C@@H](O)C1 ZINC000217650001 BG On-Demand Unstable ADH1B 0 40 CCCCCC[C@H](C)N[C@@H]1CCC[C@@H](O)C1 ZINC000217650001 BG On-Demand Unstable ADH1C 0 40 C[C@@H](NC(=O)N1CCN([C@H](C)C(=O)NC2CC2)CC1)c1ccc(-c2ccccc2)cc1 ZINC000217650012 HG On-Demand Unstable ACACA 47 40 C[C@@H](NC(=O)N1CCN([C@H](C)C(=O)NC2CC2)CC1)c1ccc(-c2ccccc2)cc1 ZINC000217650012 HG On-Demand Unstable PRCP 22 41 C[C@@H](NC(=O)N1CCN([C@H](C)C(=O)NC2CC2)CC1)c1ccc(-c2ccccc2)cc1 ZINC000217650012 HG On-Demand Unstable ACACB 18 40 C[C@@H](NC(=O)N1CCN([C@H](C)C(=O)NC2CC2)CC1)c1ccc(-c2ccccc2)cc1 ZINC000217650012 HG On-Demand Unstable BIRC3 42 34 C[C@@H](NC(=O)N1CCN([C@H](C)C(=O)NC2CC2)CC1)c1ccc(-c2ccccc2)cc1 ZINC000217650012 HG On-Demand Unstable BIRC2 41 34 C[C@@H](NC(=O)N1CCN([C@H](C)C(=O)NC2CC2)CC1)c1ccc(-c2ccccc2)cc1 ZINC000217650012 HG On-Demand Unstable BIRC8 47 33 O=C(N/C=C/c1ccccc1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217650023 FF For-Sale Unstable DRD4 25 52 O=C(N/C=C/c1ccccc1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217650023 FF For-Sale Unstable EDNRA 15 41 O=C(N/C=C/c1ccccc1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217650023 FF For-Sale Unstable BMP1 36 44 O=C(N/C=C/c1ccccc1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217650023 FF For-Sale Unstable SIGMAR1 29 55 O=C(N/C=C/c1ccccc1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217650023 FF For-Sale Unstable NOS2 70 36 O=C(N/C=C/c1ccccc1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217650023 FF For-Sale Unstable SSTR3 92 33 O=C(N/C=C/c1ccccc1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217650023 FF For-Sale Unstable FAAH 21 43 O=C(N/C=C/c1ccccc1)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217650023 FF For-Sale Unstable MCHR1 31 52 NCCCc1ccc(F)c(Br)c1F ZINC000217650082 CF For-Sale Unstable MPO 26 41 O=C(O)[C@H]1CC[C@@H]1N1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217650083 BE For-Sale Unstable CYP2D26 0 40 CCCCCC[C@@H](C)N[C@H]1CCC[C@@H](O)C1 ZINC000217650085 BG For-Sale Unstable ADH1B 0 40 CCCCCC[C@@H](C)N[C@H]1CCC[C@@H](O)C1 ZINC000217650085 BG For-Sale Unstable ADH1C 0 40 O=C(O)/C=C\c1ccc(C(=O)N2CCC(O)CC2)cc1 ZINC000217650090 CD For-Sale Unstable L3MBTL1 0 45 O=C(O)/C=C\c1ccc(C(=O)N2CCC(O)CC2)cc1 ZINC000217650090 CD For-Sale Unstable L3MBTL3 92 45 O=C(O)/C=C\c1ccc(C(=O)N2CCC(O)CC2)cc1 ZINC000217650090 CD For-Sale Unstable L3MBTL4 0 43 O=C(O)/C=C\c1ccc(C(=O)N2CCC(O)CC2)cc1 ZINC000217650090 CD For-Sale Unstable MBTD1 0 44 O=C(O)/C=C\c1ccc(C(=O)N2CCC(O)CC2)cc1 ZINC000217650090 CD For-Sale Unstable TP53BP1 0 43 O=C(O)/C=C\c1ccc(C(=O)N2CCC(O)CC2)cc1 ZINC000217650090 CD For-Sale Unstable GPR183 0 49 CCCCCNS(=O)(=O)c1ccc(NCc2ccco2)c(C(=O)O)c1 ZINC000217650100 FG In-Stock Unstable CASP3 15 41 NC(=O)COc1ccc([C@@H]2CC(=O)Oc3c2c(=O)oc2ccccc32)cc1 ZINC000217650104 FE In-Stock Unstable NQO1 17 40 C[C@H](NC(=O)N1CCN([C@H](C)C(=O)NC2CC2)CC1)c1ccc(-c2ccccc2)cc1 ZINC000217650105 HG On-Demand Unstable ACACA 47 40 C[C@H](NC(=O)N1CCN([C@H](C)C(=O)NC2CC2)CC1)c1ccc(-c2ccccc2)cc1 ZINC000217650105 HG On-Demand Unstable PRCP 22 41 C[C@H](NC(=O)N1CCN([C@H](C)C(=O)NC2CC2)CC1)c1ccc(-c2ccccc2)cc1 ZINC000217650105 HG On-Demand Unstable ACACB 18 40 C[C@H](NC(=O)N1CCN([C@H](C)C(=O)NC2CC2)CC1)c1ccc(-c2ccccc2)cc1 ZINC000217650105 HG On-Demand Unstable BIRC3 42 34 C[C@H](NC(=O)N1CCN([C@H](C)C(=O)NC2CC2)CC1)c1ccc(-c2ccccc2)cc1 ZINC000217650105 HG On-Demand Unstable BIRC2 41 34 C[C@H](NC(=O)N1CCN([C@H](C)C(=O)NC2CC2)CC1)c1ccc(-c2ccccc2)cc1 ZINC000217650105 HG On-Demand Unstable BIRC8 47 33 CCN(C/C=C\CN)Cc1ccccc1 ZINC000217650108 BE For-Sale Unstable SQLE 61 37 CCOC(=O)N1CCN(C(=O)N/C=C/c2ccccc2)CC1 ZINC000217650133 DE For-Sale Unstable P2RY12 96 43 CCOC(=O)N1CCN(C(=O)N/C=C/c2ccccc2)CC1 ZINC000217650133 DE For-Sale Unstable TGM2 23 40 CCOC(=O)N1CCN(C(=O)N/C=C/c2ccccc2)CC1 ZINC000217650133 DE For-Sale Unstable F13A1 36 40 O=C(O)[C@@H]1CC[C@H]1N1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217650162 BE For-Sale Unstable CYP2D26 0 40 CCCCCC[C@H](C)N[C@H]1CCC[C@@H](O)C1 ZINC000217650166 BG On-Demand Unstable ADH1B 0 40 CCCCCC[C@H](C)N[C@H]1CCC[C@@H](O)C1 ZINC000217650166 BG On-Demand Unstable ADH1C 0 40 Cc1nc(-c2ccccc2NC(=O)c2ccccc2C(F)(F)F)cs1 ZINC000217650186 FK In-Stock Unstable MPL 44 39 Cc1nc(-c2ccccc2NC(=O)c2ccccc2C(F)(F)F)cs1 ZINC000217650186 FK In-Stock Unstable STK33 50 37 NC(=O)COc1ccc([C@H]2CC(=O)Oc3c2c(=O)oc2ccccc32)cc1 ZINC000217650191 FE In-Stock Unstable NQO1 17 40 NCCCc1cc(Br)cc(F)c1F ZINC000217650201 CF For-Sale Unstable MPO 20 40 Cc1cccc(N2CCN(C/C=C\CN)CC2)c1C ZINC000217650215 CD For-Sale Unstable DRD2 15 43 Cc1cccc(N2CCN(C/C=C\CN)CC2)c1C ZINC000217650215 CD For-Sale Unstable HTR2A 15 42 Cc1cccc(N2CCN(C/C=C\CN)CC2)c1C ZINC000217650215 CD For-Sale Unstable HTR2C 15 42 Cc1cccc(N2CCN(C/C=C\CN)CC2)c1C ZINC000217650215 CD For-Sale Unstable DRD3 19 40 Cc1cccc(N2CCN(C/C=C\CN)CC2)c1C ZINC000217650215 CD For-Sale Unstable ABCB1 19 41 CCCCCNS(=O)(=O)c1ccc(NC[C@@H]2CCCO2)c(C(=O)O)c1 ZINC000217650223 FE In-Stock Unstable CASP3 0 40 C[C@@H](NC(=O)N1CCN(c2ncccc2C#N)CC1)c1cc(F)c(Cl)cc1Cl ZINC000217650250 HH On-Demand Unstable P2RY12 48 43 C[C@@H](NC(=O)N1CCN(c2ncccc2C#N)CC1)c1cc(F)c(Cl)cc1Cl ZINC000217650250 HH On-Demand Unstable TRPV1 15 59 NC1(CCc2ccccc2)C2CC3CC(C2)CC1C3 ZINC000217650262 CH For-Sale Unstable SLC18A2 44 39 NC1(CCc2ccccc2)C2CC3CC(C2)CC1C3 ZINC000217650262 CH For-Sale Unstable KDM1A 36 49 COc1ccc2c(c1)CCC[C@H]2N[C@@H]1CCC[C@@H](O)C1 ZINC000217650291 CF For-Sale Unstable GRIN2B 19 41 CCCCCNS(=O)(=O)c1ccc(NC[C@H]2CCCO2)c(C(=O)O)c1 ZINC000217650305 FE In-Stock Unstable CASP3 0 40 Cc1nc(-c2ccccc2NC(=O)C2CCN(S(C)(=O)=O)CC2)cs1 ZINC000217650307 GF In-Stock Unstable EPHX2 35 48 NC/C=C\CN1CCN(c2ccc(Cl)cc2)CC1 ZINC000217650327 CD For-Sale Unstable HTR1A 15 43 NC/C=C\CN1CCN(c2ccc(Cl)cc2)CC1 ZINC000217650327 CD For-Sale Unstable DRD1 0 45 NC/C=C\CN1CCN(c2ccc(Cl)cc2)CC1 ZINC000217650327 CD For-Sale Unstable DRD4 33 45 NC/C=C\CN1CCN(c2ccc(Cl)cc2)CC1 ZINC000217650327 CD For-Sale Unstable HTR7 15 40 C[C@H](NC(=O)N1CCN(c2ncccc2C#N)CC1)c1cc(F)c(Cl)cc1Cl ZINC000217650339 HH On-Demand Unstable P2RY12 48 43 C[C@H](NC(=O)N1CCN(c2ncccc2C#N)CC1)c1cc(F)c(Cl)cc1Cl ZINC000217650339 HH On-Demand Unstable TRPV1 15 59 COc1ccc2c(c1)CCC[C@@H]2N[C@@H]1CCC[C@@H](O)C1 ZINC000217650384 CF On-Demand Unstable GRIN2B 19 41 CCCCCNS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217650423 EE In-Stock Unstable CASP3 23 43 CCCCCNS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217650423 EE In-Stock Unstable KCNQ2 61 33 CCCCCNS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217650423 EE In-Stock Unstable SFRP1 50 32 O=C(N/C=C/c1ccccc1)Nc1ccc(C(F)(F)F)cc1 ZINC000217650453 DI For-Sale Anodyne EPHX1 0 41 O=C(N/C=C/c1ccccc1)Nc1ccc(C(F)(F)F)cc1 ZINC000217650453 DI For-Sale Anodyne DHODH 33 42 O=C(N/C=C/c1ccccc1)Nc1ccc(C(F)(F)F)cc1 ZINC000217650453 DI For-Sale Anodyne TRPV1 20 43 O=C(N/C=C/c1ccccc1)Nc1ccc(C(F)(F)F)cc1 ZINC000217650453 DI For-Sale Anodyne EPHX2 33 43 O=C(N/C=C/c1ccccc1)Nc1ccc(C(F)(F)F)cc1 ZINC000217650453 DI For-Sale Anodyne FPR2 20 44 O=C(N/C=C/c1ccccc1)Nc1ccc(C(F)(F)F)cc1 ZINC000217650453 DI For-Sale Anodyne PTPA 0 44 O=C(N/C=C/c1ccccc1)Nc1ccc(C(F)(F)F)cc1 ZINC000217650453 DI For-Sale Anodyne P96878_MYCTU 15 47 O=C(N/C=C/c1ccccc1)Nc1ccc(C(F)(F)F)cc1 ZINC000217650453 DI For-Sale Anodyne P95276_MYCTO 0 41 COc1ccc2c(c1)CCC[C@H]2N[C@H]1CCC[C@@H](O)C1 ZINC000217650461 CF For-Sale Unstable GRIN2B 19 41 Cc1ccc(Br)c(OCC(=O)O)c1 ZINC000217650491 BE For-Sale Unstable THRA 22 41 Cc1ccc(Br)c(OCC(=O)O)c1 ZINC000217650491 BE For-Sale Unstable THRB 19 41 Cc1ccc(Br)c(OCC(=O)O)c1 ZINC000217650491 BE For-Sale Unstable PLA2G2A 51 32 Cc1ccc(Br)c(OCC(=O)O)c1 ZINC000217650491 BE For-Sale Unstable PPARD 36 40 Cc1ccc(Br)c(OCC(=O)O)c1 ZINC000217650491 BE For-Sale Unstable PTGDR2 40 49 CCOC(=O)c1c[nH]c(=O)c2c1OC(=O)C[C@@H]2c1ccc(OC)c(OCc2ccccc2)c1 ZINC000217650506 IH In-Stock Unstable TSHR 49 34 Cc1nc(-c2ccccc2NC(=O)c2cccc(Cl)c2)cs1 ZINC000217650529 EK In-Stock Unstable GRM5 25 41 Cc1nc(-c2ccccc2NC(=O)c2cccc(Cl)c2)cs1 ZINC000217650529 EK In-Stock Unstable LUCI_LUCLA 16 41 Cc1nc(-c2ccccc2NC(=O)c2cccc(Cl)c2)cs1 ZINC000217650529 EK In-Stock Unstable STK33 49 40 Cc1nc(-c2ccccc2NC(=O)c2cccc(Cl)c2)cs1 ZINC000217650529 EK In-Stock Unstable KCNK3 61 45 Cc1nc(-c2ccccc2NC(=O)c2cccc(Cl)c2)cs1 ZINC000217650529 EK In-Stock Unstable KCNK9 43 45 CCCCCNS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217650533 FF In-Stock Unstable CASP3 16 43 CCCCCNS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217650533 FF In-Stock Unstable KCNQ2 44 33 COc1ccc2c(c1)CCC[C@@H]2N[C@H]1CCC[C@@H](O)C1 ZINC000217650549 CF On-Demand Unstable GRIN2B 19 41 CN(C/C=C\CN)Cc1ccc(Br)cc1 ZINC000217650562 CE For-Sale Unstable SHC 34 48 CCOC(=O)c1c[nH]c(=O)c2c1OC(=O)C[C@H]2c1ccc(OC)c(OCc2ccccc2)c1 ZINC000217650588 IH In-Stock Unstable TSHR 49 34 CCCCCNS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1 ZINC000217650635 FD In-Stock Unstable HTR7 21 40 CCCCCNS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1 ZINC000217650635 FD In-Stock Unstable CASP3 15 42 CCCCCNS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1 ZINC000217650635 FD In-Stock Unstable SLC6A9 17 46 O=C(N/C=C/c1ccccc1)Nc1cc(F)ccc1F ZINC000217650673 CH For-Sale Anodyne MMP1 0 47 C[C@@H](NC(=O)[C@@H]1CC[C@@H](CNC(=O)Cn2c(=O)[nH]c3ccccc3c2=O)CC1)C(=O)O ZINC000217650711 IC In-Stock Unstable AVPR1B 33 41 CCCCCNS(=O)(=O)c1ccc(NCCCOCC)c(C(=O)O)c1 ZINC000217650719 FF In-Stock Unstable CASP3 15 45 CCCCCNS(=O)(=O)c1ccc(NCCCOCC)c(C(=O)O)c1 ZINC000217650719 FF In-Stock Unstable BDKRB1 16 41 O=C(N/C=C/c1ccccc1)N1CCCC[C@H]1CCO ZINC000217650772 CF For-Sale Unstable HCRTR1 17 41 COC[C@@H]1CCCN(C(=O)c2ccc(C#CC(C)(C)O)cc2)C1 ZINC000217650777 DE In-Stock Unstable GRM3 20 61 CCCCCNS(=O)(=O)c1ccc(NCCCOC(C)C)c(C(=O)O)c1 ZINC000217650820 GG In-Stock Unstable CASP3 15 44 O=C(N/C=C/c1ccccc1)N1CCCC[C@@H]1CCO ZINC000217650849 CF For-Sale Unstable HCRTR1 17 41 COC[C@H]1CCCN(C(=O)c2ccc(C#CC(C)(C)O)cc2)C1 ZINC000217650863 DE In-Stock Unstable GRM3 20 61 CN1CCCN(C(=O)c2ccc(/C=C\C(=O)O)s2)CC1 ZINC000217650892 CD For-Sale Unstable HRH4 26 40 COC(=O)C[C@H](c1ccc2c(c1)OCO2)c1oc(CN2CCCCC2)cc(=O)c1O ZINC000217650908 HF In-Stock Unstable RORC 33 40 CCCCCNc1ccc(S(=O)(=O)NCCCCC)cc1C(=O)O ZINC000217650935 FG In-Stock Unstable CASP3 22 48 COC(=O)C[C@@H](c1ccc2c(c1)OCO2)c1oc(CN2CCCCC2)cc(=O)c1O ZINC000217650969 HF In-Stock Unstable RORC 33 40 O=C(O)/C=C\c1cccc(C(=O)NCC2CCCC2)c1 ZINC000217650978 CF For-Sale Unstable HDAC8 25 43 O=C(O)/C=C\c1cccc(C(=O)NCC2CCCC2)c1 ZINC000217650978 CF For-Sale Unstable HDAC6 15 43 O=C(O)/C=C\c1cccc(C(=O)NCC2CCCC2)c1 ZINC000217650978 CF For-Sale Unstable CACNA1I 62 43 O=C(Cn1c(=O)[nH]c2ccccc2c1=O)NC[C@@H]1CC[C@@H](C(=O)N2CCC(C(=O)O)CC2)CC1 ZINC000217650997 JC In-Stock Unstable AVPR1B 32 42 CCCCCNS(=O)(=O)c1ccc(NCCC(C)C)c(C(=O)O)c1 ZINC000217651042 FG In-Stock Unstable CASP3 22 49 O=C(Nc1ccccc1-c1csc(-c2ccccc2F)n1)c1ccccc1Cl ZINC000217651055 HK In-Stock Anodyne EPHB3 43 37 O=C(Nc1ccccc1-c1csc(-c2ccccc2F)n1)c1ccccc1Cl ZINC000217651055 HK In-Stock Anodyne NR2E3 61 39 O=C(Nc1ccccc1-c1csc(-c2ccccc2F)n1)c1ccccc1Cl ZINC000217651055 HK In-Stock Anodyne SMO 23 43 O=C(Nc1ccccc1-c1csc(-c2ccccc2F)n1)c1ccccc1Cl ZINC000217651055 HK In-Stock Anodyne STK33 44 37 O=C(Nc1ccccc1-c1csc(-c2ccccc2F)n1)c1ccccc1Cl ZINC000217651055 HK In-Stock Anodyne G2YM83_BOTF4 43 30 c1ccc(CCN[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217651056 BE On-Demand Unstable SLC18A2 43 36 c1ccc(CCN[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217651056 BE On-Demand Unstable SIGMAR1 29 60 c1ccc(CCN[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217651056 BE On-Demand Unstable SLC18A3 57 38 O=C(O)/C=C\c1ccc(F)c(C(=O)NCC2CCCC2)c1 ZINC000217651058 CF For-Sale Unstable CACNA1I 55 33 Cc1noc2nc(-c3ccc(F)cc3)cc(C(=O)N3CCN(c4ccc(O)cc4)CC3)c12 ZINC000217651061 II On-Demand Unstable SLC6A9 20 42 O=C(N/C=C/c1ccccc1)N1CCN(c2ccccn2)CC1 ZINC000217651075 DF For-Sale Unstable FAAH 22 41 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c(OC)c1 ZINC000217651078 JI In-Stock Unstable AKR1B1 0 47 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c(OC)c1 ZINC000217651078 JI In-Stock Unstable CYP1B1 57 36 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c(OC)c1 ZINC000217651078 JI In-Stock Unstable CYP1A1 43 47 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c(OC)c1 ZINC000217651078 JI In-Stock Unstable CYP1A2 33 41 c1ccc(CCN[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217651138 BE On-Demand Unstable SLC18A2 43 36 c1ccc(CCN[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217651138 BE On-Demand Unstable SIGMAR1 29 60 c1ccc(CCN[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217651138 BE On-Demand Unstable SLC18A3 57 38 CCCCCNS(=O)(=O)c1ccc(N[C@@H](C)CCC)c(C(=O)O)c1 ZINC000217651144 FG In-Stock Unstable CASP3 22 49 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c(OC)c1 ZINC000217651147 JI In-Stock Unstable AKR1B1 0 47 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c(OC)c1 ZINC000217651147 JI In-Stock Unstable CYP1B1 57 36 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c(OC)c1 ZINC000217651147 JI In-Stock Unstable CYP1A1 43 47 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c(OC)c1 ZINC000217651147 JI In-Stock Unstable CYP1A2 33 41 O=C(Nc1ccccc1-c1csc(-c2ccccc2F)n1)c1ccccc1C(F)(F)F ZINC000217651159 IK In-Stock Anodyne MPL 56 41 O=C(Nc1ccccc1-c1csc(-c2ccccc2F)n1)c1ccccc1C(F)(F)F ZINC000217651159 IK In-Stock Anodyne STK33 50 37 CCCCCNS(=O)(=O)c1ccc(N[C@H](C)CCC)c(C(=O)O)c1 ZINC000217651223 FG In-Stock Unstable CASP3 22 49 O=C(O)/C=C\c1cccc(C(=O)NCC(=O)NC2CC2)c1 ZINC000217651245 CC For-Sale Unstable CCR2 70 51 CC(C)CCNS(=O)(=O)c1ccc(Cl)c(CO)c1 ZINC000217651247 CE For-Sale Unstable TBXA2R 43 34 c1csc(CN[C@@H]2CCN3CCCC[C@@H]23)c1 ZINC000217651251 BE On-Demand Unstable VACHT_TETCF 0 41 O=C(Nc1ccccc1-c1csc(-c2ccccc2F)n1)c1cc2ccccc2oc1=O ZINC000217651282 IK In-Stock Anodyne MAOB 15 57 O=C(Nc1ccccc1-c1csc(-c2ccccc2F)n1)c1cc2ccccc2oc1=O ZINC000217651282 IK In-Stock Anodyne F12 0 40 O=C(Nc1ccccc1-c1csc(-c2ccccc2F)n1)c1cc2ccccc2oc1=O ZINC000217651282 IK In-Stock Anodyne CDC25C 0 42 O=c1n(-c2ccccc2)cnn1CCCN1CCCCC1 ZINC000217651284 CD On-Demand Unstable HTR1A 27 43 O=c1n(-c2ccccc2)cnn1CCCN1CCCCC1 ZINC000217651284 CD On-Demand Unstable HTR2A 19 43 O=c1n(-c2ccccc2)cnn1CCCN1CCCCC1 ZINC000217651284 CD On-Demand Unstable HTR7 25 42 O=c1n(-c2ccccc2)cnn1CCCN1CCCCC1 ZINC000217651284 CD On-Demand Unstable SIGMAR1 19 41 O=c1n(-c2ccccc2)cnn1CCCN1CCCCC1 ZINC000217651284 CD On-Demand Unstable HNMT 70 37 c1csc(CN[C@H]2CCN3CCCC[C@@H]23)c1 ZINC000217651338 BE On-Demand Unstable VACHT_TETCF 0 41 CCCCCNS(=O)(=O)c1ccc(N[C@@H](C)COC)c(C(=O)O)c1 ZINC000217651342 FE In-Stock Unstable CASP3 0 42 O=C(Nc1ccccc1-c1csc(-c2ccccc2F)n1)c1ccccn1 ZINC000217651386 GK In-Stock Anodyne MPL 44 38 O=C(Nc1ccccc1-c1csc(-c2ccccc2F)n1)c1ccccn1 ZINC000217651386 GK In-Stock Anodyne MAP 0 46 O=C(Nc1ccccc1-c1csc(-c2ccccc2F)n1)c1ccccn1 ZINC000217651386 GK In-Stock Anodyne GRM4 71 47 O=C(Nc1ccccc1-c1csc(-c2ccccc2F)n1)c1ccccn1 ZINC000217651386 GK In-Stock Anodyne HDAC1 18 45 O=C(Nc1ccccc1-c1csc(-c2ccccc2F)n1)c1ccccn1 ZINC000217651386 GK In-Stock Anodyne PYGM 24 40 O=C(Nc1ccccc1-c1csc(-c2ccccc2F)n1)c1ccccn1 ZINC000217651386 GK In-Stock Anodyne STK33 45 38 C[C@@H]1CN(CC[C@@H](N)c2cccc(Cl)c2)CCCO1 ZINC000217651401 CF For-Sale Unstable OPRL1 0 41 Cc1ccccc1[C@@H](C)N[C@@H](C)C(=O)Nc1nc2ccccc2s1 ZINC000217651416 EI On-Demand Unstable LCK 32 42 Cc1ccccc1[C@@H](C)N[C@@H](C)C(=O)Nc1nc2ccccc2s1 ZINC000217651416 EI On-Demand Unstable CSNK1D 34 46 Cc1ccccc1[C@@H](C)N[C@@H](C)C(=O)Nc1nc2ccccc2s1 ZINC000217651416 EI On-Demand Unstable BCL2L1 47 35 CCCCCNS(=O)(=O)c1ccc(N[C@H](C)COC)c(C(=O)O)c1 ZINC000217651425 FE In-Stock Unstable CASP3 0 42 c1cncc(CN[C@@H]2CCN3CCCC[C@@H]23)c1 ZINC000217651448 BD On-Demand Unstable ACHP_LYMST 22 43 c1cncc(CN[C@@H]2CCN3CCCC[C@@H]23)c1 ZINC000217651448 BD On-Demand Unstable NAMPT 30 42 C[C@H]1CN(CC[C@@H](N)c2cccc(Cl)c2)CCCO1 ZINC000217651475 CF For-Sale Unstable OPRL1 0 41 CC[C@@H](C)[C@H](NC(=O)[C@@H]1CC[C@@H](CNC(=O)Cn2c(=O)[nH]c3ccccc3c2=O)CC1)C(=O)O ZINC000217651485 JD In-Stock Unstable AVPR1B 32 41 CC[C@@H](C)[C@H](NC(=O)[C@@H]1CC[C@@H](CNC(=O)Cn2c(=O)[nH]c3ccccc3c2=O)CC1)C(=O)O ZINC000217651485 JD In-Stock Unstable Q7YY07_CRYPV 62 31 O=C(Nc1ccccc1-c1csc(-c2ccccc2F)n1)c1cccs1 ZINC000217651495 GK In-Stock Anodyne STK33 62 54 Cc1ccccc1[C@H](C)N[C@@H](C)C(=O)Nc1nc2ccccc2s1 ZINC000217651499 EI On-Demand Unstable LCK 32 42 Cc1ccccc1[C@H](C)N[C@@H](C)C(=O)Nc1nc2ccccc2s1 ZINC000217651499 EI On-Demand Unstable CSNK1D 34 46 Cc1ccccc1[C@H](C)N[C@@H](C)C(=O)Nc1nc2ccccc2s1 ZINC000217651499 EI On-Demand Unstable BCL2L1 47 35 COC(=O)CNC(=O)N/C=C/c1ccccc1 ZINC000217651509 BD For-Sale Unstable TLR4 22 41 c1cncc(CN[C@H]2CCN3CCCC[C@@H]23)c1 ZINC000217651531 BD On-Demand Unstable ACHP_LYMST 22 43 c1cncc(CN[C@H]2CCN3CCCC[C@@H]23)c1 ZINC000217651531 BD On-Demand Unstable NAMPT 30 42 CCCNc1ccc(S(=O)(=O)NCCC(C)C)cc1C(=O)O ZINC000217651538 EF In-Stock Unstable CASP3 16 44 Cc1ccc(Cl)cc1NC(=O)C(F)F ZINC000217651588 BF On-Demand Unstable S1PR4 26 40 Cc1ccc(Cl)cc1NC(=O)C(F)F ZINC000217651588 BF On-Demand Unstable LEF 53 37 Cc1ccc(CCC(=O)N[C@@H](C)Cc2cccnc2)cc1C ZINC000217651589 CG In-Stock Unstable TBXAS1 36 42 Cc1ccc(CCC(=O)N[C@@H](C)Cc2cccnc2)cc1C ZINC000217651589 CG In-Stock Unstable PTAFR 28 44 Cc1ccccc1[C@@H](C)N[C@H](C)C(=O)Nc1nc2ccccc2s1 ZINC000217651592 EI On-Demand Unstable LCK 32 42 Cc1ccccc1[C@@H](C)N[C@H](C)C(=O)Nc1nc2ccccc2s1 ZINC000217651592 EI On-Demand Unstable CSNK1D 34 46 Cc1ccccc1[C@@H](C)N[C@H](C)C(=O)Nc1nc2ccccc2s1 ZINC000217651592 EI On-Demand Unstable BCL2L1 47 35 O=C(Nc1ccccc1-c1csc(-c2ccccc2F)n1)c1ccco1 ZINC000217651618 FK In-Stock Anodyne KISS1R 56 37 Cc1cccnc1NC(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217651619 CF For-Sale Unstable TRPV1 16 42 COC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217651629 CG For-Sale Unstable PPIA 15 47 COC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217651629 CG For-Sale Unstable CCKAR 0 41 COC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217651629 CG For-Sale Unstable AKR1C3 29 40 COC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217651629 CG For-Sale Unstable PARP14 0 40 COC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217651629 CG For-Sale Unstable PARP15 0 40 COC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217651629 CG For-Sale Unstable KCNK3 107 41 COC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217651629 CG For-Sale Unstable KCNK9 65 38 COC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2)c1 ZINC000217651629 CG For-Sale Unstable PARP10 0 40 CC(C)CCNS(=O)(=O)c1ccc(NC(C)C)c(C(=O)O)c1 ZINC000217651641 EF In-Stock Unstable CASP3 16 43 CCCCCCCCOc1ccc([C@H](CC(N)=O)c2oc(C)cc(=O)c2O)cc1 ZINC000217651683 HI In-Stock Unstable THRA 41 37 CCCCCCCCOc1ccc([C@H](CC(N)=O)c2oc(C)cc(=O)c2O)cc1 ZINC000217651683 HI In-Stock Unstable PLA2G4B 94 39 Cc1ccc(CCC(=O)N[C@H](C)Cc2cccnc2)cc1C ZINC000217651690 CG In-Stock Unstable TBXAS1 36 42 Cc1ccc(CCC(=O)N[C@H](C)Cc2cccnc2)cc1C ZINC000217651690 CG In-Stock Unstable PTAFR 28 44 Cc1ccccc1[C@H](C)N[C@H](C)C(=O)Nc1nc2ccccc2s1 ZINC000217651691 EI On-Demand Unstable LCK 32 42 Cc1ccccc1[C@H](C)N[C@H](C)C(=O)Nc1nc2ccccc2s1 ZINC000217651691 EI On-Demand Unstable CSNK1D 34 46 Cc1ccccc1[C@H](C)N[C@H](C)C(=O)Nc1nc2ccccc2s1 ZINC000217651691 EI On-Demand Unstable BCL2L1 47 35 Cc1cccnc1NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217651710 CF For-Sale Unstable PTGER2 0 40 Cc1cccnc1NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217651710 CF For-Sale Unstable HDAC8 35 47 Cc1cccnc1NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217651710 CF For-Sale Unstable HDAC6 21 47 Cc1cccnc1NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217651710 CF For-Sale Unstable MMP1 0 42 Cc1cccnc1NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217651710 CF For-Sale Unstable KCNK3 80 39 Cc1cccnc1NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217651710 CF For-Sale Unstable KCNK9 43 38 CC(=O)Nc1ccc(CN[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217651719 CE On-Demand Unstable SSTR3 16 42 O=C(Nc1ccccc1-c1csc(-c2ccccc2F)n1)c1ccc(=O)[nH]c1 ZINC000217651724 GJ In-Stock Anodyne STK33 42 42 CCCCNc1ccc(S(=O)(=O)NCCC(C)C)cc1C(=O)O ZINC000217651747 EF In-Stock Unstable CASP3 16 45 CCCCCCCCOc1ccc([C@@H](CC(N)=O)c2oc(C)cc(=O)c2O)cc1 ZINC000217651764 HI In-Stock Unstable THRA 41 37 CCCCCCCCOc1ccc([C@@H](CC(N)=O)c2oc(C)cc(=O)c2O)cc1 ZINC000217651764 HI In-Stock Unstable PLA2G4B 78 39 CCOC(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217651767 DG For-Sale Unstable ADORA3 0 45 CCOC(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217651767 DG For-Sale Unstable F2RL3 19 40 CCOC(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217651767 DG For-Sale Unstable PDS 41 41 C[C@@H]1CCCCN1C(=O)C(F)F ZINC000217651784 AD On-Demand Unstable DPP7 25 43 O=C(O)[C@@H]1CC[C@@H]1N(Cc1ccsc1)C1CC1 ZINC000217651827 CF For-Sale Unstable GRM3 15 45 CC(C)CCNS(=O)(=O)c1ccc(NCC(C)C)c(C(=O)O)c1 ZINC000217651852 EF In-Stock Unstable CASP3 17 44 CC(C)CCNS(=O)(=O)c1ccc(NCC(C)C)c(C(=O)O)c1 ZINC000217651852 EF In-Stock Unstable MTNN 45 32 C[C@H]1CCCCN1C(=O)C(F)F ZINC000217651873 AD On-Demand Unstable DPP7 25 43 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)N1CCN(c3ccccc3)CC1)C(=O)OC2 ZINC000217651880 JI In-Stock Unstable IMPDH1 0 61 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)N1CCN(c3ccccc3)CC1)C(=O)OC2 ZINC000217651880 JI In-Stock Unstable IMPDH2 0 61 O=C(O)[C@@H]1CC[C@H]1N(Cc1ccsc1)C1CC1 ZINC000217651901 CF For-Sale Unstable GRM3 15 45 CCn1cc(NC(=O)c2ccc(/C=C\C(=O)O)cc2)cn1 ZINC000217651960 CE For-Sale Unstable PANC 52 35 CC[C@@H](C)Nc1ccc(S(=O)(=O)NCCC(C)C)cc1C(=O)O ZINC000217651962 EF In-Stock Unstable CASP3 16 41 O=C(/C=C/c1cccnc1)Nc1ccccc1-c1csc(-c2ccccc2F)n1 ZINC000217651975 HK In-Stock Anodyne HDAC1 0 44 O=C(/C=C/c1cccnc1)Nc1ccccc1-c1csc(-c2ccccc2F)n1 ZINC000217651975 HK In-Stock Anodyne MMP1 0 49 O=C(N/C=C/c1ccccc1)NCc1ccc(CO)cc1 ZINC000217651993 CF For-Sale Unstable ANPEP 17 40 O=C(N/C=C/c1ccccc1)NCc1ccc(CO)cc1 ZINC000217651993 CF For-Sale Unstable AMP1_PLAFQ 38 43 COc1ccccc1-c1c(C(N)=O)sc2cnc(Nc3ccc(-c4cnn(C)c4)cc3OC(C)C)nc12 ZINC000217651996 KK Annotated Unstable PLK1 60 41 COc1ccccc1-c1c(C(N)=O)sc2cnc(Nc3ccc(-c4cnn(C)c4)cc3OC(C)C)nc12 ZINC000217651996 KK Annotated Unstable PLK3 41 41 COc1ccccc1-c1c(C(N)=O)sc2cnc(Nc3ccc(-c4cnn(C)c4)cc3OC(C)C)nc12 ZINC000217651996 KK Annotated Unstable ALK 43 36 COc1ccccc1-c1c(C(N)=O)sc2cnc(Nc3ccc(-c4cnn(C)c4)cc3OC(C)C)nc12 ZINC000217651996 KK Annotated Unstable MAPK7 52 34 Clc1ccc(CN[C@@H]2CCN3CCCC[C@@H]23)c(Cl)c1 ZINC000217652021 CH On-Demand Unstable P2RX7 28 42 CC[C@H](C)Nc1ccc(S(=O)(=O)NCCC(C)C)cc1C(=O)O ZINC000217652046 EF In-Stock Unstable CASP3 16 41 Cc1ccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)nc1 ZINC000217652051 CF For-Sale Unstable F10 16 41 Cc1ccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)nc1 ZINC000217652051 CF For-Sale Unstable HDAC8 33 44 Cc1ccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)nc1 ZINC000217652051 CF For-Sale Unstable HDAC6 19 44 Cc1ccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)nc1 ZINC000217652051 CF For-Sale Unstable LUCI_LUCLA 49 45 Cc1ccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)nc1 ZINC000217652051 CF For-Sale Unstable KCNK3 86 41 Cc1ccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)nc1 ZINC000217652051 CF For-Sale Unstable KCNK9 47 41 Cc1cccn2c(Br)c(CC#N)nc12 ZINC000217652079 CE For-Sale Unstable BDKRB2 19 40 O=C(Nc1ccccc1-c1csc(-c2ccccc2F)n1)c1ccsc1 ZINC000217652082 GK In-Stock Anodyne HDAC1 33 42 O=C(Nc1ccccc1-c1csc(-c2ccccc2F)n1)c1ccsc1 ZINC000217652082 GK In-Stock Anodyne STK33 49 39 Cc1ccccc1CNC(=O)N/C=C/c1ccccc1 ZINC000217652095 CG For-Sale Unstable ANPEP 27 52 Cc1ccccc1CNC(=O)N/C=C/c1ccccc1 ZINC000217652095 CG For-Sale Unstable AMP1_PLAFQ 40 50 O=C(NC[C@H]1CCCN1c1nc2ccccc2o1)c1ccc(OC(F)(F)F)cc1 ZINC000217652097 HI In-Stock Unstable NOD2 17 40 Clc1ccc(CN[C@H]2CCN3CCCC[C@@H]23)c(Cl)c1 ZINC000217652104 CH On-Demand Unstable P2RX7 28 42 CC(C)CCNS(=O)(=O)c1ccc(NC(C)(C)C)c(C(=O)O)c1 ZINC000217652161 EF In-Stock Unstable CASP3 17 43 O=C(NC[C@@H]1CCCN1c1nc2ccccc2o1)c1ccc(OC(F)(F)F)cc1 ZINC000217652185 HI In-Stock Unstable NOD2 17 40 O=C(N/C=C/c1ccccc1)NCc1ccccc1Br ZINC000217652216 EH For-Sale Unstable ANPEP 24 52 O=C(N/C=C/c1ccccc1)NCc1ccccc1Br ZINC000217652216 EH For-Sale Unstable AMP1_PLAFQ 43 36 O=C(O)/C=C\c1ccc(C(=O)N2CCC(CO)CC2)cc1 ZINC000217652221 CD For-Sale Unstable GRIN2B 15 45 O=C(O)/C=C\c1ccc(C(=O)N2CCC(CO)CC2)cc1 ZINC000217652221 CD For-Sale Unstable L3MBTL3 88 42 COc1cccc(Br)c1CC(=O)O ZINC000217652247 BE For-Sale Unstable ALS 48 41 COc1cccc(Br)c1CC(=O)O ZINC000217652247 BE For-Sale Unstable PTGDR2 17 40 C=CCNc1ccc(S(=O)(=O)NCCC(C)C)cc1C(=O)O ZINC000217652269 EE In-Stock Unstable CASP3 0 41 O=C(Nc1ccccc1-c1csc(-c2ccccc2F)n1)c1ccoc1 ZINC000217652296 FK In-Stock Anodyne MPL 43 33 O=C(Nc1ccccc1-c1csc(-c2ccccc2F)n1)c1ccoc1 ZINC000217652296 FK In-Stock Anodyne STK33 46 40 Cc1cc(NC(=O)c2ccon2)ccc1/C=C\C(=O)O ZINC000217652301 CE For-Sale Unstable KCNK3 52 33 Cc1cccc(CNC(=O)N/C=C/c2ccccc2)c1 ZINC000217652329 CG For-Sale Unstable ANPEP 37 53 Cc1cccc(CNC(=O)N/C=C/c2ccccc2)c1 ZINC000217652329 CG For-Sale Unstable HDAC8 43 37 Cc1cccc(CNC(=O)N/C=C/c2ccccc2)c1 ZINC000217652329 CG For-Sale Unstable HDAC6 35 40 Cc1cccc(CNC(=O)N/C=C/c2ccccc2)c1 ZINC000217652329 CG For-Sale Unstable FBP1 16 43 Cc1cccc(CNC(=O)N/C=C/c2ccccc2)c1 ZINC000217652329 CG For-Sale Unstable AMP1_PLAFQ 52 36 Cc1cccc(CNC(=O)N/C=C/c2ccccc2)c1 ZINC000217652329 CG For-Sale Unstable E1 0 41 Cc1cccc(CNC(=O)N/C=C/c2ccccc2)c1 ZINC000217652329 CG For-Sale Unstable PDS 49 41 C=C(CC)COc1ccc(Br)cc1/C=C\C(=O)O ZINC000217652334 DH For-Sale Unstable TNFRSF1A 15 45 CC(C)C[C@H](NC(=O)[C@@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217652369 KG In-Stock Unstable PGC 49 31 CC(C)C[C@H](NC(=O)[C@@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217652369 KG In-Stock Unstable FCER2 57 33 CC(C)C[C@H](NC(=O)[C@@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217652369 KG In-Stock Unstable SSTR4 44 33 CC(C)C[C@H](NC(=O)[C@@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217652369 KG In-Stock Unstable CCKAR 17 40 CC(C)C[C@H](NC(=O)[C@@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217652369 KG In-Stock Unstable TIMP3 45 35 CC(C)C[C@H](NC(=O)[C@@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217652369 KG In-Stock Unstable CAPNS1 61 35 CC(C)C[C@H](NC(=O)[C@@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217652369 KG In-Stock Unstable HLA-DRB1 52 33 CC(C)C[C@H](NC(=O)[C@@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217652369 KG In-Stock Unstable REN 68 40 CC(C)C[C@H](NC(=O)[C@@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217652369 KG In-Stock Unstable CAPN1 74 39 CC(C)C[C@H](NC(=O)[C@@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217652369 KG In-Stock Unstable CAPN2 107 39 CC(C)C[C@H](NC(=O)[C@@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217652369 KG In-Stock Unstable FPR1 78 39 CC(C)C[C@H](NC(=O)[C@@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217652369 KG In-Stock Unstable NPR 79 35 CC(C)C[C@H](NC(=O)[C@@H](Cc1ccccc1)n1c(=O)[nH]c2ccccc2c1=O)C(=O)NC[C@@H]1CC[C@@H](C(=O)O)CC1 ZINC000217652369 KG In-Stock Unstable KISS1R 55 32 CC[C@@H]1CC[C@@H](NC)[C@@H](CCCc2ccccc2)C1 ZINC000217652379 CI For-Sale Unstable SLC18A2 34 42 CC(C)CCNS(=O)(=O)c1ccc(NC2CC2)c(C(=O)O)c1 ZINC000217652409 EE In-Stock Unstable CASP3 15 40 COc1cccc(CNC(=O)N/C=C/c2ccccc2)c1 ZINC000217652438 CG For-Sale Unstable DRD4 40 31 COc1cccc(CNC(=O)N/C=C/c2ccccc2)c1 ZINC000217652438 CG For-Sale Unstable HRH2 19 40 COc1cccc(CNC(=O)N/C=C/c2ccccc2)c1 ZINC000217652438 CG For-Sale Unstable GRIN2B 0 40 COc1cccc(CNC(=O)N/C=C/c2ccccc2)c1 ZINC000217652438 CG For-Sale Unstable ANPEP 25 55 COc1cccc(CNC(=O)N/C=C/c2ccccc2)c1 ZINC000217652438 CG For-Sale Unstable G6PC 24 42 COc1cccc(CNC(=O)N/C=C/c2ccccc2)c1 ZINC000217652438 CG For-Sale Unstable MMP13 29 42 COc1cccc(CNC(=O)N/C=C/c2ccccc2)c1 ZINC000217652438 CG For-Sale Unstable ROCK1 42 46 COc1cccc(CNC(=O)N/C=C/c2ccccc2)c1 ZINC000217652438 CG For-Sale Unstable MTNR1A 63 48 COc1cccc(CNC(=O)N/C=C/c2ccccc2)c1 ZINC000217652438 CG For-Sale Unstable MTNR1B 61 48 COc1cccc(CNC(=O)N/C=C/c2ccccc2)c1 ZINC000217652438 CG For-Sale Unstable ROCK2 53 51 COc1cccc(CNC(=O)N/C=C/c2ccccc2)c1 ZINC000217652438 CG For-Sale Unstable MMP9 19 45 COc1cccc(CNC(=O)N/C=C/c2ccccc2)c1 ZINC000217652438 CG For-Sale Unstable BACE1 16 40 COc1cccc(CNC(=O)N/C=C/c2ccccc2)c1 ZINC000217652438 CG For-Sale Unstable AMP1_PLAFQ 55 40 COc1cccc(CNC(=O)N/C=C/c2ccccc2)c1 ZINC000217652438 CG For-Sale Unstable CRTM 52 37 COc1cccc(CNC(=O)N/C=C/c2ccccc2)c1 ZINC000217652438 CG For-Sale Unstable PDS 71 46 C=C(CC)COc1ccc(/C=C\C(=O)O)cc1OCC ZINC000217652441 CH For-Sale Unstable AKR1C3 35 56 CC[C@H]1CC[C@@H](NC)[C@@H](CCCc2ccccc2)C1 ZINC000217652454 CI For-Sale Unstable SLC18A2 34 42 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)N1CCN(c2cccc(O)c2)CC1 ZINC000217652498 IH On-Demand Unstable HTR1A 25 45 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)N1CCN(c2cccc(O)c2)CC1 ZINC000217652498 IH On-Demand Unstable DRD2 32 53 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)N1CCN(c2cccc(O)c2)CC1 ZINC000217652498 IH On-Demand Unstable DRD4 75 53 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)N1CCN(c2cccc(O)c2)CC1 ZINC000217652498 IH On-Demand Unstable HTR2A 23 51 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)N1CCN(c2cccc(O)c2)CC1 ZINC000217652498 IH On-Demand Unstable DRD3 31 53 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)N1CCN(c2cccc(O)c2)CC1 ZINC000217652498 IH On-Demand Unstable SIGMAR1 34 54 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)N1CCN(c2cccc(O)c2)CC1 ZINC000217652498 IH On-Demand Unstable SSTR5 47 38 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)N1CCN(c2cccc(O)c2)CC1 ZINC000217652498 IH On-Demand Unstable CCR1 15 42 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)N1CCN(c2cccc(O)c2)CC1 ZINC000217652498 IH On-Demand Unstable CCR3 42 42 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)N1CCN(c2cccc(O)c2)CC1 ZINC000217652498 IH On-Demand Unstable MAPK1 26 41 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)N1CCN(c2cccc(O)c2)CC1 ZINC000217652498 IH On-Demand Unstable FAAH 26 47 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)N1CCN(c2cccc(O)c2)CC1 ZINC000217652498 IH On-Demand Unstable CCR2 21 44 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)N1CCN(c2cccc(O)c2)CC1 ZINC000217652498 IH On-Demand Unstable ME1 0 40 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)N1CCN(c2cccc(O)c2)CC1 ZINC000217652498 IH On-Demand Unstable CXCR3 48 40 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)N1CCN(c2cccc(O)c2)CC1 ZINC000217652498 IH On-Demand Unstable MCHR1 57 49 O=C(Nc1ccccc1-c1cn2ccccc2n1)c1ccc2nsnc2c1 ZINC000217652515 FI In-Stock Anodyne MAP3K5 43 34 CC(C)CCNS(=O)(=O)c1ccc(NC2CCCC2)c(C(=O)O)c1 ZINC000217652520 FG In-Stock Unstable CASP3 0 46 CC[C@@H]1CC[C@H](NC)[C@@H](CCCc2ccccc2)C1 ZINC000217652544 CI For-Sale Unstable SLC18A2 34 42 O=C(N/C=C/c1ccccc1)NCc1cccc(F)c1 ZINC000217652559 CG For-Sale Unstable GRIN2B 0 42 O=C(N/C=C/c1ccccc1)NCc1cccc(F)c1 ZINC000217652559 CG For-Sale Unstable ANPEP 16 51 O=C(N/C=C/c1ccccc1)NCc1cccc(F)c1 ZINC000217652559 CG For-Sale Unstable AMP1_PLAFQ 45 42 O=C(N/C=C/c1ccccc1)NCc1cccc(F)c1 ZINC000217652559 CG For-Sale Unstable PDS 36 40 C=C(CC)COc1cccc(/C=C\C(=O)O)c1 ZINC000217652561 BG For-Sale Unstable PTGER2 32 40 C=C(CC)COc1cccc(/C=C\C(=O)O)c1 ZINC000217652561 BG For-Sale Unstable CYSLTR1 17 41 C=C(CC)COc1cccc(/C=C\C(=O)O)c1 ZINC000217652561 BG For-Sale Unstable LTB4R 17 40 C=C(CC)COc1cccc(/C=C\C(=O)O)c1 ZINC000217652561 BG For-Sale Unstable AKR1C3 38 42 CC(C)CCNS(=O)(=O)c1ccc(NC2CCCCC2)c(C(=O)O)c1 ZINC000217652631 FG In-Stock Unstable CASP3 0 45 CC[C@H]1CC[C@H](NC)[C@@H](CCCc2ccccc2)C1 ZINC000217652637 CI For-Sale Unstable SLC18A2 34 42 CCN(CC)S(=O)(=O)Nc1cc(/C=C\C(=O)O)ccc1C ZINC000217652649 DE For-Sale Unstable AKR1C3 23 40 CCC[C@@H](O)CNC(=O)c1cc(N)n[nH]1 ZINC000217652666 BB For-Sale Unstable ALPL 55 39 C[C@@H](c1ccc(Br)cc1F)N1CCC[C@@H](C(=O)O)C1 ZINC000217652669 EG For-Sale Unstable SLC6A1 137 37 O=C(N/C=C/c1ccccc1)NCc1cccc(Cl)c1 ZINC000217652670 CH For-Sale Unstable GRIN2B 0 48 O=C(N/C=C/c1ccccc1)NCc1cccc(Cl)c1 ZINC000217652670 CH For-Sale Unstable ANPEP 22 51 O=C(N/C=C/c1ccccc1)NCc1cccc(Cl)c1 ZINC000217652670 CH For-Sale Unstable CACNA1B 24 43 O=C(N/C=C/c1ccccc1)NCc1cccc(Cl)c1 ZINC000217652670 CH For-Sale Unstable HDAC8 16 40 O=C(N/C=C/c1ccccc1)NCc1cccc(Cl)c1 ZINC000217652670 CH For-Sale Unstable FBP1 22 40 O=C(N/C=C/c1ccccc1)NCc1cccc(Cl)c1 ZINC000217652670 CH For-Sale Unstable AMP1_PLAFQ 47 38 O=C(N/C=C/c1ccccc1)NCc1cccc(Cl)c1 ZINC000217652670 CH For-Sale Unstable PDS 67 40 CC(C)[C@H](NC(=O)[C@@H]1CC[C@@H](CNC(=O)Cn2c(=O)[nH]c3ccccc3c2=O)CC1)C(=O)O ZINC000217652690 JC In-Stock Unstable AVPR1B 33 42 CC(C)[C@H](NC(=O)[C@@H]1CC[C@@H](CNC(=O)Cn2c(=O)[nH]c3ccccc3c2=O)CC1)C(=O)O ZINC000217652690 JC In-Stock Unstable ELANE 50 43 COc1ccc(C)c(C(=O)O)c1Br ZINC000217652695 BE For-Sale Unstable ALS 63 37 COc1ccccc1CCN1C(=O)N[C@@H](CC(=O)Nc2ccc3[nH]ccc3c2)C1=O ZINC000217652707 HF In-Stock Unstable TSHR 42 33 COc1ccccc1CCN1C(=O)N[C@@H](CC(=O)Nc2ccc3[nH]ccc3c2)C1=O ZINC000217652707 HF In-Stock Unstable ENPP1 68 33 O=C(Nc1ccccc1-c1cn2ccccc2n1)c1cc2ccccc2s1 ZINC000217652724 FK In-Stock Anodyne PIGA 0 40 O=C(O)/C=C\c1ccc(CNS(=O)(=O)c2cccs2)cc1 ZINC000217652737 DE For-Sale Unstable PTGER2 25 47 O=C(O)/C=C\c1ccc(CNS(=O)(=O)c2cccs2)cc1 ZINC000217652737 DE For-Sale Unstable PTGER4 0 47 O=C(O)/C=C\c1ccc(CNS(=O)(=O)c2cccs2)cc1 ZINC000217652737 DE For-Sale Unstable PTGER3 20 47 C[C@]12C[C@@H]3C[C@H](C1)C[C@@](NC(=O)SCc1ccccc1)(C3)C2 ZINC000217652741 DJ In-Stock Unstable EPHX2 41 46 CCC[C@H](O)CNC(=O)c1cc(N)n[nH]1 ZINC000217652749 BB For-Sale Unstable ALPL 55 39 C[C@H](c1ccc(Br)cc1F)N1CCC[C@@H](C(=O)O)C1 ZINC000217652755 EG For-Sale Unstable SLC6A1 137 37 O=C(N/C=C/c1ccccc1)NCc1cccc(Br)c1 ZINC000217652782 EH For-Sale Unstable ANPEP 35 41 O=C(N/C=C/c1ccccc1)NCc1cccc(Br)c1 ZINC000217652782 EH For-Sale Unstable HDAC6 15 43 O=C(N/C=C/c1ccccc1)NCc1cccc(Br)c1 ZINC000217652782 EH For-Sale Unstable AMP1_PLAFQ 53 37 O=C(N/C=C/c1ccccc1)NCc1cccc(Br)c1 ZINC000217652782 EH For-Sale Unstable PDS 48 40 C[C@@H](c1cc(Br)ccc1F)N1CCC[C@@H](C(=O)O)C1 ZINC000217652826 EG For-Sale Unstable SLC6A1 134 37 CC[C@@H](N[C@@H](C)C(=O)Nc1nc2ccccc2s1)c1ccc(OC)cc1 ZINC000217652828 FI On-Demand Unstable ACE 0 48 CC[C@@H](N[C@@H](C)C(=O)Nc1nc2ccccc2s1)c1ccc(OC)cc1 ZINC000217652828 FI On-Demand Unstable CSNK1D 42 45 CC[C@@H](N[C@@H](C)C(=O)Nc1nc2ccccc2s1)c1ccc(OC)cc1 ZINC000217652828 FI On-Demand Unstable PIK3CA 0 40 CC[C@@H](N[C@@H](C)C(=O)Nc1nc2ccccc2s1)c1ccc(OC)cc1 ZINC000217652828 FI On-Demand Unstable TACR3 45 39 CC[C@@H](N[C@@H](C)C(=O)Nc1nc2ccccc2s1)c1ccc(OC)cc1 ZINC000217652828 FI On-Demand Unstable LUCI_PHOPE 28 43 CC[C@@H](N[C@@H](C)C(=O)Nc1nc2ccccc2s1)c1ccc(OC)cc1 ZINC000217652828 FI On-Demand Unstable FABK 0 43 CC[C@@H](N[C@@H](C)C(=O)Nc1nc2ccccc2s1)c1ccc(OC)cc1 ZINC000217652828 FI On-Demand Unstable ISPD 0 46 CC[C@@H](N[C@@H](C)C(=O)Nc1nc2ccccc2s1)c1ccc(OC)cc1 ZINC000217652828 FI On-Demand Unstable GPR88 0 44 CSC[C@@](C)(O)CNC(=O)c1ccc(OCC(N)=O)cc1 ZINC000217652841 DC On-Demand Unstable PLA2G4B 46 35 CC(C)CCNS(=O)(=O)c1ccc(NCCO)c(C(=O)O)c1 ZINC000217652853 ED In-Stock Unstable CASP3 17 43 O=C(N/C=C/c1ccccc1)NCc1ccc(Br)cc1 ZINC000217652887 EH For-Sale Unstable ANPEP 34 43 O=C(N/C=C/c1ccccc1)NCc1ccc(Br)cc1 ZINC000217652887 EH For-Sale Unstable HDAC8 17 40 O=C(N/C=C/c1ccccc1)NCc1ccc(Br)cc1 ZINC000217652887 EH For-Sale Unstable AMP1_PLAFQ 49 45 O=C(Nc1ccc(OC(F)F)cc1)C(F)F ZINC000217652909 BE On-Demand Anodyne GUAB 0 42 CSC[C@](C)(O)CNC(=O)c1ccc(OCC(N)=O)cc1 ZINC000217652915 DC On-Demand Unstable PLA2G4B 46 35 CC[C@H](N[C@@H](C)C(=O)Nc1nc2ccccc2s1)c1ccc(OC)cc1 ZINC000217652918 FI On-Demand Unstable ACE 0 48 CC[C@H](N[C@@H](C)C(=O)Nc1nc2ccccc2s1)c1ccc(OC)cc1 ZINC000217652918 FI On-Demand Unstable CSNK1D 42 45 CC[C@H](N[C@@H](C)C(=O)Nc1nc2ccccc2s1)c1ccc(OC)cc1 ZINC000217652918 FI On-Demand Unstable PIK3CA 0 40 CC[C@H](N[C@@H](C)C(=O)Nc1nc2ccccc2s1)c1ccc(OC)cc1 ZINC000217652918 FI On-Demand Unstable TACR3 45 39 CC[C@H](N[C@@H](C)C(=O)Nc1nc2ccccc2s1)c1ccc(OC)cc1 ZINC000217652918 FI On-Demand Unstable LUCI_PHOPE 28 43 CC[C@H](N[C@@H](C)C(=O)Nc1nc2ccccc2s1)c1ccc(OC)cc1 ZINC000217652918 FI On-Demand Unstable FABK 0 43 CC[C@H](N[C@@H](C)C(=O)Nc1nc2ccccc2s1)c1ccc(OC)cc1 ZINC000217652918 FI On-Demand Unstable ISPD 0 46 CC[C@H](N[C@@H](C)C(=O)Nc1nc2ccccc2s1)c1ccc(OC)cc1 ZINC000217652918 FI On-Demand Unstable GPR88 0 44 C[C@H](c1cc(Br)ccc1F)N1CCC[C@@H](C(=O)O)C1 ZINC000217652923 EG For-Sale Unstable SLC6A1 134 37 N#Cc1ccccc1N1[C@H]2CC[C@H]1CC(C(=O)O)C2 ZINC000217652941 CE For-Sale Unstable AR 19 49 CCc1ccccc1NC(=O)N1CCN(c2cc(-n3cncn3)ncn2)CC1 ZINC000217652969 GD In-Stock Unstable PDGFRB 44 38 CC(C)CCNS(=O)(=O)c1ccc(NCCCO)c(C(=O)O)c1 ZINC000217652981 ED In-Stock Unstable CASP3 17 44 CC(C)CCNS(=O)(=O)c1ccc(NCCCO)c(C(=O)O)c1 ZINC000217652981 ED In-Stock Unstable BDKRB1 0 42 Cc1ccccc1CCNC(=O)N/C=C/c1ccccc1 ZINC000217653000 CH For-Sale Unstable MTNR1A 26 43 CC[C@@H](N[C@H](C)C(=O)Nc1nc2ccccc2s1)c1ccc(OC)cc1 ZINC000217653004 FI On-Demand Unstable ACE 0 48 CC[C@@H](N[C@H](C)C(=O)Nc1nc2ccccc2s1)c1ccc(OC)cc1 ZINC000217653004 FI On-Demand Unstable CSNK1D 42 45 CC[C@@H](N[C@H](C)C(=O)Nc1nc2ccccc2s1)c1ccc(OC)cc1 ZINC000217653004 FI On-Demand Unstable PIK3CA 0 40 CC[C@@H](N[C@H](C)C(=O)Nc1nc2ccccc2s1)c1ccc(OC)cc1 ZINC000217653004 FI On-Demand Unstable TACR3 45 39 CC[C@@H](N[C@H](C)C(=O)Nc1nc2ccccc2s1)c1ccc(OC)cc1 ZINC000217653004 FI On-Demand Unstable LUCI_PHOPE 28 43 CC[C@@H](N[C@H](C)C(=O)Nc1nc2ccccc2s1)c1ccc(OC)cc1 ZINC000217653004 FI On-Demand Unstable FABK 0 43 CC[C@@H](N[C@H](C)C(=O)Nc1nc2ccccc2s1)c1ccc(OC)cc1 ZINC000217653004 FI On-Demand Unstable ISPD 0 46 CC[C@@H](N[C@H](C)C(=O)Nc1nc2ccccc2s1)c1ccc(OC)cc1 ZINC000217653004 FI On-Demand Unstable GPR88 0 44 CC[C@H](N[C@H](C)C(=O)Nc1nc2ccccc2s1)c1ccc(OC)cc1 ZINC000217653081 FI On-Demand Unstable ACE 0 48 CC[C@H](N[C@H](C)C(=O)Nc1nc2ccccc2s1)c1ccc(OC)cc1 ZINC000217653081 FI On-Demand Unstable CSNK1D 42 45 CC[C@H](N[C@H](C)C(=O)Nc1nc2ccccc2s1)c1ccc(OC)cc1 ZINC000217653081 FI On-Demand Unstable PIK3CA 0 40 CC[C@H](N[C@H](C)C(=O)Nc1nc2ccccc2s1)c1ccc(OC)cc1 ZINC000217653081 FI On-Demand Unstable TACR3 45 39 CC[C@H](N[C@H](C)C(=O)Nc1nc2ccccc2s1)c1ccc(OC)cc1 ZINC000217653081 FI On-Demand Unstable LUCI_PHOPE 28 43 CC[C@H](N[C@H](C)C(=O)Nc1nc2ccccc2s1)c1ccc(OC)cc1 ZINC000217653081 FI On-Demand Unstable FABK 0 43 CC[C@H](N[C@H](C)C(=O)Nc1nc2ccccc2s1)c1ccc(OC)cc1 ZINC000217653081 FI On-Demand Unstable ISPD 0 46 CC[C@H](N[C@H](C)C(=O)Nc1nc2ccccc2s1)c1ccc(OC)cc1 ZINC000217653081 FI On-Demand Unstable GPR88 0 44 COCCNc1ccc(S(=O)(=O)NCCC(C)C)cc1C(=O)O ZINC000217653088 ED In-Stock Unstable CASP3 16 42 COCCNc1ccc(S(=O)(=O)NCCC(C)C)cc1C(=O)O ZINC000217653088 ED In-Stock Unstable BDKRB1 17 44 O=C(C1CCC1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217653093 CF In-Stock Unstable PREP 28 51 O=C(C1CCC1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217653093 CF In-Stock Unstable L3MBTL3 46 35 COc1ccccc1CCNC(=O)N/C=C/c1ccccc1 ZINC000217653110 CG For-Sale Unstable MTNR1A 57 43 COc1ccccc1CCNC(=O)N/C=C/c1ccccc1 ZINC000217653110 CG For-Sale Unstable MTNR1B 44 43 O=C(NC[C@@H]1CCCCO1)C1CCN(C(=O)c2ccccc2Cl)CC1 ZINC000217653162 FF In-Stock Unstable EPHX2 30 58 O=C(NC[C@@H]1CCCCO1)C1CCN(C(=O)c2ccccc2Cl)CC1 ZINC000217653162 FF In-Stock Unstable L3MBTL1 0 42 O=C(NC[C@@H]1CCCCO1)C1CCN(C(=O)c2ccccc2Cl)CC1 ZINC000217653162 FF In-Stock Unstable L3MBTL3 58 37 O=C(NC[C@@H]1CCCCO1)C1CCN(C(=O)c2ccccc2Cl)CC1 ZINC000217653162 FF In-Stock Unstable TP53BP1 0 42 O=C(C1CCC1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217653170 CF In-Stock Unstable PREP 28 51 O=C(C1CCC1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217653170 CF In-Stock Unstable L3MBTL3 46 35 COCCCNc1ccc(S(=O)(=O)NCCC(C)C)cc1C(=O)O ZINC000217653198 FE In-Stock Unstable CASP3 0 40 O=C(N/C=C/c1ccccc1)NCCc1ccccc1F ZINC000217653225 CG For-Sale Unstable MTNR1A 19 40 CCCN(CC)CCNCc1ccc2c(c1)OCO2 ZINC000217653235 CE For-Sale Unstable NOS2 60 48 COc1ccc(CCNC(=O)[C@@H](NC(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)C(C)C)cc1 ZINC000217653241 JE In-Stock Unstable CHRNA4 27 47 O=C(NC[C@H]1CCCCO1)C1CCN(C(=O)c2ccccc2Cl)CC1 ZINC000217653245 FF In-Stock Unstable EPHX2 30 58 O=C(NC[C@H]1CCCCO1)C1CCN(C(=O)c2ccccc2Cl)CC1 ZINC000217653245 FF In-Stock Unstable L3MBTL1 0 42 O=C(NC[C@H]1CCCCO1)C1CCN(C(=O)c2ccccc2Cl)CC1 ZINC000217653245 FF In-Stock Unstable L3MBTL3 58 37 O=C(NC[C@H]1CCCCO1)C1CCN(C(=O)c2ccccc2Cl)CC1 ZINC000217653245 FF In-Stock Unstable TP53BP1 0 42 CC(C)(C)C(=O)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217653275 CF In-Stock Unstable PREP 24 44 CC(C)CCNS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217653315 GG In-Stock Unstable CASP3 20 42 COC(=O)c1cc(Cl)c([N+](=O)[O-])[nH]1 ZINC000217653340 BD In-Stock Unstable CACNA1D 73 38 CC(C)(C)C(=O)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217653344 CF In-Stock Unstable PREP 24 44 CC(C)CCNS(=O)(=O)c1ccc(N[C@@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217653444 GH In-Stock Unstable CASP3 19 41 C[C@@H](c1ccc(Br)cc1F)N1CCC[C@@H](CC(=O)O)C1 ZINC000217653447 EH For-Sale Unstable GHSR 21 41 O=C(N/C=C/c1ccccc1)NCCc1ccccc1Br ZINC000217653451 EH For-Sale Unstable CA9 15 40 O=C(c1cccnc1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217653459 DE In-Stock Unstable PREP 18 45 O=C(c1cccnc1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217653459 DE In-Stock Unstable SMO 38 42 O=C(c1cccnc1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217653459 DE In-Stock Unstable L3MBTL3 44 35 C[C@H](c1ccc(Br)cc1F)N1CCC[C@@H](CC(=O)O)C1 ZINC000217653536 EH For-Sale Unstable GHSR 21 41 O=C(c1cccnc1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217653540 DE In-Stock Unstable PREP 18 45 O=C(c1cccnc1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217653540 DE In-Stock Unstable SMO 38 42 O=C(c1cccnc1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217653540 DE In-Stock Unstable L3MBTL3 44 35 CC(C)CCNS(=O)(=O)c1ccc(N[C@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217653541 GH In-Stock Unstable CASP3 19 41 COc1ccc2[nH]cc(CCNC(=O)Cn3ccc4c(NS(C)(=O)=O)cccc43)c2c1 ZINC000217653562 IF In-Stock Unstable HTR1D 26 41 COc1ccc2[nH]cc(CCNC(=O)Cn3ccc4c(NS(C)(=O)=O)cccc43)c2c1 ZINC000217653562 IF In-Stock Unstable HTR1B 33 41 COc1ccc2[nH]cc(CCNC(=O)Cn3ccc4c(NS(C)(=O)=O)cccc43)c2c1 ZINC000217653562 IF In-Stock Unstable NQO2 34 54 COc1ccc2[nH]cc(CCNC(=O)Cn3ccc4c(NS(C)(=O)=O)cccc43)c2c1 ZINC000217653562 IF In-Stock Unstable MTNR1A 96 57 COc1ccc2[nH]cc(CCNC(=O)Cn3ccc4c(NS(C)(=O)=O)cccc43)c2c1 ZINC000217653562 IF In-Stock Unstable MTNR1B 72 54 COc1ccc2[nH]cc(CCNC(=O)Cn3ccc4c(NS(C)(=O)=O)cccc43)c2c1 ZINC000217653562 IF In-Stock Unstable ABCG2 25 41 Cc1cccc(CCNC(=O)N/C=C/c2ccccc2)c1 ZINC000217653570 CH For-Sale Unstable ANPEP 18 40 Cc1cccc(CCNC(=O)N/C=C/c2ccccc2)c1 ZINC000217653570 CH For-Sale Unstable CPA1 15 41 Cc1cccc(CCNC(=O)N/C=C/c2ccccc2)c1 ZINC000217653570 CH For-Sale Unstable HDAC8 43 40 Cc1cccc(CCNC(=O)N/C=C/c2ccccc2)c1 ZINC000217653570 CH For-Sale Unstable MMP2 18 55 Cc1cccc(CCNC(=O)N/C=C/c2ccccc2)c1 ZINC000217653570 CH For-Sale Unstable HDAC1 21 40 Cc1cccc(CCNC(=O)N/C=C/c2ccccc2)c1 ZINC000217653570 CH For-Sale Unstable HDAC6 31 43 Cc1cccc(CCNC(=O)N/C=C/c2ccccc2)c1 ZINC000217653570 CH For-Sale Unstable FBP1 15 40 Cc1cccc(CCNC(=O)N/C=C/c2ccccc2)c1 ZINC000217653570 CH For-Sale Unstable AMP1_PLAFQ 36 40 Cc1cccc(CCNC(=O)N/C=C/c2ccccc2)c1 ZINC000217653570 CH For-Sale Unstable AKR1C3 16 44 C[C@@H](c1cc(Br)ccc1F)N1CCC[C@@H](CC(=O)O)C1 ZINC000217653612 EH For-Sale Unstable GHSR 21 40 CC(C)CCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217653642 GG In-Stock Unstable CA2 15 40 CC(C)CCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217653642 GG In-Stock Unstable TBXA2R 50 39 CC(C)CCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217653642 GG In-Stock Unstable CASP3 18 41 CC(C)CCNS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217653642 GG In-Stock Unstable MMP3 17 41 O=C(c1ccccn1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217653652 DE In-Stock Unstable PREP 16 42 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(OC)c(OC)c2)CC(=O)O4)cc1O ZINC000217653672 JI In-Stock Unstable AKR1B1 24 52 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(OC)c(OC)c2)CC(=O)O4)cc1O ZINC000217653672 JI In-Stock Unstable CYP1B1 69 39 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(OC)c(OC)c2)CC(=O)O4)cc1O ZINC000217653672 JI In-Stock Unstable CYP1A1 51 50 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(OC)c(OC)c2)CC(=O)O4)cc1O ZINC000217653672 JI In-Stock Unstable CYP1A2 41 47 COc1cccc(CCNC(=O)N/C=C/c2ccccc2)c1 ZINC000217653683 CG For-Sale Unstable DRD4 41 32 COc1cccc(CCNC(=O)N/C=C/c2ccccc2)c1 ZINC000217653683 CG For-Sale Unstable HRH2 26 40 COc1cccc(CCNC(=O)N/C=C/c2ccccc2)c1 ZINC000217653683 CG For-Sale Unstable NQO2 29 41 COc1cccc(CCNC(=O)N/C=C/c2ccccc2)c1 ZINC000217653683 CG For-Sale Unstable G6PC 23 40 COc1cccc(CCNC(=O)N/C=C/c2ccccc2)c1 ZINC000217653683 CG For-Sale Unstable MMP13 21 41 COc1cccc(CCNC(=O)N/C=C/c2ccccc2)c1 ZINC000217653683 CG For-Sale Unstable HDAC8 22 40 COc1cccc(CCNC(=O)N/C=C/c2ccccc2)c1 ZINC000217653683 CG For-Sale Unstable MTNR1A 114 55 COc1cccc(CCNC(=O)N/C=C/c2ccccc2)c1 ZINC000217653683 CG For-Sale Unstable MTNR1B 104 55 COc1cccc(CCNC(=O)N/C=C/c2ccccc2)c1 ZINC000217653683 CG For-Sale Unstable MMP2 17 47 COc1cccc(CCNC(=O)N/C=C/c2ccccc2)c1 ZINC000217653683 CG For-Sale Unstable ABCB1 17 40 COc1cccc(CCNC(=O)N/C=C/c2ccccc2)c1 ZINC000217653683 CG For-Sale Unstable PLM1_PLAFA 31 41 COc1cccc(CCNC(=O)N/C=C/c2ccccc2)c1 ZINC000217653683 CG For-Sale Unstable AMP1_PLAFQ 38 41 COc1cccc(CCNC(=O)N/C=C/c2ccccc2)c1 ZINC000217653683 CG For-Sale Unstable AKR1C3 18 47 COc1cccc(CCNC(=O)N/C=C/c2ccccc2)c1 ZINC000217653683 CG For-Sale Unstable CRTM 59 43 COc1cccc(CCNC(=O)N/C=C/c2ccccc2)c1 ZINC000217653683 CG For-Sale Unstable CRTH2 0 40 COc1cccc(CCNC(=O)N/C=C/c2ccccc2)c1 ZINC000217653683 CG For-Sale Unstable PDS 48 35 O=C(O)/C=C\c1ccc(C(=O)Nc2ccc(Cl)c(Cl)c2)s1 ZINC000217653687 EI For-Sale Anodyne MAOB 18 41 O=C(O)/C=C\c1ccc(C(=O)Nc2ccc(Cl)c(Cl)c2)s1 ZINC000217653687 EI For-Sale Anodyne MURB 0 41 O=C(O)/C=C\c1ccc(C(=O)Nc2ccc(Cl)c(Cl)c2)s1 ZINC000217653687 EI For-Sale Anodyne SHH 43 36 O=C(O)/C=C\c1ccc(C(=O)Nc2ccc(Cl)c(Cl)c2)s1 ZINC000217653687 EI For-Sale Anodyne P95276_MYCTO 0 41 O=C(O)/C=C\c1ccc(C(=O)Nc2ccc(Cl)c(Cl)c2)s1 ZINC000217653687 EI For-Sale Anodyne USP47 41 32 O=C(O)/C=C\c1ccc(C(=O)Nc2ccc(Cl)c(Cl)c2)s1 ZINC000217653687 EI For-Sale Anodyne PPX1 0 40 C[C@H](c1cc(Br)ccc1F)N1CCC[C@@H](CC(=O)O)C1 ZINC000217653693 EH For-Sale Unstable GHSR 21 40 COc1ccc(CCNc2ccc(S(=O)(=O)NCCC(C)C)cc2C(=O)O)cc1 ZINC000217653747 HG In-Stock Unstable TBXA2R 38 42 COc1ccc(CCNc2ccc(S(=O)(=O)NCCC(C)C)cc2C(=O)O)cc1 ZINC000217653747 HG In-Stock Unstable TBXAS1 20 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCCC(C)C)cc2C(=O)O)cc1 ZINC000217653747 HG In-Stock Unstable BMP1 87 37 COc1ccc(CCNc2ccc(S(=O)(=O)NCCC(C)C)cc2C(=O)O)cc1 ZINC000217653747 HG In-Stock Unstable CA1 15 43 COc1ccc(CCNc2ccc(S(=O)(=O)NCCC(C)C)cc2C(=O)O)cc1 ZINC000217653747 HG In-Stock Unstable MMP13 58 40 COc1ccc(CCNc2ccc(S(=O)(=O)NCCC(C)C)cc2C(=O)O)cc1 ZINC000217653747 HG In-Stock Unstable MMP2 39 40 COc1ccc(CCNc2ccc(S(=O)(=O)NCCC(C)C)cc2C(=O)O)cc1 ZINC000217653747 HG In-Stock Unstable MMP3 49 45 COc1ccc(CCNc2ccc(S(=O)(=O)NCCC(C)C)cc2C(=O)O)cc1 ZINC000217653747 HG In-Stock Unstable MMP9 47 40 COc1ccc(CCNc2ccc(S(=O)(=O)NCCC(C)C)cc2C(=O)O)cc1 ZINC000217653747 HG In-Stock Unstable PTGDR 27 41 COc1ccc(CCNc2ccc(S(=O)(=O)NCCC(C)C)cc2C(=O)O)cc1 ZINC000217653747 HG In-Stock Unstable IAP 0 44 COc1ccc(CCNc2ccc(S(=O)(=O)NCCC(C)C)cc2C(=O)O)cc1 ZINC000217653747 HG In-Stock Unstable CA9 23 42 COc1ccc(CCNc2ccc(S(=O)(=O)NCCC(C)C)cc2C(=O)O)cc1 ZINC000217653747 HG In-Stock Unstable MMP1 49 37 COc1ccc(CCNc2ccc(S(=O)(=O)NCCC(C)C)cc2C(=O)O)cc1 ZINC000217653747 HG In-Stock Unstable AKR1C3 29 45 COc1ccc(CCNc2ccc(S(=O)(=O)NCCC(C)C)cc2C(=O)O)cc1 ZINC000217653747 HG In-Stock Unstable AKR1C2 46 36 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(OC)c(OC)c2)CC(=O)O4)cc1O ZINC000217653750 JI In-Stock Unstable AKR1B1 24 52 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(OC)c(OC)c2)CC(=O)O4)cc1O ZINC000217653750 JI In-Stock Unstable CYP1B1 69 39 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(OC)c(OC)c2)CC(=O)O4)cc1O ZINC000217653750 JI In-Stock Unstable CYP1A1 51 50 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(OC)c(OC)c2)CC(=O)O4)cc1O ZINC000217653750 JI In-Stock Unstable CYP1A2 41 47 O=C(c1ccccn1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217653755 DE In-Stock Unstable PREP 16 42 CN(Cc1ccccc1)C(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217653770 DG For-Sale Unstable PTGER2 35 44 CN(Cc1ccccc1)C(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217653770 DG For-Sale Unstable PTGER4 0 44 CN(Cc1ccccc1)C(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217653770 DG For-Sale Unstable TSPO 16 42 CN(Cc1ccccc1)C(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217653770 DG For-Sale Unstable HSP90AB1 39 40 CN(Cc1ccccc1)C(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217653770 DG For-Sale Unstable HSD17B2 49 61 CN(Cc1ccccc1)C(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217653770 DG For-Sale Unstable LIMK2 36 40 O=C(NCCO)c1cc(I)c[nH]1 ZINC000217653782 CC In-Stock Unstable ALPL 41 40 O=C(N/C=C/c1ccccc1)NCCc1cccc(F)c1 ZINC000217653807 CG For-Sale Unstable CPA1 21 40 COc1ccc(CCNc2ccc(S(=O)(=O)NCCC(C)C)cc2C(=O)O)cc1OC ZINC000217653847 JG In-Stock Unstable IAP 0 45 COc1ccc(CCNc2ccc(S(=O)(=O)NCCC(C)C)cc2C(=O)O)cc1OC ZINC000217653847 JG In-Stock Unstable SCMU_MYCTU 0 44 O=C(O)/C=C\c1cccc(C(=O)N2CCC(O)CC2)c1 ZINC000217653856 CD For-Sale Unstable L3MBTL3 74 47 NC/C=C\COc1ccc(Br)cc1 ZINC000217653917 BE For-Sale Unstable SHC 37 43 O=C(N/C=C/c1ccccc1)NCCc1cccc(Cl)c1 ZINC000217653927 DH For-Sale Unstable SLC6A5 30 42 O=C(N/C=C/c1ccccc1)NCCc1cccc(Cl)c1 ZINC000217653927 DH For-Sale Unstable AMP1_PLAFQ 30 41 O=C(N/C=C/c1ccccc1)NCCc1cccc(Cl)c1 ZINC000217653927 DH For-Sale Unstable NCE103 22 40 O=C(O)/C=C\c1ccc(F)c(C(=O)N2CCC(O)CC2)c1 ZINC000217653933 CD For-Sale Unstable CCR2 70 41 COc1ccc(N2CCN(C(=O)C(F)F)CC2)cc1 ZINC000217653992 CD On-Demand Unstable CCKAR 26 40 COc1ccc(N2CCN(C(=O)C(F)F)CC2)cc1 ZINC000217653992 CD On-Demand Unstable MMP3 15 41 COc1ccc(N2CCN(C(=O)C(F)F)CC2)cc1 ZINC000217653992 CD On-Demand Unstable SLC6A9 0 45 COc1ccc(N2CCN(C(=O)C(F)F)CC2)cc1 ZINC000217653992 CD On-Demand Unstable AKR1C3 0 40 COc1cc(CN2C[C@H]3[C@@H](C2)[C@@H]3C(=O)O)cc2c1OCO2 ZINC000217653999 CD In-Stock Unstable EDNRB 45 39 COc1cc(CN2C[C@H]3[C@@H](C2)[C@@H]3C(=O)O)cc2c1OCO2 ZINC000217653999 CD In-Stock Unstable EDNRA 42 42 COc1cc(CN2C[C@H]3[C@@H](C2)[C@@H]3C(=O)O)cc2c1OCO2 ZINC000217653999 CD In-Stock Unstable ERCC5 16 48 O=C(O)/C=C\c1ccc(C(=O)N2CCC(O)CC2)c(F)c1 ZINC000217654015 CD For-Sale Unstable CCR2 73 41 COc1ccc2cc(C(=O)NC[C@@H]3CCCN4CCCC[C@H]34)[nH]c2c1 ZINC000217654033 EG In-Stock Unstable MTNR1A 44 36 O=C(N/C=C/c1ccccc1)NCCc1cccc(Br)c1 ZINC000217654046 EH For-Sale Unstable HDAC8 20 45 O=C(N/C=C/c1ccccc1)NCCc1cccc(Br)c1 ZINC000217654046 EH For-Sale Unstable HDAC6 16 45 O=C(N/C=C/c1ccccc1)NCCc1cccc(Br)c1 ZINC000217654046 EH For-Sale Unstable AMP1_PLAFQ 40 39 O=C(c1ccsc1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217654061 DG In-Stock Unstable PREP 17 43 O=C(c1ccsc1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217654061 DG In-Stock Unstable L3MBTL3 40 35 Cc1nc2ccc(NC(=O)C(F)F)cc2s1 ZINC000217654112 BF On-Demand Unstable LDHA 43 48 Cc1nc2ccc(NC(=O)C(F)F)cc2s1 ZINC000217654112 BF On-Demand Unstable PRMT3 59 33 O=C(c1ccsc1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217654133 DG In-Stock Unstable PREP 17 43 O=C(c1ccsc1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217654133 DG In-Stock Unstable L3MBTL3 40 35 Cc1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217654159 CH For-Sale Unstable HDAC8 15 43 Cc1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217654159 CH For-Sale Unstable MMP2 27 42 Cc1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217654159 CH For-Sale Unstable MMP3 18 43 Cc1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217654159 CH For-Sale Unstable SCN5A 0 46 Cc1ccc(CCNC(=O)N/C=C/c2ccccc2)cc1 ZINC000217654159 CH For-Sale Unstable AMP1_PLAFQ 29 42 Cc1cc(C(=O)NC[C@@H]2CCCN3CCCC[C@H]23)c2cc(F)ccc2n1 ZINC000217654163 FH In-Stock Unstable PREP 22 45 Cc1cc(C(=O)NC[C@@H]2CCCN3CCCC[C@H]23)c2cc(F)ccc2n1 ZINC000217654163 FH In-Stock Unstable FAP 0 45 Cc1cc(Br)c([C@@H](N)C(=O)O)s1 ZINC000217654227 CD For-Sale Unstable CACNA2D1 16 43 CSc1nc2ccc(NC(=O)C(F)F)cc2s1 ZINC000217654233 CG On-Demand Unstable LDHA 42 39 CSc1nc2ccc(NC(=O)C(F)F)cc2s1 ZINC000217654233 CG On-Demand Unstable PPXI 60 40 COc1ccc([N+](=O)[O-])cc1C(=O)NC[C@@](C)(O)CSC ZINC000217654240 DD On-Demand Unstable KCNMA1 25 43 Cn1cccc1CNC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217654256 GD In-Stock Unstable EDNRA 0 41 Cn1cccc1CNC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217654256 GD In-Stock Unstable CCKAR 22 42 O=C(N/C=C/c1ccccc1)NCCc1ccc(Cl)cc1 ZINC000217654269 DH For-Sale Unstable MMP2 35 42 O=C(N/C=C/c1ccccc1)NCCc1ccc(Cl)cc1 ZINC000217654269 DH For-Sale Unstable SLC6A5 20 40 O=C(N/C=C/c1ccccc1)NCCc1ccc(Cl)cc1 ZINC000217654269 DH For-Sale Unstable AMP1_PLAFQ 34 40 O=C(N/C=C/c1ccccc1)NCCc1ccc(Cl)cc1 ZINC000217654269 DH For-Sale Unstable NCE103 23 42 CC(C)CCNS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217654297 EE In-Stock Unstable CASP3 17 43 CC(C)CCNS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217654297 EE In-Stock Unstable KCNQ2 71 36 CC(C)CCNS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217654297 EE In-Stock Unstable SFRP1 47 33 COc1ccc([N+](=O)[O-])cc1C(=O)NC[C@](C)(O)CSC ZINC000217654324 DD On-Demand Unstable KCNMA1 25 43 CC(C)(C)OC(=O)N1CCC[C@@H]1Br ZINC000217654349 CF For-Sale Unstable PREP 18 58 CCOc1ccc(CCNC(=O)C(F)F)cc1OCC ZINC000217654367 CE On-Demand Unstable LEF 44 35 COc1ccc([C@@H]2CC(=O)Oc3ccc4c(c32)OC(=C(C)C)C4=O)c(OC)c1 ZINC000217654375 GI In-Stock Unstable MT-ND4 52 33 O=C(N/C=C/c1ccccc1)NCCc1ccc(Br)cc1 ZINC000217654376 EH For-Sale Unstable HDAC8 22 46 O=C(N/C=C/c1ccccc1)NCCc1ccc(Br)cc1 ZINC000217654376 EH For-Sale Unstable MMP2 17 53 O=C(N/C=C/c1ccccc1)NCCc1ccc(Br)cc1 ZINC000217654376 EH For-Sale Unstable HDAC6 15 46 O=C(N/C=C/c1ccccc1)NCCc1ccc(Br)cc1 ZINC000217654376 EH For-Sale Unstable AMP1_PLAFQ 35 42 O=C(N/C=C/c1ccccc1)NCCc1ccc(Br)cc1 ZINC000217654376 EH For-Sale Unstable LIG1 0 41 Cc1csc(NC(=O)c2cccc(/C=C\C(=O)O)c2)n1 ZINC000217654395 CF For-Sale Unstable MPL 48 36 Cc1csc(NC(=O)c2cccc(/C=C\C(=O)O)c2)n1 ZINC000217654395 CF For-Sale Unstable HDAC8 36 44 Cc1csc(NC(=O)c2cccc(/C=C\C(=O)O)c2)n1 ZINC000217654395 CF For-Sale Unstable HDAC6 24 44 Cc1csc(NC(=O)c2cccc(/C=C\C(=O)O)c2)n1 ZINC000217654395 CF For-Sale Unstable GCK 25 62 Cc1csc(NC(=O)c2cccc(/C=C\C(=O)O)c2)n1 ZINC000217654395 CF For-Sale Unstable KCNK3 89 40 Cc1csc(NC(=O)c2cccc(/C=C\C(=O)O)c2)n1 ZINC000217654395 CF For-Sale Unstable KCNK9 48 40 CC(C)CCNS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217654398 FF In-Stock Unstable CASP3 16 42 CC(C)CCNS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217654398 FF In-Stock Unstable KCNQ2 67 36 O=C(CCCN1CCC[C@@H]2CCCC[C@H]21)c1ccccc1 ZINC000217654402 CI On-Demand Unstable HTR2A 15 45 O=C(CCCN1CCC[C@@H]2CCCC[C@H]21)c1ccccc1 ZINC000217654402 CI On-Demand Unstable HTR2C 16 47 O=C(CCCN1CCC[C@@H]2CCCC[C@H]21)c1ccccc1 ZINC000217654402 CI On-Demand Unstable SLC6A1 75 41 O=C(CCCN1CCC[C@@H]2CCCC[C@H]21)c1ccccc1 ZINC000217654402 CI On-Demand Unstable HRH3 24 40 O=C(CCCN1CCC[C@@H]2CCCC[C@H]21)c1ccccc1 ZINC000217654402 CI On-Demand Unstable PREP 40 45 O=C(CCCN1CCC[C@@H]2CCCC[C@H]21)c1ccccc1 ZINC000217654402 CI On-Demand Unstable CYP2J2 59 42 COc1ccc(F)cc1CN1CCN(C(=O)NCCN(C)c2ccccc2)CC1 ZINC000217654417 HF On-Demand Unstable DRD4 30 42 COc1ccc(F)cc1CN1CCN(C(=O)NCCN(C)c2ccccc2)CC1 ZINC000217654417 HF On-Demand Unstable DRD3 45 39 COc1ccc(F)cc1CN1CCN(C(=O)NCCN(C)c2ccccc2)CC1 ZINC000217654417 HF On-Demand Unstable TACR1 25 40 COc1ccc(F)cc1CN1CCN(C(=O)NCCN(C)c2ccccc2)CC1 ZINC000217654417 HF On-Demand Unstable ACKR3 50 31 O=C(c1ccccc1F)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217654420 EG In-Stock Unstable PREP 15 42 CC(C)(C)OC(=O)N1CCC[C@H]1Br ZINC000217654433 CF For-Sale Unstable PREP 18 58 CSC[C@@](C)(O)CNC(=O)c1ccnc2ccccc12 ZINC000217654437 CE On-Demand Unstable PREP 28 44 CSC[C@@](C)(O)CNC(=O)c1ccnc2ccccc12 ZINC000217654437 CE On-Demand Unstable FAP 0 52 COc1ccc([C@H]2CC(=O)Oc3ccc4c(c32)OC(=C(C)C)C4=O)c(OC)c1 ZINC000217654454 GI In-Stock Unstable MT-ND4 52 33 O=C(CCCN1CCC[C@H]2CCCC[C@H]21)c1ccccc1 ZINC000217654484 CI On-Demand Unstable HTR2A 15 45 O=C(CCCN1CCC[C@H]2CCCC[C@H]21)c1ccccc1 ZINC000217654484 CI On-Demand Unstable HTR2C 16 47 O=C(CCCN1CCC[C@H]2CCCC[C@H]21)c1ccccc1 ZINC000217654484 CI On-Demand Unstable SLC6A1 75 41 O=C(CCCN1CCC[C@H]2CCCC[C@H]21)c1ccccc1 ZINC000217654484 CI On-Demand Unstable HRH3 24 40 O=C(CCCN1CCC[C@H]2CCCC[C@H]21)c1ccccc1 ZINC000217654484 CI On-Demand Unstable PREP 40 45 O=C(CCCN1CCC[C@H]2CCCC[C@H]21)c1ccccc1 ZINC000217654484 CI On-Demand Unstable CYP2J2 59 42 Cc1csc(NC(=O)c2cc(/C=C\C(=O)O)ccc2F)n1 ZINC000217654485 DF For-Sale Unstable GCK 21 47 CS(=O)(=O)c1ccc(Cl)c(NC(=O)C(F)F)c1 ZINC000217654486 CD On-Demand Unstable PTGS2 22 43 O=C(c1ccccc1F)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217654496 EG In-Stock Unstable PREP 15 42 CC(C)CCNS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1 ZINC000217654505 FD In-Stock Unstable SLC6A9 20 46 CSC[C@](C)(O)CNC(=O)c1ccnc2ccccc12 ZINC000217654509 CE On-Demand Unstable PREP 28 44 CSC[C@](C)(O)CNC(=O)c1ccnc2ccccc12 ZINC000217654509 CE On-Demand Unstable FAP 0 52 C[C@@H](N[C@@H]1CCC[C@@H](C(=O)O)C1)c1cc(Br)ccc1F ZINC000217654538 EH For-Sale Unstable SDH1 0 42 C[C@@H](NC(=O)NCCN(C)c1ccccc1)c1ccc(Br)cc1 ZINC000217654546 GH On-Demand Unstable SDH1 0 41 Cc1ccc(NC(=O)N/C=C/c2ccccc2)nc1 ZINC000217654589 CG For-Sale Unstable LUCI_LUCLA 40 42 CN1CCCN(C(=O)c2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217654595 CD For-Sale Unstable HRH4 25 42 CN1CCCN(C(=O)c2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217654595 CD For-Sale Unstable MLYCD 17 40 CN1CCCN(C(=O)c2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217654595 CD For-Sale Unstable L3MBTL3 56 45 CCOCCCNc1ccc(S(=O)(=O)NCCC(C)C)cc1C(=O)O ZINC000217654620 FF In-Stock Unstable CASP3 15 43 CCOCCCNc1ccc(S(=O)(=O)NCCC(C)C)cc1C(=O)O ZINC000217654620 FF In-Stock Unstable BDKRB1 16 41 C[C@H](NC(=O)NCCN(C)c1ccccc1)c1ccc(Br)cc1 ZINC000217654628 GH On-Demand Unstable SDH1 0 41 C[C@@H]1CN(C[C@@H]2NCCc3ccccc32)CCCO1 ZINC000217654629 CD For-Sale Unstable PRCP 47 45 C[C@H](N[C@@H]1CCC[C@@H](C(=O)O)C1)c1cc(Br)ccc1F ZINC000217654634 EH For-Sale Unstable SDH1 0 42 O=C1CC[C@@H](O)[C@@H](CO)O1 ZINC000217654677 AB For-Sale Unstable CDA 62 33 CN1CCCN(C(=O)c2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217654717 CD For-Sale Unstable HRH4 26 44 CN1CCCN(C(=O)c2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217654717 CD For-Sale Unstable PIM2 15 53 C[C@H]1CN(C[C@@H]2NCCc3ccccc32)CCCO1 ZINC000217654726 CD For-Sale Unstable PRCP 47 45 CC(C)CCNS(=O)(=O)c1ccc(NCCCOC(C)C)c(C(=O)O)c1 ZINC000217654727 GF In-Stock Unstable CASP3 15 42 O=C1CC[C@@H](O)[C@H](CO)O1 ZINC000217654750 AB For-Sale Unstable CDA 62 33 COc1ccc(OC/C=C\CN)c([N+](=O)[O-])c1 ZINC000217654821 BD For-Sale Unstable TPPP 0 47 CSC[C@@](C)(O)CNC(=O)CSCc1ccc(F)cc1 ZINC000217654826 DE On-Demand Unstable LTA4H 24 40 CCCCCNc1ccc(S(=O)(=O)NCCC(C)C)cc1C(=O)O ZINC000217654830 FG In-Stock Unstable CASP3 16 46 O=C1CC[C@H](O)[C@@H](CO)O1 ZINC000217654833 AB For-Sale Unstable CDA 62 33 C[C@H](N[C@H]1CCC[C@@H](C(=O)O)C1)c1cc(Br)ccc1F ZINC000217654835 EH For-Sale Unstable SDH1 0 42 CN(CCNC(=O)NC1CCCCCC1)c1ccccc1 ZINC000217654852 CG On-Demand Unstable CNR1 15 41 CN(CCNC(=O)NC1CCCCCC1)c1ccccc1 ZINC000217654852 CG On-Demand Unstable CNR2 20 41 CN(CCNC(=O)NC1CCCCCC1)c1ccccc1 ZINC000217654852 CG On-Demand Unstable AMY2 50 36 CN(CCNC(=O)NC1CCCCCC1)c1ccccc1 ZINC000217654852 CG On-Demand Unstable EPHX2 35 50 COC1CCN(C(=O)c2ccc(/C=C\C(=O)O)s2)CC1 ZINC000217654875 CE For-Sale Unstable L3MBTL3 17 44 CSC[C@](C)(O)CNC(=O)CSCc1ccc(F)cc1 ZINC000217654905 DE On-Demand Unstable LTA4H 24 40 O=C(N/C=C/c1ccccc1)Nc1ccc(Cl)cn1 ZINC000217654924 CH For-Sale Anodyne F10 39 40 O=C(N/C=C/c1ccccc1)Nc1ccc(Cl)cn1 ZINC000217654924 CH For-Sale Anodyne LUCI_LUCLA 35 46 C[C@@H](c1ccc(Br)cc1F)N1CC[C@@H](C(=O)O)C1 ZINC000217654925 DG For-Sale Unstable SLC6A1 43 34 CC(C)CCNc1ccc(S(=O)(=O)NCCC(C)C)cc1C(=O)O ZINC000217654931 FG In-Stock Unstable CASP3 17 45 COC1CCN(C(=O)c2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217654963 CE For-Sale Unstable L3MBTL3 84 41 CN(CCNC(=O)NCCNc1ccccc1[N+](=O)[O-])c1ccccc1 ZINC000217654970 FE On-Demand Unstable COLA 67 32 C[C@H](c1ccc(Br)cc1F)N1CC[C@@H](C(=O)O)C1 ZINC000217655003 DG For-Sale Unstable SLC6A1 43 34 N#Cc1cccc(C(=O)N2CC[C@@H](n3cc(-c4ccccc4)nn3)C2)c1 ZINC000217655014 EF In-Stock Unstable ABHD6 0 42 N#Cc1cccc(C(=O)N2CC[C@@H](n3cc(-c4ccccc4)nn3)C2)c1 ZINC000217655014 EF In-Stock Unstable MAP3K12 29 40 CC[C@@H]1CC[C@@H](NC)[C@@H](Cc2cccc(C(F)(F)F)c2)C1 ZINC000217655021 CJ For-Sale Unstable PDS 19 41 NC/C=C\COc1ccc(Cl)cc1[N+](=O)[O-] ZINC000217655037 BE For-Sale Unstable PDE7B 0 41 NC/C=C\COc1ccc(Cl)cc1[N+](=O)[O-] ZINC000217655037 BE For-Sale Unstable S1PR4 0 49 NC/C=C\COc1ccc(Cl)cc1[N+](=O)[O-] ZINC000217655037 BE For-Sale Unstable PDE7A 0 53 NC/C=C\COc1ccc(Cl)cc1[N+](=O)[O-] ZINC000217655037 BE For-Sale Unstable ENR 0 40 O=C(N/C=C/c1ccccc1)Nc1cc(Cl)ccn1 ZINC000217655040 CH For-Sale Anodyne TYK2 61 36 CCC[C@@H](C)Nc1ccc(S(=O)(=O)NCCC(C)C)cc1C(=O)O ZINC000217655049 FG In-Stock Unstable CASP3 15 43 COC1CCN(C(=O)c2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217655051 CE For-Sale Unstable L3MBTL3 54 43 N#Cc1cccc(C(=O)N2CC[C@H](n3cc(-c4ccccc4)nn3)C2)c1 ZINC000217655091 EF In-Stock Unstable ABHD6 0 42 N#Cc1cccc(C(=O)N2CC[C@H](n3cc(-c4ccccc4)nn3)C2)c1 ZINC000217655091 EF In-Stock Unstable MAP3K12 29 40 COc1cc(Nc2ncc(Br)cn2)ccc1N1CCC(N2CCN(C)CC2)CC1 ZINC000217655098 JG For-Sale Unstable LCK 15 42 COc1cc(Nc2ncc(Br)cn2)ccc1N1CCC(N2CCN(C)CC2)CC1 ZINC000217655098 JG For-Sale Unstable CCR4 40 42 COc1cc(Nc2ncc(Br)cn2)ccc1N1CCC(N2CCN(C)CC2)CC1 ZINC000217655098 JG For-Sale Unstable JAK2 23 44 COc1cc(Nc2ncc(Br)cn2)ccc1N1CCC(N2CCN(C)CC2)CC1 ZINC000217655098 JG For-Sale Unstable PAK1 73 47 COc1cc(Nc2ncc(Br)cn2)ccc1N1CCC(N2CCN(C)CC2)CC1 ZINC000217655098 JG For-Sale Unstable TNIK 55 46 COc1cc(Nc2ncc(Br)cn2)ccc1N1CCC(N2CCN(C)CC2)CC1 ZINC000217655098 JG For-Sale Unstable MAPK7 46 43 COc1cc(Nc2ncc(Br)cn2)ccc1N1CCC(N2CCN(C)CC2)CC1 ZINC000217655098 JG For-Sale Unstable STK33 15 44 C[C@@H](c1cc(Br)ccc1F)N1CC[C@@H](C(=O)O)C1 ZINC000217655101 DG For-Sale Unstable SLC6A1 41 34 Oc1ccccc1CN[C@@H]1CCN2CCCC[C@@H]12 ZINC000217655105 BE On-Demand Unstable VACHT_TETCF 0 41 Oc1ccccc1CN[C@@H]1CCN2CCCC[C@@H]12 ZINC000217655105 BE On-Demand Unstable SIGMAR1 15 44 Oc1ccccc1CN[C@@H]1CCN2CCCC[C@@H]12 ZINC000217655105 BE On-Demand Unstable SLC18A3 83 41 O=C(c1cc(Br)c(Br)[nH]1)N1CCNCC1 ZINC000217655107 ED In-Stock Unstable HRH4 31 54 CC[C@H]1CC[C@@H](NC)[C@@H](Cc2cccc(C(F)(F)F)c2)C1 ZINC000217655114 CJ For-Sale Unstable PDS 19 41 CCC[C@H](C)Nc1ccc(S(=O)(=O)NCCC(C)C)cc1C(=O)O ZINC000217655134 FG In-Stock Unstable CASP3 15 43 CN(c1ccccc1)c1cc(Cl)ccc1[N+](=O)[O-] ZINC000217655166 CI For-Sale Unstable PDE7A 19 46 Oc1ccccc1CN[C@H]1CCN2CCCC[C@@H]12 ZINC000217655182 BE On-Demand Unstable VACHT_TETCF 0 41 Oc1ccccc1CN[C@H]1CCN2CCCC[C@@H]12 ZINC000217655182 BE On-Demand Unstable SIGMAR1 15 44 Oc1ccccc1CN[C@H]1CCN2CCCC[C@@H]12 ZINC000217655182 BE On-Demand Unstable SLC18A3 83 41 C[C@H](c1cc(Br)ccc1F)N1CC[C@@H](C(=O)O)C1 ZINC000217655184 DG For-Sale Unstable SLC6A1 41 34 CC[C@@H]1CC[C@H](NC)[C@@H](Cc2cccc(C(F)(F)F)c2)C1 ZINC000217655189 CJ For-Sale Unstable PDS 19 41 O=C(/C=C/c1ccccc1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217655207 EG In-Stock Unstable PREP 23 44 COc1cc(Nc2ncc(I)cn2)ccc1N1CCC(N2CCN(C)CC2)CC1 ZINC000217655210 KG For-Sale Unstable LCK 16 42 COc1cc(Nc2ncc(I)cn2)ccc1N1CCC(N2CCN(C)CC2)CC1 ZINC000217655210 KG For-Sale Unstable CCR4 40 42 COc1cc(Nc2ncc(I)cn2)ccc1N1CCC(N2CCN(C)CC2)CC1 ZINC000217655210 KG For-Sale Unstable JAK2 30 48 COc1cc(Nc2ncc(I)cn2)ccc1N1CCC(N2CCN(C)CC2)CC1 ZINC000217655210 KG For-Sale Unstable PAK1 73 47 COc1cc(Nc2ncc(I)cn2)ccc1N1CCC(N2CCN(C)CC2)CC1 ZINC000217655210 KG For-Sale Unstable TNIK 55 46 COc1cc(Nc2ncc(I)cn2)ccc1N1CCC(N2CCN(C)CC2)CC1 ZINC000217655210 KG For-Sale Unstable MAPK7 46 43 COc1cc(Nc2ncc(I)cn2)ccc1N1CCC(N2CCN(C)CC2)CC1 ZINC000217655210 KG For-Sale Unstable STK33 15 44 N#Cc1c[nH]c(C(=O)N2CCNCC2)c1 ZINC000217655225 BB In-Stock Unstable HRH4 17 44 O=C(N/C=C/c1ccccc1)NCCCc1ccccc1 ZINC000217655265 CH For-Sale Unstable NA 0 44 O=C(N/C=C/c1ccccc1)NCCCc1ccccc1 ZINC000217655265 CH For-Sale Unstable HRH2 22 40 O=C(N/C=C/c1ccccc1)NCCCc1ccccc1 ZINC000217655265 CH For-Sale Unstable SIGMAR1 16 42 O=C(N/C=C/c1ccccc1)NCCCc1ccccc1 ZINC000217655265 CH For-Sale Unstable HDAC8 23 47 O=C(N/C=C/c1ccccc1)NCCCc1ccccc1 ZINC000217655265 CH For-Sale Unstable MTNR1A 24 40 O=C(N/C=C/c1ccccc1)NCCCc1ccccc1 ZINC000217655265 CH For-Sale Unstable MTNR1B 37 40 O=C(N/C=C/c1ccccc1)NCCCc1ccccc1 ZINC000217655265 CH For-Sale Unstable MMP2 19 55 O=C(N/C=C/c1ccccc1)NCCCc1ccccc1 ZINC000217655265 CH For-Sale Unstable HDAC1 23 50 O=C(N/C=C/c1ccccc1)NCCCc1ccccc1 ZINC000217655265 CH For-Sale Unstable HDAC2 15 50 O=C(N/C=C/c1ccccc1)NCCCc1ccccc1 ZINC000217655265 CH For-Sale Unstable HDAC6 19 47 O=C(N/C=C/c1ccccc1)NCCCc1ccccc1 ZINC000217655265 CH For-Sale Unstable FAAH 33 40 O=C(N/C=C/c1ccccc1)NCCCc1ccccc1 ZINC000217655265 CH For-Sale Unstable SCN5A 0 42 O=C(N/C=C/c1ccccc1)NCCCc1ccccc1 ZINC000217655265 CH For-Sale Unstable CES1 41 36 O=C(N/C=C/c1ccccc1)NCCCc1ccccc1 ZINC000217655265 CH For-Sale Unstable AMP1_PLAFQ 45 50 O=C(N/C=C/c1ccccc1)NCCCc1ccccc1 ZINC000217655265 CH For-Sale Unstable CRTM 45 43 CC[C@H]1CC[C@H](NC)[C@@H](Cc2cccc(C(F)(F)F)c2)C1 ZINC000217655270 CJ For-Sale Unstable PDS 19 41 O=C(/C=C/c1ccccc1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217655291 EG In-Stock Unstable PREP 23 44 C[C@H](N[C@@H]1CCN2CCCC[C@@H]12)c1ccc(Br)cc1 ZINC000217655359 DH On-Demand Unstable SDH1 0 45 O=C(N/C=C/c1ccccc1)NCCCCc1ccccc1 ZINC000217655381 CH For-Sale Unstable NA 0 43 O=C(N/C=C/c1ccccc1)NCCCCc1ccccc1 ZINC000217655381 CH For-Sale Unstable MME 22 40 O=C(N/C=C/c1ccccc1)NCCCCc1ccccc1 ZINC000217655381 CH For-Sale Unstable SIGMAR1 18 46 O=C(N/C=C/c1ccccc1)NCCCCc1ccccc1 ZINC000217655381 CH For-Sale Unstable SCN2A 23 42 O=C(N/C=C/c1ccccc1)NCCCCc1ccccc1 ZINC000217655381 CH For-Sale Unstable HDAC8 22 45 O=C(N/C=C/c1ccccc1)NCCCCc1ccccc1 ZINC000217655381 CH For-Sale Unstable MTNR1A 21 40 O=C(N/C=C/c1ccccc1)NCCCCc1ccccc1 ZINC000217655381 CH For-Sale Unstable MTNR1B 36 40 O=C(N/C=C/c1ccccc1)NCCCCc1ccccc1 ZINC000217655381 CH For-Sale Unstable MMP2 19 54 O=C(N/C=C/c1ccccc1)NCCCCc1ccccc1 ZINC000217655381 CH For-Sale Unstable HDAC1 24 49 O=C(N/C=C/c1ccccc1)NCCCCc1ccccc1 ZINC000217655381 CH For-Sale Unstable HDAC2 15 47 O=C(N/C=C/c1ccccc1)NCCCCc1ccccc1 ZINC000217655381 CH For-Sale Unstable HDAC6 19 45 O=C(N/C=C/c1ccccc1)NCCCCc1ccccc1 ZINC000217655381 CH For-Sale Unstable FAAH 53 45 O=C(N/C=C/c1ccccc1)NCCCCc1ccccc1 ZINC000217655381 CH For-Sale Unstable SCN5A 0 44 O=C(N/C=C/c1ccccc1)NCCCCc1ccccc1 ZINC000217655381 CH For-Sale Unstable CES1 56 39 O=C(N/C=C/c1ccccc1)NCCCCc1ccccc1 ZINC000217655381 CH For-Sale Unstable HDAC9 27 40 O=C(N/C=C/c1ccccc1)NCCCCc1ccccc1 ZINC000217655381 CH For-Sale Unstable HDAC7 20 40 O=C(N/C=C/c1ccccc1)NCCCCc1ccccc1 ZINC000217655381 CH For-Sale Unstable AMP1_PLAFQ 39 59 Cc1cccc(CC(=O)N2CC[C@H](n3cc(-c4ccccc4)nn3)C2)c1 ZINC000217655396 EG In-Stock Unstable HDAC8 40 38 Cc1cccc(CC(=O)N2CC[C@H](n3cc(-c4ccccc4)nn3)C2)c1 ZINC000217655396 EG In-Stock Unstable PREP 25 46 CCCNc1ccc(S(=O)(=O)N[C@@H](C)CCC)cc1C(=O)O ZINC000217655423 EF In-Stock Unstable CASP3 0 40 CCCNc1ccc(S(=O)(=O)N[C@@H](C)CCC)cc1C(=O)O ZINC000217655423 EF In-Stock Unstable LEF 47 35 CCCC(=O)c1c[nH]c(C(=O)OC)c1 ZINC000217655453 AD In-Stock Unstable GABRA1 20 42 COc1cc(OC)cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c1 ZINC000217655456 JI In-Stock Unstable AKR1B1 0 48 COc1cc(OC)cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c1 ZINC000217655456 JI In-Stock Unstable CYP1B1 57 36 COc1cc(OC)cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c1 ZINC000217655456 JI In-Stock Unstable CYP1A1 45 48 COc1cc(OC)cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c1 ZINC000217655456 JI In-Stock Unstable CYP1A2 35 40 O=C(O)[C@@H]1CC[C@@H]1N1CC[C@@H](c2ccccc2)C1 ZINC000217655465 BE For-Sale Unstable SLC6A1 0 41 O=C(O)[C@@H]1CC[C@@H]1N1CC[C@@H](c2ccccc2)C1 ZINC000217655465 BE For-Sale Unstable ERBB2 0 41 O=C(O)[C@@H]1CC[C@@H]1N1CC[C@@H](c2ccccc2)C1 ZINC000217655465 BE For-Sale Unstable VACHT_TETCF 0 49 O=C(O)[C@@H]1CC[C@@H]1N1CC[C@@H](c2ccccc2)C1 ZINC000217655465 BE For-Sale Unstable SLC18A3 110 49 O=C(O)[C@@H]1CC[C@@H]1N1CC[C@@H](c2ccccc2)C1 ZINC000217655465 BE For-Sale Unstable ADAM10 19 41 Cc1cccc(CC(=O)N2CC[C@@H](n3cc(-c4ccccc4)nn3)C2)c1 ZINC000217655479 EG In-Stock Unstable HDAC8 40 38 Cc1cccc(CC(=O)N2CC[C@@H](n3cc(-c4ccccc4)nn3)C2)c1 ZINC000217655479 EG In-Stock Unstable PREP 25 46 CCCNc1ccc(S(=O)(=O)N[C@H](C)CCC)cc1C(=O)O ZINC000217655496 EF In-Stock Unstable CASP3 0 40 CCCNc1ccc(S(=O)(=O)N[C@H](C)CCC)cc1C(=O)O ZINC000217655496 EF In-Stock Unstable LEF 47 35 C[C@H](N[C@H]1CCN2CCCC[C@@H]12)c1ccc(Br)cc1 ZINC000217655503 DH On-Demand Unstable SDH1 0 45 COc1cc(OC)cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c1 ZINC000217655536 JI In-Stock Unstable AKR1B1 0 48 COc1cc(OC)cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c1 ZINC000217655536 JI In-Stock Unstable CYP1B1 57 36 COc1cc(OC)cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c1 ZINC000217655536 JI In-Stock Unstable CYP1A1 45 48 COc1cc(OC)cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c1 ZINC000217655536 JI In-Stock Unstable CYP1A2 35 40 CN(C)S(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217655563 CD On-Demand Unstable CA2 26 48 CN(C)S(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217655563 CD On-Demand Unstable CA1 33 40 CN(C)S(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217655563 CD On-Demand Unstable CA7 15 44 CN(C)S(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217655563 CD On-Demand Unstable CA4 23 42 CN(C)S(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217655563 CD On-Demand Unstable CA14 18 48 CN(C)S(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217655563 CD On-Demand Unstable CA12 26 48 CN(C)S(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217655563 CD On-Demand Unstable CA9 25 48 CN(C)S(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217655563 CD On-Demand Unstable IDO1 30 40 CN(C)S(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217655563 CD On-Demand Unstable MTCA1 41 40 CN(C)S(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217655563 CD On-Demand Unstable P96878_MYCTU 52 40 CN(C)S(=O)(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217655563 CD On-Demand Unstable PSBA 0 41 O=C(COc1ccccc1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217655576 EF In-Stock Unstable COLA 148 43 O=C(COc1ccccc1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217655576 EF In-Stock Unstable CPT1A 122 43 O=C(COc1ccccc1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217655576 EF In-Stock Unstable CPT2 46 35 O=C(COc1ccccc1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217655576 EF In-Stock Unstable PREP 25 48 CCC[C@@H](C)NS(=O)(=O)c1ccc(NC(C)C)c(C(=O)O)c1 ZINC000217655605 EF In-Stock Unstable LEF 48 35 O=C(O)[C@@H]1CC[C@H]1N1CC[C@@H](c2ccccc2)C1 ZINC000217655629 BE For-Sale Unstable SLC6A1 0 41 O=C(O)[C@@H]1CC[C@H]1N1CC[C@@H](c2ccccc2)C1 ZINC000217655629 BE For-Sale Unstable ERBB2 0 41 O=C(O)[C@@H]1CC[C@H]1N1CC[C@@H](c2ccccc2)C1 ZINC000217655629 BE For-Sale Unstable VACHT_TETCF 0 49 O=C(O)[C@@H]1CC[C@H]1N1CC[C@@H](c2ccccc2)C1 ZINC000217655629 BE For-Sale Unstable SLC18A3 110 49 O=C(O)[C@@H]1CC[C@H]1N1CC[C@@H](c2ccccc2)C1 ZINC000217655629 BE For-Sale Unstable ADAM10 19 41 N#Cc1ccccc1CN1CCC[C@@H]2CCCC[C@H]21 ZINC000217655645 CH On-Demand Unstable DPP4 15 42 C[C@@H](c1ccc(Br)cc1F)N1CCC[C@@H](CCC(=O)O)C1 ZINC000217655653 FI For-Sale Unstable GHSR 21 40 O=C(COc1ccccc1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217655663 EF In-Stock Unstable COLA 148 43 O=C(COc1ccccc1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217655663 EF In-Stock Unstable CPT1A 122 43 O=C(COc1ccccc1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217655663 EF In-Stock Unstable CPT2 46 35 O=C(COc1ccccc1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217655663 EF In-Stock Unstable PREP 25 48 COc1cc(C(=O)CN)ncc1Br ZINC000217655681 BC For-Sale Unstable P2RX2 43 34 CCOCCNC(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217655685 CD For-Sale Unstable TNFRSF1A 19 40 CCC[C@H](C)NS(=O)(=O)c1ccc(NC(C)C)c(C(=O)O)c1 ZINC000217655690 EF In-Stock Unstable LEF 48 35 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable ACE 69 50 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable TYR 33 40 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable OPRM1 41 43 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable OPRD1 42 39 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable OPRK1 0 40 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable MME 138 51 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable ANPEP 106 45 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable TACR1 40 55 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable CTSD 33 48 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable CTRA_BOVIN 49 48 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable FCER2 89 42 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable CASP3 33 41 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable BMP1 22 43 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable TACR2 41 34 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable RNPEP 31 44 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable PFDN6 0 44 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable KLK3 71 36 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable CTSB 91 51 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable PAPA1_CARPA 83 49 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable CYSP_TRYCR 92 45 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable CTSF 43 34 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable CTSK 37 42 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable CTSL 66 50 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable CPA1 59 50 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable CACNA1B 46 38 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable CCR3 28 52 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable SLC15A1 0 45 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable PGA 43 42 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable F2R 40 39 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable NPFFR2 55 39 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable TIMP3 77 43 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable CTRB1 36 46 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable NAALAD2 31 41 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable CAPNS1 74 54 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable MMP2 26 43 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable MMP3 58 52 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable MMP8 27 44 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable GRIA1 42 32 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable MMP14 51 38 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable ECE1 57 45 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable HLA-DRB1 75 42 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable SOAT1 23 42 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable REN 48 41 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable PAM 0 53 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable CTSS 45 50 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable CAPN1 122 47 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable MMP9 36 44 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable CASP1 25 40 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable CTRC 33 40 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable CAPN2 118 45 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable KYNU 0 42 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable ACE2 100 50 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable MC1R 40 34 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable CASP6 31 40 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable CASP9 22 40 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable LAP3 49 46 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable PROTEASE 0 42 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable CTSV 40 38 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable PSENEN 0 50 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable MMP7 31 42 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable GNPAT 0 46 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable MMP1 47 63 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable FPR1 65 49 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable CTRB_BOVIN 61 39 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable POL 0 60 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable NPR 73 41 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable AMP1_PLAFQ 65 46 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable HDA106 0 58 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable RHODESAIN 0 50 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable AMPX_VIBPR 0 46 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable CARP_RHICH 0 47 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable SLC15A2 0 53 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable BLA1_STEMA 79 43 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable POLG_WNV 45 30 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable QRFPR 54 36 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable PSMB8 54 38 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable ERAP1 0 44 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable NPFFR1 61 40 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable LASB 0 43 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable IDE 0 42 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable GPR142 53 33 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable VM1B1_BOTAS 0 48 COC(=O)[C@@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655696 CD On-Demand Unstable PQSD 0 41 NC/C=C\CN1CCC(Cc2ccccc2)CC1 ZINC000217655700 BE For-Sale Unstable ACHE 25 43 NC/C=C\CN1CCC(Cc2ccccc2)CC1 ZINC000217655700 BE For-Sale Unstable SLC6A3 15 40 NC/C=C\CN1CCC(Cc2ccccc2)CC1 ZINC000217655700 BE For-Sale Unstable GRIN1 22 43 NC/C=C\CN1CCC(Cc2ccccc2)CC1 ZINC000217655700 BE For-Sale Unstable GRIN2B 71 51 NC/C=C\CN1CCC(Cc2ccccc2)CC1 ZINC000217655700 BE For-Sale Unstable SIGMAR1 52 62 NC/C=C\CN1CCC(Cc2ccccc2)CC1 ZINC000217655700 BE For-Sale Unstable CCR3 22 44 NC/C=C\CN1CCC(Cc2ccccc2)CC1 ZINC000217655700 BE For-Sale Unstable GRIN2C 24 48 NC/C=C\CN1CCC(Cc2ccccc2)CC1 ZINC000217655700 BE For-Sale Unstable GRIN3A 0 47 COc1ccccc1-c1c(C(N)=O)sc2cnc(Nc3ccc(NC4CCOCC4)cc3OC(C)C)nc12 ZINC000217655712 KK Annotated Unstable ALK 47 35 COc1ccccc1-c1c(C(N)=O)sc2cnc(Nc3ccc(NC4CCOCC4)cc3OC(C)C)nc12 ZINC000217655712 KK Annotated Unstable MAPK7 47 35 N#Cc1ccccc1CN1CCC[C@H]2CCCC[C@H]21 ZINC000217655736 CH On-Demand Unstable DPP4 15 42 C[C@H](c1ccc(Br)cc1F)N1CCC[C@@H](CCC(=O)O)C1 ZINC000217655744 FI For-Sale Unstable GHSR 21 40 C[C@@H](Cn1cncn1)NC(=O)c1n[nH]c(=O)c2ccccc12 ZINC000217655757 CC In-Stock Unstable HIS3 89 44 CCn1cc(NC(=O)c2cccc(/C=C\C(=O)O)c2)cn1 ZINC000217655768 CE For-Sale Unstable HDAC8 40 44 CCn1cc(NC(=O)c2cccc(/C=C\C(=O)O)c2)cn1 ZINC000217655768 CE For-Sale Unstable HDAC6 28 44 CCn1cc(NC(=O)c2cccc(/C=C\C(=O)O)c2)cn1 ZINC000217655768 CE For-Sale Unstable MAPK10 19 40 CCn1cc(NC(=O)c2cccc(/C=C\C(=O)O)c2)cn1 ZINC000217655768 CE For-Sale Unstable PANC 49 33 CCn1cc(NC(=O)c2cccc(/C=C\C(=O)O)c2)cn1 ZINC000217655768 CE For-Sale Unstable KCNK3 93 38 CCn1cc(NC(=O)c2cccc(/C=C\C(=O)O)c2)cn1 ZINC000217655768 CE For-Sale Unstable KCNK9 47 38 O=C(c1ccc(F)cc1Cl)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217655776 FH In-Stock Unstable P2RX7 33 51 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable ACE 69 50 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable TYR 33 40 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable OPRM1 41 43 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable OPRD1 42 39 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable OPRK1 0 40 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable MME 138 51 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable ANPEP 106 45 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable TACR1 40 55 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable CTSD 33 48 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable CTRA_BOVIN 49 48 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable FCER2 89 42 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable CASP3 33 41 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable BMP1 22 43 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable TACR2 41 34 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable RNPEP 31 44 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable PFDN6 0 44 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable KLK3 71 36 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable CTSB 91 51 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable PAPA1_CARPA 83 49 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable CYSP_TRYCR 92 45 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable CTSF 43 34 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable CTSK 37 42 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable CTSL 66 50 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable CPA1 59 50 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable CACNA1B 46 38 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable CCR3 28 52 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable SLC15A1 0 45 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable PGA 43 42 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable F2R 40 39 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable NPFFR2 55 39 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable TIMP3 77 43 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable CTRB1 36 46 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable NAALAD2 31 41 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable CAPNS1 74 54 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable MMP2 26 43 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable MMP3 58 52 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable MMP8 27 44 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable GRIA1 42 32 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable MMP14 51 38 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable ECE1 57 45 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable HLA-DRB1 75 42 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable SOAT1 23 42 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable REN 48 41 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable PAM 0 53 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable CTSS 45 50 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable CAPN1 122 47 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable MMP9 36 44 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable CASP1 25 40 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable CTRC 33 40 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable CAPN2 118 45 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable KYNU 0 42 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable ACE2 100 50 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable MC1R 40 34 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable CASP6 31 40 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable CASP9 22 40 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable LAP3 49 46 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable PROTEASE 0 42 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable CTSV 40 38 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable PSENEN 0 50 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable MMP7 31 42 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable GNPAT 0 46 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable MMP1 47 63 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable FPR1 65 49 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable CTRB_BOVIN 61 39 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable POL 0 60 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable NPR 73 41 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable AMP1_PLAFQ 65 46 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable HDA106 0 58 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable RHODESAIN 0 50 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable AMPX_VIBPR 0 46 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable CARP_RHICH 0 47 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable SLC15A2 0 53 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable BLA1_STEMA 79 43 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable POLG_WNV 45 30 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable QRFPR 54 36 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable PSMB8 54 38 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable ERAP1 0 44 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable NPFFR1 61 40 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable LASB 0 43 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable IDE 0 42 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable GPR142 53 33 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable VM1B1_BOTAS 0 48 COC(=O)[C@H](Cc1ccccc1)NC(=O)C(F)F ZINC000217655794 CD On-Demand Unstable PQSD 0 41 CCCCNc1ccc(S(=O)(=O)N[C@@H](C)CCC)cc1C(=O)O ZINC000217655797 EG In-Stock Unstable LEF 44 39 COc1cc(OC)c(F)c(CCc2cnc(N)nc2)c1F ZINC000217655825 CE For-Sale Unstable DRTS_PLABA 49 38 COc1cc(OC)c(F)c(CCc2cnc(N)nc2)c1F ZINC000217655825 CE For-Sale Unstable DRTS_TOXGO 15 40 C[C@H](Cn1cncn1)NC(=O)c1n[nH]c(=O)c2ccccc12 ZINC000217655838 CC In-Stock Unstable HIS3 89 44 NS(=O)(=O)CCNC(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217655849 CB For-Sale Unstable CA2 26 46 NS(=O)(=O)CCNC(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217655849 CB For-Sale Unstable HDA106 0 40 O=C(N/C=C/c1ccccc1)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217655855 FE For-Sale Unstable TGM2 77 40 O=C(N/C=C/c1ccccc1)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217655855 FE For-Sale Unstable F13A1 101 43 O=C(N/C=C/c1ccccc1)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217655855 FE For-Sale Unstable AKR1C3 43 37 O=C(c1ccc(F)cc1Cl)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217655864 FH In-Stock Unstable P2RX7 33 51 O=C(NC[C@@H]1CCCN2CCCC[C@H]12)c1cc(-c2ccccc2Cl)n[nH]1 ZINC000217655869 FH In-Stock Unstable ALPL 74 41 O=C(NC[C@@H]1CCCN2CCCC[C@H]12)c1cc(-c2ccccc2Cl)n[nH]1 ZINC000217655869 FH In-Stock Unstable RAC1 0 41 CCCCNc1ccc(S(=O)(=O)N[C@H](C)CCC)cc1C(=O)O ZINC000217655877 EG In-Stock Unstable LEF 44 39 O=C(O)/C=C\c1cccc(C(=O)N2CCC(CO)CC2)c1 ZINC000217655942 CD For-Sale Unstable GRIN2B 27 40 O=C(O)/C=C\c1cccc(C(=O)N2CCC(CO)CC2)c1 ZINC000217655942 CD For-Sale Unstable L3MBTL3 62 44 Cc1ccc(S(=O)(=O)N2CCN(C(=O)N/C=C/c3ccccc3)CC2)cc1 ZINC000217655961 GF For-Sale Unstable TGM2 76 41 Cc1ccc(S(=O)(=O)N2CCN(C(=O)N/C=C/c3ccccc3)CC2)cc1 ZINC000217655961 GF For-Sale Unstable F13A1 100 42 Cc1ccc(S(=O)(=O)N2CCN(C(=O)N/C=C/c3ccccc3)CC2)cc1 ZINC000217655961 GF For-Sale Unstable GPR183 0 43 O=C(c1ccc2nsnc2c1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217655966 GG In-Stock Unstable ABHD6 0 44 O=C(c1ccc2nsnc2c1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217655966 GG In-Stock Unstable L3MBTL3 70 39 CCC[C@@H](C)NS(=O)(=O)c1ccc(NCC(C)C)c(C(=O)O)c1 ZINC000217655967 EF In-Stock Unstable MTNN 41 32 COC(=O)C[C@@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(C(=O)O)cc1 ZINC000217655975 GF In-Stock Unstable KCNA5 26 41 CC[C@H]1O[C@H](OC)[C@H](O)[C@@H](O)[C@H]1O ZINC000217655979 AA For-Sale Unstable FIMH 51 43 COC(=O)c1ccn2cc([N+](=O)[O-])cc2c1O ZINC000217656007 BD In-Stock Unstable CACNA1D 55 33 COC(=O)C[C@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(C(=O)O)cc1 ZINC000217656056 GF In-Stock Unstable KCNA5 26 41 O=C(c1ccc2nsnc2c1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217656059 GG In-Stock Unstable ABHD6 0 44 O=C(c1ccc2nsnc2c1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217656059 GG In-Stock Unstable L3MBTL3 57 38 CCC[C@H](C)NS(=O)(=O)c1ccc(NCC(C)C)c(C(=O)O)c1 ZINC000217656061 EF In-Stock Unstable MTNN 41 32 CC[C@@H]1CC[C@@H](NC)[C@@H](Cc2cccc(Cl)c2)C1 ZINC000217656067 CI For-Sale Unstable CACNA1D 0 42 O=C(O)/C=C\c1ccc(C(=O)N2CCCCCCC2)s1 ZINC000217656106 CG For-Sale Unstable L3MBTL1 0 47 O=C(O)/C=C\c1ccc(C(=O)N2CCCCCCC2)s1 ZINC000217656106 CG For-Sale Unstable L3MBTL3 16 47 COc1cccc(CN(C)C/C=C\CN)c1 ZINC000217656139 BD For-Sale Unstable G6PC 24 40 CC[C@H]1CC[C@@H](NC)[C@@H](Cc2cccc(Cl)c2)C1 ZINC000217656157 CI For-Sale Unstable CACNA1D 0 42 CC[C@@H](C)[C@@H](CO)NC(=O)c1cc(O)nc2ccccc12 ZINC000217656167 CE In-Stock Unstable TACR2 26 49 CC[C@@H](C)[C@@H](CO)NC(=O)c1cc(O)nc2ccccc12 ZINC000217656167 CE In-Stock Unstable TACR3 71 45 CCC[C@@H](C)NS(=O)(=O)c1ccc(N[C@@H](C)CC)c(C(=O)O)c1 ZINC000217656171 EG In-Stock Unstable LEF 48 36 O=C(CSCc1ccccc1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217656174 GH In-Stock Unstable PREP 26 51 O=C(Nc1ccc(Br)c(C(F)(F)F)c1)C(F)F ZINC000217656191 DH On-Demand Anodyne Q8MMZ8_EIMTE 15 43 CC(C)NC(=O)CNC(=O)NC[C@H](c1ccc(Cl)cc1Cl)c1c[nH]c2ccccc12 ZINC000217656206 II On-Demand Unstable BRS3 24 40 CC(C)NC(=O)CNC(=O)NC[C@H](c1ccc(Cl)cc1Cl)c1c[nH]c2ccccc12 ZINC000217656206 II On-Demand Unstable GRPR 53 34 CC(C)NC(=O)CNC(=O)NC[C@H](c1ccc(Cl)cc1Cl)c1c[nH]c2ccccc12 ZINC000217656206 II On-Demand Unstable KISS1R 55 36 C[C@H](CC(F)(F)F)NC(=O)OC(C)(C)C ZINC000217656216 BF On-Demand Unstable PAPA1_CARPA 46 38 C[C@H](CC(F)(F)F)NC(=O)OC(C)(C)C ZINC000217656216 BF On-Demand Unstable CTSK 30 50 C[C@H](CC(F)(F)F)NC(=O)OC(C)(C)C ZINC000217656216 BF On-Demand Unstable PGA5 41 36 CCCCCCCCNCCN(CC)CCC ZINC000217656221 BH For-Sale Unstable ADH1A 0 40 CCCCCCCCNCCN(CC)CCC ZINC000217656221 BH For-Sale Unstable PAOX 18 44 CCCCCCCCNCCN(CC)CCC ZINC000217656221 BH For-Sale Unstable ADH7 0 40 CCCCCCCCNCCN(CC)CCC ZINC000217656221 BH For-Sale Unstable S1PR2 29 41 CCCCCCCCNCCN(CC)CCC ZINC000217656221 BH For-Sale Unstable ADH1B 0 40 CC[C@@H]1CC[C@H](NC)[C@@H](Cc2cccc(Cl)c2)C1 ZINC000217656238 CI For-Sale Unstable CACNA1D 0 42 CCC[C@H](C)NS(=O)(=O)c1ccc(N[C@@H](C)CC)c(C(=O)O)c1 ZINC000217656248 EG In-Stock Unstable LEF 48 36 O=C(CSCc1ccccc1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217656259 GH In-Stock Unstable PREP 26 51 Cc1ccc(/C=C\C(=O)O)cc1NS(=O)(=O)N1CCCC1 ZINC000217656265 DD For-Sale Unstable LPL 44 35 CC(C)NC(=O)CNC(=O)NC[C@@H](c1ccc(Cl)cc1Cl)c1c[nH]c2ccccc12 ZINC000217656281 II On-Demand Unstable BRS3 24 40 CC(C)NC(=O)CNC(=O)NC[C@@H](c1ccc(Cl)cc1Cl)c1c[nH]c2ccccc12 ZINC000217656281 II On-Demand Unstable GRPR 53 34 CC(C)NC(=O)CNC(=O)NC[C@@H](c1ccc(Cl)cc1Cl)c1c[nH]c2ccccc12 ZINC000217656281 II On-Demand Unstable KISS1R 55 36 CC[C@H]1CC[C@H](NC)[C@@H](Cc2cccc(Cl)c2)C1 ZINC000217656323 CI For-Sale Unstable CACNA1D 0 42 CCC[C@@H](C)NS(=O)(=O)c1ccc(N[C@H](C)CC)c(C(=O)O)c1 ZINC000217656328 EG In-Stock Unstable LEF 48 36 O=C(CCSc1ccccc1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217656374 GH In-Stock Unstable PREP 22 46 CCC[C@H](C)NS(=O)(=O)c1ccc(N[C@H](C)CC)c(C(=O)O)c1 ZINC000217656404 EG In-Stock Unstable LEF 48 36 O=C(CCSc1ccccc1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217656449 GH In-Stock Unstable PREP 22 46 COC(=O)c1ccn2cc([N+](=O)[O-])cc2c1OC ZINC000217656461 CD In-Stock Unstable CACNA1D 45 32 COCCn1cc(C(=O)NC2CC(C)(C)NC(C)(C)C2)c2ccccc21 ZINC000217656476 FG In-Stock Unstable CNR1 32 61 COCCn1cc(C(=O)NC2CC(C)(C)NC(C)(C)C2)c2ccccc21 ZINC000217656476 FG In-Stock Unstable HRH1 18 40 COCCn1cc(C(=O)NC2CC(C)(C)NC(C)(C)C2)c2ccccc21 ZINC000217656476 FG In-Stock Unstable CNR2 49 61 COCCn1cc(C(=O)NC2CC(C)(C)NC(C)(C)C2)c2ccccc21 ZINC000217656476 FG In-Stock Unstable EZH2 57 46 CC(C)(C)OC(=O)NCCNC(=O)N/C=C/c1ccccc1 ZINC000217656487 DE For-Sale Unstable PAPA1_CARPA 46 39 CC(C)(C)OC(=O)NCCNC(=O)N/C=C/c1ccccc1 ZINC000217656487 DE For-Sale Unstable CTSK 15 46 CC(C)(C)OC(=O)NCCNC(=O)N/C=C/c1ccccc1 ZINC000217656487 DE For-Sale Unstable POL 0 41 CCC[C@@H](C)NS(=O)(=O)c1ccc(NC(C)(C)C)c(C(=O)O)c1 ZINC000217656525 EG In-Stock Unstable LEF 40 34 O=C(O)C[C@H]1CCn2ncc(Br)c21 ZINC000217656537 BD For-Sale Unstable TBXA2R 49 37 O=C(c1ccc(C(F)(F)F)cc1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217656559 GI In-Stock Unstable EPHX2 21 40 O=C(c1ccc(C(F)(F)F)cc1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217656559 GI In-Stock Unstable SMO 38 44 O=C(c1ccc(C(F)(F)F)cc1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217656559 GI In-Stock Unstable L3MBTL1 0 40 O=C(c1ccc(C(F)(F)F)cc1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217656559 GI In-Stock Unstable L3MBTL3 73 40 O=C(c1ccc(C(F)(F)F)cc1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217656559 GI In-Stock Unstable SLC6A7 0 42 COC(=O)C[C@@H](c1c(O)c2ccccc2oc1=O)c1coc2ccc(OC)cc2c1=O ZINC000217656567 HG In-Stock Unstable NQO1 51 50 CC(C)(C)OC(=O)N1CCN(C(=O)N/C=C/c2ccccc2)CC1 ZINC000217656599 EF For-Sale Unstable GPR119 36 41 CCC[C@H](C)NS(=O)(=O)c1ccc(NC(C)(C)C)c(C(=O)O)c1 ZINC000217656607 EG In-Stock Unstable LEF 40 34 O=C(O)C[C@@H]1CCn2ncc(Br)c21 ZINC000217656618 BD For-Sale Unstable TBXA2R 49 37 COC(=O)C[C@H](c1c(O)c2ccccc2oc1=O)c1coc2ccc(OC)cc2c1=O ZINC000217656633 HG In-Stock Unstable NQO1 51 50 O=C(c1ccc(C(F)(F)F)cc1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217656644 GI In-Stock Unstable EPHX2 21 40 O=C(c1ccc(C(F)(F)F)cc1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217656644 GI In-Stock Unstable SMO 38 44 O=C(c1ccc(C(F)(F)F)cc1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217656644 GI In-Stock Unstable L3MBTL1 0 40 O=C(c1ccc(C(F)(F)F)cc1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217656644 GI In-Stock Unstable L3MBTL3 73 40 O=C(c1ccc(C(F)(F)F)cc1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217656644 GI In-Stock Unstable SLC6A7 0 42 CSC[C@@](C)(O)CNC(=O)COc1ccccc1[N+](=O)[O-] ZINC000217656651 DD On-Demand Unstable COLA 57 32 Cc1cc(-c2cc(C(=O)N3CCN(c4cccc(O)c4)CC3)c3c(C)noc3n2)c(C)s1 ZINC000217656653 IJ On-Demand Unstable CCKAR 28 41 CC(C)(C)OC(=O)N1CCC(NC(=O)N/C=C/c2ccccc2)CC1 ZINC000217656714 EG For-Sale Unstable EPHX2 48 42 CC(C)(C)OC(=O)N1CCC(NC(=O)N/C=C/c2ccccc2)CC1 ZINC000217656714 EG For-Sale Unstable CCR8 30 45 CC(C)(C)OC(=O)N1CCC(NC(=O)N/C=C/c2ccccc2)CC1 ZINC000217656714 EG For-Sale Unstable GPR119 44 44 CC(C)(C)OC(=O)N1CCC(NC(=O)N/C=C/c2ccccc2)CC1 ZINC000217656714 EG For-Sale Unstable SFRP1 74 42 CC(C)(C)OC(=O)N1CCC(NC(=O)N/C=C/c2ccccc2)CC1 ZINC000217656714 EG For-Sale Unstable WNT3 50 36 CSC[C@](C)(O)CNC(=O)COc1ccccc1[N+](=O)[O-] ZINC000217656736 DD On-Demand Unstable COLA 57 32 O=C(c1cc(=O)c2ccccc2o1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217656757 GG In-Stock Unstable PREP 15 42 COc1ccc(C(=O)N2CCC[C@H]2C)cc1/C=C\C(=O)O ZINC000217656759 CE For-Sale Unstable ACKR3 44 32 Cc1cc(-c2cc(C(=O)N3CCN(c4cccc(O)c4)CC3)c3c(C)noc3n2)c(C)o1 ZINC000217656768 II On-Demand Unstable CCKAR 37 43 O=C(c1cc(=O)c2ccccc2o1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217656837 GG In-Stock Unstable PREP 15 42 COc1ccc(C(=O)N2CCC[C@@H]2C)cc1/C=C\C(=O)O ZINC000217656842 CE For-Sale Unstable ACKR3 44 32 COc1cc(C2CCN(C(=O)OC(C)(C)C)CC2)ccc1Nc1ncc(OCc2c(Cl)c(OC)cc(OC)c2Cl)cn1 ZINC000217656847 KK For-Sale Unstable INSR 24 45 COc1cc(C2CCN(C(=O)OC(C)(C)C)CC2)ccc1Nc1ncc(OCc2c(Cl)c(OC)cc(OC)c2Cl)cn1 ZINC000217656847 KK For-Sale Unstable IGF1R 31 47 COc1cc(C2CCN(C(=O)OC(C)(C)C)CC2)ccc1Nc1ncc(OCc2c(Cl)c(OC)cc(OC)c2Cl)cn1 ZINC000217656847 KK For-Sale Unstable ALK 44 45 COc1cc(C2CCN(C(=O)OC(C)(C)C)CC2)ccc1Nc1ncc(OCc2c(Cl)c(OC)cc(OC)c2Cl)cn1 ZINC000217656847 KK For-Sale Unstable GPR119 50 46 COc1ccc(NC(=O)N/C=C/c2ccccc2C)cc1OC ZINC000217656851 DH For-Sale Unstable GRM4 15 42 COc1ccc(NC(=O)N/C=C/c2ccccc2C)cc1OC ZINC000217656851 DH For-Sale Unstable ENPP1 72 36 COc1ccc(NC(=O)N/C=C/c2ccccc2C)cc1OC ZINC000217656851 DH For-Sale Unstable KCNK3 38 41 CSC[C@@](C)(O)CNC(=O)c1cccnc1Cl ZINC000217656861 CD On-Demand Unstable G2YM83_BOTF4 78 40 Cc1noc2nc(-c3ccc(F)cc3)cc(C(=O)N3CCN(c4cccc(O)c4)CC3)c12 ZINC000217656870 II On-Demand Unstable SLC6A7 0 40 COc1c(C(=O)O)ccn2cc([N+](=O)[O-])cc12 ZINC000217656920 BD In-Stock Unstable AKR1C2 20 40 CSC[C@](C)(O)CNC(=O)c1cccnc1Cl ZINC000217656942 CD On-Demand Unstable G2YM83_BOTF4 78 40 Cc1ccccc1/C=C/NC(=O)NCCCN1CCCC1=O ZINC000217656971 DE For-Sale Unstable TYRO3 24 40 O=C(NCc1ccc(Oc2ccc(F)cc2)cc1)N1CCN(c2cccc(O)c2)CC1 ZINC000217656977 HI On-Demand Unstable HTR1A 15 40 O=C(NCc1ccc(Oc2ccc(F)cc2)cc1)N1CCN(c2cccc(O)c2)CC1 ZINC000217656977 HI On-Demand Unstable FAAH 19 41 O=C(NCc1ccc(Oc2ccc(F)cc2)cc1)N1CCN(c2cccc(O)c2)CC1 ZINC000217656977 HI On-Demand Unstable NPSR1 24 40 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCCc1ccc(O)cc1 ZINC000217657047 HE In-Stock Unstable TACR1 20 41 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCCc1ccc(O)cc1 ZINC000217657047 HE In-Stock Unstable CCKAR 24 40 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCCc1ccc(O)cc1 ZINC000217657047 HE In-Stock Unstable BRS3 28 45 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCCc1ccc(O)cc1 ZINC000217657047 HE In-Stock Unstable MMP8 15 44 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCCc1ccc(O)cc1 ZINC000217657047 HE In-Stock Unstable CCKBR 24 44 O=C(NCc1ccc(Oc2ccc(F)cc2)cc1)N1CCN(Cc2ccccn2)CC1 ZINC000217657098 HI On-Demand Unstable PDGFRB 23 40 O=C(NCc1ccc(Oc2ccc(F)cc2)cc1)N1CCN(Cc2ccccn2)CC1 ZINC000217657098 HI On-Demand Unstable FAAH 32 47 O=C(NCc1ccc(Oc2ccc(F)cc2)cc1)N1CCN(Cc2ccccn2)CC1 ZINC000217657098 HI On-Demand Unstable S1PR2 23 41 O=C(NCc1ccc(Oc2ccc(F)cc2)cc1)N1CCN(Cc2ccccn2)CC1 ZINC000217657098 HI On-Demand Unstable NPSR1 24 41 O=C(NCc1ccc(Oc2ccc(F)cc2)cc1)N1CCN(Cc2ccccn2)CC1 ZINC000217657098 HI On-Demand Unstable SCD 17 40 CCCOC(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217657158 CE On-Demand Unstable ACR 70 39 CCCOC(=O)c1ccc(NC(=O)C(F)F)cc1 ZINC000217657158 CE On-Demand Unstable CNGA1 0 51 CCCCCCCCOc1ccc([C@H](CC(=O)OC)c2c(O)c3ccccc3oc2=O)cc1 ZINC000217657165 JK In-Stock Unstable PLA2G4B 92 37 CCCCCCCCOc1ccc([C@H](CC(=O)OC)c2c(O)c3ccccc3oc2=O)cc1 ZINC000217657165 JK In-Stock Unstable FAAH 27 41 CCCCCCCCOc1ccc([C@H](CC(=O)OC)c2c(O)c3ccccc3oc2=O)cc1 ZINC000217657165 JK In-Stock Unstable NQO1 47 53 Cc1ccccc1/C=C/NC(=O)Nc1cccc(C(=O)O)c1 ZINC000217657183 CG For-Sale Unstable CCKAR 23 43 Cc1ccccc1/C=C/NC(=O)Nc1cccc(C(=O)O)c1 ZINC000217657183 CG For-Sale Unstable CCKBR 0 40 Cc1ccccc1/C=C/NC(=O)Nc1cccc(C(=O)O)c1 ZINC000217657183 CG For-Sale Unstable AKR1C3 41 47 Cc1ccccc1/C=C/NC(=O)Nc1cccc(C(=O)O)c1 ZINC000217657183 CG For-Sale Unstable DDX3X 0 41 Cc1ccccc1/C=C/NC(=O)Nc1cccc(C(=O)O)c1 ZINC000217657183 CG For-Sale Unstable KCNK3 105 45 Cc1ccccc1/C=C/NC(=O)Nc1cccc(C(=O)O)c1 ZINC000217657183 CG For-Sale Unstable KCNK9 58 41 CCN(C(=O)c1ccc(/C=C\C(=O)O)s1)C1CCCCC1 ZINC000217657203 DH For-Sale Unstable ACE 41 35 COc1ccccc1-c1c(C(N)=O)sc2cnc(Nc3ccc(CN4CCN(C)CC4)cc3OC(C)C)nc12 ZINC000217657209 KJ Annotated Unstable INSR 46 38 COc1ccccc1-c1c(C(N)=O)sc2cnc(Nc3ccc(CN4CCN(C)CC4)cc3OC(C)C)nc12 ZINC000217657209 KJ Annotated Unstable IGF1R 50 35 COc1ccccc1-c1c(C(N)=O)sc2cnc(Nc3ccc(CN4CCN(C)CC4)cc3OC(C)C)nc12 ZINC000217657209 KJ Annotated Unstable PLK1 65 43 COc1ccccc1-c1c(C(N)=O)sc2cnc(Nc3ccc(CN4CCN(C)CC4)cc3OC(C)C)nc12 ZINC000217657209 KJ Annotated Unstable PLK3 47 41 COc1ccccc1-c1c(C(N)=O)sc2cnc(Nc3ccc(CN4CCN(C)CC4)cc3OC(C)C)nc12 ZINC000217657209 KJ Annotated Unstable ALK 57 38 COc1ccccc1-c1c(C(N)=O)sc2cnc(Nc3ccc(CN4CCN(C)CC4)cc3OC(C)C)nc12 ZINC000217657209 KJ Annotated Unstable MAPK7 61 39 COc1ccccc1-c1c(C(N)=O)sc2cnc(Nc3ccc(CN4CCN(C)CC4)cc3OC(C)C)nc12 ZINC000217657209 KJ Annotated Unstable PLK2 29 41 Cc1cc(C)n(CCCNC(=O)NCc2ccc(Oc3ccc(F)cc3)cc2)n1 ZINC000217657214 GI On-Demand Unstable ACAT 45 36 CCCCCCCCOc1ccc([C@@H](CC(=O)OC)c2c(O)c3ccccc3oc2=O)cc1 ZINC000217657252 JK In-Stock Unstable PLA2G4B 92 37 CCCCCCCCOc1ccc([C@@H](CC(=O)OC)c2c(O)c3ccccc3oc2=O)cc1 ZINC000217657252 JK In-Stock Unstable FAAH 27 41 CCCCCCCCOc1ccc([C@@H](CC(=O)OC)c2c(O)c3ccccc3oc2=O)cc1 ZINC000217657252 JK In-Stock Unstable NQO1 47 53 COc1cccc(CNC(=O)C(F)F)c1 ZINC000217657273 BD On-Demand Unstable DRD4 43 33 COc1cccc(CNC(=O)C(F)F)c1 ZINC000217657273 BD On-Demand Unstable ANPEP 32 58 COc1cccc(CNC(=O)C(F)F)c1 ZINC000217657273 BD On-Demand Unstable NQO2 29 42 COc1cccc(CNC(=O)C(F)F)c1 ZINC000217657273 BD On-Demand Unstable PTGER3 16 42 COc1cccc(CNC(=O)C(F)F)c1 ZINC000217657273 BD On-Demand Unstable MMP13 29 41 COc1cccc(CNC(=O)C(F)F)c1 ZINC000217657273 BD On-Demand Unstable CTSK 17 42 COc1cccc(CNC(=O)C(F)F)c1 ZINC000217657273 BD On-Demand Unstable SCN3A 0 42 COc1cccc(CNC(=O)C(F)F)c1 ZINC000217657273 BD On-Demand Unstable ROCK1 46 47 COc1cccc(CNC(=O)C(F)F)c1 ZINC000217657273 BD On-Demand Unstable MTNR1A 69 51 COc1cccc(CNC(=O)C(F)F)c1 ZINC000217657273 BD On-Demand Unstable MTNR1B 59 51 COc1cccc(CNC(=O)C(F)F)c1 ZINC000217657273 BD On-Demand Unstable ROCK2 53 48 COc1cccc(CNC(=O)C(F)F)c1 ZINC000217657273 BD On-Demand Unstable DUSP3 0 42 COc1cccc(CNC(=O)C(F)F)c1 ZINC000217657273 BD On-Demand Unstable ABCB1 0 47 COc1cccc(CNC(=O)C(F)F)c1 ZINC000217657273 BD On-Demand Unstable CTSS 21 42 COc1cccc(CNC(=O)C(F)F)c1 ZINC000217657273 BD On-Demand Unstable BACE1 21 41 COc1cccc(CNC(=O)C(F)F)c1 ZINC000217657273 BD On-Demand Unstable HSD17B2 26 43 COc1cccc(CNC(=O)C(F)F)c1 ZINC000217657273 BD On-Demand Unstable AMP1_PLAFQ 58 45 COc1cccc(CNC(=O)C(F)F)c1 ZINC000217657273 BD On-Demand Unstable AKR1C3 16 40 COc1cccc(CNC(=O)C(F)F)c1 ZINC000217657273 BD On-Demand Unstable CARM1 53 44 COc1cccc(CNC(=O)C(F)F)c1 ZINC000217657273 BD On-Demand Unstable CRTM 44 36 COc1cccc(CNC(=O)C(F)F)c1 ZINC000217657273 BD On-Demand Unstable PDS 72 42 CN1CCN(C2CCN(c3ccc([N+](=O)[O-])cc3OC(F)F)CC2)CC1 ZINC000217657274 FE On-Demand Unstable ADRA1D 28 44 CN1CCN(C2CCN(c3ccc([N+](=O)[O-])cc3OC(F)F)CC2)CC1 ZINC000217657274 FE On-Demand Unstable ADRA1A 20 44 CN1CCN(C2CCN(c3ccc([N+](=O)[O-])cc3OC(F)F)CC2)CC1 ZINC000217657274 FE On-Demand Unstable ADRA1B 28 44 CN1CCN(C2CCN(c3ccc([N+](=O)[O-])cc3OC(F)F)CC2)CC1 ZINC000217657274 FE On-Demand Unstable WDR5 37 41 Cc1ccccc1/C=C/NC(=O)Nc1ccccc1[N+](=O)[O-] ZINC000217657282 CH For-Sale Unstable COLA 62 31 CSC[C@@](C)(O)CNC(=O)c1cnn2ccccc12 ZINC000217657284 CD On-Demand Unstable EPHB3 35 47 O=C(O)/C=C\c1ccc(C(=O)Nc2cccc(Cl)c2)s1 ZINC000217657297 DH For-Sale Anodyne KCNK3 81 46 O=C(O)/C=C\c1ccc(C(=O)Nc2cccc(Cl)c2)s1 ZINC000217657297 DH For-Sale Anodyne KCNK9 39 43 C[C@@H](C(=O)NC1CC1)N1CCN(C(=O)NCc2ccc(Oc3ccc(F)cc3)cc2)CC1 ZINC000217657334 IG On-Demand Unstable LTA4H 18 40 C[C@@H](C(=O)NC1CC1)N1CCN(C(=O)NCc2ccc(Oc3ccc(F)cc3)cc2)CC1 ZINC000217657334 IG On-Demand Unstable CCR3 40 35 C[C@@H](C(=O)NC1CC1)N1CCN(C(=O)NCc2ccc(Oc3ccc(F)cc3)cc2)CC1 ZINC000217657334 IG On-Demand Unstable SLC6A11 0 41 C[C@@H](C(=O)NC1CC1)N1CCN(C(=O)NCc2ccc(Oc3ccc(F)cc3)cc2)CC1 ZINC000217657334 IG On-Demand Unstable SLC6A12 0 41 O=C(Cn1c(=O)oc2ccccc21)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217657343 GE In-Stock Unstable PREP 20 41 COc1ccc(CCN2C(=O)N[C@@H](CCC(=O)Nc3ccc4c(c3)COC4=O)C2=O)cc1 ZINC000217657351 IE In-Stock Unstable KCNJ1 55 40 CSC[C@](C)(O)CNC(=O)c1cnn2ccccc12 ZINC000217657356 CD On-Demand Unstable EPHB3 35 47 Cc1ccccc1/C=C/NC(=O)Nc1cccc(O)c1 ZINC000217657389 CG For-Sale Unstable DDX3X 0 42 Cc1ccccc1/C=C/NC(=O)Nc1cccc(O)c1 ZINC000217657389 CG For-Sale Unstable KCNK3 92 40 Cc1ccccc1/C=C/NC(=O)Nc1cccc(O)c1 ZINC000217657389 CG For-Sale Unstable KCNK9 50 38 O=C(O)[C@@H]1CC[C@@H]1N1CCCc2ccccc2C1 ZINC000217657396 BE For-Sale Unstable AGTR2 42 39 O=C(O)[C@@H]1CC[C@@H]1N1CCCc2ccccc2C1 ZINC000217657396 BE For-Sale Unstable SLC18A3 56 36 O=C(O)[C@@H]1CC[C@@H]1N1CCCc2ccccc2C1 ZINC000217657396 BE For-Sale Unstable PREP 34 41 C[C@H](C(=O)NC1CC1)N1CCN(C(=O)NCc2ccc(Oc3ccc(F)cc3)cc2)CC1 ZINC000217657424 IG On-Demand Unstable LTA4H 18 40 C[C@H](C(=O)NC1CC1)N1CCN(C(=O)NCc2ccc(Oc3ccc(F)cc3)cc2)CC1 ZINC000217657424 IG On-Demand Unstable CCR3 40 35 C[C@H](C(=O)NC1CC1)N1CCN(C(=O)NCc2ccc(Oc3ccc(F)cc3)cc2)CC1 ZINC000217657424 IG On-Demand Unstable SLC6A11 0 41 C[C@H](C(=O)NC1CC1)N1CCN(C(=O)NCc2ccc(Oc3ccc(F)cc3)cc2)CC1 ZINC000217657424 IG On-Demand Unstable SLC6A12 0 41 O=C(Cn1c(=O)oc2ccccc21)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217657425 GE In-Stock Unstable PREP 20 41 Nc1ncc(CCC(=O)O)cc1Br ZINC000217657467 BD For-Sale Unstable THRA 23 47 Nc1ncc(CCC(=O)O)cc1Br ZINC000217657467 BD For-Sale Unstable THRB 30 48 Nc1ncc(CCC(=O)O)cc1Br ZINC000217657467 BD For-Sale Unstable FFAR1 55 39 CC1(C)CC(N2CCN(C(=O)OCc3ccccc3)CC2)CC(C)(C)N1 ZINC000217657475 FG For-Sale Unstable GRIN2B 25 44 CC1(C)CC(N2CCN(C(=O)OCc3ccccc3)CC2)CC(C)(C)N1 ZINC000217657475 FG For-Sale Unstable TGM2 32 41 CC1(C)CC(N2CCN(C(=O)OCc3ccccc3)CC2)CC(C)(C)N1 ZINC000217657475 FG For-Sale Unstable F13A1 45 41 CC1(C)CC(N2CCN(C(=O)OCc3ccccc3)CC2)CC(C)(C)N1 ZINC000217657475 FG For-Sale Unstable SLC12A5 70 38 O=C(O)[C@@H]1CC[C@H]1N1CCCc2ccccc2C1 ZINC000217657485 BE For-Sale Unstable AGTR2 42 39 O=C(O)[C@@H]1CC[C@H]1N1CCCc2ccccc2C1 ZINC000217657485 BE For-Sale Unstable SLC18A3 56 36 O=C(O)[C@@H]1CC[C@H]1N1CCCc2ccccc2C1 ZINC000217657485 BE For-Sale Unstable PREP 34 41 O=C(N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1)C1(c2ccc(Cl)cc2)CCCC1 ZINC000217657530 HJ In-Stock Unstable HSD11B1 0 47 O=C(NCc1ccc(CN2CCCC2)cc1)N1CCCN(S(=O)(=O)c2ccc(F)cc2)CC1 ZINC000217657552 JG On-Demand Unstable ADORA2B 46 41 O=C(NCc1ccc(CN2CCCC2)cc1)N1CCCN(S(=O)(=O)c2ccc(F)cc2)CC1 ZINC000217657552 JG On-Demand Unstable CCR3 22 49 O=C(NCc1ccc(CN2CCCC2)cc1)N1CCCN(S(=O)(=O)c2ccc(F)cc2)CC1 ZINC000217657552 JG On-Demand Unstable TGM2 54 46 O=C(NCc1ccc(CN2CCCC2)cc1)N1CCCN(S(=O)(=O)c2ccc(F)cc2)CC1 ZINC000217657552 JG On-Demand Unstable F13A1 70 46 O=C(NCc1ccc(CN2CCCC2)cc1)N1CCCN(S(=O)(=O)c2ccc(F)cc2)CC1 ZINC000217657552 JG On-Demand Unstable NAMPT 76 47 COc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)N1CCN(c3ccc(F)cc3)CC1)C(=O)OC2 ZINC000217657563 JI In-Stock Unstable IMPDH1 0 63 COc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)N1CCN(c3ccc(F)cc3)CC1)C(=O)OC2 ZINC000217657563 JI In-Stock Unstable IMPDH2 0 63 C[C@H]1C[C@@H](C)CN(C(=O)c2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217657568 CF For-Sale Unstable SRD5A2 0 40 C[C@H]1C[C@@H](C)CN(C(=O)c2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217657568 CF For-Sale Unstable L3MBTL3 43 38 O=C(O)[C@@H]1CC[C@@H]1N1CC[C@@H](N2CCCC2)C1 ZINC000217657604 BD For-Sale Unstable L3MBTL1 0 40 O=C(O)[C@@H]1CC[C@@H]1N1CC[C@@H](N2CCCC2)C1 ZINC000217657604 BD For-Sale Unstable L3MBTL3 53 37 CCOC(=O)c1ncn([C@@H]2CCN3CCC[C@@H]23)c1N ZINC000217657605 CD For-Sale Unstable GABRA1 15 40 CCOC(=O)c1ncn([C@@H]2CCN3CCC[C@@H]23)c1N ZINC000217657605 CD For-Sale Unstable GABRA5 37 40 CCOC(=O)c1ncn([C@@H]2CCN3CCC[C@@H]23)c1N ZINC000217657605 CD For-Sale Unstable GABRA3 20 40 CCOC(=O)c1ncn([C@@H]2CCN3CCC[C@@H]23)c1N ZINC000217657605 CD For-Sale Unstable GABRA2 18 40 O=C(N1CC[C@H](n2cc(-c3ccccc3)nn2)C1)C1(c2ccc(Cl)cc2)CCCC1 ZINC000217657607 HJ In-Stock Unstable HSD11B1 0 47 C[C@@H]1C[C@@H](C)CN(C(=O)CN2CCN(C(=O)NCc3ccc(CN4CCCC4)cc3)CC2)C1 ZINC000217657657 JF On-Demand Unstable DRD4 23 41 C[C@@H]1C[C@@H](C)CN(C(=O)CN2CCN(C(=O)NCc3ccc(CN4CCCC4)cc3)CC2)C1 ZINC000217657657 JF On-Demand Unstable HRH3 18 48 C[C@@H]1C[C@@H](C)CN(C(=O)CN2CCN(C(=O)NCc3ccc(CN4CCCC4)cc3)CC2)C1 ZINC000217657657 JF On-Demand Unstable MLNR 42 37 CCOC(=O)c1ncn([C@H]2CCN3CCC[C@@H]23)c1N ZINC000217657706 CD For-Sale Unstable GABRA1 15 40 CCOC(=O)c1ncn([C@H]2CCN3CCC[C@@H]23)c1N ZINC000217657706 CD For-Sale Unstable GABRA5 37 40 CCOC(=O)c1ncn([C@H]2CCN3CCC[C@@H]23)c1N ZINC000217657706 CD For-Sale Unstable GABRA3 20 40 CCOC(=O)c1ncn([C@H]2CCN3CCC[C@@H]23)c1N ZINC000217657706 CD For-Sale Unstable GABRA2 18 40 CCOc1ccc([C@@H](C)N[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217657726 CG For-Sale Unstable ACACA 0 40 C[C@H]1C[C@@H](C)CN(C(=O)CN2CCN(C(=O)NCc3ccc(CN4CCCC4)cc3)CC2)C1 ZINC000217657729 JF On-Demand Unstable DRD4 23 41 C[C@H]1C[C@@H](C)CN(C(=O)CN2CCN(C(=O)NCc3ccc(CN4CCCC4)cc3)CC2)C1 ZINC000217657729 JF On-Demand Unstable HRH3 18 48 C[C@H]1C[C@@H](C)CN(C(=O)CN2CCN(C(=O)NCc3ccc(CN4CCCC4)cc3)CC2)C1 ZINC000217657729 JF On-Demand Unstable MLNR 42 37 Cc1ccccc1/C=C/NC(=O)Nc1ccc(N)cc1 ZINC000217657748 CG For-Sale Unstable DDX3X 0 41 O=C(O)[C@@H]1CC[C@H]1N1CC[C@@H](N2CCCC2)C1 ZINC000217657773 BD For-Sale Unstable L3MBTL1 0 40 O=C(O)[C@@H]1CC[C@H]1N1CC[C@@H](N2CCCC2)C1 ZINC000217657773 BD For-Sale Unstable L3MBTL3 53 37 C[C@H]1C[C@H](C)CN(C(=O)CN2CCN(C(=O)NCc3ccc(CN4CCCC4)cc3)CC2)C1 ZINC000217657810 JF On-Demand Unstable DRD4 23 41 C[C@H]1C[C@H](C)CN(C(=O)CN2CCN(C(=O)NCc3ccc(CN4CCCC4)cc3)CC2)C1 ZINC000217657810 JF On-Demand Unstable HRH3 18 48 C[C@H]1C[C@H](C)CN(C(=O)CN2CCN(C(=O)NCc3ccc(CN4CCCC4)cc3)CC2)C1 ZINC000217657810 JF On-Demand Unstable MLNR 42 37 CCOc1ccc([C@H](C)N[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217657814 CG On-Demand Unstable ACACA 0 40 O=C(O)[C@@H]1CC[C@@H]1N1CC[C@@H](N2CCCCC2)C1 ZINC000217657861 CD For-Sale Unstable L3MBTL3 67 39 CCOc1ccc([C@@H](C)N[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217657900 CG For-Sale Unstable ACACA 0 40 COc1ccccc1-c1c(C(N)=O)sc2cnc(Nc3cc(C)c(N4CC[C@H](N(C)C)C4)cc3OC(C)C)nc12 ZINC000217657910 KK Annotated Unstable INSR 47 45 COc1ccccc1-c1c(C(N)=O)sc2cnc(Nc3cc(C)c(N4CC[C@H](N(C)C)C4)cc3OC(C)C)nc12 ZINC000217657910 KK Annotated Unstable IGF1R 44 45 COc1ccccc1-c1c(C(N)=O)sc2cnc(Nc3cc(C)c(N4CC[C@H](N(C)C)C4)cc3OC(C)C)nc12 ZINC000217657910 KK Annotated Unstable ZAP70 17 43 COc1ccccc1-c1c(C(N)=O)sc2cnc(Nc3cc(C)c(N4CC[C@H](N(C)C)C4)cc3OC(C)C)nc12 ZINC000217657910 KK Annotated Unstable ALK 51 39 COc1ccccc1-c1c(C(N)=O)sc2cnc(Nc3cc(C)c(N4CC[C@H](N(C)C)C4)cc3OC(C)C)nc12 ZINC000217657910 KK Annotated Unstable MAPK7 57 36 Cc1csc(NC(=O)c2ccc(/C=C\C(=O)O)cc2F)n1 ZINC000217657923 DF For-Sale Unstable GCK 20 47 CC(C)NS(=O)(=O)Cc1ccccc1CNC(=O)NCc1ccc(CN2CCCC2)cc1 ZINC000217657941 JG On-Demand Unstable HRH2 21 42 CC(C)NS(=O)(=O)Cc1ccccc1CNC(=O)NCc1ccc(CN2CCCC2)cc1 ZINC000217657941 JG On-Demand Unstable HRH3 15 40 CC(C)NS(=O)(=O)Cc1ccccc1CNC(=O)NCc1ccc(CN2CCCC2)cc1 ZINC000217657941 JG On-Demand Unstable SIGMAR1 21 43 CC(C)NS(=O)(=O)Cc1ccccc1CNC(=O)NCc1ccc(CN2CCCC2)cc1 ZINC000217657941 JG On-Demand Unstable F2R 40 32 CC(C)NS(=O)(=O)Cc1ccccc1CNC(=O)NCc1ccc(CN2CCCC2)cc1 ZINC000217657941 JG On-Demand Unstable BDKRB1 20 43 CC(C)NS(=O)(=O)Cc1ccccc1CNC(=O)NCc1ccc(CN2CCCC2)cc1 ZINC000217657941 JG On-Demand Unstable NPFFR1 56 34 CC(C)NS(=O)(=O)Cc1ccccc1CNC(=O)NCc1ccc(CN2CCCC2)cc1 ZINC000217657941 JG On-Demand Unstable TMPRSS11D 89 38 O=C([C@H]1CC=CCC1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217657964 DG In-Stock Unstable PREP 23 48 CCOc1ccc([C@H](C)N[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217657995 CG On-Demand Unstable ACACA 0 40 COc1ccccc1-c1c(C(N)=O)sc2cnc(Nc3cc(C)c(N4CC[C@@H](N(C)C)C4)cc3OC(C)C)nc12 ZINC000217658007 KK Annotated Unstable INSR 47 45 COc1ccccc1-c1c(C(N)=O)sc2cnc(Nc3cc(C)c(N4CC[C@@H](N(C)C)C4)cc3OC(C)C)nc12 ZINC000217658007 KK Annotated Unstable IGF1R 44 45 COc1ccccc1-c1c(C(N)=O)sc2cnc(Nc3cc(C)c(N4CC[C@@H](N(C)C)C4)cc3OC(C)C)nc12 ZINC000217658007 KK Annotated Unstable ZAP70 17 43 COc1ccccc1-c1c(C(N)=O)sc2cnc(Nc3cc(C)c(N4CC[C@@H](N(C)C)C4)cc3OC(C)C)nc12 ZINC000217658007 KK Annotated Unstable ALK 51 39 COc1ccccc1-c1c(C(N)=O)sc2cnc(Nc3cc(C)c(N4CC[C@@H](N(C)C)C4)cc3OC(C)C)nc12 ZINC000217658007 KK Annotated Unstable MAPK7 57 36 C[C@@H](C(=O)NC1CC1)N1CCN(C(=O)NCc2ccc(CN3CCCC3)cc2)CC1 ZINC000217658043 HD On-Demand Unstable HRH3 25 48 C[C@@H](C(=O)NC1CC1)N1CCN(C(=O)NCc2ccc(CN3CCCC3)cc2)CC1 ZINC000217658043 HD On-Demand Unstable SIGMAR1 21 42 C[C@@H](C(=O)NC1CC1)N1CCN(C(=O)NCc2ccc(CN3CCCC3)cc2)CC1 ZINC000217658043 HD On-Demand Unstable CCR3 17 42 C[C@@H](C(=O)NC1CC1)N1CCN(C(=O)NCc2ccc(CN3CCCC3)cc2)CC1 ZINC000217658043 HD On-Demand Unstable MCHR1 31 44 C[C@@H](C(=O)NC1CC1)N1CCN(C(=O)NCc2ccc(CN3CCCC3)cc2)CC1 ZINC000217658043 HD On-Demand Unstable BIRC2 55 35 O=C(O)[C@@H]1CC[C@H]1N1CC[C@@H](N2CCCCC2)C1 ZINC000217658045 CD For-Sale Unstable L3MBTL3 67 39 O=C([C@H]1CC=CCC1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217658052 DG In-Stock Unstable PREP 23 48 C=C(CC)COc1ccc(/C=C\C(=O)O)cc1OC ZINC000217658070 CG On-Demand Unstable PTGER2 0 48 C=C(CC)COc1ccc(/C=C\C(=O)O)cc1OC ZINC000217658070 CG On-Demand Unstable CYP1B1 18 41 C=C(CC)COc1ccc(/C=C\C(=O)O)cc1OC ZINC000217658070 CG On-Demand Unstable APP 21 45 C=C(CC)COc1ccc(/C=C\C(=O)O)cc1OC ZINC000217658070 CG On-Demand Unstable CYP1A1 21 41 C=C(CC)COc1ccc(/C=C\C(=O)O)cc1OC ZINC000217658070 CG On-Demand Unstable TUBB1 58 41 C=C(CC)COc1ccc(/C=C\C(=O)O)cc1OC ZINC000217658070 CG On-Demand Unstable AKR1C3 33 50 C=C(CC)COc1ccc(/C=C\C(=O)O)cc1OC ZINC000217658070 CG On-Demand Unstable PTPA 0 44 C=C(CC)COc1ccc(/C=C\C(=O)O)cc1OC ZINC000217658070 CG On-Demand Unstable ABCG2 16 46 Cc1ccccc1/C=C/NC(=O)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217658091 EG For-Sale Unstable CA2 19 41 Cc1ccccc1/C=C/NC(=O)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217658091 EG For-Sale Unstable LPL 56 36 Cc1ccccc1/C=C/NC(=O)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217658091 EG For-Sale Unstable CA1 45 33 Cc1ccccc1/C=C/NC(=O)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217658091 EG For-Sale Unstable MTCA1 44 41 Cc1ccccc1/C=C/NC(=O)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217658091 EG For-Sale Unstable P96878_MYCTU 56 41 CCNC(=O)CNC(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217658118 CC For-Sale Unstable CA2 25 44 C[C@H](C(=O)NC1CC1)N1CCN(C(=O)NCc2ccc(CN3CCCC3)cc2)CC1 ZINC000217658120 HD On-Demand Unstable HRH3 25 48 C[C@H](C(=O)NC1CC1)N1CCN(C(=O)NCc2ccc(CN3CCCC3)cc2)CC1 ZINC000217658120 HD On-Demand Unstable SIGMAR1 21 42 C[C@H](C(=O)NC1CC1)N1CCN(C(=O)NCc2ccc(CN3CCCC3)cc2)CC1 ZINC000217658120 HD On-Demand Unstable CCR3 17 42 C[C@H](C(=O)NC1CC1)N1CCN(C(=O)NCc2ccc(CN3CCCC3)cc2)CC1 ZINC000217658120 HD On-Demand Unstable MCHR1 31 44 C[C@H](C(=O)NC1CC1)N1CCN(C(=O)NCc2ccc(CN3CCCC3)cc2)CC1 ZINC000217658120 HD On-Demand Unstable BIRC2 55 35 O=C([C@@H]1CC=CCC1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217658128 DG In-Stock Unstable PREP 23 48 CCNC(=O)CNC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217658187 CC For-Sale Unstable HDAC8 17 44 CCNC(=O)CNC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217658187 CC For-Sale Unstable CCR2 40 35 O=C([C@@H]1CC=CCC1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217658200 DG In-Stock Unstable PREP 23 48 C=C(CC)COc1cc(/C=C\C(=O)O)ccc1OC ZINC000217658215 CG For-Sale Unstable PTGER2 0 44 C=C(CC)COc1cc(/C=C\C(=O)O)ccc1OC ZINC000217658215 CG For-Sale Unstable CYP1B1 18 41 C=C(CC)COc1cc(/C=C\C(=O)O)ccc1OC ZINC000217658215 CG For-Sale Unstable APP 20 40 C=C(CC)COc1cc(/C=C\C(=O)O)ccc1OC ZINC000217658215 CG For-Sale Unstable CYP1A1 21 41 C=C(CC)COc1cc(/C=C\C(=O)O)ccc1OC ZINC000217658215 CG For-Sale Unstable TUBB1 58 41 C=C(CC)COc1cc(/C=C\C(=O)O)ccc1OC ZINC000217658215 CG For-Sale Unstable AKR1C3 35 53 C=C(CC)COc1cc(/C=C\C(=O)O)ccc1OC ZINC000217658215 CG For-Sale Unstable PTPA 0 44 C=C(CC)COc1cc(/C=C\C(=O)O)ccc1OC ZINC000217658215 CG For-Sale Unstable ABCG2 16 46 Cc1ccccc1/C=C/NC(=O)Nc1cccc(S(=O)(=O)O)c1 ZINC000217658219 EG For-Sale Unstable KCNK3 62 37 COC(=O)c1ccc(Cc2cccc(C)c2)[nH]1 ZINC000217658266 BF In-Stock Unstable CACNA1D 46 33 O=C(NCc1nc2ccc(Cl)cc2[nH]1)c1ccc(SCCO)cc1 ZINC000217658271 FG In-Stock Unstable F9 23 43 CN1CCC(NC(=O)c2ccc(/C=C\C(=O)O)s2)CC1 ZINC000217658313 CD For-Sale Unstable HTR1F 42 32 O=C(CNS(=O)(=O)c1cccc(F)c1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217658315 ID In-Stock Unstable PREP 15 40 O=C(CNS(=O)(=O)c1cccc(F)c1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217658315 ID In-Stock Unstable ST14 60 38 O=C(CNS(=O)(=O)c1cccc(F)c1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217658315 ID In-Stock Unstable SFRP1 61 35 CN1CCC(N2CCN(c3ccc([N+](=O)[O-])cc3Cl)CC2)CC1 ZINC000217658330 EE For-Sale Unstable WDR5 43 52 C=C(CC)COc1ccc(/C=C\C(=O)O)cc1[N+](=O)[O-] ZINC000217658338 CG For-Sale Unstable AKR1C3 30 47 C[C@@H](N[C@@H]1CCC[C@@H](O)C1)c1ccc(C#N)cc1 ZINC000217658363 BF For-Sale Unstable PK7 0 47 O=C(CNS(=O)(=O)c1cccc(F)c1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217658384 ID In-Stock Unstable PREP 15 40 O=C(CNS(=O)(=O)c1cccc(F)c1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217658384 ID In-Stock Unstable ST14 60 38 O=C(CNS(=O)(=O)c1cccc(F)c1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217658384 ID In-Stock Unstable SFRP1 61 35 CC(C)C[C@@H]1CC(=O)Oc2c1c(=O)oc1ccccc21 ZINC000217658409 CG In-Stock Unstable NQO1 22 42 CN1CCC(NC(=O)c2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217658425 CD For-Sale Unstable DRD4 15 42 CN1CCC(NC(=O)c2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217658425 CD For-Sale Unstable HTR1F 50 37 CN1CCC(NC(=O)c2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217658425 CD For-Sale Unstable MAPK13 46 32 CN1CCC(NC(=O)c2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217658425 CD For-Sale Unstable SLC6A5 38 47 C[C@H](N[C@@H]1CCC[C@@H](O)C1)c1ccc(C#N)cc1 ZINC000217658452 BF On-Demand Unstable PK7 0 47 CCC[C@@H](C)NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217658453 GG In-Stock Unstable TRY2_BOVIN 49 32 CCC[C@@H](C)NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217658453 GG In-Stock Unstable ADAMTS4 46 35 CC(C)C[C@H]1CC(=O)Oc2c1c(=O)oc1ccccc21 ZINC000217658490 CG In-Stock Unstable NQO1 22 42 Cc1cccc(S(=O)(=O)NCCC(=O)N2CC[C@H](n3cc(-c4ccccc4)nn3)C2)c1 ZINC000217658496 IE In-Stock Unstable ST14 65 33 Cc1cccc(S(=O)(=O)NCCC(=O)N2CC[C@H](n3cc(-c4ccccc4)nn3)C2)c1 ZINC000217658496 IE In-Stock Unstable CCR8 41 37 CCC[C@H](C)NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217658530 GG In-Stock Unstable TRY2_BOVIN 58 33 CCC[C@H](C)NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217658530 GG In-Stock Unstable ADAMTS4 46 35 C[C@@H](N[C@H]1CCC[C@@H](O)C1)c1ccc(C#N)cc1 ZINC000217658532 BF For-Sale Unstable PK7 0 47 CN1CCC(NC(=O)c2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217658535 CD For-Sale Unstable SIGMAR1 15 45 CN1CCC(NC(=O)c2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217658535 CD For-Sale Unstable HDAC8 36 42 CN1CCC(NC(=O)c2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217658535 CD For-Sale Unstable MAPK13 51 32 CN1CCC(NC(=O)c2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217658535 CD For-Sale Unstable HDAC6 22 42 CN1CCC(NC(=O)c2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217658535 CD For-Sale Unstable SLC6A5 33 40 O=C(NCC12CC3CC(CC(C3)C1)C2)C(F)F ZINC000217658536 BF On-Demand Unstable P2RX7 22 49 O=C(NCC12CC3CC(CC(C3)C1)C2)C(F)F ZINC000217658536 BF On-Demand Unstable EPHX2 36 58 COc1ccc2nc(SC/C=C\CN)[nH]c2c1 ZINC000217658552 BE For-Sale Unstable CYP2C8 31 57 COc1ccc2nc(SC/C=C\CN)[nH]c2c1 ZINC000217658552 BE For-Sale Unstable CYP1A2 24 64 COc1ccc2nc(SC/C=C\CN)[nH]c2c1 ZINC000217658552 BE For-Sale Unstable CYP2C19 51 63 Cc1cccc(S(=O)(=O)NCCC(=O)N2CC[C@@H](n3cc(-c4ccccc4)nn3)C2)c1 ZINC000217658573 IE In-Stock Unstable ST14 65 33 Cc1cccc(S(=O)(=O)NCCC(=O)N2CC[C@@H](n3cc(-c4ccccc4)nn3)C2)c1 ZINC000217658573 IE In-Stock Unstable CCR8 41 37 COC(=O)c1ccc(Cc2cccc(F)c2)[nH]1 ZINC000217658594 BF In-Stock Unstable CACNA1D 30 41 COC(=O)c1ccc(Cc2cccc(F)c2)[nH]1 ZINC000217658594 BF In-Stock Unstable HAO2 33 42 O=C(CCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCc1cccnc1 ZINC000217658605 HF In-Stock Unstable SCN9A 0 45 O=C(CCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCc1cccnc1 ZINC000217658605 HF In-Stock Unstable NAMPT 49 37 C[C@H](N[C@H]1CCC[C@@H](O)C1)c1ccc(C#N)cc1 ZINC000217658610 BF On-Demand Unstable PK7 0 47 O=C(CCc1ccccc1Br)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217658680 II In-Stock Unstable PREP 22 47 CCN1Cc2ccccc2C[C@@H]1C(=O)NCCSc1nncn1C ZINC000217658683 ED In-Stock Unstable MMP3 43 39 CCN1Cc2ccccc2C[C@@H]1C(=O)NCCSc1nncn1C ZINC000217658683 ED In-Stock Unstable ADAM9 67 38 O=C(CCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCc1cccnc1 ZINC000217658693 HF In-Stock Unstable SCN9A 0 45 O=C(CCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCc1cccnc1 ZINC000217658693 HF In-Stock Unstable NAMPT 49 37 Cc1ccccc1/C=C/NC(=O)Nc1ccccc1C ZINC000217658750 CI For-Sale Unstable DDX3X 0 44 O=C(CCc1ccccc1Br)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217658762 II In-Stock Unstable PREP 22 47 CCN1Cc2ccccc2C[C@H]1C(=O)NCCSc1nncn1C ZINC000217658766 ED In-Stock Unstable MMP3 43 39 CCN1Cc2ccccc2C[C@H]1C(=O)NCCSc1nncn1C ZINC000217658766 ED In-Stock Unstable ADAM9 67 38 CC[C@@H]1CCCN(C(=O)c2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217658817 CG For-Sale Unstable L3MBTL3 61 38 CC[C@@H]1CCCN(C(=O)c2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217658817 CG For-Sale Unstable GPR183 0 42 Cc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217658857 DK For-Sale Unstable GUAB 0 40 Cc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217658857 DK For-Sale Unstable GRM4 37 40 Cc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217658857 DK For-Sale Unstable IMDH_CRYPV 43 41 Cc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217658857 DK For-Sale Unstable BLM 0 40 Cc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217658857 DK For-Sale Unstable P95276_MYCTO 0 48 Cc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217658857 DK For-Sale Unstable WRN 0 40 Cc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217658857 DK For-Sale Unstable KCNK3 40 34 Cc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217658857 DK For-Sale Unstable PPX1 0 43 O=C(CCc1cccc(Cl)c1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217658860 GI In-Stock Unstable PREP 25 49 CC[C@H]1CCCN(C(=O)c2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217658897 CG For-Sale Unstable L3MBTL3 61 38 CC[C@H]1CCCN(C(=O)c2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217658897 CG For-Sale Unstable GPR183 0 42 CC[C@@H](N[C@@H]1CCN2CCCC[C@@H]12)c1ccccc1O ZINC000217658933 CG For-Sale Unstable SLC18A3 57 37 O=C(CCc1cccc(Cl)c1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217658935 GI In-Stock Unstable PREP 25 49 COC(=O)c1ccc(Cc2cccc(Cl)c2)[nH]1 ZINC000217658942 BG In-Stock Unstable MAOB 22 40 Cc1ccc(NC(=O)N/C=C/c2ccccc2C)cc1Cl ZINC000217658966 DJ For-Sale Unstable LPL 41 31 CCC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217658990 GH In-Stock Unstable TRY2_BOVIN 55 32 CC[C@H](N[C@@H]1CCN2CCCC[C@@H]12)c1ccccc1O ZINC000217659015 CG On-Demand Unstable SLC18A3 57 37 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc([N+](=O)[O-])c2)CC(=O)O4)cc1O ZINC000217659024 JI In-Stock Unstable AKR1B1 0 44 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc([N+](=O)[O-])c2)CC(=O)O4)cc1O ZINC000217659024 JI In-Stock Unstable CYP1B1 48 35 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc([N+](=O)[O-])c2)CC(=O)O4)cc1O ZINC000217659024 JI In-Stock Unstable CYP1A1 36 44 O=C(CCc1c(F)cccc1Cl)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217659028 GI In-Stock Unstable PREP 26 47 COc1ccc(C(=O)C(F)F)c(F)c1 ZINC000217659046 BE In-Stock Unstable TUBB2B 23 40 COc1ccc(C(=O)C(F)F)c(F)c1 ZINC000217659046 BE In-Stock Unstable AKR1C3 27 44 COc1ccc(C(=O)C(F)F)c(F)c1 ZINC000217659046 BE In-Stock Unstable AKR1C2 59 44 CCC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217659062 GH In-Stock Unstable TRY2_BOVIN 55 32 Cc1ccccc1/C=C/NC(=O)Nc1c(C)cccc1C(C)C ZINC000217659082 DK For-Sale Unstable SOAT1 56 42 Cc1ccccc1/C=C/NC(=O)Nc1c(C)cccc1C(C)C ZINC000217659082 DK For-Sale Unstable ACAT 0 48 CC[C@@H](N[C@H]1CCN2CCCC[C@@H]12)c1ccccc1O ZINC000217659097 CG For-Sale Unstable SLC18A3 57 37 O=C(CCc1c(F)cccc1Cl)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217659105 GI In-Stock Unstable PREP 26 47 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc([N+](=O)[O-])c2)CC(=O)O4)cc1O ZINC000217659108 JI In-Stock Unstable AKR1B1 0 44 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc([N+](=O)[O-])c2)CC(=O)O4)cc1O ZINC000217659108 JI In-Stock Unstable CYP1B1 48 35 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc([N+](=O)[O-])c2)CC(=O)O4)cc1O ZINC000217659108 JI In-Stock Unstable CYP1A1 36 44 O=C(c1ccc(O)cc1F)C(F)F ZINC000217659154 AD For-Sale Anodyne CES2 33 44 CC[C@H](N[C@H]1CCN2CCCC[C@@H]12)c1ccccc1O ZINC000217659159 CG On-Demand Unstable SLC18A3 57 37 CCC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217659164 HH In-Stock Unstable BMP1 79 39 CCC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217659164 HH In-Stock Unstable MMP13 65 43 CCC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217659164 HH In-Stock Unstable MMP2 42 40 CCC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217659164 HH In-Stock Unstable MMP3 52 40 CCC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217659164 HH In-Stock Unstable MMP8 29 43 CCC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217659164 HH In-Stock Unstable MMP9 46 43 CCC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217659164 HH In-Stock Unstable PTGDR 24 40 CCC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217659164 HH In-Stock Unstable MMP7 46 38 CCC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217659164 HH In-Stock Unstable ADAMTS4 45 35 CCC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217659164 HH In-Stock Unstable CA9 19 40 CCC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217659164 HH In-Stock Unstable MMP1 48 38 CCC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217659164 HH In-Stock Unstable AKR1C2 44 35 COc1ccc(O)c(C(=O)N[C@@H]2CC[C@@H](OC)CC2)c1 ZINC000217659187 CE In-Stock Unstable EPHX2 25 40 COc1ccc(O)c(C(=O)N[C@@H]2CC[C@@H](OC)CC2)c1 ZINC000217659187 CE In-Stock Unstable PDK1 40 35 CCOc1ccccc1CCC(=O)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217659202 GH In-Stock Unstable PREP 24 45 CCC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217659245 HH In-Stock Unstable BMP1 79 39 CCC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217659245 HH In-Stock Unstable MMP13 65 43 CCC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217659245 HH In-Stock Unstable MMP2 42 40 CCC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217659245 HH In-Stock Unstable MMP3 52 40 CCC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217659245 HH In-Stock Unstable MMP8 29 43 CCC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217659245 HH In-Stock Unstable MMP9 46 43 CCC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217659245 HH In-Stock Unstable PTGDR 24 40 CCC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217659245 HH In-Stock Unstable MMP7 46 38 CCC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217659245 HH In-Stock Unstable ADAMTS4 45 35 CCC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217659245 HH In-Stock Unstable CA9 19 40 CCC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217659245 HH In-Stock Unstable MMP1 48 38 CCC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217659245 HH In-Stock Unstable AKR1C2 44 35 CCOc1ccccc1[C@@H](C)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217659270 CG For-Sale Unstable HCN1 52 36 CCOc1ccccc1[C@@H](C)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217659270 CG For-Sale Unstable HCN4 46 36 CCOc1ccccc1CCC(=O)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217659279 GH In-Stock Unstable PREP 24 45 NS(=O)(=O)CCNC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217659330 CB For-Sale Unstable CA2 18 40 NS(=O)(=O)CCNC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217659330 CB For-Sale Unstable HDAC8 23 46 C[C@@H]1CN(C[C@@](C)(C(=O)O)c2ccccc2)CCCO1 ZINC000217659338 CE For-Sale Unstable CYP2J2 50 37 CCOc1ccccc1[C@H](C)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217659340 CG On-Demand Unstable HCN1 45 35 CCOc1ccccc1[C@H](C)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217659340 CG On-Demand Unstable HCN4 46 36 CCC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217659355 JH In-Stock Unstable IAP 0 40 CCC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217659355 JH In-Stock Unstable SCMU_MYCTU 0 43 CN1CCN(c2ccc3ccccc3n2)C[C@@H](O)C1 ZINC000217659356 CD In-Stock Unstable HTR3A 43 48 CN1CCN(c2ccc3ccccc3n2)C[C@@H](O)C1 ZINC000217659356 CD In-Stock Unstable PDE1B 0 42 CN1CCN(c2ccc3ccccc3n2)C[C@@H](O)C1 ZINC000217659356 CD In-Stock Unstable SORD 32 48 NC/C=C\COc1ccc(OCc2ccccc2)cc1 ZINC000217659360 CG For-Sale Unstable MAOB 26 50 NC/C=C\COc1ccc(OCc2ccccc2)cc1 ZINC000217659360 CG For-Sale Unstable LTA4H 23 49 NC/C=C\COc1ccc(OCc2ccccc2)cc1 ZINC000217659360 CG For-Sale Unstable TAAR1 28 46 NC/C=C\COc1ccc(OCc2ccccc2)cc1 ZINC000217659360 CG For-Sale Unstable FFAR1 24 45 COC(=O)c1ccc(Cc2cccc(OC)c2)[nH]1 ZINC000217659383 BE In-Stock Unstable UPP1 41 31 COC(=O)c1ccc(Cc2cccc(OC)c2)[nH]1 ZINC000217659383 BE In-Stock Unstable ROCK2 45 37 CSc1ccc(CCC(=O)N2CC[C@H](n3cc(-c4ccccc4)nn3)C2)cc1 ZINC000217659392 GI In-Stock Unstable PREP 25 49 O=C(CCc1cc(O)no1)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217659410 DD In-Stock Unstable ACE 44 57 O=C(CCc1cc(O)no1)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217659410 DD In-Stock Unstable MME 90 47 O=C(CCc1cc(O)no1)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217659410 DD In-Stock Unstable ANPEP 60 38 O=C(CCc1cc(O)no1)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217659410 DD In-Stock Unstable CMA1 28 50 O=C(CCc1cc(O)no1)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217659410 DD In-Stock Unstable CTSB 20 41 O=C(CCc1cc(O)no1)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217659410 DD In-Stock Unstable CPA1 52 42 O=C(CCc1cc(O)no1)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217659410 DD In-Stock Unstable NAALAD2 33 46 O=C(CCc1cc(O)no1)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217659410 DD In-Stock Unstable CAPN1 24 42 O=C(CCc1cc(O)no1)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217659410 DD In-Stock Unstable ACE2 86 40 O=C(CCc1cc(O)no1)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217659410 DD In-Stock Unstable PIN1 30 42 O=C(CCc1cc(O)no1)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217659410 DD In-Stock Unstable FPR1 53 39 O=C(CCc1cc(O)no1)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217659410 DD In-Stock Unstable BLA1_STEMA 78 52 Cc1ccccc1/C=C/NC(=O)Nc1cccc(Cl)c1C ZINC000217659419 DJ For-Sale Unstable CXCL8 45 39 CCOc1ccccc1[C@@H](C)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217659424 CG For-Sale Unstable HCN1 52 36 CCOc1ccccc1[C@@H](C)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217659424 CG For-Sale Unstable HCN4 46 36 C[C@H]1CN(C[C@@](C)(C(=O)O)c2ccccc2)CCCO1 ZINC000217659429 CE For-Sale Unstable CYP2J2 50 37 CCC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217659433 JH In-Stock Unstable IAP 0 40 CCC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217659433 JH In-Stock Unstable SCMU_MYCTU 0 43 CSc1ccc(CCC(=O)N2CC[C@@H](n3cc(-c4ccccc4)nn3)C2)cc1 ZINC000217659463 GI In-Stock Unstable PREP 25 49 COc1cc(N)ccc1N(CCN1CCN(C)CC1)C(=O)OC(C)(C)C ZINC000217659478 FE For-Sale Unstable HTR1A 22 42 CCOc1ccccc1[C@H](C)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217659495 CG On-Demand Unstable HCN1 45 35 CCOc1ccccc1[C@H](C)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217659495 CG On-Demand Unstable HCN4 46 36 COC(=O)c1ccc(Cc2ccc(OC)cc2)[nH]1 ZINC000217659498 BE In-Stock Unstable SLC18A2 17 40 CCOC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2C)cc1 ZINC000217659527 DH For-Sale Unstable CA1 28 44 CCOC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2C)cc1 ZINC000217659527 DH For-Sale Unstable ACR 65 38 CCOC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2C)cc1 ZINC000217659527 DH For-Sale Unstable NOD2 17 41 O=C(O)[C@H]1c2ccsc2CCN1C(=O)/C=C\c1cccs1 ZINC000217659544 DG For-Sale Unstable TRPM8 19 41 O=C(CCc1ccc(C(F)(F)F)cc1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217659574 HI In-Stock Unstable PREP 28 49 O=C(CCc1ccc(C(F)(F)F)cc1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217659574 HI In-Stock Unstable MCHR1 25 40 CC[C@@H](N[C@@H]1CCN2CCCC[C@@H]12)c1ccc(OC)cc1 ZINC000217659604 CG For-Sale Unstable CHRM2 27 42 CC[C@@H](N[C@@H]1CCN2CCCC[C@@H]12)c1ccc(OC)cc1 ZINC000217659604 CG For-Sale Unstable CHRM4 16 42 O=C(O)/C=C\c1ccc(C(=O)N2CCCCCCC2)cc1 ZINC000217659608 CG For-Sale Unstable MLYCD 21 48 O=C(O)/C=C\c1ccc(C(=O)N2CCCCCCC2)cc1 ZINC000217659608 CG For-Sale Unstable LGB 0 40 O=C(O)/C=C\c1ccc(C(=O)N2CCCCCCC2)cc1 ZINC000217659608 CG For-Sale Unstable L3MBTL1 0 48 O=C(O)/C=C\c1ccc(C(=O)N2CCCCCCC2)cc1 ZINC000217659608 CG For-Sale Unstable L3MBTL3 91 48 O=C(O)/C=C\c1ccc(C(=O)N2CCCCCCC2)cc1 ZINC000217659608 CG For-Sale Unstable MBTD1 0 48 O=C(O)/C=C\c1ccc(C(=O)N2CCCCCCC2)cc1 ZINC000217659608 CG For-Sale Unstable HPGD 40 42 O=C(O)/C=C\c1ccc(C(=O)N2CCCCCCC2)cc1 ZINC000217659608 CG For-Sale Unstable GPR183 0 52 O=C(O)/C=C\c1ccc(C(=O)N2CCCCCCC2)cc1 ZINC000217659608 CG For-Sale Unstable SLC6A7 0 42 O=C(O)[C@@H]1c2ccsc2CCN1C(=O)/C=C\c1cccs1 ZINC000217659623 DG For-Sale Unstable TRPM8 19 41 CCN1CCN(c2cccc(Nc3ncc(Br)cn3)c2)CC1 ZINC000217659629 FG On-Demand Unstable JAK2 17 44 O=C(NC[C@H]1C[C@@H]1c1nccc2ccccc12)OCc1ccccc1 ZINC000217659638 EI For-Sale Unstable CTSB 36 42 O=C(NC[C@H]1C[C@@H]1c1nccc2ccccc12)OCc1ccccc1 ZINC000217659638 EI For-Sale Unstable CYSP_TRYCR 44 33 O=C(NC[C@H]1C[C@@H]1c1nccc2ccccc12)OCc1ccccc1 ZINC000217659638 EI For-Sale Unstable CAPNS1 51 31 O=C(NC[C@H]1C[C@@H]1c1nccc2ccccc12)OCc1ccccc1 ZINC000217659638 EI For-Sale Unstable CAPN1 51 42 O=C(NC[C@H]1C[C@@H]1c1nccc2ccccc12)OCc1ccccc1 ZINC000217659638 EI For-Sale Unstable CASP1 21 42 O=C(NC[C@H]1C[C@@H]1c1nccc2ccccc12)OCc1ccccc1 ZINC000217659638 EI For-Sale Unstable CAPN2 82 42 O=C(NC[C@H]1C[C@@H]1c1nccc2ccccc12)OCc1ccccc1 ZINC000217659638 EI For-Sale Unstable NPR 61 34 O=C(NC[C@H]1C[C@@H]1c1nccc2ccccc12)OCc1ccccc1 ZINC000217659638 EI For-Sale Unstable KDM1A 18 43 Cc1ccccc1/C=C/NC(=O)Nc1ccccc1Cl ZINC000217659646 CI For-Sale Unstable LPL 25 40 Cc1ccccc1/C=C/NC(=O)Nc1ccccc1Cl ZINC000217659646 CI For-Sale Unstable CXCL8 47 39 O=C(CCc1ccc(C(F)(F)F)cc1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217659658 HI In-Stock Unstable PREP 28 49 O=C(CCc1ccc(C(F)(F)F)cc1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217659658 HI In-Stock Unstable MCHR1 25 40 O=C(O)/C=C\c1cccc(C(=O)N2CCCCCCC2)c1 ZINC000217659687 CG For-Sale Unstable PREP 27 43 O=C(O)/C=C\c1cccc(C(=O)N2CCCCCCC2)c1 ZINC000217659687 CG For-Sale Unstable L3MBTL1 0 47 O=C(O)/C=C\c1cccc(C(=O)N2CCCCCCC2)c1 ZINC000217659687 CG For-Sale Unstable L3MBTL3 68 47 O=C(O)/C=C\c1cccc(C(=O)N2CCCCCCC2)c1 ZINC000217659687 CG For-Sale Unstable HPGD 48 42 O=C(O)/C=C\c1cccc(C(=O)N2CCCCCCC2)c1 ZINC000217659687 CG For-Sale Unstable GPR183 0 44 CC[C@H](N[C@@H]1CCN2CCCC[C@@H]12)c1ccc(OC)cc1 ZINC000217659692 CG On-Demand Unstable CHRM2 26 42 CC[C@H](N[C@@H]1CCN2CCCC[C@@H]12)c1ccc(OC)cc1 ZINC000217659692 CG On-Demand Unstable CHRM4 16 42 COCCOC(=O)[C@@H]1C(=O)C[C@](C)(O)[C@@H](C(=O)OCCOC)[C@@H]1c1ccc2c(c1)OCO2 ZINC000217659725 JC In-Stock Unstable EDNRB 64 41 COCCOC(=O)[C@@H]1C(=O)C[C@](C)(O)[C@@H](C(=O)OCCOC)[C@@H]1c1ccc2c(c1)OCO2 ZINC000217659725 JC In-Stock Unstable EDNRA 63 41 O=C1C[C@@H](c2ccco2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217659726 GH In-Stock Unstable AKR1B1 0 46 O=C1C[C@@H](c2ccco2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217659726 GH In-Stock Unstable CYP1B1 23 41 O=C1C[C@@H](c2ccco2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217659726 GH In-Stock Unstable CYP1A1 25 41 O=C1C[C@@H](c2ccco2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217659726 GH In-Stock Unstable CYP1A2 17 40 Cc1ccccc1/C=C/NC(=O)Nc1ccccc1C(C)C ZINC000217659761 CJ For-Sale Unstable ACAT 0 41 C/C=C\C=C/C(=O)N1CCc2sccc2[C@@H]1C(=O)O ZINC000217659763 CE For-Sale Unstable TRPM8 18 40 CC[C@@H](N[C@H]1CCN2CCCC[C@@H]12)c1ccc(OC)cc1 ZINC000217659773 CG For-Sale Unstable CHRM2 27 42 CC[C@@H](N[C@H]1CCN2CCCC[C@@H]12)c1ccc(OC)cc1 ZINC000217659773 CG For-Sale Unstable CHRM4 16 42 C[C@@H](N[C@@H]1CCC[C@@H](O)C1)c1cccnc1 ZINC000217659779 BE For-Sale Unstable KCNA5 40 34 Cc1ccnc2ccc(C(=O)N3CC[C@H](n4cc(-c5ccccc5)nn4)C3)cc12 ZINC000217659790 GH In-Stock Unstable L3MBTL3 40 36 O=C1C[C@H](c2ccco2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217659822 GH In-Stock Unstable AKR1B1 0 46 O=C1C[C@H](c2ccco2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217659822 GH In-Stock Unstable CYP1B1 23 41 O=C1C[C@H](c2ccco2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217659822 GH In-Stock Unstable CYP1A1 25 41 O=C1C[C@H](c2ccco2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217659822 GH In-Stock Unstable CYP1A2 17 40 NC/C=C\COc1cccc2cccnc12 ZINC000217659823 BE For-Sale Unstable CCR1 0 41 NC/C=C\COc1cccc2cccnc12 ZINC000217659823 BE For-Sale Unstable METAP2 0 41 C/C=C/C=C\C(=O)N1CCc2sccc2[C@@H]1C(=O)O ZINC000217659837 CE For-Sale Unstable TRPM8 18 40 CC[C@H](N[C@H]1CCN2CCCC[C@@H]12)c1ccc(OC)cc1 ZINC000217659843 CG On-Demand Unstable CHRM2 26 42 CC[C@H](N[C@H]1CCN2CCCC[C@@H]12)c1ccc(OC)cc1 ZINC000217659843 CG On-Demand Unstable CHRM4 16 42 C[C@H](N[C@@H]1CCC[C@@H](O)C1)c1cccnc1 ZINC000217659851 BE On-Demand Unstable KCNA5 40 34 Cc1ccnc2ccc(C(=O)N3CC[C@@H](n4cc(-c5ccccc5)nn4)C3)cc12 ZINC000217659868 GH In-Stock Unstable L3MBTL3 40 36 Cc1ccccc1/C=C/NC(=O)Nc1cccc(Cl)c1Cl ZINC000217659871 DK For-Sale Unstable CXCL8 46 39 CC(C)N(C)S(=O)(=O)Nc1ccc(/C=C\C(=O)O)cc1F ZINC000217659874 DD For-Sale Unstable TRPV1 62 34 C[C@@H](N[C@H]1CCC[C@@H](O)C1)c1cccnc1 ZINC000217659930 BE For-Sale Unstable KCNA5 40 34 C/C=C\C=C\C(=O)N1CCc2sccc2[C@@H]1C(=O)O ZINC000217659932 CE For-Sale Unstable TRPM8 18 40 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](CC(C)C)C(=O)Nc3ccc4c(c3)OCO4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217659950 KK In-Stock Unstable TUBA1A 19 62 COC(=O)CS(=O)(=O)Nc1ccc(/C=C\C(=O)O)cc1F ZINC000217659965 DC For-Sale Unstable NFE2L2 0 40 Cc1cc(CCC(=O)N2CC[C@H](n3cc(-c4ccccc4)nn3)C2)ccc1F ZINC000217659970 GH In-Stock Unstable PREP 24 45 Cc1ccccc1/C=C/NC(=O)Nc1cc(Cl)ccc1Cl ZINC000217659975 DK For-Sale Unstable CXCL8 18 41 C[C@H](N[C@H]1CCC[C@@H](O)C1)c1cccnc1 ZINC000217660017 BE On-Demand Unstable KCNA5 40 34 N#C[C@H]1CCCN1C/C=C\c1ccccc1 ZINC000217660050 BF For-Sale Unstable DPP4 27 42 COc1ccc(OCCNC(=O)c2cnn(-c3ccc(F)cc3)c2C(F)(F)F)cc1 ZINC000217660052 HH On-Demand Unstable NR3C1 25 42 COc1ccc(OCCNC(=O)c2cnn(-c3ccc(F)cc3)c2C(F)(F)F)cc1 ZINC000217660052 HH On-Demand Unstable MST1R 49 40 Cc1cc(CCC(=O)N2CC[C@@H](n3cc(-c4ccccc4)nn3)C2)ccc1F ZINC000217660054 GH In-Stock Unstable PREP 24 45 COc1ccc(NC(=O)N/C=C/c2ccccc2C)cc1Cl ZINC000217660078 DI For-Sale Unstable GRM4 22 50 COc1ccc(NC(=O)N/C=C/c2ccccc2C)cc1Cl ZINC000217660078 DI For-Sale Unstable IMPDH2 0 45 CCC[C@@H](C)NS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217660111 EE In-Stock Unstable KCNQ2 52 39 Cc1ccccc1/C=C/NC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217660185 DJ For-Sale Unstable KIT 16 42 Cc1ccccc1/C=C/NC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217660185 DJ For-Sale Unstable KDR 17 45 Cc1ccccc1/C=C/NC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217660185 DJ For-Sale Unstable TEK 30 45 Cc1ccccc1/C=C/NC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217660185 DJ For-Sale Unstable BTK 23 41 Cc1ccccc1/C=C/NC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217660185 DJ For-Sale Unstable RIPK1 44 39 Cc1ccccc1/C=C/NC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217660185 DJ For-Sale Unstable IMDH_CRYPV 49 36 Cc1ccccc1/C=C/NC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217660185 DJ For-Sale Unstable TRPM4 0 41 Cc1ccccc1/C=C/NC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217660185 DJ For-Sale Unstable KCNK3 76 47 Cc1ccccc1/C=C/NC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217660185 DJ For-Sale Unstable KCNK9 54 35 CCC[C@H](C)NS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217660191 EE In-Stock Unstable KCNQ2 52 39 OCCN1CC[C@@H](O)[C@H](O)[C@H]1CO ZINC000217660209 AA In-Stock Unstable MGAM 28 40 OCCN1CC[C@@H](O)[C@H](O)[C@H]1CO ZINC000217660209 AA In-Stock Unstable UGCG 46 36 OCCN1CC[C@@H](O)[C@H](O)[C@H]1CO ZINC000217660209 AA In-Stock Unstable GBA2 81 50 OCCN1CC[C@@H](O)[C@H](O)[C@H]1CO ZINC000217660209 AA In-Stock Unstable SI 33 58 O=C(O)[C@@H]1CC[C@@H]1N1CCCCc2ccccc21 ZINC000217660222 BF For-Sale Unstable ACE 20 40 O=C(O)[C@@H]1CC[C@@H]1N1CCCCc2ccccc21 ZINC000217660222 BF For-Sale Unstable AVPR2 34 45 O=C(O)[C@@H]1CC[C@@H]1N1CCCCc2ccccc21 ZINC000217660222 BF For-Sale Unstable SLC6A1 40 33 O=C(O)[C@@H]1CC[C@@H]1N1CCCCc2ccccc21 ZINC000217660222 BF For-Sale Unstable AVPR1A 16 42 CCCC[C@@H](CC)C(=O)NC[C@@](C)(O)CSC ZINC000217660243 CE On-Demand Unstable SLC22A20 0 42 C/C=C\C(=O)N1CCc2sccc2[C@@H]1C(=O)O ZINC000217660276 CD For-Sale Unstable TRPM8 19 42 OCCN1CC[C@@H](O)[C@H](O)[C@@H]1CO ZINC000217660289 AA For-Sale Unstable MGAM 33 58 OCCN1CC[C@@H](O)[C@H](O)[C@@H]1CO ZINC000217660289 AA For-Sale Unstable UGCG 50 36 OCCN1CC[C@@H](O)[C@H](O)[C@@H]1CO ZINC000217660289 AA For-Sale Unstable GAA 24 58 OCCN1CC[C@@H](O)[C@H](O)[C@@H]1CO ZINC000217660289 AA For-Sale Unstable GBA2 97 50 OCCN1CC[C@@H](O)[C@H](O)[C@@H]1CO ZINC000217660289 AA For-Sale Unstable SI 37 58 Cc1ccc([N+](=O)[O-])cc1OC/C=C\CN ZINC000217660300 BD For-Sale Unstable CACNA1D 49 34 CCC[C@@H](C)NS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217660302 FF In-Stock Unstable KCNQ2 51 39 O=C(O)[C@@H]1CC[C@H]1N1CCCCc2ccccc21 ZINC000217660309 BF For-Sale Unstable ACE 20 40 O=C(O)[C@@H]1CC[C@H]1N1CCCCc2ccccc21 ZINC000217660309 BF For-Sale Unstable AVPR2 34 45 O=C(O)[C@@H]1CC[C@H]1N1CCCCc2ccccc21 ZINC000217660309 BF For-Sale Unstable SLC6A1 40 33 O=C(O)[C@@H]1CC[C@H]1N1CCCCc2ccccc21 ZINC000217660309 BF For-Sale Unstable AVPR1A 16 42 COc1cccc(CN[C@@H]2CCN3CCCC[C@@H]23)c1OC ZINC000217660324 CE On-Demand Unstable TACR3 25 41 CCCC[C@H](CC)C(=O)NC[C@@](C)(O)CSC ZINC000217660327 CE On-Demand Unstable SLC22A20 0 42 Cc1noc2nc(C(C)C)cc(C(=O)Nc3ccc(Cc4ccncc4)cc3)c12 ZINC000217660329 GJ On-Demand Unstable FLT1 44 48 Cc1noc2nc(C(C)C)cc(C(=O)Nc3ccc(Cc4ccncc4)cc3)c12 ZINC000217660329 GJ On-Demand Unstable KDR 16 48 CN(CCc1ccccc1)c1ccc(F)cc1CBr ZINC000217660345 DI For-Sale Unstable AOC3 15 40 CC(=O)Nc1ccc(CC(=O)N2CC[C@H](n3cc(-c4ccccc4)nn3)C2)cc1 ZINC000217660358 GF In-Stock Unstable PREP 24 44 C/C=C\C(=O)N1CCc2sccc2[C@H]1C(=O)O ZINC000217660366 CD For-Sale Unstable TRPM8 19 42 CCC[C@H](C)NS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217660381 FF In-Stock Unstable KCNQ2 51 39 CCCC[C@@H](CC)C(=O)NC[C@](C)(O)CSC ZINC000217660407 CE On-Demand Unstable SLC22A20 0 42 COc1cccc(CN[C@H]2CCN3CCCC[C@@H]23)c1OC ZINC000217660422 CE On-Demand Unstable TACR3 25 41 CC(=O)Nc1ccc(CC(=O)N2CC[C@@H](n3cc(-c4ccccc4)nn3)C2)cc1 ZINC000217660435 GF In-Stock Unstable PREP 24 44 C(=C/c1ccccc1)\CN1CCN(C[C@@H]2[C@H]3CNC[C@H]32)CC1 ZINC000217660452 CD In-Stock Unstable ADRA2C 23 45 CCCC[C@H](CC)C(=O)NC[C@](C)(O)CSC ZINC000217660486 CE On-Demand Unstable SLC22A20 0 42 CCC[C@@H](C)NS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1 ZINC000217660513 FD In-Stock Unstable SLC6A9 20 45 CCC[C@@H](C)NS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1 ZINC000217660513 FD In-Stock Unstable MMP12 32 44 CC/C=C(\C)C(=O)N1CCc2sccc2[C@@H]1C(=O)O ZINC000217660519 CF For-Sale Unstable TRPM8 19 44 Cc1nc2ccc(C(=O)N3CC[C@H](n4cc(-c5ccccc5)nn4)C3)cc2s1 ZINC000217660535 GH In-Stock Unstable NMT1 20 40 CN(CCc1ccccc1)c1cccc(Cl)c1CBr ZINC000217660554 EJ For-Sale Unstable AOC3 15 41 CCC[C@H](C)NS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1 ZINC000217660597 FD In-Stock Unstable SLC6A9 20 45 CCC[C@H](C)NS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1 ZINC000217660597 FD In-Stock Unstable MMP12 32 44 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)NCc1c(C)nn(C)c1C)C(=O)OC2 ZINC000217660600 JH In-Stock Unstable IMPDH1 0 62 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)NCc1c(C)nn(C)c1C)C(=O)OC2 ZINC000217660600 JH In-Stock Unstable IMPDH2 0 62 CC/C=C(\C)C(=O)N1CCc2sccc2[C@H]1C(=O)O ZINC000217660614 CF For-Sale Unstable TRPM8 19 44 Cc1nc2ccc(C(=O)N3CC[C@@H](n4cc(-c5ccccc5)nn4)C3)cc2s1 ZINC000217660628 GH In-Stock Unstable NMT1 20 40 COc1ccc(Cl)cc1NC(=O)N/C=C/c1ccccc1C ZINC000217660633 DI For-Sale Unstable RBP4 24 44 COc1ccc(Cl)cc1NC(=O)N/C=C/c1ccccc1C ZINC000217660633 DI For-Sale Unstable CYSP_PLAFA 42 35 c1ccc(CCCNC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217660687 CH For-Sale Unstable SLC18A2 47 43 c1ccc(CCCNC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217660687 CH For-Sale Unstable SIGMAR1 28 44 c1ccc(CCCNC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217660687 CH For-Sale Unstable PREP 42 36 CCCCc1ccc(NC(=O)N/C=C/c2ccccc2C)cc1 ZINC000217660723 DK For-Sale Unstable SCN2A 15 48 CCCCc1ccc(NC(=O)N/C=C/c2ccccc2C)cc1 ZINC000217660723 DK For-Sale Unstable CFTR 43 35 CCCCc1ccc(NC(=O)N/C=C/c2ccccc2C)cc1 ZINC000217660723 DK For-Sale Unstable ACAT 0 50 CCN(C/C=C\CN)C1CCCCC1 ZINC000217660730 AE For-Sale Unstable ADH1A 0 41 O=C(Cc1ccccc1OCc1ccccc1)N[C@@H]1C[C@@H]2OCC[C@@H]21 ZINC000217660739 EG In-Stock Unstable PTGER2 23 41 O=C(Cc1ccccc1OCc1ccccc1)N[C@@H]1C[C@@H]2OCC[C@@H]21 ZINC000217660739 EG In-Stock Unstable PPIA 42 35 C[C@]1(N)CCC[C@H](C(=O)O)C1 ZINC000217660750 AC For-Sale Unstable GRM1 16 50 CC(=O)Nc1ccc(C(=O)N2CC[C@H](n3cc(-c4ccccc4)nn3)C2)cc1 ZINC000217660758 GF In-Stock Unstable AVPR2 61 37 CC(=O)Nc1ccc(C(=O)N2CC[C@H](n3cc(-c4ccccc4)nn3)C2)cc1 ZINC000217660758 GF In-Stock Unstable AVPR1A 47 35 CC(=O)Nc1ccc(C(=O)N2CC[C@H](n3cc(-c4ccccc4)nn3)C2)cc1 ZINC000217660758 GF In-Stock Unstable PIK3CA 18 40 CC(=O)Nc1ccc(C(=O)N2CC[C@H](n3cc(-c4ccccc4)nn3)C2)cc1 ZINC000217660758 GF In-Stock Unstable PREP 17 41 CC(=O)Nc1ccc(C(=O)N2CC[C@H](n3cc(-c4ccccc4)nn3)C2)cc1 ZINC000217660758 GF In-Stock Unstable MTOR 44 40 CC(=O)Nc1ccc(C(=O)N2CC[C@H](n3cc(-c4ccccc4)nn3)C2)cc1 ZINC000217660758 GF In-Stock Unstable EPHX2 18 41 CC(=O)Nc1ccc(C(=O)N2CC[C@H](n3cc(-c4ccccc4)nn3)C2)cc1 ZINC000217660758 GF In-Stock Unstable PIK3CG 15 40 CC(=O)Nc1ccc(C(=O)N2CC[C@H](n3cc(-c4ccccc4)nn3)C2)cc1 ZINC000217660758 GF In-Stock Unstable SMO 43 37 CC(=O)Nc1ccc(C(=O)N2CC[C@H](n3cc(-c4ccccc4)nn3)C2)cc1 ZINC000217660758 GF In-Stock Unstable L3MBTL1 0 40 CC(=O)Nc1ccc(C(=O)N2CC[C@H](n3cc(-c4ccccc4)nn3)C2)cc1 ZINC000217660758 GF In-Stock Unstable L3MBTL3 80 40 COc1ccc(CC(=O)Nc2ccc(C(=O)N/N=C/c3ccc(OC)c(CSc4nc5ccccc5o4)c3)cc2)cc1 ZINC000217660759 KK For-Sale Unstable ADCYAP1R1 60 34 C[C@@H]1CCCN1C(=O)c1cc(/C=C\C(=O)O)ccc1F ZINC000217660786 CF For-Sale Unstable TRPC6 44 33 C[C@@]1(N)CCC[C@H](C(=O)O)C1 ZINC000217660837 AC For-Sale Unstable GRM1 16 50 COc1ccc(NC(=O)N/C=C/c2ccccc2C)cc1 ZINC000217660838 CH For-Sale Unstable CA1 48 37 COc1ccc(NC(=O)N/C=C/c2ccccc2C)cc1 ZINC000217660838 CH For-Sale Unstable MTNR1B 19 46 COc1ccc(NC(=O)N/C=C/c2ccccc2C)cc1 ZINC000217660838 CH For-Sale Unstable CA12 22 44 COc1ccc(NC(=O)N/C=C/c2ccccc2C)cc1 ZINC000217660838 CH For-Sale Unstable CA9 22 44 CC(=O)Nc1ccc(C(=O)N2CC[C@@H](n3cc(-c4ccccc4)nn3)C2)cc1 ZINC000217660840 GF In-Stock Unstable AVPR2 57 37 CC(=O)Nc1ccc(C(=O)N2CC[C@@H](n3cc(-c4ccccc4)nn3)C2)cc1 ZINC000217660840 GF In-Stock Unstable AVPR1A 47 35 CC(=O)Nc1ccc(C(=O)N2CC[C@@H](n3cc(-c4ccccc4)nn3)C2)cc1 ZINC000217660840 GF In-Stock Unstable PREP 17 41 CC(=O)Nc1ccc(C(=O)N2CC[C@@H](n3cc(-c4ccccc4)nn3)C2)cc1 ZINC000217660840 GF In-Stock Unstable MTOR 43 40 CC(=O)Nc1ccc(C(=O)N2CC[C@@H](n3cc(-c4ccccc4)nn3)C2)cc1 ZINC000217660840 GF In-Stock Unstable L3MBTL1 0 40 CC(=O)Nc1ccc(C(=O)N2CC[C@@H](n3cc(-c4ccccc4)nn3)C2)cc1 ZINC000217660840 GF In-Stock Unstable L3MBTL3 70 40 C[C@H]1CCCN1C(=O)c1cc(/C=C\C(=O)O)ccc1F ZINC000217660862 CF For-Sale Unstable TRPC6 44 33 C[C@@H](CCc1ccccc1)N[C@@H]1CCC[C@@H](O)C1 ZINC000217660871 BF For-Sale Unstable ACE 42 38 C[C@@H](CCc1ccccc1)N[C@@H]1CCC[C@@H](O)C1 ZINC000217660871 BF For-Sale Unstable SLC18A2 46 39 C[C@@H](CCc1ccccc1)N[C@@H]1CCC[C@@H](O)C1 ZINC000217660871 BF For-Sale Unstable SDH1 0 42 C[C@@H](CCc1ccccc1)N[C@@H]1CCC[C@@H](O)C1 ZINC000217660871 BF For-Sale Unstable BIRC2 40 39 COc1cccc2[nH]c(C(=O)NC[C@@H]3CCCN4CCCC[C@H]34)cc12 ZINC000217660893 EG In-Stock Unstable ACKR3 49 30 C[C@@]1(N)CCC[C@@H](C(=O)O)C1 ZINC000217660931 AC For-Sale Unstable GRM1 16 50 C[C@@H]1CCCN1C(=O)c1ccc(/C=C\C(=O)O)cc1F ZINC000217660943 CF For-Sale Unstable TRPC6 43 31 C[C@H](CCc1ccccc1)N[C@@H]1CCC[C@@H](O)C1 ZINC000217660944 BF On-Demand Unstable SLC18A2 43 38 C[C@H](CCc1ccccc1)N[C@@H]1CCC[C@@H](O)C1 ZINC000217660944 BF On-Demand Unstable SDH1 0 42 C[C@H](CCc1ccccc1)N[C@@H]1CCC[C@@H](O)C1 ZINC000217660944 BF On-Demand Unstable BIRC2 40 39 Cc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)cc1Cl ZINC000217660950 DK For-Sale Unstable PYGL 20 40 Cc1noc(C)c1CCC(=O)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217660958 FF In-Stock Unstable PREP 23 44 C[C@H]1CCCN1C(=O)c1ccc(/C=C\C(=O)O)cc1F ZINC000217661015 CF For-Sale Unstable TRPC6 43 31 C[C@@H](CCc1ccccc1)N[C@H]1CCC[C@@H](O)C1 ZINC000217661022 BF For-Sale Unstable ACE 42 38 C[C@@H](CCc1ccccc1)N[C@H]1CCC[C@@H](O)C1 ZINC000217661022 BF For-Sale Unstable SLC18A2 46 39 C[C@@H](CCc1ccccc1)N[C@H]1CCC[C@@H](O)C1 ZINC000217661022 BF For-Sale Unstable SDH1 0 42 C[C@@H](CCc1ccccc1)N[C@H]1CCC[C@@H](O)C1 ZINC000217661022 BF For-Sale Unstable BIRC2 40 39 CN(CCc1ccccc1)c1ccc(CBr)cc1Cl ZINC000217661023 EJ For-Sale Unstable AOC3 15 41 COc1ccc(C2(C(=O)N[C@@H](CC(C)C)c3nc4ccccc4[nH]3)CCOCC2)cc1 ZINC000217661030 HJ In-Stock Unstable PTPN1 24 40 COc1ccc(C2(C(=O)N[C@@H](CC(C)C)c3nc4ccccc4[nH]3)CCOCC2)cc1 ZINC000217661030 HJ In-Stock Unstable MMP7 21 48 Cc1noc(C)c1CCC(=O)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217661033 FF In-Stock Unstable PREP 23 44 Cc1ccccc1/C=C/NC(=O)NCCc1ccc(O)cc1 ZINC000217661060 CG For-Sale Unstable SLC6A5 24 40 CN1C[C@H](N)[C@H](c2cccc(Cl)c2)C1 ZINC000217661079 BD In-Stock Unstable SLC6A1 25 46 CN1C[C@H](N)[C@H](c2cccc(Cl)c2)C1 ZINC000217661079 BD In-Stock Unstable DPP4 26 45 C[C@H](CCc1ccccc1)N[C@H]1CCC[C@@H](O)C1 ZINC000217661092 BF On-Demand Unstable SLC18A2 43 38 C[C@H](CCc1ccccc1)N[C@H]1CCC[C@@H](O)C1 ZINC000217661092 BF On-Demand Unstable SDH1 0 42 C[C@H](CCc1ccccc1)N[C@H]1CCC[C@@H](O)C1 ZINC000217661092 BF On-Demand Unstable BIRC2 40 39 C[C@@H](N[C@@H]1CCN2CCCC[C@@H]12)c1ccccc1Cl ZINC000217661123 CH For-Sale Unstable OPRL1 26 42 Cn1cc(CC(=O)N2CC[C@H](n3cc(-c4ccccc4)nn3)C2)c2ccccc21 ZINC000217661130 GG In-Stock Unstable PREP 23 43 CN1C[C@@H](N)[C@H](c2ccc(Cl)cc2Cl)C1 ZINC000217661182 BE In-Stock Unstable SLC6A1 0 42 CN1C[C@@H](N)[C@H](c2ccc(Cl)cc2Cl)C1 ZINC000217661182 BE In-Stock Unstable DPP4 51 63 O=C(O)/C=C\c1cccc(C(=O)Nc2cccc(Cl)c2)c1 ZINC000217661189 DH For-Sale Anodyne MAOB 15 61 O=C(O)/C=C\c1cccc(C(=O)Nc2cccc(Cl)c2)c1 ZINC000217661189 DH For-Sale Anodyne PPIA 18 49 O=C(O)/C=C\c1cccc(C(=O)Nc2cccc(Cl)c2)c1 ZINC000217661189 DH For-Sale Anodyne CPT1A 53 36 O=C(O)/C=C\c1cccc(C(=O)Nc2cccc(Cl)c2)c1 ZINC000217661189 DH For-Sale Anodyne GRM5 16 56 O=C(O)/C=C\c1cccc(C(=O)Nc2cccc(Cl)c2)c1 ZINC000217661189 DH For-Sale Anodyne CSF1R 18 45 O=C(O)/C=C\c1cccc(C(=O)Nc2cccc(Cl)c2)c1 ZINC000217661189 DH For-Sale Anodyne BTK 25 41 O=C(O)/C=C\c1cccc(C(=O)Nc2cccc(Cl)c2)c1 ZINC000217661189 DH For-Sale Anodyne LUCI_LUCLA 16 41 O=C(O)/C=C\c1cccc(C(=O)Nc2cccc(Cl)c2)c1 ZINC000217661189 DH For-Sale Anodyne TAAR1 35 57 O=C(O)/C=C\c1cccc(C(=O)Nc2cccc(Cl)c2)c1 ZINC000217661189 DH For-Sale Anodyne AKR1C3 42 50 O=C(O)/C=C\c1cccc(C(=O)Nc2cccc(Cl)c2)c1 ZINC000217661189 DH For-Sale Anodyne KCNK3 125 62 O=C(O)/C=C\c1cccc(C(=O)Nc2cccc(Cl)c2)c1 ZINC000217661189 DH For-Sale Anodyne KCNK9 65 58 Cn1cc(CC(=O)N2CC[C@@H](n3cc(-c4ccccc4)nn3)C2)c2ccccc21 ZINC000217661217 GG In-Stock Unstable PREP 23 43 CCOC(=O)COc1ccc(NC(=O)c2ccccc2I)cc1 ZINC000217661225 IG On-Demand Unstable CA1 41 38 CCOC(=O)COc1ccc(NC(=O)c2ccccc2I)cc1 ZINC000217661225 IG On-Demand Unstable PRNP 30 50 CCOC(=O)COc1ccc(NC(=O)c2ccccc2I)cc1 ZINC000217661225 IG On-Demand Unstable CA12 18 41 CCOC(=O)COc1ccc(NC(=O)c2ccccc2I)cc1 ZINC000217661225 IG On-Demand Unstable CA9 18 41 CCOC(=O)COc1ccc(NC(=O)c2ccccc2I)cc1 ZINC000217661225 IG On-Demand Unstable Q25615_ONCVO 72 37 CCOC(=O)COc1ccc(NC(=O)c2ccccc2I)cc1 ZINC000217661225 IG On-Demand Unstable KCNK3 50 39 CCOC(=O)COc1ccc(NC(=O)c2ccccc2I)cc1 ZINC000217661225 IG On-Demand Unstable KCNK9 51 39 CN(CCc1ccccc1)c1ccccc1CBr ZINC000217661241 DI For-Sale Unstable AOC3 23 47 CN1C[C@H](N)[C@H](c2ccc(Cl)cc2Cl)C1 ZINC000217661274 BE In-Stock Unstable SLC6A1 0 42 CN1C[C@H](N)[C@H](c2ccc(Cl)cc2Cl)C1 ZINC000217661274 BE In-Stock Unstable DPP4 51 63 O=C(O)/C=C\c1ccc(C(=O)Nc2cccc(F)c2)s1 ZINC000217661283 CG For-Sale Anodyne TAAR1 15 40 O=C(O)/C=C\c1ccc(C(=O)Nc2cccc(F)c2)s1 ZINC000217661283 CG For-Sale Anodyne KCNK3 83 46 O=C(O)/C=C\c1ccc(C(=O)Nc2cccc(F)c2)s1 ZINC000217661283 CG For-Sale Anodyne KCNK9 43 43 C[C@@H](N[C@H]1CCN2CCCC[C@@H]12)c1ccccc1Cl ZINC000217661287 CH For-Sale Unstable OPRL1 26 42 O=C(O)[C@@H]1CC[C@@H]1N1CCN2CCCC[C@@H]2C1 ZINC000217661319 BD For-Sale Unstable L3MBTL3 40 36 O=C(Cn1cccc1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217661338 DE In-Stock Unstable PREP 24 46 CN1C[C@@H](N)[C@H](c2ccc(Cl)c(Cl)c2)C1 ZINC000217661372 BE In-Stock Unstable SLC6A2 27 48 CN1C[C@@H](N)[C@H](c2ccc(Cl)c(Cl)c2)C1 ZINC000217661372 BE In-Stock Unstable SLC6A1 32 49 CN1C[C@@H](N)[C@H](c2ccc(Cl)c(Cl)c2)C1 ZINC000217661372 BE In-Stock Unstable SLC6A4 21 48 CN1C[C@@H](N)[C@H](c2ccc(Cl)c(Cl)c2)C1 ZINC000217661372 BE In-Stock Unstable SLC6A3 27 42 O=C(O)[C@H]1CC[C@@H]1N1CCN2CCCC[C@@H]2C1 ZINC000217661402 BD For-Sale Unstable L3MBTL3 40 36 COc1ccnc(CNC(=O)c2cc(C)nc(C)n2)c1 ZINC000217661411 CD In-Stock Unstable CHRM4 16 40 O=C(Cn1cccc1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217661418 DE In-Stock Unstable PREP 24 46 Cc1noc2nc(C(C)C)cc(C(=O)Nc3nc4ccc(Cl)cc4s3)c12 ZINC000217661439 GK On-Demand Unstable LCK 27 40 Cc1noc2nc(C(C)C)cc(C(=O)Nc3nc4ccc(Cl)cc4s3)c12 ZINC000217661439 GK On-Demand Unstable CSNK1D 41 41 Cc1noc2nc(C(C)C)cc(C(=O)Nc3nc4ccc(Cl)cc4s3)c12 ZINC000217661439 GK On-Demand Unstable HSD17B1 0 44 CN(CCc1ccccc1)c1ccc(CBr)cc1F ZINC000217661453 DI For-Sale Unstable AOC3 15 41 CN1C[C@H](N)[C@H](c2ccc(Cl)c(Cl)c2)C1 ZINC000217661465 BE In-Stock Unstable SLC6A2 27 48 CN1C[C@H](N)[C@H](c2ccc(Cl)c(Cl)c2)C1 ZINC000217661465 BE In-Stock Unstable SLC6A1 32 49 CN1C[C@H](N)[C@H](c2ccc(Cl)c(Cl)c2)C1 ZINC000217661465 BE In-Stock Unstable SLC6A4 21 48 CN1C[C@H](N)[C@H](c2ccc(Cl)c(Cl)c2)C1 ZINC000217661465 BE In-Stock Unstable SLC6A3 27 42 O=C(O)[C@@H]1CC[C@H]1N1CCN2CCCC[C@@H]2C1 ZINC000217661470 BD For-Sale Unstable L3MBTL3 40 36 O=C(O)/C=C\c1cccc(C(=O)NCc2ccccn2)c1 ZINC000217661478 CE For-Sale Unstable HDAC8 23 44 CCC[C@H](C)NS(=O)(=O)c1ccc(N[C@H](C)CCC)c(C(=O)O)c1 ZINC000217661520 FG In-Stock Unstable LEF 51 36 O=C(c1ccc(-n2cccc2)cc1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217661531 GH In-Stock Unstable PREP 15 42 O=C(c1ccc(-n2cccc2)cc1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217661531 GH In-Stock Unstable L3MBTL3 73 40 O=C(NCc1n[nH]c(=O)[nH]1)c1cc(-c2ccc(F)cc2)nc2ccccc12 ZINC000217661538 FE On-Demand Unstable ACACB 23 44 O=C(NCc1n[nH]c(=O)[nH]1)c1cc(-c2ccc(F)cc2)nc2ccccc12 ZINC000217661538 FE On-Demand Unstable TACR3 31 62 O=C(NCc1n[nH]c(=O)[nH]1)c1cc(-c2ccc(F)cc2)nc2ccccc12 ZINC000217661538 FE On-Demand Unstable MT-CO2 50 42 O=C(NCc1n[nH]c(=O)[nH]1)c1cc(-c2ccc(F)cc2)nc2ccccc12 ZINC000217661538 FE On-Demand Unstable Q76353_9HIV1 0 40 O=C(O)[C@H]1CC[C@H]1N1CCN2CCCC[C@@H]2C1 ZINC000217661545 BD For-Sale Unstable L3MBTL3 40 36 Cc1noc2nc(C(C)C)cc(C(=O)Nc3nc(-c4ccc(F)cc4)cs3)c12 ZINC000217661570 GK On-Demand Unstable MPL 44 36 Cc1noc2nc(C(C)C)cc(C(=O)Nc3nc(-c4ccc(F)cc4)cs3)c12 ZINC000217661570 GK On-Demand Unstable ROCK1 20 42 Cc1noc2nc(C(C)C)cc(C(=O)Nc3nc(-c4ccc(F)cc4)cs3)c12 ZINC000217661570 GK On-Demand Unstable CAPN1 16 41 Cc1ccccc1NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217661576 CG For-Sale Unstable EPHX1 0 47 Cc1ccccc1NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217661576 CG For-Sale Unstable PTGER2 30 42 Cc1ccccc1NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217661576 CG For-Sale Unstable HDAC8 37 51 Cc1ccccc1NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217661576 CG For-Sale Unstable MMP2 0 57 Cc1ccccc1NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217661576 CG For-Sale Unstable HDAC6 26 51 Cc1ccccc1NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217661576 CG For-Sale Unstable MMP9 0 57 Cc1ccccc1NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217661576 CG For-Sale Unstable TTR 0 44 Cc1ccccc1NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217661576 CG For-Sale Unstable MMP1 0 57 Cc1ccccc1NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217661576 CG For-Sale Unstable FABH 0 40 Cc1ccccc1NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217661576 CG For-Sale Unstable RHOA 0 40 Cc1ccccc1NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217661576 CG For-Sale Unstable KCNK3 103 45 Cc1ccccc1NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217661576 CG For-Sale Unstable KCNK9 53 45 CCC[C@H](C)Nc1ccc(S(=O)(=O)N[C@@H](C)CCC)cc1C(=O)O ZINC000217661599 FG In-Stock Unstable LEF 51 36 O=C(c1ccc(-n2cccc2)cc1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217661615 GH In-Stock Unstable PREP 15 42 O=C(c1ccc(-n2cccc2)cc1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217661615 GH In-Stock Unstable L3MBTL3 73 40 CCC[C@@H](C)Nc1ccc(S(=O)(=O)N[C@H](C)CCC)cc1C(=O)O ZINC000217661677 FG In-Stock Unstable LEF 51 36 O=C(CN1CCc2ccccc2C1)NCCc1noc(C2CCCC2)n1 ZINC000217661688 FE In-Stock Unstable COLA 42 40 O=C(CN1CCc2ccccc2C1)NCCc1noc(C2CCCC2)n1 ZINC000217661688 FE In-Stock Unstable CPT1A 35 40 O=C(CN1CCc2ccccc2C1)NCCc1noc(C2CCCC2)n1 ZINC000217661688 FE In-Stock Unstable SMO 50 36 CCc1ccc(-c2csc(NC(=O)c3cc(C4CC4)on3)n2)cc1 ZINC000217661696 EI On-Demand Unstable MPL 50 38 CCc1ccc(-c2csc(NC(=O)c3cc(C4CC4)on3)n2)cc1 ZINC000217661696 EI On-Demand Unstable SPHK2 49 33 CCc1ccc(-c2csc(NC(=O)c3cc(C4CC4)on3)n2)cc1 ZINC000217661696 EI On-Demand Unstable SPHK1 45 33 CCc1ccc(-c2csc(NC(=O)c3cc(C4CC4)on3)n2)cc1 ZINC000217661696 EI On-Demand Unstable TRPA1 15 43 CN(CCc1ccccc1)c1ncc(CBr)cn1 ZINC000217661697 DG For-Sale Unstable AOC3 15 44 CN1C[C@@H](N)[C@H](c2cccc3ccccc23)C1 ZINC000217661716 BE In-Stock Unstable DPP4 0 41 O=C(CCn1cnc2ccccc2c1=O)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217661724 HF In-Stock Unstable PREP 19 43 CCC[C@H](C)Nc1ccc(S(=O)(=O)N[C@H](C)CCC)cc1C(=O)O ZINC000217661762 FG In-Stock Unstable LEF 51 36 CN1C[C@H](N)[C@H](c2cccc3ccccc23)C1 ZINC000217661804 BE In-Stock Unstable DPP4 0 41 O=C(CCn1cnc2ccccc2c1=O)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217661809 HF In-Stock Unstable PREP 19 43 Cc1noc2nc(C(C)C)cc(C(=O)Nc3nc(-c4cc(F)ccc4F)cs3)c12 ZINC000217661817 HK On-Demand Unstable MPL 40 39 Cc1ccccc1/C=C/NC(=O)NC1CCCCC1 ZINC000217661855 CH For-Sale Unstable FAAH 15 40 Cc1ccccc1/C=C/NC(=O)NC1CCCCC1 ZINC000217661855 CH For-Sale Unstable EPHX2 29 48 COc1cccc([C@@H]2CN(C)C[C@@H]2N)c1 ZINC000217661941 BD In-Stock Unstable DPP4 0 50 COC(=O)Cn1cnc2c(Cl)nc(Cl)nc21 ZINC000217661944 CD For-Sale Unstable P2RY1 33 41 COc1ccc2[nH]c(C(=O)NC[C@@H]3CCCN4CCCC[C@H]34)cc2c1 ZINC000217661966 EG In-Stock Unstable DRD3 15 47 COc1ccc2[nH]c(C(=O)NC[C@@H]3CCCN4CCCC[C@H]34)cc2c1 ZINC000217661966 EG In-Stock Unstable PYGL 75 42 COc1ccc2[nH]c(C(=O)NC[C@@H]3CCCN4CCCC[C@H]34)cc2c1 ZINC000217661966 EG In-Stock Unstable MAPKAPK2 0 41 COc1ccc2[nH]c(C(=O)NC[C@@H]3CCCN4CCCC[C@H]34)cc2c1 ZINC000217661966 EG In-Stock Unstable MTNR1A 41 38 COc1ccc2[nH]c(C(=O)NC[C@@H]3CCCN4CCCC[C@H]34)cc2c1 ZINC000217661966 EG In-Stock Unstable TUBB2B 40 43 COc1ccc2[nH]c(C(=O)NC[C@@H]3CCCN4CCCC[C@H]34)cc2c1 ZINC000217661966 EG In-Stock Unstable FPR2 22 41 COc1cccc([C@H]2CN(C)C[C@@H]2N)c1 ZINC000217662026 BD In-Stock Unstable DPP4 0 50 CN(CCc1ccccc1)c1ccc(CBr)cc1 ZINC000217662046 DI For-Sale Unstable AOC3 18 48 C[C@@H]1CN(CC[C@@H](O)c2ccccc2)CCCO1 ZINC000217662065 BE On-Demand Unstable CCR5 30 40 CC(=O)NCCCc1ccc(-c2csc(NC(=O)c3cc(C4CC4)on3)n2)cc1 ZINC000217662068 HH On-Demand Unstable SPHK2 53 34 CC(=O)NCCCc1ccc(-c2csc(NC(=O)c3cc(C4CC4)on3)n2)cc1 ZINC000217662068 HH On-Demand Unstable SPHK1 55 34 Cc1ccccc1/C=C/NC(=O)N1CCC(C(=O)O)CC1 ZINC000217662097 CE For-Sale Unstable SLC6A1 73 37 O=C(c1ccc(Cl)c(Cl)c1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217662130 GI In-Stock Unstable HSD11B1 15 41 O=C(c1ccc(Cl)c(Cl)c1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217662130 GI In-Stock Unstable CCR3 25 41 O=C(c1ccc(Cl)c(Cl)c1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217662130 GI In-Stock Unstable ABHD6 0 41 O=C(c1ccc(Cl)c(Cl)c1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217662130 GI In-Stock Unstable L3MBTL1 0 41 O=C(c1ccc(Cl)c(Cl)c1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217662130 GI In-Stock Unstable L3MBTL3 70 41 O=C(O)c1cc(Br)c(F)c(I)c1 ZINC000217662150 EF For-Sale Anodyne TPMT 0 54 C[C@H]1CN(CC[C@@H](O)c2ccccc2)CCCO1 ZINC000217662152 BE On-Demand Unstable CCR5 30 40 CCCCCCCCCC(=O)NC[C@@](C)(O)CSC ZINC000217662189 CG For-Sale Unstable NOD1 43 35 CCCCCCCCCC(=O)NC[C@@](C)(O)CSC ZINC000217662189 CG For-Sale Unstable CQSS 53 33 CN(C)C(=O)CN(C)C(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217662196 CD For-Sale Unstable HSD17B2 32 40 O=C(c1ccc(Cl)c(Cl)c1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217662209 GI In-Stock Unstable HSD11B1 15 41 O=C(c1ccc(Cl)c(Cl)c1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217662209 GI In-Stock Unstable CCR3 25 41 O=C(c1ccc(Cl)c(Cl)c1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217662209 GI In-Stock Unstable ABHD6 0 41 O=C(c1ccc(Cl)c(Cl)c1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217662209 GI In-Stock Unstable L3MBTL1 0 41 O=C(c1ccc(Cl)c(Cl)c1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217662209 GI In-Stock Unstable L3MBTL3 70 41 Cc1ccccc1/C=C/NC(=O)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217662211 HK For-Sale Unstable OPRL1 15 42 Cc1ccccc1/C=C/NC(=O)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217662211 HK For-Sale Unstable NMUR2 0 47 Cc1ccccc1/C=C/NC(=O)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217662211 HK For-Sale Unstable NMUR1 0 47 CCCCCCCCCC(=O)NC[C@](C)(O)CSC ZINC000217662278 CG For-Sale Unstable NOD1 43 35 CCCCCCCCCC(=O)NC[C@](C)(O)CSC ZINC000217662278 CG For-Sale Unstable CQSS 53 33 Cc1noc2nc(C(C)C)cc(C(=O)Nc3cccc(Cl)c3)c12 ZINC000217662307 EJ On-Demand Unstable PSBA 0 40 Cc1noc2nc(C(C)C)cc(C(=O)Nc3cccc(Cl)c3)c12 ZINC000217662307 EJ On-Demand Unstable KCNK3 86 41 Cc1noc2nc(C(C)C)cc(C(=O)Nc3cccc(Cl)c3)c12 ZINC000217662307 EJ On-Demand Unstable KCNK9 66 41 Cc1cnc(C(=O)N2CC[C@H](n3cc(-c4ccccc4)nn3)C2)cn1 ZINC000217662333 EE In-Stock Unstable PREP 23 44 O=C(NCc1cccs1)C(F)F ZINC000217662343 AD On-Demand Unstable ADAM17 0 43 O=C(NCc1cccs1)C(F)F ZINC000217662343 AD On-Demand Unstable CA5B 30 40 O=C(NCc1cccs1)C(F)F ZINC000217662343 AD On-Demand Unstable CA5A 29 40 O=C(NCc1cccs1)C(F)F ZINC000217662343 AD On-Demand Unstable CTSC 35 44 CCOc1ccc([C@@H]2CN(C)C[C@@H]2N)cc1 ZINC000217662345 BD In-Stock Unstable SLC6A1 24 42 CCOc1ccc([C@@H]2CN(C)C[C@@H]2N)cc1 ZINC000217662345 BD In-Stock Unstable CACNA2D2 51 34 CN(C)C(=O)CN(C)C(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217662384 CC For-Sale Unstable HSD17B2 15 40 CN1CCN(C(=O)c2cnc(N)s2)CC1 ZINC000217662413 BC For-Sale Unstable HRH4 29 40 Cc1cnc(C(=O)N2CC[C@@H](n3cc(-c4ccccc4)nn3)C2)cn1 ZINC000217662418 EE In-Stock Unstable PREP 23 44 CCOc1ccc([C@H]2CN(C)C[C@@H]2N)cc1 ZINC000217662425 BD In-Stock Unstable SLC6A1 24 42 CCOc1ccc([C@H]2CN(C)C[C@@H]2N)cc1 ZINC000217662425 BD In-Stock Unstable CACNA2D2 51 34 O=C(C(F)F)N1CC=C(c2ccccc2)CC1 ZINC000217662471 BF On-Demand Unstable ADAM10 34 41 CN(C)[C@@H]1[C@H]2CC[C@@H]1CN(C(=O)c1cccc(N3CCOCC3)c1)C2 ZINC000217662473 ED In-Stock Unstable AKR1C3 28 44 O=C(O)[C@H]1c2ccsc2CCN1C/C=C\c1ccccc1 ZINC000217662484 CG For-Sale Unstable TRPM8 17 40 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@@H]1CC[C@@H](C)O1 ZINC000217662510 CD On-Demand Unstable FKBP12.6 0 53 CC(C)N1CCN(C(=O)c2ccc(/C=C\C(=O)O)s2)CC1 ZINC000217662517 DE For-Sale Unstable HRH3 22 55 O=C(c1ccc(Br)o1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217662537 GG In-Stock Unstable PREP 18 42 CCCCNC(=O)N/C=C/c1ccccc1C ZINC000217662564 BG For-Sale Unstable ACAT 0 49 O=C(O)[C@@H]1c2ccsc2CCN1C/C=C\c1ccccc1 ZINC000217662576 CG For-Sale Unstable TRPM8 17 40 CN(Cc1cccnc1)C(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217662592 DF For-Sale Unstable TBXAS1 26 61 CN(Cc1cccnc1)C(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217662592 DF For-Sale Unstable HSD17B2 39 47 CN(Cc1cccnc1)C(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217662592 DF For-Sale Unstable NR1D1 43 38 O=C(c1ccc(Br)o1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217662611 GG In-Stock Unstable PREP 18 42 O=C1C[C@@H](c2ccc(OCc3ccccn3)cc2)c2c(c3ccccc3oc2=O)O1 ZINC000217662619 GI In-Stock Unstable MAOB 17 50 CCCN[C@H](c1cccnc1)[C@@]1(N(C)C)CCC[C@@H](C)C1 ZINC000217662651 CH For-Sale Unstable KCNA5 0 42 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@H]1CC[C@@H](C)O1 ZINC000217662653 CD On-Demand Unstable FKBP12.6 0 53 O=C1C[C@H](c2ccc(OCc3ccccn3)cc2)c2c(c3ccccc3oc2=O)O1 ZINC000217662694 GI In-Stock Unstable MAOB 15 50 C/C=C\CN1CCc2sccc2[C@@H]1C(=O)O ZINC000217662714 BE For-Sale Unstable TRPM8 17 40 O=C(c1cccc(Br)c1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217662731 GH In-Stock Unstable PREP 20 42 O=C(c1cccc(Br)c1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217662731 GH In-Stock Unstable L3MBTL3 53 40 CN1C[C@@H](N)[C@H](c2ccc(OCc3ccccc3)cc2)C1 ZINC000217662740 CF In-Stock Unstable MAOB 18 44 CN1C[C@@H](N)[C@H](c2ccc(OCc3ccccc3)cc2)C1 ZINC000217662740 CF In-Stock Unstable LTA4H 40 48 CN1C[C@@H](N)[C@H](c2ccc(OCc3ccccc3)cc2)C1 ZINC000217662740 CF In-Stock Unstable HRH3 15 46 CN1C[C@@H](N)[C@H](c2ccc(OCc3ccccc3)cc2)C1 ZINC000217662740 CF In-Stock Unstable KDM1A 17 40 CSC[C@@](C)(O)CNC(=O)c1ccc(NC(N)=O)cc1 ZINC000217662782 CD On-Demand Unstable F3 48 33 CC(=O)c1ccccc1OCCN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217662802 HH On-Demand Unstable HTR1A 56 40 CC(=O)c1ccccc1OCCN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217662802 HH On-Demand Unstable DRD2 51 40 CC(=O)c1ccccc1OCCN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217662802 HH On-Demand Unstable DRD1 18 42 CC(=O)c1ccccc1OCCN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217662802 HH On-Demand Unstable HRH2 0 40 CC(=O)c1ccccc1OCCN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217662802 HH On-Demand Unstable ADRA1D 28 45 CC(=O)c1ccccc1OCCN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217662802 HH On-Demand Unstable HTR2A 33 41 CC(=O)c1ccccc1OCCN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217662802 HH On-Demand Unstable HTR2C 26 41 CC(=O)c1ccccc1OCCN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217662802 HH On-Demand Unstable SLC6A1 60 39 CC(=O)c1ccccc1OCCN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217662802 HH On-Demand Unstable SLC6A4 21 40 CC(=O)c1ccccc1OCCN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217662802 HH On-Demand Unstable ADRA1A 24 45 CC(=O)c1ccccc1OCCN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217662802 HH On-Demand Unstable HRH1 28 42 CC(=O)c1ccccc1OCCN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217662802 HH On-Demand Unstable DRD3 52 37 CC(=O)c1ccccc1OCCN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217662802 HH On-Demand Unstable HTR4 44 43 CC(=O)c1ccccc1OCCN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217662802 HH On-Demand Unstable DRD5 18 42 CC(=O)c1ccccc1OCCN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217662802 HH On-Demand Unstable LTA4H 42 40 CC(=O)c1ccccc1OCCN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217662802 HH On-Demand Unstable THRB 22 44 CC(=O)c1ccccc1OCCN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217662802 HH On-Demand Unstable HTR7 40 46 CC(=O)c1ccccc1OCCN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217662802 HH On-Demand Unstable HRH3 17 40 CC(=O)c1ccccc1OCCN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217662802 HH On-Demand Unstable ABCB1 45 45 CC(=O)c1ccccc1OCCN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217662802 HH On-Demand Unstable PSMB2 47 38 CC(=O)c1ccccc1OCCN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217662802 HH On-Demand Unstable PSMB1 41 38 CC(=O)c1ccccc1OCCN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217662802 HH On-Demand Unstable HCN1 66 34 CC(=O)c1ccccc1OCCN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217662802 HH On-Demand Unstable HCN4 48 34 CC(C)(C)OC(=O)NNc1ccc(C(F)(F)F)cc1 ZINC000217662805 CH For-Sale Unstable DHODH 28 41 O=C(c1cccc(Br)c1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217662816 GH In-Stock Unstable PREP 20 42 O=C(c1cccc(Br)c1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217662816 GH In-Stock Unstable L3MBTL3 50 38 CN1C[C@H](N)[C@H](c2ccc(OCc3ccccc3)cc2)C1 ZINC000217662819 CF In-Stock Unstable MAOB 18 44 CN1C[C@H](N)[C@H](c2ccc(OCc3ccccc3)cc2)C1 ZINC000217662819 CF In-Stock Unstable LTA4H 40 48 CN1C[C@H](N)[C@H](c2ccc(OCc3ccccc3)cc2)C1 ZINC000217662819 CF In-Stock Unstable HRH3 15 46 CN1C[C@H](N)[C@H](c2ccc(OCc3ccccc3)cc2)C1 ZINC000217662819 CF In-Stock Unstable KDM1A 17 40 CCCN[C@H](c1cccnc1)[C@]1(N(C)C)CCC[C@@H](C)C1 ZINC000217662830 CH For-Sale Unstable KCNA5 0 42 COc1ccc(N2C(=O)[C@@H]3[C@@H]4CCCN4[C@]4(C(=O)N(Cc5ccccc5)c5ccccc54)[C@@H]3C2=O)cc1 ZINC000217662863 JH In-Stock Unstable SCN9A 0 41 CSC[C@](C)(O)CNC(=O)c1ccc(NC(N)=O)cc1 ZINC000217662873 CD On-Demand Unstable F3 48 33 C[C@@H](CCc1ccc2c(c1)OCO2)N[C@@H]1CCC[C@@H](O)C1 ZINC000217662906 CF For-Sale Unstable NOS2 65 33 C[C@@H](CCc1ccc2c(c1)OCO2)N[C@@H]1CCC[C@@H](O)C1 ZINC000217662906 CF For-Sale Unstable SSTR3 102 34 Fc1ccc(SCCN2CCN(CCOc3ccccc3Cl)CC2)cc1 ZINC000217662910 GI On-Demand Unstable HTR1A 25 48 Fc1ccc(SCCN2CCN(CCOc3ccccc3Cl)CC2)cc1 ZINC000217662910 GI On-Demand Unstable DRD2 29 42 Fc1ccc(SCCN2CCN(CCOc3ccccc3Cl)CC2)cc1 ZINC000217662910 GI On-Demand Unstable DRD1 16 48 Fc1ccc(SCCN2CCN(CCOc3ccccc3Cl)CC2)cc1 ZINC000217662910 GI On-Demand Unstable DRD4 18 48 Fc1ccc(SCCN2CCN(CCOc3ccccc3Cl)CC2)cc1 ZINC000217662910 GI On-Demand Unstable HTR2A 23 48 Fc1ccc(SCCN2CCN(CCOc3ccccc3Cl)CC2)cc1 ZINC000217662910 GI On-Demand Unstable SLC6A4 30 43 Fc1ccc(SCCN2CCN(CCOc3ccccc3Cl)CC2)cc1 ZINC000217662910 GI On-Demand Unstable DRD3 15 48 Fc1ccc(SCCN2CCN(CCOc3ccccc3Cl)CC2)cc1 ZINC000217662910 GI On-Demand Unstable SLC6A3 43 43 Fc1ccc(SCCN2CCN(CCOc3ccccc3Cl)CC2)cc1 ZINC000217662910 GI On-Demand Unstable DRD5 19 42 Fc1ccc(SCCN2CCN(CCOc3ccccc3Cl)CC2)cc1 ZINC000217662910 GI On-Demand Unstable LTA4H 32 46 Fc1ccc(SCCN2CCN(CCOc3ccccc3Cl)CC2)cc1 ZINC000217662910 GI On-Demand Unstable HTR7 19 48 Fc1ccc(SCCN2CCN(CCOc3ccccc3Cl)CC2)cc1 ZINC000217662910 GI On-Demand Unstable SIGMAR1 15 45 C[C@@H]1CN(CC[C@@H](O)c2cccc(Br)c2)CCCO1 ZINC000217662915 EF For-Sale Unstable SLC18A3 0 41 O=C(CC(c1ccccc1)c1ccccc1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217662927 HJ In-Stock Unstable PREP 26 46 C[C@H]1CN(CC[C@@H](O)c2cccc(Br)c2)CCCO1 ZINC000217662987 EF For-Sale Unstable SLC18A3 0 41 C[C@H](CCc1ccc2c(c1)OCO2)N[C@@H]1CCC[C@@H](O)C1 ZINC000217662990 CF On-Demand Unstable SSTR3 102 34 O=C(CC(c1ccccc1)c1ccccc1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217663003 HJ In-Stock Unstable PREP 26 46 Cc1ccccc1/C=C/NC(=O)N1CCCc2ccccc21 ZINC000217663029 CI For-Sale Unstable AVPR2 61 48 Cc1ccccc1/C=C/NC(=O)N1CCCc2ccccc21 ZINC000217663029 CI For-Sale Unstable AVPR1A 17 45 O=C(O)/C=C\c1ccc(C(=O)N2CCC[C@H](CO)C2)cc1 ZINC000217663031 CD For-Sale Unstable L3MBTL3 56 39 C[C@@H](CCc1ccc2c(c1)OCO2)N[C@H]1CCC[C@@H](O)C1 ZINC000217663077 CF For-Sale Unstable NOS2 65 33 C[C@@H](CCc1ccc2c(c1)OCO2)N[C@H]1CCC[C@@H](O)C1 ZINC000217663077 CF For-Sale Unstable SSTR3 102 34 O=C(O)/C=C\c1ccc(C(=O)N2CCC[C@@H](CO)C2)cc1 ZINC000217663107 CD For-Sale Unstable L3MBTL3 56 39 CN1C[C@H](C(N)=O)[C@H](c2cccc(N)c2)C1 ZINC000217663117 BC In-Stock Unstable SLC6A1 0 50 O=C(CSc1nc2ccccc2s1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217663124 HI In-Stock Unstable PREP 16 41 Cc1ccccc1/C=C/NC(=O)NCCc1ccccc1 ZINC000217663134 CH For-Sale Unstable MTNR1A 17 45 Cc1ccccc1/C=C/NC(=O)NCCc1ccccc1 ZINC000217663134 CH For-Sale Unstable MTNR1B 24 45 Cc1ccccc1/C=C/NC(=O)NCCc1ccccc1 ZINC000217663134 CH For-Sale Unstable SCN5A 0 40 Cc1ccccc1/C=C/NC(=O)NCCc1ccccc1 ZINC000217663134 CH For-Sale Unstable AMP1_PLAFQ 24 42 C[C@H](CCc1ccc2c(c1)OCO2)N[C@H]1CCC[C@@H](O)C1 ZINC000217663170 CF On-Demand Unstable SSTR3 102 34 COc1cc(CCC(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)on1 ZINC000217663194 ED In-Stock Unstable CHRNA4 28 47 O=C(CSc1nc2ccccc2s1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217663204 HI In-Stock Unstable PREP 16 41 CN1C[C@@H](C(N)=O)[C@H](c2cccc(N)c2)C1 ZINC000217663205 BC In-Stock Unstable SLC6A1 0 50 Brc1ccc(CN[C@@H]2CCN3CCCC[C@@H]23)s1 ZINC000217663254 DG On-Demand Unstable VACHT_TETCF 0 42 Cc1ccccc1/C=C/NC(=O)NC1CCCC1 ZINC000217663258 BG For-Sale Unstable EPHX2 25 45 O[C@@H](COc1ccccc1Cl)CN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217663259 IG On-Demand Unstable ADRB2 52 51 O[C@@H](COc1ccccc1Cl)CN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217663259 IG On-Demand Unstable ADRB1 17 45 O[C@@H](COc1ccccc1Cl)CN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217663259 IG On-Demand Unstable HTR1A 15 43 O[C@@H](COc1ccccc1Cl)CN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217663259 IG On-Demand Unstable SLC6A4 21 43 O[C@@H](COc1ccccc1Cl)CN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217663259 IG On-Demand Unstable SLC6A3 24 44 O[C@@H](COc1ccccc1Cl)CN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217663259 IG On-Demand Unstable ADRB3 53 51 O[C@@H](COc1ccccc1Cl)CN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217663259 IG On-Demand Unstable LTA4H 35 40 O[C@@H](COc1ccccc1Cl)CN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217663259 IG On-Demand Unstable ACOX1 40 31 O[C@@H](COc1ccccc1Cl)CN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217663259 IG On-Demand Unstable CCR1 15 43 O[C@@H](COc1ccccc1Cl)CN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217663259 IG On-Demand Unstable ABCB1 109 52 O[C@@H](COc1ccccc1Cl)CN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217663259 IG On-Demand Unstable HSP90AB1 38 44 O[C@@H](COc1ccccc1Cl)CN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217663259 IG On-Demand Unstable PSMB2 47 36 O[C@@H](COc1ccccc1Cl)CN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217663259 IG On-Demand Unstable PSMB1 41 37 BrCc1ccccc1N1CCCCc2ccccc21 ZINC000217663269 DK For-Sale Unstable AVPR2 21 40 COc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)NC[C@@H]1C[C@H]3C=C[C@@H]1C3)C(=O)OC2 ZINC000217663305 IH In-Stock Unstable IMPDH1 0 67 COc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)NC[C@@H]1C[C@H]3C=C[C@@H]1C3)C(=O)OC2 ZINC000217663305 IH In-Stock Unstable IMPDH2 0 67 COc1cc(/C=C/C(=O)N2CC[C@H](n3cc(-c4ccccc4)nn3)C2)cc(OC)c1OC ZINC000217663321 IG In-Stock Unstable PREP 18 40 COc1cc(/C=C/C(=O)N2CC[C@H](n3cc(-c4ccccc4)nn3)C2)cc(OC)c1OC ZINC000217663321 IG In-Stock Unstable CCR2 50 37 Brc1ccc(CN[C@H]2CCN3CCCC[C@@H]23)s1 ZINC000217663333 DG On-Demand Unstable VACHT_TETCF 0 42 O[C@H](COc1ccccc1Cl)CN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217663338 IG On-Demand Unstable ADRB2 52 51 O[C@H](COc1ccccc1Cl)CN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217663338 IG On-Demand Unstable ADRB1 17 45 O[C@H](COc1ccccc1Cl)CN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217663338 IG On-Demand Unstable HTR1A 15 43 O[C@H](COc1ccccc1Cl)CN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217663338 IG On-Demand Unstable SLC6A4 21 43 O[C@H](COc1ccccc1Cl)CN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217663338 IG On-Demand Unstable SLC6A3 24 44 O[C@H](COc1ccccc1Cl)CN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217663338 IG On-Demand Unstable ADRB3 53 51 O[C@H](COc1ccccc1Cl)CN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217663338 IG On-Demand Unstable LTA4H 35 40 O[C@H](COc1ccccc1Cl)CN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217663338 IG On-Demand Unstable ACOX1 40 31 O[C@H](COc1ccccc1Cl)CN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217663338 IG On-Demand Unstable CCR1 15 43 O[C@H](COc1ccccc1Cl)CN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217663338 IG On-Demand Unstable ABCB1 109 52 O[C@H](COc1ccccc1Cl)CN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217663338 IG On-Demand Unstable HSP90AB1 38 44 O[C@H](COc1ccccc1Cl)CN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217663338 IG On-Demand Unstable PSMB2 47 36 O[C@H](COc1ccccc1Cl)CN1CCN(CCOc2ccccc2Cl)CC1 ZINC000217663338 IG On-Demand Unstable PSMB1 41 37 CNC(=O)[C@@H]1CN(C)C[C@@H]1c1cccc(N)c1 ZINC000217663344 BC In-Stock Unstable SLC6A1 27 47 Cc1ccccc1/C=C/NC(=O)NCc1ccccc1Cl ZINC000217663374 DI For-Sale Unstable CXCL8 42 33 Cc1ccccc1/C=C/NC(=O)NCc1ccccc1Cl ZINC000217663374 DI For-Sale Unstable P2RX7 43 45 COc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)NC[C@H]1C[C@H]3C=C[C@@H]1C3)C(=O)OC2 ZINC000217663396 IH In-Stock Unstable IMPDH1 0 67 COc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)NC[C@H]1C[C@H]3C=C[C@@H]1C3)C(=O)OC2 ZINC000217663396 IH In-Stock Unstable IMPDH2 0 67 COc1cc(/C=C/C(=O)N2CC[C@@H](n3cc(-c4ccccc4)nn3)C2)cc(OC)c1OC ZINC000217663402 IG In-Stock Unstable PREP 18 40 COc1cc(/C=C/C(=O)N2CC[C@@H](n3cc(-c4ccccc4)nn3)C2)cc(OC)c1OC ZINC000217663402 IG In-Stock Unstable CCR2 50 37 O=C1CCN(C(=O)c2ccc(=O)[nH]c2)CC1 ZINC000217663405 BC On-Demand Unstable L3MBTL3 61 39 CNC(=O)[C@H]1CN(C)C[C@@H]1c1cccc(N)c1 ZINC000217663429 BC In-Stock Unstable SLC6A1 27 47 COc1ccc(CCNC(=O)N/C=C/c2ccccc2C)cc1OC ZINC000217663488 EH For-Sale Unstable MTNR1A 18 43 COc1ccc(CCNC(=O)N/C=C/c2ccccc2C)cc1OC ZINC000217663488 EH For-Sale Unstable MTNR1B 21 45 COc1ccc(CCNC(=O)N/C=C/c2ccccc2C)cc1OC ZINC000217663488 EH For-Sale Unstable NCE103 16 46 COc1ccc(CCNC(=O)N/C=C/c2ccccc2C)cc1OC ZINC000217663488 EH For-Sale Unstable ABCG2 16 43 Cc1c(C(=O)N2CC[C@H](n3cc(-c4ccccc4)nn3)C2)cnn1-c1ccccc1 ZINC000217663519 GH In-Stock Unstable PREP 15 41 O=C(O)/C=C\c1cccc(C(=O)NCc2ccncc2)c1 ZINC000217663543 CE For-Sale Unstable HDAC8 22 43 O=C(O)/C=C\c1cccc(C(=O)NCc2ccncc2)c1 ZINC000217663543 CE For-Sale Unstable NAMPT 55 42 C=CCNc1ccc(S(=O)(=O)N[C@@H](C)COC)cc1C(=O)O ZINC000217663565 ED In-Stock Unstable ADAMTS4 40 31 CCCOC[C@@H](NC(=O)OC(C)(C)C)C(=O)O ZINC000217663568 BD In-Stock Unstable PAPA1_CARPA 52 50 CCCOC[C@@H](NC(=O)OC(C)(C)C)C(=O)O ZINC000217663568 BD In-Stock Unstable CTSK 24 48 CCCOC[C@@H](NC(=O)OC(C)(C)C)C(=O)O ZINC000217663568 BD In-Stock Unstable PGA5 41 36 CCCOC[C@@H](NC(=O)OC(C)(C)C)C(=O)O ZINC000217663568 BD In-Stock Unstable FPR1 40 44 CCCOc1ccc(NC(=O)C(F)F)cc1OCCC ZINC000217663582 CG On-Demand Unstable ENPP1 46 30 Cc1c(C(=O)N2CC[C@@H](n3cc(-c4ccccc4)nn3)C2)cnn1-c1ccccc1 ZINC000217663601 GH In-Stock Unstable PREP 15 41 Cc1noc2nc(C(C)C)cc(C(=O)N3CCCN(Cc4ccc(Cl)cc4)CC3)c12 ZINC000217663631 IJ On-Demand Unstable LSS 16 40 C=CCNc1ccc(S(=O)(=O)N[C@H](C)COC)cc1C(=O)O ZINC000217663634 ED In-Stock Unstable ADAMTS4 40 31 Cc1nonc1CC(=O)N1CCCC[C@@H]1c1ccc(F)cc1 ZINC000217663643 DF In-Stock Unstable KCNA5 15 41 Cc1nonc1CC(=O)N1CCCC[C@@H]1c1ccc(F)cc1 ZINC000217663643 DF In-Stock Unstable CPT1A 85 40 CCOc1ccc(NC(=O)C(F)F)cc1OCC ZINC000217663702 CF On-Demand Unstable ENPP1 65 33 CCOc1ccc(NC(=O)C(F)F)cc1OCC ZINC000217663702 CF On-Demand Unstable KCNK3 38 40 CCOc1ccc(NC(=O)C(F)F)cc1OCC ZINC000217663702 CF On-Demand Unstable KCNK9 33 40 COC(=O)[C@H](CCSC)NC(=O)CCn1cc(C(C)=O)c2ccccc21 ZINC000217663703 GF In-Stock Unstable CNR1 29 46 COC(=O)[C@H](CCSC)NC(=O)CCn1cc(C(C)=O)c2ccccc21 ZINC000217663703 GF In-Stock Unstable CNR2 27 46 CCCCOCCCNC(=O)N/C=C/c1ccccc1C ZINC000217663704 CG For-Sale Unstable ACAT 0 43 BrC1(Br)C[C@H]1OCc1ccccc1 ZINC000217663730 DG For-Sale Unstable GRM2 18 41 Cc1nonc1CC(=O)N1CCCC[C@H]1c1ccc(F)cc1 ZINC000217663739 DF In-Stock Unstable KCNA5 15 41 Cc1nonc1CC(=O)N1CCCC[C@H]1c1ccc(F)cc1 ZINC000217663739 DF In-Stock Unstable CPT1A 85 40 CN1C[C@H](C(=O)O)[C@H](c2cccc(N)c2)C1 ZINC000217663747 BC In-Stock Unstable SLC6A1 23 53 CN1C[C@H](C(=O)O)[C@H](c2cccc(N)c2)C1 ZINC000217663747 BC In-Stock Unstable GRM3 24 40 COC[C@@H](C)NS(=O)(=O)c1ccc(NC2CC2)c(C(=O)O)c1 ZINC000217663749 ED In-Stock Unstable MMP13 23 40 COC[C@@H](C)NS(=O)(=O)c1ccc(NC2CC2)c(C(=O)O)c1 ZINC000217663749 ED In-Stock Unstable MMP2 15 40 Cc1c(C(=O)O)cc2ccccc2c1-c1ccccc1 ZINC000217663801 CJ For-Sale Unstable DHODH 32 41 Cc1c(C(=O)O)cc2ccccc2c1-c1ccccc1 ZINC000217663801 CJ For-Sale Unstable TSPO 18 63 Cc1c(C(=O)O)cc2ccccc2c1-c1ccccc1 ZINC000217663801 CJ For-Sale Unstable MT-CO2 51 40 c1ccc(CN[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217663817 BE On-Demand Unstable VACHT_TETCF 0 43 c1ccc(CN[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217663817 BE On-Demand Unstable SIGMAR1 18 43 c1ccc(CN[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217663817 BE On-Demand Unstable SLC18A3 66 43 Cc1ccccc1/C=C/NC(=O)NCc1cccnc1 ZINC000217663821 CF For-Sale Unstable PTAFR 30 41 Cc1ccccc1/C=C/NC(=O)NCc1cccnc1 ZINC000217663821 CF For-Sale Unstable NAMPT 80 51 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cc(OC)c3c(c2)OCO3)CC(=O)O4)cc1O ZINC000217663823 KI In-Stock Unstable AKR1B1 0 49 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cc(OC)c3c(c2)OCO3)CC(=O)O4)cc1O ZINC000217663823 KI In-Stock Unstable CYP1B1 56 35 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cc(OC)c3c(c2)OCO3)CC(=O)O4)cc1O ZINC000217663823 KI In-Stock Unstable CYP1A1 37 44 COC[C@H](C)NS(=O)(=O)c1ccc(NC2CC2)c(C(=O)O)c1 ZINC000217663828 ED In-Stock Unstable MMP13 23 40 COC[C@H](C)NS(=O)(=O)c1ccc(NC2CC2)c(C(=O)O)c1 ZINC000217663828 ED In-Stock Unstable MMP2 15 40 CN1C[C@@H](C(=O)O)[C@H](c2cccc(N)c2)C1 ZINC000217663829 BC In-Stock Unstable SLC6A1 0 53 CN1C[C@@H](C(=O)O)[C@H](c2cccc(N)c2)C1 ZINC000217663829 BC In-Stock Unstable GRM3 24 40 CN(Cc1ccon1)C(=O)c1ccc(CN2CCCCCC2)cc1 ZINC000217663854 EG In-Stock Unstable PLM2_PLAFA 29 40 C=C(CNS(=O)(=O)c1ccc([N+](=O)[O-])cc1)c1ccccc1 ZINC000217663874 DF On-Demand Unstable MMP2 18 41 C=C(CNS(=O)(=O)c1ccc([N+](=O)[O-])cc1)c1ccccc1 ZINC000217663874 DF On-Demand Unstable MMP9 16 43 C=C(CNS(=O)(=O)c1ccc([N+](=O)[O-])cc1)c1ccccc1 ZINC000217663874 DF On-Demand Unstable MMP1 24 41 c1ccc(CN[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217663892 BE On-Demand Unstable VACHT_TETCF 0 43 c1ccc(CN[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217663892 BE On-Demand Unstable SIGMAR1 18 43 c1ccc(CN[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217663892 BE On-Demand Unstable SLC18A3 66 43 Cc1noc2nc(C(C)C)cc(C(=O)Nc3ncc(Cc4ccccc4)s3)c12 ZINC000217663896 GJ On-Demand Unstable CDK5 21 41 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cc(OC)c3c(c2)OCO3)CC(=O)O4)cc1O ZINC000217663900 KI In-Stock Unstable AKR1B1 0 49 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cc(OC)c3c(c2)OCO3)CC(=O)O4)cc1O ZINC000217663900 KI In-Stock Unstable CYP1B1 56 35 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cc(OC)c3c(c2)OCO3)CC(=O)O4)cc1O ZINC000217663900 KI In-Stock Unstable CYP1A1 37 44 O=C(Cn1nnc2ccccc21)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217663922 FE In-Stock Unstable PREP 22 45 O=C(Cn1nnc2ccccc21)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217663922 FE In-Stock Unstable MGLL 0 40 COC[C@@H](C)NS(=O)(=O)c1ccc(NC2CCCC2)c(C(=O)O)c1 ZINC000217663937 FE In-Stock Unstable MMP13 28 41 COC[C@@H](C)NS(=O)(=O)c1ccc(NC2CCCC2)c(C(=O)O)c1 ZINC000217663937 FE In-Stock Unstable MMP2 19 41 CN1C[C@H](C(N)=O)[C@H](c2ccc(N)cc2)C1 ZINC000217663945 BC In-Stock Unstable SLC6A1 60 52 CN1C[C@H](C(N)=O)[C@H](c2ccc(N)cc2)C1 ZINC000217663945 BC In-Stock Unstable SLC6A4 16 52 CN1C[C@H](C(N)=O)[C@H](c2ccc(N)cc2)C1 ZINC000217663945 BC In-Stock Unstable SLC6A3 21 48 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cc(C(C)C)nc4onc(C)c34)CC2)cc1 ZINC000217663992 JI On-Demand Unstable SSTR5 46 37 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cc(C(C)C)nc4onc(C)c34)CC2)cc1 ZINC000217663992 JI On-Demand Unstable PDK1 40 34 Cc1cc(NS(=O)(=O)N2CCCC2)ccc1/C=C\C(=O)O ZINC000217663993 DD For-Sale Unstable LPL 44 35 O=C(Cn1nnc2ccccc21)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217664009 FE In-Stock Unstable PREP 22 45 O=C(Cn1nnc2ccccc21)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217664009 FE In-Stock Unstable MGLL 0 40 COC[C@H](C)NS(=O)(=O)c1ccc(NC2CCCC2)c(C(=O)O)c1 ZINC000217664010 FE In-Stock Unstable MMP13 20 41 COC[C@H](C)NS(=O)(=O)c1ccc(NC2CCCC2)c(C(=O)O)c1 ZINC000217664010 FE In-Stock Unstable MMP2 15 41 CN1C[C@@H](C(N)=O)[C@H](c2ccc(N)cc2)C1 ZINC000217664044 BC In-Stock Unstable SLC6A1 60 52 CN1C[C@@H](C(N)=O)[C@H](c2ccc(N)cc2)C1 ZINC000217664044 BC In-Stock Unstable SLC6A4 16 52 CN1C[C@@H](C(N)=O)[C@H](c2ccc(N)cc2)C1 ZINC000217664044 BC In-Stock Unstable SLC6A3 21 48 BrCc1ccc(N2CCCCc3ccccc32)cc1 ZINC000217664056 DK For-Sale Unstable AVPR2 15 42 Cc1ccccc1/C=C/NC(=O)N1CCC(Cc2ccccc2)CC1 ZINC000217664061 EJ For-Sale Unstable CHRM2 15 43 Cc1ccccc1/C=C/NC(=O)N1CCC(Cc2ccccc2)CC1 ZINC000217664061 EJ For-Sale Unstable GRIN2B 88 47 Cc1ccccc1/C=C/NC(=O)N1CCC(Cc2ccccc2)CC1 ZINC000217664061 EJ For-Sale Unstable SIGMAR1 21 44 Cc1ccccc1/C=C/NC(=O)N1CCC(Cc2ccccc2)CC1 ZINC000217664061 EJ For-Sale Unstable CCR3 54 43 O=C(NCc1ccccc1F)C(F)F ZINC000217664087 BD On-Demand Unstable CXCL8 23 42 O=C(NCc1ccccc1F)C(F)F ZINC000217664087 BD On-Demand Unstable AMP1_PLAFQ 47 39 COc1cccc(-c2cc(C(=O)N3CC[C@H](n4cc(-c5ccccc5)nn4)C3)n(C)n2)c1 ZINC000217664115 IG In-Stock Unstable PREP 24 41 COC[C@@H](C)NS(=O)(=O)c1ccc(NC2CCCCC2)c(C(=O)O)c1 ZINC000217664121 FE In-Stock Unstable MMP13 21 42 COC[C@@H](C)NS(=O)(=O)c1ccc(NC2CCCCC2)c(C(=O)O)c1 ZINC000217664121 FE In-Stock Unstable MMP2 15 42 C[C@@H]1CN(CC[C@@H](O)c2ccc(F)cc2)CCCO1 ZINC000217664140 CE For-Sale Unstable SLC6A3 21 46 CNC(=O)[C@@H]1CN(C)C[C@@H]1c1ccc(N)cc1 ZINC000217664163 BC In-Stock Unstable SLC6A1 111 58 CNC(=O)[C@@H]1CN(C)C[C@@H]1c1ccc(N)cc1 ZINC000217664163 BC In-Stock Unstable SLC6A4 23 49 CNC(=O)[C@@H]1CN(C)C[C@@H]1c1ccc(N)cc1 ZINC000217664163 BC In-Stock Unstable SLC6A3 35 45 COc1cccc(-c2cc(C(=O)N3CC[C@@H](n4cc(-c5ccccc5)nn4)C3)n(C)n2)c1 ZINC000217664202 IG In-Stock Unstable PREP 24 41 COC[C@H](C)NS(=O)(=O)c1ccc(NC2CCCCC2)c(C(=O)O)c1 ZINC000217664206 FE In-Stock Unstable MMP13 25 42 COC[C@H](C)NS(=O)(=O)c1ccc(NC2CCCCC2)c(C(=O)O)c1 ZINC000217664206 FE In-Stock Unstable MMP2 19 42 C[C@H]1CN(CC[C@@H](O)c2ccc(F)cc2)CCCO1 ZINC000217664218 CE For-Sale Unstable SLC6A3 21 46 O=C(NCc1cccc(C(F)(F)F)c1)C(F)F ZINC000217664220 CF On-Demand Unstable DEF 0 54 O=C(NCc1cccc(C(F)(F)F)c1)C(F)F ZINC000217664220 CF On-Demand Unstable CCR2 78 44 O=C(NCc1cccc(C(F)(F)F)c1)C(F)F ZINC000217664220 CF On-Demand Unstable AMP1_PLAFQ 31 44 O=C(NCc1cccc(C(F)(F)F)c1)C(F)F ZINC000217664220 CF On-Demand Unstable PHES 0 44 O=C(NCc1cccc(C(F)(F)F)c1)C(F)F ZINC000217664220 CF On-Demand Unstable CARM1 60 37 O=C(NCc1cccc(C(F)(F)F)c1)C(F)F ZINC000217664220 CF On-Demand Unstable PDS 66 47 Cc1noc2nc(C(C)C)cc(C(=O)NCc3ccc(OC(F)(F)F)cc3)c12 ZINC000217664222 GI On-Demand Unstable PPARA 21 46 CNC(=O)[C@H]1CN(C)C[C@@H]1c1ccc(N)cc1 ZINC000217664257 BC In-Stock Unstable SLC6A1 111 58 CNC(=O)[C@H]1CN(C)C[C@@H]1c1ccc(N)cc1 ZINC000217664257 BC In-Stock Unstable SLC6A4 23 49 CNC(=O)[C@H]1CN(C)C[C@@H]1c1ccc(N)cc1 ZINC000217664257 BC In-Stock Unstable SLC6A3 35 45 COc1ccc(CCNC(=O)N/C=C/c2ccccc2C)cc1 ZINC000217664282 DH For-Sale Unstable MTNR1A 69 45 COc1ccc(CCNC(=O)N/C=C/c2ccccc2C)cc1 ZINC000217664282 DH For-Sale Unstable MTNR1B 62 45 COc1ccc(CCNC(=O)N/C=C/c2ccccc2C)cc1 ZINC000217664282 DH For-Sale Unstable CA9 18 45 O=C(c1ccoc1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217664310 DF In-Stock Unstable PREP 17 42 O=C(c1ccoc1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217664310 DF In-Stock Unstable L3MBTL3 41 35 COc1ccc(Br)cc1CN[C@@H]1CCN2CCCC[C@@H]12 ZINC000217664319 EG On-Demand Unstable TACR1 34 40 COc1ccc(Br)cc1CN[C@@H]1CCN2CCCC[C@@H]12 ZINC000217664319 EG On-Demand Unstable QRFPR 41 35 COc1cc2c(cc1OC)CN(C(=O)C(F)F)CC2 ZINC000217664328 CD On-Demand Unstable SLC18A2 52 38 COc1cc2c(cc1OC)CN(C(=O)C(F)F)CC2 ZINC000217664328 CD On-Demand Unstable ABCB1B 51 34 COc1cc2c(cc1OC)CN(C(=O)C(F)F)CC2 ZINC000217664328 CD On-Demand Unstable ABCB1 25 51 Cc1noc2nc(C(C)C)cc(C(=O)Nc3cccc(Br)c3)c12 ZINC000217664340 FJ On-Demand Unstable KCNK3 79 38 Cc1noc2nc(C(C)C)cc(C(=O)Nc3cccc(Br)c3)c12 ZINC000217664340 FJ On-Demand Unstable KCNK9 64 37 CN1C[C@@H](C(=O)N(C)C)[C@@H](c2ccc(N)cc2)C1 ZINC000217664372 BD In-Stock Unstable SLC6A1 40 58 CN1C[C@@H](C(=O)N(C)C)[C@@H](c2ccc(N)cc2)C1 ZINC000217664372 BD In-Stock Unstable SLC6A3 15 45 Cc1ccccc1/C=C/NC(=O)NC[C@@H]1CCCO1 ZINC000217664400 CE For-Sale Unstable OXTR 26 40 Cc1ccccc1/C=C/NC(=O)NC[C@@H]1CCCO1 ZINC000217664400 CE For-Sale Unstable AVPR1A 17 40 Cc1ccccc1/C=C/NC(=O)NC[C@@H]1CCCO1 ZINC000217664400 CE For-Sale Unstable PDE8B 16 41 COc1ccc(Br)cc1CN[C@H]1CCN2CCCC[C@@H]12 ZINC000217664401 EG On-Demand Unstable TACR1 34 40 COc1ccc(Br)cc1CN[C@H]1CCN2CCCC[C@@H]12 ZINC000217664401 EG On-Demand Unstable QRFPR 41 35 O=C(c1ccoc1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217664407 DF In-Stock Unstable PREP 17 42 O=C(c1ccoc1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217664407 DF In-Stock Unstable L3MBTL3 41 35 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cc(OC)c(OC)cc2OC)CC(=O)O4)cc1O ZINC000217664423 KI In-Stock Unstable AKR1B1 22 49 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cc(OC)c(OC)cc2OC)CC(=O)O4)cc1O ZINC000217664423 KI In-Stock Unstable CYP1B1 58 36 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cc(OC)c(OC)cc2OC)CC(=O)O4)cc1O ZINC000217664423 KI In-Stock Unstable CYP1A1 43 49 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cc(OC)c(OC)cc2OC)CC(=O)O4)cc1O ZINC000217664423 KI In-Stock Unstable CYP1A2 34 42 CN1C[C@H](c2ccc(N)cc2)[C@@H](C(=O)N(C)C)C1 ZINC000217664431 BD In-Stock Unstable SLC6A1 40 58 CN1C[C@H](c2ccc(N)cc2)[C@@H](C(=O)N(C)C)C1 ZINC000217664431 BD In-Stock Unstable SLC6A3 15 45 O=C(NC[C@@H]1COc2ccccc2O1)C(F)F ZINC000217664450 BD On-Demand Unstable HTR1A 0 47 O=C(NC[C@@H]1COc2ccccc2O1)C(F)F ZINC000217664450 BD On-Demand Unstable UBLCP1 0 41 CCOc1ccc([C@@H]2CCCN2C(=O)c2cc(C(C)C)nc3onc(C)c23)cc1 ZINC000217664471 GK On-Demand Unstable COLA 58 36 CCOc1ccc([C@@H]2CCCN2C(=O)c2cc(C(C)C)nc3onc(C)c23)cc1 ZINC000217664471 GK On-Demand Unstable CPT1A 57 36 Cc1ccccc1/C=C/NC(=O)NC[C@H]1CCCO1 ZINC000217664484 CE For-Sale Unstable OXTR 26 40 Cc1ccccc1/C=C/NC(=O)NC[C@H]1CCCO1 ZINC000217664484 CE For-Sale Unstable AVPR1A 17 40 Cc1ccccc1/C=C/NC(=O)NC[C@H]1CCCO1 ZINC000217664484 CE For-Sale Unstable PDE8B 16 41 COc1ccc2cc(C(=O)N3CC[C@H](n4cc(-c5ccccc5)nn4)C3)[nH]c2c1 ZINC000217664504 GH In-Stock Unstable GRIN2B 30 46 COc1ccc2cc(C(=O)N3CC[C@H](n4cc(-c5ccccc5)nn4)C3)[nH]c2c1 ZINC000217664504 GH In-Stock Unstable FPR2 33 51 COc1ccc2cc(C(=O)N3CC[C@H](n4cc(-c5ccccc5)nn4)C3)[nH]c2c1 ZINC000217664504 GH In-Stock Unstable AKR1C3 17 40 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cc(OC)c(OC)cc2OC)CC(=O)O4)cc1O ZINC000217664509 KI In-Stock Unstable AKR1B1 22 49 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cc(OC)c(OC)cc2OC)CC(=O)O4)cc1O ZINC000217664509 KI In-Stock Unstable CYP1B1 58 36 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cc(OC)c(OC)cc2OC)CC(=O)O4)cc1O ZINC000217664509 KI In-Stock Unstable CYP1A1 43 49 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cc(OC)c(OC)cc2OC)CC(=O)O4)cc1O ZINC000217664509 KI In-Stock Unstable CYP1A2 34 42 O=C(NC[C@H]1COc2ccccc2O1)C(F)F ZINC000217664548 BD On-Demand Unstable HTR1A 0 47 O=C(NC[C@H]1COc2ccccc2O1)C(F)F ZINC000217664548 BD On-Demand Unstable UBLCP1 0 41 CCOc1ccc([C@H]2CCCN2C(=O)c2cc(C(C)C)nc3onc(C)c23)cc1 ZINC000217664549 GK On-Demand Unstable COLA 58 36 CCOc1ccc([C@H]2CCCN2C(=O)c2cc(C(C)C)nc3onc(C)c23)cc1 ZINC000217664549 GK On-Demand Unstable CPT1A 57 36 CN1C[C@H](C(=O)O)[C@H](c2ccc(N)cc2)C1 ZINC000217664557 BC In-Stock Unstable SLC6A1 70 55 CN1C[C@H](C(=O)O)[C@H](c2ccc(N)cc2)C1 ZINC000217664557 BC In-Stock Unstable SLC6A4 19 55 CN1C[C@H](C(=O)O)[C@H](c2ccc(N)cc2)C1 ZINC000217664557 BC In-Stock Unstable SLC6A3 24 45 Cc1ccccc1/C=C/NC(=O)NCc1ccc(Cl)cc1 ZINC000217664578 DI For-Sale Unstable U38 0 40 Cc1ccccc1/C=C/NC(=O)NCc1ccc(Cl)cc1 ZINC000217664578 DI For-Sale Unstable AMP1_PLAFQ 22 40 CCCCCNC(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217664589 CF For-Sale Unstable DRD2 17 41 CCCCCNC(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217664589 CF For-Sale Unstable DRD4 40 30 CCCCCNC(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217664589 CF For-Sale Unstable DRD3 37 41 CCCCCNC(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217664589 CF For-Sale Unstable LTB4R 28 41 CCCCCNC(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217664589 CF For-Sale Unstable PLA2G4B 31 40 CCCCCNC(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217664589 CF For-Sale Unstable HDAC9 16 41 CCCCCNC(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217664589 CF For-Sale Unstable PTGDR 19 43 COc1ccc2cc(C(=O)N3CC[C@@H](n4cc(-c5ccccc5)nn4)C3)[nH]c2c1 ZINC000217664594 GH In-Stock Unstable GRIN2B 30 46 COc1ccc2cc(C(=O)N3CC[C@@H](n4cc(-c5ccccc5)nn4)C3)[nH]c2c1 ZINC000217664594 GH In-Stock Unstable FPR2 33 51 COc1ccc2cc(C(=O)N3CC[C@@H](n4cc(-c5ccccc5)nn4)C3)[nH]c2c1 ZINC000217664594 GH In-Stock Unstable AKR1C3 17 40 CN(Cc1ccccc1)C(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217664625 HF In-Stock Unstable HTR1D 38 41 CN(Cc1ccccc1)C(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217664625 HF In-Stock Unstable HTR1B 30 41 CN(Cc1ccccc1)C(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217664625 HF In-Stock Unstable EDNRA 27 42 CN(Cc1ccccc1)C(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217664625 HF In-Stock Unstable TACR1 31 46 CN(Cc1ccccc1)C(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217664625 HF In-Stock Unstable MC4R 44 46 CN(Cc1ccccc1)C(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217664625 HF In-Stock Unstable TACR2 63 44 CN(Cc1ccccc1)C(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217664625 HF In-Stock Unstable CCKAR 39 41 CN(Cc1ccccc1)C(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217664625 HF In-Stock Unstable MMP14 42 33 CN(Cc1ccccc1)C(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217664625 HF In-Stock Unstable MMP11 46 33 CN(Cc1ccccc1)C(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217664625 HF In-Stock Unstable CCKBR 45 38 CN(Cc1ccccc1)C(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217664625 HF In-Stock Unstable GHSR 44 37 CN(Cc1ccccc1)C(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217664625 HF In-Stock Unstable MC1R 22 43 CN1C[C@@H](C(=O)O)[C@H](c2ccc(N)cc2)C1 ZINC000217664632 BC In-Stock Unstable SLC6A1 70 55 CN1C[C@@H](C(=O)O)[C@H](c2ccc(N)cc2)C1 ZINC000217664632 BC In-Stock Unstable SLC6A4 19 55 CN1C[C@@H](C(=O)O)[C@H](c2ccc(N)cc2)C1 ZINC000217664632 BC In-Stock Unstable SLC6A3 24 45 C=C(CC)COc1ccc(Cl)cc1/C=C\C(=O)O ZINC000217664652 CH For-Sale Unstable PTGER3 17 41 C=C(CC)COc1ccc(Cl)cc1/C=C\C(=O)O ZINC000217664652 CH For-Sale Unstable PTGDR2 39 40 C=C(CC)COc1ccc(Cl)cc1/C=C\C(=O)O ZINC000217664652 CH For-Sale Unstable AKR1C3 23 40 CCCCN(C)C(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217664667 CF For-Sale Unstable THRA 45 43 CCCCN(C)C(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217664667 CF For-Sale Unstable THRB 24 43 O=C(Cc1ccc2c(c1)OCO2)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217664698 GF In-Stock Unstable PREP 20 43 O=C(Cc1ccc2c(c1)OCO2)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217664698 GF In-Stock Unstable NOS2 60 34 O=C(Cc1ccc2c(c1)OCO2)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217664698 GF In-Stock Unstable SSTR3 74 34 Cc1ccccc1/C=C/NC(=O)N[C@H](C)c1ccccc1 ZINC000217664700 CI For-Sale Unstable KCNQ2 47 36 CC(C)c1ccc([C@@H]2CN(C)C[C@@H]2C(=O)O)cc1 ZINC000217664749 BF In-Stock Unstable SLC6A1 100 52 CC(C)c1ccc([C@@H]2CN(C)C[C@@H]2C(=O)O)cc1 ZINC000217664749 BF In-Stock Unstable SLC6A4 22 52 CC(C)c1ccc([C@@H]2CN(C)C[C@@H]2C(=O)O)cc1 ZINC000217664749 BF In-Stock Unstable SLC6A3 30 46 CCCCN(C)C(=O)c1cc(/C=C\C(=O)O)ccc1F ZINC000217664750 CF For-Sale Unstable AKR1C3 28 40 O=C(Cc1ccc2c(c1)OCO2)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217664768 GF In-Stock Unstable PREP 20 43 O=C(Cc1ccc2c(c1)OCO2)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217664768 GF In-Stock Unstable NOS2 60 34 O=C(Cc1ccc2c(c1)OCO2)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217664768 GF In-Stock Unstable SSTR3 74 34 C=C(CC)COc1c(/C=C\C(=O)O)cccc1OCC ZINC000217664770 CH For-Sale Unstable PTGER2 17 41 C=C(CC)COc1c(/C=C\C(=O)O)cccc1OCC ZINC000217664770 CH For-Sale Unstable PTGER3 21 41 Cc1ccccc1/C=C/NC(=O)N[C@@H](C)c1ccccc1 ZINC000217664774 CI For-Sale Unstable KCNQ2 47 36 COc1ccc(NC(C)=O)cc1NC(=O)C(F)F ZINC000217664812 CD On-Demand Unstable ENPP1 50 30 CC(C)c1ccc([C@H]2CN(C)C[C@@H]2C(=O)O)cc1 ZINC000217664829 BF In-Stock Unstable SLC6A1 100 52 CC(C)c1ccc([C@H]2CN(C)C[C@@H]2C(=O)O)cc1 ZINC000217664829 BF In-Stock Unstable SLC6A4 22 52 CC(C)c1ccc([C@H]2CN(C)C[C@@H]2C(=O)O)cc1 ZINC000217664829 BF In-Stock Unstable SLC6A3 30 46 O=C(O)/C=C\c1cccc(C(=O)Nc2cccc(F)c2)c1 ZINC000217664836 CG For-Sale Anodyne MMP2 0 61 O=C(O)/C=C\c1cccc(C(=O)Nc2cccc(F)c2)c1 ZINC000217664836 CG For-Sale Anodyne MMP9 0 57 O=C(O)/C=C\c1cccc(C(=O)Nc2cccc(F)c2)c1 ZINC000217664836 CG For-Sale Anodyne MMP1 0 61 O=C(O)/C=C\c1cccc(C(=O)Nc2cccc(F)c2)c1 ZINC000217664836 CG For-Sale Anodyne BTK 19 41 O=C(O)/C=C\c1cccc(C(=O)Nc2cccc(F)c2)c1 ZINC000217664836 CG For-Sale Anodyne TAAR1 40 44 O=C(O)/C=C\c1cccc(C(=O)Nc2cccc(F)c2)c1 ZINC000217664836 CG For-Sale Anodyne AKR1C3 47 38 O=C(O)/C=C\c1cccc(C(=O)Nc2cccc(F)c2)c1 ZINC000217664836 CG For-Sale Anodyne RHOA 0 43 O=C(O)/C=C\c1cccc(C(=O)Nc2cccc(F)c2)c1 ZINC000217664836 CG For-Sale Anodyne PARP14 0 44 O=C(O)/C=C\c1cccc(C(=O)Nc2cccc(F)c2)c1 ZINC000217664836 CG For-Sale Anodyne KCNK3 129 62 O=C(O)/C=C\c1cccc(C(=O)Nc2cccc(F)c2)c1 ZINC000217664836 CG For-Sale Anodyne KCNK9 73 58 O=C(O)/C=C\c1cccc(C(=O)Nc2cccc(F)c2)c1 ZINC000217664836 CG For-Sale Anodyne PARP10 0 44 C[C@@H](O)c1cc2n(n1)CCCN(Cc1cc(Cl)ccc1OCC(N)=O)C2 ZINC000217664865 GD In-Stock Unstable PTGER1 40 40 CC(=O)NCC(=O)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217664884 DC In-Stock Unstable PREP 33 44 C=C(CC)COc1ccc(OC)cc1/C=C\C(=O)O ZINC000217664895 CG For-Sale Unstable PTGER2 41 43 C=C(CC)COc1ccc(OC)cc1/C=C\C(=O)O ZINC000217664895 CG For-Sale Unstable PTGER4 23 43 C=C(CC)COc1ccc(OC)cc1/C=C\C(=O)O ZINC000217664895 CG For-Sale Unstable CYP1B1 35 40 C=C(CC)COc1ccc(OC)cc1/C=C\C(=O)O ZINC000217664895 CG For-Sale Unstable PTGER3 18 43 C=C(CC)COc1ccc(OC)cc1/C=C\C(=O)O ZINC000217664895 CG For-Sale Unstable LTB4R 34 40 C=C(CC)COc1ccc(OC)cc1/C=C\C(=O)O ZINC000217664895 CG For-Sale Unstable CYP1A1 34 40 C=C(CC)COc1ccc(OC)cc1/C=C\C(=O)O ZINC000217664895 CG For-Sale Unstable CYP1A2 15 40 C=C(CC)COc1ccc(OC)cc1/C=C\C(=O)O ZINC000217664895 CG For-Sale Unstable CYSP_PLAFA 40 42 N#CCCCCNS(=O)(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217664899 DD On-Demand Unstable TBXAS1 23 40 CN(C)[C@@H](CNC(=O)CN1CCN(CCOc2ccccc2Cl)CC1)c1ccccc1 ZINC000217664907 IF On-Demand Unstable SLC6A3 19 40 CN1C[C@H](C(=O)O)[C@H](c2ccc(C(C)(C)C)cc2)C1 ZINC000217664931 CF In-Stock Unstable SLC6A4 16 54 CN1C[C@H](C(=O)O)[C@H](c2ccc(C(C)(C)C)cc2)C1 ZINC000217664931 CF In-Stock Unstable SLC6A3 21 44 C[C@H](O)c1cc2n(n1)CCCN(Cc1cc(Cl)ccc1OCC(N)=O)C2 ZINC000217664950 GD In-Stock Unstable PTGER1 40 40 CC(=O)NCC(=O)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217664968 DC In-Stock Unstable PREP 33 44 CN(C)[C@H](CNC(=O)CN1CCN(CCOc2ccccc2Cl)CC1)c1ccccc1 ZINC000217664979 IF On-Demand Unstable SLC6A3 19 40 COc1ccc(CNC(=O)N/C=C/c2ccccc2C)cc1 ZINC000217665007 CG For-Sale Unstable ANPEP 24 44 COc1ccc(CNC(=O)N/C=C/c2ccccc2C)cc1 ZINC000217665007 CG For-Sale Unstable PTGER4 0 43 COc1ccc(CNC(=O)N/C=C/c2ccccc2C)cc1 ZINC000217665007 CG For-Sale Unstable MTNR1A 23 47 COc1ccc(CNC(=O)N/C=C/c2ccccc2C)cc1 ZINC000217665007 CG For-Sale Unstable MTNR1B 18 47 COc1ccc(CNC(=O)N/C=C/c2ccccc2C)cc1 ZINC000217665007 CG For-Sale Unstable CA9 18 43 COc1ccc(CNC(=O)N/C=C/c2ccccc2C)cc1 ZINC000217665007 CG For-Sale Unstable KCNJ2 0 42 CN(C)CCCNC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217665016 CD For-Sale Unstable HDAC8 18 43 CN1C[C@@H](C(=O)O)[C@H](c2ccc(C(C)(C)C)cc2)C1 ZINC000217665019 CF In-Stock Unstable SLC6A4 16 54 CN1C[C@@H](C(=O)O)[C@H](c2ccc(C(C)(C)C)cc2)C1 ZINC000217665019 CF In-Stock Unstable SLC6A3 21 44 COc1ccc(CN(C)C(=O)C(F)F)cc1 ZINC000217665065 BD On-Demand Unstable BMP1 51 40 O=C(Cc1cccnc1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217665082 EE In-Stock Unstable C3AR1 43 38 O=C(Cc1cccnc1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217665082 EE In-Stock Unstable PREP 26 49 O=C(Cc1cccc(O)c1)N[C@@H]1CCCC[C@@H]1CO ZINC000217665151 CD On-Demand Unstable SSTR3 25 50 COC(=O)C[C@@H](C1=C(O)C(=O)c2ccccc2C1=O)c1cccc(O)c1 ZINC000217665154 FF In-Stock Unstable KCNA5 32 40 O=C(Cc1cccnc1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217665169 EE In-Stock Unstable C3AR1 43 38 O=C(Cc1cccnc1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217665169 EE In-Stock Unstable PREP 26 49 COc1ccc(NC(=O)C(F)F)cc1S(N)(=O)=O ZINC000217665182 CC For-Sale Unstable CA2 36 44 COc1ccc(NC(=O)C(F)F)cc1S(N)(=O)=O ZINC000217665182 CC For-Sale Unstable CA1 35 43 COc1ccc(NC(=O)C(F)F)cc1S(N)(=O)=O ZINC000217665182 CC For-Sale Unstable COLA 47 33 COc1ccc(NC(=O)C(F)F)cc1S(N)(=O)=O ZINC000217665182 CC For-Sale Unstable CPT1A 44 33 COc1ccc(NC(=O)C(F)F)cc1S(N)(=O)=O ZINC000217665182 CC For-Sale Unstable CPT2 43 32 COc1ccc(NC(=O)C(F)F)cc1S(N)(=O)=O ZINC000217665182 CC For-Sale Unstable CA14 22 44 COc1ccc(NC(=O)C(F)F)cc1S(N)(=O)=O ZINC000217665182 CC For-Sale Unstable CA12 35 43 COc1ccc(NC(=O)C(F)F)cc1S(N)(=O)=O ZINC000217665182 CC For-Sale Unstable CA9 33 43 COc1ccc(NC(=O)C(F)F)cc1S(N)(=O)=O ZINC000217665182 CC For-Sale Unstable ENPP1 49 30 COc1ccc(NC(=O)C(F)F)cc1S(N)(=O)=O ZINC000217665182 CC For-Sale Unstable P96878_MYCTU 43 42 N#Cc1ccc(OCCN2CCC[C@@H]3CCCC[C@H]32)cc1 ZINC000217665205 CH For-Sale Unstable LTA4H 44 40 N#Cc1ccc(OCCN2CCC[C@@H]3CCCC[C@H]32)cc1 ZINC000217665205 CH For-Sale Unstable HRH3 51 60 N#Cc1ccc(OCCN2CCC[C@@H]3CCCC[C@H]32)cc1 ZINC000217665205 CH For-Sale Unstable CHRNA10 41 40 N#Cc1ccc(OCCN2CCC[C@@H]3CCCC[C@H]32)cc1 ZINC000217665205 CH For-Sale Unstable PSMB1 40 35 N#Cc1ccc(OCCN2CCC[C@@H]3CCCC[C@H]32)cc1 ZINC000217665205 CH For-Sale Unstable MEN1 52 45 COC(=O)C[C@H](C1=C(O)C(=O)c2ccccc2C1=O)c1cccc(O)c1 ZINC000217665226 FF In-Stock Unstable KCNA5 32 40 O=C(Cc1cccc(O)c1)N[C@H]1CCCC[C@@H]1CO ZINC000217665231 CD On-Demand Unstable SSTR3 25 50 O=C(c1ccc(F)cc1Cl)N1CCCO[C@@H](CN2CCCC2)C1 ZINC000217665238 EF In-Stock Unstable SLC6A1 33 43 O=C(c1ccc(F)cc1Cl)N1CCCO[C@@H](CN2CCCC2)C1 ZINC000217665238 EF In-Stock Unstable P2RX7 28 44 COC[C@@H](C)NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217665243 GE In-Stock Unstable TRY2_BOVIN 43 31 COC[C@@H](C)NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217665243 GE In-Stock Unstable ADAMTS4 55 34 Cc1ccccc1/C=C/NC(=O)NCc1ccc2c(c1)OCO2 ZINC000217665245 DG For-Sale Unstable PDE5A 35 42 Cc1ccccc1/C=C/NC(=O)NCc1ccc2c(c1)OCO2 ZINC000217665245 DG For-Sale Unstable BMP1 44 39 Cc1ccccc1/C=C/NC(=O)NCc1ccc2c(c1)OCO2 ZINC000217665245 DG For-Sale Unstable SCN9A 28 43 Cc1ccccc1/C=C/NC(=O)NCc1ccc2c(c1)OCO2 ZINC000217665245 DG For-Sale Unstable NOS2 92 35 Cc1ccccc1/C=C/NC(=O)NCc1ccc2c(c1)OCO2 ZINC000217665245 DG For-Sale Unstable MCHR1 17 46 Oc1cccc(CN[C@@H]2CCN3CCCC[C@@H]23)c1 ZINC000217665269 BE On-Demand Unstable SIGMAR1 15 40 Oc1cccc(CN[C@@H]2CCN3CCCC[C@@H]23)c1 ZINC000217665269 BE On-Demand Unstable SLC18A3 40 35 O=C(Cc1ccsc1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217665271 EG In-Stock Unstable PREP 24 46 COc1ccc(C(=O)NCC2CCC2)cc1/C=C\C(=O)O ZINC000217665289 CE For-Sale Unstable CACNA1I 56 37 COc1ccc(C(=O)NCC2CCC2)cc1/C=C\C(=O)O ZINC000217665289 CE For-Sale Unstable ACKR3 46 33 N#Cc1ccc(OCCN2CCC[C@H]3CCCC[C@H]32)cc1 ZINC000217665290 CH For-Sale Unstable LTA4H 44 40 N#Cc1ccc(OCCN2CCC[C@H]3CCCC[C@H]32)cc1 ZINC000217665290 CH For-Sale Unstable HRH3 51 60 N#Cc1ccc(OCCN2CCC[C@H]3CCCC[C@H]32)cc1 ZINC000217665290 CH For-Sale Unstable CHRNA10 41 40 N#Cc1ccc(OCCN2CCC[C@H]3CCCC[C@H]32)cc1 ZINC000217665290 CH For-Sale Unstable PSMB1 40 35 N#Cc1ccc(OCCN2CCC[C@H]3CCCC[C@H]32)cc1 ZINC000217665290 CH For-Sale Unstable MEN1 52 45 O=C(Cc1cccc(O)c1)N[C@@H]1CCCC[C@H]1CO ZINC000217665320 CD On-Demand Unstable SSTR3 25 50 COC[C@H](C)NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217665328 GE In-Stock Unstable TRY2_BOVIN 52 35 COC[C@H](C)NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217665328 GE In-Stock Unstable MMP12 42 37 COC[C@H](C)NS(=O)(=O)c1ccc(NCc2ccccc2)c(C(=O)O)c1 ZINC000217665328 GE In-Stock Unstable ADAMTS4 55 34 O=C(c1ccc(F)cc1Cl)N1CCCO[C@H](CN2CCCC2)C1 ZINC000217665329 EF In-Stock Unstable SLC6A1 33 43 O=C(c1ccc(F)cc1Cl)N1CCCO[C@H](CN2CCCC2)C1 ZINC000217665329 EF In-Stock Unstable P2RX7 28 44 CN1C[C@H](C(=O)O)[C@H](c2ccccc2F)C1 ZINC000217665339 BD In-Stock Unstable MC4R 23 51 CN1C[C@H](C(=O)O)[C@H](c2ccccc2F)C1 ZINC000217665339 BD In-Stock Unstable HSD17B2 0 43 Oc1cccc(CN[C@H]2CCN3CCCC[C@@H]23)c1 ZINC000217665340 BE On-Demand Unstable SIGMAR1 15 40 Oc1cccc(CN[C@H]2CCN3CCCC[C@@H]23)c1 ZINC000217665340 BE On-Demand Unstable SLC18A3 40 35 O=C(CCn1cnc2sc3c(c2c1=O)CCCCC3)Nc1cccc(F)c1 ZINC000217665347 GH On-Demand Unstable HTR1B 20 40 O=C(Cc1ccsc1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217665356 EG In-Stock Unstable PREP 24 46 CC(C)C[C@@H](C)NC(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217665366 CF For-Sale Unstable CTSL 15 40 Cc1ccccc1/C=C/NC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217665370 EE For-Sale Unstable CA2 104 56 Cc1ccccc1/C=C/NC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217665370 EE For-Sale Unstable CA6 15 40 Cc1ccccc1/C=C/NC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217665370 EE For-Sale Unstable CA1 99 56 Cc1ccccc1/C=C/NC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217665370 EE For-Sale Unstable CA7 38 48 Cc1ccccc1/C=C/NC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217665370 EE For-Sale Unstable CA5B 46 48 Cc1ccccc1/C=C/NC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217665370 EE For-Sale Unstable CA4 76 56 Cc1ccccc1/C=C/NC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217665370 EE For-Sale Unstable CA5A 57 48 Cc1ccccc1/C=C/NC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217665370 EE For-Sale Unstable CA14 34 48 Cc1ccccc1/C=C/NC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217665370 EE For-Sale Unstable CA12 84 56 Cc1ccccc1/C=C/NC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217665370 EE For-Sale Unstable CA9 88 51 Cc1ccccc1/C=C/NC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217665370 EE For-Sale Unstable UREA_CANEN 27 42 Cc1ccccc1/C=C/NC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217665370 EE For-Sale Unstable IDO1 0 44 Cc1ccccc1/C=C/NC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217665370 EE For-Sale Unstable CYNT 40 41 Cc1ccccc1/C=C/NC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217665370 EE For-Sale Unstable NCE103 44 46 Cc1ccccc1/C=C/NC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217665370 EE For-Sale Unstable MTCA1 64 56 Cc1ccccc1/C=C/NC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217665370 EE For-Sale Unstable P96878_MYCTU 80 56 O=C(Cc1cccc(O)c1)N[C@H]1CCCC[C@H]1CO ZINC000217665417 CD On-Demand Unstable SSTR3 25 50 CC(C)C[C@H](C)NC(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217665436 CF For-Sale Unstable CTSL 15 40 O=C(c1ccc(C(F)(F)F)nc1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217665453 GG In-Stock Unstable SFRP1 31 45 O=C(c1ccc(C(F)(F)F)nc1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217665453 GG In-Stock Unstable L3MBTL3 41 37 COC[C@@H](C)NS(=O)(=O)c1ccc(N[C@@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217665454 GF In-Stock Unstable ADAMTS4 41 32 C[C@@H](N[C@@H]1CCN2CCCC[C@@H]12)c1ccc(Cl)c(Cl)c1 ZINC000217665459 DI For-Sale Unstable OPRK1 0 42 C[C@@H](N[C@@H]1CCN2CCCC[C@@H]12)c1ccc(Cl)c(Cl)c1 ZINC000217665459 DI For-Sale Unstable SLC6A3 15 47 CN1C[C@H](C(=O)O)[C@H](c2cccc(F)c2)C1 ZINC000217665463 BD In-Stock Unstable SLC6A3 17 47 CN1C[C@H](C(=O)O)[C@H](c2cccc(F)c2)C1 ZINC000217665463 BD In-Stock Unstable MC4R 0 47 CN1C[C@H](C(=O)O)[C@H](c2cccc(F)c2)C1 ZINC000217665463 BD In-Stock Unstable CCR5 103 40 CCN(CCC(=O)Nc1cccc(S(=O)(=O)N2CCCC2)c1)Cc1ccccc1 ZINC000217665468 HG On-Demand Unstable LPL 44 38 CCN(CCC(=O)Nc1cccc(S(=O)(=O)N2CCCC2)c1)Cc1ccccc1 ZINC000217665468 HG On-Demand Unstable CA4 15 41 CCN(CCC(=O)Nc1cccc(S(=O)(=O)N2CCCC2)c1)Cc1ccccc1 ZINC000217665468 HG On-Demand Unstable TGM2 47 48 CCN(CCC(=O)Nc1cccc(S(=O)(=O)N2CCCC2)c1)Cc1ccccc1 ZINC000217665468 HG On-Demand Unstable ST14 43 39 CCN(CCC(=O)Nc1cccc(S(=O)(=O)N2CCCC2)c1)Cc1ccccc1 ZINC000217665468 HG On-Demand Unstable F13A1 74 48 CCN(CCC(=O)Nc1cccc(S(=O)(=O)N2CCCC2)c1)Cc1ccccc1 ZINC000217665468 HG On-Demand Unstable AKR1C3 44 42 CCN(CCC(=O)Nc1cccc(S(=O)(=O)N2CCCC2)c1)Cc1ccccc1 ZINC000217665468 HG On-Demand Unstable RORC 18 42 CCN(CCC(=O)Nc1cccc(S(=O)(=O)N2CCCC2)c1)Cc1ccccc1 ZINC000217665468 HG On-Demand Unstable NAMPT 23 43 Cc1ccccc1/C=C/NC(=O)NCc1ccccc1 ZINC000217665485 CG For-Sale Unstable ANPEP 27 42 Cc1ccccc1/C=C/NC(=O)NCc1ccccc1 ZINC000217665485 CG For-Sale Unstable PDS 47 35 CC(C)C[C@@H](C)NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217665515 CF For-Sale Unstable CTSK 15 40 CC(C)C[C@@H](C)NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217665515 CF For-Sale Unstable CTSL 18 40 CC(C)C[C@@H](C)NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217665515 CF For-Sale Unstable HDAC8 21 44 CC(C)C[C@@H](C)NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217665515 CF For-Sale Unstable CAPN1 24 40 O=C(c1ccc(C(F)(F)F)nc1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217665530 GG In-Stock Unstable SFRP1 25 45 COC[C@H](C)NS(=O)(=O)c1ccc(N[C@@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217665532 GF In-Stock Unstable ADAMTS4 41 32 C[C@H](N[C@@H]1CCN2CCCC[C@@H]12)c1ccc(Cl)c(Cl)c1 ZINC000217665540 DI On-Demand Unstable OPRK1 0 42 C[C@H](N[C@@H]1CCN2CCCC[C@@H]12)c1ccc(Cl)c(Cl)c1 ZINC000217665540 DI On-Demand Unstable SLC6A3 15 47 CN1C[C@H](C(=O)O)[C@H](c2c(F)cccc2Cl)C1 ZINC000217665597 CE In-Stock Unstable SLC6A1 50 37 NC/C=C\CSc1nnnn1-c1ccccc1 ZINC000217665602 BD For-Sale Unstable CELA2A 31 45 CC(C)C[C@H](C)NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217665605 CF For-Sale Unstable CTSK 15 40 CC(C)C[C@H](C)NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217665605 CF For-Sale Unstable CTSL 18 40 CC(C)C[C@H](C)NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217665605 CF For-Sale Unstable HDAC8 21 44 CC(C)C[C@H](C)NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217665605 CF For-Sale Unstable CAPN1 24 40 C[C@@H](N[C@H]1CCN2CCCC[C@@H]12)c1ccc(Cl)c(Cl)c1 ZINC000217665613 DI For-Sale Unstable OPRK1 0 42 C[C@@H](N[C@H]1CCN2CCCC[C@@H]12)c1ccc(Cl)c(Cl)c1 ZINC000217665613 DI For-Sale Unstable SLC6A3 15 47 COC[C@@H](C)NS(=O)(=O)c1ccc(N[C@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217665630 GF In-Stock Unstable ADAMTS4 41 32 COc1ccc(C(=O)N2CC[C@H](n3cc(-c4ccccc4)nn3)C2)cn1 ZINC000217665635 EE In-Stock Unstable PREP 19 42 COc1ccc(C(=O)N2CC[C@H](n3cc(-c4ccccc4)nn3)C2)cn1 ZINC000217665635 EE In-Stock Unstable L3MBTL3 41 37 CCOC(=O)N1CCN(Cc2cc(C)c(O)c(C)c2)CC1 ZINC000217665642 CE On-Demand Unstable MGLL 0 40 CN1C[C@@H](C(=O)O)[C@H](c2c(F)cccc2Cl)C1 ZINC000217665676 CE In-Stock Unstable SLC6A1 50 37 O=C(O)/C=C\c1ccc(C(=O)N2CCS(=O)(=O)CC2)cc1 ZINC000217665701 DC For-Sale Unstable L3MBTL3 47 36 O=C(O)/C=C\c1ccc(C(=O)N2CCS(=O)(=O)CC2)cc1 ZINC000217665701 DC For-Sale Unstable GPR183 0 49 C[C@H](N[C@H]1CCN2CCCC[C@@H]12)c1ccc(Cl)c(Cl)c1 ZINC000217665702 DI On-Demand Unstable OPRK1 0 42 C[C@H](N[C@H]1CCN2CCCC[C@@H]12)c1ccc(Cl)c(Cl)c1 ZINC000217665702 DI On-Demand Unstable SLC6A3 15 47 C[C@@H]1CCCCN1CCC(=O)Nc1ccc2c(c1)CCC2 ZINC000217665708 CG On-Demand Unstable HRH3 64 50 C[C@@H]1CCCCN1CCC(=O)Nc1ccc2c(c1)CCC2 ZINC000217665708 CG On-Demand Unstable PTPRF 41 31 C[C@@H]1CCCCN1CCC(=O)Nc1ccc2c(c1)CCC2 ZINC000217665708 CG On-Demand Unstable TERT 20 45 C[C@@H]1CCCCN1CCC(=O)Nc1ccc2c(c1)CCC2 ZINC000217665708 CG On-Demand Unstable CALCRL 63 33 COC[C@H](C)NS(=O)(=O)c1ccc(N[C@H](C)c2ccccc2)c(C(=O)O)c1 ZINC000217665710 GF In-Stock Unstable ADAMTS4 41 32 COc1ccc(C(=O)N2CC[C@@H](n3cc(-c4ccccc4)nn3)C2)cn1 ZINC000217665713 EE In-Stock Unstable PREP 19 42 COc1ccc(C(=O)N2CC[C@@H](n3cc(-c4ccccc4)nn3)C2)cn1 ZINC000217665713 EE In-Stock Unstable L3MBTL3 41 37 O=c1cc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)oc(CN2CCc3ccccc3C2)c1O ZINC000217665744 JF In-Stock Unstable CHRNA4 29 51 O=C(O)/C=C\c1cccc(C(=O)N2CCS(=O)(=O)CC2)c1 ZINC000217665792 DC For-Sale Unstable GPR183 0 42 C[C@H]1CCCCN1CCC(=O)Nc1ccc2c(c1)CCC2 ZINC000217665795 CG On-Demand Unstable HRH3 64 50 C[C@H]1CCCCN1CCC(=O)Nc1ccc2c(c1)CCC2 ZINC000217665795 CG On-Demand Unstable PTPRF 41 31 C[C@H]1CCCCN1CCC(=O)Nc1ccc2c(c1)CCC2 ZINC000217665795 CG On-Demand Unstable TERT 20 45 C[C@H]1CCCCN1CCC(=O)Nc1ccc2c(c1)CCC2 ZINC000217665795 CG On-Demand Unstable CALCRL 63 33 CN1C[C@H](C(=O)O)[C@H](c2ccccc2Cl)C1 ZINC000217665796 BE In-Stock Unstable SLC6A1 48 35 CC(=O)NC1CCN(c2ccc3ccccc3n2)CC1 ZINC000217665801 CE On-Demand Unstable HTR3A 40 52 CC(=O)NC1CCN(c2ccc3ccccc3n2)CC1 ZINC000217665801 CE On-Demand Unstable SORD 21 46 CC(=O)NC1CCN(c2ccc3ccccc3n2)CC1 ZINC000217665801 CE On-Demand Unstable SMO 48 39 COC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217665814 GE In-Stock Unstable MMP13 33 41 COC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217665814 GE In-Stock Unstable TRY2_BOVIN 43 34 COC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217665814 GE In-Stock Unstable ADAMTS4 51 34 Brc1ccccc1CN[C@@H]1CCN2CCCC[C@@H]12 ZINC000217665820 DG On-Demand Unstable VACHT_TETCF 0 44 COc1cc([C@@H]2CC(=O)Oc3c2c(=O)oc2ccccc32)cc(OC)c1O ZINC000217665848 FF In-Stock Unstable NQO1 44 38 COc1ccc([C@@H](C)N[C@@H]2CCC[C@@H](O)C2)cc1 ZINC000217665857 BF For-Sale Unstable NPBWR1 35 40 CN(Cc1ccncc1)C(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217665864 DF For-Sale Unstable HSD17B2 32 48 COC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccccc2)c(C(=O)O)c1 ZINC000217665895 GE In-Stock Unstable ADAMTS4 51 34 Brc1ccccc1CN[C@H]1CCN2CCCC[C@@H]12 ZINC000217665907 DG On-Demand Unstable VACHT_TETCF 0 44 CN(C)c1ccc(C(=O)N[C@@H]2CCCC[C@@H]2CO)cc1 ZINC000217665913 CE On-Demand Unstable SSTR3 29 44 COc1cc([C@H]2CC(=O)Oc3c2c(=O)oc2ccccc32)cc(OC)c1O ZINC000217665924 FF In-Stock Unstable NQO1 44 38 COc1ccc([C@H](C)N[C@@H]2CCC[C@@H](O)C2)cc1 ZINC000217665940 BF On-Demand Unstable NPBWR1 35 40 C=C(C)CN(CC)CCC(=O)Nc1sc2c(c1C#N)CC[C@@H](C)C2 ZINC000217665946 EH On-Demand Unstable MURF 0 40 C=C(C)CN(CC)CCC(=O)Nc1sc2c(c1C#N)CC[C@@H](C)C2 ZINC000217665946 EH On-Demand Unstable VIPR1 26 41 CN(C)c1ccc(C(=O)N[C@H]2CCCC[C@@H]2CO)cc1 ZINC000217665987 CE On-Demand Unstable SSTR3 29 44 COC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217666009 HE In-Stock Unstable BMP1 68 38 COC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217666009 HE In-Stock Unstable MMP13 63 46 COC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217666009 HE In-Stock Unstable MMP2 39 40 COC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217666009 HE In-Stock Unstable MMP3 41 40 COC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217666009 HE In-Stock Unstable MMP8 28 46 COC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217666009 HE In-Stock Unstable MMP9 45 46 COC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217666009 HE In-Stock Unstable PTGDR 21 40 COC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217666009 HE In-Stock Unstable MMP7 29 40 COC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217666009 HE In-Stock Unstable ADAMTS4 51 35 COC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217666009 HE In-Stock Unstable CA9 19 41 COC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217666009 HE In-Stock Unstable MMP1 44 38 COC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217666009 HE In-Stock Unstable AKR1C2 45 35 COc1ccc([C@@H](C)N[C@H]2CCC[C@@H](O)C2)cc1 ZINC000217666015 BF For-Sale Unstable NPBWR1 35 40 N#Cc1cccc(CN2CCC[C@@H]3CCCC[C@H]32)c1 ZINC000217666043 CH On-Demand Unstable SLC18A3 15 41 C=C(C)CN(CC)CCC(=O)Nc1sc2c(c1C#N)CC[C@H](C)C2 ZINC000217666044 EH On-Demand Unstable MURF 0 40 C=C(C)CN(CC)CCC(=O)Nc1sc2c(c1C#N)CC[C@H](C)C2 ZINC000217666044 EH On-Demand Unstable VIPR1 26 41 CN1C[C@H](C(=O)O)[C@H](c2ccc(Cl)c(Cl)c2)C1 ZINC000217666070 CF In-Stock Unstable SLC6A4 28 51 CN1C[C@H](C(=O)O)[C@H](c2ccc(Cl)c(Cl)c2)C1 ZINC000217666070 CF In-Stock Unstable SLC6A3 34 57 CN(C)c1ccc(C(=O)N[C@@H]2CCCC[C@H]2CO)cc1 ZINC000217666079 CE On-Demand Unstable SSTR3 29 44 COc1ccc2c(ccn2C[C@@H](C(=O)O)C(F)(F)F)c1 ZINC000217666090 CF For-Sale Unstable PPARG 18 40 COc1ccc2c(ccn2C[C@@H](C(=O)O)C(F)(F)F)c1 ZINC000217666090 CF For-Sale Unstable PPARA 15 43 COc1ccc2c(ccn2C[C@@H](C(=O)O)C(F)(F)F)c1 ZINC000217666090 CF For-Sale Unstable MTNR1A 42 35 COc1ccc2c(ccn2C[C@@H](C(=O)O)C(F)(F)F)c1 ZINC000217666090 CF For-Sale Unstable AKR1C3 19 44 COc1ccc([C@H](C)N[C@H]2CCC[C@@H](O)C2)cc1 ZINC000217666096 BF On-Demand Unstable NPBWR1 35 40 O=C(COCc1nc2ccccc2[nH]1)NCc1nc(-c2ccccc2)n[nH]1 ZINC000217666099 FE In-Stock Unstable CYSP_TRYCR 0 47 O=C(COCc1nc2ccccc2[nH]1)NCc1nc(-c2ccccc2)n[nH]1 ZINC000217666099 FE In-Stock Unstable PIN1 32 41 O=C(COCc1nc2ccccc2[nH]1)NCc1nc(-c2ccccc2)n[nH]1 ZINC000217666099 FE In-Stock Unstable FABK 0 44 COC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217666103 HE In-Stock Unstable BMP1 68 38 COC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217666103 HE In-Stock Unstable MMP13 63 46 COC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217666103 HE In-Stock Unstable MMP2 39 40 COC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217666103 HE In-Stock Unstable MMP3 41 40 COC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217666103 HE In-Stock Unstable MMP8 28 46 COC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217666103 HE In-Stock Unstable MMP9 45 46 COC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217666103 HE In-Stock Unstable PTGDR 21 40 COC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217666103 HE In-Stock Unstable MMP7 29 40 COC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217666103 HE In-Stock Unstable ADAMTS4 51 35 COC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217666103 HE In-Stock Unstable CA9 19 41 COC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217666103 HE In-Stock Unstable MMP1 44 38 COC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)cc2)c(C(=O)O)c1 ZINC000217666103 HE In-Stock Unstable AKR1C2 45 35 O=C(O)/C=C\c1ccc(C(=O)Nc2ccc(F)cc2Cl)s1 ZINC000217666108 EH For-Sale Anodyne PYGL 0 41 CN(C)c1ccc(C(=O)N[C@H]2CCCC[C@H]2CO)cc1 ZINC000217666154 CE On-Demand Unstable SSTR3 29 44 N#Cc1cccc(CN2CCC[C@H]3CCCC[C@H]32)c1 ZINC000217666162 CH On-Demand Unstable SLC18A3 15 41 COc1ccc2c(ccn2C[C@H](C(=O)O)C(F)(F)F)c1 ZINC000217666168 CF For-Sale Unstable PPARG 18 40 COc1ccc2c(ccn2C[C@H](C(=O)O)C(F)(F)F)c1 ZINC000217666168 CF For-Sale Unstable PPARA 15 43 COc1ccc2c(ccn2C[C@H](C(=O)O)C(F)(F)F)c1 ZINC000217666168 CF For-Sale Unstable MTNR1A 42 35 COc1ccc2c(ccn2C[C@H](C(=O)O)C(F)(F)F)c1 ZINC000217666168 CF For-Sale Unstable AKR1C3 19 44 CCOc1cccc([C@@H]2CN(C)C[C@@H]2C(=O)O)c1 ZINC000217666190 BD In-Stock Unstable SLC6A1 34 49 CCOc1cccc([C@@H]2CN(C)C[C@@H]2C(=O)O)c1 ZINC000217666190 BD In-Stock Unstable CCKAR 41 32 CCOc1cccc([C@@H]2CN(C)C[C@@H]2C(=O)O)c1 ZINC000217666190 BD In-Stock Unstable CCR5 71 37 CCOc1cccc([C@@H]2CN(C)C[C@@H]2C(=O)O)c1 ZINC000217666190 BD In-Stock Unstable PDS 59 34 COC(=O)[C@@H]1Cc2ccccc2CN1CCC(=O)Nc1cc(Cl)ccc1Cl ZINC000217666199 HH On-Demand Unstable CFTR 48 37 COC(=O)[C@@H]1Cc2ccccc2CN1CCC(=O)Nc1cc(Cl)ccc1Cl ZINC000217666199 HH On-Demand Unstable ADAM9 55 33 NCCc1ccc(Br)c(Cl)c1O ZINC000217666212 CE For-Sale Unstable TAAR1 17 41 COC[C@@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217666219 JE In-Stock Unstable ADAMTS4 41 32 O=S(=O)(CCc1ccccc1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217666237 GF In-Stock Unstable PREP 22 47 CCOc1cccc([C@H]2CN(C)C[C@@H]2C(=O)O)c1 ZINC000217666260 BD In-Stock Unstable SLC6A1 34 49 CCOc1cccc([C@H]2CN(C)C[C@@H]2C(=O)O)c1 ZINC000217666260 BD In-Stock Unstable CCKAR 41 32 CCOc1cccc([C@H]2CN(C)C[C@@H]2C(=O)O)c1 ZINC000217666260 BD In-Stock Unstable CCR5 71 37 CCOc1cccc([C@H]2CN(C)C[C@@H]2C(=O)O)c1 ZINC000217666260 BD In-Stock Unstable PDS 59 34 COC(=O)[C@H]1Cc2ccccc2CN1CCC(=O)Nc1cc(Cl)ccc1Cl ZINC000217666282 HH On-Demand Unstable CFTR 48 37 COC(=O)[C@H]1Cc2ccccc2CN1CCC(=O)Nc1cc(Cl)ccc1Cl ZINC000217666282 HH On-Demand Unstable ADAM9 55 33 COC[C@H](C)NS(=O)(=O)c1ccc(NCCc2ccc(OC)c(OC)c2)c(C(=O)O)c1 ZINC000217666297 JE In-Stock Unstable ADAMTS4 41 32 O=S(=O)(CCc1ccccc1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217666322 GF In-Stock Unstable PREP 22 47 CCOc1ccc([C@@H]2CN(C)C[C@@H]2C(=O)O)cc1 ZINC000217666372 BD In-Stock Unstable SLC6A1 101 50 CCOc1ccc([C@@H]2CN(C)C[C@@H]2C(=O)O)cc1 ZINC000217666372 BD In-Stock Unstable SLC6A4 22 50 CCOc1ccc([C@@H]2CN(C)C[C@@H]2C(=O)O)cc1 ZINC000217666372 BD In-Stock Unstable SLC6A3 33 49 C[C@@H](CN1CCCOCC1)[C@@H](O)c1ccccc1 ZINC000217666383 BE For-Sale Unstable PLK1 0 43 C[C@@H](CN1CCCOCC1)[C@@H](O)c1ccccc1 ZINC000217666383 BE For-Sale Unstable ABCB1 0 40 COC(=O)[C@@H]1Cc2ccccc2CN1CCC(=O)Nc1cccc(Cl)c1 ZINC000217666396 FG On-Demand Unstable CFTR 57 41 COC(=O)[C@@H]1Cc2ccccc2CN1CCC(=O)Nc1cccc(Cl)c1 ZINC000217666396 FG On-Demand Unstable ADAM9 56 33 c1ccc2c(c1)CCC[C@H]2N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217666419 CG For-Sale Unstable SLC18A3 55 36 c1ccc2c(c1)CCC[C@H]2N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217666419 CG For-Sale Unstable KCNN3 22 42 Cc1cc(S(=O)(=O)N2CC[C@H](n3cc(-c4ccccc4)nn3)C2)ccc1F ZINC000217666437 GG In-Stock Unstable CA5B 17 41 Cc1cc(S(=O)(=O)N2CC[C@H](n3cc(-c4ccccc4)nn3)C2)ccc1F ZINC000217666437 GG In-Stock Unstable LEF 47 34 CCOc1ccc([C@H]2CN(C)C[C@@H]2C(=O)O)cc1 ZINC000217666461 BD In-Stock Unstable SLC6A1 101 50 CCOc1ccc([C@H]2CN(C)C[C@@H]2C(=O)O)cc1 ZINC000217666461 BD In-Stock Unstable SLC6A4 22 50 CCOc1ccc([C@H]2CN(C)C[C@@H]2C(=O)O)cc1 ZINC000217666461 BD In-Stock Unstable SLC6A3 33 49 C[C@H](CN1CCCOCC1)[C@@H](O)c1ccccc1 ZINC000217666463 BE For-Sale Unstable PLK1 0 43 C[C@H](CN1CCCOCC1)[C@@H](O)c1ccccc1 ZINC000217666463 BE For-Sale Unstable ABCB1 0 40 COC(=O)[C@H]1Cc2ccccc2CN1CCC(=O)Nc1cccc(Cl)c1 ZINC000217666474 FG On-Demand Unstable CFTR 57 41 COC(=O)[C@H]1Cc2ccccc2CN1CCC(=O)Nc1cccc(Cl)c1 ZINC000217666474 FG On-Demand Unstable ADAM9 56 33 Cc1cc(S(=O)(=O)N2CC[C@@H](n3cc(-c4ccccc4)nn3)C2)ccc1F ZINC000217666509 GG In-Stock Unstable CA5B 17 41 Cc1cc(S(=O)(=O)N2CC[C@@H](n3cc(-c4ccccc4)nn3)C2)ccc1F ZINC000217666509 GG In-Stock Unstable LEF 47 34 CSC[C@@](C)(O)CNC(=O)Cc1ccc(C)c(C)c1 ZINC000217666541 CE On-Demand Unstable TRPV1 20 43 Cc1ccccc1/C=C/NC(=O)NCCCCCC(=O)O ZINC000217666549 CF For-Sale Unstable HDAC8 15 45 Cc1ccccc1/C=C/NC(=O)NCCCCCC(=O)O ZINC000217666549 CF For-Sale Unstable EPHX2 23 43 COC(=O)[C@@H]1Cc2ccccc2CN1CCC(=O)Nc1ccc(Br)cc1F ZINC000217666577 IH On-Demand Unstable ADAM9 61 35 CCCOc1ccc([C@@H]2CN(C)C[C@@H]2C(=O)O)cc1 ZINC000217666581 CE In-Stock Unstable SLC6A1 77 47 CCCOc1ccc([C@@H]2CN(C)C[C@@H]2C(=O)O)cc1 ZINC000217666581 CE In-Stock Unstable SLC6A3 24 41 CCCOc1ccc([C@@H]2CN(C)C[C@@H]2C(=O)O)cc1 ZINC000217666581 CE In-Stock Unstable PLA2G4B 61 34 COc1ccc([C@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1OC ZINC000217666586 KH In-Stock Unstable CYP1B1 63 42 COc1ccc([C@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1OC ZINC000217666586 KH In-Stock Unstable CYP1A1 47 42 COc1ccc([C@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1OC ZINC000217666586 KH In-Stock Unstable CYP1A2 41 42 COc1ccc([C@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1OC ZINC000217666586 KH In-Stock Unstable RORC 53 37 CCOC(=O)[C@@H](NCCNC(C)=O)c1ccccc1 ZINC000217666599 CD For-Sale Unstable MTNR1A 59 43 CCOC(=O)[C@@H](NCCNC(C)=O)c1ccccc1 ZINC000217666599 CD For-Sale Unstable MTNR1B 58 44 CSC[C@](C)(O)CNC(=O)Cc1ccc(C)c(C)c1 ZINC000217666627 CE On-Demand Unstable TRPV1 20 43 CCCOc1ccc([C@H]2CN(C)C[C@@H]2C(=O)O)cc1 ZINC000217666657 CE In-Stock Unstable SLC6A1 77 47 CCCOc1ccc([C@H]2CN(C)C[C@@H]2C(=O)O)cc1 ZINC000217666657 CE In-Stock Unstable SLC6A3 24 41 CCCOc1ccc([C@H]2CN(C)C[C@@H]2C(=O)O)cc1 ZINC000217666657 CE In-Stock Unstable PLA2G4B 61 34 Cc1cc(=O)cc(C(=O)N2CCC(C(=O)N3CCCCC3)CC2)o1 ZINC000217666659 ED In-Stock Unstable L3MBTL1 0 41 Cc1cc(=O)cc(C(=O)N2CCC(C(=O)N3CCCCC3)CC2)o1 ZINC000217666659 ED In-Stock Unstable L3MBTL3 49 41 COC(=O)[C@H]1Cc2ccccc2CN1CCC(=O)Nc1ccc(Br)cc1F ZINC000217666662 IH On-Demand Unstable ADAM9 61 35 COC(=O)[C@@H](O)CNC(=O)c1ccc([N+](=O)[O-])cc1C ZINC000217666664 CC On-Demand Unstable CACNA1C 55 37 COc1ccc([C@@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1OC ZINC000217666673 KH In-Stock Unstable CYP1B1 63 42 COc1ccc([C@@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1OC ZINC000217666673 KH In-Stock Unstable CYP1A1 47 42 COc1ccc([C@@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1OC ZINC000217666673 KH In-Stock Unstable CYP1A2 41 42 COc1ccc([C@@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1OC ZINC000217666673 KH In-Stock Unstable RORC 53 37 CCOC(=O)[C@H](NCCNC(C)=O)c1ccccc1 ZINC000217666685 CD For-Sale Unstable MTNR1A 59 43 CCOC(=O)[C@H](NCCNC(C)=O)c1ccccc1 ZINC000217666685 CD For-Sale Unstable MTNR1B 58 44 NC(=O)c1n[nH]c2cc(Cl)ccc12 ZINC000217666720 AD For-Sale Unstable GRIN1 23 48 NC(=O)c1n[nH]c2cc(Cl)ccc12 ZINC000217666720 AD For-Sale Unstable SGK1 54 39 NC(=O)c1n[nH]c2cc(Cl)ccc12 ZINC000217666720 AD For-Sale Unstable ALPL 44 37 NC(=O)[C@H]1CCCN1C(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217666731 CC For-Sale Unstable PREP 54 50 COC(=O)[C@H](O)CNC(=O)c1ccc([N+](=O)[O-])cc1C ZINC000217666742 CC On-Demand Unstable CACNA1C 55 37 CN1C[C@H](C(=O)O)[C@H](c2ccc3c(c2)OCO3)C1 ZINC000217666761 BD In-Stock Unstable SLC6A1 0 45 CN1C[C@H](C(=O)O)[C@H](c2ccc3c(c2)OCO3)C1 ZINC000217666761 BD In-Stock Unstable EDNRB 66 41 CN1C[C@H](C(=O)O)[C@H](c2ccc3c(c2)OCO3)C1 ZINC000217666761 BD In-Stock Unstable EDNRA 77 45 CN1C[C@H](C(=O)O)[C@H](c2ccc3c(c2)OCO3)C1 ZINC000217666761 BD In-Stock Unstable TERT 0 42 CCN[C@@H]1CC[C@@H](CC)C[C@@H]1CCCc1ccccc1 ZINC000217666763 CJ For-Sale Unstable SLC18A2 32 41 COC(=O)[C@@H]1Cc2ccccc2CN1CCC(=O)NCc1ccccc1Cl ZINC000217666769 GF On-Demand Unstable HTR7 17 41 COC(=O)[C@@H]1Cc2ccccc2CN1CCC(=O)NCc1ccccc1Cl ZINC000217666769 GF On-Demand Unstable P2RX7 79 43 COC(=O)[C@@H]1Cc2ccccc2CN1CCC(=O)NCc1ccccc1Cl ZINC000217666769 GF On-Demand Unstable ADAM9 60 33 COc1ccc(CCC(=O)Nc2ccc3nc[nH]c(=O)c3c2)cc1 ZINC000217666784 DF In-Stock Unstable MTNR1A 21 41 COc1ccc(CCC(=O)Nc2ccc3nc[nH]c(=O)c3c2)cc1 ZINC000217666784 DF In-Stock Unstable MTNR1B 18 41 COc1ccc(CCC(=O)Nc2ccc3nc[nH]c(=O)c3c2)cc1 ZINC000217666784 DF In-Stock Unstable MCHR1 24 40 COc1ccc(CCC(=O)Nc2ccc3nc[nH]c(=O)c3c2)cc1 ZINC000217666784 DF In-Stock Unstable ENPP1 57 33 COc1ccc(CCC(=O)Nc2ccc3nc[nH]c(=O)c3c2)cc1 ZINC000217666784 DF In-Stock Unstable QTRT1 0 48 NC(=O)[C@@H]1CCCN1C(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217666809 CC For-Sale Unstable PREP 54 50 CCN[C@H]1CC[C@@H](CC)C[C@@H]1CCCc1ccccc1 ZINC000217666838 CJ For-Sale Unstable SLC18A2 32 41 CN1C[C@@H](C(=O)O)[C@H](c2ccc3c(c2)OCO3)C1 ZINC000217666856 BD In-Stock Unstable SLC6A1 0 45 CN1C[C@@H](C(=O)O)[C@H](c2ccc3c(c2)OCO3)C1 ZINC000217666856 BD In-Stock Unstable EDNRB 66 41 CN1C[C@@H](C(=O)O)[C@H](c2ccc3c(c2)OCO3)C1 ZINC000217666856 BD In-Stock Unstable EDNRA 77 45 CN1C[C@@H](C(=O)O)[C@H](c2ccc3c(c2)OCO3)C1 ZINC000217666856 BD In-Stock Unstable TERT 0 42 COC(=O)[C@H]1Cc2ccccc2CN1CCC(=O)NCc1ccccc1Cl ZINC000217666867 GF On-Demand Unstable HTR7 17 41 COC(=O)[C@H]1Cc2ccccc2CN1CCC(=O)NCc1ccccc1Cl ZINC000217666867 GF On-Demand Unstable P2RX7 79 43 COC(=O)[C@H]1Cc2ccccc2CN1CCC(=O)NCc1ccccc1Cl ZINC000217666867 GF On-Demand Unstable ADAM9 60 33 NC(=O)[C@H]1CCCN1C(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217666887 CC For-Sale Unstable PREP 62 51 COC(=O)C[C@H](c1c(O)c2ccccc2oc1=O)c1cc2ccc(OC)cc2n(C)c1=O ZINC000217666904 IG In-Stock Unstable NQO1 36 50 CCN[C@@H]1CC[C@H](CC)C[C@@H]1CCCc1ccccc1 ZINC000217666927 CJ For-Sale Unstable SLC18A2 32 41 Cc1ccccc1/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O ZINC000217666934 CF For-Sale Unstable ACE 19 43 Cc1ccccc1/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O ZINC000217666934 CF For-Sale Unstable FOLH1 59 41 Cc1ccccc1/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O ZINC000217666934 CF For-Sale Unstable MME 45 46 Cc1ccccc1/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O ZINC000217666934 CF For-Sale Unstable ANPEP 41 48 Cc1ccccc1/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O ZINC000217666934 CF For-Sale Unstable RNPEP 23 45 Cc1ccccc1/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O ZINC000217666934 CF For-Sale Unstable CTSK 20 40 Cc1ccccc1/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O ZINC000217666934 CF For-Sale Unstable NAALAD2 29 40 Cc1ccccc1/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O ZINC000217666934 CF For-Sale Unstable CAPNS1 56 34 Cc1ccccc1/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O ZINC000217666934 CF For-Sale Unstable CAPN1 57 43 Cc1ccccc1/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O ZINC000217666934 CF For-Sale Unstable CAPN2 54 34 Cc1ccccc1/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O ZINC000217666934 CF For-Sale Unstable LAP3 16 45 Cc1ccccc1/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O ZINC000217666934 CF For-Sale Unstable FPR1 84 44 Cc1ccccc1/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O ZINC000217666934 CF For-Sale Unstable NPR 66 36 Cc1ccccc1/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O ZINC000217666934 CF For-Sale Unstable AMP1_PLAFQ 22 45 CN1C[C@H](C(=O)O)[C@H](c2ccc(OCc3ccccc3)cc2)C1 ZINC000217666961 DF In-Stock Unstable MAOB 23 42 CN1C[C@H](C(=O)O)[C@H](c2ccc(OCc3ccccc3)cc2)C1 ZINC000217666961 DF In-Stock Unstable SLC6A1 91 51 CN1C[C@H](C(=O)O)[C@H](c2ccc(OCc3ccccc3)cc2)C1 ZINC000217666961 DF In-Stock Unstable SLC6A4 22 51 CN1C[C@H](C(=O)O)[C@H](c2ccc(OCc3ccccc3)cc2)C1 ZINC000217666961 DF In-Stock Unstable SLC6A3 36 44 CN1C[C@H](C(=O)O)[C@H](c2ccc(OCc3ccccc3)cc2)C1 ZINC000217666961 DF In-Stock Unstable LTA4H 38 44 CN1C[C@H](C(=O)O)[C@H](c2ccc(OCc3ccccc3)cc2)C1 ZINC000217666961 DF In-Stock Unstable ADAM17 27 40 CN1C[C@H](C(=O)O)[C@H](c2ccc(OCc3ccccc3)cc2)C1 ZINC000217666961 DF In-Stock Unstable GYS1 48 37 CN1C[C@H](C(=O)O)[C@H](c2ccc(OCc3ccccc3)cc2)C1 ZINC000217666961 DF In-Stock Unstable FFAR1 47 47 CN1C[C@H](C(=O)O)[C@H](c2ccc(OCc3ccccc3)cc2)C1 ZINC000217666961 DF In-Stock Unstable FFAR4 40 38 COC(=O)[C@@H]1Cc2ccccc2CN1CCC(=O)N[C@@H]1CCCc2ccccc21 ZINC000217666970 GG On-Demand Unstable HTR7 23 54 COC(=O)[C@@H]1Cc2ccccc2CN1CCC(=O)N[C@@H]1CCCc2ccccc21 ZINC000217666970 GG On-Demand Unstable ADAM9 54 32 COC(=O)[C@@H]1Cc2ccccc2CN1CCC(=O)N[C@@H]1CCCc2ccccc21 ZINC000217666970 GG On-Demand Unstable BIRC3 27 41 NC(=O)[C@@H]1CCCN1C(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217666978 CC For-Sale Unstable PREP 62 51 COC[C@@H](C)NS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217666989 ED In-Stock Unstable SLC6A9 18 40 COC(=O)C[C@@H](c1c(O)c2ccccc2oc1=O)c1cc2ccc(OC)cc2n(C)c1=O ZINC000217666991 IG In-Stock Unstable NQO1 36 50 CCN[C@H]1CC[C@H](CC)C[C@@H]1CCCc1ccccc1 ZINC000217666998 CJ For-Sale Unstable SLC18A2 32 41 Cc1ccccc1/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O ZINC000217667020 CF For-Sale Unstable ACE 19 43 Cc1ccccc1/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O ZINC000217667020 CF For-Sale Unstable FOLH1 59 41 Cc1ccccc1/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O ZINC000217667020 CF For-Sale Unstable MME 45 46 Cc1ccccc1/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O ZINC000217667020 CF For-Sale Unstable ANPEP 41 48 Cc1ccccc1/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O ZINC000217667020 CF For-Sale Unstable RNPEP 23 45 Cc1ccccc1/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O ZINC000217667020 CF For-Sale Unstable CTSK 20 40 Cc1ccccc1/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O ZINC000217667020 CF For-Sale Unstable NAALAD2 29 40 Cc1ccccc1/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O ZINC000217667020 CF For-Sale Unstable CAPNS1 56 34 Cc1ccccc1/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O ZINC000217667020 CF For-Sale Unstable CAPN1 57 43 Cc1ccccc1/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O ZINC000217667020 CF For-Sale Unstable CAPN2 54 34 Cc1ccccc1/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O ZINC000217667020 CF For-Sale Unstable LAP3 16 45 Cc1ccccc1/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O ZINC000217667020 CF For-Sale Unstable FPR1 84 44 Cc1ccccc1/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O ZINC000217667020 CF For-Sale Unstable NPR 66 36 Cc1ccccc1/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O ZINC000217667020 CF For-Sale Unstable AMP1_PLAFQ 22 45 COc1ccccc1NC(=S)Nc1ccc(N)cc1 ZINC000217667024 CG For-Sale Unstable PDGFRA 29 42 COc1ccccc1NC(=S)Nc1ccc(N)cc1 ZINC000217667024 CG For-Sale Unstable UREA_CANEN 16 40 Oc1cccc(N2CCN(C[C@@H]3[C@H]4CNC[C@H]43)CC2)c1 ZINC000217667025 CC In-Stock Unstable HTR7 21 43 CN1C[C@@H](C(=O)O)[C@H](c2ccc(OCc3ccccc3)cc2)C1 ZINC000217667050 DF In-Stock Unstable MAOB 23 42 CN1C[C@@H](C(=O)O)[C@H](c2ccc(OCc3ccccc3)cc2)C1 ZINC000217667050 DF In-Stock Unstable SLC6A1 91 51 CN1C[C@@H](C(=O)O)[C@H](c2ccc(OCc3ccccc3)cc2)C1 ZINC000217667050 DF In-Stock Unstable SLC6A4 22 51 CN1C[C@@H](C(=O)O)[C@H](c2ccc(OCc3ccccc3)cc2)C1 ZINC000217667050 DF In-Stock Unstable SLC6A3 36 44 CN1C[C@@H](C(=O)O)[C@H](c2ccc(OCc3ccccc3)cc2)C1 ZINC000217667050 DF In-Stock Unstable LTA4H 38 44 CN1C[C@@H](C(=O)O)[C@H](c2ccc(OCc3ccccc3)cc2)C1 ZINC000217667050 DF In-Stock Unstable ADAM17 27 40 CN1C[C@@H](C(=O)O)[C@H](c2ccc(OCc3ccccc3)cc2)C1 ZINC000217667050 DF In-Stock Unstable GYS1 48 37 CN1C[C@@H](C(=O)O)[C@H](c2ccc(OCc3ccccc3)cc2)C1 ZINC000217667050 DF In-Stock Unstable FFAR1 47 47 CN1C[C@@H](C(=O)O)[C@H](c2ccc(OCc3ccccc3)cc2)C1 ZINC000217667050 DF In-Stock Unstable FFAR4 40 38 NC(=O)C1CCN(C(=O)c2ccc(/C=C\C(=O)O)s2)CC1 ZINC000217667056 DD For-Sale Unstable L3MBTL1 0 47 NC(=O)C1CCN(C(=O)c2ccc(/C=C\C(=O)O)s2)CC1 ZINC000217667056 DD For-Sale Unstable L3MBTL3 40 31 COC(=O)[C@H]1Cc2ccccc2CN1CCC(=O)N[C@@H]1CCCc2ccccc21 ZINC000217667059 GG On-Demand Unstable HTR7 23 54 COC(=O)[C@H]1Cc2ccccc2CN1CCC(=O)N[C@@H]1CCCc2ccccc21 ZINC000217667059 GG On-Demand Unstable ADAM9 54 32 COC(=O)[C@H]1Cc2ccccc2CN1CCC(=O)N[C@@H]1CCCc2ccccc21 ZINC000217667059 GG On-Demand Unstable BIRC3 27 41 COC[C@H](C)NS(=O)(=O)c1ccc(N2CCCC2)c(C(=O)O)c1 ZINC000217667066 ED In-Stock Unstable SLC6A9 18 40 CSCC[C@@H](NC(=O)N/C=C/c1ccccc1C)C(=O)O ZINC000217667132 DE For-Sale Unstable FOLH1 24 43 CSCC[C@@H](NC(=O)N/C=C/c1ccccc1C)C(=O)O ZINC000217667132 DE For-Sale Unstable NAALAD2 49 37 CSCC[C@@H](NC(=O)N/C=C/c1ccccc1C)C(=O)O ZINC000217667132 DE For-Sale Unstable PAM 0 43 CSCC[C@@H](NC(=O)N/C=C/c1ccccc1C)C(=O)O ZINC000217667132 DE For-Sale Unstable FPR1 43 42 CSCC[C@@H](NC(=O)N/C=C/c1ccccc1C)C(=O)O ZINC000217667132 DE For-Sale Unstable SLC15A2 0 42 CSCC[C@@H](NC(=O)N/C=C/c1ccccc1C)C(=O)O ZINC000217667132 DE For-Sale Unstable FPRL2 0 42 COc1cccc([C@@H]2CN(C)C[C@@H]2C(=O)O)c1OC ZINC000217667162 CD In-Stock Unstable ADRA1B 42 33 CCCN(CC)CCN[C@@H]1CCCc2ccc(O)cc21 ZINC000217667178 CG On-Demand Unstable HTR1A 0 43 CCCN(CC)CCN[C@@H]1CCCc2ccc(O)cc21 ZINC000217667178 CG On-Demand Unstable DRD2 0 43 COC[C@@H](C)NS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217667183 FD In-Stock Unstable SLC6A9 18 41 CSCC[C@H](NC(=O)N/C=C/c1ccccc1C)C(=O)O ZINC000217667224 DE For-Sale Unstable FOLH1 24 43 CSCC[C@H](NC(=O)N/C=C/c1ccccc1C)C(=O)O ZINC000217667224 DE For-Sale Unstable NAALAD2 49 37 CSCC[C@H](NC(=O)N/C=C/c1ccccc1C)C(=O)O ZINC000217667224 DE For-Sale Unstable PAM 0 43 CSCC[C@H](NC(=O)N/C=C/c1ccccc1C)C(=O)O ZINC000217667224 DE For-Sale Unstable FPR1 43 42 CSCC[C@H](NC(=O)N/C=C/c1ccccc1C)C(=O)O ZINC000217667224 DE For-Sale Unstable SLC15A2 0 42 CSCC[C@H](NC(=O)N/C=C/c1ccccc1C)C(=O)O ZINC000217667224 DE For-Sale Unstable FPRL2 0 42 COc1cccc([C@H]2CN(C)C[C@@H]2C(=O)O)c1OC ZINC000217667231 CD In-Stock Unstable ADRA1B 42 33 CCCN(CC)CCN[C@H]1CCCc2ccc(O)cc21 ZINC000217667265 CG On-Demand Unstable HTR1A 0 43 CCCN(CC)CCN[C@H]1CCCc2ccc(O)cc21 ZINC000217667265 CG On-Demand Unstable DRD2 0 43 COC[C@H](C)NS(=O)(=O)c1ccc(N2CCCCC2)c(C(=O)O)c1 ZINC000217667266 FD In-Stock Unstable SLC6A9 18 41 COc1ccc([C@@H](C)NC(=O)N/C=C/c2ccccc2C)cc1OC ZINC000217667342 EI For-Sale Unstable KCNQ2 47 37 COc1ccc([C@@H]2CN(C)C[C@@H]2C(=O)O)cc1OC ZINC000217667362 CD In-Stock Unstable SLC6A3 22 40 COc1ccc([C@@H]2CN(C)C[C@@H]2C(=O)O)cc1OC ZINC000217667362 CD In-Stock Unstable PDE4B 15 53 COC(=O)[C@@H]1Cc2ccccc2CN1CCC(=O)Nc1c(C)nn(-c2ccccc2)c1C ZINC000217667369 IG On-Demand Unstable ADAM9 54 33 COC[C@@H](C)NS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1 ZINC000217667373 FC In-Stock Unstable SLC6A9 21 44 COC[C@@H](C)NS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1 ZINC000217667373 FC In-Stock Unstable MMP12 41 43 O=S(=O)(Cc1cccc(Cl)c1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217667402 HG In-Stock Unstable PTPN2 19 40 O=S(=O)(Cc1cccc(Cl)c1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217667402 HG In-Stock Unstable PTPN1 17 40 COc1ccc([C@H](C)NC(=O)N/C=C/c2ccccc2C)cc1OC ZINC000217667416 EI For-Sale Unstable KCNQ2 47 37 COC(=O)[C@H]1Cc2ccccc2CN1CCC(=O)Nc1c(C)nn(-c2ccccc2)c1C ZINC000217667427 IG On-Demand Unstable ADAM9 54 33 COc1ccc([C@H]2CN(C)C[C@@H]2C(=O)O)cc1OC ZINC000217667464 CD In-Stock Unstable SLC6A3 22 40 COc1ccc([C@H]2CN(C)C[C@@H]2C(=O)O)cc1OC ZINC000217667464 CD In-Stock Unstable PDE4B 15 53 O=S(=O)(Cc1cccc(Cl)c1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217667482 HG In-Stock Unstable PTPN2 19 40 O=S(=O)(Cc1cccc(Cl)c1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217667482 HG In-Stock Unstable PTPN1 17 40 COC[C@H](C)NS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1 ZINC000217667490 FC In-Stock Unstable SLC6A9 21 44 COC[C@H](C)NS(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)O)c1 ZINC000217667490 FC In-Stock Unstable MMP12 41 43 COc1ccc([C@@H](C)NC(=O)N/C=C/c2ccccc2C)cc1 ZINC000217667549 DI For-Sale Unstable ACACA 22 42 COc1ccc([C@@H](C)NC(=O)N/C=C/c2ccccc2C)cc1 ZINC000217667549 DI For-Sale Unstable ACACB 23 42 O=S(=O)(c1cccc2ccccc12)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217667577 HH In-Stock Unstable HTR6 25 42 CCCCCCCN[C@@H]1CCN2CCCC[C@@H]12 ZINC000217667608 BG For-Sale Unstable GLB1 33 42 COC(=O)[C@@H](O)CNC(=O)c1cc(Cl)c(I)cc1OC ZINC000217667614 HD On-Demand Unstable HTR4 65 47 Cn1ncc2c(=O)n(C[C@@H](C(=O)O)C(F)(F)F)cnc21 ZINC000217667629 CC For-Sale Unstable Q9M629_MAIZE 48 35 COc1ccc([C@H](C)NC(=O)N/C=C/c2ccccc2C)cc1 ZINC000217667640 DI For-Sale Unstable ACACA 22 42 COc1ccc([C@H](C)NC(=O)N/C=C/c2ccccc2C)cc1 ZINC000217667640 DI For-Sale Unstable ACACB 23 42 O=S(=O)(c1cccc2ccccc12)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217667657 HH In-Stock Unstable HTR6 25 42 CCCCCCCN[C@H]1CCN2CCCC[C@@H]12 ZINC000217667691 BG For-Sale Unstable GLB1 33 42 Cn1ncc2c(=O)n(C[C@H](C(=O)O)C(F)(F)F)cnc21 ZINC000217667705 CC For-Sale Unstable Q9M629_MAIZE 48 35 O=S(=O)(c1ccc2c(c1)CCCC2)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217667769 HG In-Stock Unstable AKR1C3 25 40 COC(=O)[C@@H]1CN(C)C[C@@H]1c1cccnc1 ZINC000217667789 BC In-Stock Unstable SLC6A1 97 48 COC(=O)[C@@H]1CN(C)C[C@@H]1c1cccnc1 ZINC000217667789 BC In-Stock Unstable CHRNA2 38 40 COC(=O)[C@@H]1CN(C)C[C@@H]1c1cccnc1 ZINC000217667789 BC In-Stock Unstable CRTY 0 40 COC(=O)[C@@H](O)CNC(=O)CCCOc1cccc(C)c1 ZINC000217667839 CC On-Demand Unstable MTNR1A 33 41 COC(=O)[C@@H](O)CNC(=O)CCCOc1cccc(C)c1 ZINC000217667839 CC On-Demand Unstable MTNR1B 26 41 O=S(=O)(c1ccc2c(c1)CCCC2)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217667847 HG In-Stock Unstable AKR1C3 25 40 COC(=O)[C@H]1CN(C)C[C@@H]1c1cccnc1 ZINC000217667888 BC In-Stock Unstable SLC6A1 97 48 COC(=O)[C@H]1CN(C)C[C@@H]1c1cccnc1 ZINC000217667888 BC In-Stock Unstable CHRNA2 38 40 COC(=O)[C@H]1CN(C)C[C@@H]1c1cccnc1 ZINC000217667888 BC In-Stock Unstable CRTY 0 40 O=C1C[C@@H](c2ccc(C(=O)O)cc2)c2c(ccc3c(=O)c(-c4ccc(O)cc4)coc23)O1 ZINC000217667920 II In-Stock Unstable ALDH2 94 38 COC(=O)[C@H](O)CNC(=O)CCCOc1cccc(C)c1 ZINC000217667923 CC On-Demand Unstable MTNR1A 33 41 COC(=O)[C@H](O)CNC(=O)CCCOc1cccc(C)c1 ZINC000217667923 CC On-Demand Unstable MTNR1B 26 41 CCOc1ccc(S(=O)(=O)N2CC[C@H](n3cc(-c4ccccc4)nn3)C2)cc1F ZINC000217667962 HG In-Stock Unstable PDE5A 25 40 CCCCCNC(=O)c1cc(/C=C\C(=O)O)ccc1F ZINC000217667979 CF For-Sale Unstable PYGL 0 40 CCCCCNC(=O)c1cc(/C=C\C(=O)O)ccc1F ZINC000217667979 CF For-Sale Unstable AKR1C3 35 40 CCCCCNC(=O)c1cc(/C=C\C(=O)O)ccc1F ZINC000217667979 CF For-Sale Unstable ASAH1 69 34 O=C1C[C@H](c2ccc(C(=O)O)cc2)c2c(ccc3c(=O)c(-c4ccc(O)cc4)coc23)O1 ZINC000217667992 II In-Stock Unstable ALDH2 94 38 COC(=O)[C@@H]1CN(C)C[C@@H]1c1ccccc1F ZINC000217668004 BD In-Stock Unstable SLC6A1 68 54 COC(=O)[C@@H]1CN(C)C[C@@H]1c1ccccc1F ZINC000217668004 BD In-Stock Unstable SLC6A4 17 49 COC(=O)[C@@H]1CN(C)C[C@@H]1c1ccccc1F ZINC000217668004 BD In-Stock Unstable SLC6A3 28 49 CCOc1ccc(S(=O)(=O)N2CC[C@@H](n3cc(-c4ccccc4)nn3)C2)cc1F ZINC000217668043 HG In-Stock Unstable PDE5A 25 40 CCN(CCC(=O)NCc1ccccc1Cl)CC(=O)Nc1c(F)cccc1F ZINC000217668045 HH On-Demand Unstable P2RX7 48 40 CCCCCNC(=O)c1ccc(/C=C\C(=O)O)cc1F ZINC000217668071 CF For-Sale Unstable PYGL 0 40 CCCCCNC(=O)c1ccc(/C=C\C(=O)O)cc1F ZINC000217668071 CF For-Sale Unstable ASAH1 69 34 COC(=O)[C@H]1CN(C)C[C@@H]1c1ccccc1F ZINC000217668093 BD In-Stock Unstable SLC6A1 68 54 COC(=O)[C@H]1CN(C)C[C@@H]1c1ccccc1F ZINC000217668093 BD In-Stock Unstable SLC6A4 17 49 COC(=O)[C@H]1CN(C)C[C@@H]1c1ccccc1F ZINC000217668093 BD In-Stock Unstable SLC6A3 28 49 CC(C)[C@@H](CO)NC(=O)Cc1ccc2c(c1)CCC(C)(C)O2 ZINC000217668105 DE In-Stock Unstable DAGLA 22 40 CCN(CCC(=O)N[C@@H]1CCCc2ccccc21)CC(=O)Nc1c(F)cccc1F ZINC000217668170 HH On-Demand Unstable BDKRB1 29 40 COC(=O)[C@@H]1CN(C)C[C@@H]1c1cccc(F)c1 ZINC000217668204 BD In-Stock Unstable SLC6A2 15 47 COC(=O)[C@@H]1CN(C)C[C@@H]1c1cccc(F)c1 ZINC000217668204 BD In-Stock Unstable SLC6A1 125 57 COC(=O)[C@@H]1CN(C)C[C@@H]1c1cccc(F)c1 ZINC000217668204 BD In-Stock Unstable SLC6A4 31 47 COC(=O)[C@@H]1CN(C)C[C@@H]1c1cccc(F)c1 ZINC000217668204 BD In-Stock Unstable SLC6A3 49 59 COC(=O)[C@@H]1CN(C)C[C@@H]1c1cccc(F)c1 ZINC000217668204 BD In-Stock Unstable CCR5 96 36 C[C@@H](N[C@@H]1CCC[C@@H](O)C1)c1cccc(C(F)(F)F)c1 ZINC000217668251 CH For-Sale Unstable CCR2 25 40 CCS(=O)(=O)Nc1ccc(C(=O)N2CCCC[C@@H]2c2ccccn2)cc1 ZINC000217668261 FG In-Stock Unstable COLA 104 41 CCS(=O)(=O)Nc1ccc(C(=O)N2CCCC[C@@H]2c2ccccn2)cc1 ZINC000217668261 FG In-Stock Unstable CPT1A 95 41 CCN(CCC(=O)N[C@H]1CCCc2ccccc21)CC(=O)Nc1c(F)cccc1F ZINC000217668262 HH On-Demand Unstable BDKRB1 29 40 COC(=O)[C@H]1CN(C)C[C@@H]1c1cccc(F)c1 ZINC000217668289 BD In-Stock Unstable SLC6A2 15 47 COC(=O)[C@H]1CN(C)C[C@@H]1c1cccc(F)c1 ZINC000217668289 BD In-Stock Unstable SLC6A1 125 57 COC(=O)[C@H]1CN(C)C[C@@H]1c1cccc(F)c1 ZINC000217668289 BD In-Stock Unstable SLC6A4 31 47 COC(=O)[C@H]1CN(C)C[C@@H]1c1cccc(F)c1 ZINC000217668289 BD In-Stock Unstable SLC6A3 49 59 COC(=O)[C@H]1CN(C)C[C@@H]1c1cccc(F)c1 ZINC000217668289 BD In-Stock Unstable CCR5 96 36 CCCCN(CC)C(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217668319 CG For-Sale Unstable OPRD1 19 41 C[C@H](N[C@@H]1CCC[C@@H](O)C1)c1cccc(C(F)(F)F)c1 ZINC000217668342 CH On-Demand Unstable CCR2 25 40 CCS(=O)(=O)Nc1ccc(C(=O)N2CCCC[C@H]2c2ccccn2)cc1 ZINC000217668344 FG In-Stock Unstable COLA 104 41 CCS(=O)(=O)Nc1ccc(C(=O)N2CCCC[C@H]2c2ccccn2)cc1 ZINC000217668344 FG In-Stock Unstable CPT1A 95 41 O=C(O)/C=C\c1cccc(C(=O)Nc2ccc(Cl)cc2)c1 ZINC000217668396 DH For-Sale Anodyne MAOB 18 49 O=C(O)/C=C\c1cccc(C(=O)Nc2ccc(Cl)cc2)c1 ZINC000217668396 DH For-Sale Anodyne ABAT 25 40 O=C(O)/C=C\c1cccc(C(=O)Nc2ccc(Cl)cc2)c1 ZINC000217668396 DH For-Sale Anodyne CPT1A 54 37 O=C(O)/C=C\c1cccc(C(=O)Nc2ccc(Cl)cc2)c1 ZINC000217668396 DH For-Sale Anodyne PRNP 19 51 O=C(O)/C=C\c1cccc(C(=O)Nc2ccc(Cl)cc2)c1 ZINC000217668396 DH For-Sale Anodyne TAAR1 17 44 O=C(O)/C=C\c1cccc(C(=O)Nc2ccc(Cl)cc2)c1 ZINC000217668396 DH For-Sale Anodyne AKR1C3 36 47 O=C(O)/C=C\c1cccc(C(=O)Nc2ccc(Cl)cc2)c1 ZINC000217668396 DH For-Sale Anodyne SMO 15 45 O=C(O)/C=C\c1cccc(C(=O)Nc2ccc(Cl)cc2)c1 ZINC000217668396 DH For-Sale Anodyne IMDH_CRYPV 16 41 O=C(O)/C=C\c1cccc(C(=O)Nc2ccc(Cl)cc2)c1 ZINC000217668396 DH For-Sale Anodyne Q25615_ONCVO 35 42 O=C(O)/C=C\c1cccc(C(=O)Nc2ccc(Cl)cc2)c1 ZINC000217668396 DH For-Sale Anodyne KCNK3 106 51 O=C(O)/C=C\c1cccc(C(=O)Nc2ccc(Cl)cc2)c1 ZINC000217668396 DH For-Sale Anodyne KCNK9 53 46 COC(=O)[C@@H]1CN(C)C[C@@H]1c1ccc(F)cc1 ZINC000217668404 BD In-Stock Unstable SLC6A2 15 58 COC(=O)[C@@H]1CN(C)C[C@@H]1c1ccc(F)cc1 ZINC000217668404 BD In-Stock Unstable SLC6A1 180 68 COC(=O)[C@@H]1CN(C)C[C@@H]1c1ccc(F)cc1 ZINC000217668404 BD In-Stock Unstable SLC6A4 37 68 COC(=O)[C@@H]1CN(C)C[C@@H]1c1ccc(F)cc1 ZINC000217668404 BD In-Stock Unstable SLC6A3 68 58 C[C@@H](N[C@H]1CCC[C@@H](O)C1)c1cccc(C(F)(F)F)c1 ZINC000217668438 CH For-Sale Unstable CCR2 25 40 COC(=O)[C@H]1CN(C)C[C@@H]1c1ccc(F)cc1 ZINC000217668489 BD In-Stock Unstable SLC6A2 15 58 COC(=O)[C@H]1CN(C)C[C@@H]1c1ccc(F)cc1 ZINC000217668489 BD In-Stock Unstable SLC6A1 180 68 COC(=O)[C@H]1CN(C)C[C@@H]1c1ccc(F)cc1 ZINC000217668489 BD In-Stock Unstable SLC6A4 37 68 COC(=O)[C@H]1CN(C)C[C@@H]1c1ccc(F)cc1 ZINC000217668489 BD In-Stock Unstable SLC6A3 68 58 C[C@H](N[C@H]1CCC[C@@H](O)C1)c1cccc(C(F)(F)F)c1 ZINC000217668520 CH On-Demand Unstable CCR2 25 40 CCc1cccc(CC)c1NC(=O)N/C=C/c1ccccc1C ZINC000217668611 DJ For-Sale Unstable ACAT 0 42 COC(=O)[C@@H]1CN(C)C[C@@H]1c1cccc(Br)c1 ZINC000217668618 CE In-Stock Unstable SLC6A1 101 52 COC[C@H](C)NS(=O)(=O)c1ccc(N[C@H](C)COC)c(C(=O)O)c1 ZINC000217668694 FD In-Stock Unstable MMP12 45 34 COC(=O)[C@H]1CN(C)C[C@@H]1c1cccc(Br)c1 ZINC000217668695 CE In-Stock Unstable SLC6A1 101 52 Cc1ccccc1/C=C/NC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217668712 EK For-Sale Unstable EPHX1 0 46 Cc1ccccc1/C=C/NC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217668712 EK For-Sale Unstable CA1 46 47 Cc1ccccc1/C=C/NC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217668712 EK For-Sale Unstable RAF1 27 43 Cc1ccccc1/C=C/NC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217668712 EK For-Sale Unstable NPY5R 22 40 Cc1ccccc1/C=C/NC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217668712 EK For-Sale Unstable CA12 19 47 Cc1ccccc1/C=C/NC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217668712 EK For-Sale Unstable CA9 19 47 Cc1ccccc1/C=C/NC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217668712 EK For-Sale Unstable Q8MMZ8_EIMTE 43 43 Cc1ccccc1/C=C/NC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217668712 EK For-Sale Unstable F13A1 15 40 O=S(=O)(c1ccc(OC(F)(F)F)cc1)N1CC[C@@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217668746 IG In-Stock Unstable EPHX2 18 50 COC[C@H](C)Nc1ccc(S(=O)(=O)N[C@@H](C)COC)cc1C(=O)O ZINC000217668783 FD In-Stock Unstable MMP12 45 34 COC(=O)[C@@H]1CN(C)C[C@@H]1c1cccc(N)c1 ZINC000217668813 BD In-Stock Unstable SLC6A1 99 52 COC(=O)[C@@H]1CN(C)C[C@@H]1c1cccc(N)c1 ZINC000217668813 BD In-Stock Unstable SLC6A3 39 41 CCN1CCC[C@@H]1CNC(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217668816 DE For-Sale Unstable DRD2 38 49 CCN1CCC[C@@H]1CNC(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217668816 DE For-Sale Unstable PFG6PD 0 45 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](CC(C)C)C(=O)N3CCc4[nH]c5ccccc5c4C3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217668835 KK In-Stock Unstable TUBA1A 16 57 O=S(=O)(c1ccc(OC(F)(F)F)cc1)N1CC[C@H](n2cc(-c3ccccc3)nn2)C1 ZINC000217668839 IG In-Stock Unstable EPHX2 18 50 COC[C@@H](C)Nc1ccc(S(=O)(=O)N[C@H](C)COC)cc1C(=O)O ZINC000217668862 FD In-Stock Unstable MMP12 45 34 CC1=CC[C@](N)(Cc2ccccc2)C1 ZINC000217668882 AF For-Sale Unstable KDM1A 25 41 COC(=O)[C@H]1CN(C)C[C@@H]1c1cccc(N)c1 ZINC000217668895 BD In-Stock Unstable SLC6A1 99 52 COC(=O)[C@H]1CN(C)C[C@@H]1c1cccc(N)c1 ZINC000217668895 BD In-Stock Unstable SLC6A3 39 41 COc1ccc(OC)c(NC(=O)N/C=C/c2ccccc2C)c1 ZINC000217668922 DH For-Sale Unstable CYP1B1 43 41 COc1ccc(OC)c(NC(=O)N/C=C/c2ccccc2C)c1 ZINC000217668922 DH For-Sale Unstable MTNR1A 22 49 COc1ccc(OC)c(NC(=O)N/C=C/c2ccccc2C)c1 ZINC000217668922 DH For-Sale Unstable MTNR1B 22 49 COc1ccc(OC)c(NC(=O)N/C=C/c2ccccc2C)c1 ZINC000217668922 DH For-Sale Unstable ABCG2 15 40 COc1ccc(OC)c(NC(=O)N/C=C/c2ccccc2C)c1 ZINC000217668922 DH For-Sale Unstable AKR1C2 45 34 COC[C@H](C)Nc1ccc(S(=O)(=O)N[C@H](C)COC)cc1C(=O)O ZINC000217668957 FD In-Stock Unstable MMP12 45 34 CC1=CC[C@@](N)(Cc2ccccc2)C1 ZINC000217668978 AF For-Sale Unstable KDM1A 25 41 COC(=O)[C@@H]1CN(C)C[C@@H]1c1ccc(N)cc1 ZINC000217668999 BD In-Stock Unstable SLC6A1 167 58 COC(=O)[C@@H]1CN(C)C[C@@H]1c1ccc(N)cc1 ZINC000217668999 BD In-Stock Unstable SLC6A4 31 58 COC(=O)[C@@H]1CN(C)C[C@@H]1c1ccc(N)cc1 ZINC000217668999 BD In-Stock Unstable SLC6A3 61 54 CCc1cccc(C)c1NC(=O)N/C=C/c1ccccc1C ZINC000217669021 CJ For-Sale Unstable S1PR4 0 40 CCc1cccc(C)c1NC(=O)N/C=C/c1ccccc1C ZINC000217669021 CJ For-Sale Unstable ACAT 0 41 OC/C=C\c1cccc(OCc2ccccc2)c1 ZINC000217669023 BG For-Sale Unstable ALOX5 17 43 OC/C=C\c1cccc(OCc2ccccc2)c1 ZINC000217669023 BG For-Sale Unstable MAOB 45 41 OC/C=C\c1cccc(OCc2ccccc2)c1 ZINC000217669023 BG For-Sale Unstable PTGER2 29 49 OC/C=C\c1cccc(OCc2ccccc2)c1 ZINC000217669023 BG For-Sale Unstable ACR 20 40 OC/C=C\c1cccc(OCc2ccccc2)c1 ZINC000217669023 BG For-Sale Unstable FFAR1 23 45 CO[P@](=O)(O)CCCCCCCCCCCCCCCCCCC(=O)O ZINC000217669049 GK For-Sale Unstable FABP4 16 46 CO[P@](=O)(O)CCCCCCCCCCCCCCCCCCC(=O)O ZINC000217669049 GK For-Sale Unstable FABP5 15 46 COC(=O)[C@H]1CN(C)C[C@@H]1c1ccc(N)cc1 ZINC000217669071 BD In-Stock Unstable SLC6A1 167 58 COC(=O)[C@H]1CN(C)C[C@@H]1c1ccc(N)cc1 ZINC000217669071 BD In-Stock Unstable SLC6A4 31 58 COC(=O)[C@H]1CN(C)C[C@@H]1c1ccc(N)cc1 ZINC000217669071 BD In-Stock Unstable SLC6A3 61 54 Cc1cc(C)c(NC(=O)N/C=C/c2ccccc2C)c(C)c1 ZINC000217669136 CJ For-Sale Unstable PYGL 40 37 CCN(CCC(=O)Nc1cccc(S(=O)(=O)N2CCCC2)c1)Cc1cccs1 ZINC000217669156 HG On-Demand Unstable LPL 44 36 COC(=O)[C@@H]1CN(C)C[C@@H]1c1ccccc1Cl ZINC000217669189 CE In-Stock Unstable SLC6A1 71 54 COC(=O)[C@@H]1CN(C)C[C@@H]1c1ccccc1Cl ZINC000217669189 CE In-Stock Unstable SLC6A3 29 52 COC(=O)[C@H]1CN(C)C[C@@H]1c1ccccc1Cl ZINC000217669268 CE In-Stock Unstable SLC6A1 0 54 COC(=O)[C@H]1CN(C)C[C@@H]1c1ccccc1Cl ZINC000217669268 CE In-Stock Unstable SLC6A4 0 52 COC(=O)[C@H]1CN(C)C[C@@H]1c1ccccc1Cl ZINC000217669268 CE In-Stock Unstable SLC6A3 29 52 O=C(O)/C=C\c1ccc(F)c(C(=O)NCC2CCC2)c1 ZINC000217669269 CE For-Sale Unstable CACNA1I 55 33 CCCCCCCCCCNCCN(CC)CCC ZINC000217669301 CI For-Sale Unstable PAOX 18 44 CCCCCCCCCCNCCN(CC)CCC ZINC000217669301 CI For-Sale Unstable S1PR2 17 41 COC(=O)[C@@H]1CN(C)C[C@@H]1c1cccc(Cl)c1 ZINC000217669378 CE In-Stock Unstable SLC6A2 15 47 COC(=O)[C@@H]1CN(C)C[C@@H]1c1cccc(Cl)c1 ZINC000217669378 CE In-Stock Unstable SLC6A1 146 56 COC(=O)[C@@H]1CN(C)C[C@@H]1c1cccc(Cl)c1 ZINC000217669378 CE In-Stock Unstable SLC6A4 32 56 COC(=O)[C@@H]1CN(C)C[C@@H]1c1cccc(Cl)c1 ZINC000217669378 CE In-Stock Unstable SLC6A3 54 56 COC(=O)[C@@H]1CN(C)C[C@@H]1c1cccc(Cl)c1 ZINC000217669378 CE In-Stock Unstable MDM2 67 34 CCNC(=O)Cc1cc(OC)c(OC)cc1N ZINC000217669409 BC In-Stock Unstable HTR4 40 36 CC[C@@H](N[C@@H]1CCC[C@@H](O)C1)c1ccc(Cl)cc1 ZINC000217669413 CH For-Sale Unstable SLC6A1 24 43 COc1nc(NCCc2ccc(F)cc2)nc(-c2ccc(OC)c(S(=O)(=O)NC3CC3)c2)n1 ZINC000217669455 JF Annotated Unstable ADRA1D 21 40 COc1nc(NCCc2ccc(F)cc2)nc(-c2ccc(OC)c(S(=O)(=O)NC3CC3)c2)n1 ZINC000217669455 JF Annotated Unstable ADRA1B 26 40 COC(=O)[C@H]1CN(C)C[C@@H]1c1cccc(Cl)c1 ZINC000217669467 CE In-Stock Unstable SLC6A1 146 56 COC(=O)[C@H]1CN(C)C[C@@H]1c1cccc(Cl)c1 ZINC000217669467 CE In-Stock Unstable SLC6A4 32 56 COC(=O)[C@H]1CN(C)C[C@@H]1c1cccc(Cl)c1 ZINC000217669467 CE In-Stock Unstable SLC6A3 54 56 COC(=O)[C@H]1CN(C)C[C@@H]1c1cccc(Cl)c1 ZINC000217669467 CE In-Stock Unstable MDM2 53 32 Cc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217669484 EI For-Sale Unstable DDX3X 0 41 Cc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217669484 EI For-Sale Unstable IMDH_CRYPV 33 47 Cc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217669484 EI For-Sale Unstable BLM 0 46 CC[C@H](N[C@@H]1CCC[C@@H](O)C1)c1ccc(Cl)cc1 ZINC000217669496 CH On-Demand Unstable SLC6A1 24 43 CCN(CC)C(=O)Cc1cc(OC)c(OC)cc1N ZINC000217669519 CD In-Stock Unstable HTR4 17 40 COc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)NCC(=O)c1ccccc1)C(=O)OC2 ZINC000217669572 IH In-Stock Unstable IMPDH1 0 82 COc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)NCC(=O)c1ccccc1)C(=O)OC2 ZINC000217669572 IH In-Stock Unstable IMPDH2 0 82 COC(=O)[C@@H]1CN(C)C[C@@H]1c1cccc([N+](=O)[O-])c1 ZINC000217669573 CD In-Stock Unstable SLC6A4 18 49 COC(=O)[C@@H]1CN(C)C[C@@H]1c1cccc([N+](=O)[O-])c1 ZINC000217669573 CD In-Stock Unstable SLC6A3 28 49 COC(=O)[C@@H]1CN(C)C[C@@H]1c1cccc([N+](=O)[O-])c1 ZINC000217669573 CD In-Stock Unstable CACNA1C 69 42 COC(=O)[C@@H]1CN(C)C[C@@H]1c1cccc([N+](=O)[O-])c1 ZINC000217669573 CD In-Stock Unstable CACNA1D 101 42 CC[C@@H](N[C@H]1CCC[C@@H](O)C1)c1ccc(Cl)cc1 ZINC000217669576 CH For-Sale Unstable SLC6A1 24 43 Cn1nccc1NS(=O)(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217669585 DD On-Demand Unstable OXTR 40 37 COc1cc([N+](=O)[O-])ccc1NC(=O)N/C=C/c1ccccc1C ZINC000217669605 EH For-Sale Unstable EPHX1 0 54 COc1cc([N+](=O)[O-])ccc1NC(=O)N/C=C/c1ccccc1C ZINC000217669605 EH For-Sale Unstable CACNA1D 55 33 COc1cc([N+](=O)[O-])ccc1NC(=O)N/C=C/c1ccccc1C ZINC000217669605 EH For-Sale Unstable KCNMA1 29 54 COc1cc([N+](=O)[O-])ccc1NC(=O)N/C=C/c1ccccc1C ZINC000217669605 EH For-Sale Unstable DDX3X 0 44 COC(=O)[C@@H](O)CNC(=O)COc1ccccc1C#N ZINC000217669606 CB On-Demand Unstable ADRB1 53 42 COC(=O)[C@@H](O)CNC(=O)COc1ccccc1C#N ZINC000217669606 CB On-Demand Unstable CASR 41 41 COC(=O)[C@@H](O)CNC(=O)COc1ccccc1C#N ZINC000217669606 CB On-Demand Unstable CYP2D6 15 41 CCCNC(=O)Cc1cc(OC)c(OC)cc1N ZINC000217669646 CD In-Stock Unstable HTR4 42 37 CCCNC(=O)Cc1cc(OC)c(OC)cc1N ZINC000217669646 CD In-Stock Unstable CAN2 0 40 COC(=O)[C@H]1CN(C)C[C@@H]1c1cccc([N+](=O)[O-])c1 ZINC000217669655 CD In-Stock Unstable SLC6A4 18 49 COC(=O)[C@H]1CN(C)C[C@@H]1c1cccc([N+](=O)[O-])c1 ZINC000217669655 CD In-Stock Unstable SLC6A3 28 49 COC(=O)[C@H]1CN(C)C[C@@H]1c1cccc([N+](=O)[O-])c1 ZINC000217669655 CD In-Stock Unstable CACNA1C 69 42 COC(=O)[C@H]1CN(C)C[C@@H]1c1cccc([N+](=O)[O-])c1 ZINC000217669655 CD In-Stock Unstable CACNA1D 101 42 CC[C@H](N[C@H]1CCC[C@@H](O)C1)c1ccc(Cl)cc1 ZINC000217669665 CH On-Demand Unstable SLC6A1 24 43 COC(=O)[C@H](O)CNC(=O)COc1ccccc1C#N ZINC000217669692 CB On-Demand Unstable ADRB1 53 42 COC(=O)[C@H](O)CNC(=O)COc1ccccc1C#N ZINC000217669692 CB On-Demand Unstable CASR 41 41 COC(=O)[C@H](O)CNC(=O)COc1ccccc1C#N ZINC000217669692 CB On-Demand Unstable CYP2D6 15 41 O=C(CCN1CCN([C@@H]2CCS(=O)(=O)C2)CC1)N[C@@H]1CCCc2ccccc21 ZINC000217669727 HD On-Demand Unstable HTR7 17 57 O=C(CCN1CCN([C@@H]2CCS(=O)(=O)C2)CC1)N[C@@H]1CCCc2ccccc21 ZINC000217669727 HD On-Demand Unstable HTR3B 0 46 Cc1ccccc1/C=C/NC(=O)Nc1ccc([N+](=O)[O-])cc1 ZINC000217669731 CH For-Sale Unstable NMBR 55 33 Cc1ccccc1/C=C/NC(=O)Nc1ccc([N+](=O)[O-])cc1 ZINC000217669731 CH For-Sale Unstable MMP8 15 41 COC(=O)[C@@H]1CN(C)C[C@@H]1c1ccc([N+](=O)[O-])cc1 ZINC000217669758 CD In-Stock Unstable SLC6A4 27 45 COC(=O)[C@@H]1CN(C)C[C@@H]1c1ccc([N+](=O)[O-])cc1 ZINC000217669758 CD In-Stock Unstable SLC6A3 49 58 COC(=O)[C@@H]1CN(C)C[C@@H]1c1ccc([N+](=O)[O-])cc1 ZINC000217669758 CD In-Stock Unstable SLC27A4 51 34 COC(=O)Nc1ccc(S(=O)(=O)N2CC[C@H](n3cc(-c4ccccc4)nn3)C2)cc1 ZINC000217669771 IF In-Stock Unstable TGM2 66 42 COC(=O)Nc1ccc(S(=O)(=O)N2CC[C@H](n3cc(-c4ccccc4)nn3)C2)cc1 ZINC000217669771 IF In-Stock Unstable F13A1 96 42 COC(=O)Nc1ccc(S(=O)(=O)N2CC[C@H](n3cc(-c4ccccc4)nn3)C2)cc1 ZINC000217669771 IF In-Stock Unstable RAC1 0 40 COC(=O)Nc1ccc(S(=O)(=O)N2CC[C@H](n3cc(-c4ccccc4)nn3)C2)cc1 ZINC000217669771 IF In-Stock Unstable TGM6 0 41 O=C(CCN1CCN([C@H]2CCS(=O)(=O)C2)CC1)N[C@@H]1CCCc2ccccc21 ZINC000217669805 HD On-Demand Unstable HTR7 17 57 O=C(CCN1CCN([C@H]2CCS(=O)(=O)C2)CC1)N[C@@H]1CCCc2ccccc21 ZINC000217669805 HD On-Demand Unstable HTR3B 0 46 Cc1ccccc1/C=C/NC(=O)Nc1cccc([N+](=O)[O-])c1 ZINC000217669829 CH For-Sale Unstable CACNA1D 64 33 Cc1ccccc1/C=C/NC(=O)Nc1cccc([N+](=O)[O-])c1 ZINC000217669829 CH For-Sale Unstable TRPM8 0 48 Cc1ccccc1/C=C/NC(=O)Nc1cccc([N+](=O)[O-])c1 ZINC000217669829 CH For-Sale Unstable KCNK3 44 36 COC(=O)Nc1ccc(S(=O)(=O)N2CC[C@@H](n3cc(-c4ccccc4)nn3)C2)cc1 ZINC000217669852 IF In-Stock Unstable TGM2 66 42 COC(=O)Nc1ccc(S(=O)(=O)N2CC[C@@H](n3cc(-c4ccccc4)nn3)C2)cc1 ZINC000217669852 IF In-Stock Unstable F13A1 96 42 COC(=O)Nc1ccc(S(=O)(=O)N2CC[C@@H](n3cc(-c4ccccc4)nn3)C2)cc1 ZINC000217669852 IF In-Stock Unstable RAC1 0 40 COC(=O)Nc1ccc(S(=O)(=O)N2CC[C@@H](n3cc(-c4ccccc4)nn3)C2)cc1 ZINC000217669852 IF In-Stock Unstable TGM6 0 41 COC(=O)[C@H]1CN(C)C[C@@H]1c1ccc([N+](=O)[O-])cc1 ZINC000217669856 CD In-Stock Unstable SLC6A4 27 45 COC(=O)[C@H]1CN(C)C[C@@H]1c1ccc([N+](=O)[O-])cc1 ZINC000217669856 CD In-Stock Unstable SLC6A3 49 58 COC(=O)[C@H]1CN(C)C[C@@H]1c1ccc([N+](=O)[O-])cc1 ZINC000217669856 CD In-Stock Unstable SLC27A4 51 34 CCCCNC(=O)Cc1cc(OC)c(OC)cc1N ZINC000217669872 CD In-Stock Unstable HTR4 38 40 CCCCNC(=O)Cc1cc(OC)c(OC)cc1N ZINC000217669872 CD In-Stock Unstable ACAT 0 42 CCCCNC(=O)Cc1cc(OC)c(OC)cc1N ZINC000217669872 CD In-Stock Unstable CAN2 0 44 O=C(CCN1CCN([C@@H]2CCS(=O)(=O)C2)CC1)N[C@H]1CCCc2ccccc21 ZINC000217669880 HD On-Demand Unstable HTR7 17 57 O=C(CCN1CCN([C@@H]2CCS(=O)(=O)C2)CC1)N[C@H]1CCCc2ccccc21 ZINC000217669880 HD On-Demand Unstable HTR3B 0 46 CC(C)NC(=O)CNC(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217669886 CD For-Sale Unstable CA2 27 46 Cc1ccn(C[C@@H](C(=O)O)C(F)(F)F)c(=O)c1 ZINC000217669888 BD For-Sale Unstable IDH1 63 35 COc1ccc([C@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2oc(C)cc(=O)c2O)c(OC)c1 ZINC000217669909 JI In-Stock Unstable RORC 40 40 COC(=O)[C@H]1CN(C)C[C@@H]1c1ccccc1OC ZINC000217669936 BD In-Stock Unstable SLC6A1 49 54 COC(=O)[C@H]1CN(C)C[C@@H]1c1ccccc1OC ZINC000217669936 BD In-Stock Unstable SLC6A3 22 48 Cc1ccccc1/C=C/NC(=O)Nc1cc([N+](=O)[O-])ccc1Cl ZINC000217669950 EI For-Sale Unstable DDX3X 0 46 O=C(CCN1CCN([C@H]2CCS(=O)(=O)C2)CC1)N[C@H]1CCCc2ccccc21 ZINC000217669961 HD On-Demand Unstable HTR7 17 57 O=C(CCN1CCN([C@H]2CCS(=O)(=O)C2)CC1)N[C@H]1CCCc2ccccc21 ZINC000217669961 HD On-Demand Unstable HTR3B 0 46 O=C(C1CCC1)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217669963 CE In-Stock Unstable PREP 30 51 O=C(C1CCC1)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217669963 CE In-Stock Unstable FIMH 20 41 Cc1ccn(C[C@H](C(=O)O)C(F)(F)F)c(=O)c1 ZINC000217669969 BD For-Sale Unstable IDH1 63 35 CC(C)NC(=O)CNC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217669985 CD For-Sale Unstable HDAC8 19 43 CC(C)NC(=O)CNC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217669985 CD For-Sale Unstable CCR2 47 40 COc1ccc([C@@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2oc(C)cc(=O)c2O)c(OC)c1 ZINC000217669986 JI In-Stock Unstable RORC 40 40 COC(=O)[C@@H]1CN(C)C[C@@H]1c1cccc(OC)c1 ZINC000217670054 BD In-Stock Unstable DRD4 43 33 COC(=O)[C@@H]1CN(C)C[C@@H]1c1cccc(OC)c1 ZINC000217670054 BD In-Stock Unstable SLC6A1 114 55 COC(=O)[C@@H]1CN(C)C[C@@H]1c1cccc(OC)c1 ZINC000217670054 BD In-Stock Unstable SLC6A3 42 41 COc1ccc(C(=O)N[C@H](C)C(C)C)cc1/C=C\C(=O)O ZINC000217670067 CF For-Sale Unstable TNFRSF1A 23 40 O=C(CCN1CCN([C@@H]2CCS(=O)(=O)C2)CC1)NC(c1ccccc1)c1ccccc1 ZINC000217670068 IE On-Demand Unstable PRCP 34 52 O=C(CCN1CCN([C@@H]2CCS(=O)(=O)C2)CC1)NC(c1ccccc1)c1ccccc1 ZINC000217670068 IE On-Demand Unstable XIAP 41 34 O=C(CCN1CCN([C@@H]2CCS(=O)(=O)C2)CC1)NC(c1ccccc1)c1ccccc1 ZINC000217670068 IE On-Demand Unstable BIRC8 56 34 O=C(c1cnccn1)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217670073 DD In-Stock Unstable PREP 20 44 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccsc2)CC(=O)O4)cc1O ZINC000217670102 II In-Stock Unstable AKR1B1 22 48 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccsc2)CC(=O)O4)cc1O ZINC000217670102 II In-Stock Unstable CYP1B1 50 48 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccsc2)CC(=O)O4)cc1O ZINC000217670102 II In-Stock Unstable CYP1A1 39 48 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccsc2)CC(=O)O4)cc1O ZINC000217670102 II In-Stock Unstable CYP1A2 30 40 COC(=O)[C@H]1CN(C)C[C@@H]1c1cccc(OC)c1 ZINC000217670136 BD In-Stock Unstable DRD4 43 33 COC(=O)[C@H]1CN(C)C[C@@H]1c1cccc(OC)c1 ZINC000217670136 BD In-Stock Unstable SLC6A1 114 55 COC(=O)[C@H]1CN(C)C[C@@H]1c1cccc(OC)c1 ZINC000217670136 BD In-Stock Unstable SLC6A3 42 41 CCC[C@@H](NCCN(CC)CCC)c1ccc(Cl)cc1 ZINC000217670148 CJ For-Sale Unstable UTS2 43 35 O=C(CCN1CCN([C@H]2CCS(=O)(=O)C2)CC1)NC(c1ccccc1)c1ccccc1 ZINC000217670156 IE On-Demand Unstable PRCP 34 52 O=C(CCN1CCN([C@H]2CCS(=O)(=O)C2)CC1)NC(c1ccccc1)c1ccccc1 ZINC000217670156 IE On-Demand Unstable XIAP 41 34 O=C(CCN1CCN([C@H]2CCS(=O)(=O)C2)CC1)NC(c1ccccc1)c1ccccc1 ZINC000217670156 IE On-Demand Unstable BIRC8 56 34 COc1ccc(C(=O)N[C@@H](C)C(C)C)cc1/C=C\C(=O)O ZINC000217670159 CF For-Sale Unstable TNFRSF1A 23 40 Cc1ccccc1C(=O)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217670178 DF In-Stock Unstable PREP 19 43 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccsc2)CC(=O)O4)cc1O ZINC000217670187 II In-Stock Unstable AKR1B1 22 48 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccsc2)CC(=O)O4)cc1O ZINC000217670187 II In-Stock Unstable CYP1B1 50 48 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccsc2)CC(=O)O4)cc1O ZINC000217670187 II In-Stock Unstable CYP1A1 39 48 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccsc2)CC(=O)O4)cc1O ZINC000217670187 II In-Stock Unstable CYP1A2 30 40 CCC[C@H](NCCN(CC)CCC)c1ccc(Cl)cc1 ZINC000217670221 CJ For-Sale Unstable UTS2 43 35 c1cnc2c(-c3ccc(N(c4ccc(-c5cccc6cccnc56)cc4)c4ccc(-c5cccc6cccnc56)cc4)cc3)cccc2c1 ZINC000217670258 KK For-Sale Anodyne CCR1 18 52 c1cnc2c(-c3ccc(N(c4ccc(-c5cccc6cccnc56)cc4)c4ccc(-c5cccc6cccnc56)cc4)cc3)cccc2c1 ZINC000217670258 KK For-Sale Anodyne METAP2 17 45 O=C(CCN1CCN([C@@H]2CCS(=O)(=O)C2)CC1)Nc1ccccc1-c1ccccc1 ZINC000217670264 IE On-Demand Unstable CHRM3 22 45 O=C(CCN1CCN([C@@H]2CCS(=O)(=O)C2)CC1)Nc1ccccc1-c1ccccc1 ZINC000217670264 IE On-Demand Unstable PRCP 15 41 COC(=O)[C@@H]1CN(C)C[C@@H]1c1ccc(OC)cc1 ZINC000217670269 BD In-Stock Unstable SLC6A2 16 58 COC(=O)[C@@H]1CN(C)C[C@@H]1c1ccc(OC)cc1 ZINC000217670269 BD In-Stock Unstable SLC6A1 176 58 COC(=O)[C@@H]1CN(C)C[C@@H]1c1ccc(OC)cc1 ZINC000217670269 BD In-Stock Unstable SLC6A4 35 56 COC(=O)[C@@H]1CN(C)C[C@@H]1c1ccc(OC)cc1 ZINC000217670269 BD In-Stock Unstable SLC6A3 64 54 COC(=O)[C@@H]1CN(C)C[C@@H]1c1ccc(OC)cc1 ZINC000217670269 BD In-Stock Unstable CACNA1S 40 33 COc1cc(N)c(CC(=O)NCC(C)C)cc1OC ZINC000217670279 CD In-Stock Unstable TRPV1 15 42 Cc1ccccc1/C=C/NC(=O)N1CCN(c2ccc(F)cc2)CC1 ZINC000217670282 EH For-Sale Unstable AKR1C3 0 43 O=C(CCN1CCN([C@H]2CCS(=O)(=O)C2)CC1)Nc1ccccc1-c1ccccc1 ZINC000217670352 IE On-Demand Unstable CHRM3 22 45 O=C(CCN1CCN([C@H]2CCS(=O)(=O)C2)CC1)Nc1ccccc1-c1ccccc1 ZINC000217670352 IE On-Demand Unstable PRCP 15 41 COC(=O)[C@H]1CN(C)C[C@@H]1c1ccc(OC)cc1 ZINC000217670354 BD In-Stock Unstable SLC6A2 16 58 COC(=O)[C@H]1CN(C)C[C@@H]1c1ccc(OC)cc1 ZINC000217670354 BD In-Stock Unstable SLC6A1 176 58 COC(=O)[C@H]1CN(C)C[C@@H]1c1ccc(OC)cc1 ZINC000217670354 BD In-Stock Unstable SLC6A4 35 56 COC(=O)[C@H]1CN(C)C[C@@H]1c1ccc(OC)cc1 ZINC000217670354 BD In-Stock Unstable SLC6A3 64 54 COC(=O)[C@H]1CN(C)C[C@@H]1c1ccc(OC)cc1 ZINC000217670354 BD In-Stock Unstable CACNA1S 40 33 COc1cc(N)c(CC(=O)NC2CC2)cc1OC ZINC000217670384 CD In-Stock Unstable HTR4 69 45 Cc1nnsc1C(=O)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217670387 ED In-Stock Unstable PREP 19 42 COC(=O)[C@@H](O)CNC(=O)c1ccc(S(C)(=O)=O)cc1 ZINC000217670395 DB On-Demand Unstable CA2 39 43 COC(=O)[C@@H](O)CNC(=O)c1ccc(S(C)(=O)=O)cc1 ZINC000217670395 DB On-Demand Unstable PTGS2 17 44 COC(=O)[C@@H](O)CNC(=O)c1ccc(S(C)(=O)=O)cc1 ZINC000217670395 DB On-Demand Unstable CA1 19 42 COC(=O)[C@@H](O)CNC(=O)c1ccc(S(C)(=O)=O)cc1 ZINC000217670395 DB On-Demand Unstable CA4 15 42 COC(=O)[C@@H](O)CNC(=O)c1ccc(S(C)(=O)=O)cc1 ZINC000217670395 DB On-Demand Unstable CA14 21 44 COC(=O)[C@@H](O)CNC(=O)c1ccc(S(C)(=O)=O)cc1 ZINC000217670395 DB On-Demand Unstable ITGAV 47 38 COC(=O)[C@@H](O)CNC(=O)c1ccc(S(C)(=O)=O)cc1 ZINC000217670395 DB On-Demand Unstable LOX1.1 49 35 COC(=O)[C@@H](O)CNC(=O)c1ccc(S(C)(=O)=O)cc1 ZINC000217670395 DB On-Demand Unstable O49150_SOLTU 53 36 COC(=O)[C@@H](O)CNC(=O)c1ccc(S(C)(=O)=O)cc1 ZINC000217670395 DB On-Demand Unstable CYNT 25 40 COC(=O)[C@@H]1CN(C)C[C@@H]1c1ccc2c(c1)OCO2 ZINC000217670469 CD In-Stock Unstable SLC6A3 37 41 COC(=O)[C@@H]1CN(C)C[C@@H]1c1ccc2c(c1)OCO2 ZINC000217670469 CD In-Stock Unstable EDNRB 66 41 COC(=O)[C@@H]1CN(C)C[C@@H]1c1ccc2c(c1)OCO2 ZINC000217670469 CD In-Stock Unstable EDNRA 70 43 CCC=C=CC(=O)c1ccccc1 ZINC000217670477 AF For-Sale Unstable PA 15 41 COC(=O)[C@H](O)CNC(=O)c1ccc(S(C)(=O)=O)cc1 ZINC000217670482 DB On-Demand Unstable CA2 39 43 COC(=O)[C@H](O)CNC(=O)c1ccc(S(C)(=O)=O)cc1 ZINC000217670482 DB On-Demand Unstable PTGS2 17 44 COC(=O)[C@H](O)CNC(=O)c1ccc(S(C)(=O)=O)cc1 ZINC000217670482 DB On-Demand Unstable CA1 19 42 COC(=O)[C@H](O)CNC(=O)c1ccc(S(C)(=O)=O)cc1 ZINC000217670482 DB On-Demand Unstable CA4 15 42 COC(=O)[C@H](O)CNC(=O)c1ccc(S(C)(=O)=O)cc1 ZINC000217670482 DB On-Demand Unstable CA14 21 44 COC(=O)[C@H](O)CNC(=O)c1ccc(S(C)(=O)=O)cc1 ZINC000217670482 DB On-Demand Unstable ITGAV 47 38 COC(=O)[C@H](O)CNC(=O)c1ccc(S(C)(=O)=O)cc1 ZINC000217670482 DB On-Demand Unstable LOX1.1 49 35 COC(=O)[C@H](O)CNC(=O)c1ccc(S(C)(=O)=O)cc1 ZINC000217670482 DB On-Demand Unstable O49150_SOLTU 53 36 COC(=O)[C@H](O)CNC(=O)c1ccc(S(C)(=O)=O)cc1 ZINC000217670482 DB On-Demand Unstable CYNT 25 40 COc1cc2cc(C(=O)NC[C@@H]3CCCN4CCCC[C@H]34)[nH]c2cc1OC ZINC000217670485 FG In-Stock Unstable PYGL 44 38 N#Cc1cccc(C(=O)N2CC(n3cc(-c4ccccc4)nn3)C2)c1 ZINC000217670487 EF In-Stock Unstable ABHD6 0 41 CCOc1ccc(NC(=O)N/C=C/c2ccccc2C)cc1 ZINC000217670498 CI For-Sale Unstable CA1 43 41 CCOc1ccc(NC(=O)N/C=C/c2ccccc2C)cc1 ZINC000217670498 CI For-Sale Unstable CA12 17 41 CCOc1ccc(NC(=O)N/C=C/c2ccccc2C)cc1 ZINC000217670498 CI For-Sale Unstable CA9 19 41 COC(=O)[C@H]1CN(C)C[C@@H]1c1ccc2c(c1)OCO2 ZINC000217670551 CD In-Stock Unstable SLC6A3 37 41 COC(=O)[C@H]1CN(C)C[C@@H]1c1ccc2c(c1)OCO2 ZINC000217670551 CD In-Stock Unstable EDNRB 66 41 COC(=O)[C@H]1CN(C)C[C@@H]1c1ccc2c(c1)OCO2 ZINC000217670551 CD In-Stock Unstable EDNRA 70 43 O=C(O)c1cc(F)c(O)c(Br)c1O ZINC000217670557 CD For-Sale Anodyne AKR1C2 65 50 O=C(O)c1cc(F)c(O)c(Br)c1O ZINC000217670557 CD For-Sale Anodyne AKR1C1 63 50 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(OC)c(OCC(N)=O)c2)CC(=O)O4)cc1O ZINC000217670588 KG In-Stock Unstable AKR1B1 0 46 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(OC)c(OCC(N)=O)c2)CC(=O)O4)cc1O ZINC000217670588 KG In-Stock Unstable CYP1B1 55 34 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(OC)c(OCC(N)=O)c2)CC(=O)O4)cc1O ZINC000217670588 KG In-Stock Unstable CYP1A1 41 44 O=C(/C=C/c1ccccc1)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217670595 EG In-Stock Unstable HDAC8 42 34 O=C(/C=C/c1ccccc1)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217670595 EG In-Stock Unstable PREP 21 44 O=C(O)/C=C\c1ccc(C(=O)NCc2cccnc2)s1 ZINC000217670600 CE For-Sale Unstable TBXAS1 27 62 O=C(O)/C=C\c1ccc(C(=O)NCc2cccnc2)s1 ZINC000217670600 CE For-Sale Unstable CHRNA7 27 40 O=C(O)/C=C\c1ccc(C(=O)NCc2cccnc2)s1 ZINC000217670600 CE For-Sale Unstable HDAC1 15 43 O=C(O)/C=C\c1ccc(C(=O)NCc2cccnc2)s1 ZINC000217670600 CE For-Sale Unstable SCD1 22 42 O=C(O)/C=C\c1ccc(C(=O)NCc2cccnc2)s1 ZINC000217670600 CE For-Sale Unstable SCD 25 42 O=C(O)/C=C\c1ccc(C(=O)NCc2cccnc2)s1 ZINC000217670600 CE For-Sale Unstable NAMPT 87 42 COc1cc(N)c(CC(=O)NC2CCCCC2)cc1OC ZINC000217670617 CE In-Stock Unstable HTR4 67 45 COc1cc(N)c(CC(=O)NC2CCCCC2)cc1OC ZINC000217670617 CE In-Stock Unstable EPHX2 20 44 COc1cc(N)c(CC(=O)NC2CCCCC2)cc1OC ZINC000217670617 CE In-Stock Unstable STK17B 40 35 COC(=O)[C@@H]1CN(C)C[C@@H]1c1ccc(OC)c(OC)c1 ZINC000217670647 CD In-Stock Unstable SLC6A3 44 39 COC(=O)[C@@H]1CN(C)C[C@@H]1c1ccc(OC)c(OC)c1 ZINC000217670647 CD In-Stock Unstable PDE4B 21 58 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(OC)c(OCC(N)=O)c2)CC(=O)O4)cc1O ZINC000217670663 KG In-Stock Unstable AKR1B1 0 46 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(OC)c(OCC(N)=O)c2)CC(=O)O4)cc1O ZINC000217670663 KG In-Stock Unstable CYP1B1 55 34 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(OC)c(OCC(N)=O)c2)CC(=O)O4)cc1O ZINC000217670663 KG In-Stock Unstable CYP1A1 41 44 C[C@@H](c1nc2ccccc2s1)N(C)CCC(=O)NCc1ccccc1Cl ZINC000217670677 GJ On-Demand Unstable P2RX7 19 41 C[C@@H](c1nc2ccccc2s1)N(C)CCC(=O)NCc1ccccc1Cl ZINC000217670677 GJ On-Demand Unstable SLC6A12 0 40 O=C(O)/C=C\c1cccc(C(=O)NCc2cccnc2)c1 ZINC000217670680 CE For-Sale Unstable TBXAS1 59 54 O=C(O)/C=C\c1cccc(C(=O)NCc2cccnc2)c1 ZINC000217670680 CE For-Sale Unstable PTAFR 29 41 O=C(O)/C=C\c1cccc(C(=O)NCc2cccnc2)c1 ZINC000217670680 CE For-Sale Unstable HDAC8 18 50 O=C(O)/C=C\c1cccc(C(=O)NCc2cccnc2)c1 ZINC000217670680 CE For-Sale Unstable HDAC1 15 42 O=C(O)/C=C\c1cccc(C(=O)NCc2cccnc2)c1 ZINC000217670680 CE For-Sale Unstable HDAC6 15 50 O=C(O)/C=C\c1cccc(C(=O)NCc2cccnc2)c1 ZINC000217670680 CE For-Sale Unstable NAMPT 97 46 O=C(O)c1cc(Br)c(O)c(F)c1O ZINC000217670694 CD For-Sale Anodyne AKR1C2 68 59 O=C(O)c1cc(Br)c(O)c(F)c1O ZINC000217670694 CD For-Sale Anodyne AKR1C1 65 59 COc1ccc(C(=O)N2CC(n3cc(-c4ccccc4)nn3)C2)cc1 ZINC000217670713 EF In-Stock Unstable AVPR1A 19 42 COc1ccc(C(=O)N2CC(n3cc(-c4ccccc4)nn3)C2)cc1 ZINC000217670713 EF In-Stock Unstable SLC18A3 15 42 COc1ccc(C(=O)N2CC(n3cc(-c4ccccc4)nn3)C2)cc1 ZINC000217670713 EF In-Stock Unstable PREP 21 43 COc1ccc(C(=O)N2CC(n3cc(-c4ccccc4)nn3)C2)cc1 ZINC000217670713 EF In-Stock Unstable SLC6A7 0 42 COc1cc(N)c(CC(=O)N2CCCC2)cc1OC ZINC000217670718 CD In-Stock Unstable HTR4 65 42 COC(=O)[C@H]1CN(C)C[C@@H]1c1ccc(OC)c(OC)c1 ZINC000217670739 CD In-Stock Unstable SLC6A3 44 39 COC(=O)[C@H]1CN(C)C[C@@H]1c1ccc(OC)c(OC)c1 ZINC000217670739 CD In-Stock Unstable PDE4B 21 58 CCCNC[C@@H](c1ccccc1)N1CCCO[C@@H](C)C1 ZINC000217670740 CF For-Sale Unstable CCR3 42 39 C[C@H](c1nc2ccccc2s1)N(C)CCC(=O)NCc1ccccc1Cl ZINC000217670760 GJ On-Demand Unstable P2RX7 19 41 C[C@H](c1nc2ccccc2s1)N(C)CCC(=O)NCc1ccccc1Cl ZINC000217670760 GJ On-Demand Unstable SLC6A12 0 40 Cc1cc(NS(=O)(=O)c2cccs2)ccc1/C=C\C(=O)O ZINC000217670768 DF For-Sale Unstable PTGER3 23 43 CSCC[C@H](Nc1nc(C)cc(C)n1)C(=O)N1CCc2c([nH]c3ccccc23)C1 ZINC000217670785 HH In-Stock Unstable SSTR4 50 34 CSCC[C@H](Nc1nc(C)cc(C)n1)C(=O)N1CCc2c([nH]c3ccccc23)C1 ZINC000217670785 HH In-Stock Unstable SSTR5 40 34 CCCNC[C@H](c1ccccc1)N1CCCO[C@@H](C)C1 ZINC000217670812 CF For-Sale Unstable CCR3 42 39 O=C(Cc1ccc(F)cc1)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217670830 EF In-Stock Unstable PREP 24 46 CC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2C)c1 ZINC000217670833 CH For-Sale Unstable CCR3 18 41 CC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2C)c1 ZINC000217670833 CH For-Sale Unstable AKR1C3 24 44 CC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2C)c1 ZINC000217670833 CH For-Sale Unstable KCNK3 101 43 CC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2C)c1 ZINC000217670833 CH For-Sale Unstable KCNK9 53 40 COC(=O)[C@@H]1CN(C)C[C@@H]1c1cccs1 ZINC000217670840 BD In-Stock Unstable SLC6A1 82 47 COC(=O)[C@@H]1CN(C)C[C@@H]1c1cccs1 ZINC000217670840 BD In-Stock Unstable SLC6A4 22 40 COC(=O)[C@@H]1CN(C)C[C@@H]1c1cccs1 ZINC000217670840 BD In-Stock Unstable SLC6A3 29 46 COc1cc(N)c(CC(=O)N2CCCCC2)cc1OC ZINC000217670844 CD In-Stock Unstable HTR4 61 42 CSCC[C@@H](Nc1nc(C)cc(C)n1)C(=O)N1CCc2c([nH]c3ccccc23)C1 ZINC000217670876 HH In-Stock Unstable SSTR4 50 34 CSCC[C@@H](Nc1nc(C)cc(C)n1)C(=O)N1CCc2c([nH]c3ccccc23)C1 ZINC000217670876 HH In-Stock Unstable SSTR5 40 34 N#Cc1ccccc1NC(=O)CCN1CCN(S(=O)(=O)c2ccc(F)cc2F)CC1 ZINC000217670904 IE On-Demand Unstable HTR2A 17 46 N#Cc1ccccc1NC(=O)CCN1CCN(S(=O)(=O)c2ccc(F)cc2F)CC1 ZINC000217670904 IE On-Demand Unstable TRPV4 46 38 COC(=O)[C@H]1CN(C)C[C@@H]1c1cccs1 ZINC000217670925 BD In-Stock Unstable SLC6A1 82 47 COC(=O)[C@H]1CN(C)C[C@@H]1c1cccs1 ZINC000217670925 BD In-Stock Unstable SLC6A4 22 40 COC(=O)[C@H]1CN(C)C[C@@H]1c1cccs1 ZINC000217670925 BD In-Stock Unstable SLC6A3 29 46 CCc1ccc(CCN2[C@H]3CC[C@H]2CC(=O)C3)cc1 ZINC000217670953 CF On-Demand Unstable Q8WSF8_APLCA 17 42 COc1cc(N)c(CC(=O)N2CCOCC2)cc1OC ZINC000217670970 CC In-Stock Unstable HTR4 52 35 CCOC(=O)[C@H](c1ccccc1)N1C[C@H](C)O[C@@H](C)C1 ZINC000217670972 CE On-Demand Unstable NPY2R 38 40 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccnn2C)CC(=O)O4)cc1O ZINC000217670991 IG In-Stock Unstable AKR1B1 0 47 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccnn2C)CC(=O)O4)cc1O ZINC000217670991 IG In-Stock Unstable CYP1B1 56 35 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccnn2C)CC(=O)O4)cc1O ZINC000217670991 IG In-Stock Unstable CYP1A1 40 47 COC(=O)[C@@H](O)CNC(=O)c1ccc(C)c(OC)c1 ZINC000217671024 CC On-Demand Unstable DRD4 43 35 COC(=O)[C@@H](O)CNC(=O)c1ccc(C)c(OC)c1 ZINC000217671024 CC On-Demand Unstable CYSLTR1 40 34 COC(=O)[C@@H]1CN(C)C[C@@H]1c1ccco1 ZINC000217671032 BD In-Stock Unstable SLC6A1 42 48 COC(=O)[C@@H]1CN(C)C[C@@H]1c1ccco1 ZINC000217671032 BD In-Stock Unstable SLC6A3 19 56 COc1cc(N)c(CC(=O)N2CCC(C)CC2)cc1OC ZINC000217671074 CE In-Stock Unstable HTR4 64 46 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccnn2C)CC(=O)O4)cc1O ZINC000217671082 IG In-Stock Unstable AKR1B1 0 47 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccnn2C)CC(=O)O4)cc1O ZINC000217671082 IG In-Stock Unstable CYP1B1 56 35 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccnn2C)CC(=O)O4)cc1O ZINC000217671082 IG In-Stock Unstable CYP1A1 40 47 Cn1nccc1NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217671090 CD For-Sale Unstable HDAC8 32 44 Cn1nccc1NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217671090 CD For-Sale Unstable HDAC6 19 44 Cn1nccc1NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217671090 CD For-Sale Unstable KCNK3 75 36 COC(=O)[C@H](O)CNC(=O)c1ccc(C)c(OC)c1 ZINC000217671099 CC On-Demand Unstable DRD4 43 35 COC(=O)[C@H](O)CNC(=O)c1ccc(C)c(OC)c1 ZINC000217671099 CC On-Demand Unstable CYSLTR1 40 34 COC(=O)[C@H]1CN(C)C[C@@H]1c1ccco1 ZINC000217671118 BD In-Stock Unstable SLC6A1 42 48 COC(=O)[C@H]1CN(C)C[C@@H]1c1ccco1 ZINC000217671118 BD In-Stock Unstable SLC6A3 19 56 COc1cc(N)c(CC(=O)N2CCCCCC2)cc1OC ZINC000217671153 CE In-Stock Unstable HTR4 61 42 CCOC(=O)[C@@H](c1ccccc1)N(C)Cc1ccccc1 ZINC000217671188 CG On-Demand Unstable BLAIMP-1 0 40 COCc1cccc(C(=O)NC[C@@H](O)C(=O)OC)c1 ZINC000217671213 CC On-Demand Unstable DRD4 42 33 COC(=O)[C@@H]1CN(C)C[C@@H]1c1ccc(C)o1 ZINC000217671229 BD In-Stock Unstable SLC6A1 31 46 c1cc2c(cc1CN[C@@H]1CCN3CCCC[C@@H]13)OCO2 ZINC000217671246 CE For-Sale Unstable NOS2 55 37 O=C(O)Cc1cc(Br)cc(F)c1F ZINC000217671247 CE For-Sale Unstable AKR1B1 15 43 COc1cc(N)c(CC(=O)Nc2ccccc2)cc1OC ZINC000217671264 CE In-Stock Unstable TSHR 65 32 COc1cc(N)c(CC(=O)Nc2ccccc2)cc1OC ZINC000217671264 CE In-Stock Unstable CPT1A 45 32 COc1cc(N)c(CC(=O)Nc2ccccc2)cc1OC ZINC000217671264 CE In-Stock Unstable CA5B 36 40 COc1cc(N)c(CC(=O)Nc2ccccc2)cc1OC ZINC000217671264 CE In-Stock Unstable CA5A 41 40 COc1cc(N)c(CC(=O)Nc2ccccc2)cc1OC ZINC000217671264 CE In-Stock Unstable MTNR1B 22 42 COc1cc(N)c(CC(=O)Nc2ccccc2)cc1OC ZINC000217671264 CE In-Stock Unstable HDAC1 16 40 COc1cc(N)c(CC(=O)Nc2ccccc2)cc1OC ZINC000217671264 CE In-Stock Unstable HDAC2 19 42 COc1cc(N)c(CC(=O)Nc2ccccc2)cc1OC ZINC000217671264 CE In-Stock Unstable MAPK9 0 42 COc1cc(N)c(CC(=O)Nc2ccccc2)cc1OC ZINC000217671264 CE In-Stock Unstable ACR 19 40 COc1cc(N)c(CC(=O)Nc2ccccc2)cc1OC ZINC000217671264 CE In-Stock Unstable MAPK8 18 42 COc1cc(N)c(CC(=O)Nc2ccccc2)cc1OC ZINC000217671264 CE In-Stock Unstable ENPP1 58 35 COc1cc(N)c(CC(=O)Nc2ccccc2)cc1OC ZINC000217671264 CE In-Stock Unstable GLMU 0 45 COc1cc(N)c(CC(=O)Nc2ccccc2)cc1OC ZINC000217671264 CE In-Stock Unstable KCNK3 45 41 COc1cc(N)c(CC(=O)Nc2ccccc2)cc1OC ZINC000217671264 CE In-Stock Unstable KCNK9 39 41 CCOC(=O)[C@H](c1ccccc1)N(C)Cc1ccccc1 ZINC000217671271 CG On-Demand Unstable BLAIMP-1 0 40 O=C(O)/C=C\c1ccc(F)c(C(=O)Nc2nccs2)c1 ZINC000217671277 CF For-Sale Anodyne MAP1 129 49 O=C(O)/C=C\c1ccc(F)c(C(=O)Nc2nccs2)c1 ZINC000217671277 CF For-Sale Anodyne GCK 25 41 COCc1cccc(C(=O)NC[C@H](O)C(=O)OC)c1 ZINC000217671281 CC On-Demand Unstable DRD4 42 33 COc1ccc(C)cc1NC(=O)N/C=C/c1ccccc1C ZINC000217671293 CI For-Sale Unstable EPHX1 0 40 CCOc1ccccc1C(=O)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217671296 EG In-Stock Unstable HCRTR1 45 34 CCOc1ccccc1C(=O)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217671296 EG In-Stock Unstable PREP 20 43 CCOc1ccccc1C(=O)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217671296 EG In-Stock Unstable HCN1 43 34 CCOc1ccccc1C(=O)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217671296 EG In-Stock Unstable HCN4 43 34 COC(=O)[C@H]1CN(C)C[C@@H]1c1ccc(C)o1 ZINC000217671313 BD In-Stock Unstable SLC6A1 31 46 c1cc2c(cc1CN[C@H]1CCN3CCCC[C@@H]13)OCO2 ZINC000217671315 CE For-Sale Unstable NOS2 55 37 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)NCCCn3ccnc3)[C@H]21 ZINC000217671330 JE In-Stock Unstable QPCT 35 44 O=C(O)/C=C\c1ccc(C(=O)Nc2nccs2)c(F)c1 ZINC000217671361 CF For-Sale Anodyne MAP1 129 49 O=C(O)/C=C\c1ccc(C(=O)Nc2nccs2)c(F)c1 ZINC000217671361 CF For-Sale Anodyne GCK 25 41 COc1cc(N)c(CC(=O)Nc2ccc(C)cc2)cc1OC ZINC000217671362 DF In-Stock Unstable CA12 18 41 COc1cc(N)c(CC(=O)Nc2ccc(C)cc2)cc1OC ZINC000217671362 DF In-Stock Unstable CA9 18 41 COc1cc(N)c(CC(=O)Nc2ccc(C)cc2)cc1OC ZINC000217671362 DF In-Stock Unstable ENPP1 61 37 C[C@H]1N[C@@H](CO)Cc2ccccc21 ZINC000217671377 AD For-Sale Unstable PNMT 20 50 COC(=O)[C@@H](O)CNC(=O)COc1ccc(Cl)c(Cl)c1 ZINC000217671388 DD On-Demand Unstable GRIN1 46 42 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)NCCCn3ccnc3)[C@@H]21 ZINC000217671403 JE In-Stock Unstable QPCT 35 44 O=C(COc1ccccc1F)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217671407 FF In-Stock Unstable PREP 22 45 Cc1ccccc1-c1ccc(C(=O)N2CCN3CCC[C@@H]3C2)cc1 ZINC000217671408 DH In-Stock Unstable AVPR2 26 45 Cc1ccccc1-c1ccc(C(=O)N2CCN3CCC[C@@H]3C2)cc1 ZINC000217671408 DH In-Stock Unstable AVPR1A 25 41 Cc1ccccc1-c1ccc(C(=O)N2CCN3CCC[C@@H]3C2)cc1 ZINC000217671408 DH In-Stock Unstable INHA 25 49 Cc1ccccc1-c1ccc(C(=O)N2CCN3CCC[C@@H]3C2)cc1 ZINC000217671408 DH In-Stock Unstable HRH3 28 52 Cc1ccccc1-c1ccc(C(=O)N2CCN3CCC[C@@H]3C2)cc1 ZINC000217671408 DH In-Stock Unstable HSD11B1 15 40 Cc1ccccc1-c1ccc(C(=O)N2CCN3CCC[C@@H]3C2)cc1 ZINC000217671408 DH In-Stock Unstable L3MBTL1 0 54 Cc1ccccc1-c1ccc(C(=O)N2CCN3CCC[C@@H]3C2)cc1 ZINC000217671408 DH In-Stock Unstable L3MBTL3 104 54 Cc1ccccc1-c1ccc(C(=O)N2CCN3CCC[C@@H]3C2)cc1 ZINC000217671408 DH In-Stock Unstable L3MBTL4 0 41 Cc1ccccc1-c1ccc(C(=O)N2CCN3CCC[C@@H]3C2)cc1 ZINC000217671408 DH In-Stock Unstable MBTD1 0 45 Cc1ccccc1-c1ccc(C(=O)N2CCN3CCC[C@@H]3C2)cc1 ZINC000217671408 DH In-Stock Unstable TP53BP1 0 41 Cc1ccccc1-c1ccc(C(=O)N2CCN3CCC[C@@H]3C2)cc1 ZINC000217671408 DH In-Stock Unstable SLC6A7 0 54 Cc1cccc(NC(=O)N/C=C/c2ccccc2C)c1 ZINC000217671409 CI For-Sale Unstable CCKAR 24 51 Cc1cccc(NC(=O)N/C=C/c2ccccc2C)c1 ZINC000217671409 CI For-Sale Unstable KDR 18 40 Cc1cccc(NC(=O)N/C=C/c2ccccc2C)c1 ZINC000217671409 CI For-Sale Unstable DDX3X 0 43 Cc1cccc(NC(=O)N/C=C/c2ccccc2C)c1 ZINC000217671409 CI For-Sale Unstable KCNK3 110 47 Cc1cccc(NC(=O)N/C=C/c2ccccc2C)c1 ZINC000217671409 CI For-Sale Unstable KCNK9 65 47 Cc1ccc([C@@H]2CN(C)C[C@H]2CO)cc1 ZINC000217671440 BD In-Stock Unstable SLC6A1 64 55 Cc1ccc([C@@H]2CN(C)C[C@H]2CO)cc1 ZINC000217671440 BD In-Stock Unstable SLC6A4 21 44 Cc1ccc([C@@H]2CN(C)C[C@H]2CO)cc1 ZINC000217671440 BD In-Stock Unstable SLC6A3 26 55 CC[C@@H](C)NC(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217671441 CE For-Sale Unstable TNFRSF1A 23 41 C[C@@H]1N[C@@H](CO)Cc2ccccc21 ZINC000217671448 AD For-Sale Unstable PNMT 20 50 COc1cc(N)c(CC(=O)Nc2cccc(C)c2)cc1OC ZINC000217671465 DF In-Stock Unstable PDGFRB 26 40 COc1cc(N)c(CC(=O)Nc2cccc(C)c2)cc1OC ZINC000217671465 DF In-Stock Unstable KIT 20 42 COc1cc(N)c(CC(=O)Nc2cccc(C)c2)cc1OC ZINC000217671465 DF In-Stock Unstable KDR 19 43 COc1cc(N)c(CC(=O)Nc2cccc(C)c2)cc1OC ZINC000217671465 DF In-Stock Unstable FLT3 19 41 COc1cc(N)c(CC(=O)Nc2cccc(C)c2)cc1OC ZINC000217671465 DF In-Stock Unstable CSF1R 17 42 COc1cc(N)c(CC(=O)Nc2cccc(C)c2)cc1OC ZINC000217671465 DF In-Stock Unstable ENPP1 59 35 COc1cc(N)c(CC(=O)Nc2cccc(C)c2)cc1OC ZINC000217671465 DF In-Stock Unstable PSBA 0 43 COc1cc(N)c(CC(=O)Nc2cccc(C)c2)cc1OC ZINC000217671465 DF In-Stock Unstable KCNK3 68 44 COc1cc(N)c(CC(=O)Nc2cccc(C)c2)cc1OC ZINC000217671465 DF In-Stock Unstable KCNK9 74 44 COC(=O)[C@H](O)CNC(=O)COc1ccc(Cl)c(Cl)c1 ZINC000217671473 DD On-Demand Unstable GRIN1 46 42 Cc1ccccc1-c1ccc(C(=O)N2CCN3CCC[C@H]3C2)cc1 ZINC000217671501 DH In-Stock Unstable AVPR2 26 45 Cc1ccccc1-c1ccc(C(=O)N2CCN3CCC[C@H]3C2)cc1 ZINC000217671501 DH In-Stock Unstable AVPR1A 25 41 Cc1ccccc1-c1ccc(C(=O)N2CCN3CCC[C@H]3C2)cc1 ZINC000217671501 DH In-Stock Unstable INHA 25 49 Cc1ccccc1-c1ccc(C(=O)N2CCN3CCC[C@H]3C2)cc1 ZINC000217671501 DH In-Stock Unstable HRH3 28 52 Cc1ccccc1-c1ccc(C(=O)N2CCN3CCC[C@H]3C2)cc1 ZINC000217671501 DH In-Stock Unstable HSD11B1 15 40 Cc1ccccc1-c1ccc(C(=O)N2CCN3CCC[C@H]3C2)cc1 ZINC000217671501 DH In-Stock Unstable L3MBTL1 0 54 Cc1ccccc1-c1ccc(C(=O)N2CCN3CCC[C@H]3C2)cc1 ZINC000217671501 DH In-Stock Unstable L3MBTL3 104 54 Cc1ccccc1-c1ccc(C(=O)N2CCN3CCC[C@H]3C2)cc1 ZINC000217671501 DH In-Stock Unstable L3MBTL4 0 41 Cc1ccccc1-c1ccc(C(=O)N2CCN3CCC[C@H]3C2)cc1 ZINC000217671501 DH In-Stock Unstable MBTD1 0 45 Cc1ccccc1-c1ccc(C(=O)N2CCN3CCC[C@H]3C2)cc1 ZINC000217671501 DH In-Stock Unstable TP53BP1 0 41 Cc1ccccc1-c1ccc(C(=O)N2CCN3CCC[C@H]3C2)cc1 ZINC000217671501 DH In-Stock Unstable SLC6A7 0 54 Cc1ccc([C@@H]2CN(C)C[C@@H]2CO)cc1 ZINC000217671513 BD In-Stock Unstable SLC6A1 64 55 Cc1ccc([C@@H]2CN(C)C[C@@H]2CO)cc1 ZINC000217671513 BD In-Stock Unstable SLC6A4 21 44 Cc1ccc([C@@H]2CN(C)C[C@@H]2CO)cc1 ZINC000217671513 BD In-Stock Unstable SLC6A3 26 55 Cc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217671516 FK For-Sale Unstable GUAB 0 48 Cc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217671516 FK For-Sale Unstable RAF1 34 47 Cc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217671516 FK For-Sale Unstable Q8MMZ8_EIMTE 55 47 Cc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217671516 FK For-Sale Unstable BRAF 16 42 Cc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217671516 FK For-Sale Unstable PTPA 0 45 Cc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217671516 FK For-Sale Unstable IMDH_CRYPV 40 50 Cc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217671516 FK For-Sale Unstable BLM 0 45 CC[C@H](C)NC(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217671520 CE For-Sale Unstable TNFRSF1A 23 41 O=C(CCSc1ccccc1)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217671523 FH In-Stock Unstable PREP 22 46 O=C(CCSc1ccccc1)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217671523 FH In-Stock Unstable FIMH 19 40 C[C@@H]1N[C@H](CO)Cc2ccccc21 ZINC000217671533 AD For-Sale Unstable PNMT 20 50 COc1cc(N)c(CC(=O)Nc2ccccc2C)cc1OC ZINC000217671576 DF In-Stock Unstable EPHX1 0 40 COc1cc(N)c(CC(=O)Nc2ccccc2C)cc1OC ZINC000217671576 DF In-Stock Unstable MAPK9 0 40 COc1cc(N)c(CC(=O)Nc2ccccc2C)cc1OC ZINC000217671576 DF In-Stock Unstable MAPK10 0 40 COc1cc(N)c(CC(=O)Nc2ccccc2C)cc1OC ZINC000217671576 DF In-Stock Unstable MAPK8 16 40 COc1cc(N)c(CC(=O)Nc2ccccc2C)cc1OC ZINC000217671576 DF In-Stock Unstable DDX3X 0 42 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccn2)c1 ZINC000217671603 CE For-Sale Anodyne HDAC8 27 50 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccn2)c1 ZINC000217671603 CE For-Sale Anodyne GRM5 17 52 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccn2)c1 ZINC000217671603 CE For-Sale Anodyne LUCI_LUCLA 36 43 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccn2)c1 ZINC000217671603 CE For-Sale Anodyne KCNK3 93 45 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccn2)c1 ZINC000217671603 CE For-Sale Anodyne KCNK9 45 38 Cc1ccccc1/C=C/NC(=O)Nc1ccc(N)cc1Cl ZINC000217671633 DI For-Sale Unstable DDX3X 0 42 CC(C)c1ccc([C@@H]2CN(C)C[C@@H]2CO)cc1 ZINC000217671646 BE In-Stock Unstable SLC6A1 51 55 CC(C)c1ccc([C@@H]2CN(C)C[C@@H]2CO)cc1 ZINC000217671646 BE In-Stock Unstable SLC6A4 15 41 CC(C)c1ccc([C@@H]2CN(C)C[C@@H]2CO)cc1 ZINC000217671646 BE In-Stock Unstable SLC6A3 18 55 O=C(c1cccc(C(F)(F)F)c1)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217671647 FH In-Stock Unstable CCR2 42 38 O=C(c1cccc(C(F)(F)F)c1)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217671647 FH In-Stock Unstable ABHD6 0 41 COc1cc(N)c(CC(=O)Nc2ccccc2F)cc1OC ZINC000217671684 DF In-Stock Unstable CA5B 17 41 COc1cc(N)c(CC(=O)Nc2ccccc2F)cc1OC ZINC000217671684 DF In-Stock Unstable CA5A 20 41 COc1cc(N)c(CC(=O)Nc2ccccc2F)cc1OC ZINC000217671684 DF In-Stock Unstable MAPK9 0 40 COc1cc(N)c(CC(=O)Nc2ccccc2F)cc1OC ZINC000217671684 DF In-Stock Unstable MAPK8 15 40 COc1cc(N)c(CC(=O)Nc2ccccc2F)cc1OC ZINC000217671684 DF In-Stock Unstable PDGFRA 15 41 COc1cc(N)c(CC(=O)Nc2ccccc2F)cc1OC ZINC000217671684 DF In-Stock Unstable GLMU 0 43 O=C(O)/C=C\c1ccc(F)c(C(=O)Nc2ccccn2)c1 ZINC000217671685 CF For-Sale Anodyne MMP9 0 40 O=C(O)/C=C\c1ccc(F)c(C(=O)Nc2ccccn2)c1 ZINC000217671685 CF For-Sale Anodyne MMP1 0 40 Cn1nccc1NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217671696 DD For-Sale Unstable HDAC8 36 49 Cn1nccc1NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217671696 DD For-Sale Unstable HDAC1 15 49 Cn1nccc1NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217671696 DD For-Sale Unstable HDAC6 16 49 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(O)cc2)CC(=O)O4)cc1O ZINC000217671704 II In-Stock Unstable AKR1B1 26 50 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(O)cc2)CC(=O)O4)cc1O ZINC000217671704 II In-Stock Unstable CYP1B1 67 37 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(O)cc2)CC(=O)O4)cc1O ZINC000217671704 II In-Stock Unstable CYP1A1 50 52 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(O)cc2)CC(=O)O4)cc1O ZINC000217671704 II In-Stock Unstable CYP1A2 40 48 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(O)cc2)CC(=O)O4)cc1O ZINC000217671704 II In-Stock Unstable ABCG2 0 41 CC(C)c1ccc([C@H]2CN(C)C[C@@H]2CO)cc1 ZINC000217671738 BE In-Stock Unstable SLC6A1 51 55 CC(C)c1ccc([C@H]2CN(C)C[C@@H]2CO)cc1 ZINC000217671738 BE In-Stock Unstable SLC6A4 15 41 CC(C)c1ccc([C@H]2CN(C)C[C@@H]2CO)cc1 ZINC000217671738 BE In-Stock Unstable SLC6A3 18 55 O=C(/C=C/c1ccc2c(c1)OCO2)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217671759 FF In-Stock Unstable DYRK2 42 35 COC(=O)[C@@H](O)CNC(=O)CSc1ccc(C)cc1 ZINC000217671776 CC On-Demand Unstable FAS 47 37 NC(=O)CCCNC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217671780 CC For-Sale Unstable HDAC8 16 44 NC(=O)CCCNC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217671780 CC For-Sale Unstable HDA106 0 43 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(O)cc2)CC(=O)O4)cc1O ZINC000217671781 II In-Stock Unstable AKR1B1 26 50 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(O)cc2)CC(=O)O4)cc1O ZINC000217671781 II In-Stock Unstable CYP1B1 67 37 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(O)cc2)CC(=O)O4)cc1O ZINC000217671781 II In-Stock Unstable CYP1A1 50 52 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(O)cc2)CC(=O)O4)cc1O ZINC000217671781 II In-Stock Unstable CYP1A2 40 48 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(O)cc2)CC(=O)O4)cc1O ZINC000217671781 II In-Stock Unstable ABCG2 0 41 CCN[C@@H]1CC[C@@H](CC)C[C@@H]1Cc1cccc(Cl)c1 ZINC000217671789 CJ For-Sale Unstable CACNA1D 0 41 COc1cc(N)c(CC(=O)Nc2cccc(F)c2)cc1OC ZINC000217671790 DF In-Stock Unstable PDGFRB 27 44 COc1cc(N)c(CC(=O)Nc2cccc(F)c2)cc1OC ZINC000217671790 DF In-Stock Unstable AURKB 30 44 COc1cc(N)c(CC(=O)Nc2cccc(F)c2)cc1OC ZINC000217671790 DF In-Stock Unstable PDGFRA 21 43 COc1cc(N)c(CC(=O)Nc2cccc(F)c2)cc1OC ZINC000217671790 DF In-Stock Unstable FLT3 18 44 COc1cc(N)c(CC(=O)Nc2cccc(F)c2)cc1OC ZINC000217671790 DF In-Stock Unstable CSF1R 19 43 COc1cc(N)c(CC(=O)Nc2cccc(F)c2)cc1OC ZINC000217671790 DF In-Stock Unstable AURKA 27 44 COc1cc(N)c(CC(=O)Nc2cccc(F)c2)cc1OC ZINC000217671790 DF In-Stock Unstable ENPP1 58 37 COc1cc(N)c(CC(=O)Nc2cccc(F)c2)cc1OC ZINC000217671790 DF In-Stock Unstable KCNK3 57 40 COc1cc(N)c(CC(=O)Nc2cccc(F)c2)cc1OC ZINC000217671790 DF In-Stock Unstable KCNK9 53 40 CC(=O)c1ccc(NC(=O)CCN2CCN(Cc3cc(=O)n4ccsc4n3)CC2)cc1 ZINC000217671796 IE On-Demand Unstable CHRNA7 15 43 COC[C@@H](C)NC(=O)CNCCCN1CCCC[C@@H]1C ZINC000217671819 CC For-Sale Unstable HRH3 33 40 COC(=O)[C@H](O)CNC(=O)CSc1ccc(C)cc1 ZINC000217671850 CC On-Demand Unstable FAS 47 37 CN1C[C@@H](CO)[C@H](c2ccc(C(C)(C)C)cc2)C1 ZINC000217671863 BF In-Stock Unstable SLC6A1 31 52 O=C(N1CC(n2cc(-c3ccccc3)nn2)C1)C1(c2ccccc2)CCOCC1 ZINC000217671875 GG In-Stock Unstable PREP 15 40 CCN[C@H]1CC[C@@H](CC)C[C@@H]1Cc1cccc(Cl)c1 ZINC000217671883 CJ For-Sale Unstable CACNA1D 0 41 COc1cc(N)c(CC(=O)Nc2ccc(F)cc2)cc1OC ZINC000217671892 DF In-Stock Unstable KDR 20 41 COc1cc(N)c(CC(=O)Nc2ccc(F)cc2)cc1OC ZINC000217671892 DF In-Stock Unstable CA12 16 40 COc1cc(N)c(CC(=O)Nc2ccc(F)cc2)cc1OC ZINC000217671892 DF In-Stock Unstable PDGFRA 36 41 COc1cc(N)c(CC(=O)Nc2ccc(F)cc2)cc1OC ZINC000217671892 DF In-Stock Unstable CSF1R 18 40 COc1cc(N)c(CC(=O)Nc2ccc(F)cc2)cc1OC ZINC000217671892 DF In-Stock Unstable CA9 15 40 COc1cc(N)c(CC(=O)Nc2ccc(F)cc2)cc1OC ZINC000217671892 DF In-Stock Unstable ENPP1 64 41 COc1cc(N)c(CC(=O)Nc2ccc(F)cc2)cc1OC ZINC000217671892 DF In-Stock Unstable DRTS_TRYCR 53 32 CN1CCN(C(=O)C[C@H](c2ccc(O)cc2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)CC1 ZINC000217671895 KH In-Stock Unstable RORC 42 33 CN1C[C@H](CO)[C@H](c2ccc(C(C)(C)C)cc2)C1 ZINC000217671947 BF In-Stock Unstable SLC6A1 31 52 Cc1ccccc1/C=C/NC(=O)Nc1cccc(Cl)c1 ZINC000217671965 CI For-Sale Unstable PPIA 18 40 Cc1ccccc1/C=C/NC(=O)Nc1cccc(Cl)c1 ZINC000217671965 CI For-Sale Unstable DDX3X 0 41 Cc1ccccc1/C=C/NC(=O)Nc1cccc(Cl)c1 ZINC000217671965 CI For-Sale Unstable IMDH_CRYPV 18 42 Cc1ccccc1/C=C/NC(=O)Nc1cccc(Cl)c1 ZINC000217671965 CI For-Sale Unstable PSBA 0 46 Cc1ccccc1/C=C/NC(=O)Nc1cccc(Cl)c1 ZINC000217671965 CI For-Sale Unstable KCNK3 87 44 Cc1ccccc1/C=C/NC(=O)Nc1cccc(Cl)c1 ZINC000217671965 CI For-Sale Unstable KCNK9 51 44 CCN[C@@H]1CC[C@H](CC)C[C@@H]1Cc1cccc(Cl)c1 ZINC000217671972 CJ For-Sale Unstable CACNA1D 0 41 O=C(CCS(=O)(=O)c1ccccc1)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217671976 GE In-Stock Unstable PREP 23 48 CN1CCN(C(=O)C[C@@H](c2ccc(O)cc2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)CC1 ZINC000217671986 KH In-Stock Unstable RORC 42 33 COc1cc(N)c(CC(=O)Nc2cccc(C(F)(F)F)c2)cc1OC ZINC000217671999 FG In-Stock Unstable KIT 15 46 COc1cc(N)c(CC(=O)Nc2cccc(C(F)(F)F)c2)cc1OC ZINC000217671999 FG In-Stock Unstable KDR 20 41 COc1cc(N)c(CC(=O)Nc2cccc(C(F)(F)F)c2)cc1OC ZINC000217671999 FG In-Stock Unstable SLC1A1 20 40 COc1cc(N)c(CC(=O)Nc2cccc(C(F)(F)F)c2)cc1OC ZINC000217671999 FG In-Stock Unstable SLC1A3 18 40 COc1cc(N)c(CC(=O)Nc2cccc(C(F)(F)F)c2)cc1OC ZINC000217671999 FG In-Stock Unstable FLT4 16 40 COc1cc(N)c(CC(=O)Nc2cccc(C(F)(F)F)c2)cc1OC ZINC000217671999 FG In-Stock Unstable SLC1A2 34 40 COc1cc(N)c(CC(=O)Nc2cccc(C(F)(F)F)c2)cc1OC ZINC000217671999 FG In-Stock Unstable CSF1R 15 46 COc1cc(N)c(CC(=O)Nc2cccc(C(F)(F)F)c2)cc1OC ZINC000217671999 FG In-Stock Unstable PHES 0 43 COc1cc(N)c(CC(=O)Nc2cccc(C(F)(F)F)c2)cc1OC ZINC000217671999 FG In-Stock Unstable ENPP1 55 33 COc1cc(N)c(CC(=O)Nc2cccc(C(F)(F)F)c2)cc1OC ZINC000217671999 FG In-Stock Unstable KCNK3 54 41 COc1cc(N)c(CC(=O)Nc2cccc(C(F)(F)F)c2)cc1OC ZINC000217671999 FG In-Stock Unstable KCNK9 44 40 COc1cc(N)c(CC(=O)Nc2cccc(C(F)(F)F)c2)cc1OC ZINC000217671999 FG In-Stock Unstable PDS 42 37 Cc1ncn(CCNC(=O)CCn2cncn2)c1C ZINC000217672009 CC In-Stock Unstable HIS3 46 33 O=C(CCN1CCN(Cc2cc(=O)n3ccsc3n2)CC1)Nc1cccc(Cl)c1 ZINC000217672034 IF On-Demand Unstable HTR1A 21 43 COC(=O)[C@H](O)CNC(=O)c1ccccc1O ZINC000217672046 BB For-Sale Unstable KCNA3 17 44 CCN[C@H]1CC[C@H](CC)C[C@@H]1Cc1cccc(Cl)c1 ZINC000217672050 CJ For-Sale Unstable CACNA1D 0 41 Cc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)cc1 ZINC000217672076 CI For-Sale Unstable GUAB 0 40 Cc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)cc1 ZINC000217672076 CI For-Sale Unstable P95276_MYCTO 0 41 Cc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)cc1 ZINC000217672076 CI For-Sale Unstable PSBA 0 40 O=C(CCc1cccc(OCc2ccccc2)c1)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217672082 IJ In-Stock Unstable PREP 26 49 O=C(CCc1cccc(OCc2ccccc2)c1)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217672082 IJ In-Stock Unstable FAAH 23 44 O=C(CCc1cccc(OCc2ccccc2)c1)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217672082 IJ In-Stock Unstable FFAR1 47 44 COC(=O)[C@H](CC(C)C)NC(=O)c1cn(C(C)C)c(=O)c2ccccc12 ZINC000217672092 FF In-Stock Unstable CAPNS1 47 36 COC(=O)[C@H](CC(C)C)NC(=O)c1cn(C(C)C)c(=O)c2ccccc12 ZINC000217672092 FF In-Stock Unstable CAPN1 37 40 COC(=O)[C@H](CC(C)C)NC(=O)c1cn(C(C)C)c(=O)c2ccccc12 ZINC000217672092 FF In-Stock Unstable CAPN2 60 34 COC(=O)[C@H](CC(C)C)NC(=O)c1cn(C(C)C)c(=O)c2ccccc12 ZINC000217672092 FF In-Stock Unstable NPR 66 35 COc1cc(N)c(CC(=O)Nc2ccc(Cl)cc2)cc1OC ZINC000217672122 DG In-Stock Unstable HTR2A 21 42 COc1cc(N)c(CC(=O)Nc2ccc(Cl)cc2)cc1OC ZINC000217672122 DG In-Stock Unstable PTGS2 0 43 COc1cc(N)c(CC(=O)Nc2ccc(Cl)cc2)cc1OC ZINC000217672122 DG In-Stock Unstable HTR4 49 35 COc1cc(N)c(CC(=O)Nc2ccc(Cl)cc2)cc1OC ZINC000217672122 DG In-Stock Unstable F10 47 32 COc1cc(N)c(CC(=O)Nc2ccc(Cl)cc2)cc1OC ZINC000217672122 DG In-Stock Unstable CSNK1D 16 41 COc1cc(N)c(CC(=O)Nc2ccc(Cl)cc2)cc1OC ZINC000217672122 DG In-Stock Unstable COLA 46 38 COc1cc(N)c(CC(=O)Nc2ccc(Cl)cc2)cc1OC ZINC000217672122 DG In-Stock Unstable CPT1A 44 31 COc1cc(N)c(CC(=O)Nc2ccc(Cl)cc2)cc1OC ZINC000217672122 DG In-Stock Unstable KDR 21 41 COc1cc(N)c(CC(=O)Nc2ccc(Cl)cc2)cc1OC ZINC000217672122 DG In-Stock Unstable CA12 16 40 COc1cc(N)c(CC(=O)Nc2ccc(Cl)cc2)cc1OC ZINC000217672122 DG In-Stock Unstable PDGFRA 31 41 COc1cc(N)c(CC(=O)Nc2ccc(Cl)cc2)cc1OC ZINC000217672122 DG In-Stock Unstable CSF1R 22 40 COc1cc(N)c(CC(=O)Nc2ccc(Cl)cc2)cc1OC ZINC000217672122 DG In-Stock Unstable CA9 20 40 COc1cc(N)c(CC(=O)Nc2ccc(Cl)cc2)cc1OC ZINC000217672122 DG In-Stock Unstable ENPP1 62 38 COc1cc(N)c(CC(=O)Nc2ccc(Cl)cc2)cc1OC ZINC000217672122 DG In-Stock Unstable DRTS_TRYCR 53 32 O=C(CCN1CCN(Cc2cc(=O)n3ccsc3n2)CC1)Nc1cccc(F)c1 ZINC000217672157 HE On-Demand Unstable CHRNA7 17 41 COc1cc(CN2CCC[C@@H](N)C2)ccc1OCCN1CCCC1 ZINC000217672173 EE In-Stock Unstable ACHE 21 46 COc1cc(CN2CCC[C@@H](N)C2)ccc1OCCN1CCCC1 ZINC000217672173 EE In-Stock Unstable LTA4H 35 41 COc1cc(CN2CCC[C@@H](N)C2)ccc1OCCN1CCCC1 ZINC000217672173 EE In-Stock Unstable HRH3 36 41 COc1cc(CN2CCC[C@@H](N)C2)ccc1OCCN1CCCC1 ZINC000217672173 EE In-Stock Unstable SIGMAR1 15 44 COc1cc(CN2CCC[C@@H](N)C2)ccc1OCCN1CCCC1 ZINC000217672173 EE In-Stock Unstable SSTR5 47 38 COc1cc(CN2CCC[C@@H](N)C2)ccc1OCCN1CCCC1 ZINC000217672173 EE In-Stock Unstable UTS2R 30 43 COc1cc(CN2CCC[C@@H](N)C2)ccc1OCCN1CCCC1 ZINC000217672173 EE In-Stock Unstable MCHR1 22 42 COc1cc(CN2CCC[C@@H](N)C2)ccc1OCCN1CCCC1 ZINC000217672173 EE In-Stock Unstable PSMB2 45 38 COc1cc(CN2CCC[C@@H](N)C2)ccc1OCCN1CCCC1 ZINC000217672173 EE In-Stock Unstable EHMT2 89 40 COc1ccc(CCC(=O)N2CC(n3cc(-c4ccccc4)nn3)C2)cc1Br ZINC000217672181 IH In-Stock Unstable PREP 24 46 CCOC(=O)[C@@H]1C(=O)C2=C(C[C@@H]1c1cccs1)N(c1cccc(C(F)(F)F)c1)C(=O)C[C@@H]2c1cccc([N+](=O)[O-])c1 ZINC000217672205 KK In-Stock Unstable CACNA1C 46 35 CCOC(=O)[C@@H]1C(=O)C2=C(C[C@@H]1c1cccs1)N(c1cccc(C(F)(F)F)c1)C(=O)C[C@@H]2c1cccc([N+](=O)[O-])c1 ZINC000217672205 KK In-Stock Unstable CACNA1D 67 35 COc1cc(N)c(CC(=O)Nc2cccc(Cl)c2)cc1OC ZINC000217672228 DG In-Stock Unstable HTR4 37 41 COc1cc(N)c(CC(=O)Nc2cccc(Cl)c2)cc1OC ZINC000217672228 DG In-Stock Unstable CSNK1D 21 41 COc1cc(N)c(CC(=O)Nc2cccc(Cl)c2)cc1OC ZINC000217672228 DG In-Stock Unstable CPT1A 45 31 COc1cc(N)c(CC(=O)Nc2cccc(Cl)c2)cc1OC ZINC000217672228 DG In-Stock Unstable CSF1R 22 44 COc1cc(N)c(CC(=O)Nc2cccc(Cl)c2)cc1OC ZINC000217672228 DG In-Stock Unstable ENPP1 59 36 COc1cc(N)c(CC(=O)Nc2cccc(Cl)c2)cc1OC ZINC000217672228 DG In-Stock Unstable PSBA 0 45 COc1cc(N)c(CC(=O)Nc2cccc(Cl)c2)cc1OC ZINC000217672228 DG In-Stock Unstable KCNK3 52 40 COc1cc(N)c(CC(=O)Nc2cccc(Cl)c2)cc1OC ZINC000217672228 DG In-Stock Unstable KCNK9 43 40 COc1cc(CN2CCC[C@H](N)C2)ccc1OCCN1CCCC1 ZINC000217672256 EE In-Stock Unstable ACHE 21 46 COc1cc(CN2CCC[C@H](N)C2)ccc1OCCN1CCCC1 ZINC000217672256 EE In-Stock Unstable LTA4H 35 41 COc1cc(CN2CCC[C@H](N)C2)ccc1OCCN1CCCC1 ZINC000217672256 EE In-Stock Unstable HRH3 36 41 COc1cc(CN2CCC[C@H](N)C2)ccc1OCCN1CCCC1 ZINC000217672256 EE In-Stock Unstable SIGMAR1 15 44 COc1cc(CN2CCC[C@H](N)C2)ccc1OCCN1CCCC1 ZINC000217672256 EE In-Stock Unstable SSTR5 47 38 COc1cc(CN2CCC[C@H](N)C2)ccc1OCCN1CCCC1 ZINC000217672256 EE In-Stock Unstable UTS2R 30 43 COc1cc(CN2CCC[C@H](N)C2)ccc1OCCN1CCCC1 ZINC000217672256 EE In-Stock Unstable MCHR1 22 42 COc1cc(CN2CCC[C@H](N)C2)ccc1OCCN1CCCC1 ZINC000217672256 EE In-Stock Unstable PSMB2 45 38 COc1cc(CN2CCC[C@H](N)C2)ccc1OCCN1CCCC1 ZINC000217672256 EE In-Stock Unstable EHMT2 89 40 O=C(CCN1CCN(Cc2cc(=O)n3ccsc3n2)CC1)Nc1cccc2ccccc12 ZINC000217672274 IG On-Demand Unstable PRKDC 72 40 O=C(CCc1ccc(Cl)c(Cl)c1)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217672281 HI In-Stock Unstable PREP 23 48 Cc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccccc2)CC1 ZINC000217672305 EG For-Sale Unstable DRD4 50 40 Cc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccccc2)CC1 ZINC000217672305 EG For-Sale Unstable ACHE 28 42 Cc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccccc2)CC1 ZINC000217672305 EG For-Sale Unstable SIGMAR1 52 43 Cc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccccc2)CC1 ZINC000217672305 EG For-Sale Unstable FAAH 27 49 Cc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccccc2)CC1 ZINC000217672305 EG For-Sale Unstable MGLL 0 43 Cc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccccc2)CC1 ZINC000217672305 EG For-Sale Unstable NPFFR1 45 33 CC[C@@H](N[C@@H]1CCC[C@@H](O)C1)c1ccc(F)cc1 ZINC000217672308 CG For-Sale Unstable SLC6A3 15 43 COc1cc(N)c(CC(=O)Nc2ccccc2Cl)cc1OC ZINC000217672339 DG In-Stock Unstable HTR4 70 41 COc1cc(N)c(CC(=O)Nc2ccccc2Cl)cc1OC ZINC000217672339 DG In-Stock Unstable KCNQ2 39 44 COc1cc(N)c(CC(=O)Nc2ccccc2Cl)cc1OC ZINC000217672339 DG In-Stock Unstable PTGER3 15 41 COc1cc(N)c(CC(=O)Nc2ccccc2Cl)cc1OC ZINC000217672339 DG In-Stock Unstable CA5B 17 41 COc1cc(N)c(CC(=O)Nc2ccccc2Cl)cc1OC ZINC000217672339 DG In-Stock Unstable CA5A 20 41 COc1cc(N)c(CC(=O)Nc2ccccc2Cl)cc1OC ZINC000217672339 DG In-Stock Unstable MAPK9 0 40 COc1cc(N)c(CC(=O)Nc2ccccc2Cl)cc1OC ZINC000217672339 DG In-Stock Unstable MAPK8 15 40 COc1cc(N)c(CC(=O)Nc2ccccc2Cl)cc1OC ZINC000217672339 DG In-Stock Unstable CSF1R 17 42 COc1cc(N)c(CC(=O)Nc2ccccc2Cl)cc1OC ZINC000217672339 DG In-Stock Unstable CA9 16 42 COc1ccc(CCC(=O)N2CC(n3cc(-c4ccccc4)nn3)C2)c(OC)c1 ZINC000217672385 GF In-Stock Unstable PREP 24 46 CCOC(=O)[C@@H]1C(=O)C2=C(C[C@H]1c1cccs1)N(c1cccc(C(F)(F)F)c1)C(=O)C[C@@H]2c1cccc([N+](=O)[O-])c1 ZINC000217672386 KK In-Stock Unstable CACNA1C 46 35 CCOC(=O)[C@@H]1C(=O)C2=C(C[C@H]1c1cccs1)N(c1cccc(C(F)(F)F)c1)C(=O)C[C@@H]2c1cccc([N+](=O)[O-])c1 ZINC000217672386 KK In-Stock Unstable CACNA1D 67 35 CCOC(=O)[C@@H](Nc1ccc(C)c(C)c1)c1ccccc1 ZINC000217672394 CI On-Demand Unstable NPY5R 22 40 CCOC(=O)[C@@H](Nc1ccc(C)c(C)c1)c1ccccc1 ZINC000217672394 CI On-Demand Unstable DHOD 0 41 CC[C@H](N[C@@H]1CCC[C@@H](O)C1)c1ccc(F)cc1 ZINC000217672395 CG On-Demand Unstable SLC6A3 15 43 COc1ccc(NC(=O)Cc2cc(OC)c(OC)cc2N)cc1 ZINC000217672446 DE In-Stock Unstable TSHR 54 33 COc1ccc(NC(=O)Cc2cc(OC)c(OC)cc2N)cc1 ZINC000217672446 DE In-Stock Unstable PDGFRB 45 44 COc1ccc(NC(=O)Cc2cc(OC)c(OC)cc2N)cc1 ZINC000217672446 DE In-Stock Unstable CA1 26 41 COc1ccc(NC(=O)Cc2cc(OC)c(OC)cc2N)cc1 ZINC000217672446 DE In-Stock Unstable MTNR1A 43 43 COc1ccc(NC(=O)Cc2cc(OC)c(OC)cc2N)cc1 ZINC000217672446 DE In-Stock Unstable MTNR1B 39 45 COc1ccc(NC(=O)Cc2cc(OC)c(OC)cc2N)cc1 ZINC000217672446 DE In-Stock Unstable MAPK9 23 46 COc1ccc(NC(=O)Cc2cc(OC)c(OC)cc2N)cc1 ZINC000217672446 DE In-Stock Unstable ACR 42 32 COc1ccc(NC(=O)Cc2cc(OC)c(OC)cc2N)cc1 ZINC000217672446 DE In-Stock Unstable CA12 22 53 COc1ccc(NC(=O)Cc2cc(OC)c(OC)cc2N)cc1 ZINC000217672446 DE In-Stock Unstable MAPK8 19 44 COc1ccc(NC(=O)Cc2cc(OC)c(OC)cc2N)cc1 ZINC000217672446 DE In-Stock Unstable PDGFRA 53 42 COc1ccc(NC(=O)Cc2cc(OC)c(OC)cc2N)cc1 ZINC000217672446 DE In-Stock Unstable FLT3 19 44 COc1ccc(NC(=O)Cc2cc(OC)c(OC)cc2N)cc1 ZINC000217672446 DE In-Stock Unstable CSF1R 23 44 COc1ccc(NC(=O)Cc2cc(OC)c(OC)cc2N)cc1 ZINC000217672446 DE In-Stock Unstable CA9 30 53 COc1ccc(NC(=O)Cc2cc(OC)c(OC)cc2N)cc1 ZINC000217672446 DE In-Stock Unstable ENPP1 65 39 COc1ccc(NC(=O)Cc2cc(OC)c(OC)cc2N)cc1 ZINC000217672446 DE In-Stock Unstable DRTS_TRYCR 53 32 CN1C[C@@H](CO)[C@H](c2cccc(F)c2)C1 ZINC000217672449 BD In-Stock Unstable CCR5 104 40 CCOC(=O)[C@H](Nc1ccc(C)c(C)c1)c1ccccc1 ZINC000217672474 CI On-Demand Unstable NPY5R 22 40 CCOC(=O)[C@H](Nc1ccc(C)c(C)c1)c1ccccc1 ZINC000217672474 CI On-Demand Unstable DHOD 0 41 CC[C@@H](N[C@H]1CCC[C@@H](O)C1)c1ccc(F)cc1 ZINC000217672488 CG For-Sale Unstable SLC6A3 15 43 Cc1ccccc1CCC(=O)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217672509 EG In-Stock Unstable PREP 24 47 CN1C[C@H](CO)[C@H](c2cccc(F)c2)C1 ZINC000217672530 BD In-Stock Unstable CCR5 104 40 CCOc1ccccc1C(=O)NC[C@@H](O)C(=O)OC ZINC000217672538 CC On-Demand Unstable KCNA3 35 48 CCOc1ccccc1C(=O)NC[C@@H](O)C(=O)OC ZINC000217672538 CC On-Demand Unstable HCN1 79 46 CCOc1ccccc1C(=O)NC[C@@H](O)C(=O)OC ZINC000217672538 CC On-Demand Unstable HCN4 67 45 CCOc1ccccc1C(=O)NC[C@@H](O)C(=O)OC ZINC000217672538 CC On-Demand Unstable KCNK3 63 51 CCOc1ccccc1C(=O)NC[C@@H](O)C(=O)OC ZINC000217672538 CC On-Demand Unstable KCNK9 48 51 COc1cccc(NC(=O)Cc2cc(OC)c(OC)cc2N)c1 ZINC000217672561 DE In-Stock Unstable PDGFRB 44 52 COc1cccc(NC(=O)Cc2cc(OC)c(OC)cc2N)c1 ZINC000217672561 DE In-Stock Unstable TRPV1 0 43 COc1cccc(NC(=O)Cc2cc(OC)c(OC)cc2N)c1 ZINC000217672561 DE In-Stock Unstable MTNR1A 40 51 COc1cccc(NC(=O)Cc2cc(OC)c(OC)cc2N)c1 ZINC000217672561 DE In-Stock Unstable MTNR1B 40 51 COc1cccc(NC(=O)Cc2cc(OC)c(OC)cc2N)c1 ZINC000217672561 DE In-Stock Unstable MAPK9 15 41 COc1cccc(NC(=O)Cc2cc(OC)c(OC)cc2N)c1 ZINC000217672561 DE In-Stock Unstable FLT4 23 52 COc1cccc(NC(=O)Cc2cc(OC)c(OC)cc2N)c1 ZINC000217672561 DE In-Stock Unstable ACR 19 40 COc1cccc(NC(=O)Cc2cc(OC)c(OC)cc2N)c1 ZINC000217672561 DE In-Stock Unstable MAPK8 19 41 COc1cccc(NC(=O)Cc2cc(OC)c(OC)cc2N)c1 ZINC000217672561 DE In-Stock Unstable PDGFRA 21 43 COc1cccc(NC(=O)Cc2cc(OC)c(OC)cc2N)c1 ZINC000217672561 DE In-Stock Unstable FLT3 19 52 COc1cccc(NC(=O)Cc2cc(OC)c(OC)cc2N)c1 ZINC000217672561 DE In-Stock Unstable CSF1R 24 44 COc1cccc(NC(=O)Cc2cc(OC)c(OC)cc2N)c1 ZINC000217672561 DE In-Stock Unstable ENPP1 59 35 COc1cccc(NC(=O)Cc2cc(OC)c(OC)cc2N)c1 ZINC000217672561 DE In-Stock Unstable PSBA 0 50 COc1cccc(NC(=O)Cc2cc(OC)c(OC)cc2N)c1 ZINC000217672561 DE In-Stock Unstable KCNK3 60 44 COc1cccc(NC(=O)Cc2cc(OC)c(OC)cc2N)c1 ZINC000217672561 DE In-Stock Unstable KCNK9 54 44 CN(Cc1ccoc1)C(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217672571 CF For-Sale Unstable HSD17B2 23 42 CC[C@H](N[C@H]1CCC[C@@H](O)C1)c1ccc(F)cc1 ZINC000217672575 CG On-Demand Unstable SLC6A3 15 43 CCOc1ccccc1C(=O)NC[C@H](O)C(=O)OC ZINC000217672615 CC On-Demand Unstable KCNA3 35 48 CCOc1ccccc1C(=O)NC[C@H](O)C(=O)OC ZINC000217672615 CC On-Demand Unstable HCN1 79 46 CCOc1ccccc1C(=O)NC[C@H](O)C(=O)OC ZINC000217672615 CC On-Demand Unstable HCN4 67 45 CCOc1ccccc1C(=O)NC[C@H](O)C(=O)OC ZINC000217672615 CC On-Demand Unstable KCNK3 63 51 CCOc1ccccc1C(=O)NC[C@H](O)C(=O)OC ZINC000217672615 CC On-Demand Unstable KCNK9 48 51 O=C(CCc1ccc(Cl)c(F)c1)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217672619 GH In-Stock Unstable PREP 22 45 Cc1ccccc1/C=C/NC(=O)NC1CCCCCCCCCCC1 ZINC000217672621 EK For-Sale Unstable FAAH 15 40 Cc1ccccc1/C=C/NC(=O)NC1CCCCCCCCCCC1 ZINC000217672621 EK For-Sale Unstable EPHX2 29 48 CN1C[C@@H](CO)[C@H](c2ccccc2Cl)C1 ZINC000217672641 BD In-Stock Unstable SLC6A1 35 49 COc1ccccc1NC(=O)Cc1cc(OC)c(OC)cc1N ZINC000217672672 DE In-Stock Unstable CSNK1D 15 40 COc1ccccc1NC(=O)Cc1cc(OC)c(OC)cc1N ZINC000217672672 DE In-Stock Unstable MAPK9 0 44 COc1ccccc1NC(=O)Cc1cc(OC)c(OC)cc1N ZINC000217672672 DE In-Stock Unstable MAPK10 0 41 COc1ccccc1NC(=O)Cc1cc(OC)c(OC)cc1N ZINC000217672672 DE In-Stock Unstable MAPK8 17 44 FC(F)(F)C1CCN(c2ccc(CBr)cc2)CC1 ZINC000217672680 DI For-Sale Unstable L3MBTL3 38 41 COc1cccc(N2C[C@H](C(=O)NC[C@@H]3CCCN4CCCC[C@H]34)CC2=O)c1 ZINC000217672699 GE In-Stock Unstable DRD4 42 32 O=C(CCN1CCN(Cc2cc(=O)n3ccsc3n2)CC1)NCc1ccccc1Cl ZINC000217672709 IE On-Demand Unstable HTR1A 18 41 O=C(CCN1CCN(Cc2cc(=O)n3ccsc3n2)CC1)NCc1ccccc1Cl ZINC000217672709 IE On-Demand Unstable HTR2A 16 41 O=C(CCN1CCN(Cc2cc(=O)n3ccsc3n2)CC1)NCc1ccccc1Cl ZINC000217672709 IE On-Demand Unstable HTR7 43 41 Cn1ncc2c(=O)n(C[C@@H](C(=O)O)C(F)(F)F)nnc21 ZINC000217672712 CB For-Sale Unstable Q9M629_MAIZE 62 39 CN1C[C@H](CO)[C@H](c2ccccc2Cl)C1 ZINC000217672733 BD In-Stock Unstable SLC6A1 35 49 S=C=Nc1ccc2occc2c1 ZINC000217672734 AG For-Sale Reactive CYP2A6 16 46 Cc1ccccc1/C=C/NC(=O)NCCN1CCOCC1 ZINC000217672745 CD For-Sale Unstable CNR1 22 44 Cc1ccccc1/C=C/NC(=O)NCCN1CCOCC1 ZINC000217672745 CD For-Sale Unstable DRD4 43 34 Cc1ccccc1/C=C/NC(=O)NCCN1CCOCC1 ZINC000217672745 CD For-Sale Unstable CASR 43 36 Cc1ccccc1/C=C/NC(=O)NCCN1CCOCC1 ZINC000217672745 CD For-Sale Unstable PTGDS 44 38 Cc1ccccc1/C=C/NC(=O)NCCN1CCOCC1 ZINC000217672745 CD For-Sale Unstable EPHX2 18 47 Cc1ccccc1/C=C/NC(=O)NCCN1CCOCC1 ZINC000217672745 CD For-Sale Unstable HPGDS 24 42 COc1cccc(N2C[C@@H](C(=O)NC[C@@H]3CCCN4CCCC[C@H]34)CC2=O)c1 ZINC000217672777 GE In-Stock Unstable DRD4 42 32 COc1ccc(NC(=O)Cc2cc(OC)c(OC)cc2N)cc1OC ZINC000217672782 EE In-Stock Unstable TRPV1 0 42 COc1ccc(NC(=O)Cc2cc(OC)c(OC)cc2N)cc1OC ZINC000217672782 EE In-Stock Unstable MAPK9 0 41 COc1ccc(NC(=O)Cc2cc(OC)c(OC)cc2N)cc1OC ZINC000217672782 EE In-Stock Unstable IMPDH2 0 42 COc1ccc(NC(=O)Cc2cc(OC)c(OC)cc2N)cc1OC ZINC000217672782 EE In-Stock Unstable ENPP1 78 47 COc1ccc(NC(=O)Cc2cc(OC)c(OC)cc2N)cc1OC ZINC000217672782 EE In-Stock Unstable IMDH_CRYPV 16 40 COc1ccc(NC(=O)Cc2cc(OC)c(OC)cc2N)cc1OC ZINC000217672782 EE In-Stock Unstable DRTS_TRYCR 60 38 Cn1ncc2c(=O)n(C[C@H](C(=O)O)C(F)(F)F)nnc21 ZINC000217672799 CB For-Sale Unstable Q9M629_MAIZE 62 39 COc1ccc(S(=O)(=O)N2CCCC2)cc1/C=C\C(=O)O ZINC000217672838 DD For-Sale Unstable PKM 23 40 COc1ccc(S(=O)(=O)N2CCCC2)cc1/C=C\C(=O)O ZINC000217672838 DD For-Sale Unstable AKR1C3 54 44 CSC[C@@](C)(O)CNC(=O)CNC(=O)Nc1ccccc1 ZINC000217672851 DD On-Demand Unstable F7 27 42 CN1C[C@@H](CO)[C@H](c2cccc(Cl)c2)C1 ZINC000217672861 BD In-Stock Unstable SLC6A1 46 52 CN1C[C@@H](CO)[C@H](c2cccc(Cl)c2)C1 ZINC000217672861 BD In-Stock Unstable SLC6A4 18 49 CN1C[C@@H](CO)[C@H](c2cccc(Cl)c2)C1 ZINC000217672861 BD In-Stock Unstable SLC6A3 21 52 CN1C[C@@H](CO)[C@H](c2cccc(Cl)c2)C1 ZINC000217672861 BD In-Stock Unstable HSD17B2 0 41 CN1C[C@@H](CO)[C@H](c2cccc(Cl)c2)C1 ZINC000217672861 BD In-Stock Unstable MDM2 74 34 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(C(=O)O)cc2)CC(=O)O4)cc1O ZINC000217672873 JI In-Stock Unstable AKR1B1 0 47 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(C(=O)O)cc2)CC(=O)O4)cc1O ZINC000217672873 JI In-Stock Unstable CYP1B1 56 36 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(C(=O)O)cc2)CC(=O)O4)cc1O ZINC000217672873 JI In-Stock Unstable CYP1A1 43 47 COc1cc(N)c(CC(=O)Nc2ccc(C)c(C)c2)cc1OC ZINC000217672884 DG In-Stock Unstable ENPP1 65 38 O=C(O)/C=C\c1ccc(S(=O)(=O)N2CCCC2)c(Cl)c1 ZINC000217672927 DE For-Sale Unstable EPHX2 16 41 Cc1nc(C=O)nc2ccc(Br)cc12 ZINC000217672928 CF For-Sale Unstable PRS 40 39 CSC[C@](C)(O)CNC(=O)CNC(=O)Nc1ccccc1 ZINC000217672929 DD On-Demand Unstable F7 27 42 CN1C[C@H](CO)[C@H](c2cccc(Cl)c2)C1 ZINC000217672934 BD In-Stock Unstable SLC6A1 46 52 CN1C[C@H](CO)[C@H](c2cccc(Cl)c2)C1 ZINC000217672934 BD In-Stock Unstable SLC6A4 18 49 CN1C[C@H](CO)[C@H](c2cccc(Cl)c2)C1 ZINC000217672934 BD In-Stock Unstable SLC6A3 21 52 CN1C[C@H](CO)[C@H](c2cccc(Cl)c2)C1 ZINC000217672934 BD In-Stock Unstable HSD17B2 0 41 CN1C[C@H](CO)[C@H](c2cccc(Cl)c2)C1 ZINC000217672934 BD In-Stock Unstable MDM2 74 34 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(C(=O)O)cc2)CC(=O)O4)cc1O ZINC000217672950 JI In-Stock Unstable AKR1B1 0 47 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(C(=O)O)cc2)CC(=O)O4)cc1O ZINC000217672950 JI In-Stock Unstable CYP1B1 56 36 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(C(=O)O)cc2)CC(=O)O4)cc1O ZINC000217672950 JI In-Stock Unstable CYP1A1 43 47 COC(=O)[C@@H](O)CNC(=O)COc1ccc(Cl)cc1 ZINC000217672953 CC On-Demand Unstable TRAR 21 42 CC(=O)Nc1ccc(CC(=O)N2CC(n3cc(-c4ccccc4)nn3)C2)cc1 ZINC000217672985 GF In-Stock Unstable PREP 23 44 O=C(O)c1cnc(NCCN2CCOCC2)[nH]c1=O ZINC000217673000 CB In-Stock Unstable STAT6 47 32 COC(=O)[C@H](O)CNC(=O)COc1ccc(Cl)cc1 ZINC000217673043 CC On-Demand Unstable TRAR 21 42 CN1C[C@@H](CO)[C@H](c2ccc(Cl)cc2)C1 ZINC000217673053 BD In-Stock Unstable SLC6A1 105 75 CN1C[C@@H](CO)[C@H](c2ccc(Cl)cc2)C1 ZINC000217673053 BD In-Stock Unstable SLC6A4 27 56 CN1C[C@@H](CO)[C@H](c2ccc(Cl)cc2)C1 ZINC000217673053 BD In-Stock Unstable SLC6A3 32 75 CN1C[C@@H](CO)[C@H](c2ccc(Cl)cc2)C1 ZINC000217673053 BD In-Stock Unstable CHRNA9 0 41 Cc1ccccc1/C=C/NC(=O)NCCN1CCNCC1 ZINC000217673087 CD For-Sale Unstable DRD4 41 32 COCCNS(=O)(=O)c1ccc(/C=C\C(=O)O)cc1Cl ZINC000217673093 DD For-Sale Unstable PTGDR2 15 40 CN1C[C@H](CO)[C@H](c2ccc(Cl)cc2)C1 ZINC000217673152 BD In-Stock Unstable SLC6A1 105 75 CN1C[C@H](CO)[C@H](c2ccc(Cl)cc2)C1 ZINC000217673152 BD In-Stock Unstable SLC6A4 27 56 CN1C[C@H](CO)[C@H](c2ccc(Cl)cc2)C1 ZINC000217673152 BD In-Stock Unstable SLC6A3 32 75 CN1C[C@H](CO)[C@H](c2ccc(Cl)cc2)C1 ZINC000217673152 BD In-Stock Unstable CHRNA9 0 41 Cc1ccc(CNC(=O)N/C=C/c2ccccc2C)cc1 ZINC000217673194 CH For-Sale Unstable ANPEP 15 42 O=C(c1cnn(-c2ccccc2)n1)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217673207 FE In-Stock Unstable PREP 15 42 O=C(O)c1cnc(NCCCn2ccnc2)[nH]c1=O ZINC000217673227 CC In-Stock Unstable TBXAS1 48 42 C[C@@H]1CCCN([C@H](C)C(=O)Nc2ccc(C#N)cc2)C1 ZINC000217673236 CF In-Stock Unstable DHODH 25 40 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)NCCc3c[nH]cn3)[C@H]21 ZINC000217673248 JE In-Stock Unstable HRH3 28 42 COc1ccc(S(=O)(=O)NCC(N)=O)cc1/C=C\C(=O)O ZINC000217673267 DB For-Sale Unstable PTGDR2 16 40 O=C(c1ccccc1Br)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217673302 GG In-Stock Unstable PREP 15 43 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)NCCc3c[nH]cn3)[C@@H]21 ZINC000217673334 JE In-Stock Unstable HRH3 28 42 CCCCOc1ccc(C(=O)NC[C@@H](O)C(=O)OC)cc1 ZINC000217673354 CD On-Demand Unstable THRA 30 40 CCCCOc1ccc(C(=O)NC[C@@H](O)C(=O)OC)cc1 ZINC000217673354 CD On-Demand Unstable KCNQ1 0 53 CCCCOc1ccc(C(=O)NC[C@@H](O)C(=O)OC)cc1 ZINC000217673354 CD On-Demand Unstable SLC2A1 0 47 CCCCOc1ccc(C(=O)NC[C@@H](O)C(=O)OC)cc1 ZINC000217673354 CD On-Demand Unstable PLA2G4B 88 46 CCCCOc1ccc(C(=O)NC[C@@H](O)C(=O)OC)cc1 ZINC000217673354 CD On-Demand Unstable LMGT2 0 47 CC(=O)NCC(=O)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217673422 CC In-Stock Unstable PREP 29 45 CCCCOc1ccc(C(=O)NC[C@H](O)C(=O)OC)cc1 ZINC000217673433 CD On-Demand Unstable KCNQ1 0 53 Cc1ccccc1/C=C/NC(=O)NCCCN1CCOCC1 ZINC000217673436 DD For-Sale Unstable HTR1A 20 40 Cc1ccccc1/C=C/NC(=O)NCCCN1CCOCC1 ZINC000217673436 DD For-Sale Unstable CNR1 0 43 Cc1ccccc1/C=C/NC(=O)NCCCN1CCOCC1 ZINC000217673436 DD For-Sale Unstable ADRA1D 18 41 Cc1ccccc1/C=C/NC(=O)NCCCN1CCOCC1 ZINC000217673436 DD For-Sale Unstable ADRA1A 30 41 Cc1ccccc1/C=C/NC(=O)NCCCN1CCOCC1 ZINC000217673436 DD For-Sale Unstable ADRA1B 18 41 Cc1ccccc1/C=C/NC(=O)NCCCN1CCOCC1 ZINC000217673436 DD For-Sale Unstable DRD3 44 39 Cc1ccccc1/C=C/NC(=O)NCCCN1CCOCC1 ZINC000217673436 DD For-Sale Unstable CASR 40 36 Cc1ccccc1/C=C/NC(=O)NCCCN1CCOCC1 ZINC000217673436 DD For-Sale Unstable TACR2 29 42 Cc1ccccc1/C=C/NC(=O)NCCCN1CCOCC1 ZINC000217673436 DD For-Sale Unstable EPHX2 22 44 COc1ccccc1[C@@H]1CN(C)C[C@@H]1CO ZINC000217673467 BD In-Stock Unstable HTR1A 17 43 COc1ccccc1[C@@H]1CN(C)C[C@@H]1CO ZINC000217673467 BD In-Stock Unstable ADRA1B 41 35 O=C(Cc1cccnc1)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217673540 DD In-Stock Unstable PREP 26 49 COC(=O)[C@@H](O)CNC(=O)CCc1ccc(OC)cc1 ZINC000217673542 CC On-Demand Unstable BMP1 51 44 COC(=O)[C@@H](O)CNC(=O)CCc1ccc(OC)cc1 ZINC000217673542 CC On-Demand Unstable MTNR1A 49 43 COC(=O)[C@@H](O)CNC(=O)CCc1ccc(OC)cc1 ZINC000217673542 CC On-Demand Unstable MMP12 22 48 COC(=O)[C@@H](O)CNC(=O)CCc1ccc(OC)cc1 ZINC000217673542 CC On-Demand Unstable MMP1 34 40 COC(=O)[C@@H](O)CNC(=O)CCc1ccc(OC)cc1 ZINC000217673542 CC On-Demand Unstable PPO2 24 42 COc1ccccc1[C@H]1CN(C)C[C@@H]1CO ZINC000217673545 BD In-Stock Unstable HTR1A 17 43 COc1ccccc1[C@H]1CN(C)C[C@@H]1CO ZINC000217673545 BD In-Stock Unstable ADRA1B 41 35 COC(=O)[C@H](O)CNC(=O)CCc1ccc(OC)cc1 ZINC000217673609 CC On-Demand Unstable ADRB3 16 40 COC(=O)[C@H](O)CNC(=O)CCc1ccc(OC)cc1 ZINC000217673609 CC On-Demand Unstable BMP1 51 44 COC(=O)[C@H](O)CNC(=O)CCc1ccc(OC)cc1 ZINC000217673609 CC On-Demand Unstable MMP13 20 48 COC(=O)[C@H](O)CNC(=O)CCc1ccc(OC)cc1 ZINC000217673609 CC On-Demand Unstable MTNR1A 49 43 COC(=O)[C@H](O)CNC(=O)CCc1ccc(OC)cc1 ZINC000217673609 CC On-Demand Unstable MMP8 18 48 COC(=O)[C@H](O)CNC(=O)CCc1ccc(OC)cc1 ZINC000217673609 CC On-Demand Unstable MMP12 22 48 COC(=O)[C@H](O)CNC(=O)CCc1ccc(OC)cc1 ZINC000217673609 CC On-Demand Unstable CA9 18 45 COC(=O)[C@H](O)CNC(=O)CCc1ccc(OC)cc1 ZINC000217673609 CC On-Demand Unstable MMP1 34 40 COC(=O)[C@H](O)CNC(=O)CCc1ccc(OC)cc1 ZINC000217673609 CC On-Demand Unstable AOC3 15 40 COC(=O)[C@H](O)CNC(=O)CCc1ccc(OC)cc1 ZINC000217673609 CC On-Demand Unstable PPO2 24 42 Cc1ccccc1/C=C/NC(=O)N(C)Cc1ccccc1 ZINC000217673638 CH For-Sale Unstable LIMK2 23 41 O=C(Cc1ccsc1)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217673640 DF In-Stock Unstable PREP 24 46 COc1cccc([C@@H]2CN(C)C[C@@H]2CO)c1 ZINC000217673654 BD In-Stock Unstable DRD4 42 32 COc1cccc([C@@H]2CN(C)C[C@@H]2CO)c1 ZINC000217673654 BD In-Stock Unstable SLC6A1 0 42 CN1C(=O)[C@@H]2CC[C@H]1CN(C(=O)CN1CCc3ccccc3C1)C2 ZINC000217673655 ED In-Stock Unstable CHRNA6 0 40 CN1C(=O)[C@@H]2CC[C@H]1CN(C(=O)CN1CCc3ccccc3C1)C2 ZINC000217673655 ED In-Stock Unstable NOD2 40 33 CN(C)C(=O)CNS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217673661 DC For-Sale Unstable AKR1C3 24 40 COc1cccc([C@H]2CN(C)C[C@@H]2CO)c1 ZINC000217673736 BD In-Stock Unstable DRD4 42 32 COc1cccc([C@H]2CN(C)C[C@@H]2CO)c1 ZINC000217673736 BD In-Stock Unstable SLC6A1 0 42 C[C@@H]1C[C@@H](C)CN([C@H](C)C(=O)Nc2ccc(C#N)cc2)C1 ZINC000217673783 CF In-Stock Unstable DHODH 25 41 CSC[C@@](C)(O)CNC(=O)c1sc(-c2cccs2)nc1C ZINC000217673811 EG On-Demand Unstable SCD1 23 40 Clc1cc2nc(-c3ccc(-c4ccccc4)cc3)c(Cl)cc2[nH]1 ZINC000217673849 EK For-Sale Anodyne PRCP 17 40 Clc1cc2nc(-c3ccc(-c4ccccc4)cc3)c(Cl)cc2[nH]1 ZINC000217673849 EK For-Sale Anodyne NR2E3 43 32 COc1ccc([C@@H]2CN(C)C[C@@H]2CO)cc1 ZINC000217673860 BD In-Stock Unstable SLC6A1 68 51 COc1ccc([C@@H]2CN(C)C[C@@H]2CO)cc1 ZINC000217673860 BD In-Stock Unstable SLC6A4 17 41 COc1ccc([C@@H]2CN(C)C[C@@H]2CO)cc1 ZINC000217673860 BD In-Stock Unstable SLC6A3 24 51 COc1ccc([C@@H]2CN(C)C[C@@H]2CO)cc1 ZINC000217673860 BD In-Stock Unstable CACNA1S 47 36 Cc1csc(NC(=O)N/C=C/c2ccccc2C)n1 ZINC000217673877 CH For-Sale Unstable ROCK1 17 40 Cc1csc(NC(=O)N/C=C/c2ccccc2C)n1 ZINC000217673877 CH For-Sale Unstable GCK 18 47 COCCC[C@@H]1CCCCN1C(=O)C(=O)c1ccco1 ZINC000217673898 CE In-Stock Unstable FKBP1A 47 36 CSC[C@](C)(O)CNC(=O)c1sc(-c2cccs2)nc1C ZINC000217673901 EG On-Demand Unstable SCD1 23 40 COC(=O)[C@@H](O)CNC(=O)c1ccc(OCC(N)=O)cc1 ZINC000217673906 CA On-Demand Unstable PLA2G4B 41 35 COC(=O)[C@@H](O)CNC(=O)c1ccc(OCC(N)=O)cc1 ZINC000217673906 CA On-Demand Unstable ACR 48 33 COc1ccc([C@H]2CN(C)C[C@@H]2CO)cc1 ZINC000217673951 BD In-Stock Unstable SLC6A1 68 51 COc1ccc([C@H]2CN(C)C[C@@H]2CO)cc1 ZINC000217673951 BD In-Stock Unstable SLC6A4 17 41 COc1ccc([C@H]2CN(C)C[C@@H]2CO)cc1 ZINC000217673951 BD In-Stock Unstable SLC6A3 24 51 COc1ccc([C@H]2CN(C)C[C@@H]2CO)cc1 ZINC000217673951 BD In-Stock Unstable CACNA1S 47 36 CCOC(=O)[C@@H](NCc1ccncc1)c1ccccc1 ZINC000217673957 CE On-Demand Unstable CAPN2 23 41 COCCC[C@H]1CCCCN1C(=O)C(=O)c1ccco1 ZINC000217673986 CE In-Stock Unstable FKBP1A 47 36 COC(=O)[C@H](O)CNC(=O)c1ccc(OCC(N)=O)cc1 ZINC000217673991 CA On-Demand Unstable PLA2G4B 41 35 COC(=O)[C@H](O)CNC(=O)c1ccc(OCC(N)=O)cc1 ZINC000217673991 CA On-Demand Unstable ACR 48 33 COc1ccc(C(=O)N(C)C2CC2)cc1/C=C\C(=O)O ZINC000217674020 CE For-Sale Unstable ACKR3 41 34 COCCn1cnc2c1c(=O)n(CCC(=O)Nc1cccc(F)c1)c(=O)n2Cc1ccccc1 ZINC000217674046 JE On-Demand Unstable ADORA2B 27 42 CN1C[C@@H](CO)[C@H](c2ccc3c(c2)OCO3)C1 ZINC000217674065 BD In-Stock Unstable EDNRB 59 38 CN1C[C@@H](CO)[C@H](c2ccc3c(c2)OCO3)C1 ZINC000217674065 BD In-Stock Unstable EDNRA 64 41 CN1C[C@@H](CO)[C@H](c2ccc3c(c2)OCO3)C1 ZINC000217674065 BD In-Stock Unstable SCN9A 0 40 CN1C[C@@H](CO)[C@H](c2ccc3c(c2)OCO3)C1 ZINC000217674065 BD In-Stock Unstable PDE11A 42 32 CN1C[C@@H](CO)[C@H](c2ccc3c(c2)OCO3)C1 ZINC000217674065 BD In-Stock Unstable DYRK2 53 35 COc1cccc(NC(=O)N/C=C/c2ccccc2C)c1 ZINC000217674126 CH For-Sale Unstable MTNR1A 25 46 COc1cccc(NC(=O)N/C=C/c2ccccc2C)c1 ZINC000217674126 CH For-Sale Unstable MTNR1B 30 46 COc1cccc(NC(=O)N/C=C/c2ccccc2C)c1 ZINC000217674126 CH For-Sale Unstable TAAR1 32 43 COc1cccc(NC(=O)N/C=C/c2ccccc2C)c1 ZINC000217674126 CH For-Sale Unstable AKR1C3 18 42 COc1cccc(NC(=O)N/C=C/c2ccccc2C)c1 ZINC000217674126 CH For-Sale Unstable KCNK3 95 48 COc1cccc(NC(=O)N/C=C/c2ccccc2C)c1 ZINC000217674126 CH For-Sale Unstable KCNK9 66 39 CN1C[C@H](CO)[C@H](c2ccc3c(c2)OCO3)C1 ZINC000217674139 BD In-Stock Unstable EDNRB 59 38 CN1C[C@H](CO)[C@H](c2ccc3c(c2)OCO3)C1 ZINC000217674139 BD In-Stock Unstable EDNRA 64 41 CN1C[C@H](CO)[C@H](c2ccc3c(c2)OCO3)C1 ZINC000217674139 BD In-Stock Unstable SCN9A 0 40 CN1C[C@H](CO)[C@H](c2ccc3c(c2)OCO3)C1 ZINC000217674139 BD In-Stock Unstable PDE11A 42 32 CN1C[C@H](CO)[C@H](c2ccc3c(c2)OCO3)C1 ZINC000217674139 BD In-Stock Unstable DYRK2 53 35 COc1ccc2ncc(C(=O)NCCc3c[nH]cn3)c(O)c2c1 ZINC000217674208 DD In-Stock Unstable HRH3 55 44 COc1ccc2ncc(C(=O)NCCc3c[nH]cn3)c(O)c2c1 ZINC000217674208 DD In-Stock Unstable HRH4 21 43 COc1ccc2ncc(C(=O)NCCc3c[nH]cn3)c(O)c2c1 ZINC000217674208 DD In-Stock Unstable MTNR1A 59 44 COc1ccc2ncc(C(=O)NCCc3c[nH]cn3)c(O)c2c1 ZINC000217674208 DD In-Stock Unstable MTNR1B 48 43 CSC[C@@](C)(O)CNC(=O)c1ccc2c(c1)CCC(=O)N2 ZINC000217674228 DD On-Demand Unstable HDAC9 21 52 COc1ccc([C@@H]2CN(C)C[C@@H]2CO)cc1OC ZINC000217674245 CD In-Stock Unstable SLC6A1 26 45 Cc1ccccc1/C=C/NC(=O)Nc1cc(Cl)ccc1O ZINC000217674250 DI For-Sale Unstable KCNMA1 32 48 O=C(O)c1cnc(N2CCC(Cc3ccccc3)CC2)[nH]c1=O ZINC000217674284 DD In-Stock Unstable GRIN2B 77 42 O=C(O)c1cnc(N2CCC(Cc3ccccc3)CC2)[nH]c1=O ZINC000217674284 DD In-Stock Unstable SIGMAR1 16 40 O=C(O)c1cnc(N2CCC(Cc3ccccc3)CC2)[nH]c1=O ZINC000217674284 DD In-Stock Unstable CCR3 39 40 O=C(O)c1cnc(N2CCC(Cc3ccccc3)CC2)[nH]c1=O ZINC000217674284 DD In-Stock Unstable BRS3 23 42 O=C(O)c1cnc(N2CCC(Cc3ccccc3)CC2)[nH]c1=O ZINC000217674284 DD In-Stock Unstable GRIN3A 0 43 Cc1cccc(NC(=O)c2ccc(/C=C\C(=O)O)s2)c1 ZINC000217674285 CG For-Sale Unstable CCKAR 19 41 Cc1cccc(NC(=O)c2ccc(/C=C\C(=O)O)s2)c1 ZINC000217674285 CG For-Sale Unstable KCNK3 119 47 Cc1cccc(NC(=O)c2ccc(/C=C\C(=O)O)s2)c1 ZINC000217674285 CG For-Sale Unstable KCNK9 80 47 O=S(=O)(c1ccc(F)c(Cl)c1)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217674310 GF In-Stock Unstable CA5B 17 40 O=S(=O)(c1ccc(F)c(Cl)c1)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217674310 GF In-Stock Unstable CA5A 17 40 CSC[C@](C)(O)CNC(=O)c1ccc2c(c1)CCC(=O)N2 ZINC000217674320 DD On-Demand Unstable HDAC9 21 52 c1ccc2c(c1)CCCC[C@H]2N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217674342 CH For-Sale Unstable SLC18A3 55 36 c1ccc2c(c1)CCCC[C@H]2N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217674342 CH For-Sale Unstable KCNN3 15 44 COc1ccc(C(=O)N2CCOCC2)cc1/C=C\C(=O)O ZINC000217674349 CD For-Sale Unstable ITGAL 44 43 COc1ccc(C(=O)N2CCOCC2)cc1/C=C\C(=O)O ZINC000217674349 CD For-Sale Unstable AKR1C3 0 40 COc1ccc(C(=O)N2CCOCC2)cc1/C=C\C(=O)O ZINC000217674349 CD For-Sale Unstable LRRK2 31 45 O=C(O)c1cnc(NCc2cccnc2)[nH]c1=O ZINC000217674400 BC In-Stock Unstable NAMPT 44 42 O=S(=O)(c1ccc2c(c1)OCCO2)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217674424 GD In-Stock Unstable PKM 39 53 CCOC(=O)[C@@H](N[C@@H](CC)CO)c1ccccc1 ZINC000217674429 CD On-Demand Unstable CAPN2 29 42 CCOC(=O)[C@@H](N[C@@H](CC)CO)c1ccccc1 ZINC000217674429 CD On-Demand Unstable COL4A3BP 0 41 O=C(O)/C=C\c1ccc(C(=O)Nc2ccccn2)c(F)c1 ZINC000217674438 CF For-Sale Anodyne MMP9 0 40 O=C(O)/C=C\c1ccc(C(=O)Nc2ccccn2)c(F)c1 ZINC000217674438 CF For-Sale Anodyne MMP1 0 40 Cc1ccccc1/C=C/NC(=O)Nc1nccs1 ZINC000217674450 CG For-Sale Unstable MAP 0 46 Cc1ccccc1/C=C/NC(=O)Nc1nccs1 ZINC000217674450 CG For-Sale Unstable MAP1 123 39 CCOC(=O)[C@H](N[C@@H](CC)CO)c1ccccc1 ZINC000217674513 CD On-Demand Unstable CAPN2 29 42 CCOC(=O)[C@H](N[C@@H](CC)CO)c1ccccc1 ZINC000217674513 CD On-Demand Unstable COL4A3BP 0 41 COc1ccc(CCNc2ncc(C(=O)O)c(=O)[nH]2)cc1OC ZINC000217674517 DD In-Stock Unstable CNR2 37 41 COc1ccc(CCNc2ncc(C(=O)O)c(=O)[nH]2)cc1OC ZINC000217674517 DD In-Stock Unstable BRS3 28 41 COc1ccc(CCNc2ncc(C(=O)O)c(=O)[nH]2)cc1OC ZINC000217674517 DD In-Stock Unstable ABCG2 15 43 COc1ccc(CCNc2ncc(C(=O)O)c(=O)[nH]2)cc1OC ZINC000217674517 DD In-Stock Unstable ENPP1 49 30 COc1ccc(CCNc2ncc(C(=O)O)c(=O)[nH]2)cc1OC ZINC000217674517 DD In-Stock Unstable SCMU_MYCTU 0 42 COc1ccc(CCNc2ncc(C(=O)O)c(=O)[nH]2)cc1OC ZINC000217674517 DD In-Stock Unstable DRTS_TRYCR 43 30 CSc1cccc(NC(=O)N/C=C/c2ccccc2C)c1 ZINC000217674565 CJ For-Sale Unstable DDX3X 0 40 CSc1cccc(NC(=O)N/C=C/c2ccccc2C)c1 ZINC000217674565 CJ For-Sale Unstable KCNK3 67 38 OCc1cc2n(n1)CCN(c1ncnc3[nH]ccc13)C2 ZINC000217674592 CC In-Stock Unstable AKT2 47 44 OCc1cc2n(n1)CCN(c1ncnc3[nH]ccc13)C2 ZINC000217674592 CC In-Stock Unstable AKT3 35 40 OCc1cc2n(n1)CCN(c1ncnc3[nH]ccc13)C2 ZINC000217674592 CC In-Stock Unstable ROCK2 41 39 OCc1cc2n(n1)CCN(c1ncnc3[nH]ccc13)C2 ZINC000217674592 CC In-Stock Unstable AKT1 24 45 CCOC(=O)[C@@H](N[C@H](CC)CO)c1ccccc1 ZINC000217674599 CD On-Demand Unstable CAPN2 29 42 CCOC(=O)[C@@H](N[C@H](CC)CO)c1ccccc1 ZINC000217674599 CD On-Demand Unstable COL4A3BP 0 41 Cc1ccccc1/C=C/NC(=O)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217674674 IG For-Sale Unstable LPL 58 46 Cc1ccccc1/C=C/NC(=O)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217674674 IG For-Sale Unstable LIPG 24 46 CCOC(=O)[C@H](N[C@H](CC)CO)c1ccccc1 ZINC000217674678 CD On-Demand Unstable CAPN2 29 42 CCOC(=O)[C@H](N[C@H](CC)CO)c1ccccc1 ZINC000217674678 CD On-Demand Unstable COL4A3BP 0 41 CC(C)N(Cc1ccccc1)C[C@@H](C(=O)O)C(F)(F)F ZINC000217674700 CG For-Sale Unstable CPA1 40 43 CC(C)N(Cc1ccccc1)C[C@@H](C(=O)O)C(F)(F)F ZINC000217674700 CG For-Sale Unstable CES1 17 40 O=Cc1cc(C(=O)O)cc(C=O)c1O ZINC000217674761 AC For-Sale Anodyne TPMT 57 39 O=Cc1cc(C(=O)O)cc(C=O)c1O ZINC000217674761 AC For-Sale Anodyne HCAR1 0 40 CC(C)N(Cc1ccccc1)C[C@H](C(=O)O)C(F)(F)F ZINC000217674784 CG For-Sale Unstable CPA1 40 43 CC(C)N(Cc1ccccc1)C[C@H](C(=O)O)C(F)(F)F ZINC000217674784 CG For-Sale Unstable CES1 17 40 Cc1ccccc1/C=C/NC(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000217674789 EE For-Sale Unstable CA2 121 55 Cc1ccccc1/C=C/NC(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000217674789 EE For-Sale Unstable CA1 101 55 Cc1ccccc1/C=C/NC(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000217674789 EE For-Sale Unstable CA7 60 54 Cc1ccccc1/C=C/NC(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000217674789 EE For-Sale Unstable CA5B 56 54 Cc1ccccc1/C=C/NC(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000217674789 EE For-Sale Unstable CA4 79 55 Cc1ccccc1/C=C/NC(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000217674789 EE For-Sale Unstable CA5A 64 54 Cc1ccccc1/C=C/NC(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000217674789 EE For-Sale Unstable CA14 47 52 Cc1ccccc1/C=C/NC(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000217674789 EE For-Sale Unstable CA12 76 52 Cc1ccccc1/C=C/NC(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000217674789 EE For-Sale Unstable CA9 89 54 Cc1ccccc1/C=C/NC(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000217674789 EE For-Sale Unstable CYNT 35 45 Cc1ccccc1/C=C/NC(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000217674789 EE For-Sale Unstable MTCA1 48 52 Cc1ccccc1/C=C/NC(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000217674789 EE For-Sale Unstable P96878_MYCTU 62 52 COC(=O)c1ccc(CN[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217674826 CE On-Demand Unstable SLC18A3 44 35 COC(=O)c1ccc(CN[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217674826 CE On-Demand Unstable SSTR3 23 44 COC(=O)c1ccc(CN[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217674826 CE On-Demand Unstable L3MBTL3 55 35 CCOC(=O)[C@@H](NCC1CCCCC1)c1ccccc1 ZINC000217674850 CG On-Demand Unstable METAP2 34 44 Cc1ccccc1/C=C/NC(=O)Nc1cccnc1Cl ZINC000217674897 CH For-Sale Unstable G2YM83_BOTF4 66 34 CN(CC(F)(F)F)C(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217674900 CE For-Sale Unstable MLYCD 16 42 C[C@@H]1CCc2ccccc2N1C[C@@H](C(=O)O)C(F)(F)F ZINC000217674918 CG For-Sale Unstable ACE 25 40 COC(=O)c1ccc(CN[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217674928 CE On-Demand Unstable SLC18A3 44 35 COC(=O)c1ccc(CN[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217674928 CE On-Demand Unstable SSTR3 23 44 COC(=O)c1ccc(CN[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217674928 CE On-Demand Unstable L3MBTL3 55 35 CCOC(=O)[C@H](NCC1CCCCC1)c1ccccc1 ZINC000217674933 CG On-Demand Unstable METAP2 34 44 C[C@H]1CCc2ccccc2N1C[C@@H](C(=O)O)C(F)(F)F ZINC000217674999 CG For-Sale Unstable ACE 25 40 O=S(=O)(N1CCCC1)N1CC(n2cc(-c3ccccc3)nn2)C1 ZINC000217675032 ED In-Stock Unstable PREP 16 45 Cc1ccccc1[C@@H](C)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217675043 CG For-Sale Unstable SLC18A3 36 41 Cc1ccccc1[C@H](C)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217675128 CG On-Demand Unstable SLC18A3 33 41 C[C@@H]1Cc2ccccc2N1C[C@@H](C(=O)O)C(F)(F)F ZINC000217675141 CF For-Sale Unstable DRD4 21 40 C[C@@H]1Cc2ccccc2N1C[C@@H](C(=O)O)C(F)(F)F ZINC000217675141 CF For-Sale Unstable TPP2 51 32 CSC[C@@](C)(O)CNC(=O)CCc1ccc(C)cc1 ZINC000217675188 CE On-Demand Unstable FFAR1 17 41 C[C@H]1Cc2ccccc2N1C[C@@H](C(=O)O)C(F)(F)F ZINC000217675210 CF For-Sale Unstable DRD4 21 40 C[C@H]1Cc2ccccc2N1C[C@@H](C(=O)O)C(F)(F)F ZINC000217675210 CF For-Sale Unstable TPP2 51 32 Cc1ccccc1[C@@H](C)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217675212 CG For-Sale Unstable SLC18A3 36 41 C=CCn1c(SCCC(=O)Nc2sc3c(c2C#N)CCC3)nnc1-c1ccccc1F ZINC000217675247 JJ On-Demand Unstable MAPK10 17 46 C=CCn1c(SCCC(=O)Nc2sc3c(c2C#N)CCC3)nnc1-c1ccccc1F ZINC000217675247 JJ On-Demand Unstable VIPR1 28 47 CSC[C@](C)(O)CNC(=O)CCc1ccc(C)cc1 ZINC000217675270 CE On-Demand Unstable FFAR1 17 41 Cc1ccccc1[C@H](C)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217675296 CG On-Demand Unstable SLC18A3 33 41 O=C(CCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCc1ccccc1 ZINC000217675375 HH In-Stock Unstable SCN9A 0 40 O=C(CCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCc1ccccc1 ZINC000217675460 HH In-Stock Unstable SCN9A 0 40 CCOC(=O)[C@@H](NCCCN(C)C)c1ccccc1 ZINC000217675510 CD For-Sale Unstable THRA 42 37 CCOC(=O)[C@@H](NCCCN(C)C)c1ccccc1 ZINC000217675510 CD For-Sale Unstable AMY2 48 36 CC(C)CCN(C)C(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217675538 CF For-Sale Unstable AKR1C3 36 42 CCCCOC(=O)Cc1cc(OC)c(OC)cc1N ZINC000217675549 CE In-Stock Unstable PLA2G4B 40 40 CCCCOC(=O)Cc1cc(OC)c(OC)cc1N ZINC000217675549 CE In-Stock Unstable ACAT 0 41 CCOC(=O)[C@H](NCCCN(C)C)c1ccccc1 ZINC000217675603 CD For-Sale Unstable THRA 42 37 CCOC(=O)[C@H](NCCCN(C)C)c1ccccc1 ZINC000217675603 CD For-Sale Unstable AMY2 48 36 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)c1cccnc1)C2 ZINC000217675636 DC In-Stock Unstable GLRA1 16 45 CCN(C[C@@H](C(=O)O)C(F)(F)F)c1ccccc1 ZINC000217675676 CF For-Sale Unstable NR1H3 0 46 CCN(C[C@@H](C(=O)O)C(F)(F)F)c1ccccc1 ZINC000217675676 CF For-Sale Unstable NR1H2 29 46 CCN(C[C@H](C(=O)O)C(F)(F)F)c1ccccc1 ZINC000217675762 CF For-Sale Unstable NR1H3 0 46 CCN(C[C@H](C(=O)O)C(F)(F)F)c1ccccc1 ZINC000217675762 CF For-Sale Unstable NR1H2 29 46 CCC(=O)N(c1ccccc1)C1CCN(CCCCc2ccccc2)CC1 ZINC000217675765 FJ For-Sale Unstable CHRM2 19 45 CCC(=O)N(c1ccccc1)C1CCN(CCCCc2ccccc2)CC1 ZINC000217675765 FJ For-Sale Unstable HTR1A 22 46 CCC(=O)N(c1ccccc1)C1CCN(CCCCc2ccccc2)CC1 ZINC000217675765 FJ For-Sale Unstable CHRM1 26 43 CCC(=O)N(c1ccccc1)C1CCN(CCCCc2ccccc2)CC1 ZINC000217675765 FJ For-Sale Unstable DRD2 28 53 CCC(=O)N(c1ccccc1)C1CCN(CCCCc2ccccc2)CC1 ZINC000217675765 FJ For-Sale Unstable FKBP1A 31 40 CCC(=O)N(c1ccccc1)C1CCN(CCCCc2ccccc2)CC1 ZINC000217675765 FJ For-Sale Unstable DRD4 23 47 CCC(=O)N(c1ccccc1)C1CCN(CCCCc2ccccc2)CC1 ZINC000217675765 FJ For-Sale Unstable ACHE 17 49 CCC(=O)N(c1ccccc1)C1CCN(CCCCc2ccccc2)CC1 ZINC000217675765 FJ For-Sale Unstable HTR2A 25 55 CCC(=O)N(c1ccccc1)C1CCN(CCCCc2ccccc2)CC1 ZINC000217675765 FJ For-Sale Unstable HTR2C 15 50 CCC(=O)N(c1ccccc1)C1CCN(CCCCc2ccccc2)CC1 ZINC000217675765 FJ For-Sale Unstable SLC6A4 19 42 CCC(=O)N(c1ccccc1)C1CCN(CCCCc2ccccc2)CC1 ZINC000217675765 FJ For-Sale Unstable HRH1 30 50 CCC(=O)N(c1ccccc1)C1CCN(CCCCc2ccccc2)CC1 ZINC000217675765 FJ For-Sale Unstable OPRM1 40 86 CCC(=O)N(c1ccccc1)C1CCN(CCCCc2ccccc2)CC1 ZINC000217675765 FJ For-Sale Unstable DRD3 17 42 CCC(=O)N(c1ccccc1)C1CCN(CCCCc2ccccc2)CC1 ZINC000217675765 FJ For-Sale Unstable OPRD1 41 86 CCC(=O)N(c1ccccc1)C1CCN(CCCCc2ccccc2)CC1 ZINC000217675765 FJ For-Sale Unstable OPRK1 26 86 CCC(=O)N(c1ccccc1)C1CCN(CCCCc2ccccc2)CC1 ZINC000217675765 FJ For-Sale Unstable SLC6A3 19 45 CCC(=O)N(c1ccccc1)C1CCN(CCCCc2ccccc2)CC1 ZINC000217675765 FJ For-Sale Unstable CHRM3 25 40 CCC(=O)N(c1ccccc1)C1CCN(CCCCc2ccccc2)CC1 ZINC000217675765 FJ For-Sale Unstable GRIN2B 31 43 CCC(=O)N(c1ccccc1)C1CCN(CCCCc2ccccc2)CC1 ZINC000217675765 FJ For-Sale Unstable LTA4H 15 41 CCC(=O)N(c1ccccc1)C1CCN(CCCCc2ccccc2)CC1 ZINC000217675765 FJ For-Sale Unstable HTR7 25 41 CCC(=O)N(c1ccccc1)C1CCN(CCCCc2ccccc2)CC1 ZINC000217675765 FJ For-Sale Unstable HRH3 17 46 CCC(=O)N(c1ccccc1)C1CCN(CCCCc2ccccc2)CC1 ZINC000217675765 FJ For-Sale Unstable SIGMAR1 88 57 CCC(=O)N(c1ccccc1)C1CCN(CCCCc2ccccc2)CC1 ZINC000217675765 FJ For-Sale Unstable CCR3 23 40 CCC(=O)N(c1ccccc1)C1CCN(CCCCc2ccccc2)CC1 ZINC000217675765 FJ For-Sale Unstable KCNA3 19 46 CCC(=O)N(c1ccccc1)C1CCN(CCCCc2ccccc2)CC1 ZINC000217675765 FJ For-Sale Unstable CCR4 17 42 CCC(=O)N(c1ccccc1)C1CCN(CCCCc2ccccc2)CC1 ZINC000217675765 FJ For-Sale Unstable CCR5 66 44 CCC(=O)N(c1ccccc1)C1CCN(CCCCc2ccccc2)CC1 ZINC000217675765 FJ For-Sale Unstable PREP 45 37 CCC(=O)N(c1ccccc1)C1CCN(CCCCc2ccccc2)CC1 ZINC000217675765 FJ For-Sale Unstable ABCB1 15 86 CCC(=O)N(c1ccccc1)C1CCN(CCCCc2ccccc2)CC1 ZINC000217675765 FJ For-Sale Unstable PLM2_PLAFA 16 41 CCC(=O)N(c1ccccc1)C1CCN(CCCCc2ccccc2)CC1 ZINC000217675765 FJ For-Sale Unstable CACNA1G 25 45 CCC(=O)N(c1ccccc1)C1CCN(CCCCc2ccccc2)CC1 ZINC000217675765 FJ For-Sale Unstable CYP2J2 58 45 Cc1occc1CN(C)C(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217675798 DG For-Sale Unstable HSD17B2 27 40 Cc1c(NC(=O)CCOc2ccc(Cl)cc2Br)c(=O)n(-c2ccccc2)n1C ZINC000217675823 JI On-Demand Unstable IGF1R 18 41 Cc1c(NC(=O)CCOc2ccc(Cl)cc2Br)c(=O)n(-c2ccccc2)n1C ZINC000217675823 JI On-Demand Unstable FPR2 51 46 COC(=O)[C@@H](O)CNC(=O)c1cnc2ccccn2c1=O ZINC000217675831 CA On-Demand Unstable POLR1A 59 37 N#Cc1cc(Br)ccc1[C@@H]1CCNC1 ZINC000217675874 CE For-Sale Unstable IKBKB 26 41 COC(=O)[C@H](O)CNC(=O)c1cnc2ccccn2c1=O ZINC000217675923 CA On-Demand Unstable POLR1A 59 37 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)c1cccc(C#N)c1)C2 ZINC000217675929 ED In-Stock Unstable EZH2 55 36 Cc1cc(S(=O)(=O)N2CCCC2)ccc1/C=C\C(=O)O ZINC000217675983 CD For-Sale Unstable LPL 47 37 Cc1cc(S(=O)(=O)N2CCCC2)ccc1/C=C\C(=O)O ZINC000217675983 CD For-Sale Unstable CASP3 0 40 Cc1cc(S(=O)(=O)N2CCCC2)ccc1/C=C\C(=O)O ZINC000217675983 CD For-Sale Unstable F13A1 46 41 Cc1cc(S(=O)(=O)N2CCCC2)ccc1/C=C\C(=O)O ZINC000217675983 CD For-Sale Unstable AKR1C3 51 39 COC(=O)[C@@H](O)CNC(=O)Cc1cccc(O)c1 ZINC000217676032 CB On-Demand Unstable TRPV1 24 40 Cc1c(C(=O)O)cnc(=S)n1Cc1ccccc1 ZINC000217676121 CF In-Stock Unstable AGTR1 66 41 Cc1c(C(=O)O)cnc(=S)n1Cc1ccccc1 ZINC000217676121 CF In-Stock Unstable AGTR1B 52 37 Cc1c(C(=O)O)cnc(=S)n1Cc1ccccc1 ZINC000217676121 CF In-Stock Unstable PLA2G2A 66 40 COC(=O)[C@H](O)CNC(=O)Cc1cccc(O)c1 ZINC000217676130 CB On-Demand Unstable TRPV1 24 40 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCc1cccc(O)c1O ZINC000217676140 CH For-Sale Unstable TRPM8 17 46 Oc1cccc(-c2c3cn[nH]c3nc3c2oc2c(O)c(O)ccc23)c1 ZINC000217676188 EH In-Stock Clean HSD17B1 52 40 Oc1cccc(-c2c3cn[nH]c3nc3c2oc2c(O)c(O)ccc23)c1 ZINC000217676188 EH In-Stock Clean HSD17B2 28 40 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCc1cccc(O)c1O ZINC000217676209 CH For-Sale Unstable TRPM8 17 46 Brc1nc2ccccc2n1C1CCC1 ZINC000217676213 CH For-Sale Unstable RPS6KB1 32 48 COc1ccc([C@@H](C)N[C@@H]2CCC[C@@H](O)C2)cc1OC ZINC000217676221 CF For-Sale Unstable PDE4A 35 41 COc1ccc([C@@H](C)N[C@@H]2CCC[C@@H](O)C2)cc1OC ZINC000217676221 CF For-Sale Unstable PDE4B 20 41 COc1ccc([C@@H](C)N[C@@H]2CCC[C@@H](O)C2)cc1OC ZINC000217676221 CF For-Sale Unstable PDE4D 20 41 COc1ccc([C@@H](C)N[C@@H]2CCC[C@@H](O)C2)cc1OC ZINC000217676221 CF For-Sale Unstable PDE4C 15 41 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)CCc1ccccc1)C2 ZINC000217676225 ED In-Stock Unstable SLC6A3 15 40 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)CCc1ccccc1)C2 ZINC000217676225 ED In-Stock Unstable GRIN2B 23 50 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)CCc1ccccc1)C2 ZINC000217676225 ED In-Stock Unstable SIGMAR1 19 45 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)CCc1ccccc1)C2 ZINC000217676225 ED In-Stock Unstable NAAA 23 48 C[C@H]1CN(S(=O)(=O)c2cccc([C@H](C)N)c2)CCCO1 ZINC000217676232 CD For-Sale Unstable AKR1C3 41 33 COC(=O)[C@@H](O)CNC(=O)COc1ccc(Br)cc1 ZINC000217676239 EC On-Demand Unstable TRAR 21 42 COC(=O)[C@@H](O)CNC(=O)COc1ccc(Br)cc1 ZINC000217676239 EC On-Demand Unstable FAS 17 46 CC(=O)Cc1cccc(O)c1C(=O)O ZINC000217676255 AD In-Stock Unstable PLCG1 0 49 CC(=O)Cc1cccc(O)c1C(=O)O ZINC000217676255 AD In-Stock Unstable KAT5 0 43 CC(=O)Cc1cccc(O)c1C(=O)O ZINC000217676255 AD In-Stock Unstable G3PG_TRYCR 0 57 CC(=O)Cc1cccc(O)c1C(=O)O ZINC000217676255 AD In-Stock Unstable SAE1 0 57 CC(=O)Cc1cccc(O)c1C(=O)O ZINC000217676255 AD In-Stock Unstable CYP73A1 0 44 CCCCCNC(=O)N/C=C/c1ccccc1C ZINC000217676257 BG For-Sale Unstable ASAH1 76 34 CCCCCNC(=O)N/C=C/c1ccccc1C ZINC000217676257 BG For-Sale Unstable ACAT 0 55 CC[C@@H](C)NS(=O)(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217676261 DD For-Sale Unstable PTGER2 22 40 CC[C@@H](C)NS(=O)(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217676261 DD For-Sale Unstable MMP12 65 39 CC[C@@H](C)NS(=O)(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217676261 DD For-Sale Unstable ADAMTS4 51 34 CC[C@@H](C)NS(=O)(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217676261 DD For-Sale Unstable LEF 30 42 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCc1cccc(O)c1O ZINC000217676283 CH For-Sale Unstable TRPM8 17 46 COc1ccc([C@H](C)N[C@@H]2CCC[C@@H](O)C2)cc1OC ZINC000217676309 CF On-Demand Unstable PDE4B 20 41 COc1ccc([C@H](C)N[C@@H]2CCC[C@@H](O)C2)cc1OC ZINC000217676309 CF On-Demand Unstable PDE4D 20 41 COC(=O)[C@H](O)CNC(=O)COc1ccc(Br)cc1 ZINC000217676320 EC On-Demand Unstable TRAR 21 42 COC(=O)[C@H](O)CNC(=O)COc1ccc(Br)cc1 ZINC000217676320 EC On-Demand Unstable FAS 17 46 COc1ccccc1-n1cc(C(=O)O)cnc1=S ZINC000217676346 CE In-Stock Unstable HTR1A 32 40 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCc1cccc(O)c1O ZINC000217676359 CH For-Sale Unstable TRPM8 17 46 Cc1ccccc1/C=C/NC(=O)Nc1ccccc1 ZINC000217676367 CH For-Sale Unstable LPL 41 38 CC[C@H](C)NS(=O)(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217676368 DD For-Sale Unstable PTGER2 22 40 CC[C@H](C)NS(=O)(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217676368 DD For-Sale Unstable MMP12 65 39 CC[C@H](C)NS(=O)(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217676368 DD For-Sale Unstable ADAMTS4 51 34 CC[C@H](C)NS(=O)(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217676368 DD For-Sale Unstable LEF 30 42 COc1ccc([C@@H](C)N[C@H]2CCC[C@@H](O)C2)cc1OC ZINC000217676380 CF For-Sale Unstable PDE4A 35 41 COc1ccc([C@@H](C)N[C@H]2CCC[C@@H](O)C2)cc1OC ZINC000217676380 CF For-Sale Unstable PDE4B 20 41 COc1ccc([C@@H](C)N[C@H]2CCC[C@@H](O)C2)cc1OC ZINC000217676380 CF For-Sale Unstable PDE4D 20 41 COc1ccc([C@@H](C)N[C@H]2CCC[C@@H](O)C2)cc1OC ZINC000217676380 CF For-Sale Unstable PDE4C 15 41 COc1cccc(-n2c(C)c(C(=O)O)cnc2=S)c1 ZINC000217676451 CF In-Stock Unstable DHODH 16 40 COc1cccc(-n2c(C)c(C(=O)O)cnc2=S)c1 ZINC000217676451 CF In-Stock Unstable AKR1C3 24 40 COc1cccc(-n2c(C)c(C(=O)O)cnc2=S)c1 ZINC000217676451 CF In-Stock Unstable AKR1C2 50 38 COC(=O)[C@@H](O)CNC(=O)CNC(=O)c1cccc(Cl)c1 ZINC000217676455 DB On-Demand Unstable DRD4 44 37 COC(=O)[C@@H](O)CNC(=O)CNC(=O)c1cccc(Cl)c1 ZINC000217676455 DB On-Demand Unstable CTSL 15 42 COC(=O)[C@@H](O)CNC(=O)CNC(=O)c1cccc(Cl)c1 ZINC000217676455 DB On-Demand Unstable CCR2 43 41 COC(=O)[C@@H](O)CNC(=O)CNC(=O)c1cccc(Cl)c1 ZINC000217676455 DB On-Demand Unstable CTSV 35 42 COC(=O)[C@@H](O)CNC(=O)CNC(=O)c1cccc(Cl)c1 ZINC000217676455 DB On-Demand Unstable CACNA1I 32 43 COc1ccc([C@H](C)N[C@H]2CCC[C@@H](O)C2)cc1OC ZINC000217676469 CF On-Demand Unstable PDE4B 20 41 COc1ccc([C@H](C)N[C@H]2CCC[C@@H](O)C2)cc1OC ZINC000217676469 CF On-Demand Unstable PDE4D 20 41 C[C@@H](N[C@@H]1CCN2CCCC[C@@H]12)c1cccs1 ZINC000217676477 CG For-Sale Unstable VACHT_TETCF 0 44 CCOC(=O)[C@@H]1CCCN(C(=O)N/C=C/c2ccccc2C)C1 ZINC000217676481 DF For-Sale Unstable SLC6A1 100 40 CC(C)c1cc(C(=O)N[C@@H](C)Cn2cncn2)nc(N)n1 ZINC000217676507 CC In-Stock Unstable HIS3 87 40 COC(=O)[C@H](O)CNC(=O)CNC(=O)c1cccc(Cl)c1 ZINC000217676534 DB On-Demand Unstable DRD4 44 37 COC(=O)[C@H](O)CNC(=O)CNC(=O)c1cccc(Cl)c1 ZINC000217676534 DB On-Demand Unstable CTSL 15 42 COC(=O)[C@H](O)CNC(=O)CNC(=O)c1cccc(Cl)c1 ZINC000217676534 DB On-Demand Unstable CCR2 43 41 COC(=O)[C@H](O)CNC(=O)CNC(=O)c1cccc(Cl)c1 ZINC000217676534 DB On-Demand Unstable CTSV 35 42 COC(=O)[C@H](O)CNC(=O)CNC(=O)c1cccc(Cl)c1 ZINC000217676534 DB On-Demand Unstable CACNA1I 32 43 C[C@H](N[C@@H]1CCN2CCCC[C@@H]12)c1cccs1 ZINC000217676563 CG On-Demand Unstable VACHT_TETCF 0 44 CCOC(=O)[C@H]1CCCN(C(=O)N/C=C/c2ccccc2C)C1 ZINC000217676568 DF For-Sale Unstable SLC6A1 100 40 COc1cccc(-n2cc(C(=O)O)cnc2=S)c1 ZINC000217676569 CE In-Stock Unstable DRD4 41 32 COc1cccc(-n2cc(C(=O)O)cnc2=S)c1 ZINC000217676569 CE In-Stock Unstable CCKAR 15 40 CC(C)c1cc(C(=O)N[C@H](C)Cn2cncn2)nc(N)n1 ZINC000217676593 CC In-Stock Unstable HIS3 87 40 CC(C)Cc1cc(O)c(-c2ccccc2Cl)c(=O)[nH]1 ZINC000217676618 CH Annotated Unstable WEE1 47 34 CCN(C[C@@H](C(=O)O)C(F)(F)F)c1cccc(C)c1 ZINC000217676632 CG For-Sale Unstable CETP 0 44 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC)cc1O ZINC000217676648 CB On-Demand Unstable MTNR1A 58 40 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC)cc1O ZINC000217676648 CB On-Demand Unstable MTNR1B 46 40 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC)cc1O ZINC000217676648 CB On-Demand Unstable AKR1C2 50 36 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC)cc1O ZINC000217676648 CB On-Demand Unstable AKR1B10 30 41 C[C@@H](N[C@H]1CCN2CCCC[C@@H]12)c1cccs1 ZINC000217676654 CG For-Sale Unstable VACHT_TETCF 0 44 COc1ccc(-n2c(C)c(C(=O)O)cnc2=S)c(OC)c1 ZINC000217676689 DF In-Stock Unstable LUCI_LUCLA 15 40 COc1ccc(-n2c(C)c(C(=O)O)cnc2=S)c(OC)c1 ZINC000217676689 DF In-Stock Unstable AKR1C2 50 35 CCN(C[C@H](C(=O)O)C(F)(F)F)c1cccc(C)c1 ZINC000217676719 CG For-Sale Unstable CETP 0 44 COC(=O)[C@H](O)CNC(=O)c1ccc(OC)cc1O ZINC000217676725 CB For-Sale Unstable MTNR1A 58 40 COC(=O)[C@H](O)CNC(=O)c1ccc(OC)cc1O ZINC000217676725 CB For-Sale Unstable MTNR1B 46 40 COC(=O)[C@H](O)CNC(=O)c1ccc(OC)cc1O ZINC000217676725 CB For-Sale Unstable AKR1C2 40 36 COC(=O)[C@H](O)CNC(=O)c1ccc(OC)cc1O ZINC000217676725 CB For-Sale Unstable AKR1B10 30 41 C[C@H](N[C@H]1CCN2CCCC[C@@H]12)c1cccs1 ZINC000217676730 CG On-Demand Unstable VACHT_TETCF 0 44 COC(=O)c1cc(-c2ccccc2Cl)nn1C ZINC000217676805 CF In-Stock Unstable ALPL 21 43 COC(=O)c1cc(-c2ccccc2Cl)nn1C ZINC000217676805 CF In-Stock Unstable MT-CYB 49 39 CC(C)CCNS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217676806 CE For-Sale Unstable HDAC8 17 46 CC(C)CCNS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217676806 CE For-Sale Unstable AKR1C3 37 45 CCOc1ccc(OCC(=O)NC[C@@H](O)C(=O)OC)cc1 ZINC000217676831 CC On-Demand Unstable PLA2G4B 60 33 COc1cc2c(cc1OC)[C@@H](c1cccnc1)N(C(=O)c1cnc[nH]1)CC2 ZINC000217676834 FF In-Stock Unstable MTNR1B 20 40 Cc1nc2c3ccccc3nc(SCc3cnn(-c4ccccc4)c3)n2n1 ZINC000217676846 FI On-Demand Unstable PDE10A 20 65 O=C(O)/C=C\c1cccc(C(=O)Nc2cnccn2)c1 ZINC000217676882 CD For-Sale Anodyne KCNK3 60 38 Cc1c(C(=O)O)cnc(=S)n1-c1ccccc1 ZINC000217676897 BF In-Stock Unstable SLC9A2 0 43 CCOc1ccc(OCC(=O)NC[C@H](O)C(=O)OC)cc1 ZINC000217676920 CC On-Demand Unstable PLA2G4B 60 33 COc1cc2c(cc1OC)[C@H](c1cccnc1)N(C(=O)c1cnc[nH]1)CC2 ZINC000217676932 FF In-Stock Unstable MTNR1B 20 40 CS(=O)(=O)Nc1ccc(-c2csc(NC(=O)c3c[nH]nc3-c3ccc(Cl)cc3)n2)cc1 ZINC000217676957 JI On-Demand Unstable MPL 29 45 CS(=O)(=O)Nc1ccc(-c2csc(NC(=O)c3c[nH]nc3-c3ccc(Cl)cc3)n2)cc1 ZINC000217676957 JI On-Demand Unstable ROCK1 19 42 CS(=O)(=O)Nc1ccc(-c2csc(NC(=O)c3c[nH]nc3-c3ccc(Cl)cc3)n2)cc1 ZINC000217676957 JI On-Demand Unstable U38 0 49 COc1ccc([C@@H](C#N)N2CCN(C(=O)CSc3ccc(Cl)c(C(F)(F)F)c3)CC2)cc1 ZINC000217677056 JJ On-Demand Unstable PTAFR 41 40 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)COc1ccccc1F)C2 ZINC000217677090 FD In-Stock Unstable LUXN 0 40 CCc1ccc(NC(=O)N/C=C/c2ccccc2C)cc1 ZINC000217677093 CI For-Sale Unstable FPR2 15 42 COc1cccc(-n2c(C)c(C(=O)O)cnc2=O)c1 ZINC000217677099 CD In-Stock Unstable HPD 20 45 COc1cccc(-n2c(C)c(C(=O)O)cnc2=O)c1 ZINC000217677099 CD In-Stock Unstable DHODH 16 40 COc1cccc(-n2c(C)c(C(=O)O)cnc2=O)c1 ZINC000217677099 CD In-Stock Unstable AKR1C3 28 40 COc1cccc(-n2c(C)c(C(=O)O)cnc2=O)c1 ZINC000217677099 CD In-Stock Unstable AKR1C2 51 38 O=C(O)c1[nH]nc(-c2cccc([N+](=O)[O-])c2)c1Br ZINC000217677121 DE In-Stock Bother FBP1 0 44 O=C(O)c1[nH]nc(-c2cccc([N+](=O)[O-])c2)c1Br ZINC000217677121 DE In-Stock Bother HAO2 79 38 COc1ccc([C@H](C#N)N2CCN(C(=O)CSc3ccc(Cl)c(C(F)(F)F)c3)CC2)cc1 ZINC000217677124 JJ On-Demand Unstable PTAFR 41 40 Cc1cccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)c1 ZINC000217677137 CG For-Sale Unstable MAOB 0 60 Cc1cccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)c1 ZINC000217677137 CG For-Sale Unstable KIT 17 41 Cc1cccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)c1 ZINC000217677137 CG For-Sale Unstable CCKAR 23 48 Cc1cccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)c1 ZINC000217677137 CG For-Sale Unstable HDAC8 27 55 Cc1cccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)c1 ZINC000217677137 CG For-Sale Unstable KDR 16 41 Cc1cccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)c1 ZINC000217677137 CG For-Sale Unstable MMP2 0 57 Cc1cccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)c1 ZINC000217677137 CG For-Sale Unstable NR1H4 15 43 Cc1cccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)c1 ZINC000217677137 CG For-Sale Unstable HDAC6 19 55 Cc1cccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)c1 ZINC000217677137 CG For-Sale Unstable F12 0 41 Cc1cccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)c1 ZINC000217677137 CG For-Sale Unstable MMP9 0 57 Cc1cccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)c1 ZINC000217677137 CG For-Sale Unstable TTR 0 42 Cc1cccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)c1 ZINC000217677137 CG For-Sale Unstable CSF1R 24 45 Cc1cccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)c1 ZINC000217677137 CG For-Sale Unstable MMP1 0 57 Cc1cccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)c1 ZINC000217677137 CG For-Sale Unstable TAAR1 47 44 Cc1cccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)c1 ZINC000217677137 CG For-Sale Unstable AKR1C3 54 42 Cc1cccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)c1 ZINC000217677137 CG For-Sale Unstable DDR1 28 41 Cc1cccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)c1 ZINC000217677137 CG For-Sale Unstable TRPM8 0 51 Cc1cccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)c1 ZINC000217677137 CG For-Sale Unstable RHOA 0 43 Cc1cccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)c1 ZINC000217677137 CG For-Sale Unstable PARP14 0 45 Cc1cccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)c1 ZINC000217677137 CG For-Sale Unstable PARP15 0 45 Cc1cccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)c1 ZINC000217677137 CG For-Sale Unstable KCNK3 155 64 Cc1cccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)c1 ZINC000217677137 CG For-Sale Unstable KCNK9 101 64 Cc1cccc(NC(=O)c2cccc(/C=C\C(=O)O)c2)c1 ZINC000217677137 CG For-Sale Unstable PARP10 0 45 CCOC(=O)[C@H]1C[C@@H]1c1ccc(OC)c(OC)c1 ZINC000217677177 CE For-Sale Unstable SLC6A1 59 49 CCOC(=O)[C@H]1C[C@@H]1c1ccc(OC)c(OC)c1 ZINC000217677177 CE For-Sale Unstable SLC6A4 15 40 CCOC(=O)[C@H]1C[C@@H]1c1ccc(OC)c(OC)c1 ZINC000217677177 CE For-Sale Unstable SLC6A3 29 40 CN(C[C@@H]1CCCO1)C[C@H](C(=O)O)C(F)(F)F ZINC000217677202 CD For-Sale Unstable OXTR 27 43 CN(C[C@@H]1CCCO1)C[C@H](C(=O)O)C(F)(F)F ZINC000217677202 CD For-Sale Unstable AVPR1A 0 41 COc1cccc(-n2cc(C(=O)O)cnc2=O)c1 ZINC000217677210 BC In-Stock Unstable DRD4 42 33 COc1cccc(-n2cc(C(=O)O)cnc2=O)c1 ZINC000217677210 BC In-Stock Unstable HPD 19 42 COc1cccc(-n2cc(C(=O)O)cnc2=O)c1 ZINC000217677210 BC In-Stock Unstable CCKAR 24 40 COc1cccc(-n2cc(C(=O)O)cnc2=O)c1 ZINC000217677210 BC In-Stock Unstable HPGD 28 47 COc1cccc(-n2cc(C(=O)O)cnc2=O)c1 ZINC000217677210 BC In-Stock Unstable CYSK1 41 35 O=C(COc1ccccc1Br)Nc1cccc(-c2nnc3n2CCCCC3)c1 ZINC000217677263 II On-Demand Unstable PTPN2 46 33 O=C(COc1ccccc1Br)Nc1cccc(-c2nnc3n2CCCCC3)c1 ZINC000217677263 II On-Demand Unstable PTPN1 41 33 CCOc1ccc(CC(=O)NC2C[C@@H]3CC[C@H](C2)N3S(C)(=O)=O)cc1 ZINC000217677276 FD In-Stock Unstable AVPR1A 0 43 CCOc1ccc(CC(=O)NC2C[C@@H]3CC[C@H](C2)N3S(C)(=O)=O)cc1 ZINC000217677276 FD In-Stock Unstable MMP13 46 42 CCOc1ccc(CC(=O)NC2C[C@@H]3CC[C@H](C2)N3S(C)(=O)=O)cc1 ZINC000217677276 FD In-Stock Unstable MMP2 23 41 CCOc1ccc(CC(=O)NC2C[C@@H]3CC[C@H](C2)N3S(C)(=O)=O)cc1 ZINC000217677276 FD In-Stock Unstable MMP1 34 42 COc1ccc(C[C@@H](C)N[C@@H]2CCC[C@@H](O)C2)cc1 ZINC000217677308 CF For-Sale Unstable SLC18A2 23 40 Cc1ccccc1/C=C/NC(=O)NC1CC(C)(C)NC(C)(C)C1 ZINC000217677311 DH For-Sale Unstable EZH2 53 40 Cc1ccc(-n2c(C)c(C(=O)O)cnc2=O)c(C)c1 ZINC000217677318 CD In-Stock Unstable HPD 15 43 O=C(O)/C=C\c1ccc(F)c(C(=O)N2CCOCC2)c1 ZINC000217677325 CD For-Sale Unstable PARP1 30 40 O=C(O)/C=C\c1ccc(F)c(C(=O)N2CCOCC2)c1 ZINC000217677325 CD For-Sale Unstable AKR1C3 36 40 O=C(O)/C=C\c1ccc(C(=O)N2CCOCC2)c(F)c1 ZINC000217677389 CD For-Sale Unstable AKR1C3 54 37 COc1ccc(C[C@H](C)N[C@@H]2CCC[C@@H](O)C2)cc1 ZINC000217677401 CF On-Demand Unstable SLC18A2 23 40 COC(=O)[C@@H](O)CNC(=O)[C@@H](C)Oc1cccc(Cl)c1 ZINC000217677425 DC On-Demand Unstable MTNR1A 19 43 COC(=O)[C@@H](O)CNC(=O)[C@@H](C)Oc1cccc(Cl)c1 ZINC000217677425 DC On-Demand Unstable MTNR1B 20 43 COc1ccc(C[C@@H](C)N[C@H]2CCC[C@@H](O)C2)cc1 ZINC000217677478 CF For-Sale Unstable SLC18A2 23 40 COC(=O)[C@H](O)CNC(=O)[C@@H](C)Oc1cccc(Cl)c1 ZINC000217677507 DC On-Demand Unstable MTNR1A 19 43 COC(=O)[C@H](O)CNC(=O)[C@@H](C)Oc1cccc(Cl)c1 ZINC000217677507 DC On-Demand Unstable MTNR1B 20 43 CSc1ccccc1C(=O)Nc1nc2ccccc2nc1N1CCCC1 ZINC000217677563 FI On-Demand Unstable KCNQ2 40 32 COc1ccc(C[C@H](C)N[C@H]2CCC[C@@H](O)C2)cc1 ZINC000217677565 CF On-Demand Unstable SLC18A2 23 40 COC(=O)[C@@H](O)CNC(=O)[C@H](C)Oc1cccc(Cl)c1 ZINC000217677585 DC On-Demand Unstable MTNR1A 19 43 COC(=O)[C@@H](O)CNC(=O)[C@H](C)Oc1cccc(Cl)c1 ZINC000217677585 DC On-Demand Unstable MTNR1B 20 43 COC(=O)C[C@H](c1ccc(-c2ccc(C(=O)O)cc2)o1)c1c(O)c2ccccc2oc1=O ZINC000217677628 II In-Stock Unstable NQO1 35 47 COC(=O)C[C@H](c1ccc(-c2ccc(C(=O)O)cc2)o1)c1c(O)c2ccccc2oc1=O ZINC000217677628 II In-Stock Unstable TNKS 26 45 CC(C)c1ccc(NS(=O)(=O)CCCCO)cc1 ZINC000217677631 CE For-Sale Unstable TBXA2R 16 55 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)CCSc1ccccc1)C2 ZINC000217677639 FE In-Stock Unstable TNKS 64 33 COc1cccc(-n2c(N)c(C(=O)O)cnc2=S)c1 ZINC000217677664 CD In-Stock Unstable AKR1C2 50 34 COC(=O)[C@H](O)CNC(=O)[C@H](C)Oc1cccc(Cl)c1 ZINC000217677681 DC On-Demand Unstable MTNR1A 19 43 COC(=O)[C@H](O)CNC(=O)[C@H](C)Oc1cccc(Cl)c1 ZINC000217677681 DC On-Demand Unstable MTNR1B 20 43 C[C@@H]1CCCN(C(=O)c2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217677696 CF For-Sale Unstable L3MBTL3 70 42 C[C@@H]1CCCN(C(=O)c2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217677696 CF For-Sale Unstable HPGD 15 46 COC(=O)C[C@@H](c1ccc(-c2ccc(C(=O)O)cc2)o1)c1c(O)c2ccccc2oc1=O ZINC000217677727 II In-Stock Unstable NQO1 35 47 COC(=O)C[C@@H](c1ccc(-c2ccc(C(=O)O)cc2)o1)c1c(O)c2ccccc2oc1=O ZINC000217677727 II In-Stock Unstable TNKS 26 45 CCOC(=O)[C@@H](Nc1ccc(CC)cc1)c1ccccc1 ZINC000217677755 CH On-Demand Unstable TIMP3 48 31 CCOC(=O)[C@@H](Nc1ccc(CC)cc1)c1ccccc1 ZINC000217677755 CH On-Demand Unstable CAPN2 52 33 CSC[C@@](C)(O)CNC(=O)CCc1cccnc1 ZINC000217677756 CD On-Demand Unstable TBXAS1 31 42 CSC[C@@](C)(O)CNC(=O)CCc1cccnc1 ZINC000217677756 CD On-Demand Unstable PTAFR 28 40 CSC[C@@](C)(O)CNC(=O)CCc1cccnc1 ZINC000217677756 CD On-Demand Unstable C3AR1 41 37 CSC[C@@](C)(O)CNC(=O)CCc1cccnc1 ZINC000217677756 CD On-Demand Unstable NAMPT 21 44 C[C@H]1CCCN(C(=O)c2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217677766 CF For-Sale Unstable L3MBTL3 70 42 C[C@H]1CCCN(C(=O)c2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217677766 CF For-Sale Unstable HPGD 15 46 Cc1nc(NCCN)cc(Nc2ccccc2)n1 ZINC000217677792 BD In-Stock Unstable AGPAT2 45 37 COC(=O)[C@@H](O)CNC(=O)c1cc(OC)ccc1OC ZINC000217677793 CB On-Demand Unstable MTNR1A 52 40 COC(=O)[C@@H](O)CNC(=O)c1cc(OC)ccc1OC ZINC000217677793 CB On-Demand Unstable MTNR1B 43 40 COC(=O)[C@@H](O)CNC(=O)c1cc(OC)ccc1OC ZINC000217677793 CB On-Demand Unstable AKR1C2 48 33 CSC[C@](C)(O)CNC(=O)CCc1cccnc1 ZINC000217677837 CD On-Demand Unstable TBXAS1 31 42 CSC[C@](C)(O)CNC(=O)CCc1cccnc1 ZINC000217677837 CD On-Demand Unstable PTAFR 28 40 CSC[C@](C)(O)CNC(=O)CCc1cccnc1 ZINC000217677837 CD On-Demand Unstable C3AR1 41 37 CSC[C@](C)(O)CNC(=O)CCc1cccnc1 ZINC000217677837 CD On-Demand Unstable NAMPT 21 44 CCOC(=O)[C@H](Nc1ccc(CC)cc1)c1ccccc1 ZINC000217677838 CH On-Demand Unstable TIMP3 56 31 CCOC(=O)[C@H](Nc1ccc(CC)cc1)c1ccccc1 ZINC000217677838 CH On-Demand Unstable CAPN2 52 33 CCOC(=O)[C@H](Nc1ccc(CC)cc1)c1ccccc1 ZINC000217677838 CH On-Demand Unstable NPR 41 33 O=C(O)/C=C\c1cccc(C(=O)Nc2ccncc2)c1 ZINC000217677852 CE For-Sale Anodyne PRNP 17 42 O=C(O)/C=C\c1cccc(C(=O)Nc2ccncc2)c1 ZINC000217677852 CE For-Sale Anodyne ROCK2 28 42 O=C(O)/C=C\c1cccc(C(=O)Nc2ccncc2)c1 ZINC000217677852 CE For-Sale Anodyne TYK2 30 44 O=C(O)/C=C\c1cccc(C(=O)Nc2ccncc2)c1 ZINC000217677852 CE For-Sale Anodyne CSF1R 17 40 O=C(O)/C=C\c1cccc(C(=O)Nc2ccncc2)c1 ZINC000217677852 CE For-Sale Anodyne TAAR1 23 41 O=C(O)/C=C\c1cccc(C(=O)Nc2ccncc2)c1 ZINC000217677852 CE For-Sale Anodyne KCNK3 116 55 O=C(O)/C=C\c1cccc(C(=O)Nc2ccncc2)c1 ZINC000217677852 CE For-Sale Anodyne KCNK9 60 46 COC(=O)[C@H](O)CNC(=O)c1cc(OC)ccc1OC ZINC000217677884 CB On-Demand Unstable MTNR1A 52 40 COC(=O)[C@H](O)CNC(=O)c1cc(OC)ccc1OC ZINC000217677884 CB On-Demand Unstable MTNR1B 43 40 COC(=O)[C@H](O)CNC(=O)c1cc(OC)ccc1OC ZINC000217677884 CB On-Demand Unstable AKR1C2 48 33 CCN(Cc1ccccc1)C(=O)N/C=C/c1ccccc1C ZINC000217677908 CI For-Sale Unstable TSPO 20 41 CCN(Cc1ccccc1)C(=O)N/C=C/c1ccccc1C ZINC000217677908 CI For-Sale Unstable LIMK2 18 40 COc1ccc(Nc2cc(NCCN)nc(C)n2)cc1 ZINC000217677920 CD In-Stock Unstable GALR2 58 43 COc1ccc(Nc2cc(NCCN)nc(C)n2)cc1 ZINC000217677920 CD In-Stock Unstable AGPAT2 62 40 O=C(O)/C=C\c1ccc(F)c(C(=O)Nc2ccncc2)c1 ZINC000217677951 CF For-Sale Anodyne MMP1 0 40 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217677993 DC On-Demand Unstable GCGR 47 51 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217677993 DC On-Demand Unstable GRIN2B 23 42 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217677993 DC On-Demand Unstable TRPV1 0 52 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217677993 DC On-Demand Unstable ACR 48 33 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217677993 DC On-Demand Unstable GIPR 56 51 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217677993 DC On-Demand Unstable SHH 40 34 CCC[C@@H]1CC[C@@H](N)[C@@H](CCc2ccc([N+](=O)[O-])cc2)C1 ZINC000217677997 CI For-Sale Unstable KCNJ1 22 40 Cc1nc(NCCN)cc(Nc2ccc(Cl)cc2)n1 ZINC000217678030 CF In-Stock Unstable AGPAT2 78 51 Cc1nc(NCCN)cc(Nc2ccc(Cl)cc2)n1 ZINC000217678030 CF In-Stock Unstable PETD 0 40 O=C(O)/C=C\c1ccc(C(=O)Nc2ccncc2)c(F)c1 ZINC000217678048 CF For-Sale Anodyne MMP1 0 40 COC(=O)[C@H](O)CNC(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217678084 DC On-Demand Unstable GCGR 47 51 COC(=O)[C@H](O)CNC(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217678084 DC On-Demand Unstable GRIN2B 23 42 COC(=O)[C@H](O)CNC(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217678084 DC On-Demand Unstable TRPV1 0 52 COC(=O)[C@H](O)CNC(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217678084 DC On-Demand Unstable ACR 48 33 COC(=O)[C@H](O)CNC(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217678084 DC On-Demand Unstable GIPR 56 51 COC(=O)[C@H](O)CNC(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217678084 DC On-Demand Unstable SHH 40 34 CCC[C@H]1CC[C@@H](N)[C@@H](CCc2ccc([N+](=O)[O-])cc2)C1 ZINC000217678093 CI For-Sale Unstable KCNJ1 22 40 COc1ccc(Cl)cc1C(=O)NC1C[C@@H]2CC[C@H](C1)N2S(C)(=O)=O ZINC000217678109 FE In-Stock Unstable DRD2 26 45 COc1ccc(Cl)cc1C(=O)NC1C[C@@H]2CC[C@H](C1)N2S(C)(=O)=O ZINC000217678109 FE In-Stock Unstable DRD3 0 41 COc1ccc(Cl)cc1C(=O)NC1C[C@@H]2CC[C@H](C1)N2S(C)(=O)=O ZINC000217678109 FE In-Stock Unstable COLA 70 36 COc1ccc(Cl)cc1C(=O)NC1C[C@@H]2CC[C@H](C1)N2S(C)(=O)=O ZINC000217678109 FE In-Stock Unstable CPT1A 44 30 COc1ccc(Cl)cc1C(=O)NC1C[C@@H]2CC[C@H](C1)N2S(C)(=O)=O ZINC000217678109 FE In-Stock Unstable CPT2 46 35 COc1ccc(Cl)cc1C(=O)NC1C[C@@H]2CC[C@H](C1)N2S(C)(=O)=O ZINC000217678109 FE In-Stock Unstable CPT1B 52 35 Cc1ccc(Nc2cc(NCCN)nc(C)n2)cc1 ZINC000217678138 CE In-Stock Unstable AGPAT2 56 40 CCC[C@@H]1CC[C@H](N)[C@@H](CCc2ccc([N+](=O)[O-])cc2)C1 ZINC000217678178 CI For-Sale Unstable KCNJ1 22 40 COC(=O)[C@@H](O)CNC(=O)CSc1ccccc1 ZINC000217678227 CC On-Demand Unstable FAS 73 49 CCC[C@H]1CC[C@H](N)[C@@H](CCc2ccc([N+](=O)[O-])cc2)C1 ZINC000217678263 CI For-Sale Unstable KCNJ1 22 40 COC(=O)[C@H](O)CNC(=O)CSc1ccccc1 ZINC000217678293 CC On-Demand Unstable FAS 73 49 C[C@@H](CCc1ccccc1)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217678299 CG For-Sale Unstable SLC18A2 41 36 C[C@@H](CCc1ccccc1)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217678299 CG For-Sale Unstable SIGMAR1 22 49 C[C@@H](CCc1ccccc1)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217678299 CG For-Sale Unstable SLC18A3 36 43 O=C(O)/C=C\c1ccc(C(=O)NCCc2cccnc2)s1 ZINC000217678301 DE For-Sale Unstable TBXAS1 44 60 O=C(O)/C=C\c1ccc(C(=O)NCCc2cccnc2)s1 ZINC000217678301 DE For-Sale Unstable PTAFR 28 44 O=C(O)/C=C\c1ccc(C(=O)NCCc2cccnc2)s1 ZINC000217678301 DE For-Sale Unstable CHRNA7 33 41 CCOC(=O)[C@@H](Nc1ccc(C)c(F)c1)c1ccccc1 ZINC000217678341 CH On-Demand Unstable DHODH 21 41 CCOC(=O)[C@@H](Nc1ccc(C)c(F)c1)c1ccccc1 ZINC000217678341 CH On-Demand Unstable NPY2R 51 34 CCOC(=O)[C@@H](Nc1ccc(C)c(F)c1)c1ccccc1 ZINC000217678341 CH On-Demand Unstable FPR2 19 41 CCOC(=O)[C@@H](Nc1ccc(C)c(F)c1)c1ccccc1 ZINC000217678341 CH On-Demand Unstable DHOD 0 44 Cc1nc(Nc2ccc(Cl)cc2)cc(N2CCNCC2)n1 ZINC000217678360 DF In-Stock Unstable PRKD1 49 40 Cc1nc(Nc2ccc(Cl)cc2)cc(N2CCNCC2)n1 ZINC000217678360 DF In-Stock Unstable GALR2 48 39 Cc1nc(Nc2ccc(Cl)cc2)cc(N2CCNCC2)n1 ZINC000217678360 DF In-Stock Unstable AGPAT2 52 41 Cc1nc(Nc2ccc(Cl)cc2)cc(N2CCNCC2)n1 ZINC000217678360 DF In-Stock Unstable PKD2 0 47 Cc1nc(Nc2ccc(Cl)cc2)cc(N2CCNCC2)n1 ZINC000217678360 DF In-Stock Unstable KARS 56 37 COc1ccc(C(=O)NCC(C)(C)C)cc1/C=C\C(=O)O ZINC000217678382 CF For-Sale Unstable LTB4R 27 40 COc1ccc(C(=O)NCC(C)(C)C)cc1/C=C\C(=O)O ZINC000217678382 CF For-Sale Unstable COLA 24 43 COc1ccc(C(=O)NCC(C)(C)C)cc1/C=C\C(=O)O ZINC000217678382 CF For-Sale Unstable CPT1A 43 30 C[C@H](CCc1ccccc1)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217678395 CG On-Demand Unstable SLC18A2 41 36 C[C@H](CCc1ccccc1)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217678395 CG On-Demand Unstable SLC18A3 29 42 Cc1ccccc1/C=C/NC(=O)N(Cc1ccccc1)Cc1ccccc1 ZINC000217678411 FK For-Sale Unstable PTGES 22 41 CCOC(=O)[C@H](Nc1ccc(C)c(F)c1)c1ccccc1 ZINC000217678432 CH On-Demand Unstable DHODH 21 41 CCOC(=O)[C@H](Nc1ccc(C)c(F)c1)c1ccccc1 ZINC000217678432 CH On-Demand Unstable NPY2R 51 34 CCOC(=O)[C@H](Nc1ccc(C)c(F)c1)c1ccccc1 ZINC000217678432 CH On-Demand Unstable FPR2 19 41 CCOC(=O)[C@H](Nc1ccc(C)c(F)c1)c1ccccc1 ZINC000217678432 CH On-Demand Unstable DHOD 0 44 Cc1nc(Nc2ccc(F)cc2)cc(N2CCNCC2)n1 ZINC000217678452 CE In-Stock Unstable PRKD1 49 41 Cc1nc(Nc2ccc(F)cc2)cc(N2CCNCC2)n1 ZINC000217678452 CE In-Stock Unstable GALR2 58 45 Cc1nc(Nc2ccc(F)cc2)cc(N2CCNCC2)n1 ZINC000217678452 CE In-Stock Unstable PKD2 0 47 Cc1nc(Nc2ccc(F)cc2)cc(N2CCNCC2)n1 ZINC000217678452 CE In-Stock Unstable KARS 62 38 C[C@@H](CCc1ccccc1)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217678495 CG For-Sale Unstable SLC18A2 41 36 C[C@@H](CCc1ccccc1)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217678495 CG For-Sale Unstable SIGMAR1 22 49 C[C@@H](CCc1ccccc1)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217678495 CG For-Sale Unstable SLC18A3 36 43 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)c1ccc(C(F)(F)F)cc1)C2 ZINC000217678497 GE In-Stock Unstable CCR2 61 39 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)c1ccc(C(F)(F)F)cc1)C2 ZINC000217678497 GE In-Stock Unstable SLC6A5 36 46 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)c1ccc(C(F)(F)F)cc1)C2 ZINC000217678497 GE In-Stock Unstable EPHX2 25 48 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)c1ccc(C(F)(F)F)cc1)C2 ZINC000217678497 GE In-Stock Unstable ELOVL6 0 45 Cc1ccccc1/C=C/NC(=O)N(CCO)Cc1ccccc1 ZINC000217678521 DG For-Sale Unstable LIMK2 20 40 CSC[C@@](C)(O)CNC(=O)c1ccc(CS(C)(=O)=O)cc1 ZINC000217678550 ED On-Demand Unstable CYNT 24 40 Cc1cccc(Nc2cc(N3CCNCC3)nc(C)n2)c1 ZINC000217678569 CE In-Stock Unstable PRKD1 50 42 Cc1cccc(Nc2cc(N3CCNCC3)nc(C)n2)c1 ZINC000217678569 CE In-Stock Unstable GALR2 50 38 Cc1cccc(Nc2cc(N3CCNCC3)nc(C)n2)c1 ZINC000217678569 CE In-Stock Unstable PKD2 0 48 Cc1cccc(Nc2cc(N3CCNCC3)nc(C)n2)c1 ZINC000217678569 CE In-Stock Unstable KARS 61 36 COc1cc2c(cc1OC)CN(Cc1cc(=O)c(O)c(CN3CCCC3)o1)CC2 ZINC000217678576 HF In-Stock Unstable ABCB1B 61 35 COc1cc2c(cc1OC)CN(Cc1cc(=O)c(O)c(CN3CCCC3)o1)CC2 ZINC000217678576 HF In-Stock Unstable ABCB1 23 48 CCC[C@@H](O)CNc1ccncc1N ZINC000217678580 AD For-Sale Unstable AMO_PEA 41 36 C[C@H](CCc1ccccc1)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217678582 CG On-Demand Unstable SLC18A2 41 36 C[C@H](CCc1ccccc1)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217678582 CG On-Demand Unstable SLC18A3 29 42 C[C@@H](NC1CCC(O)CC1)C(=O)N1CCCCC1 ZINC000217678604 CD On-Demand Unstable DPP7 33 40 CSC[C@](C)(O)CNC(=O)c1ccc(CS(C)(=O)=O)cc1 ZINC000217678634 ED On-Demand Unstable CYNT 24 40 COc1ccc(NC(=O)N/C=C/c2ccccc2C)c(OC)c1 ZINC000217678637 DH For-Sale Unstable CYP1B1 40 47 COc1ccc(NC(=O)N/C=C/c2ccccc2C)c(OC)c1 ZINC000217678637 DH For-Sale Unstable MTNR1A 22 46 COc1ccc(NC(=O)N/C=C/c2ccccc2C)c(OC)c1 ZINC000217678637 DH For-Sale Unstable MTNR1B 21 46 COc1ccc(NC(=O)N/C=C/c2ccccc2C)c(OC)c1 ZINC000217678637 DH For-Sale Unstable AKR1C2 44 33 CCC[C@H](O)CNc1ccncc1N ZINC000217678670 AD For-Sale Unstable AMO_PEA 41 36 COc1cccc2cc(C(=O)NC3C[C@@H]4CC[C@H](C3)N4S(C)(=O)=O)oc12 ZINC000217678674 GE In-Stock Unstable DRD2 19 40 COc1cccc2cc(C(=O)NC3C[C@@H]4CC[C@H](C3)N4S(C)(=O)=O)oc12 ZINC000217678674 GE In-Stock Unstable HTR3A 26 49 CCCNc1ccc(C(=O)N2CCCC2)cc1N ZINC000217678680 BE In-Stock Unstable L3MBTL1 0 44 CCCNc1ccc(C(=O)N2CCCC2)cc1N ZINC000217678680 BE In-Stock Unstable L3MBTL3 68 44 CCCNc1ccc(C(=O)N2CCCC2)cc1N ZINC000217678680 BE In-Stock Unstable HPGD 35 42 C[C@H](NC1CCC(O)CC1)C(=O)N1CCCCC1 ZINC000217678689 CD On-Demand Unstable DPP7 33 40 CCC[C@@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678775 EI On-Demand Unstable ADRB1 17 40 CCC[C@@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678775 EI On-Demand Unstable ACE 48 44 CCC[C@@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678775 EI On-Demand Unstable OPRM1 37 41 CCC[C@@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678775 EI On-Demand Unstable OPRD1 29 41 CCC[C@@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678775 EI On-Demand Unstable MME 81 45 CCC[C@@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678775 EI On-Demand Unstable SDH1 0 49 CCC[C@@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678775 EI On-Demand Unstable KCNQ2 26 47 CCC[C@@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678775 EI On-Demand Unstable ACACA 22 42 CCC[C@@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678775 EI On-Demand Unstable NPY1R 23 42 CCC[C@@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678775 EI On-Demand Unstable KLK3 50 34 CCC[C@@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678775 EI On-Demand Unstable CTSB 49 38 CCC[C@@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678775 EI On-Demand Unstable CTSK 39 40 CCC[C@@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678775 EI On-Demand Unstable CAPNS1 59 34 CCC[C@@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678775 EI On-Demand Unstable MMP3 47 43 CCC[C@@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678775 EI On-Demand Unstable GRIA1 56 39 CCC[C@@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678775 EI On-Demand Unstable SOAT1 27 46 CCC[C@@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678775 EI On-Demand Unstable YARS 58 43 CCC[C@@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678775 EI On-Demand Unstable CAPN1 75 43 CCC[C@@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678775 EI On-Demand Unstable CAPN2 106 43 CCC[C@@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678775 EI On-Demand Unstable ACE2 60 39 CCC[C@@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678775 EI On-Demand Unstable NPR 59 35 CCC[C@@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678775 EI On-Demand Unstable SLC15A2 0 40 CCC[C@@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678775 EI On-Demand Unstable GLI1 0 42 CCC[C@@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678775 EI On-Demand Unstable GPR88 0 44 CNC(=O)c1cc(N)ccc1N1CCCC1 ZINC000217678798 BD In-Stock Unstable KCNQ2 72 35 CCC[C@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678864 EI On-Demand Unstable ADRB1 17 40 CCC[C@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678864 EI On-Demand Unstable ACE 48 44 CCC[C@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678864 EI On-Demand Unstable OPRM1 37 41 CCC[C@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678864 EI On-Demand Unstable OPRD1 29 41 CCC[C@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678864 EI On-Demand Unstable MME 81 45 CCC[C@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678864 EI On-Demand Unstable SDH1 0 49 CCC[C@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678864 EI On-Demand Unstable KCNQ2 26 47 CCC[C@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678864 EI On-Demand Unstable ACACA 22 42 CCC[C@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678864 EI On-Demand Unstable NPY1R 23 42 CCC[C@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678864 EI On-Demand Unstable KLK3 50 34 CCC[C@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678864 EI On-Demand Unstable CTSB 49 38 CCC[C@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678864 EI On-Demand Unstable CTSK 39 40 CCC[C@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678864 EI On-Demand Unstable CAPNS1 59 34 CCC[C@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678864 EI On-Demand Unstable MMP3 47 43 CCC[C@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678864 EI On-Demand Unstable GRIA1 56 39 CCC[C@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678864 EI On-Demand Unstable SOAT1 27 46 CCC[C@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678864 EI On-Demand Unstable YARS 58 43 CCC[C@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678864 EI On-Demand Unstable CAPN1 75 43 CCC[C@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678864 EI On-Demand Unstable CAPN2 106 43 CCC[C@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678864 EI On-Demand Unstable ACE2 60 39 CCC[C@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678864 EI On-Demand Unstable NPR 59 35 CCC[C@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678864 EI On-Demand Unstable SLC15A2 0 40 CCC[C@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678864 EI On-Demand Unstable GLI1 0 42 CCC[C@H](C(=O)N[C@@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678864 EI On-Demand Unstable GPR88 0 44 C/C=C(/Cl)c1ccc(OC)cc1 ZINC000217678888 AG For-Sale Unstable CYP1B1 50 39 CCOC(=O)[C@@H]1C[C@@H]1c1ccc(F)cc1F ZINC000217678917 BF On-Demand Unstable PRCP 44 32 CCCNc1ccc(N)cc1C(=O)N(C)C ZINC000217678928 BD In-Stock Unstable CXCR2 54 33 CCCNc1ccc(N)cc1C(=O)N(C)C ZINC000217678928 BD In-Stock Unstable CXCR1 47 33 CCC[C@@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678945 EI On-Demand Unstable ADRB1 17 40 CCC[C@@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678945 EI On-Demand Unstable ACE 48 44 CCC[C@@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678945 EI On-Demand Unstable OPRM1 37 41 CCC[C@@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678945 EI On-Demand Unstable OPRD1 29 41 CCC[C@@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678945 EI On-Demand Unstable MME 81 45 CCC[C@@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678945 EI On-Demand Unstable SDH1 0 49 CCC[C@@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678945 EI On-Demand Unstable KCNQ2 26 47 CCC[C@@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678945 EI On-Demand Unstable ACACA 22 42 CCC[C@@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678945 EI On-Demand Unstable NPY1R 23 42 CCC[C@@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678945 EI On-Demand Unstable KLK3 50 34 CCC[C@@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678945 EI On-Demand Unstable CTSB 49 38 CCC[C@@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678945 EI On-Demand Unstable CTSK 39 40 CCC[C@@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678945 EI On-Demand Unstable CAPNS1 59 34 CCC[C@@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678945 EI On-Demand Unstable MMP3 47 43 CCC[C@@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678945 EI On-Demand Unstable GRIA1 56 39 CCC[C@@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678945 EI On-Demand Unstable SOAT1 27 46 CCC[C@@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678945 EI On-Demand Unstable YARS 58 43 CCC[C@@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678945 EI On-Demand Unstable CAPN1 75 43 CCC[C@@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678945 EI On-Demand Unstable CAPN2 106 43 CCC[C@@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678945 EI On-Demand Unstable ACE2 60 39 CCC[C@@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678945 EI On-Demand Unstable NPR 59 35 CCC[C@@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678945 EI On-Demand Unstable SLC15A2 0 40 CCC[C@@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678945 EI On-Demand Unstable GLI1 0 42 CCC[C@@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217678945 EI On-Demand Unstable GPR88 0 44 COc1ccccc1N(C)C[C@@H](C(=O)O)C(F)(F)F ZINC000217678952 CE For-Sale Unstable SLC6A9 17 40 CCOC(=O)[C@H]1C[C@@H]1c1ccc(F)cc1F ZINC000217678999 BF On-Demand Unstable PRCP 44 32 CCC[C@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217679018 EI On-Demand Unstable ADRB1 17 40 CCC[C@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217679018 EI On-Demand Unstable ACE 48 44 CCC[C@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217679018 EI On-Demand Unstable OPRM1 37 41 CCC[C@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217679018 EI On-Demand Unstable OPRD1 29 41 CCC[C@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217679018 EI On-Demand Unstable MME 81 45 CCC[C@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217679018 EI On-Demand Unstable SDH1 0 49 CCC[C@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217679018 EI On-Demand Unstable KCNQ2 26 47 CCC[C@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217679018 EI On-Demand Unstable ACACA 22 42 CCC[C@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217679018 EI On-Demand Unstable NPY1R 23 42 CCC[C@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217679018 EI On-Demand Unstable KLK3 50 34 CCC[C@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217679018 EI On-Demand Unstable CTSB 49 38 CCC[C@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217679018 EI On-Demand Unstable CTSK 39 40 CCC[C@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217679018 EI On-Demand Unstable CAPNS1 59 34 CCC[C@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217679018 EI On-Demand Unstable MMP3 47 43 CCC[C@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217679018 EI On-Demand Unstable GRIA1 56 39 CCC[C@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217679018 EI On-Demand Unstable SOAT1 27 46 CCC[C@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217679018 EI On-Demand Unstable YARS 58 43 CCC[C@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217679018 EI On-Demand Unstable CAPN1 75 43 CCC[C@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217679018 EI On-Demand Unstable CAPN2 106 43 CCC[C@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217679018 EI On-Demand Unstable ACE2 60 39 CCC[C@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217679018 EI On-Demand Unstable NPR 59 35 CCC[C@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217679018 EI On-Demand Unstable SLC15A2 0 40 CCC[C@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217679018 EI On-Demand Unstable GLI1 0 42 CCC[C@H](C(=O)N[C@H](C)CCc1ccc(O)cc1)c1ccccc1 ZINC000217679018 EI On-Demand Unstable GPR88 0 44 COc1ccc(Cn2ncnc2CCn2c(C)cccc2=O)cc1 ZINC000217679025 DE In-Stock Unstable PROKR1 52 32 COc1ccc(Cn2ncnc2CCn2c(C)cccc2=O)cc1 ZINC000217679025 DE In-Stock Unstable NPBWR1 73 40 COc1ccccc1N(C)C[C@H](C(=O)O)C(F)(F)F ZINC000217679041 CE For-Sale Unstable SLC6A9 17 40 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)/C=C/c1ccc3c(c1)OCO3)C2 ZINC000217679073 GD In-Stock Unstable DYRK2 67 36 CCOC(=O)[C@@H]1C[C@H]1c1ccc(F)cc1F ZINC000217679090 BF On-Demand Unstable PRCP 44 32 CCOc1cccc(CN[C@@H]2CCN3CCCC[C@@H]23)c1O ZINC000217679104 CF On-Demand Unstable HCN1 41 33 CCOc1cccc(CN[C@@H]2CCN3CCCC[C@@H]23)c1O ZINC000217679104 CF On-Demand Unstable HCN4 42 35 Cc1nc(Nc2ccc(Cl)cc2)cc(N2CCC[C@@H](C(=O)O)C2)n1 ZINC000217679133 EG In-Stock Unstable SLC6A1 94 37 Cc1nc(Nc2ccc(Cl)cc2)cc(N2CCC[C@@H](C(=O)O)C2)n1 ZINC000217679133 EG In-Stock Unstable GALR2 52 38 Cc1nc(Nc2ccc(Cl)cc2)cc(N2CCC[C@@H](C(=O)O)C2)n1 ZINC000217679133 EG In-Stock Unstable GPBAR1 30 52 O=C(N[C@@H]1CCOC2(CCOCC2)C1)c1ccccc1N1CCOCC1 ZINC000217679155 FD In-Stock Unstable HTR3A 16 41 COc1cccc(N(C)C[C@@H](C(=O)O)C(F)(F)F)c1 ZINC000217679167 CE For-Sale Unstable MTNR1A 34 43 COc1cccc(N(C)C[C@@H](C(=O)O)C(F)(F)F)c1 ZINC000217679167 CE For-Sale Unstable MTNR1B 35 43 COc1cccc(N(C)C[C@@H](C(=O)O)C(F)(F)F)c1 ZINC000217679167 CE For-Sale Unstable HSD17B2 28 45 CCOC(=O)[C@H]1C[C@H]1c1ccc(F)cc1F ZINC000217679174 BF On-Demand Unstable PRCP 44 32 CCOc1cccc(CN[C@H]2CCN3CCCC[C@@H]23)c1O ZINC000217679183 CF On-Demand Unstable HCN1 41 33 CCOc1cccc(CN[C@H]2CCN3CCCC[C@@H]23)c1O ZINC000217679183 CF On-Demand Unstable HCN4 42 35 CSC[C@](C)(O)CNC(=O)/C=C/c1ccc(C)cc1 ZINC000217679220 CE On-Demand Unstable HDAC8 15 40 CSC[C@](C)(O)CNC(=O)/C=C/c1ccc(C)cc1 ZINC000217679220 CE On-Demand Unstable HDAC1 15 40 Cc1nc(Nc2ccc(Cl)cc2)cc(N2CCC[C@H](C(=O)O)C2)n1 ZINC000217679236 EG In-Stock Unstable SLC6A1 94 37 Cc1nc(Nc2ccc(Cl)cc2)cc(N2CCC[C@H](C(=O)O)C2)n1 ZINC000217679236 EG In-Stock Unstable GALR2 52 38 Cc1nc(Nc2ccc(Cl)cc2)cc(N2CCC[C@H](C(=O)O)C2)n1 ZINC000217679236 EG In-Stock Unstable GPBAR1 30 52 O=C(N[C@H]1CCOC2(CCOCC2)C1)c1ccccc1N1CCOCC1 ZINC000217679244 FD In-Stock Unstable HTR3A 16 41 COC(=O)[C@@H](O)CNC(=O)c1cc(Cl)ccc1O ZINC000217679247 CC On-Demand Unstable KCNMA1 29 48 COc1cccc(N(C)C[C@H](C(=O)O)C(F)(F)F)c1 ZINC000217679261 CE For-Sale Unstable MTNR1A 34 43 COc1cccc(N(C)C[C@H](C(=O)O)C(F)(F)F)c1 ZINC000217679261 CE For-Sale Unstable MTNR1B 35 43 COc1cccc(N(C)C[C@H](C(=O)O)C(F)(F)F)c1 ZINC000217679261 CE For-Sale Unstable HSD17B2 28 45 CCC1CCN(C(=O)c2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217679278 CG For-Sale Unstable GRIN2B 21 44 CCC1CCN(C(=O)c2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217679278 CG For-Sale Unstable L3MBTL1 0 41 CCC1CCN(C(=O)c2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217679278 CG For-Sale Unstable L3MBTL3 91 41 CCC1CCN(C(=O)c2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217679278 CG For-Sale Unstable MBTD1 0 40 CCC1CCN(C(=O)c2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217679278 CG For-Sale Unstable GPR183 0 48 C[C@@H](N[C@@H]1CCN2CCCC[C@@H]12)c1ccccc1F ZINC000217679309 CG For-Sale Unstable SLC18A3 40 36 COC(=O)[C@H](O)CNC(=O)c1cc(Cl)ccc1O ZINC000217679331 CC For-Sale Unstable KCNMA1 29 48 COC(=O)[C@H](O)CNC(=O)c1cc(Cl)ccc1O ZINC000217679331 CC For-Sale Unstable U38 0 41 COC(=O)[C@H](O)CNC(=O)c1cc(Cl)ccc1O ZINC000217679331 CC For-Sale Unstable TMPRSS4 0 42 CCCCN(CCCC)C(=O)N/C=C/c1ccccc1C ZINC000217679332 CJ For-Sale Unstable TSPO 30 40 N#Cc1ccc(S(=O)(=O)NCCF)cc1 ZINC000217679350 BC On-Demand Unstable TBXA2R 22 43 COc1ccc2occ([C@@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(O)cc6)oc5c43)c(=O)c2c1 ZINC000217679354 JI In-Stock Unstable ALDH2 56 40 COc1ccc2occ([C@@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(O)cc6)oc5c43)c(=O)c2c1 ZINC000217679354 JI In-Stock Unstable AKR1B1 0 41 COc1ccc2occ([C@@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(O)cc6)oc5c43)c(=O)c2c1 ZINC000217679354 JI In-Stock Unstable CYP1B1 40 42 COc1ccc2occ([C@@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(O)cc6)oc5c43)c(=O)c2c1 ZINC000217679354 JI In-Stock Unstable CYP1A1 33 42 COc1ccc2occ([C@@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(O)cc6)oc5c43)c(=O)c2c1 ZINC000217679354 JI In-Stock Unstable CYP1A2 24 42 O=C(O)/C=C\c1cccc(S(=O)(=O)NC2CCCCC2)c1 ZINC000217679368 DE For-Sale Unstable HDAC8 15 50 O=C(O)/C=C\c1cccc(S(=O)(=O)NC2CCCCC2)c1 ZINC000217679368 DE For-Sale Unstable SFRP1 128 38 O=C(O)/C=C\c1cccc(S(=O)(=O)NC2CCCCC2)c1 ZINC000217679368 DE For-Sale Unstable WNT3 87 38 O=C(O)/C=C\c1cccc(S(=O)(=O)NC2CCCCC2)c1 ZINC000217679368 DE For-Sale Unstable BRD4 0 46 CCCn1c(-c2ccccc2)ncc(C(=O)O)c1=O ZINC000217679371 CE In-Stock Unstable ADORA1 28 42 CCCn1c(-c2ccccc2)ncc(C(=O)O)c1=O ZINC000217679371 CE In-Stock Unstable ADORA2A 26 43 CCCn1c(-c2ccccc2)ncc(C(=O)O)c1=O ZINC000217679371 CE In-Stock Unstable ADORA2B 49 43 CCCn1c(-c2ccccc2)ncc(C(=O)O)c1=O ZINC000217679371 CE In-Stock Unstable CTRA_BOVIN 42 32 CCCn1c(-c2ccccc2)ncc(C(=O)O)c1=O ZINC000217679371 CE In-Stock Unstable AGTR1B 47 43 CCCn1c(-c2ccccc2)ncc(C(=O)O)c1=O ZINC000217679371 CE In-Stock Unstable CTRC 45 38 O=C(NC[C@@H]1CCCO1)[C@@H]1CC[C@@H](CNC(=O)[C@@H]2Cc3ccccc3CN2)CC1 ZINC000217679437 GD In-Stock Unstable PDE8B 21 40 COc1ccc2occ([C@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(O)cc6)oc5c43)c(=O)c2c1 ZINC000217679443 JI In-Stock Unstable ALDH2 56 40 COc1ccc2occ([C@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(O)cc6)oc5c43)c(=O)c2c1 ZINC000217679443 JI In-Stock Unstable AKR1B1 0 41 COc1ccc2occ([C@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(O)cc6)oc5c43)c(=O)c2c1 ZINC000217679443 JI In-Stock Unstable CYP1B1 40 42 COc1ccc2occ([C@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(O)cc6)oc5c43)c(=O)c2c1 ZINC000217679443 JI In-Stock Unstable CYP1A1 33 42 COc1ccc2occ([C@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(O)cc6)oc5c43)c(=O)c2c1 ZINC000217679443 JI In-Stock Unstable CYP1A2 24 42 CCCNS(=O)(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217679444 CD For-Sale Unstable AKR1C3 15 42 C[C@@H](N[C@H]1CCN2CCCC[C@@H]12)c1ccccc1F ZINC000217679486 CG For-Sale Unstable SLC18A3 40 36 O=C(O)c1cnc(-c2ccccc2)n(C2CC2)c1=O ZINC000217679500 CD In-Stock Unstable NS5B 0 41 O=C(NC[C@H]1CCCO1)[C@@H]1CC[C@@H](CNC(=O)[C@@H]2Cc3ccccc3CN2)CC1 ZINC000217679529 GD In-Stock Unstable PDE8B 21 40 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable ADRB2 20 50 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable ADRB1 29 47 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable ACE 58 46 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable OPRM1 46 41 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable OPRD1 42 41 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable ADRB3 36 47 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable MME 97 48 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable ANPEP 54 39 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable SDH1 0 49 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable NPY1R 39 53 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable KLK3 56 35 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable CTSB 54 45 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable PAPA1_CARPA 45 33 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable CTSK 33 40 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable CTSL 44 45 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable ACACB 15 42 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable CAPNS1 61 34 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable MMP3 51 45 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable MMP8 17 47 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable GRIA1 53 41 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable SOAT1 18 63 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable HDAC5 15 45 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable YARS 61 46 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable CTSS 18 45 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable CAPN1 68 46 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable MMP9 15 47 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable CAPN2 79 41 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable ACE2 63 38 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable LAP3 41 39 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable MMP1 21 45 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable POL 0 40 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable NPR 57 33 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable SLC15A2 0 43 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679542 FJ On-Demand Unstable GLI1 0 43 COc1cc([C@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2oc(C)cc(=O)c2O)cc2c1OCO2 ZINC000217679569 KH In-Stock Unstable RORC 46 35 C[C@@H](C(=O)Nc1ccccc1)N1CCC[C@@H](O)C1 ZINC000217679577 BD In-Stock Unstable ACE 30 41 C[C@@H](C(=O)Nc1ccccc1)N1CCC[C@@H](O)C1 ZINC000217679577 BD In-Stock Unstable KCNQ2 16 40 C[C@@H](C(=O)Nc1ccccc1)N1CCC[C@@H](O)C1 ZINC000217679577 BD In-Stock Unstable XIAP 43 35 C[C@@H](C(=O)Nc1ccccc1)N1CCC[C@@H](O)C1 ZINC000217679577 BD In-Stock Unstable BIRC2 56 38 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable ADRB2 20 50 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable ADRB1 29 47 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable ACE 58 46 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable OPRM1 46 41 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable OPRD1 42 41 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable ADRB3 36 47 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable MME 97 48 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable ANPEP 54 39 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable SDH1 0 49 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable NPY1R 39 53 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable KLK3 56 35 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable CTSB 54 45 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable PAPA1_CARPA 45 33 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable CTSK 33 40 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable CTSL 44 45 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable ACACB 15 42 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable CAPNS1 61 34 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable MMP3 51 45 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable MMP8 17 47 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable GRIA1 53 41 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable SOAT1 18 63 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable HDAC5 15 45 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable YARS 61 46 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable CTSS 18 45 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable CAPN1 68 46 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable MMP9 15 47 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable CAPN2 79 41 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable ACE2 63 38 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable LAP3 41 39 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable MMP1 21 45 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable POL 0 40 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable NPR 57 33 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable SLC15A2 0 43 C[C@H](CCc1ccc(O)cc1)NC(=O)C(c1ccccc1)c1ccccc1 ZINC000217679632 FJ On-Demand Unstable GLI1 0 43 COc1cc([C@@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2oc(C)cc(=O)c2O)cc2c1OCO2 ZINC000217679667 KH In-Stock Unstable RORC 46 35 CCOC(=O)[C@@H](c1ccccc1)N1CCC[C@@H](O)C1 ZINC000217679709 CD On-Demand Unstable CHRM1 26 51 CCOC(=O)[C@@H](c1ccccc1)N1CCC[C@@H](O)C1 ZINC000217679709 CD On-Demand Unstable SLC6A1 84 40 CCOC(=O)[C@@H](c1ccccc1)N1CCC[C@@H](O)C1 ZINC000217679709 CD On-Demand Unstable P2RY12 51 38 CCOC(=O)[C@@H](c1ccccc1)N1CCC[C@@H](O)C1 ZINC000217679709 CD On-Demand Unstable CHRM3 24 51 CCOC(=O)[C@@H](c1ccccc1)N1CCC[C@@H](O)C1 ZINC000217679709 CD On-Demand Unstable NPY2R 24 40 CCOC(=O)[C@@H](c1ccccc1)N1CCC[C@@H](O)C1 ZINC000217679709 CD On-Demand Unstable AMY2 44 31 CCOC(=O)[C@@H](c1ccccc1)N1CCC[C@@H](O)C1 ZINC000217679709 CD On-Demand Unstable FKBP12.6 0 40 CC[C@H](C)[C@@H](N[C@H](C)CC)C(N)=O ZINC000217679711 AD For-Sale Unstable LASB 0 45 CC[C@H](C)[C@@H](N[C@H](C)CC)C(N)=O ZINC000217679711 AD For-Sale Unstable SPSB2 0 41 COc1cc(C=O)ccc1NC(=O)OC(C)(C)C ZINC000217679739 CF For-Sale Unstable TUBB1 41 33 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(C)(C)Oc1ccc(Cl)cc1 ZINC000217679749 FI On-Demand Unstable ADRB1 28 42 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(C)(C)Oc1ccc(Cl)cc1 ZINC000217679749 FI On-Demand Unstable AVPR1A 20 40 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(C)(C)Oc1ccc(Cl)cc1 ZINC000217679749 FI On-Demand Unstable ADRB3 23 46 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(C)(C)Oc1ccc(Cl)cc1 ZINC000217679749 FI On-Demand Unstable ACACA 23 40 C[C@@H](CCc1ccc(O)cc1)NC(=O)C(C)(C)Oc1ccc(Cl)cc1 ZINC000217679749 FI On-Demand Unstable GRIA1 46 37 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)NCc3cccn3C(C)C)[C@H]21 ZINC000217679780 JH In-Stock Unstable TSHR 41 31 CC[C@H](C)[C@H](N[C@H](C)CC)C(N)=O ZINC000217679799 AD For-Sale Unstable LASB 0 45 CC[C@H](C)[C@H](N[C@H](C)CC)C(N)=O ZINC000217679799 AD For-Sale Unstable SPSB2 0 41 CCOC(=O)[C@H](c1ccccc1)N1CCC[C@@H](O)C1 ZINC000217679801 CD On-Demand Unstable CHRM1 26 51 CCOC(=O)[C@H](c1ccccc1)N1CCC[C@@H](O)C1 ZINC000217679801 CD On-Demand Unstable SLC6A1 84 40 CCOC(=O)[C@H](c1ccccc1)N1CCC[C@@H](O)C1 ZINC000217679801 CD On-Demand Unstable OPRM1 0 44 CCOC(=O)[C@H](c1ccccc1)N1CCC[C@@H](O)C1 ZINC000217679801 CD On-Demand Unstable OPRK1 0 40 CCOC(=O)[C@H](c1ccccc1)N1CCC[C@@H](O)C1 ZINC000217679801 CD On-Demand Unstable P2RY12 51 38 CCOC(=O)[C@H](c1ccccc1)N1CCC[C@@H](O)C1 ZINC000217679801 CD On-Demand Unstable CHRM3 24 51 CCOC(=O)[C@H](c1ccccc1)N1CCC[C@@H](O)C1 ZINC000217679801 CD On-Demand Unstable NPY2R 24 40 CCOC(=O)[C@H](c1ccccc1)N1CCC[C@@H](O)C1 ZINC000217679801 CD On-Demand Unstable AMY2 44 31 CCOC(=O)[C@H](c1ccccc1)N1CCC[C@@H](O)C1 ZINC000217679801 CD On-Demand Unstable FKBP12.6 0 40 C[C@H](CCc1ccc(O)cc1)NC(=O)C(C)(C)Oc1ccc(Cl)cc1 ZINC000217679833 FI On-Demand Unstable ADRB1 28 42 C[C@H](CCc1ccc(O)cc1)NC(=O)C(C)(C)Oc1ccc(Cl)cc1 ZINC000217679833 FI On-Demand Unstable AVPR1A 20 40 C[C@H](CCc1ccc(O)cc1)NC(=O)C(C)(C)Oc1ccc(Cl)cc1 ZINC000217679833 FI On-Demand Unstable ADRB3 23 46 C[C@H](CCc1ccc(O)cc1)NC(=O)C(C)(C)Oc1ccc(Cl)cc1 ZINC000217679833 FI On-Demand Unstable ACACA 23 40 C[C@H](CCc1ccc(O)cc1)NC(=O)C(C)(C)Oc1ccc(Cl)cc1 ZINC000217679833 FI On-Demand Unstable GRIA1 46 37 O=C(NC1CCCCC1)[C@@H]1C[C@H]2C[C@H]2N1 ZINC000217679848 BD On-Demand Unstable EPHX2 29 40 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)NCc3cccn3C(C)C)[C@@H]21 ZINC000217679869 JH In-Stock Unstable TSHR 41 31 COC(=O)[C@@H](O)CNC(=O)CCc1cccc(OC)c1 ZINC000217679877 CC On-Demand Unstable DRD4 40 32 COC(=O)[C@@H](O)CNC(=O)CCc1cccc(OC)c1 ZINC000217679877 CC On-Demand Unstable MTNR1A 63 51 COC(=O)[C@@H](O)CNC(=O)CCc1cccc(OC)c1 ZINC000217679877 CC On-Demand Unstable MTNR1B 61 51 COC(=O)[C@@H](O)CNC(=O)CCc1cccc(OC)c1 ZINC000217679877 CC On-Demand Unstable CRTM 46 35 O=C(O)/C=C\c1cccc(S(=O)(=O)N2CCCCCC2)c1 ZINC000217679893 DE For-Sale Unstable LPL 45 38 O=C(O)/C=C\c1cccc(S(=O)(=O)N2CCCCCC2)c1 ZINC000217679893 DE For-Sale Unstable HDAC8 22 44 O=C(O)/C=C\c1cccc(S(=O)(=O)N2CCCCCC2)c1 ZINC000217679893 DE For-Sale Unstable AKR1C3 68 43 O=C(O)/C=C\c1cccc(S(=O)(=O)N2CCCCCC2)c1 ZINC000217679893 DE For-Sale Unstable AKR1C1 24 42 COC(=O)[C@H](O)CNC(=O)CCc1cccc(OC)c1 ZINC000217679948 CC On-Demand Unstable DRD4 40 32 COC(=O)[C@H](O)CNC(=O)CCc1cccc(OC)c1 ZINC000217679948 CC On-Demand Unstable MTNR1A 63 51 COC(=O)[C@H](O)CNC(=O)CCc1cccc(OC)c1 ZINC000217679948 CC On-Demand Unstable MTNR1B 61 51 COC(=O)[C@H](O)CNC(=O)CCc1cccc(OC)c1 ZINC000217679948 CC On-Demand Unstable CRTM 46 35 C[C@@H]1CN(S(=O)(=O)c2cccc(/C=C\C(=O)O)c2)CCO1 ZINC000217679982 DD For-Sale Unstable AKR1C3 54 36 COc1cccc(CN[C@@H]2CCN3CCCC[C@@H]23)c1O ZINC000217680063 CE On-Demand Unstable TACR3 25 40 C[C@H]1CN(S(=O)(=O)c2cccc(/C=C\C(=O)O)c2)CCO1 ZINC000217680064 DD For-Sale Unstable AKR1C3 54 36 CCN(C[C@@H](C(=O)O)C(F)(F)F)c1ccc(C)cc1 ZINC000217680148 CG For-Sale Unstable NR1H2 0 41 COc1cccc(CN[C@H]2CCN3CCCC[C@@H]23)c1O ZINC000217680157 CE On-Demand Unstable TACR3 25 40 O=C(O)/C=C\c1cccc(S(=O)(=O)Nc2cccnc2)c1 ZINC000217680158 DD For-Sale Anodyne TBXAS1 26 43 O=C(O)/C=C\c1cccc(S(=O)(=O)Nc2cccnc2)c1 ZINC000217680158 DD For-Sale Anodyne HDAC1 0 60 O=C(O)/C=C\c1cccc(S(=O)(=O)Nc2cccnc2)c1 ZINC000217680158 DD For-Sale Anodyne RHOA 0 44 O=C(O)/C=C\c1cccc(S(=O)(=O)Nc2cccnc2)c1 ZINC000217680158 DD For-Sale Anodyne NAMPT 31 48 CCOc1ccccc1OCC(=O)NC[C@@](C)(O)CSC ZINC000217680161 DD On-Demand Unstable HCN1 41 31 CCOc1ccccc1OCC(=O)NC[C@@](C)(O)CSC ZINC000217680161 DD On-Demand Unstable HCN4 40 31 COCCn1ccc2c(NC(=O)CC/C(C)=C/Cc3c(O)c4c(c(C)c3OC)COC4=O)cccc21 ZINC000217680191 JJ In-Stock Unstable IMPDH1 0 68 COCCn1ccc2c(NC(=O)CC/C(C)=C/Cc3c(O)c4c(c(C)c3OC)COC4=O)cccc21 ZINC000217680191 JJ In-Stock Unstable IMPDH2 0 68 CCN(C[C@H](C(=O)O)C(F)(F)F)c1ccc(C)cc1 ZINC000217680235 CG For-Sale Unstable NR1H2 0 41 CCOc1ccccc1OCC(=O)NC[C@](C)(O)CSC ZINC000217680245 DD On-Demand Unstable HCN1 41 31 CCOc1ccccc1OCC(=O)NC[C@](C)(O)CSC ZINC000217680245 DD On-Demand Unstable HCN4 40 31 Cc1cc(S(=O)(=O)NCCC(C)C)ccc1/C=C\C(=O)O ZINC000217680255 DE For-Sale Unstable LEF 52 35 COc1ccc(C(=O)N2CCC[C@@H](c3nc(C)n[nH]3)C2)o1 ZINC000217680294 CD In-Stock Unstable GRM3 15 41 O=C(CN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCc1cccnc1 ZINC000217680310 GF In-Stock Unstable SCN9A 0 45 O=C(CN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCc1cccnc1 ZINC000217680310 GF In-Stock Unstable NAMPT 47 38 CCC[C@@H](C)N[C@@H](C(=O)OCC)c1ccccc1 ZINC000217680336 BG On-Demand Unstable CAPN2 59 35 CCC[C@@H](C)N[C@@H](C(=O)OCC)c1ccccc1 ZINC000217680336 BG On-Demand Unstable GPR88 0 40 COc1ccc(C(=O)N2CCC[C@H](c3nc(C)n[nH]3)C2)o1 ZINC000217680376 CD In-Stock Unstable GRM3 15 41 O=C(CN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCc1cccnc1 ZINC000217680385 GF In-Stock Unstable SCN9A 0 45 O=C(CN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCc1cccnc1 ZINC000217680385 GF In-Stock Unstable NAMPT 41 35 CCC[C@H](C)N[C@@H](C(=O)OCC)c1ccccc1 ZINC000217680426 BG On-Demand Unstable CAPN2 59 35 CCC[C@H](C)N[C@@H](C(=O)OCC)c1ccccc1 ZINC000217680426 BG On-Demand Unstable GPR88 0 40 COC(=O)[C@@H](O)CNC(=O)Cc1ccc(OC(F)F)cc1 ZINC000217680446 DC On-Demand Unstable CA9 19 40 COc1cc2c(cc1OC)CC(=O)N(CC(=O)NCCN(C)C)C=C2 ZINC000217680498 EC In-Stock Unstable HCN2 0 44 CCC[C@@H](C)N[C@H](C(=O)OCC)c1ccccc1 ZINC000217680511 BG On-Demand Unstable CAPN2 59 35 CCC[C@@H](C)N[C@H](C(=O)OCC)c1ccccc1 ZINC000217680511 BG On-Demand Unstable GPR88 0 40 COC(=O)[C@H](O)CNC(=O)Cc1ccc(OC(F)F)cc1 ZINC000217680533 DC On-Demand Unstable CA9 19 40 Cc1cccc(N(C)C[C@@H](C(=O)O)C(F)(F)F)c1 ZINC000217680537 CF For-Sale Unstable HSD17B2 15 42 Cc1ccccc1/C=C/NC(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000217680592 EK For-Sale Unstable EPHX1 0 43 Cc1ccccc1/C=C/NC(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000217680592 EK For-Sale Unstable P95276_MYCTO 0 43 COc1ccc2c(c1OC)C(=O)O[C@@H]2CC(=O)Nc1ccc(C(=O)O)cc1 ZINC000217680596 FF In-Stock Unstable FDFT1 15 41 CCC[C@H](C)N[C@H](C(=O)OCC)c1ccccc1 ZINC000217680602 BG On-Demand Unstable CAPN2 59 35 CCC[C@H](C)N[C@H](C(=O)OCC)c1ccccc1 ZINC000217680602 BG On-Demand Unstable GPR88 0 40 Cc1cccc(N(C)C[C@H](C(=O)O)C(F)(F)F)c1 ZINC000217680623 CF For-Sale Unstable HSD17B2 15 42 COc1ccc2c(c1OC)C(=O)O[C@H]2CC(=O)Nc1ccc(C(=O)O)cc1 ZINC000217680676 FF In-Stock Unstable FDFT1 15 41 CSC[C@@](C)(O)CNC(=O)CSc1ccc([N+](=O)[O-])cc1 ZINC000217680744 ED On-Demand Unstable FAS 26 42 Cc1ccnc(NC(=O)c2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217680787 CF For-Sale Unstable KCNK3 54 38 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)CCc1ccc(Cl)c(C(F)(F)F)c1)C2 ZINC000217680788 IG In-Stock Unstable Q8MMZ8_EIMTE 25 40 COc1cc2c(c(OC)c1OC)-c1ccc(N3C[C@@]4(C)C[C@@H]3CC(C)(C)C4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217680812 KK In-Stock Unstable AVPR1A 20 40 COc1cc2c(c(OC)c1OC)-c1ccc(N3C[C@@]4(C)C[C@@H]3CC(C)(C)C4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217680812 KK In-Stock Unstable TUBA1A 18 64 CSC[C@](C)(O)CNC(=O)CSc1ccc([N+](=O)[O-])cc1 ZINC000217680825 ED On-Demand Unstable FAS 26 42 Cc1cccc(NC(=O)N/C=C/c2ccccc2C)n1 ZINC000217680826 CG For-Sale Unstable GRM5 18 47 Cc1cccc(NC(=O)N/C=C/c2ccccc2C)n1 ZINC000217680826 CG For-Sale Unstable SORT1 16 40 CCOC(=O)[C@@H](NC[C@@H](C)O)c1ccccc1 ZINC000217680828 BD On-Demand Unstable CAPN2 42 35 CCOC(=O)[C@@H](NC[C@@H](C)O)c1ccccc1 ZINC000217680828 BD On-Demand Unstable METAP2 22 42 COc1ccc(NC(=O)OC(C)(C)C)cc1C=O ZINC000217680830 CF For-Sale Unstable ENPP1 55 31 CCOC(=O)[C@H](NC[C@@H](C)O)c1ccccc1 ZINC000217680908 BD On-Demand Unstable CAPN2 42 35 CCOC(=O)[C@H](NC[C@@H](C)O)c1ccccc1 ZINC000217680908 BD On-Demand Unstable METAP2 22 42 CSCC[C@@H](NC(N)=O)C(=O)NC[C@@](C)(O)CSC ZINC000217680939 DC On-Demand Unstable LASB 0 40 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCCc1ccc(O)cc1 ZINC000217680954 IE In-Stock Unstable TACR1 18 40 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCCc1ccc(O)cc1 ZINC000217680954 IE In-Stock Unstable CCKAR 22 43 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCCc1ccc(O)cc1 ZINC000217680954 IE In-Stock Unstable BRS3 27 42 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCCc1ccc(O)cc1 ZINC000217680954 IE In-Stock Unstable MC5R 34 42 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCCc1ccc(O)cc1 ZINC000217680954 IE In-Stock Unstable CCKBR 21 43 CCOC(=O)[C@@H](NC[C@H](C)O)c1ccccc1 ZINC000217680997 BD On-Demand Unstable CAPN2 42 35 CCOC(=O)[C@@H](NC[C@H](C)O)c1ccccc1 ZINC000217680997 BD On-Demand Unstable METAP2 22 42 CSCC[C@H](NC(N)=O)C(=O)NC[C@@](C)(O)CSC ZINC000217681016 DC On-Demand Unstable LASB 0 40 CC[C@@H](CCO)NC(=O)CCC(=O)O ZINC000217681045 BC For-Sale Unstable PLA2G2C 0 46 CC[C@@H](CCO)NC(=O)CCC(=O)O ZINC000217681045 BC For-Sale Unstable GNPAT 0 40 CC[C@@H](CCO)NC(=O)CCC(=O)O ZINC000217681045 BC For-Sale Unstable Q6UB75_PIG 0 43 CC[C@@H](CCO)NC(=O)CCC(=O)O ZINC000217681045 BC For-Sale Unstable KDM2A 40 39 O=C(CC[C@@H]1NC(=O)N(CCc2ccccc2)C1=O)NCCc1ccc(O)cc1 ZINC000217681048 GD In-Stock Unstable NCE103 18 41 O=C(CC[C@@H]1NC(=O)N(CCc2ccccc2)C1=O)NCCc1ccc(O)cc1 ZINC000217681048 GD In-Stock Unstable CAN2 0 41 CCOC(=O)[C@H](NC[C@H](C)O)c1ccccc1 ZINC000217681093 BD On-Demand Unstable CAPN2 42 35 CCOC(=O)[C@H](NC[C@H](C)O)c1ccccc1 ZINC000217681093 BD On-Demand Unstable METAP2 22 42 CSCC[C@@H](NC(N)=O)C(=O)NC[C@](C)(O)CSC ZINC000217681106 DC On-Demand Unstable LASB 0 40 CC[C@H](CCO)NC(=O)CCC(=O)O ZINC000217681130 BC For-Sale Unstable PLA2G2C 0 46 CC[C@H](CCO)NC(=O)CCC(=O)O ZINC000217681130 BC For-Sale Unstable GNPAT 0 40 CC[C@H](CCO)NC(=O)CCC(=O)O ZINC000217681130 BC For-Sale Unstable Q6UB75_PIG 0 43 CC[C@H](CCO)NC(=O)CCC(=O)O ZINC000217681130 BC For-Sale Unstable KDM2A 40 39 Cc1ccccc1/C=C/NC(=O)Nc1cccnc1 ZINC000217681186 CG For-Sale Unstable NAMPT 29 46 CSCC[C@H](NC(N)=O)C(=O)NC[C@](C)(O)CSC ZINC000217681201 DC On-Demand Unstable LASB 0 40 CC[C@@H](CCO)NC(=O)CCCCC(=O)O ZINC000217681250 BC On-Demand Unstable PLA2G2C 0 55 CC[C@@H](CCO)NC(=O)CCCCC(=O)O ZINC000217681250 BC On-Demand Unstable Q6UB75_PIG 0 54 CC[C@@H](CCO)NC(=O)CCCCC(=O)O ZINC000217681250 BC On-Demand Unstable SLC22A20 0 41 CC[C@@H](CCO)NC(=O)CCCCC(=O)O ZINC000217681250 BC On-Demand Unstable NOD1 60 40 CC[C@@H](CCO)NC(=O)CCCCC(=O)O ZINC000217681250 BC On-Demand Unstable COL4A3BP 0 45 CCN(CC)C(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217681292 CE For-Sale Unstable OPRD1 28 40 CCN(CC)C(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217681292 CE For-Sale Unstable TNFRSF1A 29 42 CCN(CC)C(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217681292 CE For-Sale Unstable ACKR3 44 34 CC[C@H](CCO)NC(=O)CCCCC(=O)O ZINC000217681329 BC On-Demand Unstable PLA2G2C 0 55 CC[C@H](CCO)NC(=O)CCCCC(=O)O ZINC000217681329 BC On-Demand Unstable Q6UB75_PIG 0 54 CC[C@H](CCO)NC(=O)CCCCC(=O)O ZINC000217681329 BC On-Demand Unstable SLC22A20 0 41 CC[C@H](CCO)NC(=O)CCCCC(=O)O ZINC000217681329 BC On-Demand Unstable NOD1 60 40 CC[C@H](CCO)NC(=O)CCCCC(=O)O ZINC000217681329 BC On-Demand Unstable COL4A3BP 0 45 C[C@@H]1CCCN(C(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217681374 CF For-Sale Unstable PREP 34 42 C[C@@H]1CCCN(C(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217681374 CF For-Sale Unstable L3MBTL3 43 40 C[C@@H]1CCCN(C(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217681374 CF For-Sale Unstable HPGD 26 48 COc1ccc(CNC(=O)CCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@H]23)cc1 ZINC000217681383 IH In-Stock Unstable HTR7 27 45 COc1ccc(CNC(=O)CCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@H]23)cc1 ZINC000217681383 IH In-Stock Unstable SCN9A 0 52 COc1ccc(CNC(=O)CCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@H]23)cc1 ZINC000217681383 IH In-Stock Unstable PROKR1 47 32 CCC[C@@H]1CC[C@@H](N)[C@@H](CCc2ccccc2[N+](=O)[O-])C1 ZINC000217681417 CI For-Sale Unstable COLA 74 33 COc1ccc(CNC(=O)CCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@@H]23)cc1 ZINC000217681466 IH In-Stock Unstable HTR7 27 45 COc1ccc(CNC(=O)CCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@@H]23)cc1 ZINC000217681466 IH In-Stock Unstable SCN9A 0 52 COc1ccc(CNC(=O)CCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@@H]23)cc1 ZINC000217681466 IH In-Stock Unstable PROKR1 47 32 C[C@H]1CCCN(C(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217681467 CF For-Sale Unstable PREP 34 42 C[C@H]1CCCN(C(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217681467 CF For-Sale Unstable L3MBTL3 43 40 C[C@H]1CCCN(C(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217681467 CF For-Sale Unstable HPGD 26 48 CCC[C@H]1CC[C@@H](N)[C@@H](CCc2ccccc2[N+](=O)[O-])C1 ZINC000217681495 CI For-Sale Unstable COLA 74 33 CCN(C[C@@H](C(=O)O)C(F)(F)F)c1ccc(F)cc1 ZINC000217681504 CF For-Sale Unstable NR1H2 0 41 CCC[C@@H]1CC[C@H](N)[C@@H](CCc2ccccc2[N+](=O)[O-])C1 ZINC000217681589 CI For-Sale Unstable COLA 74 33 CCN(C[C@H](C(=O)O)C(F)(F)F)c1ccc(F)cc1 ZINC000217681598 CF For-Sale Unstable NR1H2 0 41 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)c1cccc(OCc3ccccc3)c1)C2 ZINC000217681619 HF In-Stock Unstable PLG 19 46 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)c1cccc(OCc3ccccc3)c1)C2 ZINC000217681619 HF In-Stock Unstable DRD4 41 32 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)c1cccc(OCc3ccccc3)c1)C2 ZINC000217681619 HF In-Stock Unstable HTR3A 15 43 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)c1cccc(OCc3ccccc3)c1)C2 ZINC000217681619 HF In-Stock Unstable KCNH2 43 41 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)c1cccc(OCc3ccccc3)c1)C2 ZINC000217681619 HF In-Stock Unstable F10 15 46 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)c1cccc(OCc3ccccc3)c1)C2 ZINC000217681619 HF In-Stock Unstable LTA4H 17 43 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)c1cccc(OCc3ccccc3)c1)C2 ZINC000217681619 HF In-Stock Unstable EDNRA 0 40 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)c1cccc(OCc3ccccc3)c1)C2 ZINC000217681619 HF In-Stock Unstable MMP26 0 42 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)c1cccc(OCc3ccccc3)c1)C2 ZINC000217681619 HF In-Stock Unstable TRY2_BOVIN 47 34 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)c1cccc(OCc3ccccc3)c1)C2 ZINC000217681619 HF In-Stock Unstable ADAM17 29 40 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)c1cccc(OCc3ccccc3)c1)C2 ZINC000217681619 HF In-Stock Unstable MMP15 0 42 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)c1cccc(OCc3ccccc3)c1)C2 ZINC000217681619 HF In-Stock Unstable MMP16 0 42 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)c1cccc(OCc3ccccc3)c1)C2 ZINC000217681619 HF In-Stock Unstable GRM5 15 43 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)c1cccc(OCc3ccccc3)c1)C2 ZINC000217681619 HF In-Stock Unstable GHSR 15 41 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)c1cccc(OCc3ccccc3)c1)C2 ZINC000217681619 HF In-Stock Unstable SLC6A5 41 46 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)c1cccc(OCc3ccccc3)c1)C2 ZINC000217681619 HF In-Stock Unstable ST14 40 46 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)c1cccc(OCc3ccccc3)c1)C2 ZINC000217681619 HF In-Stock Unstable ADAMTS4 29 40 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)c1cccc(OCc3ccccc3)c1)C2 ZINC000217681619 HF In-Stock Unstable MCHR1 19 43 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)c1cccc(OCc3ccccc3)c1)C2 ZINC000217681619 HF In-Stock Unstable SENP1 0 40 O=C(c1ccc(=O)n(Cc2ccccc2Cl)c1)N1CCN(C(=O)[C@@H]2CCCO2)CC1 ZINC000217681631 IE On-Demand Unstable L3MBTL3 49 35 CCOC(=O)[C@@H](Nc1cccc(CC)c1)c1ccccc1 ZINC000217681670 CH On-Demand Unstable CAPN2 62 33 CCOC(=O)[C@@H](Nc1cccc(CC)c1)c1ccccc1 ZINC000217681670 CH On-Demand Unstable NPR 42 33 CCOC(=O)[C@@H](Nc1cccc(CC)c1)c1ccccc1 ZINC000217681670 CH On-Demand Unstable PPASE1 0 50 CCOC(=O)[C@@H](Nc1cccc(CC)c1)c1ccccc1 ZINC000217681670 CH On-Demand Unstable PDS 46 37 CCC[C@H]1CC[C@H](N)[C@@H](CCc2ccccc2[N+](=O)[O-])C1 ZINC000217681672 CI For-Sale Unstable COLA 74 33 O=C(c1ccc(=O)n(Cc2ccccc2Cl)c1)N1CCN(C(=O)[C@H]2CCCO2)CC1 ZINC000217681719 IE On-Demand Unstable L3MBTL3 49 35 O=C(O)[C@@H](CN1CC[C@@H](c2ccccc2)C1)C(F)(F)F ZINC000217681722 CF For-Sale Unstable TACR1 15 42 O=C(O)[C@@H](CN1CC[C@@H](c2ccccc2)C1)C(F)(F)F ZINC000217681722 CF For-Sale Unstable SIGMAR1 25 46 O=C(O)[C@@H](CN1CC[C@@H](c2ccccc2)C1)C(F)(F)F ZINC000217681722 CF For-Sale Unstable PRCP 23 46 O=C(O)[C@@H](CN1CC[C@@H](c2ccccc2)C1)C(F)(F)F ZINC000217681722 CF For-Sale Unstable CCR5 104 37 O=C(O)[C@@H](CN1CC[C@@H](c2ccccc2)C1)C(F)(F)F ZINC000217681722 CF For-Sale Unstable SLC18A3 66 50 O=C(O)[C@@H](CN1CC[C@@H](c2ccccc2)C1)C(F)(F)F ZINC000217681722 CF For-Sale Unstable CCR2 24 44 O=C(O)[C@@H](CN1CC[C@@H](c2ccccc2)C1)C(F)(F)F ZINC000217681722 CF For-Sale Unstable RBP4 40 37 O=C(O)[C@@H](CN1CC[C@@H](c2ccccc2)C1)C(F)(F)F ZINC000217681722 CF For-Sale Unstable MGEA5 24 40 CCOC(=O)[C@H](Nc1cccc(CC)c1)c1ccccc1 ZINC000217681752 CH On-Demand Unstable CAPN2 62 33 CCOC(=O)[C@H](Nc1cccc(CC)c1)c1ccccc1 ZINC000217681752 CH On-Demand Unstable NPR 42 33 CCOC(=O)[C@H](Nc1cccc(CC)c1)c1ccccc1 ZINC000217681752 CH On-Demand Unstable PPASE1 0 50 CCOC(=O)[C@H](Nc1cccc(CC)c1)c1ccccc1 ZINC000217681752 CH On-Demand Unstable PDS 46 37 CC[C@@H](CCO)NC(=O)CCCC(=O)O ZINC000217681824 BC On-Demand Unstable PLA2G2C 0 51 CC[C@@H](CCO)NC(=O)CCCC(=O)O ZINC000217681824 BC On-Demand Unstable Q6UB75_PIG 0 50 CC[C@@H](CCO)NC(=O)CCCC(=O)O ZINC000217681824 BC On-Demand Unstable NOD1 57 37 CC[C@@H](CCO)NC(=O)CCCC(=O)O ZINC000217681824 BC On-Demand Unstable COL4A3BP 0 42 Cc1ccccc1CNC(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217681884 DG For-Sale Unstable PTGER2 28 41 CC[C@H](CCO)NC(=O)CCCC(=O)O ZINC000217681900 BC On-Demand Unstable PLA2G2C 0 51 CC[C@H](CCO)NC(=O)CCCC(=O)O ZINC000217681900 BC On-Demand Unstable Q6UB75_PIG 0 50 CC[C@H](CCO)NC(=O)CCCC(=O)O ZINC000217681900 BC On-Demand Unstable NOD1 57 37 CC[C@H](CCO)NC(=O)CCCC(=O)O ZINC000217681900 BC On-Demand Unstable COL4A3BP 0 42 CC[C@@H](N[C@@H]1CCN2CCCC[C@@H]12)c1cccc(Cl)c1 ZINC000217681938 CI For-Sale Unstable OPRL1 0 40 Cc1cccc(CNC(=O)c2ccc(/C=C\C(=O)O)s2)c1 ZINC000217681958 DG For-Sale Unstable HDAC1 15 44 Cc1cccc(CNC(=O)c2ccc(/C=C\C(=O)O)s2)c1 ZINC000217681958 DG For-Sale Unstable HSD17B2 29 40 Cc1cccc(CNC(=O)c2ccc(/C=C\C(=O)O)s2)c1 ZINC000217681958 DG For-Sale Unstable SCD1 17 40 Cc1cccc(CNC(=O)c2ccc(/C=C\C(=O)O)s2)c1 ZINC000217681958 DG For-Sale Unstable SCD 16 40 CC[C@H](N[C@@H]1CCN2CCCC[C@@H]12)c1cccc(Cl)c1 ZINC000217682012 CI On-Demand Unstable OPRL1 0 40 CCOC(=O)[C@@H](c1ccccc1)N1CCC[C@@H](CO)C1 ZINC000217682027 CD On-Demand Unstable CHRM1 22 49 CCOC(=O)[C@@H](c1ccccc1)N1CCC[C@@H](CO)C1 ZINC000217682027 CD On-Demand Unstable SLC6A1 76 38 CCOC(=O)[C@@H](c1ccccc1)N1CCC[C@@H](CO)C1 ZINC000217682027 CD On-Demand Unstable CHRM3 22 49 CCOC(=O)[C@@H](c1ccccc1)N1CCC[C@@H](CO)C1 ZINC000217682027 CD On-Demand Unstable FKBP12.6 0 41 CC(=O)Nc1cccc(NC(=O)N/C=C/c2ccccc2C)c1 ZINC000217682037 DH For-Sale Unstable KCNK3 114 44 CC(=O)Nc1cccc(NC(=O)N/C=C/c2ccccc2C)c1 ZINC000217682037 DH For-Sale Unstable KCNK9 76 41 NC(=O)c1ccc(NC(=O)CCCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@H]23)cc1 ZINC000217682082 JG In-Stock Unstable TOP1 0 40 CC[C@@H](N[C@H]1CCN2CCCC[C@@H]12)c1cccc(Cl)c1 ZINC000217682090 CI For-Sale Unstable OPRL1 0 40 CCOC(=O)[C@H](c1ccccc1)N1CCC[C@@H](CO)C1 ZINC000217682123 CD On-Demand Unstable CHRM1 22 49 CCOC(=O)[C@H](c1ccccc1)N1CCC[C@@H](CO)C1 ZINC000217682123 CD On-Demand Unstable SLC6A1 76 38 CCOC(=O)[C@H](c1ccccc1)N1CCC[C@@H](CO)C1 ZINC000217682123 CD On-Demand Unstable CHRM3 22 49 CCOC(=O)[C@H](c1ccccc1)N1CCC[C@@H](CO)C1 ZINC000217682123 CD On-Demand Unstable FKBP12.6 0 41 CCCOc1cccc(C(=O)NC[C@@H](O)C(=O)OC)c1 ZINC000217682140 CC On-Demand Unstable DRD4 48 38 CCCOc1cccc(C(=O)NC[C@@H](O)C(=O)OC)c1 ZINC000217682140 CC On-Demand Unstable PLA2G4B 43 44 CCCOc1cccc(C(=O)NC[C@@H](O)C(=O)OC)c1 ZINC000217682140 CC On-Demand Unstable PDS 43 32 NC(=O)c1ccc(NC(=O)CCCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@@H]23)cc1 ZINC000217682152 JG In-Stock Unstable TOP1 0 40 CC[C@H](N[C@H]1CCN2CCCC[C@@H]12)c1cccc(Cl)c1 ZINC000217682159 CI On-Demand Unstable OPRL1 0 40 COc1ccc(C(=O)N2CCC[C@@H](C(=O)O)C2)c(F)c1 ZINC000217682196 CD In-Stock Unstable SLC6A1 129 41 COc1ccc(C(=O)N2CCC[C@@H](C(=O)O)C2)c(F)c1 ZINC000217682196 CD In-Stock Unstable GRM3 20 60 COc1ccc(C(=O)N2CCC[C@@H](C(=O)O)C2)c(F)c1 ZINC000217682196 CD In-Stock Unstable MTNR1B 20 44 COc1ccc(C(=O)N2CCC[C@@H](C(=O)O)C2)c(F)c1 ZINC000217682196 CD In-Stock Unstable SLC6A11 0 45 COc1ccc(C(=O)N2CCC[C@@H](C(=O)O)C2)c(F)c1 ZINC000217682196 CD In-Stock Unstable SLC6A13 0 45 CCCOc1cccc(C(=O)NC[C@H](O)C(=O)OC)c1 ZINC000217682205 CC On-Demand Unstable DRD4 48 38 CCCOc1cccc(C(=O)NC[C@H](O)C(=O)OC)c1 ZINC000217682205 CC On-Demand Unstable PLA2G4B 43 44 CCCOc1cccc(C(=O)NC[C@H](O)C(=O)OC)c1 ZINC000217682205 CC On-Demand Unstable PDS 43 32 O=C(O)[C@@H](CN1CC[C@@H](O)C1)C(F)(F)F ZINC000217682253 BC For-Sale Unstable OPRK1 18 40 COc1ccc(C(=O)N2CCC[C@H](C(=O)O)C2)c(F)c1 ZINC000217682258 CD In-Stock Unstable SLC6A1 129 41 COc1ccc(C(=O)N2CCC[C@H](C(=O)O)C2)c(F)c1 ZINC000217682258 CD In-Stock Unstable GRM3 20 60 COc1ccc(C(=O)N2CCC[C@H](C(=O)O)C2)c(F)c1 ZINC000217682258 CD In-Stock Unstable MTNR1B 20 44 COc1ccc(C(=O)N2CCC[C@H](C(=O)O)C2)c(F)c1 ZINC000217682258 CD In-Stock Unstable SLC6A11 0 45 COc1ccc(C(=O)N2CCC[C@H](C(=O)O)C2)c(F)c1 ZINC000217682258 CD In-Stock Unstable SLC6A13 0 45 COc1ccc([C@@H](C)N[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217682291 CF For-Sale Unstable CHRM2 29 45 COc1ccc([C@@H](C)N[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217682291 CF For-Sale Unstable CHRM4 17 45 CC(C)[C@H](NC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)C(=O)NCc1cccn1C ZINC000217682298 ID In-Stock Unstable CHRNA4 27 44 CC(C)c1noc2ncc(C(=O)NCCCN3CCCCC3)cc12 ZINC000217682306 EF On-Demand Unstable DRD3 41 36 CC(C)c1noc2ncc(C(=O)NCCCN3CCCCC3)cc12 ZINC000217682306 EF On-Demand Unstable CHRNA7 25 43 CC(C)c1noc2ncc(C(=O)NCCCN3CCCCC3)cc12 ZINC000217682306 EF On-Demand Unstable HNMT 46 34 COC(=O)[C@@H](O)CNC(=O)Cc1ccc(OC)c(OC)c1 ZINC000217682324 CB On-Demand Unstable TRPV1 25 45 COC(=O)[C@@H](O)CNC(=O)Cc1ccc(OC)c(OC)c1 ZINC000217682324 CB On-Demand Unstable MT-ND1 26 43 COC(=O)[C@@H](O)CNC(=O)Cc1ccc(OC)c(OC)c1 ZINC000217682324 CB On-Demand Unstable NCE103 30 51 COC(=O)[C@@H](O)CNC(=O)Cc1ccc(OC)c(OC)c1 ZINC000217682324 CB On-Demand Unstable ENPP1 49 30 COC(=O)[C@@H](O)CNC(=O)Cc1ccc(OC)c(OC)c1 ZINC000217682324 CB On-Demand Unstable P96878_MYCTU 17 51 O=C1C=C(C(=O)O)N[C@@H](C(=O)O)C1 ZINC000217682336 AA For-Sale Unstable CAD 48 38 COc1ccc(C(=O)N2CCC(C(=O)O)CC2)c(F)c1 ZINC000217682358 CD On-Demand Unstable CHRM2 22 41 COc1ccc(C(=O)N2CCC(C(=O)O)CC2)c(F)c1 ZINC000217682358 CD On-Demand Unstable OXTR 0 42 COc1ccc(C(=O)N2CCC(C(=O)O)CC2)c(F)c1 ZINC000217682358 CD On-Demand Unstable AKR1C2 52 37 COc1ccc(C(=O)N2CCC(C(=O)O)CC2)c(F)c1 ZINC000217682358 CD On-Demand Unstable L3MBTL3 49 38 Cc1nccn1CC[C@@H]1CCCCN1C(=O)c1n[nH]c(=O)c2ccccc12 ZINC000217682369 FF In-Stock Unstable PARP1 27 40 COc1ccc([C@H](C)N[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217682377 CF On-Demand Unstable CHRM2 27 45 COC(=O)[C@H](O)CNC(=O)Cc1ccc(OC)c(OC)c1 ZINC000217682413 CB On-Demand Unstable TRPV1 25 45 COC(=O)[C@H](O)CNC(=O)Cc1ccc(OC)c(OC)c1 ZINC000217682413 CB On-Demand Unstable MT-ND1 26 43 COC(=O)[C@H](O)CNC(=O)Cc1ccc(OC)c(OC)c1 ZINC000217682413 CB On-Demand Unstable NCE103 30 51 COC(=O)[C@H](O)CNC(=O)Cc1ccc(OC)c(OC)c1 ZINC000217682413 CB On-Demand Unstable ENPP1 49 30 COC(=O)[C@H](O)CNC(=O)Cc1ccc(OC)c(OC)c1 ZINC000217682413 CB On-Demand Unstable P96878_MYCTU 17 51 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)c1cc(Br)ccc1Cl)C2 ZINC000217682438 HF In-Stock Unstable HTR4 38 43 CCOC(=O)[C@@H](c1ccccc1)N1CCCN(C)CC1 ZINC000217682443 CD On-Demand Unstable MC4R 25 44 CCOC(=O)[C@@H](c1ccccc1)N1CCCN(C)CC1 ZINC000217682443 CD On-Demand Unstable NPY2R 41 37 CCOC(=O)[C@@H](c1ccccc1)N1CCCN(C)CC1 ZINC000217682443 CD On-Demand Unstable NMUR2 0 45 CCOC(=O)[C@@H](c1ccccc1)N1CCCN(C)CC1 ZINC000217682443 CD On-Demand Unstable NMUR1 0 45 Cc1nccn1CC[C@H]1CCCCN1C(=O)c1n[nH]c(=O)c2ccccc12 ZINC000217682453 FF In-Stock Unstable PARP1 27 40 COc1ccc([C@@H](C)N[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217682460 CF For-Sale Unstable CHRM2 29 45 COc1ccc([C@@H](C)N[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217682460 CF For-Sale Unstable CHRM4 17 45 CCOC(=O)[C@H](c1ccccc1)N1CCCN(C)CC1 ZINC000217682521 CD On-Demand Unstable MC4R 25 44 CCOC(=O)[C@H](c1ccccc1)N1CCCN(C)CC1 ZINC000217682521 CD On-Demand Unstable NPY2R 41 37 CCOC(=O)[C@H](c1ccccc1)N1CCCN(C)CC1 ZINC000217682521 CD On-Demand Unstable NMUR2 0 45 CCOC(=O)[C@H](c1ccccc1)N1CCCN(C)CC1 ZINC000217682521 CD On-Demand Unstable NMUR1 0 45 O=C(O)[C@@H](CN1CC[C@@H](N2CCCC2)C1)C(F)(F)F ZINC000217682524 CD For-Sale Unstable L3MBTL3 41 38 COc1ccc([C@H](C)N[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217682534 CF On-Demand Unstable CHRM2 27 45 COC(=O)[C@@H](O)CNC(=O)C(C)(C)Oc1ccc(Cl)cc1 ZINC000217682556 DD On-Demand Unstable FABP1 15 45 CSC/C=C(\NC(C)=O)C(=O)O ZINC000217682570 AC For-Sale Unstable DPEP1 69 40 c1ccc2c(c1)CC[C@H]2N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217682622 CF For-Sale Unstable SIGMAR1 0 43 c1ccc2c(c1)CC[C@H]2N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217682622 CF For-Sale Unstable SLC18A3 52 40 COC(=O)[C@H](O)CNC(=O)C(C)(C)Oc1ccc(Cl)cc1 ZINC000217682630 DD On-Demand Unstable FABP1 15 45 CSC/C=C(/NC(C)=O)C(=O)O ZINC000217682648 AC For-Sale Unstable DPEP1 69 40 CCN(CCNC(=O)c1cnn(-c2ccccc2)c1C(F)(F)F)c1cccc(C)c1 ZINC000217682681 HI On-Demand Unstable MST1R 55 41 O=C(O)CCNC(=O)c1ccc2c(c1)[C@@H]1C=CC[C@@H]1[C@@H](c1cc(C(F)(F)F)cc(C(F)(F)F)c1)N2 ZINC000217682693 JK In-Stock Unstable GCGR 53 43 O=C(O)CCNC(=O)c1ccc2c(c1)[C@@H]1C=CC[C@@H]1[C@@H](c1cc(C(F)(F)F)cc(C(F)(F)F)c1)N2 ZINC000217682693 JK In-Stock Unstable GIPR 44 43 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)c1ccc(-n3cccc3)cc1)C2 ZINC000217682738 FE In-Stock Unstable AOC2 0 45 O=C(O)CCNC(=O)c1ccc2c(c1)[C@@H]1C=CC[C@H]1[C@@H](c1cc(C(F)(F)F)cc(C(F)(F)F)c1)N2 ZINC000217682783 JK In-Stock Unstable GCGR 53 43 O=C(O)CCNC(=O)c1ccc2c(c1)[C@@H]1C=CC[C@H]1[C@@H](c1cc(C(F)(F)F)cc(C(F)(F)F)c1)N2 ZINC000217682783 JK In-Stock Unstable GIPR 44 43 CCC1CCN(C(=O)c2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217682836 CG For-Sale Unstable L3MBTL1 0 43 CCC1CCN(C(=O)c2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217682836 CG For-Sale Unstable L3MBTL3 66 43 CCC1CCN(C(=O)c2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217682836 CG For-Sale Unstable GPR183 0 42 O=C(c1cccc(OCc2cn3ccccc3n2)c1)N1CCN(CCN2CCCC2)CC1 ZINC000217682883 IF On-Demand Unstable DRD4 42 34 O=C(c1cccc(OCc2cn3ccccc3n2)c1)N1CCN(CCN2CCCC2)CC1 ZINC000217682883 IF On-Demand Unstable HRH3 19 43 O=C(c1cccc(OCc2cn3ccccc3n2)c1)N1CCN(CCN2CCCC2)CC1 ZINC000217682883 IF On-Demand Unstable PARP1 15 40 CC(=O)N1CCC(C(=O)NC2C[C@@H]3CC[C@H](C2)N3S(C)(=O)=O)CC1 ZINC000217682921 FC In-Stock Unstable EPHX2 29 41 C[C@@H](N[C@@H]1CCN2CCCC[C@@H]12)c1ccccc1 ZINC000217682944 BF For-Sale Unstable SLC18A3 56 38 O=C(O)CCNC(=O)c1ccc2c(c1)[C@@H]1C=CC[C@@H]1[C@@H](c1ccc(C(F)(F)F)cc1)N2 ZINC000217682954 IJ In-Stock Unstable GCGR 63 41 O=C(O)CCNC(=O)c1ccc2c(c1)[C@@H]1C=CC[C@@H]1[C@@H](c1ccc(C(F)(F)F)cc1)N2 ZINC000217682954 IJ In-Stock Unstable GIPR 46 41 O=C(c1ccc(=O)n(Cc2ccccc2Cl)c1)N1CCN(CCN2CCCC2)CC1 ZINC000217682994 IE On-Demand Unstable HRH3 17 40 O=C(c1ccc(=O)n(Cc2ccccc2Cl)c1)N1CCN(CCN2CCCC2)CC1 ZINC000217682994 IE On-Demand Unstable L3MBTL3 43 36 C[C@H](N[C@@H]1CCN2CCCC[C@@H]12)c1ccccc1 ZINC000217683016 BF On-Demand Unstable SLC18A3 50 38 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cc3cc5c(cc3[nH]c2=O)OCCO5)CC(=O)O4)cc1O ZINC000217683024 KH In-Stock Unstable AKR1B1 0 41 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cc3cc5c(cc3[nH]c2=O)OCCO5)CC(=O)O4)cc1O ZINC000217683024 KH In-Stock Unstable CYP1A1 27 41 O=C(O)CCNC(=O)c1ccc2c(c1)[C@@H]1C=CC[C@H]1[C@@H](c1ccc(C(F)(F)F)cc1)N2 ZINC000217683035 IJ In-Stock Unstable GCGR 63 41 O=C(O)CCNC(=O)c1ccc2c(c1)[C@@H]1C=CC[C@H]1[C@@H](c1ccc(C(F)(F)F)cc1)N2 ZINC000217683035 IJ In-Stock Unstable GIPR 46 41 CCOC(=O)[C@@H](c1ccccc1)N1CCCCCCC1 ZINC000217683071 CH For-Sale Unstable CHRM2 21 44 CCOC(=O)[C@@H](c1ccccc1)N1CCCCCCC1 ZINC000217683071 CH For-Sale Unstable CHRM1 30 70 CCOC(=O)[C@@H](c1ccccc1)N1CCCCCCC1 ZINC000217683071 CH For-Sale Unstable FKBP1A 27 40 CCOC(=O)[C@@H](c1ccccc1)N1CCCCCCC1 ZINC000217683071 CH For-Sale Unstable OPRK1 18 41 CCOC(=O)[C@@H](c1ccccc1)N1CCCCCCC1 ZINC000217683071 CH For-Sale Unstable OPRL1 16 40 CCOC(=O)[C@@H](c1ccccc1)N1CCCCCCC1 ZINC000217683071 CH For-Sale Unstable SLC6A3 22 48 CCOC(=O)[C@@H](c1ccccc1)N1CCCCCCC1 ZINC000217683071 CH For-Sale Unstable CHRM3 22 70 CCOC(=O)[C@@H](c1ccccc1)N1CCCCCCC1 ZINC000217683071 CH For-Sale Unstable KCNQ2 55 42 CCOC(=O)[C@@H](c1ccccc1)N1CCCCCCC1 ZINC000217683071 CH For-Sale Unstable NPY2R 55 45 CCOC(=O)[C@@H](c1ccccc1)N1CCCCCCC1 ZINC000217683071 CH For-Sale Unstable AMY2 46 33 C[C@@H](N[C@H]1CCN2CCCC[C@@H]12)c1ccccc1 ZINC000217683093 BF For-Sale Unstable SLC18A3 56 38 CC[C@@H](C)NS(=O)(=O)c1ccc(/C=C\C(=O)O)c(C)c1 ZINC000217683095 CE For-Sale Unstable MMP12 44 34 CC[C@@H](C)NS(=O)(=O)c1ccc(/C=C\C(=O)O)c(C)c1 ZINC000217683095 CE For-Sale Unstable LEF 64 46 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cc3cc5c(cc3[nH]c2=O)OCCO5)CC(=O)O4)cc1O ZINC000217683101 KH In-Stock Unstable AKR1B1 0 41 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cc3cc5c(cc3[nH]c2=O)OCCO5)CC(=O)O4)cc1O ZINC000217683101 KH In-Stock Unstable CYP1A1 27 41 CCCn1c(C)c(C(=O)N2CCN(CCN3CCCC3)CC2)c2cc(OC)ccc21 ZINC000217683111 HG On-Demand Unstable CNR1 21 46 CCCn1c(C)c(C(=O)N2CCN(CCN3CCCC3)CC2)c2cc(OC)ccc21 ZINC000217683111 HG On-Demand Unstable DRD4 43 33 CCCn1c(C)c(C(=O)N2CCN(CCN3CCCC3)CC2)c2cc(OC)ccc21 ZINC000217683111 HG On-Demand Unstable AVPR1B 20 43 CCCn1c(C)c(C(=O)N2CCN(CCN3CCCC3)CC2)c2cc(OC)ccc21 ZINC000217683111 HG On-Demand Unstable CNR2 19 50 CCCn1c(C)c(C(=O)N2CCN(CCN3CCCC3)CC2)c2cc(OC)ccc21 ZINC000217683111 HG On-Demand Unstable PTGDS 46 44 CCOC(=O)[C@H](c1ccccc1)N1CCCCCCC1 ZINC000217683156 CH For-Sale Unstable CHRM2 21 44 CCOC(=O)[C@H](c1ccccc1)N1CCCCCCC1 ZINC000217683156 CH For-Sale Unstable CHRM1 30 70 CCOC(=O)[C@H](c1ccccc1)N1CCCCCCC1 ZINC000217683156 CH For-Sale Unstable FKBP1A 27 40 CCOC(=O)[C@H](c1ccccc1)N1CCCCCCC1 ZINC000217683156 CH For-Sale Unstable OPRK1 18 41 CCOC(=O)[C@H](c1ccccc1)N1CCCCCCC1 ZINC000217683156 CH For-Sale Unstable OPRL1 16 40 CCOC(=O)[C@H](c1ccccc1)N1CCCCCCC1 ZINC000217683156 CH For-Sale Unstable SLC6A3 22 48 CCOC(=O)[C@H](c1ccccc1)N1CCCCCCC1 ZINC000217683156 CH For-Sale Unstable CHRM3 22 70 CCOC(=O)[C@H](c1ccccc1)N1CCCCCCC1 ZINC000217683156 CH For-Sale Unstable KCNQ2 55 42 CCOC(=O)[C@H](c1ccccc1)N1CCCCCCC1 ZINC000217683156 CH For-Sale Unstable NPY2R 55 45 CCOC(=O)[C@H](c1ccccc1)N1CCCCCCC1 ZINC000217683156 CH For-Sale Unstable AMY2 46 33 CNC(=O)c1cc(F)cc(Cl)c1 ZINC000217683161 AD In-Stock Unstable CACNA1I 43 33 C[C@H](N[C@H]1CCN2CCCC[C@@H]12)c1ccccc1 ZINC000217683175 BF On-Demand Unstable SLC18A3 50 38 CC[C@H](C)NS(=O)(=O)c1ccc(/C=C\C(=O)O)c(C)c1 ZINC000217683177 CE For-Sale Unstable MMP12 44 34 CC[C@H](C)NS(=O)(=O)c1ccc(/C=C\C(=O)O)c(C)c1 ZINC000217683177 CE For-Sale Unstable LEF 64 46 O=C(Cn1cc(Br)c(=O)[nH]c1=O)N1CCN(CCN2CCCC2)CC1 ZINC000217683227 HB On-Demand Unstable GRIA3 19 43 O=C(Cn1cc(Br)c(=O)[nH]c1=O)N1CCN(CCN2CCCC2)CC1 ZINC000217683227 HB On-Demand Unstable GRIK5 24 43 C=C(C)CNC[C@@H](C)NC(=O)OC(C)(C)C ZINC000217683251 BE For-Sale Unstable CTSK 22 55 Cc1ccccc1/C=C/NC(=O)Nc1ccccc1N1CCOCC1 ZINC000217683313 EH For-Sale Unstable KCNQ2 83 42 Cc1ccccc1/C=C/NC(=O)Nc1ccccc1N1CCOCC1 ZINC000217683313 EH For-Sale Unstable CSF1R 0 46 Cc1ccccc1/C=C/NC(=O)Nc1ccccc1N1CCOCC1 ZINC000217683313 EH For-Sale Unstable AKR1C3 0 40 CS(=O)(=O)N1CCN(C(=O)c2cnn(-c3ccccc3)c2C(F)(F)F)CC1 ZINC000217683341 HD On-Demand Unstable SLC6A9 26 40 CS(=O)(=O)N1CCN(C(=O)c2cnn(-c3ccccc3)c2C(F)(F)F)CC1 ZINC000217683341 HD On-Demand Unstable MST1R 43 36 C[C@H](N[C@@H]1CCN2CCCC[C@@H]12)c1cccc(Br)c1 ZINC000217683382 DH On-Demand Unstable MBTD1 0 52 CCCCCC[C@@H](C)NCCN(CC)CCC ZINC000217683385 BH For-Sale Unstable ADH1B 0 44 CCCCCC[C@@H](C)NCCN(CC)CCC ZINC000217683385 BH For-Sale Unstable ADH1C 0 44 CCCCCC[C@@H](C)NCCN(CC)CCC ZINC000217683385 BH For-Sale Unstable Q6UB75_PIG 0 46 COC(=O)C[C@H](c1oc(CN2CCCCC2)cc(=O)c1O)c1ccnc2ccccc12 ZINC000217683407 HH In-Stock Unstable HNMT 50 37 Cc1ccccc1/C=C/NC(=O)Nc1ccc(N2CCN(C)CC2)cc1 ZINC000217683445 FH For-Sale Unstable LCK 20 42 Cc1ccccc1/C=C/NC(=O)Nc1ccc(N2CCN(C)CC2)cc1 ZINC000217683445 FH For-Sale Unstable PRNP 41 49 Cc1ccccc1/C=C/NC(=O)Nc1ccc(N2CCN(C)CC2)cc1 ZINC000217683445 FH For-Sale Unstable MTOR 21 43 CCOC(=O)[C@H](N[C@@H]1CCCC[C@@H]1C)c1ccccc1 ZINC000217683453 CG On-Demand Unstable AMY2 49 35 COc1ccc(S(=O)(=O)NC2CC2)cc1/C=C\C(=O)O ZINC000217683459 CD For-Sale Unstable ADRA1D 24 44 COc1ccc(S(=O)(=O)NC2CC2)cc1/C=C\C(=O)O ZINC000217683459 CD For-Sale Unstable ADRA1A 17 44 COc1ccc(S(=O)(=O)NC2CC2)cc1/C=C\C(=O)O ZINC000217683459 CD For-Sale Unstable ADRA1B 31 44 COc1ccc(S(=O)(=O)NC2CC2)cc1/C=C\C(=O)O ZINC000217683459 CD For-Sale Unstable SFRP1 97 34 COc1ccc(S(=O)(=O)NC2CC2)cc1/C=C\C(=O)O ZINC000217683459 CD For-Sale Unstable WNT3 58 32 O=C(O)CCNC(=O)c1ccc2c(c1)[C@@H]1C=CC[C@@H]1[C@@H](c1cccc(C(F)(F)F)c1)N2 ZINC000217683463 IJ In-Stock Unstable GCGR 52 41 O=C(O)CCNC(=O)c1ccc2c(c1)[C@@H]1C=CC[C@@H]1[C@@H](c1cccc(C(F)(F)F)c1)N2 ZINC000217683463 IJ In-Stock Unstable CCR2 49 37 CCCCCC[C@H](C)NCCN(CC)CCC ZINC000217683467 BH For-Sale Unstable ADH1B 0 44 CCCCCC[C@H](C)NCCN(CC)CCC ZINC000217683467 BH For-Sale Unstable ADH1C 0 44 CCCCCC[C@H](C)NCCN(CC)CCC ZINC000217683467 BH For-Sale Unstable Q6UB75_PIG 0 46 COC(=O)C[C@@H](c1oc(CN2CCCCC2)cc(=O)c1O)c1ccnc2ccccc12 ZINC000217683498 HH In-Stock Unstable HNMT 50 37 COc1ccc(S(=O)(=O)NCC2CC2)cc1/C=C\C(=O)O ZINC000217683540 DD For-Sale Unstable NPY2R 65 42 COc1ccc(S(=O)(=O)NCC2CC2)cc1/C=C\C(=O)O ZINC000217683540 DD For-Sale Unstable NPY5R 15 42 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)c1cccc3ccccc13)C2 ZINC000217683556 FF In-Stock Unstable HTR3A 41 43 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)c1cccc3ccccc13)C2 ZINC000217683556 FF In-Stock Unstable HTR4 50 45 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)c1cccc3ccccc13)C2 ZINC000217683556 FF In-Stock Unstable CCR3 20 40 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)c1cccc3ccccc13)C2 ZINC000217683556 FF In-Stock Unstable CCR8 60 37 Cc1ccccc1/C=C/NC(=O)Nc1ccc(N2CCCCC2)cc1 ZINC000217683566 EJ For-Sale Unstable LPL 45 37 Cc1ccccc1/C=C/NC(=O)Nc1ccc(N2CCCCC2)cc1 ZINC000217683566 EJ For-Sale Unstable KCNQ2 19 44 C[C@H](N[C@H]1CCN2CCCC[C@@H]12)c1cccc(Br)c1 ZINC000217683569 DH On-Demand Unstable MBTD1 0 52 O=C(O)CCNC(=O)c1ccc2c(c1)[C@@H]1C=CC[C@H]1[C@@H](c1cccc(C(F)(F)F)c1)N2 ZINC000217683570 IJ In-Stock Unstable GCGR 52 41 O=C(O)CCNC(=O)c1ccc2c(c1)[C@@H]1C=CC[C@H]1[C@@H](c1cccc(C(F)(F)F)c1)N2 ZINC000217683570 IJ In-Stock Unstable CCR2 49 37 Cc1cc(CNC(=O)c2cc(-c3cccs3)on2)ccc1F ZINC000217683608 DH On-Demand Unstable S1PR4 0 43 CCOC(=O)[C@H](N[C@H]1CCCC[C@@H]1C)c1ccccc1 ZINC000217683612 CG On-Demand Unstable AMY2 49 35 CC(C)NC(=O)CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12 ZINC000217683621 GG In-Stock Unstable TOP1 22 43 O=C(O)/C=C\c1ccc(S(=O)(=O)NCC2CC2)c(Cl)c1 ZINC000217683628 DE For-Sale Unstable NPY2R 59 41 O=C(O)/C=C\c1ccc(S(=O)(=O)NCC2CC2)c(Cl)c1 ZINC000217683628 DE For-Sale Unstable NPY5R 17 41 CCCCN(C[C@@H](C(=O)O)C(F)(F)F)c1ccccc1 ZINC000217683649 CH For-Sale Unstable AMY2 54 31 CSC[C@@](C)(O)CNC(=O)c1ccc2ncccc2c1 ZINC000217683687 CE On-Demand Unstable CCR3 17 40 CC(C)NC(=O)CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12 ZINC000217683708 GG In-Stock Unstable TOP1 22 43 O=C(O)/C=C\c1cc(Cl)c(S(=O)(=O)NCC2CC2)c(Cl)c1 ZINC000217683724 FF For-Sale Unstable NPY2R 43 37 CCC[C@@H](O)CNC(=O)CCC(=O)O ZINC000217683729 BC On-Demand Unstable KDM2A 40 39 CCCCN(C[C@H](C(=O)O)C(F)(F)F)c1ccccc1 ZINC000217683733 CH For-Sale Unstable AMY2 54 31 CSC[C@](C)(O)CNC(=O)c1ccc2ncccc2c1 ZINC000217683770 CE On-Demand Unstable CCR3 17 40 CCCCN(C)S(=O)(=O)c1ccc(/C=C\C(=O)O)cc1Cl ZINC000217683806 EF For-Sale Unstable NR0B2 0 40 CCC[C@H](O)CNC(=O)CCC(=O)O ZINC000217683813 BC On-Demand Unstable KDM2A 40 39 CC(C)C[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217683819 HD In-Stock Unstable SSTR2 41 37 CC(C)C[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217683819 HD In-Stock Unstable EDNRA 40 43 CC(C)C[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217683819 HD In-Stock Unstable TACR1 29 40 CC(C)C[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217683819 HD In-Stock Unstable CCKAR 41 38 CC(C)C[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217683819 HD In-Stock Unstable BRS3 26 41 CC(C)C[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217683819 HD In-Stock Unstable NMBR 45 32 CC(C)C[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217683819 HD In-Stock Unstable MMP2 21 40 CC(C)C[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217683819 HD In-Stock Unstable MMP8 30 40 CC(C)C[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217683819 HD In-Stock Unstable GRPR 71 38 CC(C)C[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217683819 HD In-Stock Unstable CCKBR 40 37 CC(C)C[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217683819 HD In-Stock Unstable GHSR 60 39 CC(C)C[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217683819 HD In-Stock Unstable MMP9 17 40 CC(C)C[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217683819 HD In-Stock Unstable SLC15A2 0 43 CC(C)C[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217683819 HD In-Stock Unstable KISS1R 66 32 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)c1ccccc1Br)C2 ZINC000217683842 GE In-Stock Unstable HTR4 39 40 COC(=O)C[C@H](c1cc(OC)c2c(c1)OCO2)c1c(O)cc(C)n(CCc2ccc(O)cc2)c1=O ZINC000217683934 JG In-Stock Unstable RORC 40 38 CCC[C@@H](O)CNC(=O)CCCCC(=O)O ZINC000217683937 BC On-Demand Unstable FABP2 0 44 CCC[C@@H](O)CNC(=O)CCCCC(=O)O ZINC000217683937 BC On-Demand Unstable FABP4 17 44 CCC[C@@H](O)CNC(=O)CCCCC(=O)O ZINC000217683937 BC On-Demand Unstable PLA2G2C 0 44 CCC[C@@H](O)CNC(=O)CCCCC(=O)O ZINC000217683937 BC On-Demand Unstable Q6UB75_PIG 0 43 CCC[C@@H](O)CNC(=O)CCCCC(=O)O ZINC000217683937 BC On-Demand Unstable FABP3 33 41 CCC[C@@H](O)CNC(=O)CCCCC(=O)O ZINC000217683937 BC On-Demand Unstable FABP5 15 44 CCC[C@@H](O)CNC(=O)CCCCC(=O)O ZINC000217683937 BC On-Demand Unstable SLC22A20 0 45 CCC[C@@H](O)CNC(=O)CCCCC(=O)O ZINC000217683937 BC On-Demand Unstable NOD1 50 37 CCC[C@@H](O)CNC(=O)CCCCC(=O)O ZINC000217683937 BC On-Demand Unstable CQSS 43 37 Cc1ccccc1/C=C/NC(=O)Nc1cccc2ccccc12 ZINC000217683987 DJ For-Sale Unstable CHAT 65 39 O=C(CCc1ccccc1)N1C[C@H]2CNC[C@@H](C2)C1 ZINC000217684008 CD For-Sale Unstable CHRNA7 22 57 COC(=O)C[C@@H](c1cc(OC)c2c(c1)OCO2)c1c(O)cc(C)n(CCc2ccc(O)cc2)c1=O ZINC000217684010 JG In-Stock Unstable RORC 40 38 CCC[C@H](O)CNC(=O)CCCCC(=O)O ZINC000217684021 BC On-Demand Unstable FABP2 0 44 CCC[C@H](O)CNC(=O)CCCCC(=O)O ZINC000217684021 BC On-Demand Unstable FABP4 17 44 CCC[C@H](O)CNC(=O)CCCCC(=O)O ZINC000217684021 BC On-Demand Unstable PLA2G2C 0 44 CCC[C@H](O)CNC(=O)CCCCC(=O)O ZINC000217684021 BC On-Demand Unstable Q6UB75_PIG 0 43 CCC[C@H](O)CNC(=O)CCCCC(=O)O ZINC000217684021 BC On-Demand Unstable FABP3 33 41 CCC[C@H](O)CNC(=O)CCCCC(=O)O ZINC000217684021 BC On-Demand Unstable FABP5 15 44 CCC[C@H](O)CNC(=O)CCCCC(=O)O ZINC000217684021 BC On-Demand Unstable SLC22A20 0 45 CCC[C@H](O)CNC(=O)CCCCC(=O)O ZINC000217684021 BC On-Demand Unstable NOD1 50 37 CCC[C@H](O)CNC(=O)CCCCC(=O)O ZINC000217684021 BC On-Demand Unstable CQSS 43 37 Cc1[nH]c2ccccc2c1CC(=O)NCc1c[nH]c(=O)[nH]c1=O ZINC000217684069 DC In-Stock Unstable GRIN1 19 43 Cc1[nH]c2ccccc2c1CC(=O)NCc1c[nH]c(=O)[nH]c1=O ZINC000217684069 DC In-Stock Unstable P2RX7 26 44 Cc1ccnc(NC(=O)c2cccc(/C=C\C(=O)O)c2)c1 ZINC000217684085 CF For-Sale Unstable LCK 18 42 Cc1ccnc(NC(=O)c2cccc(/C=C\C(=O)O)c2)c1 ZINC000217684085 CF For-Sale Unstable HDAC8 31 45 Cc1ccnc(NC(=O)c2cccc(/C=C\C(=O)O)c2)c1 ZINC000217684085 CF For-Sale Unstable HDAC6 18 45 Cc1ccnc(NC(=O)c2cccc(/C=C\C(=O)O)c2)c1 ZINC000217684085 CF For-Sale Unstable KCNK3 95 45 Cc1ccnc(NC(=O)c2cccc(/C=C\C(=O)O)c2)c1 ZINC000217684085 CF For-Sale Unstable KCNK9 50 45 COC(=O)C/C=C\CNC(=O)OC(C)(C)C ZINC000217684096 BD For-Sale Unstable CTSK 21 40 COC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2C)cc1 ZINC000217684112 DH For-Sale Unstable ACR 54 39 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)CNC(=O)OCc1ccccc1)C2 ZINC000217684118 GC In-Stock Unstable CTSB 46 45 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)CNC(=O)OCc1ccccc1)C2 ZINC000217684118 GC In-Stock Unstable CYSP_TRYCR 54 40 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)CNC(=O)OCc1ccccc1)C2 ZINC000217684118 GC In-Stock Unstable CTSK 28 45 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)CNC(=O)OCc1ccccc1)C2 ZINC000217684118 GC In-Stock Unstable CTSL 38 45 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)CNC(=O)OCc1ccccc1)C2 ZINC000217684118 GC In-Stock Unstable PREP 21 44 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)CNC(=O)OCc1ccccc1)C2 ZINC000217684118 GC In-Stock Unstable CAPNS1 62 33 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)CNC(=O)OCc1ccccc1)C2 ZINC000217684118 GC In-Stock Unstable CTSS 18 42 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)CNC(=O)OCc1ccccc1)C2 ZINC000217684118 GC In-Stock Unstable CAPN1 73 35 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)CNC(=O)OCc1ccccc1)C2 ZINC000217684118 GC In-Stock Unstable CAPN2 115 35 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)CNC(=O)OCc1ccccc1)C2 ZINC000217684118 GC In-Stock Unstable TGM2 33 41 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)CNC(=O)OCc1ccccc1)C2 ZINC000217684118 GC In-Stock Unstable POL 0 41 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)CNC(=O)OCc1ccccc1)C2 ZINC000217684118 GC In-Stock Unstable NPR 62 34 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)CNC(=O)OCc1ccccc1)C2 ZINC000217684118 GC In-Stock Unstable F13A1 31 41 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)CNC(=O)OCc1ccccc1)C2 ZINC000217684118 GC In-Stock Unstable NAAA 30 41 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)CNC(=O)OCc1ccccc1)C2 ZINC000217684118 GC In-Stock Unstable SLC12A5 53 35 COc1ccc(-c2csc(Nc3ccc(Cl)cc3)n2)cc1N ZINC000217684141 EJ In-Stock Unstable MAOA 0 40 COc1ccc(-c2csc(Nc3ccc(Cl)cc3)n2)cc1N ZINC000217684141 EJ In-Stock Unstable MAOB 26 44 COc1ccc(-c2csc(Nc3ccc(Cl)cc3)n2)cc1N ZINC000217684141 EJ In-Stock Unstable SPHK2 55 40 COc1ccc(-c2csc(Nc3ccc(Cl)cc3)n2)cc1N ZINC000217684141 EJ In-Stock Unstable SPHK1 41 57 COc1ccc(-c2csc(Nc3ccc(Cl)cc3)n2)cc1N ZINC000217684141 EJ In-Stock Unstable PLAU 22 44 COc1ccc(-c2csc(Nc3ccc(Cl)cc3)n2)cc1N ZINC000217684141 EJ In-Stock Unstable AGPAT2 58 48 COc1ccc(-c2csc(Nc3ccc(Cl)cc3)n2)cc1N ZINC000217684141 EJ In-Stock Unstable VCP 20 52 COc1ccc(-c2csc(Nc3ccc(Cl)cc3)n2)cc1N ZINC000217684141 EJ In-Stock Unstable TRPC6 40 38 O=C(Cn1c(=O)ccn(Cc2ccccc2)c1=O)N1CCN(Cc2cccnc2)CC1 ZINC000217684181 HC On-Demand Unstable DRD4 22 41 O=C(Cn1c(=O)ccn(Cc2ccccc2)c1=O)N1CCN(Cc2cccnc2)CC1 ZINC000217684181 HC On-Demand Unstable ACHE 16 45 O=C(Cn1c(=O)ccn(Cc2ccccc2)c1=O)N1CCN(Cc2cccnc2)CC1 ZINC000217684181 HC On-Demand Unstable PTAFR 15 57 O=C(Cn1c(=O)ccn(Cc2ccccc2)c1=O)N1CCN(Cc2cccnc2)CC1 ZINC000217684181 HC On-Demand Unstable SIGMAR1 27 40 O=C(Cn1c(=O)ccn(Cc2ccccc2)c1=O)N1CCN(Cc2cccnc2)CC1 ZINC000217684181 HC On-Demand Unstable FAAH 22 44 O=C(Cn1c(=O)ccn(Cc2ccccc2)c1=O)N1CCN(Cc2cccnc2)CC1 ZINC000217684181 HC On-Demand Unstable MGLL 0 40 O=C(CN1CCOC1=O)NCc1cnn(Cc2ccccc2)c1 ZINC000217684238 DC In-Stock Unstable ITK 0 40 COc1ccc(-c2csc(NS(=O)(=O)c3ccccc3)n2)cc1N ZINC000217684266 FG In-Stock Unstable MAOA 0 57 COc1ccc(-c2csc(NS(=O)(=O)c3ccccc3)n2)cc1N ZINC000217684266 FG In-Stock Unstable NPY5R 15 42 COc1ccc(NC(C)=O)cc1NC(=O)CCCCCNc1ccc2c(cc1=O)[C@@H](NC(C)=O)CCc1cc(OC)c(OC)c(OC)c1-2 ZINC000217684299 KK In-Stock Unstable TUBA1A 18 65 O=C(c1cnn(-c2ccccc2)c1C(F)(F)F)N1CCN(Cc2cccnc2)CC1 ZINC000217684341 HG On-Demand Unstable FAAH 18 42 O=C(c1cnn(-c2ccccc2)c1C(F)(F)F)N1CCN(Cc2cccnc2)CC1 ZINC000217684341 HG On-Demand Unstable MST1R 45 34 O=C(c1cnn(-c2ccccc2)c1C(F)(F)F)N1CCN(Cc2cccnc2)CC1 ZINC000217684341 HG On-Demand Unstable SCD 16 40 CC1CCN(C(=O)c2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217684349 CF For-Sale Unstable L3MBTL3 70 46 CC1CCN(C(=O)c2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217684349 CF For-Sale Unstable TRPC6 42 35 Cc1ccccc1/C=C/NC(=O)Nc1ccc2ccccc2c1 ZINC000217684353 DJ For-Sale Unstable IMDH_CRYPV 32 43 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)Nc1ccc(Cl)c(Cl)c1)C2 ZINC000217684373 GG In-Stock Unstable EPHX2 50 56 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)Nc1ccc(Cl)c(Cl)c1)C2 ZINC000217684373 GG In-Stock Unstable VATB 0 41 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)Nc1ccc(Cl)c(Cl)c1)C2 ZINC000217684373 GG In-Stock Unstable ENV 45 35 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)Nc1ccc(Cl)c(Cl)c1)C2 ZINC000217684373 GG In-Stock Unstable P95276_MYCTO 0 45 CS(=O)(=O)N1[C@H]2CC[C@H]1CC(NC(=O)Nc1ccc(Cl)c(Cl)c1)C2 ZINC000217684373 GG In-Stock Unstable PPX1 0 41 COc1ccc(C(=O)NCC(C)C)cc1/C=C\C(=O)O ZINC000217684429 CE For-Sale Unstable F3 87 40 O=C(O)CCNC(=O)c1ccc2c(c1)[C@@H]1C=CC[C@@H]1[C@@H](C(c1ccccc1)c1ccccc1)N2 ZINC000217684475 JK In-Stock Unstable GCGR 41 37 CCC[C@@H](O)CNC(=O)CCCC(=O)O ZINC000217684482 BC On-Demand Unstable PLA2G2C 0 40 CCC[C@@H](O)CNC(=O)CCCC(=O)O ZINC000217684482 BC On-Demand Unstable Q6UB75_PIG 0 40 CCC[C@@H](O)CNC(=O)CCCC(=O)O ZINC000217684482 BC On-Demand Unstable SLC22A20 0 41 COc1ccc(C(=O)NCC(N)=O)cc1/C=C\C(=O)O ZINC000217684515 CC For-Sale Unstable ABCG2 16 46 O=C(O)CCNC(=O)c1ccc2c(c1)[C@@H]1C=CC[C@H]1[C@@H](C(c1ccccc1)c1ccccc1)N2 ZINC000217684551 JK In-Stock Unstable GCGR 41 37 CCC[C@H](O)CNC(=O)CCCC(=O)O ZINC000217684562 BC On-Demand Unstable PLA2G2C 0 40 CCC[C@H](O)CNC(=O)CCCC(=O)O ZINC000217684562 BC On-Demand Unstable Q6UB75_PIG 0 40 CCC[C@H](O)CNC(=O)CCCC(=O)O ZINC000217684562 BC On-Demand Unstable SLC22A20 0 41 O=Cc1ccnc(-c2ccc(OC(F)(F)F)cc2)c1 ZINC000217684567 CG For-Sale Anodyne SCN10A 28 49 COC(=O)[C@@H](O)CNC(=O)Cc1ccccc1OC ZINC000217684578 CB On-Demand Unstable ANPEP 27 48 COC(=O)[C@@H](O)CNC(=O)Cc1ccccc1OC ZINC000217684578 CB On-Demand Unstable TACR1 27 40 COC(=O)[C@@H](O)CNC(=O)Cc1ccccc1OC ZINC000217684578 CB On-Demand Unstable TRPV1 23 40 COC(=O)[C@@H](O)CNC(=O)Cc1ccccc1OC ZINC000217684578 CB On-Demand Unstable KCNA3 19 41 COC(=O)[C@@H](O)CNC(=O)Cc1ccccc1OC ZINC000217684578 CB On-Demand Unstable MBTPS1 42 35 COc1cc2c(c(OC)c1OC)-c1ccc(NCCCC(=O)Nc3ccc(Cn4cncn4)cc3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217684596 KI In-Stock Unstable TUBA1A 15 57 COc1cc2c(c(OC)c1OC)-c1ccc(NCCCC(=O)Nc3ccc(Cn4cncn4)cc3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217684596 KI In-Stock Unstable TPPP 0 54 O=C(O)/C=C\c1ccc(C(=O)N2CCNC(=O)C2)cc1 ZINC000217684597 CC For-Sale Unstable GPR183 0 42 COC(=O)[C@H](O)CNC(=O)Cc1ccccc1OC ZINC000217684674 CB On-Demand Unstable ANPEP 27 48 COC(=O)[C@H](O)CNC(=O)Cc1ccccc1OC ZINC000217684674 CB On-Demand Unstable TACR1 27 40 COC(=O)[C@H](O)CNC(=O)Cc1ccccc1OC ZINC000217684674 CB On-Demand Unstable TRPV1 23 40 COC(=O)[C@H](O)CNC(=O)Cc1ccccc1OC ZINC000217684674 CB On-Demand Unstable KCNA3 19 41 COC(=O)[C@H](O)CNC(=O)Cc1ccccc1OC ZINC000217684674 CB On-Demand Unstable MBTPS1 42 35 O=C(O)/C=C\c1ccc(C(=O)NCCC2CCCC2)s1 ZINC000217684692 CG For-Sale Unstable SIRT3 47 38 O=C(O)/C=C\c1ccc(C(=O)NCCC2CCCC2)s1 ZINC000217684692 CG For-Sale Unstable SIRT2 51 41 O=C(O)/C=C\c1ccc(C(=O)NCCC2CCCC2)s1 ZINC000217684692 CG For-Sale Unstable SIRT1 47 38 O=C(NCCn1ccnc1)[C@H]1[C@H]2C=C[C@@H](C2)[C@H]1C(=O)O ZINC000217684748 CC For-Sale Unstable TBXAS1 32 40 O=C(O)/C=C\c1ccc(C(=O)NCCC2CCCC2)cc1 ZINC000217684780 CG For-Sale Unstable LDLR 0 49 COC(=O)[C@@H](O)CNC(=O)c1ccc(C)c([N+](=O)[O-])c1 ZINC000217684790 CC On-Demand Unstable GSTM2 40 34 CCOC(=O)[C@@H](NC1CCC(C)CC1)c1ccccc1 ZINC000217684821 CG On-Demand Unstable CHRM1 17 40 O=C(CSCCN1CCOCC1)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217684855 HH On-Demand Unstable CASR 32 45 O=C(CSCCN1CCOCC1)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217684855 HH On-Demand Unstable EPHX2 28 48 COC(=O)[C@H](O)CNC(=O)c1ccc(C)c([N+](=O)[O-])c1 ZINC000217684869 CC On-Demand Unstable GSTM2 40 34 O=C(O)/C=C\c1cccc(C(=O)NCCC2CCCC2)c1 ZINC000217684889 CG For-Sale Unstable DRD4 41 31 O=C(O)/C=C\c1cccc(C(=O)NCCC2CCCC2)c1 ZINC000217684889 CG For-Sale Unstable HDAC8 17 42 O=C(O)/C=C\c1cccc(C(=O)NCCC2CCCC2)c1 ZINC000217684889 CG For-Sale Unstable LDLR 0 46 Cc1cc(I)ccc1NC(=O)CSCCN1CCOCC1 ZINC000217684969 HF On-Demand Unstable CNR1 15 40 Cc1ccccc1/C=C/NC(=O)NCCCNC=O ZINC000217685029 CD For-Sale Unstable ACAT 0 43 O=C(c1cc(-c2ccccc2)n2c1NCC2)N1CCCC1 ZINC000217685090 CF In-Stock Unstable NPSR1 15 45 O=C(c1cc(-c2ccccc2)n2c1NCC2)N1CCCC1 ZINC000217685090 CF In-Stock Unstable L3MBTL1 0 41 O=C(c1cc(-c2ccccc2)n2c1NCC2)N1CCCC1 ZINC000217685090 CF In-Stock Unstable L3MBTL3 48 41 O=C(c1cc(-c2ccccc2)n2c1NCC2)N1CCCC1 ZINC000217685090 CF In-Stock Unstable TP53BP1 0 40 COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OCC(=O)O ZINC000217685095 KG In-Stock Unstable ALOX5 0 42 COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OCC(=O)O ZINC000217685095 KG In-Stock Unstable AKR1B1 0 42 COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OCC(=O)O ZINC000217685095 KG In-Stock Unstable CYP1B1 51 39 COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OCC(=O)O ZINC000217685095 KG In-Stock Unstable CYP1A1 49 39 COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OCC(=O)O ZINC000217685095 KG In-Stock Unstable ABCB1A 23 43 Cc1ccccc1C(=O)NCC1C[C@@H]2CC[C@H](C1)N2 ZINC000217685123 CE For-Sale Unstable CCR8 51 35 COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OCC(=O)O ZINC000217685191 KG In-Stock Unstable ALOX5 0 42 COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OCC(=O)O ZINC000217685191 KG In-Stock Unstable AKR1B1 0 42 COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OCC(=O)O ZINC000217685191 KG In-Stock Unstable CYP1B1 51 39 COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OCC(=O)O ZINC000217685191 KG In-Stock Unstable CYP1A1 49 39 COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OCC(=O)O ZINC000217685191 KG In-Stock Unstable ABCB1A 23 43 COc1cccc(N2C[C@@]34C=C[C@@H](O3)[C@@H](C(=O)NCCc3c[nH]c5ccccc35)[C@H]4C2=O)c1 ZINC000217685198 IF In-Stock Unstable NQO2 17 40 COc1cccc(N2C[C@@]34C=C[C@@H](O3)[C@@H](C(=O)NCCc3c[nH]c5ccccc35)[C@H]4C2=O)c1 ZINC000217685198 IF In-Stock Unstable MTNR1A 31 41 COc1cccc(N2C[C@@]34C=C[C@@H](O3)[C@@H](C(=O)NCCc3c[nH]c5ccccc35)[C@H]4C2=O)c1 ZINC000217685198 IF In-Stock Unstable MTNR1B 22 40 COc1cccc(N2C[C@@]34C=C[C@@H](O3)[C@@H](C(=O)NCCc3c[nH]c5ccccc35)[C@H]4C2=O)c1 ZINC000217685198 IF In-Stock Unstable CCKBR 25 41 Clc1ccc(Nc2ncnc(Cl)c2-c2ccccc2)cc1 ZINC000217685210 DK In-Stock Anodyne EGFR 31 45 Clc1ccc(Nc2ncnc(Cl)c2-c2ccccc2)cc1 ZINC000217685210 DK In-Stock Anodyne ADK 26 42 Clc1ccc(Nc2ncnc(Cl)c2-c2ccccc2)cc1 ZINC000217685210 DK In-Stock Anodyne MKNK1 16 45 Cc1ccccc1/C=C/NC(=O)N1C[C@@]2(C)C[C@H]1CC(C)(C)C2 ZINC000217685316 DJ For-Sale Unstable AVPR2 17 53 Cc1ccccc1/C=C/NC(=O)N1C[C@@]2(C)C[C@H]1CC(C)(C)C2 ZINC000217685316 DJ For-Sale Unstable AVPR1A 42 53 COc1ccc(Nc2ncnc(Cl)c2-c2ccccc2)cc1 ZINC000217685319 DJ In-Stock Unstable EGFR 44 50 COc1ccc(Nc2ncnc(Cl)c2-c2ccccc2)cc1 ZINC000217685319 DJ In-Stock Unstable ERBB2 21 45 COc1ccc(Nc2ncnc(Cl)c2-c2ccccc2)cc1 ZINC000217685319 DJ In-Stock Unstable ADK 21 44 COc1ccc(Nc2ncnc(Cl)c2-c2ccccc2)cc1 ZINC000217685319 DJ In-Stock Unstable ABCG2 0 50 COc1ccc(Nc2ncnc(Cl)c2-c2ccccc2)cc1 ZINC000217685319 DJ In-Stock Unstable DYRK1B 19 41 C[C@@H](N[C@@H]1CCN2CCCC[C@@H]12)c1ccc2c(c1)OCO2 ZINC000217685346 CF For-Sale Unstable CHRM2 33 40 C[C@@H](N[C@@H]1CCN2CCCC[C@@H]12)c1ccc2c(c1)OCO2 ZINC000217685346 CF For-Sale Unstable KCNQ2 21 41 Cc1cccc(C(=O)NCC2C[C@@H]3CC[C@H](C2)N3)c1 ZINC000217685382 CE For-Sale Unstable CACNA1I 58 44 Cc1cccc(C(=O)NCC2C[C@@H]3CC[C@H](C2)N3)c1 ZINC000217685382 CE For-Sale Unstable KCNK3 59 43 Cc1cccc(C(=O)NCC2C[C@@H]3CC[C@H](C2)N3)c1 ZINC000217685382 CE For-Sale Unstable KCNK9 48 43 COC(=O)C[C@H](c1cccc(O)c1)c1oc(CN2CCOCC2)cc(=O)c1O ZINC000217685390 GD In-Stock Unstable CASR 43 37 C[C@H](N[C@@H]1CCN2CCCC[C@@H]12)c1ccc2c(c1)OCO2 ZINC000217685430 CF On-Demand Unstable CHRM2 33 40 CSC[C@@](C)(O)CNC(=O)[C@@H](C)Oc1cccc(F)c1 ZINC000217685473 DD On-Demand Unstable PDS 22 40 CN(C[C@@H]1CCCO1)C(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217685475 CE For-Sale Unstable OXTR 29 46 CN(C[C@@H]1CCCO1)C(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217685475 CE For-Sale Unstable AVPR1A 19 43 COC(=O)C[C@@H](c1cccc(O)c1)c1oc(CN2CCOCC2)cc(=O)c1O ZINC000217685481 GD In-Stock Unstable CASR 43 37 C[C@@H](N[C@H]1CCN2CCCC[C@@H]12)c1ccc2c(c1)OCO2 ZINC000217685503 CF For-Sale Unstable CHRM2 33 40 C[C@@H](N[C@H]1CCN2CCCC[C@@H]12)c1ccc2c(c1)OCO2 ZINC000217685503 CF For-Sale Unstable KCNQ2 21 41 Cc1ccccc1/C=C/NC(=O)Nc1cccc(N(C)C)c1 ZINC000217685519 CH For-Sale Unstable KCNK3 71 43 CCOC(=O)[C@@H](c1ccccc1)N1CCC(=O)CC1 ZINC000217685529 CD For-Sale Unstable CHRM2 15 43 CCOC(=O)[C@@H](c1ccccc1)N1CCC(=O)CC1 ZINC000217685529 CD For-Sale Unstable CHRM1 24 53 CCOC(=O)[C@@H](c1ccccc1)N1CCC(=O)CC1 ZINC000217685529 CD For-Sale Unstable SLC6A3 15 43 CCOC(=O)[C@@H](c1ccccc1)N1CCC(=O)CC1 ZINC000217685529 CD For-Sale Unstable CHRM3 24 53 CCOC(=O)[C@@H](c1ccccc1)N1CCC(=O)CC1 ZINC000217685529 CD For-Sale Unstable KCNQ2 42 36 CCOC(=O)[C@@H](c1ccccc1)N1CCC(=O)CC1 ZINC000217685529 CD For-Sale Unstable NPY2R 51 44 CCOC(=O)[C@@H](c1ccccc1)N1CCC(=O)CC1 ZINC000217685529 CD For-Sale Unstable KCNA3 15 40 CSC[C@](C)(O)CNC(=O)[C@@H](C)Oc1cccc(F)c1 ZINC000217685532 DD On-Demand Unstable PDS 22 40 COC(=O)[C@@H](O)CNC(=O)c1cc(OC)ccc1Br ZINC000217685558 EC On-Demand Unstable MTNR1A 49 39 COC(=O)[C@@H](O)CNC(=O)c1cc(OC)ccc1Br ZINC000217685558 EC On-Demand Unstable MTNR1B 41 39 CN(C[C@H]1CCCO1)C(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217685564 CE For-Sale Unstable OXTR 29 46 CN(C[C@H]1CCCO1)C(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217685564 CE For-Sale Unstable AVPR1A 19 43 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1cnco1 ZINC000217685571 CD In-Stock Unstable ACE 50 49 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1cnco1 ZINC000217685571 CD In-Stock Unstable FOLH1 23 43 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1cnco1 ZINC000217685571 CD In-Stock Unstable MME 112 50 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1cnco1 ZINC000217685571 CD In-Stock Unstable ANPEP 96 43 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1cnco1 ZINC000217685571 CD In-Stock Unstable FCER2 60 32 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1cnco1 ZINC000217685571 CD In-Stock Unstable CTSB 40 45 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1cnco1 ZINC000217685571 CD In-Stock Unstable PAPA1_CARPA 49 41 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1cnco1 ZINC000217685571 CD In-Stock Unstable CYSP_TRYCR 49 35 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1cnco1 ZINC000217685571 CD In-Stock Unstable CPA1 63 46 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1cnco1 ZINC000217685571 CD In-Stock Unstable C3AR1 41 34 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1cnco1 ZINC000217685571 CD In-Stock Unstable ITGA4 42 47 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1cnco1 ZINC000217685571 CD In-Stock Unstable CTRB1 33 40 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1cnco1 ZINC000217685571 CD In-Stock Unstable NAALAD2 34 48 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1cnco1 ZINC000217685571 CD In-Stock Unstable CAPNS1 45 37 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1cnco1 ZINC000217685571 CD In-Stock Unstable ECE1 49 44 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1cnco1 ZINC000217685571 CD In-Stock Unstable PAM 0 40 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1cnco1 ZINC000217685571 CD In-Stock Unstable CAPN1 49 47 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1cnco1 ZINC000217685571 CD In-Stock Unstable MMP9 19 44 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1cnco1 ZINC000217685571 CD In-Stock Unstable ACE2 99 44 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1cnco1 ZINC000217685571 CD In-Stock Unstable PIN1 40 35 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1cnco1 ZINC000217685571 CD In-Stock Unstable CPA3 0 40 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1cnco1 ZINC000217685571 CD In-Stock Unstable MMP1 17 40 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1cnco1 ZINC000217685571 CD In-Stock Unstable FPR1 60 43 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1cnco1 ZINC000217685571 CD In-Stock Unstable RHODESAIN 0 44 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1cnco1 ZINC000217685571 CD In-Stock Unstable PSMB5 43 40 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1cnco1 ZINC000217685571 CD In-Stock Unstable SLC15A2 0 51 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1cnco1 ZINC000217685571 CD In-Stock Unstable BLA1_STEMA 82 43 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1cnco1 ZINC000217685571 CD In-Stock Unstable NPFFR1 43 33 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1cnco1 ZINC000217685571 CD In-Stock Unstable BLAIMP-1 0 40 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1cnco1 ZINC000217685571 CD In-Stock Unstable GPR142 57 34 C[C@H](N[C@H]1CCN2CCCC[C@@H]12)c1ccc2c(c1)OCO2 ZINC000217685585 CF On-Demand Unstable CHRM2 33 40 CCOC(=O)[C@H](c1ccccc1)N1CCC(=O)CC1 ZINC000217685609 CD For-Sale Unstable CHRM2 15 43 CCOC(=O)[C@H](c1ccccc1)N1CCC(=O)CC1 ZINC000217685609 CD For-Sale Unstable CHRM1 24 53 CCOC(=O)[C@H](c1ccccc1)N1CCC(=O)CC1 ZINC000217685609 CD For-Sale Unstable SLC6A3 15 43 CCOC(=O)[C@H](c1ccccc1)N1CCC(=O)CC1 ZINC000217685609 CD For-Sale Unstable CHRM3 24 53 CCOC(=O)[C@H](c1ccccc1)N1CCC(=O)CC1 ZINC000217685609 CD For-Sale Unstable KCNQ2 42 36 CCOC(=O)[C@H](c1ccccc1)N1CCC(=O)CC1 ZINC000217685609 CD For-Sale Unstable NPY2R 51 44 CSC[C@@](C)(O)CNC(=O)[C@H](C)Oc1cccc(F)c1 ZINC000217685621 DD On-Demand Unstable PDS 22 40 COC(=O)[C@H](O)CNC(=O)c1cc(OC)ccc1Br ZINC000217685633 EC On-Demand Unstable MTNR1A 49 39 COC(=O)[C@H](O)CNC(=O)c1cc(OC)ccc1Br ZINC000217685633 EC On-Demand Unstable MTNR1B 41 39 Cc1ccccc1/C=C/NC(=O)Nc1nc2c(s1)CN(C)CC2 ZINC000217685638 EG For-Sale Unstable F10 24 45 COc1ccc(C)cc1NC(=O)[C@@H](SCCN1CCOCC1)c1ccccc1 ZINC000217685639 HH On-Demand Unstable CASR 64 42 O=C(C1CCC1)N1CC[C@@H](n2ccnn2)C1 ZINC000217685650 BC In-Stock Unstable L3MBTL3 44 35 Cc1ccc(C(=O)NCC2C[C@@H]3CC[C@H](C2)N3)cc1 ZINC000217685651 CE For-Sale Unstable GRIN2B 16 40 Cc1ccc(C(=O)NCC2C[C@@H]3CC[C@H](C2)N3)cc1 ZINC000217685651 CE For-Sale Unstable CACNA1I 61 44 Nc1nc(-c2ccc(Cl)cc2)ccc1C(=O)O ZINC000217685675 BF In-Stock Unstable DRTS_PLAFK 15 40 Nc1nc(-c2ccc(Cl)cc2)ccc1C(=O)O ZINC000217685675 BF In-Stock Unstable PRS 60 39 Nc1nc(-c2ccc(Cl)cc2)ccc1C(=O)O ZINC000217685675 BF In-Stock Unstable KMO 0 44 Cc1nc(NC(=O)c2cccc(/C=C\C(=O)O)c2)sc1C ZINC000217685679 DG For-Sale Unstable LCK 29 45 Cc1nc(NC(=O)c2cccc(/C=C\C(=O)O)c2)sc1C ZINC000217685679 DG For-Sale Unstable HDAC8 39 44 Cc1nc(NC(=O)c2cccc(/C=C\C(=O)O)c2)sc1C ZINC000217685679 DG For-Sale Unstable HDAC6 23 44 Cc1nc(NC(=O)c2cccc(/C=C\C(=O)O)c2)sc1C ZINC000217685679 DG For-Sale Unstable RHOA 0 40 Cc1nc(NC(=O)c2cccc(/C=C\C(=O)O)c2)sc1C ZINC000217685679 DG For-Sale Unstable KCNK3 77 38 Cc1nc(NC(=O)c2cccc(/C=C\C(=O)O)c2)sc1C ZINC000217685679 DG For-Sale Unstable KCNK9 46 38 CC(C)(C)OC(=O)N1CCC[C@@H]1C1(O)CCCC1 ZINC000217685692 CF For-Sale Unstable PREP 21 56 CSC[C@](C)(O)CNC(=O)[C@H](C)Oc1cccc(F)c1 ZINC000217685709 DD On-Demand Unstable PDS 22 40 CC[C@@H](N[C@@H]1CCN2CCCC[C@@H]12)c1ccc(Cl)cc1 ZINC000217685712 CI For-Sale Unstable SLC6A1 0 41 COc1ccc(C)cc1NC(=O)[C@H](SCCN1CCOCC1)c1ccccc1 ZINC000217685721 HH On-Demand Unstable CASR 64 42 O=C(C1CCC1)N1CC[C@H](n2ccnn2)C1 ZINC000217685730 BC In-Stock Unstable L3MBTL3 44 35 CCCCC[C@@H](C)NC(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217685767 CH For-Sale Unstable NOD1 68 38 CC[C@H](N[C@@H]1CCN2CCCC[C@@H]12)c1ccc(Cl)cc1 ZINC000217685808 CI On-Demand Unstable SLC6A1 0 41 COc1ccc(Cc2nc(C)cc(SCC(=O)O)n2)cc1 ZINC000217685815 DF In-Stock Unstable PTGS2 0 43 COc1ccc(Cc2nc(C)cc(SCC(=O)O)n2)cc1 ZINC000217685815 DF In-Stock Unstable IDH1 20 40 O=C(c1ccccc1F)N1CC[C@H](n2ccnn2)C1 ZINC000217685828 CD In-Stock Unstable L3MBTL1 0 42 O=C(c1ccccc1F)N1CC[C@H](n2ccnn2)C1 ZINC000217685828 CD In-Stock Unstable L3MBTL3 37 42 O=C(c1ccccc1F)N1CC[C@H](n2ccnn2)C1 ZINC000217685828 CD In-Stock Unstable TP53BP1 0 42 CCCCC[C@H](C)NC(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217685864 CH For-Sale Unstable NOD1 68 38 Clc1nc(-c2ccco2)nc2c1oc1ccccc12 ZINC000217685883 CI In-Stock Anodyne PIM3 22 47 O=C(c1ccccc1F)N1CC[C@@H](n2ccnn2)C1 ZINC000217685908 CD In-Stock Unstable L3MBTL1 0 42 O=C(c1ccccc1F)N1CC[C@@H](n2ccnn2)C1 ZINC000217685908 CD In-Stock Unstable L3MBTL3 37 42 O=C(c1ccccc1F)N1CC[C@@H](n2ccnn2)C1 ZINC000217685908 CD In-Stock Unstable TP53BP1 0 42 CC[C@@H](N[C@H]1CCN2CCCC[C@@H]12)c1ccc(Cl)cc1 ZINC000217685913 CI For-Sale Unstable SLC6A1 0 41 COc1ccc(-c2csc(Nc3ccc(C)c(C)c3)n2)cc1N ZINC000217685928 EJ In-Stock Unstable MAOB 0 44 COc1ccc(-c2csc(Nc3ccc(C)c(C)c3)n2)cc1N ZINC000217685928 EJ In-Stock Unstable SPHK2 45 35 COc1ccc(-c2csc(Nc3ccc(C)c(C)c3)n2)cc1N ZINC000217685928 EJ In-Stock Unstable SPHK1 35 40 COc1ccc(-c2csc(Nc3ccc(C)c(C)c3)n2)cc1N ZINC000217685928 EJ In-Stock Unstable PLAU 15 43 COc1ccc(-c2csc(Nc3ccc(C)c(C)c3)n2)cc1N ZINC000217685928 EJ In-Stock Unstable VCP 19 44 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC)cc1F ZINC000217685932 CC On-Demand Unstable MTNR1A 46 39 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC)cc1F ZINC000217685932 CC On-Demand Unstable MTNR1B 40 39 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC)cc1F ZINC000217685932 CC On-Demand Unstable AKR1C2 40 35 CCCCC[C@@H](C)NC(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217685935 CG For-Sale Unstable FOLH1 15 40 CCCCC[C@@H](C)NC(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217685935 CG For-Sale Unstable CTSG 28 43 CCCCC[C@@H](C)NC(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217685935 CG For-Sale Unstable CTRB1 28 43 CCCCC[C@@H](C)NC(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217685935 CG For-Sale Unstable CELA2A 23 43 CC[C@H](N[C@H]1CCN2CCCC[C@@H]12)c1ccc(Cl)cc1 ZINC000217685974 CI On-Demand Unstable SLC6A1 0 41 COc1ccc(NC(=O)[C@@H](SCCN2CCOCC2)c2ccccc2)cc1Cl ZINC000217686014 HI On-Demand Unstable HTR2A 31 40 COc1ccc(NC(=O)[C@@H](SCCN2CCOCC2)c2ccccc2)cc1Cl ZINC000217686014 HI On-Demand Unstable HTR2C 15 42 COc1ccc(NC(=O)[C@@H](SCCN2CCOCC2)c2ccccc2)cc1Cl ZINC000217686014 HI On-Demand Unstable HTR4 30 40 COc1ccc(NC(=O)[C@@H](SCCN2CCOCC2)c2ccccc2)cc1Cl ZINC000217686014 HI On-Demand Unstable CASR 71 46 COc1ccc(NC(=O)[C@@H](SCCN2CCOCC2)c2ccccc2)cc1Cl ZINC000217686014 HI On-Demand Unstable TACR2 27 40 COc1ccc(NC(=O)[C@@H](SCCN2CCOCC2)c2ccccc2)cc1Cl ZINC000217686014 HI On-Demand Unstable NPY2R 53 37 COc1ccc(NC(=O)[C@@H](SCCN2CCOCC2)c2ccccc2)cc1Cl ZINC000217686014 HI On-Demand Unstable EPHX2 22 44 COc1ccc(NC(=O)[C@@H](SCCN2CCOCC2)c2ccccc2)cc1Cl ZINC000217686014 HI On-Demand Unstable MCHR1 15 43 COc1ccc(NC(=O)[C@@H](SCCN2CCOCC2)c2ccccc2)cc1Cl ZINC000217686014 HI On-Demand Unstable ENPP1 54 32 CCCCC[C@H](C)NC(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217686019 CG For-Sale Unstable FOLH1 15 40 CCCCC[C@H](C)NC(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217686019 CG For-Sale Unstable CTSG 28 43 CCCCC[C@H](C)NC(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217686019 CG For-Sale Unstable CTRB1 28 43 CCCCC[C@H](C)NC(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217686019 CG For-Sale Unstable CELA2A 23 43 COC(=O)[C@H](O)CNC(=O)c1ccc(OC)cc1F ZINC000217686021 CC On-Demand Unstable MTNR1A 46 39 COC(=O)[C@H](O)CNC(=O)c1ccc(OC)cc1F ZINC000217686021 CC On-Demand Unstable MTNR1B 40 39 COC(=O)[C@H](O)CNC(=O)c1ccc(OC)cc1F ZINC000217686021 CC On-Demand Unstable AKR1C2 40 35 COc1ccc(-c2csc(Nc3ccccc3C)n2)cc1N ZINC000217686035 DI In-Stock Unstable CCR4 15 46 COc1ccc(-c2csc(Nc3ccccc3C)n2)cc1N ZINC000217686035 DI In-Stock Unstable PLAU 15 44 COc1ccc(-c2csc(Nc3ccccc3C)n2)cc1N ZINC000217686035 DI In-Stock Unstable VCP 16 41 O=C1[C@H]2[C@@H]3C=C[C@@H]([C@H]4C[C@@H]34)[C@H]2C(=O)N1CCc1ccccc1 ZINC000217686067 CE In-Stock Unstable ALDH1A1 25 41 COc1ccc(NC(=O)[C@H](SCCN2CCOCC2)c2ccccc2)cc1Cl ZINC000217686089 HI On-Demand Unstable HTR2A 31 40 COc1ccc(NC(=O)[C@H](SCCN2CCOCC2)c2ccccc2)cc1Cl ZINC000217686089 HI On-Demand Unstable HTR2C 15 42 COc1ccc(NC(=O)[C@H](SCCN2CCOCC2)c2ccccc2)cc1Cl ZINC000217686089 HI On-Demand Unstable HTR4 30 40 COc1ccc(NC(=O)[C@H](SCCN2CCOCC2)c2ccccc2)cc1Cl ZINC000217686089 HI On-Demand Unstable CASR 71 46 COc1ccc(NC(=O)[C@H](SCCN2CCOCC2)c2ccccc2)cc1Cl ZINC000217686089 HI On-Demand Unstable TACR2 27 40 COc1ccc(NC(=O)[C@H](SCCN2CCOCC2)c2ccccc2)cc1Cl ZINC000217686089 HI On-Demand Unstable NPY2R 53 37 COc1ccc(NC(=O)[C@H](SCCN2CCOCC2)c2ccccc2)cc1Cl ZINC000217686089 HI On-Demand Unstable EPHX2 22 44 COc1ccc(NC(=O)[C@H](SCCN2CCOCC2)c2ccccc2)cc1Cl ZINC000217686089 HI On-Demand Unstable MCHR1 15 43 COc1ccc(NC(=O)[C@H](SCCN2CCOCC2)c2ccccc2)cc1Cl ZINC000217686089 HI On-Demand Unstable ENPP1 54 32 CCC(C)(C)NS(=O)(=O)c1ccc(/C=C\C(=O)O)cc1Cl ZINC000217686096 EF For-Sale Unstable NR0B2 0 47 CC(C)(C)c1nc(Cl)c2oc3ccccc3c2n1 ZINC000217686110 CI In-Stock Unstable PIM3 22 45 COc1ccc(CCNC(=O)CCCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@H]23)cc1 ZINC000217686138 JH In-Stock Unstable SCN9A 0 45 COc1ccc(CCNC(=O)CCCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@H]23)cc1 ZINC000217686138 JH In-Stock Unstable MTNR1A 48 38 COc1ccc(CCNC(=O)CCCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@H]23)cc1 ZINC000217686138 JH In-Stock Unstable MTNR1B 41 36 COc1ccc(-c2csc(Nc3ccc(F)cc3)n2)cc1N ZINC000217686141 DI In-Stock Unstable MAOA 0 40 COc1ccc(-c2csc(Nc3ccc(F)cc3)n2)cc1N ZINC000217686141 DI In-Stock Unstable MAOB 30 56 COc1ccc(-c2csc(Nc3ccc(F)cc3)n2)cc1N ZINC000217686141 DI In-Stock Unstable SPHK2 51 36 COc1ccc(-c2csc(Nc3ccc(F)cc3)n2)cc1N ZINC000217686141 DI In-Stock Unstable SPHK1 47 43 COc1ccc(-c2csc(Nc3ccc(F)cc3)n2)cc1N ZINC000217686141 DI In-Stock Unstable PLAU 20 42 COc1ccc(-c2csc(Nc3ccc(F)cc3)n2)cc1N ZINC000217686141 DI In-Stock Unstable VCP 20 49 O=C(O)/C=C\c1cc(Cl)c(S(=O)(=O)NC2CC2)c(Cl)c1 ZINC000217686174 EF For-Sale Unstable SFRP1 44 33 C[C@@H](SCCN1CCOCC1)C(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217686195 GH On-Demand Unstable LTA4H 53 45 C[C@@H](SCCN1CCOCC1)C(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217686195 GH On-Demand Unstable CASR 53 44 C[C@@H](SCCN1CCOCC1)C(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217686195 GH On-Demand Unstable TACR2 33 55 C[C@@H](SCCN1CCOCC1)C(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217686195 GH On-Demand Unstable RAF1 17 41 C[C@@H](SCCN1CCOCC1)C(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217686195 GH On-Demand Unstable NPY5R 0 43 C[C@@H](SCCN1CCOCC1)C(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217686195 GH On-Demand Unstable MAP2K1 18 43 C[C@@H](SCCN1CCOCC1)C(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217686195 GH On-Demand Unstable EPHX2 28 51 C[C@@H](SCCN1CCOCC1)C(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217686195 GH On-Demand Unstable MCHR1 15 44 C[C@@H](SCCN1CCOCC1)C(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217686195 GH On-Demand Unstable Q8MMZ8_EIMTE 25 41 Cc1ccccc1/C=C/NC(=O)Nc1cccc(Br)c1 ZINC000217686206 EJ For-Sale Unstable DDX3X 0 41 Cc1ccccc1/C=C/NC(=O)Nc1cccc(Br)c1 ZINC000217686206 EJ For-Sale Unstable KCNK3 84 39 Cc1ccccc1/C=C/NC(=O)Nc1cccc(Br)c1 ZINC000217686206 EJ For-Sale Unstable KCNK9 49 37 CC[C@H](C(=O)N1CC[C@H](n2ccnn2)C1)c1ccccc1 ZINC000217686219 CE In-Stock Unstable KCNQ2 40 38 COc1ccc(CCNC(=O)CCCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@@H]23)cc1 ZINC000217686226 JH In-Stock Unstable SCN9A 0 45 COc1ccc(CCNC(=O)CCCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@@H]23)cc1 ZINC000217686226 JH In-Stock Unstable MTNR1A 48 38 COc1ccc(CCNC(=O)CCCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@@H]23)cc1 ZINC000217686226 JH In-Stock Unstable MTNR1B 41 36 Cc1nc(CN(C)Cc2ccccc2/C=C\C(=O)O)cs1 ZINC000217686248 DG For-Sale Unstable PTGER2 48 42 Cc1nc(CN(C)Cc2ccccc2/C=C\C(=O)O)cs1 ZINC000217686248 DG For-Sale Unstable PTGER3 19 42 Cc1nc(CN(C)Cc2ccccc2/C=C\C(=O)O)cs1 ZINC000217686248 DG For-Sale Unstable PTGDR 0 41 Cc1cc(S(=O)(=O)NCC2CC2)ccc1/C=C\C(=O)O ZINC000217686258 CD For-Sale Unstable NPY2R 64 43 Cc1cc(S(=O)(=O)NCC2CC2)ccc1/C=C\C(=O)O ZINC000217686258 CD For-Sale Unstable NPY5R 20 43 Cc1cc(S(=O)(=O)NCC2CC2)ccc1/C=C\C(=O)O ZINC000217686258 CD For-Sale Unstable LEF 38 41 C[C@H](SCCN1CCOCC1)C(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217686287 GH On-Demand Unstable LTA4H 53 45 C[C@H](SCCN1CCOCC1)C(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217686287 GH On-Demand Unstable CASR 53 44 C[C@H](SCCN1CCOCC1)C(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217686287 GH On-Demand Unstable TACR2 33 55 C[C@H](SCCN1CCOCC1)C(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217686287 GH On-Demand Unstable RAF1 17 41 C[C@H](SCCN1CCOCC1)C(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217686287 GH On-Demand Unstable NPY5R 0 43 C[C@H](SCCN1CCOCC1)C(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217686287 GH On-Demand Unstable MAP2K1 18 43 C[C@H](SCCN1CCOCC1)C(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217686287 GH On-Demand Unstable EPHX2 28 51 C[C@H](SCCN1CCOCC1)C(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217686287 GH On-Demand Unstable MCHR1 15 44 C[C@H](SCCN1CCOCC1)C(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217686287 GH On-Demand Unstable Q8MMZ8_EIMTE 25 41 CC[C@@H](C(=O)N1CC[C@H](n2ccnn2)C1)c1ccccc1 ZINC000217686301 CE In-Stock Unstable KCNQ2 40 38 Cc1ccc(/C=C\C(=O)O)cc1S(=O)(=O)NCC1CC1 ZINC000217686341 CD For-Sale Unstable NPY2R 61 36 O=C(CCCCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)Nc1nccs1 ZINC000217686349 II In-Stock Unstable MAP 0 41 O=C(CCCCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)Nc1nccs1 ZINC000217686349 II In-Stock Unstable MAP1 60 41 c1ccc(Cn2nnnc2-c2ccccn2)cc1 ZINC000217686360 BD On-Demand Unstable P2RX7 16 45 COc1ccc(-c2csc(Nc3ccccc3)n2)cc1N ZINC000217686374 CI In-Stock Unstable MAOA 0 40 COc1ccc(-c2csc(Nc3ccccc3)n2)cc1N ZINC000217686374 CI In-Stock Unstable MAOB 0 43 COc1ccc(-c2csc(Nc3ccccc3)n2)cc1N ZINC000217686374 CI In-Stock Unstable SPHK2 47 36 COc1ccc(-c2csc(Nc3ccccc3)n2)cc1N ZINC000217686374 CI In-Stock Unstable SPHK1 38 42 COc1ccc(-c2csc(Nc3ccccc3)n2)cc1N ZINC000217686374 CI In-Stock Unstable PLAU 22 46 COc1ccc(-c2csc(Nc3ccccc3)n2)cc1N ZINC000217686374 CI In-Stock Unstable VCP 21 51 CC[C@H](C(=O)N1CC[C@@H](n2ccnn2)C1)c1ccccc1 ZINC000217686381 CE In-Stock Unstable KCNQ2 40 38 O=C(CSCCN1CCOCC1)Nc1ccccc1I ZINC000217686395 HE On-Demand Unstable CASR 49 37 CSC[C@@](C)(O)CNC(=O)Cc1c(C)nn(C)c1C ZINC000217686416 CC On-Demand Unstable P2RX7 30 46 O=C(CCCCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)Nc1nccs1 ZINC000217686426 II In-Stock Unstable MAP 0 41 O=C(CCCCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)Nc1nccs1 ZINC000217686426 II In-Stock Unstable MAP1 60 41 ClCc1nc(Cl)c2oc3ccccc3c2n1 ZINC000217686470 CH In-Stock Unstable PIM3 0 45 CC[C@@H](C(=O)N1CC[C@@H](n2ccnn2)C1)c1ccccc1 ZINC000217686475 CE In-Stock Unstable KCNQ2 40 38 CSC[C@](C)(O)CNC(=O)Cc1c(C)nn(C)c1C ZINC000217686497 CC On-Demand Unstable P2RX7 30 46 CC[C@@H](CCO)NS(=O)(=O)CCCC(=O)O ZINC000217686500 CB For-Sale Unstable CPT1A 17 43 COc1ccc(-c2csc(NS(=O)(=O)c3ccc(C)cc3)n2)cc1N ZINC000217686506 GH In-Stock Unstable MAOA 0 52 COc1ccc(-c2csc(NS(=O)(=O)c3ccc(C)cc3)n2)cc1N ZINC000217686506 GH In-Stock Unstable CA1 15 40 COc1ccc(-c2csc(NS(=O)(=O)c3ccc(C)cc3)n2)cc1N ZINC000217686506 GH In-Stock Unstable CA4 20 40 COc1ccc(-c2csc(NS(=O)(=O)c3ccc(C)cc3)n2)cc1N ZINC000217686506 GH In-Stock Unstable NPY5R 0 40 COc1ccc(-c2csc(NS(=O)(=O)c3ccc(C)cc3)n2)cc1N ZINC000217686506 GH In-Stock Unstable GHSR 0 41 COc1ccc(-c2csc(NS(=O)(=O)c3ccc(C)cc3)n2)cc1N ZINC000217686506 GH In-Stock Unstable SREBF2 0 45 CC(C)[C@@H](CO)NC(=O)CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217686529 HD In-Stock Unstable EDNRA 23 40 CC(C)[C@@H](CO)NC(=O)CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217686529 HD In-Stock Unstable CCKAR 42 36 CC(C)[C@@H](CO)NC(=O)CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217686529 HD In-Stock Unstable GHSR 60 40 Cc1ccccc1/C=C/NC(=O)Nc1ccc(C(C)(C)C)cc1 ZINC000217686531 DK For-Sale Unstable TRPV1 22 44 O=C(O)c1cc(Cl)c(Br)cc1O ZINC000217686552 CF For-Sale Anodyne APP 32 40 O=C(O)c1cc(Cl)c(Br)cc1O ZINC000217686552 CF For-Sale Anodyne AKR1C2 70 44 O=C(O)c1cc(Cl)c(Br)cc1O ZINC000217686552 CF For-Sale Anodyne AKR1C1 67 44 CC[C@H](CCO)NS(=O)(=O)CCCC(=O)O ZINC000217686594 CB For-Sale Unstable CPT1A 17 43 O=C(O)/C=C\c1ccc(S(=O)(=O)NCC(F)(F)F)c(Cl)c1 ZINC000217686608 EE For-Sale Unstable NR0B2 0 40 CC1CCN(C(=O)COc2ccc(C(=N)N)cc2)CC1 ZINC000217686614 CD In-Stock Unstable F2 29 45 CC1CCN(C(=O)COc2ccc(C(=N)N)cc2)CC1 ZINC000217686614 CD In-Stock Unstable PLG 18 40 CC1CCN(C(=O)COc2ccc(C(=N)N)cc2)CC1 ZINC000217686614 CD In-Stock Unstable HTR1D 15 41 CC1CCN(C(=O)COc2ccc(C(=N)N)cc2)CC1 ZINC000217686614 CD In-Stock Unstable HTR1B 18 41 CC1CCN(C(=O)COc2ccc(C(=N)N)cc2)CC1 ZINC000217686614 CD In-Stock Unstable F10 25 45 CC1CCN(C(=O)COc2ccc(C(=N)N)cc2)CC1 ZINC000217686614 CD In-Stock Unstable PRSS2 69 35 CC1CCN(C(=O)COc2ccc(C(=N)N)cc2)CC1 ZINC000217686614 CD In-Stock Unstable SAT1 0 42 CC1CCN(C(=O)COc2ccc(C(=N)N)cc2)CC1 ZINC000217686614 CD In-Stock Unstable CPT1A 63 36 CC1CCN(C(=O)COc2ccc(C(=N)N)cc2)CC1 ZINC000217686614 CD In-Stock Unstable PLAU 36 45 CC1CCN(C(=O)COc2ccc(C(=N)N)cc2)CC1 ZINC000217686614 CD In-Stock Unstable ACR 50 42 CC1CCN(C(=O)COc2ccc(C(=N)N)cc2)CC1 ZINC000217686614 CD In-Stock Unstable ST14 46 45 CC1CCN(C(=O)COc2ccc(C(=N)N)cc2)CC1 ZINC000217686614 CD In-Stock Unstable GPR183 0 42 O=C(CSCCN1CCOCC1)Nc1cccc(I)c1 ZINC000217686615 HE On-Demand Unstable CASR 59 42 O=C(CSCCN1CCOCC1)Nc1cccc(I)c1 ZINC000217686615 HE On-Demand Unstable EPHX2 30 47 COCCCNC(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217686682 CD For-Sale Unstable DRD4 41 31 COCCCNC(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217686682 CD For-Sale Unstable DRD3 28 42 COCCCNC(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217686682 CD For-Sale Unstable REN 15 41 COCCCNC(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217686682 CD For-Sale Unstable HDAC9 15 40 Cc1cc(SCC(=O)O)nc(Cc2ccc(F)cc2)n1 ZINC000217686723 CF In-Stock Unstable ACAT 43 35 CCc1ccc(-c2csc(NC(=O)CSCCN3CCOCC3)n2)cc1 ZINC000217686738 GG On-Demand Unstable CASR 35 47 CCc1ccc(-c2csc(NC(=O)CSCCN3CCOCC3)n2)cc1 ZINC000217686738 GG On-Demand Unstable HDAC9 15 40 CCc1ccc(-c2csc(NC(=O)CSCCN3CCOCC3)n2)cc1 ZINC000217686738 GG On-Demand Unstable TRPA1 21 53 CCC[C@@H]1CC[C@@H](N)[C@@H](CCCc2ccccc2)C1 ZINC000217686789 CJ For-Sale Unstable SLC18A2 43 44 COC(=O)[C@H](C)NC(=O)c1cccc(-c2cc3ccccc3oc2=O)c1 ZINC000217686841 FF In-Stock Unstable MAOB 16 43 COc1ccc(-c2ccc(C(=O)O)c(NC3CCCCC3)n2)cc1 ZINC000217686845 EI In-Stock Unstable MMP13 0 45 COc1ccc(-c2ccc(C(=O)O)c(NC3CCCCC3)n2)cc1 ZINC000217686845 EI In-Stock Unstable CCR4 0 42 COc1ccc(-c2ccc(C(=O)O)c(NC3CCCCC3)n2)cc1 ZINC000217686845 EI In-Stock Unstable SYK 0 41 COc1ccc(-c2ccc(C(=O)O)c(NC3CCCCC3)n2)cc1 ZINC000217686845 EI In-Stock Unstable AKR1C2 50 38 Cc1ccc(-c2cc(NC(=O)CSCCN3CCOCC3)n(-c3ccccc3)n2)cc1 ZINC000217686849 IH On-Demand Unstable TNF 50 45 Cc1ccc(-c2cc(NC(=O)CSCCN3CCOCC3)n(-c3ccccc3)n2)cc1 ZINC000217686849 IH On-Demand Unstable CASR 52 36 Cc1ccc(-c2cc(NC(=O)CSCCN3CCOCC3)n(-c3ccccc3)n2)cc1 ZINC000217686849 IH On-Demand Unstable MAPK14 29 45 Cc1ccc(-c2cc(NC(=O)CSCCN3CCOCC3)n(-c3ccccc3)n2)cc1 ZINC000217686849 IH On-Demand Unstable NR1H4 15 42 Cc1ccc(-c2cc(NC(=O)CSCCN3CCOCC3)n(-c3ccccc3)n2)cc1 ZINC000217686849 IH On-Demand Unstable PTK2B 21 45 Cc1ccc(-c2cc(NC(=O)CSCCN3CCOCC3)n(-c3ccccc3)n2)cc1 ZINC000217686849 IH On-Demand Unstable DDR2 18 45 COC(=O)[C@@H](O)CNC(=O)Cc1ccc(NC(C)=O)cc1 ZINC000217686861 CB On-Demand Unstable PLAU 15 40 COC(=O)[C@@H](O)CNC(=O)Cc1ccc(NC(C)=O)cc1 ZINC000217686861 CB On-Demand Unstable CA9 19 42 CC[C@@H]1CCCCN1C(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217686869 CG For-Sale Unstable ABHD11 0 42 CCC[C@H]1CC[C@@H](N)[C@@H](CCCc2ccccc2)C1 ZINC000217686874 CJ For-Sale Unstable SLC18A2 43 44 COC(=O)[C@H](O)CNC(=O)Cc1ccc(NC(C)=O)cc1 ZINC000217686948 CB On-Demand Unstable PLAU 15 40 COC(=O)[C@H](O)CNC(=O)Cc1ccc(NC(C)=O)cc1 ZINC000217686948 CB On-Demand Unstable CA9 19 42 CCC[C@@H]1CC[C@H](N)[C@@H](CCCc2ccccc2)C1 ZINC000217686952 CJ For-Sale Unstable SLC18A2 43 44 O=C(CN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)Nc1nccs1 ZINC000217686953 GF In-Stock Unstable MAP 0 43 O=C(CN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)Nc1nccs1 ZINC000217686953 GF In-Stock Unstable MAP1 103 38 O=C(CSCCN1CCOCC1)Nc1sc2c(c1C(=O)c1ccccc1)CCCC2 ZINC000217686963 IH On-Demand Unstable CNR1 18 49 O=C(CSCCN1CCOCC1)Nc1sc2c(c1C(=O)c1ccccc1)CCCC2 ZINC000217686963 IH On-Demand Unstable CNR2 15 49 O=C(CSCCN1CCOCC1)Nc1sc2c(c1C(=O)c1ccccc1)CCCC2 ZINC000217686963 IH On-Demand Unstable CASR 48 36 O=C(CSCCN1CCOCC1)Nc1sc2c(c1C(=O)c1ccccc1)CCCC2 ZINC000217686963 IH On-Demand Unstable EPHX2 18 41 O=C(CSCCN1CCOCC1)Nc1sc2c(c1C(=O)c1ccccc1)CCCC2 ZINC000217686963 IH On-Demand Unstable FLT3 19 49 O=C(CSCCN1CCOCC1)Nc1sc2c(c1C(=O)c1ccccc1)CCCC2 ZINC000217686963 IH On-Demand Unstable VIPR1 24 42 CC[C@H]1CCCCN1C(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217686964 CG For-Sale Unstable ABHD11 0 42 CC(C)c1nc(Cl)c2oc3ccccc3c2n1 ZINC000217687006 BI In-Stock Unstable PIM3 0 44 O=C(CN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)Nc1nccs1 ZINC000217687014 GF In-Stock Unstable MAP 0 43 O=C(CN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)Nc1nccs1 ZINC000217687014 GF In-Stock Unstable MAP1 103 38 CCC[C@H]1CC[C@H](N)[C@@H](CCCc2ccccc2)C1 ZINC000217687029 CJ For-Sale Unstable SLC18A2 43 44 CC[C@@H]1CCCCN1C(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217687042 CG For-Sale Unstable L3MBTL3 62 36 CC[C@@H]1CCCCN1C(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217687042 CG For-Sale Unstable ABHD11 0 40 CC[C@@H]1CCCCN1C(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217687042 CG For-Sale Unstable GPR183 0 40 O=Cc1c(N2CCCC2)ncnc1N1CCOCC1 ZINC000217687064 CC In-Stock Unstable LIPA 41 35 O=C(CSCCN1CCOCC1)Nc1cc(-c2ccccc2)nn1-c1ccccc1 ZINC000217687069 HH On-Demand Unstable TNF 29 43 O=C(CSCCN1CCOCC1)Nc1cc(-c2ccccc2)nn1-c1ccccc1 ZINC000217687069 HH On-Demand Unstable CASR 55 39 CC[C@H]1CCCCN1C(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217687130 CG For-Sale Unstable L3MBTL3 62 36 CC[C@H]1CCCCN1C(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217687130 CG For-Sale Unstable ABHD11 0 40 CC[C@H]1CCCCN1C(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217687130 CG For-Sale Unstable GPR183 0 40 Oc1ccc(Cl)cc1CN[C@@H]1CCN2CCCC[C@@H]12 ZINC000217687158 CF On-Demand Unstable SLC18A3 15 41 CCCCCCCCC(=O)NC[C@@](C)(O)CSC ZINC000217687180 CF For-Sale Unstable CNR1 0 51 CCCCCCCCC(=O)NC[C@@](C)(O)CSC ZINC000217687180 CF For-Sale Unstable FAAH 0 51 CCCCCCCCC(=O)NC[C@@](C)(O)CSC ZINC000217687180 CF For-Sale Unstable NOD1 43 35 CCCCCCCCC(=O)NC[C@@](C)(O)CSC ZINC000217687180 CF For-Sale Unstable CQSS 53 33 CC(C)(C)c1cc(NC(=O)CSCCN2CCOCC2)n(-c2ccccc2)n1 ZINC000217687181 HG On-Demand Unstable TNF 64 53 CC(C)(C)c1cc(NC(=O)CSCCN2CCOCC2)n(-c2ccccc2)n1 ZINC000217687181 HG On-Demand Unstable CASR 45 37 CC(C)(C)c1cc(NC(=O)CSCCN2CCOCC2)n(-c2ccccc2)n1 ZINC000217687181 HG On-Demand Unstable MAPK14 37 59 CC(C)(C)c1cc(NC(=O)CSCCN2CCOCC2)n(-c2ccccc2)n1 ZINC000217687181 HG On-Demand Unstable MAPK9 16 53 CC(C)(C)c1cc(NC(=O)CSCCN2CCOCC2)n(-c2ccccc2)n1 ZINC000217687181 HG On-Demand Unstable EPHB2 15 53 CC(C)(C)c1cc(NC(=O)CSCCN2CCOCC2)n(-c2ccccc2)n1 ZINC000217687181 HG On-Demand Unstable ZAK 15 53 CC(C)(C)c1cc(NC(=O)CSCCN2CCOCC2)n(-c2ccccc2)n1 ZINC000217687181 HG On-Demand Unstable STK10 15 53 CC(C)(C)c1cc(NC(=O)CSCCN2CCOCC2)n(-c2ccccc2)n1 ZINC000217687181 HG On-Demand Unstable PTK2B 33 53 CC(C)(C)c1cc(NC(=O)CSCCN2CCOCC2)n(-c2ccccc2)n1 ZINC000217687181 HG On-Demand Unstable DDR2 40 53 CC(C)(C)c1cc(NC(=O)CSCCN2CCOCC2)n(-c2ccccc2)n1 ZINC000217687181 HG On-Demand Unstable CDK8 15 53 Cc1ccccc1/C=C/NC(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000217687187 FE For-Sale Unstable CA2 114 62 Cc1ccccc1/C=C/NC(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000217687187 FE For-Sale Unstable CA1 98 62 Cc1ccccc1/C=C/NC(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000217687187 FE For-Sale Unstable CA7 56 56 Cc1ccccc1/C=C/NC(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000217687187 FE For-Sale Unstable CA5B 57 56 Cc1ccccc1/C=C/NC(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000217687187 FE For-Sale Unstable CA4 74 57 Cc1ccccc1/C=C/NC(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000217687187 FE For-Sale Unstable CA5A 63 56 Cc1ccccc1/C=C/NC(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000217687187 FE For-Sale Unstable CA14 46 53 Cc1ccccc1/C=C/NC(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000217687187 FE For-Sale Unstable CA12 74 62 Cc1ccccc1/C=C/NC(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000217687187 FE For-Sale Unstable CA9 86 62 Cc1ccccc1/C=C/NC(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000217687187 FE For-Sale Unstable CYNT 32 47 Cc1ccccc1/C=C/NC(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000217687187 FE For-Sale Unstable NCE103 35 54 Cc1ccccc1/C=C/NC(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000217687187 FE For-Sale Unstable MTCA1 43 39 Cc1ccccc1/C=C/NC(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000217687187 FE For-Sale Unstable P96878_MYCTU 56 46 Cc1ccccc1/C=C/NC(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000217687187 FE For-Sale Unstable A6YCJ1_9METZ 25 50 CC[C@@H]1CCCCN1C(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217687205 CG For-Sale Unstable PREP 41 44 CC[C@@H]1CCCCN1C(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217687205 CG For-Sale Unstable ABHD11 0 40 CN(CC(=O)O)c1ncc(CN2CCC[C@@H](c3ccc(C(=O)O)cc3)C2)cn1 ZINC000217687253 GE In-Stock Unstable LTA4H 18 41 Oc1ccc(Cl)cc1CN[C@H]1CCN2CCCC[C@@H]12 ZINC000217687257 CF On-Demand Unstable SLC18A3 15 41 CCCCCCCCC(=O)NC[C@](C)(O)CSC ZINC000217687272 CF For-Sale Unstable CNR1 0 51 CCCCCCCCC(=O)NC[C@](C)(O)CSC ZINC000217687272 CF For-Sale Unstable FAAH 0 51 CCCCCCCCC(=O)NC[C@](C)(O)CSC ZINC000217687272 CF For-Sale Unstable NOD1 43 35 CCCCCCCCC(=O)NC[C@](C)(O)CSC ZINC000217687272 CF For-Sale Unstable CQSS 53 33 Cc1ccccc1/C=C/NC(=O)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217687298 GK For-Sale Unstable PTPA 0 45 CC[C@H]1CCCCN1C(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217687305 CG For-Sale Unstable PREP 41 44 CC[C@H]1CCCCN1C(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217687305 CG For-Sale Unstable ABHD11 0 40 Cc1cc(=O)c(O)c([C@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccccc2)o1 ZINC000217687330 II In-Stock Unstable SSTR4 44 34 CC1CCN(C(=O)c2cc(/C=C\C(=O)O)ccc2F)CC1 ZINC000217687384 CF For-Sale Unstable CCR2 54 40 CC1CCN(C(=O)c2cc(/C=C\C(=O)O)ccc2F)CC1 ZINC000217687384 CF For-Sale Unstable PARP1 44 34 CC1CCN(C(=O)c2cc(/C=C\C(=O)O)ccc2F)CC1 ZINC000217687384 CF For-Sale Unstable TRPC6 27 41 Cc1cc(=O)c(O)c([C@@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccccc2)o1 ZINC000217687396 II In-Stock Unstable SSTR4 44 34 COc1cccc(Nc2ncnc(Cl)c2-c2ccccc2)c1 ZINC000217687426 DJ In-Stock Unstable ABL1 0 51 COc1cccc(Nc2ncnc(Cl)c2-c2ccccc2)c1 ZINC000217687426 DJ In-Stock Unstable EGFR 86 58 COc1cccc(Nc2ncnc(Cl)c2-c2ccccc2)c1 ZINC000217687426 DJ In-Stock Unstable ERBB2 32 43 COc1cccc(Nc2ncnc(Cl)c2-c2ccccc2)c1 ZINC000217687426 DJ In-Stock Unstable PIK3R1 0 41 COc1cccc(Nc2ncnc(Cl)c2-c2ccccc2)c1 ZINC000217687426 DJ In-Stock Unstable FBP1 22 46 COc1cccc(Nc2ncnc(Cl)c2-c2ccccc2)c1 ZINC000217687426 DJ In-Stock Unstable MKNK1 23 46 COc1cccc(Nc2ncnc(Cl)c2-c2ccccc2)c1 ZINC000217687426 DJ In-Stock Unstable AHK4 0 47 COc1cccc(Nc2ncnc(Cl)c2-c2ccccc2)c1 ZINC000217687426 DJ In-Stock Unstable AHK3 0 54 COc1cccc(Nc2ncnc(Cl)c2-c2ccccc2)c1 ZINC000217687426 DJ In-Stock Unstable CKX2 0 47 CC[C@H]1C(=O)N[C@H]1Cc1ccccc1 ZINC000217687455 AD For-Sale Unstable SLC18A2 28 40 CC[C@H]1C(=O)N[C@H]1Cc1ccccc1 ZINC000217687455 AD For-Sale Unstable GALR1 58 46 CC[C@H]1C(=O)N[C@H]1Cc1ccccc1 ZINC000217687455 AD For-Sale Unstable GALR2 27 46 CC[C@H]1C(=O)N[C@H]1Cc1ccccc1 ZINC000217687455 AD For-Sale Unstable PROTEASE 0 44 COC(=O)[C@@H](O)CNC(=O)c1ccc(SC)cc1 ZINC000217687457 CC On-Demand Unstable ITGAV 40 36 CC1CCN(C(=O)c2ccc(/C=C\C(=O)O)cc2F)CC1 ZINC000217687471 CF For-Sale Unstable CCR2 63 40 CC[C@H](C)[C@H](NC(=O)CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)c1nc2ccccc2[nH]1 ZINC000217687483 IG In-Stock Unstable PLCD1 0 41 CC[C@H](C)[C@H](NC(=O)CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)c1nc2ccccc2[nH]1 ZINC000217687483 IG In-Stock Unstable AGAL_COFAR 0 44 CC[C@H](C)[C@H](NC(=O)CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)c1nc2ccccc2[nH]1 ZINC000217687483 IG In-Stock Unstable CYTH3 0 41 CC[C@H](C)[C@H](NC(=O)CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)c1nc2ccccc2[nH]1 ZINC000217687483 IG In-Stock Unstable HLCS 0 45 CC[C@H](C)[C@H](NC(=O)CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)c1nc2ccccc2[nH]1 ZINC000217687483 IG In-Stock Unstable BIRA 0 42 O=C(c1ccc(-n2cccc2)cc1)N1CC[C@H](n2ccnn2)C1 ZINC000217687506 DE In-Stock Unstable L3MBTL1 0 45 O=C(c1ccc(-n2cccc2)cc1)N1CC[C@H](n2ccnn2)C1 ZINC000217687506 DE In-Stock Unstable L3MBTL3 69 45 O=C(c1ccc(-n2cccc2)cc1)N1CC[C@H](n2ccnn2)C1 ZINC000217687506 DE In-Stock Unstable L3MBTL4 0 41 O=C(c1ccc(-n2cccc2)cc1)N1CC[C@H](n2ccnn2)C1 ZINC000217687506 DE In-Stock Unstable MBTD1 0 41 O=C(c1ccc(-n2cccc2)cc1)N1CC[C@H](n2ccnn2)C1 ZINC000217687506 DE In-Stock Unstable TP53BP1 0 41 O=C(c1ccc(-n2cccc2)cc1)N1CC[C@H](n2ccnn2)C1 ZINC000217687506 DE In-Stock Unstable SLC6A7 0 49 O=C(Nc1ccccc1C(=O)O)c1cnco1 ZINC000217687511 BD In-Stock Anodyne HCAR2 41 42 O=C(Nc1ccccc1C(=O)O)c1cnco1 ZINC000217687511 BD In-Stock Anodyne AKR1C2 44 43 CC[C@H]1C(=O)N[C@@H]1Cc1ccccc1 ZINC000217687537 AD For-Sale Unstable SLC18A2 28 40 CC[C@H]1C(=O)N[C@@H]1Cc1ccccc1 ZINC000217687537 AD For-Sale Unstable GALR1 58 46 CC[C@H]1C(=O)N[C@@H]1Cc1ccccc1 ZINC000217687537 AD For-Sale Unstable GALR2 27 46 CC[C@H]1C(=O)N[C@@H]1Cc1ccccc1 ZINC000217687537 AD For-Sale Unstable PROTEASE 0 44 COC(=O)[C@H](O)CNC(=O)c1ccc(SC)cc1 ZINC000217687548 CC On-Demand Unstable ITGAV 40 36 CN(C)[C@@H]1CCCN(c2ccc(CBr)cn2)C1 ZINC000217687557 CF For-Sale Unstable MCHR1 0 44 COc1ccc(C(=O)NC(C)(C)C)cc1/C=C\C(=O)O ZINC000217687559 CE For-Sale Unstable LTB4R 22 40 COc1ccc(C(=O)NC(C)(C)C)cc1/C=C\C(=O)O ZINC000217687559 CE For-Sale Unstable CPT1A 20 45 COc1ccc(C(=O)NC(C)(C)C)cc1/C=C\C(=O)O ZINC000217687559 CE For-Sale Unstable TNFRSF1A 24 42 O=C(c1ccc(-n2cccc2)cc1)N1CC[C@@H](n2ccnn2)C1 ZINC000217687580 DE In-Stock Unstable L3MBTL1 0 45 O=C(c1ccc(-n2cccc2)cc1)N1CC[C@@H](n2ccnn2)C1 ZINC000217687580 DE In-Stock Unstable L3MBTL3 69 45 O=C(c1ccc(-n2cccc2)cc1)N1CC[C@@H](n2ccnn2)C1 ZINC000217687580 DE In-Stock Unstable L3MBTL4 0 41 O=C(c1ccc(-n2cccc2)cc1)N1CC[C@@H](n2ccnn2)C1 ZINC000217687580 DE In-Stock Unstable MBTD1 0 41 O=C(c1ccc(-n2cccc2)cc1)N1CC[C@@H](n2ccnn2)C1 ZINC000217687580 DE In-Stock Unstable TP53BP1 0 41 O=C(c1ccc(-n2cccc2)cc1)N1CC[C@@H](n2ccnn2)C1 ZINC000217687580 DE In-Stock Unstable SLC6A7 0 49 COc1ccc2[nH]cc(-c3csc(NC(=O)CCCCCNc4ccc5c(cc4=O)[C@@H](NC(C)=O)CCc4cc(OC)c(OC)c(OC)c4-5)n3)c2c1 ZINC000217687591 KK In-Stock Unstable TUBA1A 15 52 C[C@@H](SCCN1CCOCC1)C(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217687595 HH On-Demand Unstable LTA4H 49 48 C[C@@H](SCCN1CCOCC1)C(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217687595 HH On-Demand Unstable CASR 56 40 C[C@@H](SCCN1CCOCC1)C(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217687595 HH On-Demand Unstable TACR2 35 55 C[C@@H](SCCN1CCOCC1)C(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217687595 HH On-Demand Unstable MMP13 19 41 C[C@@H](SCCN1CCOCC1)C(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217687595 HH On-Demand Unstable CTSK 18 41 C[C@@H](SCCN1CCOCC1)C(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217687595 HH On-Demand Unstable SCN2A 19 43 C[C@@H](SCCN1CCOCC1)C(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217687595 HH On-Demand Unstable ADAM17 31 43 C[C@@H](SCCN1CCOCC1)C(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217687595 HH On-Demand Unstable MMP2 18 43 C[C@@H](SCCN1CCOCC1)C(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217687595 HH On-Demand Unstable MMP3 16 40 C[C@@H](SCCN1CCOCC1)C(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217687595 HH On-Demand Unstable CAPN1 21 41 C[C@@H](SCCN1CCOCC1)C(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217687595 HH On-Demand Unstable MMP9 17 43 C[C@@H](SCCN1CCOCC1)C(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217687595 HH On-Demand Unstable CAPN2 25 41 C[C@@H](SCCN1CCOCC1)C(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217687595 HH On-Demand Unstable EPHX2 29 55 C[C@@H](SCCN1CCOCC1)C(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217687595 HH On-Demand Unstable ADAMTS4 40 35 C[C@@H](SCCN1CCOCC1)C(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217687595 HH On-Demand Unstable NPR 57 33 CC[C@@H]1C(=O)N[C@@H]1Cc1ccccc1 ZINC000217687606 AD For-Sale Unstable SLC18A2 28 40 CC[C@@H]1C(=O)N[C@@H]1Cc1ccccc1 ZINC000217687606 AD For-Sale Unstable GALR1 58 46 CC[C@@H]1C(=O)N[C@@H]1Cc1ccccc1 ZINC000217687606 AD For-Sale Unstable GALR2 27 46 CC[C@@H]1C(=O)N[C@@H]1Cc1ccccc1 ZINC000217687606 AD For-Sale Unstable PROTEASE 0 44 COc1cccc(Nc2nc(-c3ccc(OC)c(N)c3)cs2)c1 ZINC000217687641 EI In-Stock Unstable MAOA 21 48 COc1cccc(Nc2nc(-c3ccc(OC)c(N)c3)cs2)c1 ZINC000217687641 EI In-Stock Unstable MAOB 26 48 CN(C)[C@H]1CCCN(c2ccc(CBr)cn2)C1 ZINC000217687647 CF For-Sale Unstable MCHR1 0 44 C[C@H](SCCN1CCOCC1)C(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217687672 HH On-Demand Unstable LTA4H 49 48 C[C@H](SCCN1CCOCC1)C(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217687672 HH On-Demand Unstable CASR 56 40 C[C@H](SCCN1CCOCC1)C(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217687672 HH On-Demand Unstable TACR2 35 55 C[C@H](SCCN1CCOCC1)C(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217687672 HH On-Demand Unstable MMP13 19 41 C[C@H](SCCN1CCOCC1)C(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217687672 HH On-Demand Unstable CTSK 18 41 C[C@H](SCCN1CCOCC1)C(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217687672 HH On-Demand Unstable SCN2A 19 43 C[C@H](SCCN1CCOCC1)C(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217687672 HH On-Demand Unstable ADAM17 31 43 C[C@H](SCCN1CCOCC1)C(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217687672 HH On-Demand Unstable MMP2 18 43 C[C@H](SCCN1CCOCC1)C(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217687672 HH On-Demand Unstable MMP3 16 40 C[C@H](SCCN1CCOCC1)C(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217687672 HH On-Demand Unstable CAPN1 21 41 C[C@H](SCCN1CCOCC1)C(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217687672 HH On-Demand Unstable MMP9 17 43 C[C@H](SCCN1CCOCC1)C(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217687672 HH On-Demand Unstable CAPN2 25 41 C[C@H](SCCN1CCOCC1)C(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217687672 HH On-Demand Unstable EPHX2 29 55 C[C@H](SCCN1CCOCC1)C(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217687672 HH On-Demand Unstable ADAMTS4 40 35 C[C@H](SCCN1CCOCC1)C(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217687672 HH On-Demand Unstable NPR 57 33 O=C(O)/C=C\c1ccc(F)c(C(=O)N2CCNC(=O)C2)c1 ZINC000217687721 CC For-Sale Unstable PARP1 49 46 Cc1ccccc1/C=C/NC(=O)Nc1ccc(F)c(Cl)c1 ZINC000217687726 DJ For-Sale Unstable P95276_MYCTO 0 42 Cc1ccc2nc(-c3ccc(NC(=O)[C@@H](C)SCCN4CCOCC4)cc3)sc2c1 ZINC000217687800 IJ On-Demand Unstable CASR 53 46 Cc1ccc2nc(-c3ccc(NC(=O)[C@@H](C)SCCN4CCOCC4)cc3)sc2c1 ZINC000217687800 IJ On-Demand Unstable APP 23 45 CCCNc1ncnc(Cl)c1-c1ccccc1 ZINC000217687837 BH In-Stock Unstable HTT 0 41 CCN(CC)c1ccc(NC(=O)N/C=C/c2ccccc2C)cc1 ZINC000217687842 DJ For-Sale Unstable GHSR 0 43 Cc1ccc2nc(-c3ccc(NC(=O)[C@H](C)SCCN4CCOCC4)cc3)sc2c1 ZINC000217687872 IJ On-Demand Unstable CASR 53 46 Cc1ccc2nc(-c3ccc(NC(=O)[C@H](C)SCCN4CCOCC4)cc3)sc2c1 ZINC000217687872 IJ On-Demand Unstable APP 23 45 O=C(c1ccoc1)N1CC[C@H](n2ccnn2)C1 ZINC000217687879 BC In-Stock Unstable L3MBTL1 0 41 O=C(c1ccoc1)N1CC[C@H](n2ccnn2)C1 ZINC000217687879 BC In-Stock Unstable L3MBTL3 56 41 COC(=O)[C@@H](O)CNC(=O)c1ccccc1[N+](=O)[O-] ZINC000217687887 CB On-Demand Unstable CCR3 0 41 COC(=O)[C@@H](O)CNC(=O)c1ccccc1[N+](=O)[O-] ZINC000217687887 CB On-Demand Unstable COLA 95 37 COC(=O)[C@@H](O)CNC(=O)c1ccccc1[N+](=O)[O-] ZINC000217687887 CB On-Demand Unstable KCNMA1 18 40 COC(=O)[C@@H](O)CNC(=O)c1ccccc1[N+](=O)[O-] ZINC000217687887 CB On-Demand Unstable DAC 17 57 O=C(O)/C=C\c1ccc(C(=O)NCCC2CCCCC2)s1 ZINC000217687903 DH For-Sale Unstable SIRT3 46 38 O=C(O)/C=C\c1ccc(C(=O)NCCC2CCCCC2)s1 ZINC000217687903 DH For-Sale Unstable SIRT2 50 41 O=C(O)/C=C\c1ccc(C(=O)NCCC2CCCCC2)s1 ZINC000217687903 DH For-Sale Unstable SIRT1 46 38 CSC[C@@](C)(O)CNC(=O)c1ccc(NS(C)(=O)=O)cc1 ZINC000217687925 EC On-Demand Unstable TRPV1 22 47 Nc1ncncc1C(=O)OCc1ccccc1 ZINC000217687933 BD In-Stock Unstable 17HSDCL 0 43 Cc1ccccc1/C=C/NC(=O)NCc1ccc(F)cc1 ZINC000217687936 CH For-Sale Unstable ANPEP 16 42 Cc1ccccc1/C=C/NC(=O)NCc1ccc(F)cc1 ZINC000217687936 CH For-Sale Unstable AMP1_PLAFQ 15 42 Fc1cccc(Nc2ncnc(Cl)c2-c2ccccc2)c1 ZINC000217687945 CJ In-Stock Anodyne EGFR 83 56 Fc1cccc(Nc2ncnc(Cl)c2-c2ccccc2)c1 ZINC000217687945 CJ In-Stock Anodyne ERBB2 50 38 Fc1cccc(Nc2ncnc(Cl)c2-c2ccccc2)c1 ZINC000217687945 CJ In-Stock Anodyne CD38 18 44 Fc1cccc(Nc2ncnc(Cl)c2-c2ccccc2)c1 ZINC000217687945 CJ In-Stock Anodyne AHK3 0 44 Fc1cccc(Nc2ncnc(Cl)c2-c2ccccc2)c1 ZINC000217687945 CJ In-Stock Anodyne CKX2 0 44 O=C(c1ccoc1)N1CC[C@@H](n2ccnn2)C1 ZINC000217687949 BC In-Stock Unstable L3MBTL1 0 41 O=C(c1ccoc1)N1CC[C@@H](n2ccnn2)C1 ZINC000217687949 BC In-Stock Unstable L3MBTL3 56 41 COC(=O)[C@H](O)CNC(=O)c1ccccc1[N+](=O)[O-] ZINC000217687966 CB On-Demand Unstable CCR3 0 41 COC(=O)[C@H](O)CNC(=O)c1ccccc1[N+](=O)[O-] ZINC000217687966 CB On-Demand Unstable COLA 95 37 COC(=O)[C@H](O)CNC(=O)c1ccccc1[N+](=O)[O-] ZINC000217687966 CB On-Demand Unstable KCNMA1 18 40 COC(=O)[C@H](O)CNC(=O)c1ccccc1[N+](=O)[O-] ZINC000217687966 CB On-Demand Unstable DAC 17 57 CCn1c2ccccc2c2cc(NC(=O)[C@@H](C)SCCN3CCOCC3)ccc21 ZINC000217687972 HI On-Demand Unstable CNR1 21 46 CCn1c2ccccc2c2cc(NC(=O)[C@@H](C)SCCN3CCOCC3)ccc21 ZINC000217687972 HI On-Demand Unstable CNR2 25 46 CCn1c2ccccc2c2cc(NC(=O)[C@@H](C)SCCN3CCOCC3)ccc21 ZINC000217687972 HI On-Demand Unstable CASR 43 37 CCn1c2ccccc2c2cc(NC(=O)[C@@H](C)SCCN3CCOCC3)ccc21 ZINC000217687972 HI On-Demand Unstable NPY2R 25 68 CCn1c2ccccc2c2cc(NC(=O)[C@@H](C)SCCN3CCOCC3)ccc21 ZINC000217687972 HI On-Demand Unstable ADCY5 19 40 CCn1c2ccccc2c2cc(NC(=O)[C@@H](C)SCCN3CCOCC3)ccc21 ZINC000217687972 HI On-Demand Unstable NPY5R 16 56 CCn1c2ccccc2c2cc(NC(=O)[C@@H](C)SCCN3CCOCC3)ccc21 ZINC000217687972 HI On-Demand Unstable PTGDS 47 40 CCn1c2ccccc2c2cc(NC(=O)[C@@H](C)SCCN3CCOCC3)ccc21 ZINC000217687972 HI On-Demand Unstable MCHR2 45 38 CCn1c2ccccc2c2cc(NC(=O)[C@@H](C)SCCN3CCOCC3)ccc21 ZINC000217687972 HI On-Demand Unstable RAC1 0 47 CSC[C@](C)(O)CNC(=O)c1ccc(NS(C)(=O)=O)cc1 ZINC000217688012 EC On-Demand Unstable TRPV1 22 47 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2C)CC1 ZINC000217688044 FH For-Sale Unstable DRD1 35 42 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2C)CC1 ZINC000217688044 FH For-Sale Unstable DRD3 24 41 CCn1c2ccccc2c2cc(NC(=O)[C@H](C)SCCN3CCOCC3)ccc21 ZINC000217688049 HI On-Demand Unstable CNR1 21 46 CCn1c2ccccc2c2cc(NC(=O)[C@H](C)SCCN3CCOCC3)ccc21 ZINC000217688049 HI On-Demand Unstable CNR2 25 46 CCn1c2ccccc2c2cc(NC(=O)[C@H](C)SCCN3CCOCC3)ccc21 ZINC000217688049 HI On-Demand Unstable CASR 43 37 CCn1c2ccccc2c2cc(NC(=O)[C@H](C)SCCN3CCOCC3)ccc21 ZINC000217688049 HI On-Demand Unstable NPY2R 25 68 CCn1c2ccccc2c2cc(NC(=O)[C@H](C)SCCN3CCOCC3)ccc21 ZINC000217688049 HI On-Demand Unstable ADCY5 19 40 CCn1c2ccccc2c2cc(NC(=O)[C@H](C)SCCN3CCOCC3)ccc21 ZINC000217688049 HI On-Demand Unstable NPY5R 16 56 CCn1c2ccccc2c2cc(NC(=O)[C@H](C)SCCN3CCOCC3)ccc21 ZINC000217688049 HI On-Demand Unstable PTGDS 47 40 CCn1c2ccccc2c2cc(NC(=O)[C@H](C)SCCN3CCOCC3)ccc21 ZINC000217688049 HI On-Demand Unstable MCHR2 45 38 CCn1c2ccccc2c2cc(NC(=O)[C@H](C)SCCN3CCOCC3)ccc21 ZINC000217688049 HI On-Demand Unstable RAC1 0 47 COC(=O)[C@@H](O)CNC(=O)c1cccc([N+](=O)[O-])c1C ZINC000217688060 CC On-Demand Unstable CACNA1D 62 33 COC(=O)[C@@H](O)CNC(=O)c1cccc([N+](=O)[O-])c1C ZINC000217688060 CC On-Demand Unstable COLA 83 33 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)Nc3cccc4c3ccn4C(C)C)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217688063 KK In-Stock Unstable TUBA1A 17 60 C[C@H]1CN(S(=O)(=O)c2cccc([C@H](C)O)c2)CCCO1 ZINC000217688122 CD For-Sale Unstable AKR1C3 51 35 COC(=O)[C@H](O)CNC(=O)c1cccc([N+](=O)[O-])c1C ZINC000217688153 CC On-Demand Unstable CACNA1D 62 33 COC(=O)[C@H](O)CNC(=O)c1cccc([N+](=O)[O-])c1C ZINC000217688153 CC On-Demand Unstable COLA 83 33 CCN(C[C@@H]1CCCO1)C(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217688155 DE For-Sale Unstable OXTR 27 42 CCN(C[C@@H]1CCCO1)C(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217688155 DE For-Sale Unstable AVPR1A 0 40 COc1ccccc1N1C[C@H](C(=O)NC[C@@H]2CCCN3CCCC[C@H]23)CC1=O ZINC000217688178 GE In-Stock Unstable HTR1A 41 43 COc1ccccc1N1C[C@H](C(=O)NC[C@@H]2CCCN3CCCC[C@H]23)CC1=O ZINC000217688178 GE In-Stock Unstable DRD2 40 47 COc1ccccc1N1C[C@H](C(=O)NC[C@@H]2CCCN3CCCC[C@H]23)CC1=O ZINC000217688178 GE In-Stock Unstable DRD4 20 42 COc1ccccc1N1C[C@H](C(=O)NC[C@@H]2CCCN3CCCC[C@H]23)CC1=O ZINC000217688178 GE In-Stock Unstable HTR2A 18 43 COc1ccccc1N1C[C@H](C(=O)NC[C@@H]2CCCN3CCCC[C@H]23)CC1=O ZINC000217688178 GE In-Stock Unstable ADRA1A 36 41 Cn1c(C(=O)NCCc2noc(C3CCC3)n2)cc2ccccc21 ZINC000217688234 DF In-Stock Unstable SMO 50 40 CCN(C[C@H]1CCCO1)C(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217688244 DE For-Sale Unstable OXTR 27 42 CCN(C[C@H]1CCCO1)C(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217688244 DE For-Sale Unstable AVPR1A 0 40 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC)c(OC)c1 ZINC000217688256 CB On-Demand Unstable F3 62 38 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC)c(OC)c1 ZINC000217688256 CB On-Demand Unstable MT-ND1 26 43 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC)c(OC)c1 ZINC000217688256 CB On-Demand Unstable ABCG2 19 44 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC)c(OC)c1 ZINC000217688256 CB On-Demand Unstable ENPP1 53 31 COc1ccccc1N1C[C@@H](C(=O)NC[C@@H]2CCCN3CCCC[C@H]23)CC1=O ZINC000217688266 GE In-Stock Unstable HTR1A 53 48 COc1ccccc1N1C[C@@H](C(=O)NC[C@@H]2CCCN3CCCC[C@H]23)CC1=O ZINC000217688266 GE In-Stock Unstable DRD2 46 47 COc1ccccc1N1C[C@@H](C(=O)NC[C@@H]2CCCN3CCCC[C@H]23)CC1=O ZINC000217688266 GE In-Stock Unstable DRD4 23 42 COc1ccccc1N1C[C@@H](C(=O)NC[C@@H]2CCCN3CCCC[C@H]23)CC1=O ZINC000217688266 GE In-Stock Unstable ADRA1D 41 36 COc1ccccc1N1C[C@@H](C(=O)NC[C@@H]2CCCN3CCCC[C@H]23)CC1=O ZINC000217688266 GE In-Stock Unstable HTR2A 18 43 COc1ccccc1N1C[C@@H](C(=O)NC[C@@H]2CCCN3CCCC[C@H]23)CC1=O ZINC000217688266 GE In-Stock Unstable ADRA1A 37 41 COc1ccccc1N1C[C@@H](C(=O)NC[C@@H]2CCCN3CCCC[C@H]23)CC1=O ZINC000217688266 GE In-Stock Unstable DRD3 49 39 COc1ccccc1N1C[C@@H](C(=O)NC[C@@H]2CCCN3CCCC[C@H]23)CC1=O ZINC000217688266 GE In-Stock Unstable SLC18A3 28 40 OCc1ccn(Cc2ccc(Cl)cc2)n1 ZINC000217688274 BE In-Stock Unstable HDAC7 21 45 CC[C@@H](O)c1cccc(S(=O)(=O)N2CCCO[C@@H](C)C2)c1 ZINC000217688282 DD For-Sale Unstable AKR1C3 41 34 Clc1ncnc(NC2CC2)c1-c1ccccc1 ZINC000217688288 BG In-Stock Unstable TNK2 44 37 CCC[C@@H](N[C@@H]1CCN2CCC[C@@H]12)c1ccc(Cl)cc1 ZINC000217688293 CI For-Sale Unstable SLC6A1 0 42 CN(C[C@@H]1CCCO1)C(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217688334 CE For-Sale Unstable OXTR 27 43 CN(C[C@@H]1CCCO1)C(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217688334 CE For-Sale Unstable AVPR1A 18 43 COC(=O)[C@H](O)CNC(=O)c1ccc(OC)c(OC)c1 ZINC000217688342 CB On-Demand Unstable F3 62 38 COC(=O)[C@H](O)CNC(=O)c1ccc(OC)c(OC)c1 ZINC000217688342 CB On-Demand Unstable MT-ND1 26 43 COC(=O)[C@H](O)CNC(=O)c1ccc(OC)c(OC)c1 ZINC000217688342 CB On-Demand Unstable ABCG2 19 44 COC(=O)[C@H](O)CNC(=O)c1ccc(OC)c(OC)c1 ZINC000217688342 CB On-Demand Unstable ENPP1 53 31 CC[C@H](O)c1cccc(S(=O)(=O)N2CCCO[C@@H](C)C2)c1 ZINC000217688360 DD For-Sale Unstable AKR1C3 41 34 CCC[C@H](N[C@@H]1CCN2CCC[C@@H]12)c1ccc(Cl)cc1 ZINC000217688381 CI For-Sale Unstable SLC6A1 0 42 OCc1ccn(Cc2cccc(Cl)c2)n1 ZINC000217688395 BE In-Stock Unstable HDAC7 21 41 CN(C[C@H]1CCCO1)C(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217688430 CE For-Sale Unstable OXTR 27 43 CN(C[C@H]1CCCO1)C(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217688430 CE For-Sale Unstable AVPR1A 18 43 Cc1ccccc1/C=C/NC(=O)NC1CCCCCC1 ZINC000217688437 CH For-Sale Unstable FAAH 15 40 Cc1ccccc1/C=C/NC(=O)NC1CCCCCC1 ZINC000217688437 CH For-Sale Unstable EPHX2 29 48 CCC[C@@H](N[C@H]1CCN2CCC[C@@H]12)c1ccc(Cl)cc1 ZINC000217688449 CI For-Sale Unstable SLC6A1 0 42 O=C(CSCCN1CCOCC1)Nc1cc(C(F)(F)F)ccc1-n1cncn1 ZINC000217688465 HE On-Demand Unstable EPHX2 16 40 O=C(Nc1cccc(Cl)c1)N1CC[C@H](n2ccnn2)C1 ZINC000217688479 CE In-Stock Unstable FAAH 17 45 O=C(Nc1cccc(Cl)c1)N1CC[C@H](n2ccnn2)C1 ZINC000217688479 CE In-Stock Unstable EPHX2 17 48 N=C(N)c1ccc(OCC(=O)N2CCCCC2)cc1 ZINC000217688524 CD In-Stock Unstable F2 18 46 N=C(N)c1ccc(OCC(=O)N2CCCCC2)cc1 ZINC000217688524 CD In-Stock Unstable PRSS1 16 43 N=C(N)c1ccc(OCC(=O)N2CCCCC2)cc1 ZINC000217688524 CD In-Stock Unstable HTR1D 15 40 N=C(N)c1ccc(OCC(=O)N2CCCCC2)cc1 ZINC000217688524 CD In-Stock Unstable HTR1B 18 40 N=C(N)c1ccc(OCC(=O)N2CCCCC2)cc1 ZINC000217688524 CD In-Stock Unstable F10 20 45 N=C(N)c1ccc(OCC(=O)N2CCCCC2)cc1 ZINC000217688524 CD In-Stock Unstable HRH3 16 40 N=C(N)c1ccc(OCC(=O)N2CCCCC2)cc1 ZINC000217688524 CD In-Stock Unstable SAT1 0 46 N=C(N)c1ccc(OCC(=O)N2CCCCC2)cc1 ZINC000217688524 CD In-Stock Unstable CPT1A 79 38 N=C(N)c1ccc(OCC(=O)N2CCCCC2)cc1 ZINC000217688524 CD In-Stock Unstable CPT2 41 34 N=C(N)c1ccc(OCC(=O)N2CCCCC2)cc1 ZINC000217688524 CD In-Stock Unstable PLA2G4B 40 34 N=C(N)c1ccc(OCC(=O)N2CCCCC2)cc1 ZINC000217688524 CD In-Stock Unstable PLAU 37 43 N=C(N)c1ccc(OCC(=O)N2CCCCC2)cc1 ZINC000217688524 CD In-Stock Unstable ACR 72 46 N=C(N)c1ccc(OCC(=O)N2CCCCC2)cc1 ZINC000217688524 CD In-Stock Unstable ST14 48 46 N=C(N)c1ccc(OCC(=O)N2CCCCC2)cc1 ZINC000217688524 CD In-Stock Unstable PSMB2 48 38 N=C(N)c1ccc(OCC(=O)N2CCCCC2)cc1 ZINC000217688524 CD In-Stock Unstable PSMB1 42 38 N=C(N)c1ccc(OCC(=O)N2CCCCC2)cc1 ZINC000217688524 CD In-Stock Unstable GPR183 0 45 CCC[C@H](N[C@H]1CCN2CCC[C@@H]12)c1ccc(Cl)cc1 ZINC000217688532 CI For-Sale Unstable SLC6A1 0 42 O=C(Nc1cccc(Cl)c1)N1CC[C@@H](n2ccnn2)C1 ZINC000217688558 CE In-Stock Unstable FAAH 17 45 O=C(Nc1cccc(Cl)c1)N1CC[C@@H](n2ccnn2)C1 ZINC000217688558 CE In-Stock Unstable EPHX2 17 48 O=C(C1CCC1)N1CCC(N2CCn3nc([C@@H](O)CO)cc3C2)CC1 ZINC000217688590 EC In-Stock Unstable L3MBTL3 50 33 COc1ccc(-c2csc(Nc3ccc(C)cc3)n2)cc1N ZINC000217688630 DI In-Stock Unstable MAOB 23 45 COc1ccc(-c2csc(Nc3ccc(C)cc3)n2)cc1N ZINC000217688630 DI In-Stock Unstable SPHK2 53 39 COc1ccc(-c2csc(Nc3ccc(C)cc3)n2)cc1N ZINC000217688630 DI In-Stock Unstable SPHK1 46 44 COc1ccc(-c2csc(Nc3ccc(C)cc3)n2)cc1N ZINC000217688630 DI In-Stock Unstable PLAU 20 44 COc1ccc(-c2csc(Nc3ccc(C)cc3)n2)cc1N ZINC000217688630 DI In-Stock Unstable AGPAT2 20 43 COc1ccc(-c2csc(Nc3ccc(C)cc3)n2)cc1N ZINC000217688630 DI In-Stock Unstable VCP 21 48 COc1ccc(-c2csc(Nc3ccc(C)cc3)n2)cc1N ZINC000217688630 DI In-Stock Unstable TRPC6 42 38 COC(=O)[C@@H](O)CNC(=O)c1ccc([N+](=O)[O-])cc1Cl ZINC000217688656 DC On-Demand Unstable CACNA1C 47 34 COC(=O)[C@@H](O)CNC(=O)c1ccc([N+](=O)[O-])cc1Cl ZINC000217688656 DC On-Demand Unstable CACNA1D 81 36 O=C(NC(c1ccccc1)c1ccccc1)N1CC[C@H](n2ccnn2)C1 ZINC000217688658 EG In-Stock Unstable XIAP 25 42 O=C(NC(c1ccccc1)c1ccccc1)N1CC[C@H](n2ccnn2)C1 ZINC000217688658 EG In-Stock Unstable BIRC3 17 42 O=C(NC(c1ccccc1)c1ccccc1)N1CC[C@H](n2ccnn2)C1 ZINC000217688658 EG In-Stock Unstable BIRC2 17 42 O=C(NC(c1ccccc1)c1ccccc1)N1CC[C@H](n2ccnn2)C1 ZINC000217688658 EG In-Stock Unstable BIRC8 57 42 O=C(C1CCC1)N1CCC(N2CCn3nc([C@H](O)CO)cc3C2)CC1 ZINC000217688666 EC In-Stock Unstable L3MBTL3 50 33 COC(=O)[C@H](O)CNC(=O)c1ccc([N+](=O)[O-])cc1Cl ZINC000217688735 DC On-Demand Unstable CACNA1C 47 34 COC(=O)[C@H](O)CNC(=O)c1ccc([N+](=O)[O-])cc1Cl ZINC000217688735 DC On-Demand Unstable CACNA1D 81 36 O=C(NC(c1ccccc1)c1ccccc1)N1CC[C@@H](n2ccnn2)C1 ZINC000217688739 EG In-Stock Unstable XIAP 25 42 O=C(NC(c1ccccc1)c1ccccc1)N1CC[C@@H](n2ccnn2)C1 ZINC000217688739 EG In-Stock Unstable BIRC3 17 42 O=C(NC(c1ccccc1)c1ccccc1)N1CC[C@@H](n2ccnn2)C1 ZINC000217688739 EG In-Stock Unstable BIRC2 17 42 O=C(NC(c1ccccc1)c1ccccc1)N1CC[C@@H](n2ccnn2)C1 ZINC000217688739 EG In-Stock Unstable BIRC8 57 42 Clc1ncnc(Nc2ccccc2)c1-c1ccccc1 ZINC000217688751 CJ In-Stock Anodyne EGFR 27 48 CNC(=O)[C@H](C)NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217688818 CC For-Sale Unstable KCNK3 87 38 CNC(=O)[C@H](C)NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217688818 CC For-Sale Unstable KCNK9 46 38 O=C(NC1CCCCC1)N1CC[C@@H](n2ccnn2)C1 ZINC000217688839 CD In-Stock Unstable EPHX2 19 51 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC)cc1OC ZINC000217688849 CB On-Demand Unstable CYP1B1 30 41 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC)cc1OC ZINC000217688849 CB On-Demand Unstable MTNR1A 52 40 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC)cc1OC ZINC000217688849 CB On-Demand Unstable MTNR1B 44 40 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC)cc1OC ZINC000217688849 CB On-Demand Unstable AKR1C2 50 36 CNC(=O)[C@@H](C)NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217688911 CC For-Sale Unstable KCNK3 87 38 CNC(=O)[C@@H](C)NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217688911 CC For-Sale Unstable KCNK9 46 38 O=C(NC1CCCCC1)N1CC[C@H](n2ccnn2)C1 ZINC000217688921 CD In-Stock Unstable EPHX2 19 51 COC(=O)[C@H](O)CNC(=O)c1ccc(OC)cc1OC ZINC000217688922 CB On-Demand Unstable CYP1B1 30 41 COC(=O)[C@H](O)CNC(=O)c1ccc(OC)cc1OC ZINC000217688922 CB On-Demand Unstable MTNR1A 52 40 COC(=O)[C@H](O)CNC(=O)c1ccc(OC)cc1OC ZINC000217688922 CB On-Demand Unstable MTNR1B 44 40 COC(=O)[C@H](O)CNC(=O)c1ccc(OC)cc1OC ZINC000217688922 CB On-Demand Unstable AKR1C2 50 36 Cc1cccnc1C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217688955 CH On-Demand Unstable ABL1 15 40 Cc1cccnc1C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217688955 CH On-Demand Unstable DHODH 15 43 Cc1cccnc1C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217688955 CH On-Demand Unstable KIT 21 46 Cc1cccnc1C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217688955 CH On-Demand Unstable TRPV1 60 67 Cc1cccnc1C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217688955 CH On-Demand Unstable P2RY1 34 46 Cc1cccnc1C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217688955 CH On-Demand Unstable MAP1 40 36 Cc1cccnc1C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217688955 CH On-Demand Unstable ATF1 33 45 Cc1cccnc1C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217688955 CH On-Demand Unstable PRNP 43 33 Cc1cccnc1C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217688955 CH On-Demand Unstable FLT1 37 45 Cc1cccnc1C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217688955 CH On-Demand Unstable KDR 30 51 Cc1cccnc1C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217688955 CH On-Demand Unstable GRM4 41 40 Cc1cccnc1C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217688955 CH On-Demand Unstable MTTP 49 41 Cc1cccnc1C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217688955 CH On-Demand Unstable NFKB1 31 45 Cc1cccnc1C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217688955 CH On-Demand Unstable EPHX2 29 51 Cc1cccnc1C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217688955 CH On-Demand Unstable TEK 47 40 Cc1cccnc1C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217688955 CH On-Demand Unstable BTK 23 41 Cc1cccnc1C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217688955 CH On-Demand Unstable BRAF 21 45 Cc1cccnc1C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217688955 CH On-Demand Unstable SHH 55 36 Cc1cccnc1C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217688955 CH On-Demand Unstable TRPM8 45 40 Cc1cccnc1C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217688955 CH On-Demand Unstable SMO 21 41 Cc1cccnc1C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217688955 CH On-Demand Unstable NAMPT 15 43 Cc1cccnc1C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217688955 CH On-Demand Unstable SLC11A2 31 50 COc1ccc(OCCNC(=O)N/C=C/c2ccccc2C)cc1 ZINC000217688969 EG For-Sale Unstable MTNR1A 40 45 COc1ccc(OCCNC(=O)N/C=C/c2ccccc2C)cc1 ZINC000217688969 EG For-Sale Unstable MTNR1B 33 45 CCCCC[C@@H](C)NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217688991 CG For-Sale Unstable CTSG 27 42 CCCCC[C@@H](C)NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217688991 CG For-Sale Unstable CTRB1 29 42 CCCCC[C@@H](C)NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217688991 CG For-Sale Unstable CELA2A 22 42 COc1cc(NC(=O)c2cnco2)c(C(=O)O)cc1OC ZINC000217689006 CD In-Stock Unstable IMPDH2 0 44 CNCCO[C@H](c1ccccc1)C1CCC1 ZINC000217689017 BF In-Stock Unstable SLC6A3 18 41 Cc1cc(C)n2nc(CC(=O)N3CCC[C@@H]3c3ccccn3)nc2n1 ZINC000217689030 EE In-Stock Unstable COLA 123 42 Cc1cc(C)n2nc(CC(=O)N3CCC[C@@H]3c3ccccn3)nc2n1 ZINC000217689030 EE In-Stock Unstable CPT1A 107 42 O=C(Nc1ccc2c(c1)OCO2)N1CC[C@H](n2ccnn2)C1 ZINC000217689045 DD In-Stock Unstable NOS2 79 37 O=C(Nc1ccc2c(c1)OCO2)N1CC[C@H](n2ccnn2)C1 ZINC000217689045 DD In-Stock Unstable TRPC3 29 41 CCCCC[C@H](C)NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217689063 CG For-Sale Unstable CTSG 27 42 CCCCC[C@H](C)NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217689063 CG For-Sale Unstable CTRB1 29 42 CCCCC[C@H](C)NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217689063 CG For-Sale Unstable CELA2A 22 42 Cc1cc(C)n2nc(CC(=O)N3CCC[C@H]3c3ccccn3)nc2n1 ZINC000217689102 EE In-Stock Unstable COLA 123 42 Cc1cc(C)n2nc(CC(=O)N3CCC[C@H]3c3ccccn3)nc2n1 ZINC000217689102 EE In-Stock Unstable CPT1A 107 42 CNCCO[C@@H](c1ccccc1)C1CCC1 ZINC000217689104 BF In-Stock Unstable SLC6A3 18 41 O=C(Nc1ccc2c(c1)OCO2)N1CC[C@@H](n2ccnn2)C1 ZINC000217689135 DD In-Stock Unstable NOS2 79 37 O=C(Nc1ccc2c(c1)OCO2)N1CC[C@@H](n2ccnn2)C1 ZINC000217689135 DD In-Stock Unstable TRPC3 29 41 CC(C)[C@H](NC(=O)c1cn(Cc2ccccc2)c2ccccc12)C(=O)O ZINC000217689178 FH In-Stock Unstable CNR1 33 55 CC(C)[C@H](NC(=O)c1cn(Cc2ccccc2)c2ccccc12)C(=O)O ZINC000217689178 FH In-Stock Unstable CNR2 25 55 CC(C)[C@H](NC(=O)c1cn(Cc2ccccc2)c2ccccc12)C(=O)O ZINC000217689178 FH In-Stock Unstable POL 0 52 CC(C)[C@H](NC(=O)c1cn(Cc2ccccc2)c2ccccc12)C(=O)O ZINC000217689178 FH In-Stock Unstable F2RL3 17 42 CC(=O)NCCNC(=O)N/C=C/c1ccccc1C ZINC000217689181 CD For-Sale Unstable MTNR1A 30 49 CC(=O)NCCNC(=O)N/C=C/c1ccccc1C ZINC000217689181 CD For-Sale Unstable MTNR1B 25 49 COc1ccccc1NC(=O)N1CC[C@H](n2ccnn2)C1 ZINC000217689244 CD In-Stock Unstable SMO 28 47 O=C(O)/C=C\c1cccc(CSc2ncccc2Cl)c1 ZINC000217689277 DI For-Sale Unstable LTB4R 17 41 COC(=O)c1cccc(COc2ccc3occ(-c4ccc(OC)c(OC)c4)c3c2)c1 ZINC000217689301 HK In-Stock Unstable ALDH2 68 33 COC(=O)c1cccc(COc2ccc3occ(-c4ccc(OC)c(OC)c4)c3c2)c1 ZINC000217689301 HK In-Stock Unstable MAOB 47 51 COC(=O)c1cccc(COc2ccc3occ(-c4ccc(OC)c(OC)c4)c3c2)c1 ZINC000217689301 HK In-Stock Unstable PRKCZ 21 41 COC(=O)c1cccc(COc2ccc3occ(-c4ccc(OC)c(OC)c4)c3c2)c1 ZINC000217689301 HK In-Stock Unstable PRKCI 0 41 COC(=O)c1cccc(COc2ccc3occ(-c4ccc(OC)c(OC)c4)c3c2)c1 ZINC000217689301 HK In-Stock Unstable GYS1 56 41 COC(=O)c1cccc(COc2ccc3occ(-c4ccc(OC)c(OC)c4)c3c2)c1 ZINC000217689301 HK In-Stock Unstable ADAMTS4 21 46 CCC(C)(C)NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217689303 CE For-Sale Unstable HDAC8 18 47 CCC(C)(C)NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217689303 CE For-Sale Unstable AKR1C3 26 40 COc1ccccc1NC(=O)N1CC[C@@H](n2ccnn2)C1 ZINC000217689327 CD In-Stock Unstable SMO 28 47 C[C@@H](N[C@@H]1CCN2CCCC[C@@H]12)c1ccccc1O ZINC000217689359 CF For-Sale Unstable SLC18A3 68 39 Cc1ccccc1/C=C/NC(=O)NC12CC3CC(CC(C3)C1)C2 ZINC000217689394 DI For-Sale Unstable CNR2 19 42 Cc1ccccc1/C=C/NC(=O)NC12CC3CC(CC(C3)C1)C2 ZINC000217689394 DI For-Sale Unstable EPHX2 107 50 CC(C)C[C@H](NC(=O)CCCC[C@H]1CCSS1)c1nc2ccccc2[nH]1 ZINC000217689412 GK In-Stock Unstable PTPN1 33 41 CC(C)C[C@H](NC(=O)CCCC[C@H]1CCSS1)c1nc2ccccc2[nH]1 ZINC000217689412 GK In-Stock Unstable MMP7 22 52 COC(=O)[C@@H](O)CNC(=O)[C@@H](C)Oc1cccc(C)c1 ZINC000217689415 CC On-Demand Unstable MTNR1A 24 45 O=C(Nc1ccccc1F)N1CC[C@H](n2ccnn2)C1 ZINC000217689426 CD In-Stock Unstable RBP4 54 37 COc1ccccc1Nc1ncnc(Cl)c1-c1ccccc1 ZINC000217689438 DJ In-Stock Unstable EGFR 34 44 COc1ccccc1Nc1ncnc(Cl)c1-c1ccccc1 ZINC000217689438 DJ In-Stock Unstable FLT1 0 40 C[C@H](N[C@@H]1CCN2CCCC[C@@H]12)c1ccccc1O ZINC000217689439 CF On-Demand Unstable SLC18A3 55 39 CN(C)[C@@H]1CCCN(c2cc(Cl)ccc2CBr)C1 ZINC000217689461 EH For-Sale Unstable NOS3 16 40 COC(=O)[C@H](O)CNC(=O)[C@@H](C)Oc1cccc(C)c1 ZINC000217689490 CC On-Demand Unstable MTNR1A 24 45 CC(C)C[C@H](NC(=O)CCCC[C@@H]1CCSS1)c1nc2ccccc2[nH]1 ZINC000217689493 GK In-Stock Unstable PTPN1 33 41 CC(C)C[C@H](NC(=O)CCCC[C@@H]1CCSS1)c1nc2ccccc2[nH]1 ZINC000217689493 GK In-Stock Unstable MMP7 22 52 O=C(Nc1ccccc1F)N1CC[C@@H](n2ccnn2)C1 ZINC000217689507 CD In-Stock Unstable RBP4 54 37 C[C@@H](N[C@H]1CCN2CCCC[C@@H]12)c1ccccc1O ZINC000217689532 CF For-Sale Unstable SLC18A3 68 39 CN(C)[C@H]1CCCN(c2cc(Cl)ccc2CBr)C1 ZINC000217689537 EH For-Sale Unstable NOS3 16 40 COC(=O)[C@@H](O)CNC(=O)[C@H](C)Oc1cccc(C)c1 ZINC000217689565 CC On-Demand Unstable MTNR1A 24 45 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cc3ccccc3n(CC(C)C)c2=O)CC(=O)O4)cc1O ZINC000217689609 KK In-Stock Unstable CYP1B1 46 33 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cc3ccccc3n(CC(C)C)c2=O)CC(=O)O4)cc1O ZINC000217689609 KK In-Stock Unstable CYP1A1 32 40 O=S(=O)(c1ccc(-c2cccc(C(F)(F)F)c2)cc1)N1CC[C@H](n2ccnn2)C1 ZINC000217689611 HH In-Stock Unstable CACNA1B 45 33 C[C@H](N[C@H]1CCN2CCCC[C@@H]12)c1ccccc1O ZINC000217689615 CF On-Demand Unstable SLC18A3 55 39 CN(Cc1cccc2cnccc12)C(=O)Cc1ccccn1 ZINC000217689633 CF In-Stock Unstable TRPV1 31 40 COC(=O)[C@H](O)CNC(=O)[C@H](C)Oc1cccc(C)c1 ZINC000217689644 CC On-Demand Unstable MTNR1A 24 45 CN(C)[C@@H]1CCCN(c2ccc(Cl)cc2CBr)C1 ZINC000217689645 EH For-Sale Unstable NOS2 21 42 CN(C)[C@@H]1CCCN(c2ccc(Cl)cc2CBr)C1 ZINC000217689645 EH For-Sale Unstable NOS3 21 42 O=C(O)COc1ccc(NC(=O)c2cnco2)cc1 ZINC000217689680 CD In-Stock Unstable P4HTM 0 43 O=S(=O)(c1ccc(-c2cccc(C(F)(F)F)c2)cc1)N1CC[C@@H](n2ccnn2)C1 ZINC000217689705 HH In-Stock Unstable CACNA1B 45 33 CC(C)N(C)S(=O)(=O)c1ccc(/C=C\C(=O)O)cc1Cl ZINC000217689708 DE For-Sale Unstable NR0B2 0 40 Cc1ccccc1/C=C/NC(=O)N1c2ccccc2C[C@H]1C ZINC000217689712 CI For-Sale Unstable DRD4 25 46 Cc1ccccc1/C=C/NC(=O)N1c2ccccc2C[C@H]1C ZINC000217689712 CI For-Sale Unstable TPP2 53 34 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cc3ccccc3n(CC(C)C)c2=O)CC(=O)O4)cc1O ZINC000217689716 KK In-Stock Unstable CYP1B1 46 33 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cc3ccccc3n(CC(C)C)c2=O)CC(=O)O4)cc1O ZINC000217689716 KK In-Stock Unstable CYP1A1 32 40 CN(C)[C@H]1CCCN(c2ccc(Cl)cc2CBr)C1 ZINC000217689729 EH For-Sale Unstable NOS2 21 42 CN(C)[C@H]1CCCN(c2ccc(Cl)cc2CBr)C1 ZINC000217689729 EH For-Sale Unstable NOS3 21 42 CCO/C=C/C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217689740 CG On-Demand Unstable TRPV1 20 47 CCO/C=C/C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217689740 CG On-Demand Unstable EPHX2 24 40 CCO/C=C/C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217689740 CG On-Demand Unstable ACR 20 41 COC(=O)[C@@H](O)CNC(=O)c1ccc([N+](=O)[O-])cc1F ZINC000217689769 CB On-Demand Unstable CACNA1C 49 34 COC(=O)[C@@H](O)CNC(=O)c1ccc([N+](=O)[O-])cc1F ZINC000217689769 CB On-Demand Unstable CACNA1D 81 35 Cc1ccccc1/C=C/NC(=O)N1c2ccccc2C[C@@H]1C ZINC000217689792 CI For-Sale Unstable DRD4 25 46 Cc1ccccc1/C=C/NC(=O)N1c2ccccc2C[C@@H]1C ZINC000217689792 CI For-Sale Unstable TPP2 53 34 O=C(c1cnccn1)N1CCC(n2ccnn2)CC1 ZINC000217689813 CC In-Stock Unstable L3MBTL3 43 32 COC(=O)[C@H](O)CNC(=O)c1ccc([N+](=O)[O-])cc1F ZINC000217689851 CB On-Demand Unstable CACNA1C 49 34 COC(=O)[C@H](O)CNC(=O)c1ccc([N+](=O)[O-])cc1F ZINC000217689851 CB On-Demand Unstable CACNA1D 81 35 O=C(O)/C=C\c1cccc(S(=O)(=O)NCC(F)(F)F)c1 ZINC000217689872 DD For-Sale Unstable AKR1C3 34 42 O=C(O)/C=C\c1cccc(S(=O)(=O)NCC(F)(F)F)c1 ZINC000217689872 DD For-Sale Unstable SFRP1 55 32 O=C(O)/C=C\c1ccccc1CSc1ncccc1Cl ZINC000217689905 DI For-Sale Unstable PTGER2 39 48 O=C(O)/C=C\c1ccccc1CSc1ncccc1Cl ZINC000217689905 DI For-Sale Unstable PTGER4 21 44 O=C(O)/C=C\c1ccccc1CSc1ncccc1Cl ZINC000217689905 DI For-Sale Unstable PTGER3 20 51 O=C(O)/C=C\c1ccccc1CSc1ncccc1Cl ZINC000217689905 DI For-Sale Unstable PTGDR 0 43 CC[C@@H](C)[C@@H](CO)NC(=O)Cc1c(C)c2ccc(O)cc2oc1=O ZINC000217689925 ED In-Stock Unstable HSD17B3 45 54 CC[C@@H](C)[C@@H](CO)NC(=O)Cc1c(C)c2ccc(O)cc2oc1=O ZINC000217689925 ED In-Stock Unstable NQO1 54 37 Cc1cc(S(=O)(=O)NCC(F)(F)F)ccc1/C=C\C(=O)O ZINC000217689966 DD For-Sale Unstable LEF 47 34 COc1ccc(-c2csc(NS(C)(=O)=O)n2)cc1N ZINC000217690020 CD In-Stock Unstable SREBF2 0 40 OCc1ccn(Cc2ccc(F)cc2)n1 ZINC000217690036 BD In-Stock Unstable HDAC7 22 57 Cc1cc(N2C[C@]34C=C[C@@H](O3)[C@@H](C(=O)NCc3ccc5c(c3)OCO5)[C@H]4C2=O)no1 ZINC000217690065 HD In-Stock Unstable NOS2 90 33 O=C(O)/C=C\c1cc(F)ccc1CSc1ncccc1Cl ZINC000217690071 DI For-Sale Unstable PTGER2 22 40 Cc1ccccc1/C=C/NC(=O)N1CCN(c2ncccn2)CC1 ZINC000217690107 DE For-Sale Unstable SLC6A7 0 49 COc1ccc(C)cc1CN[C@@H]1CCN2CCCC[C@@H]12 ZINC000217690133 CF On-Demand Unstable TACR1 35 41 Cc1cc(N2C[C@]34C=C[C@@H](O3)[C@H](C(=O)NCc3ccc5c(c3)OCO5)[C@H]4C2=O)no1 ZINC000217690137 HD In-Stock Unstable NOS2 90 33 N=C(N)c1ccc(OCC(=O)N2CCCC2)cc1 ZINC000217690145 BC In-Stock Unstable F2 20 47 N=C(N)c1ccc(OCC(=O)N2CCCC2)cc1 ZINC000217690145 BC In-Stock Unstable PRSS1 17 44 N=C(N)c1ccc(OCC(=O)N2CCCC2)cc1 ZINC000217690145 BC In-Stock Unstable HTR1D 15 41 N=C(N)c1ccc(OCC(=O)N2CCCC2)cc1 ZINC000217690145 BC In-Stock Unstable HTR1B 19 41 N=C(N)c1ccc(OCC(=O)N2CCCC2)cc1 ZINC000217690145 BC In-Stock Unstable F10 20 45 N=C(N)c1ccc(OCC(=O)N2CCCC2)cc1 ZINC000217690145 BC In-Stock Unstable TRY1_BOVIN 54 37 N=C(N)c1ccc(OCC(=O)N2CCCC2)cc1 ZINC000217690145 BC In-Stock Unstable COLA 95 45 N=C(N)c1ccc(OCC(=O)N2CCCC2)cc1 ZINC000217690145 BC In-Stock Unstable CPT1A 87 39 N=C(N)c1ccc(OCC(=O)N2CCCC2)cc1 ZINC000217690145 BC In-Stock Unstable CPT2 45 35 N=C(N)c1ccc(OCC(=O)N2CCCC2)cc1 ZINC000217690145 BC In-Stock Unstable PLA2G4B 41 35 N=C(N)c1ccc(OCC(=O)N2CCCC2)cc1 ZINC000217690145 BC In-Stock Unstable PLAU 37 44 N=C(N)c1ccc(OCC(=O)N2CCCC2)cc1 ZINC000217690145 BC In-Stock Unstable ACR 79 47 N=C(N)c1ccc(OCC(=O)N2CCCC2)cc1 ZINC000217690145 BC In-Stock Unstable ST14 52 47 N=C(N)c1ccc(OCC(=O)N2CCCC2)cc1 ZINC000217690145 BC In-Stock Unstable PSMB2 40 36 OCc1ccn(Cc2cccc(F)c2)n1 ZINC000217690147 BD In-Stock Unstable HDAC7 21 40 O=C(O)/C=C\c1ccc(C(=O)Nc2ccc(Cl)cn2)s1 ZINC000217690199 DG For-Sale Anodyne F10 53 34 O=C(O)/C=C\c1ccc(C(=O)Nc2ccc(Cl)cn2)s1 ZINC000217690199 DG For-Sale Anodyne LUCI_LUCLA 32 42 COc1ccc(C)cc1CN[C@H]1CCN2CCCC[C@@H]12 ZINC000217690210 CF On-Demand Unstable TACR1 35 41 O=C(O)/C=C\c1cc(CSc2ncccc2Cl)ccc1F ZINC000217690218 DI For-Sale Unstable PTGER4 0 41 CCOC(=O)c1sc(NC(=O)CCCCCNc2ccc3c(cc2=O)[C@@H](NC(C)=O)CCc2cc(OC)c(OC)c(OC)c2-3)nc1C ZINC000217690226 KK In-Stock Unstable TUBA1A 15 56 CC(C)CNC[C@@H]1CC[C@@H]1N1CC[C@@H](c2ccccc2)C1 ZINC000217690238 CH For-Sale Unstable SLC18A3 52 39 CC(C)(C)c1ccc(S(=O)(=O)N2CCC(n3ccnn3)CC2)cc1 ZINC000217690251 EF In-Stock Unstable HSD11B1 22 50 O=C(O)/C=C\c1ccc(C(=O)Nc2ccc(Cl)cn2)cc1 ZINC000217690289 DG For-Sale Anodyne KLKB1 35 47 O=C(O)/C=C\c1ccc(C(=O)Nc2ccc(Cl)cn2)cc1 ZINC000217690289 DG For-Sale Anodyne F10 54 50 O=C(O)/C=C\c1ccc(C(=O)Nc2ccc(Cl)cn2)cc1 ZINC000217690289 DG For-Sale Anodyne LUCI_LUCLA 48 54 C1CCN2CC[C@@H](NC3C4CC5CC(C4)CC3C5)[C@H]2C1 ZINC000217690323 CG On-Demand Unstable CYP2D26 0 43 CCOC(=O)N1CCC(NC(=O)N/C=C/c2ccccc2C)CC1 ZINC000217690344 EF For-Sale Unstable EPHX2 31 41 CCOC(=O)N1CCC(NC(=O)N/C=C/c2ccccc2C)CC1 ZINC000217690344 EF For-Sale Unstable CCR8 56 43 COc1ccc(C(=O)N2CCCC2)cc1/C=C\C(=O)O ZINC000217690366 CE For-Sale Unstable TNFRSF1A 23 41 COc1ccc(C(=O)N2CCCC2)cc1/C=C\C(=O)O ZINC000217690366 CE For-Sale Unstable L3MBTL3 65 37 COc1ccc(C(=O)N2CCCC2)cc1/C=C\C(=O)O ZINC000217690366 CE For-Sale Unstable HPGD 40 43 NCCO[C@H](c1ccccc1)C1CCC1 ZINC000217690380 BF In-Stock Unstable AMY2 43 30 CC(C)CNC[C@@H]1CC[C@H]1N1CC[C@@H](c2ccccc2)C1 ZINC000217690406 CH For-Sale Unstable SLC18A3 52 39 Cc1n[nH]c(C)c1CNC(=O)CN(C)Cc1cccnc1 ZINC000217690431 CD In-Stock Unstable HAO2 61 40 Cc1ccccc1/C=C/NC(=O)N1CCN(c2cccc(Cl)c2)CC1 ZINC000217690436 FI For-Sale Unstable HTR1A 19 45 Cc1ccccc1/C=C/NC(=O)N1CCN(c2cccc(Cl)c2)CC1 ZINC000217690436 FI For-Sale Unstable HTR2A 15 42 c1ccc(C2CC(N[C@@H]3CCN4CCCC[C@@H]34)C2)cc1 ZINC000217690448 CG On-Demand Unstable VACHT_TETCF 0 50 c1ccc(C2CC(N[C@@H]3CCN4CCCC[C@@H]34)C2)cc1 ZINC000217690448 CG On-Demand Unstable SLC18A3 58 50 COc1ccc(C(=O)NN)cc1C#N ZINC000217690457 AC In-Stock Unstable AR 15 42 COc1ccc(C(=O)NN)cc1C#N ZINC000217690457 AC In-Stock Unstable XDH 45 37 COc1ccc(C(=O)NN)cc1C#N ZINC000217690457 AC In-Stock Unstable EZH2 41 41 COc1ccc(C(=O)NN)cc1C#N ZINC000217690457 AC In-Stock Unstable H9B8T9_CAPHI 15 51 COc1ccc(C(=O)NC2CCCC2)cc1/C=C\C(=O)O ZINC000217690458 CE For-Sale Unstable MAPK14 31 40 COc1ccc(C(=O)NC2CCCC2)cc1/C=C\C(=O)O ZINC000217690458 CE For-Sale Unstable TNFRSF1A 24 42 COc1ccc(C(=O)NC2CCCC2)cc1/C=C\C(=O)O ZINC000217690458 CE For-Sale Unstable PLAU 16 40 COc1ccc(C(=O)NC2CCCC2)cc1/C=C\C(=O)O ZINC000217690458 CE For-Sale Unstable ACKR3 40 32 COc1ccc(OC)c(Nc2nc(-c3ccc(OC)c(N)c3)cs2)c1 ZINC000217690460 FI In-Stock Unstable MAOA 0 42 COc1ccc(OC)c(Nc2nc(-c3ccc(OC)c(N)c3)cs2)c1 ZINC000217690460 FI In-Stock Unstable MAOB 0 42 NCCO[C@@H](c1ccccc1)C1CCC1 ZINC000217690462 BF In-Stock Unstable AMY2 43 30 COC(=O)[C@@H](O)CNC(=O)c1ccc([N+](=O)[O-])c(C)c1 ZINC000217690513 CC On-Demand Unstable GSTM2 49 37 O=C(O)/C=C\c1cccc(C(=O)N2CCCCCC2)c1 ZINC000217690538 CF For-Sale Unstable PREP 27 43 O=C(O)/C=C\c1cccc(C(=O)N2CCCCCC2)c1 ZINC000217690538 CF For-Sale Unstable L3MBTL3 68 47 O=C(O)/C=C\c1cccc(C(=O)N2CCCCCC2)c1 ZINC000217690538 CF For-Sale Unstable HPGD 48 42 c1ccc(C2CC(N[C@H]3CCN4CCCC[C@@H]34)C2)cc1 ZINC000217690544 CG On-Demand Unstable VACHT_TETCF 0 50 c1ccc(C2CC(N[C@H]3CCN4CCCC[C@@H]34)C2)cc1 ZINC000217690544 CG On-Demand Unstable SLC18A3 58 50 Cc1ccc2nc(-c3ccc(NC(=O)N/C=C/c4ccccc4C)cc3)sc2c1 ZINC000217690546 GK For-Sale Unstable APP 26 53 Cc1ccc(Cn2ccc(CO)n2)cc1 ZINC000217690562 BD In-Stock Unstable HDAC7 20 41 CCCNC[C@@H]1CC[C@@H]1N1CC[C@@H](c2ccccc2)C1 ZINC000217690567 CG For-Sale Unstable VACHT_TETCF 0 40 CCCNC[C@@H]1CC[C@@H]1N1CC[C@@H](c2ccccc2)C1 ZINC000217690567 CG For-Sale Unstable SLC18A3 57 40 O=C(Cc1cccs1)NCc1cncc(-c2ccsc2)c1 ZINC000217690572 DH In-Stock Unstable CA5B 36 48 O=C(Cc1cccs1)NCc1cncc(-c2ccsc2)c1 ZINC000217690572 DH In-Stock Unstable CA5A 36 48 COC(=O)[C@H](O)CNC(=O)c1ccc([N+](=O)[O-])c(C)c1 ZINC000217690594 CC On-Demand Unstable GSTM2 49 37 CCCN(CCC)C(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217690625 CG For-Sale Unstable TTR 0 40 Fc1ccc(C2CC(N[C@@H]3CCN4CCCC[C@@H]34)C2)cc1 ZINC000217690655 CG For-Sale Unstable SLC18A3 40 37 Cc1cccc(Cn2ccc(CO)n2)c1 ZINC000217690660 BD In-Stock Unstable HDAC7 23 43 Cc1ccccc1/C=C/NC(=O)Nc1ccc2c(c1)OCO2 ZINC000217690668 CH For-Sale Unstable CCR2 0 42 O=C(NCc1cncc(-c2ccsc2)c1)c1nc2ccccc2s1 ZINC000217690696 FI In-Stock Unstable NAMPT 16 47 O=C(NCc1cncc(-c2ccsc2)c1)c1nc2ccccc2s1 ZINC000217690696 FI In-Stock Unstable TMPRSS6 40 30 COc1ccc(C(=O)N(C)CCO)cc1/C=C\C(=O)O ZINC000217690717 CC For-Sale Unstable CYSP_PLAFA 41 35 Fc1ccc(C2CC(N[C@H]3CCN4CCCC[C@@H]34)C2)cc1 ZINC000217690737 CG For-Sale Unstable SLC18A3 40 37 CCCNC[C@@H]1CC[C@H]1N1CC[C@@H](c2ccccc2)C1 ZINC000217690745 CG For-Sale Unstable VACHT_TETCF 0 40 CCCNC[C@@H]1CC[C@H]1N1CC[C@@H](c2ccccc2)C1 ZINC000217690745 CG For-Sale Unstable SLC18A3 57 40 COc1ccc(CCN2C(=O)N[C@@H](CCC(=O)Nc3ccc4cc[nH]c4c3)C2=O)cc1OC ZINC000217690763 JG In-Stock Unstable ENPP1 75 36 O=C(O)c1cc2c(NC3CCCCC3)ncnc2s1 ZINC000217690808 CG In-Stock Unstable GRM1 17 45 O=C(O)c1cc2c(NC3CCCCC3)ncnc2s1 ZINC000217690808 CG In-Stock Unstable CD38 43 44 C[C@H](c1cccs1)N(C)C[C@@H](O)c1ccccc1 ZINC000217690819 CG On-Demand Unstable AOC3 32 51 CNC[C@@H]1CC[C@@H]1N1CC[C@@H](c2ccccc2)C1 ZINC000217690909 BE For-Sale Unstable VACHT_TETCF 0 43 CNC[C@@H]1CC[C@@H]1N1CC[C@@H](c2ccccc2)C1 ZINC000217690909 BE For-Sale Unstable SLC18A3 70 43 C[C@@H](c1cccs1)N(C)C[C@@H](O)c1ccccc1 ZINC000217690912 CG On-Demand Unstable AOC3 32 51 Cc1ccccc1/C=C/NC(=O)Nc1cccc(F)c1 ZINC000217690915 CH For-Sale Unstable KCNK3 91 44 Cc1ccccc1/C=C/NC(=O)Nc1cccc(F)c1 ZINC000217690915 CH For-Sale Unstable KCNK9 55 44 COC[C@H](C)N(C)C(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217690966 CD For-Sale Unstable NR1H4 49 37 COC[C@H](C)N(C)C(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217690966 CD For-Sale Unstable AKR1C3 29 40 NC[C@@H](O)c1cc(F)c(Br)cc1F ZINC000217690982 CD For-Sale Unstable ADRB1 15 52 COC[C@@H](C)N(C)C(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217691048 CD For-Sale Unstable NR1H4 49 37 COC[C@@H](C)N(C)C(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217691048 CD For-Sale Unstable AKR1C3 29 40 NC[C@H](O)c1cc(F)c(Br)cc1F ZINC000217691057 CD For-Sale Unstable ADRB1 15 52 Oc1cccc2c1CC[C@@H]2N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217691059 CF For-Sale Unstable SLC18A3 45 34 CNC[C@@H]1CC[C@H]1N1CC[C@@H](c2ccccc2)C1 ZINC000217691081 BE For-Sale Unstable VACHT_TETCF 0 43 CNC[C@@H]1CC[C@H]1N1CC[C@@H](c2ccccc2)C1 ZINC000217691081 BE For-Sale Unstable SLC18A3 70 43 COC(=O)[C@@H](O)CNC(=O)CCc1ccc(OC)c(Br)c1 ZINC000217691085 FD On-Demand Unstable TRPV1 38 40 Cc1ccccc1/C=C/NC(=O)N1CCc2ccccc21 ZINC000217691142 CH For-Sale Unstable AVPR2 42 40 Oc1cccc2c1CC[C@H]2N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217691143 CF For-Sale Unstable SLC18A3 45 34 Cc1noc(C)c1CC(=O)NCc1cncc(-c2ccsc2)c1 ZINC000217691147 EG In-Stock Unstable P2RX7 32 56 Clc1ncnc(N2CCOCC2)c1-c1ccccc1 ZINC000217691161 CF In-Stock Unstable ADK 27 46 Clc1ncnc(N2CCOCC2)c1-c1ccccc1 ZINC000217691161 CF In-Stock Unstable PIK3CA 20 42 Clc1ncnc(N2CCOCC2)c1-c1ccccc1 ZINC000217691161 CF In-Stock Unstable LRRK2 16 54 Oc1cccc2c1CC[C@@H]2N[C@H]1CCN2CCCC[C@@H]12 ZINC000217691221 CF For-Sale Unstable SLC18A3 45 34 NC[C@@H]1CC[C@@H]1N1CC[C@@H](c2ccccc2)C1 ZINC000217691227 BE For-Sale Unstable VACHT_TETCF 0 46 NC[C@@H]1CC[C@@H]1N1CC[C@@H](c2ccccc2)C1 ZINC000217691227 BE For-Sale Unstable SLC18A3 75 45 CCCCC[C@H](C(=O)O)C1CCC1 ZINC000217691228 AG In-Stock Unstable CPN1 0 40 CCCCC[C@H](C(=O)O)C1CCC1 ZINC000217691228 AG In-Stock Unstable CQSS 49 32 O=C(NCc1cncc(-c2ccsc2)c1)C1CCCC1 ZINC000217691248 CH In-Stock Unstable GRIN2B 17 53 Fc1ccc(Nc2ncnc(Cl)c2-c2ccccc2)cc1 ZINC000217691250 CJ In-Stock Anodyne EGFR 30 43 COc1ccc2ncc(C(=O)N3CCc4ccccc4C3)c(O)c2c1 ZINC000217691277 EG In-Stock Unstable DRD4 40 31 COc1ccc2ncc(C(=O)N3CCc4ccccc4C3)c(O)c2c1 ZINC000217691277 EG In-Stock Unstable OXTR 0 41 COc1ccc2ncc(C(=O)N3CCc4ccccc4C3)c(O)c2c1 ZINC000217691277 EG In-Stock Unstable MTNR1A 25 40 COc1ccc2ncc(C(=O)N3CCc4ccccc4C3)c(O)c2c1 ZINC000217691277 EG In-Stock Unstable MTNR1B 17 40 COc1ccc2ncc(C(=O)N3CCc4ccccc4C3)c(O)c2c1 ZINC000217691277 EG In-Stock Unstable HDAC6 17 40 COc1ccc2ncc(C(=O)N3CCc4ccccc4C3)c(O)c2c1 ZINC000217691277 EG In-Stock Unstable TRPC6 19 46 Oc1cccc2c1CC[C@H]2N[C@H]1CCN2CCCC[C@@H]12 ZINC000217691304 CF For-Sale Unstable SLC18A3 45 34 CCCCC[C@@H](C(=O)O)C1CCC1 ZINC000217691306 AG In-Stock Unstable CPN1 0 40 CCCCC[C@@H](C(=O)O)C1CCC1 ZINC000217691306 AG In-Stock Unstable CQSS 49 32 COC(=O)[C@@H](O)CNC(=O)Cc1ccc(OC)cc1 ZINC000217691319 CB On-Demand Unstable PTGS2 0 42 COC(=O)[C@@H](O)CNC(=O)Cc1ccc(OC)cc1 ZINC000217691319 CB On-Demand Unstable ANPEP 16 42 COC(=O)[C@@H](O)CNC(=O)Cc1ccc(OC)cc1 ZINC000217691319 CB On-Demand Unstable BMP1 62 37 COC(=O)[C@@H](O)CNC(=O)Cc1ccc(OC)cc1 ZINC000217691319 CB On-Demand Unstable MMP13 32 45 COC(=O)[C@@H](O)CNC(=O)Cc1ccc(OC)cc1 ZINC000217691319 CB On-Demand Unstable MTNR1A 53 40 COC(=O)[C@@H](O)CNC(=O)Cc1ccc(OC)cc1 ZINC000217691319 CB On-Demand Unstable MTNR1B 37 40 COC(=O)[C@@H](O)CNC(=O)Cc1ccc(OC)cc1 ZINC000217691319 CB On-Demand Unstable MMP8 24 45 COC(=O)[C@@H](O)CNC(=O)Cc1ccc(OC)cc1 ZINC000217691319 CB On-Demand Unstable MMP12 27 45 COC(=O)[C@@H](O)CNC(=O)Cc1ccc(OC)cc1 ZINC000217691319 CB On-Demand Unstable CA12 16 53 COC(=O)[C@@H](O)CNC(=O)Cc1ccc(OC)cc1 ZINC000217691319 CB On-Demand Unstable MAPK8 15 44 COC(=O)[C@@H](O)CNC(=O)Cc1ccc(OC)cc1 ZINC000217691319 CB On-Demand Unstable CA9 27 53 COC(=O)[C@@H](O)CNC(=O)Cc1ccc(OC)cc1 ZINC000217691319 CB On-Demand Unstable MMP1 47 37 COC(=O)[C@@H](O)CNC(=O)Cc1ccc(OC)cc1 ZINC000217691319 CB On-Demand Unstable DXR 18 41 COC(=O)[C@@H](O)CNC(=O)Cc1ccc(OC)cc1 ZINC000217691319 CB On-Demand Unstable CACNA1I 16 40 COC(=O)[C@@H](O)CNC(=O)Cc1ccc(OC)cc1 ZINC000217691319 CB On-Demand Unstable PROKR1 51 32 COC(=O)[C@@H](O)CNC(=O)Cc1ccc(OC)cc1 ZINC000217691319 CB On-Demand Unstable H9B8T9_CAPHI 23 46 NC[C@@H](O)c1cc(Br)cc(F)c1F ZINC000217691344 CD For-Sale Unstable ADRB1 16 55 COc1ccc(C(=O)NCc2cncc(-c3ccsc3)c2)c(OC)c1OC ZINC000217691348 GH In-Stock Unstable GRIN2B 21 48 COc1ccc(C(=O)NCc2cncc(-c3ccsc3)c2)c(OC)c1OC ZINC000217691348 GH In-Stock Unstable HCRTR2 21 40 CCOC(=O)c1ccc(-c2ccc(OC)cc2)nc1N ZINC000217691358 CF In-Stock Unstable ABCG2 0 42 Cc1ccccc1/C=C/NC(=O)NCCc1c[nH]c2ccccc12 ZINC000217691364 DH For-Sale Unstable CCKAR 61 45 Cc1ccccc1/C=C/NC(=O)NCCc1c[nH]c2ccccc12 ZINC000217691364 DH For-Sale Unstable MPO 33 41 Cc1ccccc1/C=C/NC(=O)NCCc1c[nH]c2ccccc12 ZINC000217691364 DH For-Sale Unstable BRS3 28 44 Cc1ccccc1/C=C/NC(=O)NCCc1c[nH]c2ccccc12 ZINC000217691364 DH For-Sale Unstable NMBR 49 47 Cc1ccccc1/C=C/NC(=O)NCCc1c[nH]c2ccccc12 ZINC000217691364 DH For-Sale Unstable MTNR1A 15 46 Cc1ccccc1/C=C/NC(=O)NCCc1c[nH]c2ccccc12 ZINC000217691364 DH For-Sale Unstable CCKBR 42 36 Cc1ccccc1/C=C/NC(=O)NCCc1c[nH]c2ccccc12 ZINC000217691364 DH For-Sale Unstable ALOX15 27 47 Cc1ccccc1/C=C/NC(=O)NCCc1c[nH]c2ccccc12 ZINC000217691364 DH For-Sale Unstable MMP9 15 55 COC(=O)[C@H](O)CNC(=O)Cc1ccc(OC)cc1 ZINC000217691406 CB On-Demand Unstable PTGS2 0 42 COC(=O)[C@H](O)CNC(=O)Cc1ccc(OC)cc1 ZINC000217691406 CB On-Demand Unstable ANPEP 16 42 COC(=O)[C@H](O)CNC(=O)Cc1ccc(OC)cc1 ZINC000217691406 CB On-Demand Unstable BMP1 62 37 COC(=O)[C@H](O)CNC(=O)Cc1ccc(OC)cc1 ZINC000217691406 CB On-Demand Unstable MMP13 32 45 COC(=O)[C@H](O)CNC(=O)Cc1ccc(OC)cc1 ZINC000217691406 CB On-Demand Unstable MTNR1A 53 40 COC(=O)[C@H](O)CNC(=O)Cc1ccc(OC)cc1 ZINC000217691406 CB On-Demand Unstable MTNR1B 37 40 COC(=O)[C@H](O)CNC(=O)Cc1ccc(OC)cc1 ZINC000217691406 CB On-Demand Unstable MMP8 24 45 COC(=O)[C@H](O)CNC(=O)Cc1ccc(OC)cc1 ZINC000217691406 CB On-Demand Unstable MMP12 27 45 COC(=O)[C@H](O)CNC(=O)Cc1ccc(OC)cc1 ZINC000217691406 CB On-Demand Unstable CA12 16 53 COC(=O)[C@H](O)CNC(=O)Cc1ccc(OC)cc1 ZINC000217691406 CB On-Demand Unstable MAPK8 15 44 COC(=O)[C@H](O)CNC(=O)Cc1ccc(OC)cc1 ZINC000217691406 CB On-Demand Unstable CA9 27 53 COC(=O)[C@H](O)CNC(=O)Cc1ccc(OC)cc1 ZINC000217691406 CB On-Demand Unstable MMP1 47 37 COC(=O)[C@H](O)CNC(=O)Cc1ccc(OC)cc1 ZINC000217691406 CB On-Demand Unstable DXR 18 41 COC(=O)[C@H](O)CNC(=O)Cc1ccc(OC)cc1 ZINC000217691406 CB On-Demand Unstable CACNA1I 16 40 COC(=O)[C@H](O)CNC(=O)Cc1ccc(OC)cc1 ZINC000217691406 CB On-Demand Unstable PROKR1 51 32 COC(=O)[C@H](O)CNC(=O)Cc1ccc(OC)cc1 ZINC000217691406 CB On-Demand Unstable H9B8T9_CAPHI 23 46 NC[C@@H]1CC[C@H]1N1CC[C@@H](c2ccccc2)C1 ZINC000217691408 BE For-Sale Unstable VACHT_TETCF 0 46 NC[C@@H]1CC[C@H]1N1CC[C@@H](c2ccccc2)C1 ZINC000217691408 BE For-Sale Unstable SLC18A3 75 45 CC(C)CC[C@H](C(=O)O)C1CCC1 ZINC000217691421 AF In-Stock Unstable CPN1 0 42 NC[C@H](O)c1cc(Br)cc(F)c1F ZINC000217691423 CD For-Sale Unstable ADRB1 16 55 CCOc1cc(C(=O)NCc2cncc(-c3ccsc3)c2)cc(OCC)c1OCC ZINC000217691457 IJ In-Stock Unstable GRIN2B 16 45 CC(C)(C)NC[C@@H]1CC[C@@H]1N1CC[C@@H](c2ccccc2)C1 ZINC000217691492 CH For-Sale Unstable SLC18A3 57 45 C[C@@H](Oc1ccc2c(c1)OCO2)C(=O)NCc1nnc(-c2ccccc2)o1 ZINC000217691495 FF In-Stock Unstable EDNRB 54 41 C[C@@H](Oc1ccc2c(c1)OCO2)C(=O)NCc1nnc(-c2ccccc2)o1 ZINC000217691495 FF In-Stock Unstable BMP1 43 35 CC(C)CC[C@@H](C(=O)O)C1CCC1 ZINC000217691501 AF In-Stock Unstable CPN1 0 42 COCCN(C(=O)c1ccc(/C=C\C(=O)O)cc1)C1CC1 ZINC000217691502 CE For-Sale Unstable MBTPS1 78 35 CCc1ccc(OCC(=O)NC[C@@H](O)C(=O)OC)cc1 ZINC000217691518 CC On-Demand Unstable PLA2G4B 60 36 O=C(O)c1cc2c(N3CCOCC3)nc(-c3ccccc3)nc2s1 ZINC000217691525 EF In-Stock Unstable PRKDC 39 41 O=C(O)c1cc2c(N3CCOCC3)nc(-c3ccccc3)nc2s1 ZINC000217691525 EF In-Stock Unstable PIK3CA 76 46 O=C(O)c1cc2c(N3CCOCC3)nc(-c3ccccc3)nc2s1 ZINC000217691525 EF In-Stock Unstable PIK3CD 44 42 O=C(O)c1cc2c(N3CCOCC3)nc(-c3ccccc3)nc2s1 ZINC000217691525 EF In-Stock Unstable MTOR 78 46 O=C(O)c1cc2c(N3CCOCC3)nc(-c3ccccc3)nc2s1 ZINC000217691525 EF In-Stock Unstable PIK3CG 53 44 O=C(O)c1cc2c(N3CCOCC3)nc(-c3ccccc3)nc2s1 ZINC000217691525 EF In-Stock Unstable PIK3CB 46 50 O=C(O)c1cc2c(N3CCOCC3)nc(-c3ccccc3)nc2s1 ZINC000217691525 EF In-Stock Unstable HIPK3 16 40 O=C(O)c1cc2c(N3CCOCC3)nc(-c3ccccc3)nc2s1 ZINC000217691525 EF In-Stock Unstable PIK3C2B 31 44 O=C(O)c1cc2c(N3CCOCC3)nc(-c3ccccc3)nc2s1 ZINC000217691525 EF In-Stock Unstable RIOK2 15 40 O=C(O)c1cc2c(N3CCOCC3)nc(-c3ccccc3)nc2s1 ZINC000217691525 EF In-Stock Unstable PIK3C2G 15 40 O=C(NCc1cncc(-c2ccsc2)c1)Nc1ccc(Cl)c(Cl)c1 ZINC000217691565 GK In-Stock Unstable ROCK2 22 43 O=C(NCc1cncc(-c2ccsc2)c1)Nc1ccc(Cl)c(Cl)c1 ZINC000217691565 GK In-Stock Unstable BLM 0 45 O=C(NCc1cncc(-c2ccsc2)c1)Nc1ccc(Cl)c(Cl)c1 ZINC000217691565 GK In-Stock Unstable NAMPT 41 42 O=C(NCc1cncc(-c2ccsc2)c1)Nc1ccc(Cl)c(Cl)c1 ZINC000217691565 GK In-Stock Unstable P95276_MYCTO 0 41 O=C(NCc1cncc(-c2ccsc2)c1)Nc1ccc(Cl)c(Cl)c1 ZINC000217691565 GK In-Stock Unstable WRN 0 45 C[C@H](Oc1ccc2c(c1)OCO2)C(=O)NCc1nnc(-c2ccccc2)o1 ZINC000217691581 FF In-Stock Unstable EDNRB 54 41 C[C@H](Oc1ccc2c(c1)OCO2)C(=O)NCc1nnc(-c2ccccc2)o1 ZINC000217691581 FF In-Stock Unstable BMP1 43 35 CCc1ccc(OCC(=O)NC[C@H](O)C(=O)OC)cc1 ZINC000217691597 CC On-Demand Unstable PLA2G4B 60 36 Cc1ccc(C2CC(N[C@@H]3CCN4CCCC[C@@H]34)C2)cc1 ZINC000217691604 CG On-Demand Unstable SLC18A3 23 52 COCc1n[nH]c(-c2ccc(NC(=O)CCCCCNc3ccc4c(cc3=O)[C@@H](NC(C)=O)CCc3cc(OC)c(OC)c(OC)c3-4)cc2)n1 ZINC000217691612 KK In-Stock Unstable TUBA1A 15 54 COc1ccc(-c2csc(NC(C)=O)n2)cc1N ZINC000217691642 CE In-Stock Unstable MAOA 22 40 COc1ccc(-c2csc(NC(C)=O)n2)cc1N ZINC000217691642 CE In-Stock Unstable MAOB 31 41 COc1ccc(-c2csc(NC(C)=O)n2)cc1N ZINC000217691642 CE In-Stock Unstable PIK3CA 17 43 COc1ccc(-c2csc(NC(C)=O)n2)cc1N ZINC000217691642 CE In-Stock Unstable ROCK2 21 45 COc1ccc(-c2csc(NC(C)=O)n2)cc1N ZINC000217691642 CE In-Stock Unstable HDAC9 15 40 COc1ccc(-c2csc(NC(C)=O)n2)cc1N ZINC000217691642 CE In-Stock Unstable U38 0 43 COc1ccc(-c2csc(NC(C)=O)n2)cc1N ZINC000217691642 CE In-Stock Unstable GCK 15 44 O=C(Nc1ccc(C(F)(F)F)cc1)c1nccc2ccccc12 ZINC000217691652 DJ On-Demand Anodyne PPIA 15 46 O=C(Nc1ccc(C(F)(F)F)cc1)c1nccc2ccccc12 ZINC000217691652 DJ On-Demand Anodyne KCNJ11 106 46 O=C(Nc1ccc(C(F)(F)F)cc1)c1nccc2ccccc12 ZINC000217691652 DJ On-Demand Anodyne DNMT1 24 43 O=C(Nc1ccc(C(F)(F)F)cc1)c1nccc2ccccc12 ZINC000217691652 DJ On-Demand Anodyne TRPV1 60 48 O=C(Nc1ccc(C(F)(F)F)cc1)c1nccc2ccccc12 ZINC000217691652 DJ On-Demand Anodyne UL80 20 40 O=C(Nc1ccc(C(F)(F)F)cc1)c1nccc2ccccc12 ZINC000217691652 DJ On-Demand Anodyne P2RY1 18 40 O=C(Nc1ccc(C(F)(F)F)cc1)c1nccc2ccccc12 ZINC000217691652 DJ On-Demand Anodyne ATF1 59 50 O=C(Nc1ccc(C(F)(F)F)cc1)c1nccc2ccccc12 ZINC000217691652 DJ On-Demand Anodyne AURKB 34 41 O=C(Nc1ccc(C(F)(F)F)cc1)c1nccc2ccccc12 ZINC000217691652 DJ On-Demand Anodyne FLT1 48 46 O=C(Nc1ccc(C(F)(F)F)cc1)c1nccc2ccccc12 ZINC000217691652 DJ On-Demand Anodyne KDR 33 47 O=C(Nc1ccc(C(F)(F)F)cc1)c1nccc2ccccc12 ZINC000217691652 DJ On-Demand Anodyne GRM4 35 40 O=C(Nc1ccc(C(F)(F)F)cc1)c1nccc2ccccc12 ZINC000217691652 DJ On-Demand Anodyne MTTP 45 35 O=C(Nc1ccc(C(F)(F)F)cc1)c1nccc2ccccc12 ZINC000217691652 DJ On-Demand Anodyne NFKB1 55 50 O=C(Nc1ccc(C(F)(F)F)cc1)c1nccc2ccccc12 ZINC000217691652 DJ On-Demand Anodyne EPHX2 32 48 O=C(Nc1ccc(C(F)(F)F)cc1)c1nccc2ccccc12 ZINC000217691652 DJ On-Demand Anodyne MCHR1 20 42 O=C(Nc1ccc(C(F)(F)F)cc1)c1nccc2ccccc12 ZINC000217691652 DJ On-Demand Anodyne AURKA 17 44 O=C(Nc1ccc(C(F)(F)F)cc1)c1nccc2ccccc12 ZINC000217691652 DJ On-Demand Anodyne ATR 49 38 O=C(Nc1ccc(C(F)(F)F)cc1)c1nccc2ccccc12 ZINC000217691652 DJ On-Demand Anodyne RIPK1 38 40 O=C(Nc1ccc(C(F)(F)F)cc1)c1nccc2ccccc12 ZINC000217691652 DJ On-Demand Anodyne IMDH_CRYPV 32 41 O=C(Nc1ccc(C(F)(F)F)cc1)c1nccc2ccccc12 ZINC000217691652 DJ On-Demand Anodyne KCNK3 23 40 CC(C)(C)NC[C@@H]1CC[C@H]1N1CC[C@@H](c2ccccc2)C1 ZINC000217691659 CH For-Sale Unstable SLC18A3 57 45 Cc1ccc(C2CC(N[C@H]3CCN4CCCC[C@@H]34)C2)cc1 ZINC000217691685 CG On-Demand Unstable SLC18A3 23 52 O=C(O)c1cc2c(N3CCCCC3)ncnc2s1 ZINC000217691761 CE In-Stock Unstable SIRT3 66 40 O=C(O)c1cc2c(N3CCCCC3)ncnc2s1 ZINC000217691761 CE In-Stock Unstable SIRT2 52 34 O=C(O)c1cc2c(N3CCCCC3)ncnc2s1 ZINC000217691761 CE In-Stock Unstable SIRT1 43 40 CSC[C@@](C)(O)CNC(=O)COc1cccc(Cl)c1 ZINC000217691785 DD On-Demand Unstable PDS 81 43 Cc1nonc1CC(=O)N[C@@H](C)c1nc(-c2ccccn2)no1 ZINC000217691793 DD In-Stock Unstable LUCI_PHOPE 24 40 CCNC[C@@H]1CC[C@@H]1N1CC[C@@H](c2ccccc2)C1 ZINC000217691819 CF For-Sale Unstable SLC18A3 61 42 CSC[C@](C)(O)CNC(=O)COc1cccc(Cl)c1 ZINC000217691864 DD On-Demand Unstable PDS 81 43 Cc1nonc1CC(=O)N[C@H](C)c1nc(-c2ccccn2)no1 ZINC000217691867 DD In-Stock Unstable LUCI_PHOPE 24 40 Cc1cc(SCC(=O)O)nc(COc2ccc(F)cc2)n1 ZINC000217691879 DF In-Stock Unstable FFAR1 27 45 CCNC[C@@H]1CC[C@H]1N1CC[C@@H](c2ccccc2)C1 ZINC000217691984 CF For-Sale Unstable SLC18A3 61 42 O=C(O)/C=C\c1cccc(CSc2ncccc2Br)c1 ZINC000217692071 FI For-Sale Unstable LTB4R 15 40 O=C1C[C@@H](c2cccc(O)c2)c2c(c3ccccc3oc2=O)O1 ZINC000217692091 DF In-Stock Unstable NQO1 32 45 COc1ccc(Nc2nc(-c3ccc(OC)c(N)c3)cs2)cc1 ZINC000217692115 EI In-Stock Unstable MAOA 0 44 COc1ccc(Nc2nc(-c3ccc(OC)c(N)c3)cs2)cc1 ZINC000217692115 EI In-Stock Unstable MAOB 0 45 COc1ccc(Nc2nc(-c3ccc(OC)c(N)c3)cs2)cc1 ZINC000217692115 EI In-Stock Unstable SPHK2 50 43 COc1ccc(Nc2nc(-c3ccc(OC)c(N)c3)cs2)cc1 ZINC000217692115 EI In-Stock Unstable SPHK1 39 44 COc1ccc(Nc2nc(-c3ccc(OC)c(N)c3)cs2)cc1 ZINC000217692115 EI In-Stock Unstable PLAU 0 48 COc1ccc(Nc2nc(-c3ccc(OC)c(N)c3)cs2)cc1 ZINC000217692115 EI In-Stock Unstable TRPC6 42 41 COc1ccc(Nc2nc(-c3ccc(OC)c(N)c3)cs2)cc1 ZINC000217692115 EI In-Stock Unstable TRPC3 28 41 O=C(O)/C=C\c1cccc(C(=O)NC(C2CC2)C2CC2)c1 ZINC000217692116 CF For-Sale Unstable KCNK3 44 33 CC(C)NC[C@@H]1CC[C@@H]1N1CC[C@@H](c2ccccc2)C1 ZINC000217692136 CG For-Sale Unstable VACHT_TETCF 0 43 CC(C)NC[C@@H]1CC[C@@H]1N1CC[C@@H](c2ccccc2)C1 ZINC000217692136 CG For-Sale Unstable SLC18A3 64 43 Cc1ccccc1/C=C/NC(=O)Nc1c(Cl)cccc1Cl ZINC000217692150 DK For-Sale Unstable ACAT 0 43 Fc1ccccc1C1CC(N[C@@H]2CCN3CCCC[C@@H]23)C1 ZINC000217692164 CG On-Demand Unstable SLC18A3 47 36 O=C1C[C@H](c2cccc(O)c2)c2c(c3ccccc3oc2=O)O1 ZINC000217692166 DF In-Stock Unstable NQO1 32 45 CCOC(=O)CNC(=O)Nc1nnc(CC)s1 ZINC000217692194 CC For-Sale Unstable MME 16 41 O=C(O)/C=C\c1ccc(S(=O)(=O)Nc2nccs2)c(Cl)c1 ZINC000217692206 EF For-Sale Anodyne SCN9A 0 42 NCCc1c(O)cc(F)c(Br)c1F ZINC000217692218 CD For-Sale Unstable TAAR1 15 50 COc1ccc(-c2ccc(C(=O)O)c(N)n2)cc1 ZINC000217692233 BE In-Stock Unstable PRS 56 33 COc1ccc(-c2ccc(C(=O)O)c(N)n2)cc1 ZINC000217692233 BE In-Stock Unstable AKR1C3 21 43 COc1ccc(-c2ccc(C(=O)O)c(N)n2)cc1 ZINC000217692233 BE In-Stock Unstable AKR1C2 57 43 COc1ccc(-c2ccc(C(=O)O)c(N)n2)cc1 ZINC000217692233 BE In-Stock Unstable MT-CO2 45 33 Fc1ccccc1C1CC(N[C@H]2CCN3CCCC[C@@H]23)C1 ZINC000217692249 CG On-Demand Unstable SLC18A3 47 36 CC1CC(C(=O)c2ccccc2)C1 ZINC000217692276 AF In-Stock Unstable SLC18A3 18 41 COc1ccccc1OCC(=O)N1CCc2oncc2C1 ZINC000217692295 CD In-Stock Unstable CPT2 32 43 O=C(O)/C=C\c1cccc(S(=O)(=O)Nc2nccs2)c1 ZINC000217692297 DE For-Sale Anodyne MAP 0 40 O=C(O)/C=C\c1cccc(S(=O)(=O)Nc2nccs2)c1 ZINC000217692297 DE For-Sale Anodyne MAP1 50 33 O=C(O)/C=C\c1cccc(S(=O)(=O)Nc2nccs2)c1 ZINC000217692297 DE For-Sale Anodyne SCN9A 0 48 COC(=O)[C@@H](O)CNC(=O)[C@@H]1CC(=O)N(C2CCCC2)C1 ZINC000217692299 CB On-Demand Unstable INHA 46 46 CC(C)NC[C@@H]1CC[C@H]1N1CC[C@@H](c2ccccc2)C1 ZINC000217692308 CG For-Sale Unstable VACHT_TETCF 0 43 CC(C)NC[C@@H]1CC[C@H]1N1CC[C@@H](c2ccccc2)C1 ZINC000217692308 CG For-Sale Unstable SLC18A3 64 43 CSC[C@@](C)(O)CNC(=O)Cc1ccc2ccccc2c1 ZINC000217692337 DF On-Demand Unstable GSR 39 40 O=C(O)c1ccc(NC(=O)c2cnco2)cc1 ZINC000217692339 BD In-Stock Anodyne PRNP 41 36 O=C(O)c1ccc(NC(=O)c2cnco2)cc1 ZINC000217692339 BD In-Stock Anodyne NAMPT 20 43 C[C@](O)(CNC(=O)/C=C\c1ccc(Cl)c(Cl)c1)CC(=O)O ZINC000217692344 EE For-Sale Unstable PYGL 33 64 Cc1ccccc1/C=C/NC(=O)N1CCN(c2ccccc2)CC1 ZINC000217692372 DG For-Sale Unstable AKR1C3 0 43 Cc1cc(S(=O)(=O)Nc2nccs2)ccc1/C=C\C(=O)O ZINC000217692378 DE For-Sale Unstable SCN9A 0 52 COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1NC(=O)/C(F)=C\CN(C)C ZINC000217692405 JI Annotated Unstable EGFR 184 74 COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1NC(=O)/C(F)=C\CN(C)C ZINC000217692405 JI Annotated Unstable ERBB2 105 74 COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1NC(=O)/C(F)=C\CN(C)C ZINC000217692405 JI Annotated Unstable PDGFRB 28 45 COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1NC(=O)/C(F)=C\CN(C)C ZINC000217692405 JI Annotated Unstable MAP2K5 20 40 COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1NC(=O)/C(F)=C\CN(C)C ZINC000217692405 JI Annotated Unstable AURKB 55 45 COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1NC(=O)/C(F)=C\CN(C)C ZINC000217692405 JI Annotated Unstable FLT1 25 46 COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1NC(=O)/C(F)=C\CN(C)C ZINC000217692405 JI Annotated Unstable KDR 25 46 COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1NC(=O)/C(F)=C\CN(C)C ZINC000217692405 JI Annotated Unstable ABL2 16 40 COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1NC(=O)/C(F)=C\CN(C)C ZINC000217692405 JI Annotated Unstable BLK 15 45 COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1NC(=O)/C(F)=C\CN(C)C ZINC000217692405 JI Annotated Unstable FLT4 36 45 COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1NC(=O)/C(F)=C\CN(C)C ZINC000217692405 JI Annotated Unstable FLT3 17 45 COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1NC(=O)/C(F)=C\CN(C)C ZINC000217692405 JI Annotated Unstable ERBB4 77 74 COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1NC(=O)/C(F)=C\CN(C)C ZINC000217692405 JI Annotated Unstable CSF1R 16 43 COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1NC(=O)/C(F)=C\CN(C)C ZINC000217692405 JI Annotated Unstable AURKA 44 38 COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1NC(=O)/C(F)=C\CN(C)C ZINC000217692405 JI Annotated Unstable GAK 15 40 COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1NC(=O)/C(F)=C\CN(C)C ZINC000217692405 JI Annotated Unstable EPHA2 54 49 COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1NC(=O)/C(F)=C\CN(C)C ZINC000217692405 JI Annotated Unstable EPHA8 21 40 COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1NC(=O)/C(F)=C\CN(C)C ZINC000217692405 JI Annotated Unstable EPHA5 32 40 COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1NC(=O)/C(F)=C\CN(C)C ZINC000217692405 JI Annotated Unstable EPHA6 15 45 COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1NC(=O)/C(F)=C\CN(C)C ZINC000217692405 JI Annotated Unstable MKNK1 32 58 COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1NC(=O)/C(F)=C\CN(C)C ZINC000217692405 JI Annotated Unstable TIE1 22 40 COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1NC(=O)/C(F)=C\CN(C)C ZINC000217692405 JI Annotated Unstable DDR1 15 40 COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1NC(=O)/C(F)=C\CN(C)C ZINC000217692405 JI Annotated Unstable ABCG2 16 47 COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1NC(=O)/C(F)=C\CN(C)C ZINC000217692405 JI Annotated Unstable HIPK4 15 45 O=C(c1ccc(F)cc1Cl)N1CCC[C@@H](N2CCCC2=O)C1 ZINC000217692413 DF In-Stock Unstable P2RX7 29 46 CSC[C@](C)(O)CNC(=O)Cc1ccc2ccccc2c1 ZINC000217692420 DF On-Demand Unstable GSR 39 40 C[C@@](O)(CNC(=O)/C=C\c1ccc(Cl)c(Cl)c1)CC(=O)O ZINC000217692422 EE For-Sale Unstable PYGL 33 64 CC[C@H](C(=O)O)N(C)C(=O)/C=C\c1ccc2c(c1)OCO2 ZINC000217692423 CD On-Demand Unstable EDNRB 30 48 CC[C@H](C(=O)O)N(C)C(=O)/C=C\c1ccc2c(c1)OCO2 ZINC000217692423 CD On-Demand Unstable DYRK2 66 37 CC(C)CNS(=O)(=O)c1ccc(/C=C\C(=O)O)cc1Cl ZINC000217692451 DE For-Sale Unstable NR0B2 0 40 COC(=O)[C@@H](O)CNC(=O)[C@H]1CC(=O)N(C2CCCC2)C1 ZINC000217692455 CB On-Demand Unstable INHA 46 46 COC(=O)C[C@H](c1ccc(OC)cc1)c1c(O)cc(C)n(CCc2ccc(O)cc2)c1=O ZINC000217692477 IH In-Stock Unstable RORC 36 40 CC[C@@H](C(=O)O)N(C)C(=O)/C=C\c1ccc2c(c1)OCO2 ZINC000217692512 CD On-Demand Unstable EDNRB 30 48 CC[C@@H](C(=O)O)N(C)C(=O)/C=C\c1ccc2c(c1)OCO2 ZINC000217692512 CD On-Demand Unstable DYRK2 66 37 O=C(c1ccc(F)cc1Cl)N1CCC[C@H](N2CCCC2=O)C1 ZINC000217692516 DF In-Stock Unstable P2RX7 29 46 CCCOc1ccc(C(=O)NC[C@@](C)(O)CSC)cc1 ZINC000217692543 CE For-Sale Unstable PLA2G4B 82 40 COC(=O)C[C@@H](c1ccc(OC)cc1)c1c(O)cc(C)n(CCc2ccc(O)cc2)c1=O ZINC000217692559 IH In-Stock Unstable RORC 36 40 Clc1ccc(C2CC(N[C@@H]3CCN4CCCC[C@@H]34)C2)cc1 ZINC000217692571 DH On-Demand Unstable SLC18A3 28 52 CCCCCCCCN[C@@H](CC)CCO ZINC000217692588 BG For-Sale Unstable CQSS 40 31 Cc1ccccc1/C=C/NC(=O)Nc1c(C)cccc1C ZINC000217692619 CI For-Sale Unstable S1PR4 23 41 Cc1ccccc1/C=C/NC(=O)Nc1c(C)cccc1C ZINC000217692619 CI For-Sale Unstable ACAT 0 42 CCCOc1ccc(C(=O)NC[C@](C)(O)CSC)cc1 ZINC000217692628 CE For-Sale Unstable PLA2G4B 82 40 Clc1ccc(C2CC(N[C@H]3CCN4CCCC[C@@H]34)C2)cc1 ZINC000217692648 DH On-Demand Unstable SLC18A3 28 52 CCCCCCCCN[C@H](CC)CCO ZINC000217692671 BG For-Sale Unstable CQSS 40 31 CCOC(=O)c1ccc(-c2ccc(F)cc2)nc1N ZINC000217692672 CF In-Stock Unstable GCGR 0 40 CCCC[C@H](C(=O)O)C1CCC1 ZINC000217692695 AF In-Stock Unstable CPN1 0 41 CCCC[C@H](C(=O)O)C1CCC1 ZINC000217692695 AF In-Stock Unstable SLC22A20 0 44 COc1ccc([N+](=O)[O-])cc1NC(=O)N/C=C/c1ccccc1C ZINC000217692739 EH For-Sale Unstable KCNMA1 28 54 COc1ccc([N+](=O)[O-])cc1NC(=O)N/C=C/c1ccccc1C ZINC000217692739 EH For-Sale Unstable DDX3X 0 44 CCCC[C@@H](C(=O)O)C1CCC1 ZINC000217692782 AF In-Stock Unstable CPN1 0 41 CCCC[C@@H](C(=O)O)C1CCC1 ZINC000217692782 AF In-Stock Unstable SLC22A20 0 44 O=[N+]([O-])c1cccc(CN[C@@H]2CCN3CCC[C@@H]23)c1 ZINC000217692785 CD For-Sale Unstable CACNA1D 61 36 CC(C)c1cc(C(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)n(-c2ccccc2)n1 ZINC000217692815 HG In-Stock Unstable CHRNA4 27 44 O=C(c1ccc(OC(F)(F)F)cc1)N1CCc2oncc2C1 ZINC000217692839 DF In-Stock Unstable EPHX2 39 41 O=C(O)/C=C\c1cccc(S(=O)(=O)N2CCC(O)CC2)c1 ZINC000217692844 DC For-Sale Unstable HDAC8 30 42 O=C(O)/C=C\c1cccc(S(=O)(=O)N2CCC(O)CC2)c1 ZINC000217692844 DC For-Sale Unstable HDAC1 16 44 O=C(O)/C=C\c1cccc(S(=O)(=O)N2CCC(O)CC2)c1 ZINC000217692844 DC For-Sale Unstable HDAC6 18 42 O=C(O)/C=C\c1cccc(S(=O)(=O)N2CCC(O)CC2)c1 ZINC000217692844 DC For-Sale Unstable AKR1C3 63 40 O=[N+]([O-])c1cccc(CN[C@H]2CCN3CCC[C@@H]23)c1 ZINC000217692865 CD For-Sale Unstable CACNA1D 61 36 Cc1cnc(NS(=O)(=O)c2cccc(/C=C\C(=O)O)c2)s1 ZINC000217692920 DE For-Sale Unstable HDAC8 29 48 CSC[C@@](C)(O)CNC(=O)CCc1ccccc1Cl ZINC000217692935 DF On-Demand Unstable PSMB5 30 42 NC(=O)c1ccsc1NC(=O)NC1CCCCC1 ZINC000217692966 CE For-Sale Unstable EPHX2 28 50 NC(=O)c1ccsc1NC(=O)NC1CCCCC1 ZINC000217692966 CE For-Sale Unstable CHEK1 15 41 O=[N+]([O-])c1ccc(CN[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217692987 CD For-Sale Unstable KCNJ1 25 41 CSC[C@](C)(O)CNC(=O)CCc1ccccc1Cl ZINC000217693026 DF On-Demand Unstable PSMB5 30 42 O=C(O)[C@@H](CC1CC1)C1CCC1 ZINC000217693033 AE In-Stock Unstable CPN1 0 42 O=C(O)[C@@H](CC1CC1)C1CCC1 ZINC000217693033 AE In-Stock Unstable CPB2 16 42 CN(C)CCCNS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217693034 DD For-Sale Unstable BDKRB1 0 41 CN(C)CCCNS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217693034 DD For-Sale Unstable AKR1C3 27 43 CC[C@H](C(=O)O)N(C)C(=O)/C=C\c1ccccc1[N+](=O)[O-] ZINC000217693040 CD For-Sale Unstable COLA 76 33 CC[C@H](C(=O)O)N(C)C(=O)/C=C\c1ccccc1[N+](=O)[O-] ZINC000217693040 CD For-Sale Unstable TLR4 18 46 O=[N+]([O-])c1ccc(CN[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217693054 CD For-Sale Unstable KCNJ1 25 41 COC(=O)[C@@H](O)CNC(=O)c1ccc2c(c1)CCO2 ZINC000217693069 CB On-Demand Unstable F3 62 34 CC(C)(C)NC(=O)Nc1sccc1C(N)=O ZINC000217693093 BD For-Sale Unstable MAPK8 27 54 COc1ccc(-c2csc(Nc3cccc(C)c3)n2)cc1N ZINC000217693104 DI In-Stock Unstable MAOA 0 40 COc1ccc(-c2csc(Nc3cccc(C)c3)n2)cc1N ZINC000217693104 DI In-Stock Unstable MAOB 0 41 COc1ccc(-c2csc(Nc3cccc(C)c3)n2)cc1N ZINC000217693104 DI In-Stock Unstable SPHK2 40 37 COc1ccc(-c2csc(Nc3cccc(C)c3)n2)cc1N ZINC000217693104 DI In-Stock Unstable PLAU 18 42 COc1ccc(-c2csc(Nc3cccc(C)c3)n2)cc1N ZINC000217693104 DI In-Stock Unstable VCP 18 44 CC[C@@H](C(=O)O)N(C)C(=O)/C=C\c1ccccc1[N+](=O)[O-] ZINC000217693129 CD For-Sale Unstable COLA 76 33 CC[C@@H](C(=O)O)N(C)C(=O)/C=C\c1ccccc1[N+](=O)[O-] ZINC000217693129 CD For-Sale Unstable TLR4 18 46 O=C(O)[C@H](CC1CC1)C1CCC1 ZINC000217693135 AE In-Stock Unstable CPN1 0 42 O=C(O)[C@H](CC1CC1)C1CCC1 ZINC000217693135 AE In-Stock Unstable CPB2 16 42 O=C(O)/C=C\c1cccc(C(=O)Nc2ccc(Cl)cn2)c1 ZINC000217693143 DG For-Sale Anodyne KLKB1 32 43 O=C(O)/C=C\c1cccc(C(=O)Nc2ccc(Cl)cn2)c1 ZINC000217693143 DG For-Sale Anodyne F10 50 46 O=C(O)/C=C\c1cccc(C(=O)Nc2ccc(Cl)cn2)c1 ZINC000217693143 DG For-Sale Anodyne GRM5 16 45 O=C(O)/C=C\c1cccc(C(=O)Nc2ccc(Cl)cn2)c1 ZINC000217693143 DG For-Sale Anodyne GCK 20 43 O=C(O)/C=C\c1cccc(C(=O)Nc2ccc(Cl)cn2)c1 ZINC000217693143 DG For-Sale Anodyne LUCI_LUCLA 50 54 O=C(O)/C=C\c1cccc(C(=O)Nc2ccc(Cl)cn2)c1 ZINC000217693143 DG For-Sale Anodyne AKR1C3 30 40 O=C(O)/C=C\c1cccc(C(=O)Nc2ccc(Cl)cn2)c1 ZINC000217693143 DG For-Sale Anodyne RHOA 0 44 O=C(O)/C=C\c1cccc(C(=O)Nc2ccc(Cl)cn2)c1 ZINC000217693143 DG For-Sale Anodyne KCNK3 67 41 O=C(O)/C=C\c1cccc(C(=O)Nc2ccc(Cl)cn2)c1 ZINC000217693143 DG For-Sale Anodyne KCNK9 40 36 COC(=O)[C@H](O)CNC(=O)c1ccc2c(c1)CCO2 ZINC000217693145 CB For-Sale Unstable F3 62 34 O=[N+]([O-])c1ccccc1CN[C@@H]1CCN2CCC[C@@H]12 ZINC000217693162 CD For-Sale Unstable COLA 94 33 CCCCNC(=O)Nc1sccc1C(N)=O ZINC000217693206 BD For-Sale Unstable MAPK8 26 52 C[C@](O)(CNC(=O)/C=C\c1cc(Cl)cc(Cl)c1)CC(=O)O ZINC000217693213 EE For-Sale Unstable PYGL 0 44 Cc1ccccc1/C=C/NC(=O)NCCC(C)C ZINC000217693215 BG For-Sale Unstable DNPEP 0 42 O=C(O)/C=C\c1ccc(C(=O)Nc2ccc(F)c(Cl)c2)s1 ZINC000217693231 EH For-Sale Anodyne MAOB 16 42 O=[N+]([O-])c1ccccc1CN[C@H]1CCN2CCC[C@@H]12 ZINC000217693257 CD For-Sale Unstable COLA 94 33 CC[C@H](C(=O)O)N(C)C(=O)/C=C\c1ccc(OC)cc1 ZINC000217693265 CE On-Demand Unstable PTGS2 18 45 C[C@@](O)(CNC(=O)/C=C\c1cc(Cl)cc(Cl)c1)CC(=O)O ZINC000217693314 EE For-Sale Unstable PYGL 0 44 COC(=O)[C@H](O)CNC(=O)[C@@H](NC(C)=O)C(C)C ZINC000217693341 CA For-Sale Unstable PGA 40 37 CC[C@@H](C(=O)O)N(C)C(=O)/C=C\c1ccc(OC)cc1 ZINC000217693357 CE On-Demand Unstable PTGS2 18 45 Cc1cnc(Cl)nc1N1CCN(C)[C@@H](C)C1 ZINC000217693367 BD For-Sale Unstable ADRA2A 0 42 Cc1cnc(Cl)nc1N1CCN(C)[C@@H](C)C1 ZINC000217693367 BD For-Sale Unstable ADRA2B 0 42 Cc1cnc(Cl)nc1N1CCN(C)[C@@H](C)C1 ZINC000217693367 BD For-Sale Unstable ADRA2C 0 42 C[C@@H]1CCCCN1C(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217693404 CF For-Sale Unstable PREP 26 42 C[C@@H]1CCCCN1C(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217693404 CF For-Sale Unstable L3MBTL3 48 35 O=C(c1c[nH]c2ccccc12)N1CCc2oncc2C1 ZINC000217693420 CE In-Stock Unstable AVPR1A 23 48 CCNC(=O)Nc1sccc1C(N)=O ZINC000217693454 BC For-Sale Unstable MAPK8 28 57 O=C(O)c1cccc(NC(=O)c2cnco2)c1 ZINC000217693471 BD In-Stock Anodyne ROCK2 18 40 O=C(O)c1cccc(NC(=O)c2cnco2)c1 ZINC000217693471 BD In-Stock Anodyne NR1H4 0 41 O=C(O)c1cccc(NC(=O)c2cnco2)c1 ZINC000217693471 BD In-Stock Anodyne AKR1C3 42 47 O=C(O)c1cccc(NC(=O)c2cnco2)c1 ZINC000217693471 BD In-Stock Anodyne NAMPT 16 40 O=C(O)c1cccc(NC(=O)c2cnco2)c1 ZINC000217693471 BD In-Stock Anodyne KCNK3 96 50 O=C(O)c1cccc(NC(=O)c2cnco2)c1 ZINC000217693471 BD In-Stock Anodyne KCNK9 75 40 C[C@H]1CCCCN1C(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217693496 CF For-Sale Unstable PREP 26 42 C[C@H]1CCCCN1C(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217693496 CF For-Sale Unstable L3MBTL3 48 35 COC(=O)[C@H](O)CNC(=O)[C@H](NC(C)=O)C(C)C ZINC000217693506 CA For-Sale Unstable PGA 40 37 Cc1c(C(=O)N2CCc3oncc3C2)cnn1-c1ccccc1 ZINC000217693538 DE In-Stock Unstable SLC9A2 0 47 Cc1c(C(=O)N2CCc3oncc3C2)cnn1-c1ccccc1 ZINC000217693538 DE In-Stock Unstable BCL2 24 44 O=C(Cc1c[nH]cn1)N1CCCC[C@@H]1c1ccccn1 ZINC000217693568 CE In-Stock Unstable HRH1 0 40 O=C(Cc1c[nH]cn1)N1CCCC[C@@H]1c1ccccn1 ZINC000217693568 CE In-Stock Unstable PGC 45 36 O=C(Cc1c[nH]cn1)N1CCCC[C@@H]1c1ccccn1 ZINC000217693568 CE In-Stock Unstable COLA 133 46 O=C(Cc1c[nH]cn1)N1CCCC[C@@H]1c1ccccn1 ZINC000217693568 CE In-Stock Unstable CPT1A 116 46 O=C(Cc1c[nH]cn1)N1CCCC[C@@H]1c1ccccn1 ZINC000217693568 CE In-Stock Unstable CTSE 45 36 C[C@@H]1CCCCN1C(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217693579 CF For-Sale Unstable PREP 41 46 Clc1cccc(Nc2ncnc(Cl)c2-c2ccccc2)c1 ZINC000217693584 DK In-Stock Anodyne ABL1 23 53 Clc1cccc(Nc2ncnc(Cl)c2-c2ccccc2)c1 ZINC000217693584 DK In-Stock Anodyne EGFR 75 64 Clc1cccc(Nc2ncnc(Cl)c2-c2ccccc2)c1 ZINC000217693584 DK In-Stock Anodyne ERBB2 20 49 Clc1cccc(Nc2ncnc(Cl)c2-c2ccccc2)c1 ZINC000217693584 DK In-Stock Anodyne FBP1 0 51 Clc1cccc(Nc2ncnc(Cl)c2-c2ccccc2)c1 ZINC000217693584 DK In-Stock Anodyne CD38 20 45 Clc1cccc(Nc2ncnc(Cl)c2-c2ccccc2)c1 ZINC000217693584 DK In-Stock Anodyne MKNK1 22 51 Clc1cccc(Nc2ncnc(Cl)c2-c2ccccc2)c1 ZINC000217693584 DK In-Stock Anodyne ABCG2 23 51 Clc1cccc(Nc2ncnc(Cl)c2-c2ccccc2)c1 ZINC000217693584 DK In-Stock Anodyne AHK4 0 42 Clc1cccc(Nc2ncnc(Cl)c2-c2ccccc2)c1 ZINC000217693584 DK In-Stock Anodyne CKX2 0 42 Brc1ccccc1C1CC(N[C@@H]2CCN3CCCC[C@@H]23)C1 ZINC000217693616 EH For-Sale Unstable SLC18A3 28 52 O=C(Cc1c[nH]cn1)N1CCCC[C@H]1c1ccccn1 ZINC000217693663 CE In-Stock Unstable HRH1 0 40 O=C(Cc1c[nH]cn1)N1CCCC[C@H]1c1ccccn1 ZINC000217693663 CE In-Stock Unstable PGC 45 36 O=C(Cc1c[nH]cn1)N1CCCC[C@H]1c1ccccn1 ZINC000217693663 CE In-Stock Unstable COLA 133 46 O=C(Cc1c[nH]cn1)N1CCCC[C@H]1c1ccccn1 ZINC000217693663 CE In-Stock Unstable CPT1A 116 46 O=C(Cc1c[nH]cn1)N1CCCC[C@H]1c1ccccn1 ZINC000217693663 CE In-Stock Unstable CTSE 45 36 C[C@H]1CCCCN1C(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217693676 CF For-Sale Unstable PREP 41 46 Brc1ccccc1C1CC(N[C@H]2CCN3CCCC[C@@H]23)C1 ZINC000217693684 EH For-Sale Unstable SLC18A3 28 52 c1ccc(CCCN[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217693751 BE For-Sale Unstable SLC18A2 44 39 c1ccc(CCCN[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217693751 BE For-Sale Unstable SIGMAR1 35 51 c1ccc(CCCN[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217693751 BE For-Sale Unstable SLC18A3 40 34 c1ccc(CCCN[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217693751 BE For-Sale Unstable PREP 44 37 O=C(O)/C=C\c1ccc(F)c(C(=O)NC2CCCC2)c1 ZINC000217693765 CF For-Sale Unstable CNR1 19 44 O=C(O)/C=C\c1ccc(F)c(C(=O)NC2CCCC2)c1 ZINC000217693765 CF For-Sale Unstable CNR2 23 44 O=C(c1csc(-c2ccccc2)n1)N1CCc2oncc2C1 ZINC000217693767 DF In-Stock Unstable TRPC6 41 42 O=C(c1csc(-c2ccccc2)n1)N1CCc2oncc2C1 ZINC000217693767 DF In-Stock Unstable TRPC3 26 41 c1ccc(CCCN[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217693828 BE For-Sale Unstable SLC18A2 44 39 c1ccc(CCCN[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217693828 BE For-Sale Unstable SIGMAR1 35 51 c1ccc(CCCN[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217693828 BE For-Sale Unstable SLC18A3 40 34 c1ccc(CCCN[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217693828 BE For-Sale Unstable PREP 44 37 COc1ccc(/C=C/C(=O)NC[C@@](C)(O)CSC)cc1 ZINC000217693836 CD On-Demand Unstable HDAC8 0 52 COc1ccc(/C=C/C(=O)NC[C@@](C)(O)CSC)cc1 ZINC000217693836 CD On-Demand Unstable HDAC1 0 44 COc1ccc(/C=C/C(=O)NC[C@@](C)(O)CSC)cc1 ZINC000217693836 CD On-Demand Unstable GPR183 0 40 O=C(O)/C=C\c1ccc(C(=O)NC2CCCC2)c(F)c1 ZINC000217693847 CF For-Sale Unstable CNR1 16 42 O=C(O)/C=C\c1ccc(C(=O)NC2CCCC2)c(F)c1 ZINC000217693847 CF For-Sale Unstable CNR2 24 42 COc1ccc([C@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c(OC)c1 ZINC000217693857 KH In-Stock Unstable CYP1B1 50 39 COc1ccc([C@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c(OC)c1 ZINC000217693857 KH In-Stock Unstable CYP1A1 40 39 COc1ccc([C@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c(OC)c1 ZINC000217693857 KH In-Stock Unstable ABCB1 17 42 COc1ccc([C@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c(OC)c1 ZINC000217693857 KH In-Stock Unstable RORC 0 43 COc1ccc(/C=C/C(=O)NC[C@](C)(O)CSC)cc1 ZINC000217693915 CD On-Demand Unstable HDAC8 0 52 COc1ccc(/C=C/C(=O)NC[C@](C)(O)CSC)cc1 ZINC000217693915 CD On-Demand Unstable HDAC1 0 44 COc1ccc(/C=C/C(=O)NC[C@](C)(O)CSC)cc1 ZINC000217693915 CD On-Demand Unstable GPR183 0 40 O=C(O)/C=C\c1ccc(F)c(C(=O)N2CCCCCC2)c1 ZINC000217693927 CF For-Sale Unstable PARP1 51 36 O=C(O)c1cc2c(N3CCCC3)ncnc2s1 ZINC000217693934 BD In-Stock Unstable SIRT3 67 41 O=C(O)c1cc2c(N3CCCC3)ncnc2s1 ZINC000217693934 BD In-Stock Unstable SIRT2 53 35 O=C(O)c1cc2c(N3CCCC3)ncnc2s1 ZINC000217693934 BD In-Stock Unstable SIRT1 44 41 CCCCCCN[C@@H](CC)CCO ZINC000217693939 AE For-Sale Unstable SLC6A8 40 32 CCCCCCN[C@@H](CC)CCO ZINC000217693939 AE For-Sale Unstable Q6UB75_PIG 0 47 CCCCCCN[C@@H](CC)CCO ZINC000217693939 AE For-Sale Unstable CQSS 40 31 COc1ccc([C@@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c(OC)c1 ZINC000217693943 KH In-Stock Unstable CYP1B1 50 39 COc1ccc([C@@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c(OC)c1 ZINC000217693943 KH In-Stock Unstable CYP1A1 40 39 COc1ccc([C@@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c(OC)c1 ZINC000217693943 KH In-Stock Unstable ABCB1 17 42 COc1ccc([C@@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c(OC)c1 ZINC000217693943 KH In-Stock Unstable RORC 47 43 O=S(=O)(c1cccnc1)N1CCc2oncc2C1 ZINC000217693975 CC In-Stock Unstable AKR1C3 61 44 C[C@](O)(CNC(=O)/C=C\c1ccc(Cl)cc1Cl)CC(=O)O ZINC000217693988 EE For-Sale Unstable PYGL 0 40 C[C@](O)(CNC(=O)/C=C\c1ccc(Cl)cc1Cl)CC(=O)O ZINC000217693988 EE For-Sale Unstable BOTA 31 54 CCCCCCN[C@H](CC)CCO ZINC000217694016 AE For-Sale Unstable SLC6A8 40 32 CCCCCCN[C@H](CC)CCO ZINC000217694016 AE For-Sale Unstable Q6UB75_PIG 0 47 CCCCCCN[C@H](CC)CCO ZINC000217694016 AE For-Sale Unstable CQSS 40 31 C[C@@](O)(CNC(=O)/C=C\c1ccc(Cl)cc1Cl)CC(=O)O ZINC000217694069 EE For-Sale Unstable PYGL 0 40 C[C@@](O)(CNC(=O)/C=C\c1ccc(Cl)cc1Cl)CC(=O)O ZINC000217694069 EE For-Sale Unstable BOTA 31 54 CSC[C@@](C)(O)CNC(=O)Cc1c(Cl)cccc1Cl ZINC000217694078 DF On-Demand Unstable P2RX7 18 42 O=S(=O)(c1ccccc1F)N1CCc2oncc2C1 ZINC000217694090 CD In-Stock Unstable PKM 20 42 C/C(=N/NC(N)=S)c1ccc(I)cc1 ZINC000217694135 DD For-Sale Unstable CTSL 33 45 C/C(=N/NC(N)=S)c1ccc(I)cc1 ZINC000217694135 DD For-Sale Unstable PPO2 111 82 CC[C@H](C(=O)O)N(C)C(=O)/C=C\c1cccc([N+](=O)[O-])c1 ZINC000217694138 CD For-Sale Unstable CACNA1C 51 39 CC[C@H](C(=O)O)N(C)C(=O)/C=C\c1cccc([N+](=O)[O-])c1 ZINC000217694138 CD For-Sale Unstable CACNA1D 81 39 CC[C@H](C(=O)O)N(C)C(=O)/C=C\c1cccc([N+](=O)[O-])c1 ZINC000217694138 CD For-Sale Unstable TRPM8 0 47 CC[C@@H](CCO)N[C@@H](C)Cc1ccccc1 ZINC000217694145 BE For-Sale Unstable ACE 21 42 CC[C@@H](CCO)N[C@@H](C)Cc1ccccc1 ZINC000217694145 BE For-Sale Unstable MME 74 42 CC[C@@H](CCO)N[C@@H](C)Cc1ccccc1 ZINC000217694145 BE For-Sale Unstable ANPEP 63 37 CC[C@@H](CCO)N[C@@H](C)Cc1ccccc1 ZINC000217694145 BE For-Sale Unstable ACE2 44 37 COc1cc2c(c(OC)c1OC)-c1ccc(NCCCCCC(=O)Nc3ccn(C)n3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217694166 KI In-Stock Unstable TUBA1A 17 62 COc1cc2c(c(OC)c1OC)-c1ccc(NCCCCCC(=O)Nc3ccn(C)n3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217694166 KI In-Stock Unstable TPPP 0 58 CSC[C@](C)(O)CNC(=O)Cc1c(Cl)cccc1Cl ZINC000217694172 DF On-Demand Unstable P2RX7 18 42 COC(=O)[C@@H](O)CNC(=O)c1cc(OC)cs1 ZINC000217694194 CC On-Demand Unstable TBK1 22 41 CC[C@@H](C(=O)O)N(C)C(=O)/C=C\c1cccc([N+](=O)[O-])c1 ZINC000217694217 CD For-Sale Unstable CACNA1C 51 39 CC[C@@H](C(=O)O)N(C)C(=O)/C=C\c1cccc([N+](=O)[O-])c1 ZINC000217694217 CD For-Sale Unstable CACNA1D 81 39 CC[C@@H](C(=O)O)N(C)C(=O)/C=C\c1cccc([N+](=O)[O-])c1 ZINC000217694217 CD For-Sale Unstable TRPM8 0 47 CC[C@H](CCO)N[C@@H](C)Cc1ccccc1 ZINC000217694228 BE For-Sale Unstable ACE 21 42 CC[C@H](CCO)N[C@@H](C)Cc1ccccc1 ZINC000217694228 BE For-Sale Unstable MME 74 42 CC[C@H](CCO)N[C@@H](C)Cc1ccccc1 ZINC000217694228 BE For-Sale Unstable ANPEP 63 37 CC[C@H](CCO)N[C@@H](C)Cc1ccccc1 ZINC000217694228 BE For-Sale Unstable ACE2 44 37 Cc1cc(SCC(=O)O)nc(COc2cccc(Cl)c2)n1 ZINC000217694261 DG In-Stock Unstable PDS 35 41 COC(=O)[C@H](O)CNC(=O)c1cc(OC)cs1 ZINC000217694265 CC On-Demand Unstable TBK1 22 41 CSC[C@@](C)(O)CNC(=O)/C=C/c1cccc(F)c1 ZINC000217694273 CE On-Demand Unstable IMPDH2 18 40 Cc1ccc(S(=O)(=O)N2CCc3oncc3C2)cc1C ZINC000217694304 CE In-Stock Unstable AKR1C3 63 41 CC[C@@H](CCO)N[C@H](C)Cc1ccccc1 ZINC000217694321 BE For-Sale Unstable ACE 21 42 CC[C@@H](CCO)N[C@H](C)Cc1ccccc1 ZINC000217694321 BE For-Sale Unstable MME 74 42 CC[C@@H](CCO)N[C@H](C)Cc1ccccc1 ZINC000217694321 BE For-Sale Unstable ANPEP 63 37 CC[C@@H](CCO)N[C@H](C)Cc1ccccc1 ZINC000217694321 BE For-Sale Unstable ACE2 44 37 CSC[C@](C)(O)CNC(=O)/C=C/c1cccc(F)c1 ZINC000217694361 CE On-Demand Unstable IMPDH2 18 40 CC[C@H](C(=O)O)N(C)C(=O)/C=C\c1ccccc1 ZINC000217694370 BE On-Demand Unstable NA 0 40 CC[C@H](C(=O)O)N(C)C(=O)/C=C\c1ccccc1 ZINC000217694370 BE On-Demand Unstable F3 18 44 O=C(O)c1ccc(-c2ccccc2)nc1NC1CCCCC1 ZINC000217694378 CI In-Stock Unstable ADORA1 19 44 O=C(O)c1ccc(-c2ccccc2)nc1NC1CCCCC1 ZINC000217694378 CI In-Stock Unstable P2RY12 19 40 O=C(O)c1ccc(-c2ccccc2)nc1NC1CCCCC1 ZINC000217694378 CI In-Stock Unstable PRKD1 54 34 O=C(O)c1ccc(-c2ccccc2)nc1NC1CCCCC1 ZINC000217694378 CI In-Stock Unstable GSK3A 23 41 O=C(O)c1ccc(-c2ccccc2)nc1NC1CCCCC1 ZINC000217694378 CI In-Stock Unstable ADORA3 0 42 O=C(O)c1ccc(-c2ccccc2)nc1NC1CCCCC1 ZINC000217694378 CI In-Stock Unstable MAPK8 15 46 O=C(O)c1ccc(-c2ccccc2)nc1NC1CCCCC1 ZINC000217694378 CI In-Stock Unstable TYRO3 41 37 CC[C@H](CCO)N[C@H](C)Cc1ccccc1 ZINC000217694402 BE For-Sale Unstable ACE 21 42 CC[C@H](CCO)N[C@H](C)Cc1ccccc1 ZINC000217694402 BE For-Sale Unstable MME 74 42 CC[C@H](CCO)N[C@H](C)Cc1ccccc1 ZINC000217694402 BE For-Sale Unstable ANPEP 63 37 CC[C@H](CCO)N[C@H](C)Cc1ccccc1 ZINC000217694402 BE For-Sale Unstable ACE2 44 37 CC[C@@H](C)c1ccccc1NC(=O)N/C=C/c1ccccc1C ZINC000217694441 DK For-Sale Unstable AO-ACHE 0 40 CC[C@@H](C(=O)O)N(C)C(=O)/C=C\c1ccccc1 ZINC000217694456 BE On-Demand Unstable NA 0 40 CC[C@@H](C(=O)O)N(C)C(=O)/C=C\c1ccccc1 ZINC000217694456 BE On-Demand Unstable F3 18 44 COc1cc2c(c(OC)c1OC)-c1ccc(NCCCCCC(=O)NCc3nc4ccccc4n3C)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217694484 KK In-Stock Unstable TUBA1A 16 56 Cc1cc(S(=O)(=O)N2CCc3oncc3C2)ccc1F ZINC000217694525 CD In-Stock Unstable AKR1C3 59 37 Cc1cc(S(=O)(=O)N2CCc3oncc3C2)ccc1F ZINC000217694525 CD In-Stock Unstable LEF 48 34 CC[C@H](C)c1ccccc1NC(=O)N/C=C/c1ccccc1C ZINC000217694529 DK For-Sale Unstable AO-ACHE 0 40 COc1ccccc1[C@@H]1CCCN1C(=O)CN(C)Cc1cccnc1 ZINC000217694583 EF In-Stock Unstable NPY2R 42 34 COc1ccccc1[C@@H]1CCCN1C(=O)CN(C)Cc1cccnc1 ZINC000217694583 EF In-Stock Unstable CHRNA7 34 42 COc1ccccc1[C@@H]1CCCN1C(=O)CN(C)Cc1cccnc1 ZINC000217694583 EF In-Stock Unstable COLA 78 38 COc1ccccc1[C@@H]1CCCN1C(=O)CN(C)Cc1cccnc1 ZINC000217694583 EF In-Stock Unstable CPT1A 78 36 COc1ccccc1[C@@H]1CCCN1C(=O)CN(C)Cc1cccnc1 ZINC000217694583 EF In-Stock Unstable PREP 51 36 COc1ccccc1[C@@H]1CCCN1C(=O)CN(C)Cc1cccnc1 ZINC000217694583 EF In-Stock Unstable ACKR3 51 31 Nc1ccc(Cc2noc(-c3ccccc3F)n2)cc1 ZINC000217694600 CG In-Stock Unstable LUCI_PHOPE 15 43 Cc1cc(=O)c(O)c([C@H](CC(N)=O)c2ccc3c(c2)n(C)c(=O)n3C)o1 ZINC000217694603 FC In-Stock Unstable BRPF1 0 40 CSC[C@@](C)(O)CNC(=O)c1coc2ccccc12 ZINC000217694646 CE On-Demand Unstable INHA 61 33 CCNc1cc(=O)n(CC)c(=O)[nH]1 ZINC000217694650 AB For-Sale Unstable POLC 92 40 O=S(=O)(c1cccc(Cl)c1)N1CCc2oncc2C1 ZINC000217694652 CE In-Stock Unstable AKR1C3 71 51 COc1ccccc1[C@H]1CCCN1C(=O)CN(C)Cc1cccnc1 ZINC000217694670 EF In-Stock Unstable NPY2R 42 34 COc1ccccc1[C@H]1CCCN1C(=O)CN(C)Cc1cccnc1 ZINC000217694670 EF In-Stock Unstable CHRNA7 34 42 COc1ccccc1[C@H]1CCCN1C(=O)CN(C)Cc1cccnc1 ZINC000217694670 EF In-Stock Unstable COLA 78 38 COc1ccccc1[C@H]1CCCN1C(=O)CN(C)Cc1cccnc1 ZINC000217694670 EF In-Stock Unstable CPT1A 78 36 COc1ccccc1[C@H]1CCCN1C(=O)CN(C)Cc1cccnc1 ZINC000217694670 EF In-Stock Unstable PREP 51 36 COc1ccccc1[C@H]1CCCN1C(=O)CN(C)Cc1cccnc1 ZINC000217694670 EF In-Stock Unstable ACKR3 51 31 Cc1cc(=O)c(O)c([C@@H](CC(N)=O)c2ccc3c(c2)n(C)c(=O)n3C)o1 ZINC000217694684 FC In-Stock Unstable BRPF1 0 40 CSC[C@](C)(O)CNC(=O)c1coc2ccccc12 ZINC000217694717 CE On-Demand Unstable INHA 61 33 O[C@@H]1CCO[C@@H]1OCc1ccccc1 ZINC000217694734 AD For-Sale Unstable FIMH 18 50 COCCN(C(=O)c1cccc(/C=C\C(=O)O)c1)C1CC1 ZINC000217694737 CE For-Sale Unstable MBTPS1 53 32 COCCN(C(=O)c1cccc(/C=C\C(=O)O)c1)C1CC1 ZINC000217694737 CE For-Sale Unstable ACKR3 54 35 O=S(=O)(c1ccccc1Cl)N1CCc2oncc2C1 ZINC000217694759 CE In-Stock Unstable AKR1C3 40 38 Cc1ccccc1/C=C/NC(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000217694760 EH For-Sale Unstable CHRM2 24 42 Cc1ccccc1/C=C/NC(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000217694760 EH For-Sale Unstable CHRM1 19 48 Cc1ccccc1/C=C/NC(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000217694760 EH For-Sale Unstable DRD2 25 58 Cc1ccccc1/C=C/NC(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000217694760 EH For-Sale Unstable DRD4 56 58 Cc1ccccc1/C=C/NC(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000217694760 EH For-Sale Unstable ACHE 43 48 Cc1ccccc1/C=C/NC(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000217694760 EH For-Sale Unstable DRD3 27 58 Cc1ccccc1/C=C/NC(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000217694760 EH For-Sale Unstable KCNH2 16 41 Cc1ccccc1/C=C/NC(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000217694760 EH For-Sale Unstable CHRM3 28 48 Cc1ccccc1/C=C/NC(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000217694760 EH For-Sale Unstable SIGMAR1 60 59 Cc1ccccc1/C=C/NC(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000217694760 EH For-Sale Unstable SSTR5 53 38 Cc1ccccc1/C=C/NC(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000217694760 EH For-Sale Unstable CCR3 41 48 Cc1ccccc1/C=C/NC(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000217694760 EH For-Sale Unstable SLC6A5 19 43 Cc1ccccc1/C=C/NC(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000217694760 EH For-Sale Unstable EPHX2 25 52 Cc1ccccc1/C=C/NC(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000217694760 EH For-Sale Unstable MCHR1 57 48 Cc1ccccc1/C=C/NC(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000217694760 EH For-Sale Unstable CACNA1G 26 42 Cc1ccccc1/C=C/NC(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000217694760 EH For-Sale Unstable CCR8 22 46 Cc1ccccc1/C=C/NC(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000217694760 EH For-Sale Unstable ADIPOR1 0 47 Cc1ccccc1/C=C/NC(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000217694760 EH For-Sale Unstable ADIPOR2 0 47 COC(=O)[C@@H](O)CNC(=O)Cc1ccccc1[N+](=O)[O-] ZINC000217694762 CB On-Demand Unstable CACNA1D 45 31 COC(=O)[C@@H](O)CNC(=O)Cc1ccccc1[N+](=O)[O-] ZINC000217694762 CB On-Demand Unstable COLA 111 44 COC(=O)[C@H](O)CNC(=O)Cc1ccccc1[N+](=O)[O-] ZINC000217694840 CB On-Demand Unstable CACNA1D 45 31 COC(=O)[C@H](O)CNC(=O)Cc1ccccc1[N+](=O)[O-] ZINC000217694840 CB On-Demand Unstable COLA 111 44 O[C@H]1CCO[C@@H]1OCc1ccccc1 ZINC000217694841 AD For-Sale Unstable FIMH 18 50 CCOc1ccc(S(=O)(=O)N2CCc3oncc3C2)cc1C ZINC000217694875 DE In-Stock Unstable AKR1C3 54 35 COc1ccccc1-c1nc(Cc2ccc(N)cc2)no1 ZINC000217694905 CF In-Stock Unstable LUCI_PHOPE 37 48 COc1cccc2ccc(N3CCN(Cc4ccccc4)C[C@@H](O)C3)nc12 ZINC000217694960 FF In-Stock Unstable DRD2 37 40 COc1cccc2ccc(N3CCN(Cc4ccccc4)C[C@@H](O)C3)nc12 ZINC000217694960 FF In-Stock Unstable DRD4 48 41 COc1cccc2ccc(N3CCN(Cc4ccccc4)C[C@@H](O)C3)nc12 ZINC000217694960 FF In-Stock Unstable DRD3 39 41 COC(=O)[C@@H](O)CNC(=O)c1ccc([N+](=O)[O-])cc1 ZINC000217694964 CB On-Demand Unstable CA2 18 42 COC(=O)[C@@H](O)CNC(=O)c1ccc([N+](=O)[O-])cc1 ZINC000217694964 CB On-Demand Unstable CACNA1D 60 33 COC(=O)[C@@H](O)CNC(=O)c1ccc([N+](=O)[O-])cc1 ZINC000217694964 CB On-Demand Unstable CCR3 0 41 CCOc1ccc(S(=O)(=O)N2CCc3oncc3C2)cc1F ZINC000217694986 ED In-Stock Unstable AKR1C3 54 35 CSCC[C@H](NC(=O)CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)c1nc2ccccc2n1C ZINC000217695014 JG In-Stock Unstable AGAL_COFAR 0 44 CSCC[C@H](NC(=O)CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)c1nc2ccccc2n1C ZINC000217695014 JG In-Stock Unstable BIRA 0 40 O=C(O)/C=C\c1cccc(C(=O)NCCc2ccsc2)c1 ZINC000217695026 DF For-Sale Unstable HDAC8 20 40 O=C(O)/C=C\c1cccc(C(=O)NCCc2ccsc2)c1 ZINC000217695026 DF For-Sale Unstable KDM4E 21 40 COc1ccc(-c2csc(Nc3ccccc3OC)n2)cc1N ZINC000217695034 EI In-Stock Unstable MAOB 27 42 COc1ccc(-c2csc(Nc3ccccc3OC)n2)cc1N ZINC000217695034 EI In-Stock Unstable CCR4 0 45 COC(=O)[C@H](O)CNC(=O)c1ccc([N+](=O)[O-])cc1 ZINC000217695042 CB On-Demand Unstable CA2 18 42 COC(=O)[C@H](O)CNC(=O)c1ccc([N+](=O)[O-])cc1 ZINC000217695042 CB On-Demand Unstable CACNA1D 60 33 COC(=O)[C@H](O)CNC(=O)c1ccc([N+](=O)[O-])cc1 ZINC000217695042 CB On-Demand Unstable CCR3 0 41 Cc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217695096 GG For-Sale Unstable DRD4 21 49 Cc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217695096 GG For-Sale Unstable NOS2 56 33 Cc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217695096 GG For-Sale Unstable MCHR1 29 50 CC(=O)NCCOc1ccc(C(=O)N(C)CCc2ccncc2)cc1 ZINC000217695107 ED In-Stock Unstable MTNR1A 35 42 CC(=O)NCCOc1ccc(C(=O)N(C)CCc2ccncc2)cc1 ZINC000217695107 ED In-Stock Unstable MTNR1B 35 42 O=C(O)/C=C\c1ccc(C(=O)Nc2ccc(Cl)c(F)c2)s1 ZINC000217695111 EH For-Sale Anodyne MAOB 16 42 O=C(O)/C=C\c1ccc(C(=O)Nc2ccc(Cl)c(F)c2)s1 ZINC000217695111 EH For-Sale Anodyne ENV 47 37 CCOc1cc(CN[C@@H]2CCN3CCC[C@@H]23)ccc1OC ZINC000217695118 CE For-Sale Unstable SSTR5 65 44 COc1ccc(-c2nnc(Cc3ccc(N)cc3)o2)cc1 ZINC000217695122 CF In-Stock Unstable APP 15 43 COC(=O)[C@@H](O)CNC(=O)c1cccc(OC)c1OC ZINC000217695139 CB On-Demand Unstable DRD2 18 40 COC(=O)[C@@H](O)CNC(=O)c1cccc(OC)c1OC ZINC000217695139 CB On-Demand Unstable KCNA3 35 48 COC(=O)[C@@H](O)CNC(=O)c1cccc(OC)c1OC ZINC000217695139 CB On-Demand Unstable KCNK3 45 40 COC(=O)[C@@H](O)CNC(=O)c1cccc(OC)c1OC ZINC000217695139 CB On-Demand Unstable KCNK9 34 40 CCOc1cc(CN[C@H]2CCN3CCC[C@@H]23)ccc1OC ZINC000217695195 CE For-Sale Unstable SSTR5 65 44 O=C(O)/C=C\c1ccc(C(=O)N2CCCSCC2)cc1 ZINC000217695199 CE For-Sale Unstable MLYCD 17 40 O=C(O)/C=C\c1ccc(C(=O)N2CCCSCC2)cc1 ZINC000217695199 CE For-Sale Unstable L3MBTL3 49 37 CCOC(=O)N1CCN(C(=O)N/C=C/c2ccccc2C)CC1 ZINC000217695215 DE For-Sale Unstable P2RY12 48 38 COC(=O)[C@H](O)CNC(=O)c1cccc(OC)c1OC ZINC000217695220 CB On-Demand Unstable DRD2 18 40 COC(=O)[C@H](O)CNC(=O)c1cccc(OC)c1OC ZINC000217695220 CB On-Demand Unstable KCNA3 35 48 COC(=O)[C@H](O)CNC(=O)c1cccc(OC)c1OC ZINC000217695220 CB On-Demand Unstable KCNK3 45 40 COC(=O)[C@H](O)CNC(=O)c1cccc(OC)c1OC ZINC000217695220 CB On-Demand Unstable KCNK9 34 40 Cn1c(=O)oc2ccc(S(=O)(=O)N3CCc4oncc4C3)cc21 ZINC000217695223 EC In-Stock Unstable AKR1C3 54 34 CCCOc1ccc(CN[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217695302 CF For-Sale Unstable HRH3 33 45 COC(=O)Nc1ccc(S(=O)(=O)N2CCc3oncc3C2)cc1 ZINC000217695327 ED In-Stock Unstable TGM2 62 37 COC(=O)Nc1ccc(S(=O)(=O)N2CCc3oncc3C2)cc1 ZINC000217695327 ED In-Stock Unstable F13A1 90 40 COC(=O)Nc1ccc(S(=O)(=O)N2CCc3oncc3C2)cc1 ZINC000217695327 ED In-Stock Unstable AKR1C3 56 37 COC(=O)[C@@H](O)CNC(=O)c1ccc(NC(C)=O)cc1 ZINC000217695330 CB On-Demand Unstable PRSS1 17 40 COC(=O)[C@@H](O)CNC(=O)c1ccc(NC(C)=O)cc1 ZINC000217695330 CB On-Demand Unstable PRNP 49 37 COC(=O)[C@@H](O)CNC(=O)c1ccc(NC(C)=O)cc1 ZINC000217695330 CB On-Demand Unstable F3 76 38 COC(=O)[C@@H](O)CNC(=O)c1ccc(NC(C)=O)cc1 ZINC000217695330 CB On-Demand Unstable ACR 55 40 COc1ccc(CCN2C(=O)N[C@@H](CC(=O)N3CCCC3)C2=O)cc1OC ZINC000217695339 GD In-Stock Unstable FKBP1A 41 42 COc1ccc(OC)c(CN[C@@H]2CCN3CCCC[C@@H]23)c1 ZINC000217695359 CE On-Demand Unstable TACR1 36 52 CCCOc1ccc(CN[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217695385 CF For-Sale Unstable HRH3 33 45 CCc1ccc(/C=C\C(=O)NC[C@](C)(O)CC(=O)O)cc1 ZINC000217695410 CD For-Sale Unstable HDAC8 15 40 COC(=O)[C@H](O)CNC(=O)c1ccc(NC(C)=O)cc1 ZINC000217695420 CB On-Demand Unstable PRSS1 17 40 COC(=O)[C@H](O)CNC(=O)c1ccc(NC(C)=O)cc1 ZINC000217695420 CB On-Demand Unstable PRNP 49 37 COC(=O)[C@H](O)CNC(=O)c1ccc(NC(C)=O)cc1 ZINC000217695420 CB On-Demand Unstable F3 76 38 COC(=O)[C@H](O)CNC(=O)c1ccc(NC(C)=O)cc1 ZINC000217695420 CB On-Demand Unstable ACR 55 40 COc1ccc(OC)c(CN[C@H]2CCN3CCCC[C@@H]23)c1 ZINC000217695438 CE On-Demand Unstable TACR1 36 52 O=C1CCc2cc(S(=O)(=O)N3CCc4oncc4C3)cc3c2N1CC3 ZINC000217695445 FD In-Stock Unstable CYP11B1 27 43 O=C1CCc2cc(S(=O)(=O)N3CCc4oncc4C3)cc3c2N1CC3 ZINC000217695445 FD In-Stock Unstable CYP11B2 26 44 O=C1CCc2cc(S(=O)(=O)N3CCc4oncc4C3)cc3c2N1CC3 ZINC000217695445 FD In-Stock Unstable AKR1C3 50 38 O=C(O)COc1ccc(S(=O)(=O)N2CCCC2)c2cccnc12 ZINC000217695447 ED In-Stock Unstable PTGDR2 24 40 Cc1ccc(/C=C\C(=O)O)cc1S(=O)(=O)Nc1nccs1 ZINC000217695468 DE For-Sale Unstable SCN9A 0 40 CCc1ccc(/C=C\C(=O)NC[C@@](C)(O)CC(=O)O)cc1 ZINC000217695496 CD For-Sale Unstable HDAC8 15 40 Cc1ccccc1/C=C/NC(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217695538 DJ For-Sale Unstable TRPV1 15 46 Cc1ccccc1/C=C/NC(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217695538 DJ For-Sale Unstable EPHX2 27 41 Cc1ccccc1/C=C/NC(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217695538 DJ For-Sale Unstable FPR2 19 43 CN(C)S(=O)(=O)c1ccc(OCC(=O)O)c2ncccc12 ZINC000217695558 DC In-Stock Unstable PTGDR2 31 41 COC(=O)C[C@H](c1cccnc1)c1oc(CN2CCCCC2)cc(=O)c1O ZINC000217695586 FE In-Stock Unstable KCNA5 44 40 Cc1ccccc1/C=C/NC(=O)Nc1ccc(F)cc1F ZINC000217695644 CI For-Sale Unstable SOAT1 38 44 O=C(O)/C=C\c1cccc(S(=O)(=O)N2CCOCC2)c1 ZINC000217695654 CC For-Sale Unstable LPL 20 41 O=C(O)/C=C\c1cccc(S(=O)(=O)N2CCOCC2)c1 ZINC000217695654 CC For-Sale Unstable PKM 39 41 O=C(O)/C=C\c1cccc(S(=O)(=O)N2CCOCC2)c1 ZINC000217695654 CC For-Sale Unstable AKR1C3 66 42 COC(=O)C[C@@H](c1cccnc1)c1oc(CN2CCCCC2)cc(=O)c1O ZINC000217695666 FE In-Stock Unstable KCNA5 44 40 Cc1cc(S(=O)(=O)NCC(C)C)ccc1/C=C\C(=O)O ZINC000217695718 CE For-Sale Unstable LEF 56 37 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC)cc1 ZINC000217695748 CB On-Demand Unstable CA2 17 57 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC)cc1 ZINC000217695748 CB On-Demand Unstable DRD4 40 32 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC)cc1 ZINC000217695748 CB On-Demand Unstable NQO2 15 40 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC)cc1 ZINC000217695748 CB On-Demand Unstable TRPV1 0 41 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC)cc1 ZINC000217695748 CB On-Demand Unstable MMP13 24 40 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC)cc1 ZINC000217695748 CB On-Demand Unstable CYP2D6 0 46 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC)cc1 ZINC000217695748 CB On-Demand Unstable ACR 48 33 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC)cc1 ZINC000217695748 CB On-Demand Unstable ITGAV 46 37 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC)cc1 ZINC000217695748 CB On-Demand Unstable MT-ND1 24 40 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC)cc1 ZINC000217695748 CB On-Demand Unstable MMP1 28 40 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC)cc1 ZINC000217695748 CB On-Demand Unstable AOC3 26 44 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC)cc1 ZINC000217695748 CB On-Demand Unstable CYP27B1 28 45 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC)cc1 ZINC000217695748 CB On-Demand Unstable H9B8T9_CAPHI 18 60 Cc1ccccc1C(=O)N1CCC(S(=O)(=O)c2nccn2C)CC1 ZINC000217695754 ED In-Stock Unstable CCR8 58 34 C[C@](O)(CNC(=O)/C=C\c1cc(Cl)ccc1Cl)CC(=O)O ZINC000217695776 EE For-Sale Unstable PYGL 0 42 C[C@](O)(CNC(=O)/C=C\c1cc(Cl)ccc1Cl)CC(=O)O ZINC000217695776 EE For-Sale Unstable BOTA 23 42 CC(=O)Nc1ccc(OCC(=O)O)c2ncccc12 ZINC000217695781 CD In-Stock Unstable PTGDR2 28 41 COC(=O)[C@H](O)CNC(=O)c1ccc(OC)cc1 ZINC000217695836 CB On-Demand Unstable CA2 17 57 COC(=O)[C@H](O)CNC(=O)c1ccc(OC)cc1 ZINC000217695836 CB On-Demand Unstable DRD4 40 32 COC(=O)[C@H](O)CNC(=O)c1ccc(OC)cc1 ZINC000217695836 CB On-Demand Unstable NQO2 15 40 COC(=O)[C@H](O)CNC(=O)c1ccc(OC)cc1 ZINC000217695836 CB On-Demand Unstable TRPV1 0 41 COC(=O)[C@H](O)CNC(=O)c1ccc(OC)cc1 ZINC000217695836 CB On-Demand Unstable MMP13 24 40 COC(=O)[C@H](O)CNC(=O)c1ccc(OC)cc1 ZINC000217695836 CB On-Demand Unstable CYP2D6 0 46 COC(=O)[C@H](O)CNC(=O)c1ccc(OC)cc1 ZINC000217695836 CB On-Demand Unstable ACR 48 33 COC(=O)[C@H](O)CNC(=O)c1ccc(OC)cc1 ZINC000217695836 CB On-Demand Unstable ITGAV 46 37 COC(=O)[C@H](O)CNC(=O)c1ccc(OC)cc1 ZINC000217695836 CB On-Demand Unstable MT-ND1 24 40 COC(=O)[C@H](O)CNC(=O)c1ccc(OC)cc1 ZINC000217695836 CB On-Demand Unstable MMP1 28 40 COC(=O)[C@H](O)CNC(=O)c1ccc(OC)cc1 ZINC000217695836 CB On-Demand Unstable AOC3 26 44 COC(=O)[C@H](O)CNC(=O)c1ccc(OC)cc1 ZINC000217695836 CB On-Demand Unstable CYP27B1 28 45 COC(=O)[C@H](O)CNC(=O)c1ccc(OC)cc1 ZINC000217695836 CB On-Demand Unstable H9B8T9_CAPHI 18 60 COc1ccc(F)cc1-c1ccnc2[nH]c(C3=CCN(C(=O)CC(=O)O)CC3)cc12 ZINC000217695841 HG For-Sale Unstable CSNK1G2 45 31 C[C@@](O)(CNC(=O)/C=C\c1cc(Cl)ccc1Cl)CC(=O)O ZINC000217695855 EE For-Sale Unstable PYGL 0 42 C[C@@](O)(CNC(=O)/C=C\c1cc(Cl)ccc1Cl)CC(=O)O ZINC000217695855 EE For-Sale Unstable BOTA 23 42 Cc1ccccc1/C=C/NC(=O)N1CCCC[C@@H]1CCO ZINC000217695868 CF For-Sale Unstable SLC6A1 40 34 Cn1cc(C(=O)N2CCC(Oc3cccc(F)c3)CC2)c(=O)[nH]c1=O ZINC000217695873 EC In-Stock Unstable HRH1 18 40 Cn1cc(C(=O)N2CCC(Oc3cccc(F)c3)CC2)c(=O)[nH]c1=O ZINC000217695873 EC In-Stock Unstable PRSS2 53 30 Cn1cc(C(=O)N2CCC(Oc3cccc(F)c3)CC2)c(=O)[nH]c1=O ZINC000217695873 EC In-Stock Unstable HRH3 0 43 Cn1cc(C(=O)N2CCC(Oc3cccc(F)c3)CC2)c(=O)[nH]c1=O ZINC000217695873 EC In-Stock Unstable CCR3 19 40 Cn1cc(C(=O)N2CCC(Oc3cccc(F)c3)CC2)c(=O)[nH]c1=O ZINC000217695873 EC In-Stock Unstable MLNR 25 45 O=C(O)/C=C\c1ccc(S(=O)(=O)NC2CCCC2)c(Cl)c1 ZINC000217695880 EF For-Sale Unstable CCR8 37 41 O=C(O)/C=C\c1ccc(S(=O)(=O)NC2CCCC2)c(Cl)c1 ZINC000217695880 EF For-Sale Unstable SFRP1 114 36 O=C(O)/C=C\c1ccc(S(=O)(=O)NC2CCCC2)c(Cl)c1 ZINC000217695880 EF For-Sale Unstable WNT3 76 36 CCNc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O ZINC000217695892 DC In-Stock Unstable CASP3 17 45 CCNc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O ZINC000217695892 DC In-Stock Unstable BDKRB1 0 43 COCc1cc(=O)c(O)c([C@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccc(O)c(OC)c2)o1 ZINC000217695901 KH In-Stock Unstable RORC 49 34 Cc1ccccc1/C=C/NC(=O)N1CCCC[C@H]1CCO ZINC000217695947 CF For-Sale Unstable SLC6A1 40 34 Cc1cc(S(=O)(=O)N2CCCCC2)ccc1/C=C\C(=O)O ZINC000217695966 DE For-Sale Unstable LPL 48 39 Cc1cc(S(=O)(=O)N2CCCCC2)ccc1/C=C\C(=O)O ZINC000217695966 DE For-Sale Unstable CASP3 0 41 Cc1cc(S(=O)(=O)N2CCCCC2)ccc1/C=C\C(=O)O ZINC000217695966 DE For-Sale Unstable F13A1 38 40 Cc1cc(S(=O)(=O)N2CCCCC2)ccc1/C=C\C(=O)O ZINC000217695966 DE For-Sale Unstable AKR1C3 50 39 CC(F)(F)CS(=O)(=O)c1cccc(C#N)c1 ZINC000217695973 BD For-Sale Unstable NR1H2 16 44 COCc1cc(=O)c(O)c([C@@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccc(O)c(OC)c2)o1 ZINC000217695990 KH In-Stock Unstable RORC 49 34 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NC(C)C ZINC000217696007 CD In-Stock Unstable NEU3 0 41 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NC(C)C ZINC000217696007 CD In-Stock Unstable ITGAV 41 37 CCOCCCNS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217696060 DD For-Sale Unstable AKR1C3 25 42 CCCCOc1ccc(CN[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217696113 CG For-Sale Unstable LTA4H 26 40 CCCCOc1ccc(CN[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217696113 CG For-Sale Unstable HRH3 50 48 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NCC(C)C ZINC000217696118 DD In-Stock Unstable NEU3 0 40 CC(C)=CCC/C(C)=C/CC/C(C)=C\CC/C(C)=C/CBr ZINC000217696137 FK For-Sale Unstable GGPS1 51 48 CC(C)=CCC/C(C)=C/CC/C(C)=C\CC/C(C)=C/CBr ZINC000217696137 FK For-Sale Unstable FDFT1 41 53 CC(C)=CCC/C(C)=C/CC/C(C)=C\CC/C(C)=C/CBr ZINC000217696137 FK For-Sale Unstable LSS 37 40 CC(C)=CCC/C(C)=C/CC/C(C)=C\CC/C(C)=C/CBr ZINC000217696137 FK For-Sale Unstable TRPA1 17 40 Fc1ccccc1CN[C@@H]1CCN2CCCC[C@@H]12 ZINC000217696158 BF On-Demand Unstable VACHT_TETCF 0 44 Fc1ccccc1CN[C@@H]1CCN2CCCC[C@@H]12 ZINC000217696158 BF On-Demand Unstable SLC18A3 51 37 CCCCOc1ccc(CN[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217696192 CG For-Sale Unstable LTA4H 26 40 CCCCOc1ccc(CN[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217696192 CG For-Sale Unstable HRH3 50 48 Cc1ccccc1/C=C/NC(=O)N1CCN(c2ccccn2)CC1 ZINC000217696200 DF For-Sale Unstable DRD4 28 40 Cc1ccccc1/C=C/NC(=O)N1CCN(c2ccccn2)CC1 ZINC000217696200 DF For-Sale Unstable EBP 24 43 Cn1ccnc1S(=O)(=O)C1CCN(C(=O)c2ccc(F)cc2Cl)CC1 ZINC000217696224 GE In-Stock Unstable P2RX7 26 55 CCNc1ccc(S(=O)(=O)NCCO)cc1C(=O)O ZINC000217696262 CC In-Stock Unstable CASP3 16 40 Fc1ccccc1CN[C@H]1CCN2CCCC[C@@H]12 ZINC000217696267 BF On-Demand Unstable VACHT_TETCF 0 44 Fc1ccccc1CN[C@H]1CCN2CCCC[C@@H]12 ZINC000217696267 BF On-Demand Unstable SLC18A3 51 37 CCOc1ccc(CN[C@@H]2CCN3CCC[C@@H]23)cc1OC ZINC000217696292 CE For-Sale Unstable SSTR5 60 40 CCOc1ccc(CN[C@H]2CCN3CCC[C@@H]23)cc1OC ZINC000217696380 CE For-Sale Unstable SSTR5 60 40 O=C(O)c1cc(O)n(-c2cc(C(F)(F)F)ccc2Cl)n1 ZINC000217696399 DF In-Stock Anodyne RPA1 77 42 O=C(O)/C=C\c1ccc(C(=O)NCc2cccc(F)c2)s1 ZINC000217696411 DF For-Sale Unstable HCAR2 0 43 Cn1ccnc1S(=O)(=O)C1CCN(C(=O)c2ccc(OC(F)(F)F)cc2)CC1 ZINC000217696463 HE In-Stock Unstable SLC9A1 26 41 Cn1ccnc1S(=O)(=O)C1CCN(C(=O)c2ccc(OC(F)(F)F)cc2)CC1 ZINC000217696463 HE In-Stock Unstable EPHX2 47 51 Cn1ccnc1S(=O)(=O)C1CCN(C(=O)c2ccc(OC(F)(F)F)cc2)CC1 ZINC000217696463 HE In-Stock Unstable L3MBTL3 53 35 Cn1ccnc1S(=O)(=O)C1CCN(C(=O)c2ccc(OC(F)(F)F)cc2)CC1 ZINC000217696463 HE In-Stock Unstable SLC6A7 0 46 Cc1oncc1C(=O)NC1CCN(C(=O)N2CCOCC2)CC1 ZINC000217696475 DC In-Stock Unstable CCR8 17 40 COC(=O)c1ccc(NC(=O)CCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@H]23)cc1 ZINC000217696478 JH In-Stock Unstable ACR 42 36 CCNc1ccc(S(=O)(=O)NCCC(C)C)cc1C(=O)O ZINC000217696520 DE In-Stock Unstable CASP3 16 44 CCNc1ccc(S(=O)(=O)NCCC(C)C)cc1C(=O)O ZINC000217696520 DE In-Stock Unstable BDKRB1 0 42 C[C@](O)(CNC(=O)/C=C\c1ccc(F)cc1)CC(=O)O ZINC000217696545 CD For-Sale Unstable MMP2 15 46 COC(=O)c1ccc(NC(=O)CCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@@H]23)cc1 ZINC000217696566 JH In-Stock Unstable ACR 42 36 COc1c(N)cc(S(C)(=O)=O)cc1C(=O)O ZINC000217696614 BC For-Sale Unstable MT-CO2 34 43 CNc1ccc(S(=O)(=O)NCCC(C)C)cc1C(=O)O ZINC000217696634 DD In-Stock Unstable CASP3 17 43 C[C@@](O)(CNC(=O)/C=C\c1ccc(F)cc1)CC(=O)O ZINC000217696636 CD For-Sale Unstable MMP2 15 46 COC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2C)c1 ZINC000217696766 DH For-Sale Unstable KCNK3 105 40 COC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2C)c1 ZINC000217696766 DH For-Sale Unstable KCNK9 66 38 Cn1ccnc1S(=O)(=O)C1CCN(C(=O)c2cc(-c3ccc(F)cc3)c[nH]2)CC1 ZINC000217696799 HF In-Stock Unstable HTR2B 18 41 O=C(O)/C=C\c1cccc(C(=O)NC2CCCCC2)c1 ZINC000217696811 CF For-Sale Unstable CNR1 17 40 O=C(O)/C=C\c1cccc(C(=O)NC2CCCCC2)c1 ZINC000217696811 CF For-Sale Unstable CNR2 22 42 O=C(O)/C=C\c1cccc(C(=O)NC2CCCCC2)c1 ZINC000217696811 CF For-Sale Unstable HDAC8 16 45 O=C(O)/C=C\c1cccc(C(=O)NC2CCCCC2)c1 ZINC000217696811 CF For-Sale Unstable FAAH 17 45 O=C(O)/C=C\c1cccc(C(=O)NC2CCCCC2)c1 ZINC000217696811 CF For-Sale Unstable EPHX2 18 41 O=C(O)/C=C\c1ccc(F)c(C(=O)NC2CCCCC2)c1 ZINC000217696886 CF For-Sale Unstable CNR1 23 45 O=C(O)/C=C\c1ccc(F)c(C(=O)NC2CCCCC2)c1 ZINC000217696886 CF For-Sale Unstable CNR2 29 45 CC(C)Cc1cc(C(=O)N[C@H](CO)C(C)C)c2ccccc2n1 ZINC000217696897 DG In-Stock Unstable TACR2 0 44 CC(C)Cc1cc(C(=O)N[C@H](CO)C(C)C)c2ccccc2n1 ZINC000217696897 DG In-Stock Unstable CCR1 23 41 CC(C)Cc1cc(C(=O)N[C@H](CO)C(C)C)c2ccccc2n1 ZINC000217696897 DG In-Stock Unstable TACR3 39 41 CCCCS[C@@H](C(=O)OCC)c1ccccc1 ZINC000217696948 CH For-Sale Unstable SOAT1 52 36 COC(=O)[C@@H](O)CNC(=O)c1ccccc1OC(F)F ZINC000217696950 CC On-Demand Unstable KCNA3 34 47 COC(=O)[C@@H](O)CNC(=O)c1ccccc1OC(F)F ZINC000217696950 CC On-Demand Unstable HCN1 62 36 COC(=O)[C@@H](O)CNC(=O)c1ccccc1OC(F)F ZINC000217696950 CC On-Demand Unstable HCN4 49 34 COC(=O)[C@@H](O)CNC(=O)c1ccccc1OC(F)F ZINC000217696950 CC On-Demand Unstable KCNK3 55 37 COC(=O)[C@@H](O)CNC(=O)c1ccccc1OC(F)F ZINC000217696950 CC On-Demand Unstable KCNK9 47 37 CCCCS[C@H](C(=O)OCC)c1ccccc1 ZINC000217697035 CH For-Sale Unstable SOAT1 52 36 COC(=O)[C@H](O)CNC(=O)c1ccccc1OC(F)F ZINC000217697041 CC On-Demand Unstable KCNA3 34 47 COC(=O)[C@H](O)CNC(=O)c1ccccc1OC(F)F ZINC000217697041 CC On-Demand Unstable HCN1 62 36 COC(=O)[C@H](O)CNC(=O)c1ccccc1OC(F)F ZINC000217697041 CC On-Demand Unstable HCN4 49 34 COC(=O)[C@H](O)CNC(=O)c1ccccc1OC(F)F ZINC000217697041 CC On-Demand Unstable KCNK3 55 37 COC(=O)[C@H](O)CNC(=O)c1ccccc1OC(F)F ZINC000217697041 CC On-Demand Unstable KCNK9 47 37 CC[C@@H](Nc1ccc(S(=O)(=O)CC)cc1Br)c1ccccc1 ZINC000217697062 GJ For-Sale Unstable CXCR2 15 40 CC[C@@H](Nc1ccc(S(=O)(=O)CC)cc1Br)c1ccccc1 ZINC000217697062 GJ For-Sale Unstable CA5B 16 40 CC[C@@H](Nc1ccc(S(=O)(=O)CC)cc1Br)c1ccccc1 ZINC000217697062 GJ For-Sale Unstable CA5A 18 40 CCC(CC)(CNCc1cccc(F)c1)NC(=O)OC(C)(C)C ZINC000217697074 DH On-Demand Unstable PAPA1_CARPA 21 45 CCCCc1ccc(-n2nc(C(=O)O)cc2O)cc1 ZINC000217697086 CF In-Stock Unstable INHA 82 35 CCCCc1ccc(-n2nc(C(=O)O)cc2O)cc1 ZINC000217697086 CF In-Stock Unstable AGTR1B 46 36 CCCCc1ccc(-n2nc(C(=O)O)cc2O)cc1 ZINC000217697086 CF In-Stock Unstable RPA1 88 38 COc1ccc(-n2nc(C(=O)O)cc2O)cc1OC ZINC000217697222 CD In-Stock Unstable ALS 40 34 COc1ccc(-n2nc(C(=O)O)cc2O)cc1OC ZINC000217697222 CD In-Stock Unstable RPA1 87 50 N[C@H]1CNC[C@H](Cc2ccccc2)C1 ZINC000217697317 AD For-Sale Unstable SLC18A2 23 41 CNc1ccc(C(=O)O)cc1S(=O)(=O)NCC(C)C ZINC000217697332 CD In-Stock Unstable NEU3 0 40 Cc1ccccc1/C=C/NC(=O)NCc1ccccc1Br ZINC000217697374 EI For-Sale Unstable ANPEP 15 48 CSC[C@@](C)(O)CNC(=O)[C@@H]1CCCN1C(=O)C(C)(C)C ZINC000217697376 DD On-Demand Unstable TPP2 41 41 N[C@H]1CNC[C@@H](Cc2ccccc2)C1 ZINC000217697406 AD For-Sale Unstable SLC18A2 23 41 CNc1ccc(C(=O)O)cc1S(=O)(=O)NC1CC1 ZINC000217697435 CC In-Stock Unstable CCR8 85 42 CNc1ccc(C(=O)O)cc1S(=O)(=O)NC1CC1 ZINC000217697435 CC In-Stock Unstable SFRP1 108 40 CNc1ccc(C(=O)O)cc1S(=O)(=O)NC1CC1 ZINC000217697435 CC In-Stock Unstable WNT3 82 38 CSC[C@](C)(O)CNC(=O)[C@@H]1CCCN1C(=O)C(C)(C)C ZINC000217697455 DD On-Demand Unstable TPP2 41 41 Cc1cccc(CNC(=O)N/C=C/c2ccccc2C)c1 ZINC000217697474 CH For-Sale Unstable ANPEP 20 48 C[C@@H]1CCC[C@@H](N[C@H](C)C(N)=O)C1 ZINC000217697475 AD On-Demand Unstable XPNPEP1 59 35 C[C@@H]1CCC[C@@H](N[C@H](C)C(N)=O)C1 ZINC000217697475 AD On-Demand Unstable XPNPEP2 56 35 CSC[C@@](C)(O)CNC(=O)[C@H]1CCCN1C(=O)C(C)(C)C ZINC000217697534 DD On-Demand Unstable TPP2 41 41 Cn1ccnc1S(=O)(=O)C1CCN(S(=O)(=O)c2cccc3ccccc23)CC1 ZINC000217697536 HE In-Stock Unstable NPY2R 29 44 Cn1ccnc1S(=O)(=O)C1CCN(S(=O)(=O)c2cccc3ccccc23)CC1 ZINC000217697536 HE In-Stock Unstable HTR6 25 44 COC(=O)[C@@H](O)CNC(=O)Cc1ccc(C)c(OC)c1 ZINC000217697543 CC On-Demand Unstable TRPV1 26 48 COC(=O)[C@@H](O)CNC(=O)Cc1ccc(C)c(OC)c1 ZINC000217697543 CC On-Demand Unstable NCE103 26 44 O=C(O)c1cc(O)n(-c2ccc(Cl)cc2C(F)(F)F)n1 ZINC000217697558 DF In-Stock Anodyne RPA1 65 48 C[C@@H]1CCC[C@H](N[C@H](C)C(N)=O)C1 ZINC000217697567 AD On-Demand Unstable XPNPEP1 59 35 C[C@@H]1CCC[C@H](N[C@H](C)C(N)=O)C1 ZINC000217697567 AD On-Demand Unstable XPNPEP2 56 35 COc1cccc(CNC(=O)N/C=C/c2ccccc2C)c1 ZINC000217697582 CG For-Sale Unstable DRD4 41 32 COc1cccc(CNC(=O)N/C=C/c2ccccc2C)c1 ZINC000217697582 CG For-Sale Unstable ROCK1 38 44 COc1cccc(CNC(=O)N/C=C/c2ccccc2C)c1 ZINC000217697582 CG For-Sale Unstable MTNR1A 51 47 COc1cccc(CNC(=O)N/C=C/c2ccccc2C)c1 ZINC000217697582 CG For-Sale Unstable MTNR1B 50 47 COc1cccc(CNC(=O)N/C=C/c2ccccc2C)c1 ZINC000217697582 CG For-Sale Unstable ROCK2 47 48 COc1cccc(CNC(=O)N/C=C/c2ccccc2C)c1 ZINC000217697582 CG For-Sale Unstable PDS 47 41 CSC[C@](C)(O)CNC(=O)[C@H]1CCCN1C(=O)C(C)(C)C ZINC000217697619 DD On-Demand Unstable TPP2 41 41 COC(=O)[C@H](O)CNC(=O)Cc1ccc(C)c(OC)c1 ZINC000217697629 CC On-Demand Unstable TRPV1 26 48 COC(=O)[C@H](O)CNC(=O)Cc1ccc(C)c(OC)c1 ZINC000217697629 CC On-Demand Unstable NCE103 26 44 Cn1ccnc1S(=O)(=O)C1CCN(S(=O)(=O)c2ccc(F)c(Cl)c2)CC1 ZINC000217697651 HD In-Stock Unstable PKM 35 42 C[C@H]1CCC[C@H](C)C1N[C@H](C)C(N)=O ZINC000217697677 AD For-Sale Unstable XPNPEP1 59 35 C[C@H]1CCC[C@H](C)C1N[C@H](C)C(N)=O ZINC000217697677 AD For-Sale Unstable XPNPEP2 56 35 COC(=O)[C@@H](O)CNC(=O)[C@@H]1CCCN(C(=O)C2CC2)C1 ZINC000217697740 CB On-Demand Unstable F2R 25 47 C[C@H]1CCC[C@@H](C)C1N[C@H](C)C(N)=O ZINC000217697750 AD For-Sale Unstable XPNPEP1 59 35 C[C@H]1CCC[C@@H](C)C1N[C@H](C)C(N)=O ZINC000217697750 AD For-Sale Unstable XPNPEP2 56 35 Cn1ccnc1S(=O)(=O)C1CCN(S(=O)(=O)c2ccc3c(c2)OCCO3)CC1 ZINC000217697766 IC In-Stock Unstable PKM 52 59 CCCCOc1ccc(CN2C[C@@H]3CC[C@H](C2)[C@@H]3O)cc1 ZINC000217697774 CG In-Stock Unstable LTA4H 35 40 CCCCOc1ccc(CN2C[C@@H]3CC[C@H](C2)[C@@H]3O)cc1 ZINC000217697774 CG In-Stock Unstable HRH3 35 48 CCCCOc1ccc(CN2C[C@@H]3CC[C@H](C2)[C@@H]3O)cc1 ZINC000217697774 CG In-Stock Unstable PLA2G4B 61 37 Cc1ccccc1/C=C/NC(=O)NCc1cccc(Cl)c1 ZINC000217697841 DI For-Sale Unstable PDS 45 32 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1N[C@@H](C)C(N)=O ZINC000217697859 BD For-Sale Unstable TRPM8 0 52 CCOc1ccc(S(=O)(=O)N2CCC(S(=O)(=O)c3nccn3C)CC2)cc1C ZINC000217697872 ID In-Stock Unstable PDE5A 33 43 CCC[C@@H](C)NS(=O)(=O)c1ccc(NCC)c(C(=O)O)c1 ZINC000217697878 DE In-Stock Unstable LEF 48 35 COC(=O)[C@@H](O)CNC(=O)[C@H]1CCCN(C(=O)C2CC2)C1 ZINC000217697910 CB On-Demand Unstable F2R 25 47 CSC[C@@](C)(O)CNC(=O)Cn1cncn1 ZINC000217697916 BB For-Sale Unstable HIS3 53 32 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1N[C@@H](C)C(N)=O ZINC000217697929 BD For-Sale Unstable TRPM8 0 52 CCC[C@H](C)NS(=O)(=O)c1ccc(NCC)c(C(=O)O)c1 ZINC000217697954 DE In-Stock Unstable LEF 48 35 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1N[C@@H](C)C(N)=O ZINC000217698010 BD For-Sale Unstable TRPM8 0 52 CSC[C@](C)(O)CNC(=O)Cn1cncn1 ZINC000217698013 BB For-Sale Unstable HIS3 53 32 Cc1cc(NC(=O)c2cccc(/C=C\C(=O)O)c2)no1 ZINC000217698017 CE For-Sale Unstable HDAC8 33 45 Cc1cc(NC(=O)c2cccc(/C=C\C(=O)O)c2)no1 ZINC000217698017 CE For-Sale Unstable HDAC6 15 45 Cc1cc(NC(=O)c2cccc(/C=C\C(=O)O)c2)no1 ZINC000217698017 CE For-Sale Unstable KCNK3 86 39 Cc1cc(NC(=O)c2cccc(/C=C\C(=O)O)c2)no1 ZINC000217698017 CE For-Sale Unstable KCNK9 43 39 CCC(CC)(CNCc1ccc(F)cc1)NC(=O)OC(C)(C)C ZINC000217698061 DH On-Demand Unstable PAPA1_CARPA 20 41 CCc1ccccc1-n1nc(C(=O)O)cc1O ZINC000217698070 BD In-Stock Unstable RPA1 71 41 Cc1ccccc1/C=C/NC(=O)NCCc1ccccc1C ZINC000217698076 CH For-Sale Unstable MTNR1A 25 45 CC(C)[C@H]1CC[C@H](C)C[C@@H]1N[C@@H](C)C(N)=O ZINC000217698096 BD For-Sale Unstable TRPM8 0 52 COc1ccc(CCN2C(=O)N[C@@H](CCC(=O)N[C@H](CO)c3ccccc3)C2=O)cc1 ZINC000217698101 ID In-Stock Unstable GPR88 0 45 Cc1n[nH]c(C)c1CCNC(=O)[C@@]1(c2ccccc2)CC12CCCC2 ZINC000217698179 EH In-Stock Unstable HAO2 58 35 CCN(CCO)C(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217698194 CD For-Sale Unstable ACKR3 44 33 CNc1ccc(C(=O)O)cc1S(=O)(=O)NC(C)(C)C ZINC000217698200 CD In-Stock Unstable NEU3 0 41 COc1ccccc1CCNC(=O)N/C=C/c1ccccc1C ZINC000217698204 DH For-Sale Unstable MTNR1A 34 43 COc1ccccc1CCNC(=O)N/C=C/c1ccccc1C ZINC000217698204 DH For-Sale Unstable MTNR1B 25 43 COc1ccc(CCN2C(=O)N[C@@H](CCC(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)C2=O)cc1OC ZINC000217698232 KD In-Stock Unstable CHRNA4 27 45 Cc1n[nH]c(C)c1CCNC(=O)[C@]1(c2ccccc2)CC12CCCC2 ZINC000217698279 EH In-Stock Unstable HAO2 58 35 CNc1ccc(S(=O)(=O)NCCC2=CCCCC2)cc1C(=O)O ZINC000217698303 EF In-Stock Unstable TBXA2R 49 37 COC(=O)Nc1ccc(S(=O)(=O)N2CCC(S(=O)(=O)c3nccn3C)CC2)cc1 ZINC000217698313 ID In-Stock Unstable EPHX2 26 46 COC(=O)Nc1ccc(S(=O)(=O)N2CCC(S(=O)(=O)c3nccn3C)CC2)cc1 ZINC000217698313 ID In-Stock Unstable TGM2 79 44 COC(=O)Nc1ccc(S(=O)(=O)N2CCC(S(=O)(=O)c3nccn3C)CC2)cc1 ZINC000217698313 ID In-Stock Unstable F13A1 96 42 COC(=O)Nc1ccc(S(=O)(=O)N2CCC(S(=O)(=O)c3nccn3C)CC2)cc1 ZINC000217698313 ID In-Stock Unstable NAMPT 37 41 COC(=O)Nc1ccc(S(=O)(=O)N2CCC(S(=O)(=O)c3nccn3C)CC2)cc1 ZINC000217698313 ID In-Stock Unstable TGM6 0 44 COC(=O)[C@@H](O)CNC(=O)c1cccc(C)c1[N+](=O)[O-] ZINC000217698336 CC On-Demand Unstable CACNA1D 62 33 CCCCN(C(=O)c1ccc(/C=C\C(=O)O)cc1)C1CC1 ZINC000217698353 CG For-Sale Unstable PLM2_PLAFA 40 34 CCCCN(C(=O)c1ccc(/C=C\C(=O)O)cc1)C1CC1 ZINC000217698353 CG For-Sale Unstable MBTPS1 60 34 COC(=O)[C@H](O)CNC(=O)c1cccc(C)c1[N+](=O)[O-] ZINC000217698425 CC On-Demand Unstable CACNA1D 62 33 Cc1ccccc1/C=C/NC(=O)NCCc1ccccc1Cl ZINC000217698442 DI For-Sale Unstable CXCL8 41 34 CCCCN(C(=O)c1cccc(/C=C\C(=O)O)c1)C1CC1 ZINC000217698457 CG For-Sale Unstable ACE 26 40 C[C@](O)(CNC(=O)/C=C\c1ccccc1)CC(=O)O ZINC000217698484 CD For-Sale Unstable HDAC8 52 37 C[C@](O)(CNC(=O)/C=C\c1ccccc1)CC(=O)O ZINC000217698484 CD For-Sale Unstable F3 18 43 C[C@](O)(CNC(=O)/C=C\c1ccccc1)CC(=O)O ZINC000217698484 CD For-Sale Unstable MMP2 22 55 C[C@](O)(CNC(=O)/C=C\c1ccccc1)CC(=O)O ZINC000217698484 CD For-Sale Unstable HDAC1 33 42 C[C@](O)(CNC(=O)/C=C\c1ccccc1)CC(=O)O ZINC000217698484 CD For-Sale Unstable HDAC4 21 42 C[C@](O)(CNC(=O)/C=C\c1ccccc1)CC(=O)O ZINC000217698484 CD For-Sale Unstable HDAC6 37 51 C[C@](O)(CNC(=O)/C=C\c1ccccc1)CC(=O)O ZINC000217698484 CD For-Sale Unstable MMP9 19 55 C[C@](O)(CNC(=O)/C=C\c1ccccc1)CC(=O)O ZINC000217698484 CD For-Sale Unstable HDAC9 26 42 C[C@](O)(CNC(=O)/C=C\c1ccccc1)CC(=O)O ZINC000217698484 CD For-Sale Unstable HDAC7 40 42 C[C@](O)(CNC(=O)/C=C\c1ccccc1)CC(=O)O ZINC000217698484 CD For-Sale Unstable MMP1 0 44 O=S(=O)(NC[C@H]1CCCN1c1nc2ccccc2o1)c1cccs1 ZINC000217698509 FF In-Stock Unstable NPY1R 41 32 COC(=O)[C@@H](O)CNC(=O)c1cccc(OC)c1 ZINC000217698544 CB On-Demand Unstable PRSS1 22 42 COC(=O)[C@@H](O)CNC(=O)c1cccc(OC)c1 ZINC000217698544 CB On-Demand Unstable DRD4 62 48 COC(=O)[C@@H](O)CNC(=O)c1cccc(OC)c1 ZINC000217698544 CB On-Demand Unstable F10 17 40 COC(=O)[C@@H](O)CNC(=O)c1cccc(OC)c1 ZINC000217698544 CB On-Demand Unstable NQO2 17 43 COC(=O)[C@@H](O)CNC(=O)c1cccc(OC)c1 ZINC000217698544 CB On-Demand Unstable MTNR1A 47 47 COC(=O)[C@@H](O)CNC(=O)c1cccc(OC)c1 ZINC000217698544 CB On-Demand Unstable MTNR1B 48 47 COC(=O)[C@@H](O)CNC(=O)c1cccc(OC)c1 ZINC000217698544 CB On-Demand Unstable ACR 24 42 COC(=O)[C@@H](O)CNC(=O)c1cccc(OC)c1 ZINC000217698544 CB On-Demand Unstable ITGAV 38 43 COC(=O)[C@@H](O)CNC(=O)c1cccc(OC)c1 ZINC000217698544 CB On-Demand Unstable HSD17B2 22 42 COC(=O)[C@@H](O)CNC(=O)c1cccc(OC)c1 ZINC000217698544 CB On-Demand Unstable TAAR1 25 41 COC(=O)[C@@H](O)CNC(=O)c1cccc(OC)c1 ZINC000217698544 CB On-Demand Unstable KCNK3 28 50 CCC[C@@H](C)NS(=O)(=O)c1ccc(NC)c(C(=O)O)c1 ZINC000217698559 DD In-Stock Unstable MMP12 47 37 CCC[C@@H](C)NS(=O)(=O)c1ccc(NC)c(C(=O)O)c1 ZINC000217698559 DD In-Stock Unstable LEF 51 36 C[C@@](O)(CNC(=O)/C=C\c1ccccc1)CC(=O)O ZINC000217698576 CD For-Sale Unstable HDAC8 52 37 C[C@@](O)(CNC(=O)/C=C\c1ccccc1)CC(=O)O ZINC000217698576 CD For-Sale Unstable F3 18 43 C[C@@](O)(CNC(=O)/C=C\c1ccccc1)CC(=O)O ZINC000217698576 CD For-Sale Unstable MMP2 22 55 C[C@@](O)(CNC(=O)/C=C\c1ccccc1)CC(=O)O ZINC000217698576 CD For-Sale Unstable HDAC1 33 42 C[C@@](O)(CNC(=O)/C=C\c1ccccc1)CC(=O)O ZINC000217698576 CD For-Sale Unstable HDAC4 21 42 C[C@@](O)(CNC(=O)/C=C\c1ccccc1)CC(=O)O ZINC000217698576 CD For-Sale Unstable HDAC6 37 51 C[C@@](O)(CNC(=O)/C=C\c1ccccc1)CC(=O)O ZINC000217698576 CD For-Sale Unstable MMP9 19 55 C[C@@](O)(CNC(=O)/C=C\c1ccccc1)CC(=O)O ZINC000217698576 CD For-Sale Unstable HDAC9 26 42 C[C@@](O)(CNC(=O)/C=C\c1ccccc1)CC(=O)O ZINC000217698576 CD For-Sale Unstable HDAC7 40 42 C[C@@](O)(CNC(=O)/C=C\c1ccccc1)CC(=O)O ZINC000217698576 CD For-Sale Unstable MMP1 0 44 C[C@@](O)(CNC(=O)/C=C\c1ccccc1)CC(=O)O ZINC000217698576 CD For-Sale Unstable IMA1 0 43 O=S(=O)(NC[C@@H]1CCCN1c1nc2ccccc2o1)c1cccs1 ZINC000217698592 FF In-Stock Unstable NPY1R 41 32 COc1ccc(Cc2ccccn2)cc1OC ZINC000217698603 BF Annotated Unstable FOLA 22 47 COc1ccc(Cc2ccccn2)cc1OC ZINC000217698603 BF Annotated Unstable DRTS_PLAFK 39 42 COc1ccc(Cc2ccccn2)cc1OC ZINC000217698603 BF Annotated Unstable DRTS_PLABA 21 47 COc1ccc(Cc2ccccn2)cc1OC ZINC000217698603 BF Annotated Unstable Q9XSW7_PIG 0 51 COc1ccc(Cc2ccccn2)cc1OC ZINC000217698603 BF Annotated Unstable TTR 0 42 COc1ccc(Cc2ccccn2)cc1OC ZINC000217698603 BF Annotated Unstable PDEB1 0 43 COC(=O)[C@H](O)CNC(=O)c1cccc(OC)c1 ZINC000217698632 CB On-Demand Unstable PRSS1 22 42 COC(=O)[C@H](O)CNC(=O)c1cccc(OC)c1 ZINC000217698632 CB On-Demand Unstable DRD4 62 48 COC(=O)[C@H](O)CNC(=O)c1cccc(OC)c1 ZINC000217698632 CB On-Demand Unstable F10 17 40 COC(=O)[C@H](O)CNC(=O)c1cccc(OC)c1 ZINC000217698632 CB On-Demand Unstable NQO2 17 43 COC(=O)[C@H](O)CNC(=O)c1cccc(OC)c1 ZINC000217698632 CB On-Demand Unstable MTNR1A 47 47 COC(=O)[C@H](O)CNC(=O)c1cccc(OC)c1 ZINC000217698632 CB On-Demand Unstable MTNR1B 48 47 COC(=O)[C@H](O)CNC(=O)c1cccc(OC)c1 ZINC000217698632 CB On-Demand Unstable ACR 24 42 COC(=O)[C@H](O)CNC(=O)c1cccc(OC)c1 ZINC000217698632 CB On-Demand Unstable ITGAV 38 43 COC(=O)[C@H](O)CNC(=O)c1cccc(OC)c1 ZINC000217698632 CB On-Demand Unstable HSD17B2 22 42 COC(=O)[C@H](O)CNC(=O)c1cccc(OC)c1 ZINC000217698632 CB On-Demand Unstable TAAR1 25 41 COC(=O)[C@H](O)CNC(=O)c1cccc(OC)c1 ZINC000217698632 CB On-Demand Unstable KCNK3 28 50 CCC[C@H](C)NS(=O)(=O)c1ccc(NC)c(C(=O)O)c1 ZINC000217698637 DD In-Stock Unstable MMP12 47 37 CCC[C@H](C)NS(=O)(=O)c1ccc(NC)c(C(=O)O)c1 ZINC000217698637 DD In-Stock Unstable LEF 51 36 CC[C@H](C(=O)O)N(C)C(=O)/C=C\c1cccc(OC)c1 ZINC000217698653 CE For-Sale Unstable AHR 18 41 CC[C@H](C(=O)O)N(C)C(=O)/C=C\c1cccc(OC)c1 ZINC000217698653 CE For-Sale Unstable NR1H4 31 40 CC[C@H](C(=O)O)N(C)C(=O)/C=C\c1cccc(OC)c1 ZINC000217698653 CE For-Sale Unstable AKR1C3 19 41 c1ccc2c(c1)CC(N[C@@H]1CCN3CCCC[C@@H]13)C2 ZINC000217698718 CE On-Demand Unstable VACHT_TETCF 0 43 COC(=O)[C@@H](O)CNC(=O)c1cccc(OC(F)F)c1 ZINC000217698728 CC On-Demand Unstable DRD4 49 39 CC[C@@H](C(=O)O)N(C)C(=O)/C=C\c1cccc(OC)c1 ZINC000217698745 CE For-Sale Unstable AHR 18 41 CC[C@@H](C(=O)O)N(C)C(=O)/C=C\c1cccc(OC)c1 ZINC000217698745 CE For-Sale Unstable NR1H4 31 40 CC[C@@H](C(=O)O)N(C)C(=O)/C=C\c1cccc(OC)c1 ZINC000217698745 CE For-Sale Unstable AKR1C3 19 41 CSc1ccccc1-n1nc(C(=O)O)cc1O ZINC000217698749 CD In-Stock Unstable RPA1 68 39 COc1cccc(CCNC(=O)N/C=C/c2ccccc2C)c1 ZINC000217698780 DH For-Sale Unstable DRD4 43 33 COc1cccc(CCNC(=O)N/C=C/c2ccccc2C)c1 ZINC000217698780 DH For-Sale Unstable MTNR1A 89 52 COc1cccc(CCNC(=O)N/C=C/c2ccccc2C)c1 ZINC000217698780 DH For-Sale Unstable MTNR1B 81 52 COc1cccc(CCNC(=O)N/C=C/c2ccccc2C)c1 ZINC000217698780 DH For-Sale Unstable CRTM 54 39 COC(=O)[C@H](O)CNC(=O)c1cccc(OC(F)F)c1 ZINC000217698805 CC On-Demand Unstable DRD4 49 39 Cc1cc(C)c(-n2nc(C(=O)O)cc2O)c(C)c1 ZINC000217698849 BE In-Stock Unstable RPA1 66 40 CC[C@H](C(=O)O)N(C)C(=O)/C=C\c1ccccc1OC ZINC000217698859 CE For-Sale Unstable AKR1B10 28 40 C[C@](O)(CNC(=O)/C=C\c1ccc(Br)cc1)CC(=O)O ZINC000217698886 ED For-Sale Unstable HDAC2 15 40 C[C@](O)(CNC(=O)/C=C\c1ccc(Br)cc1)CC(=O)O ZINC000217698886 ED For-Sale Unstable HDAC6 17 40 COc1ccc(CNC(=O)CN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@H]23)cc1OC ZINC000217698902 JG In-Stock Unstable TSHR 50 34 COc1ccc(CNC(=O)CN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@H]23)cc1OC ZINC000217698902 JG In-Stock Unstable HCRTR1 20 44 COc1ccc(CNC(=O)CN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@H]23)cc1OC ZINC000217698902 JG In-Stock Unstable SCN9A 0 40 CC[C@@H](C(=O)O)N(C)C(=O)/C=C\c1ccccc1OC ZINC000217698941 CE For-Sale Unstable AKR1B10 28 40 Nc1cccc(-n2nc(C(=O)O)cc2O)c1 ZINC000217698969 BC In-Stock Unstable RPA1 87 48 COc1ccc(CNC(=O)CN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@@H]23)cc1OC ZINC000217698980 JG In-Stock Unstable TSHR 50 34 COc1ccc(CNC(=O)CN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@@H]23)cc1OC ZINC000217698980 JG In-Stock Unstable HCRTR1 20 44 COc1ccc(CNC(=O)CN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@@H]23)cc1OC ZINC000217698980 JG In-Stock Unstable SCN9A 0 40 C[C@@](O)(CNC(=O)/C=C\c1ccc(Br)cc1)CC(=O)O ZINC000217698990 ED For-Sale Unstable HDAC2 15 40 C[C@@](O)(CNC(=O)/C=C\c1ccc(Br)cc1)CC(=O)O ZINC000217698990 ED For-Sale Unstable HDAC6 17 40 Cc1ccccc1/C=C/NC(=O)NCCc1cccc(Cl)c1 ZINC000217699009 DI For-Sale Unstable LMGT2 0 44 C[C@H](NC(=O)c1ccc2c(ccn2Cc2ccccc2)c1)C(=O)O ZINC000217699082 DF In-Stock Unstable MME 34 42 C[C@H](NC(=O)c1ccc2c(ccn2Cc2ccccc2)c1)C(=O)O ZINC000217699082 DF In-Stock Unstable PTGER4 21 43 C[C@H](NC(=O)c1ccc2c(ccn2Cc2ccccc2)c1)C(=O)O ZINC000217699082 DF In-Stock Unstable GLO1 20 41 C[C@H](NC(=O)c1ccc2c(ccn2Cc2ccccc2)c1)C(=O)O ZINC000217699082 DF In-Stock Unstable SLC15A1 0 40 C[C@H](NC(=O)c1ccc2c(ccn2Cc2ccccc2)c1)C(=O)O ZINC000217699082 DF In-Stock Unstable PTGDR 0 41 C[C@H](NC(=O)c1ccc2c(ccn2Cc2ccccc2)c1)C(=O)O ZINC000217699082 DF In-Stock Unstable SLC15A2 0 44 C[C@](O)(CNC(=O)/C=C\c1ccc(O)cc1)CC(=O)O ZINC000217699084 CC For-Sale Unstable HDAC8 15 48 C[C@](O)(CNC(=O)/C=C\c1ccc(O)cc1)CC(=O)O ZINC000217699084 CC For-Sale Unstable F3 26 44 C[C@](O)(CNC(=O)/C=C\c1ccc(O)cc1)CC(=O)O ZINC000217699084 CC For-Sale Unstable MMP2 15 55 C[C@](O)(CNC(=O)/C=C\c1ccc(O)cc1)CC(=O)O ZINC000217699084 CC For-Sale Unstable MMP9 15 55 C[C@](O)(CNC(=O)/C=C\c1ccc(O)cc1)CC(=O)O ZINC000217699084 CC For-Sale Unstable MMP1 23 48 C[C@](O)(CNC(=O)/C=C\c1ccc(O)cc1)CC(=O)O ZINC000217699084 CC For-Sale Unstable SSSIM 16 49 C[C@](O)(CNC(=O)/C=C\c1ccc(O)cc1)CC(=O)O ZINC000217699084 CC For-Sale Unstable IMA1 0 43 C[C@@](O)(CNC(=O)/C=C\c1ccc(O)cc1)CC(=O)O ZINC000217699178 CC For-Sale Unstable HDAC8 15 48 C[C@@](O)(CNC(=O)/C=C\c1ccc(O)cc1)CC(=O)O ZINC000217699178 CC For-Sale Unstable F3 26 44 C[C@@](O)(CNC(=O)/C=C\c1ccc(O)cc1)CC(=O)O ZINC000217699178 CC For-Sale Unstable MMP2 15 55 C[C@@](O)(CNC(=O)/C=C\c1ccc(O)cc1)CC(=O)O ZINC000217699178 CC For-Sale Unstable MMP9 15 55 C[C@@](O)(CNC(=O)/C=C\c1ccc(O)cc1)CC(=O)O ZINC000217699178 CC For-Sale Unstable MMP1 23 48 C[C@@](O)(CNC(=O)/C=C\c1ccc(O)cc1)CC(=O)O ZINC000217699178 CC For-Sale Unstable SSSIM 16 49 C[C@@](O)(CNC(=O)/C=C\c1ccc(O)cc1)CC(=O)O ZINC000217699178 CC For-Sale Unstable IMA1 0 43 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)NC3CCCCCC3)[C@H]21 ZINC000217699193 JH In-Stock Unstable NTSR2 44 38 CCC(CC)(CNCc1ccccc1)NC(=O)OC(C)(C)C ZINC000217699215 DH On-Demand Unstable CTSB 15 42 CCC(CC)(CNCc1ccccc1)NC(=O)OC(C)(C)C ZINC000217699215 DH On-Demand Unstable PAPA1_CARPA 40 40 CCC(CC)(CNCc1ccccc1)NC(=O)OC(C)(C)C ZINC000217699215 DH On-Demand Unstable CTSK 16 47 CCC(CC)(CNCc1ccccc1)NC(=O)OC(C)(C)C ZINC000217699215 DH On-Demand Unstable FPR1 45 37 CCC(CC)(CNCc1ccccc1)NC(=O)OC(C)(C)C ZINC000217699215 DH On-Demand Unstable PDS 48 35 O=C(O)/C=C\c1ccc(C(=O)N2CCCC[C@@H]2CO)cc1 ZINC000217699264 CD For-Sale Unstable PREP 27 40 O=C(O)/C=C\c1ccc(C(=O)N2CCCC[C@@H]2CO)cc1 ZINC000217699264 CD For-Sale Unstable L3MBTL3 62 37 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)NC3CCCCCC3)[C@@H]21 ZINC000217699274 JH In-Stock Unstable NTSR2 44 38 CNc1ccc(S(=O)(=O)NC[C@@H]2CCCO2)cc1C(=O)O ZINC000217699278 DC In-Stock Unstable BDKRB1 0 46 C[C@](O)(CNC(=O)/C=C\c1cccc(Cl)c1)CC(=O)O ZINC000217699285 CD For-Sale Unstable PYGL 25 46 C[C@](O)(CNC(=O)/C=C\c1cccc(Cl)c1)CC(=O)O ZINC000217699285 CD For-Sale Unstable HDAC8 41 35 C[C@](O)(CNC(=O)/C=C\c1cccc(Cl)c1)CC(=O)O ZINC000217699285 CD For-Sale Unstable MMP2 15 43 C[C@](O)(CNC(=O)/C=C\c1cccc(Cl)c1)CC(=O)O ZINC000217699285 CD For-Sale Unstable MMP9 0 45 C[C@](O)(CNC(=O)/C=C\c1cccc(Cl)c1)CC(=O)O ZINC000217699285 CD For-Sale Unstable MMP1 0 48 CSc1ccccc1N[C@@H](C)C(=O)Nc1ccccc1 ZINC000217699335 CH For-Sale Unstable LPL 44 35 O=C(O)/C=C\c1ccc(C(=O)N2CCCC[C@H]2CO)cc1 ZINC000217699358 CD For-Sale Unstable PREP 27 40 O=C(O)/C=C\c1ccc(C(=O)N2CCCC[C@H]2CO)cc1 ZINC000217699358 CD For-Sale Unstable L3MBTL3 62 37 CNc1ccc(S(=O)(=O)NC[C@H]2CCCO2)cc1C(=O)O ZINC000217699368 DC In-Stock Unstable BDKRB1 0 46 C[C@@](O)(CNC(=O)/C=C\c1cccc(Cl)c1)CC(=O)O ZINC000217699376 CD For-Sale Unstable PYGL 25 46 C[C@@](O)(CNC(=O)/C=C\c1cccc(Cl)c1)CC(=O)O ZINC000217699376 CD For-Sale Unstable HDAC8 41 35 C[C@@](O)(CNC(=O)/C=C\c1cccc(Cl)c1)CC(=O)O ZINC000217699376 CD For-Sale Unstable MMP2 15 43 C[C@@](O)(CNC(=O)/C=C\c1cccc(Cl)c1)CC(=O)O ZINC000217699376 CD For-Sale Unstable MMP9 0 45 C[C@@](O)(CNC(=O)/C=C\c1cccc(Cl)c1)CC(=O)O ZINC000217699376 CD For-Sale Unstable MMP1 0 48 C[C@@](O)(CNC(=O)/C=C\c1cccc(Cl)c1)CC(=O)O ZINC000217699376 CD For-Sale Unstable TUBA4A 0 42 CSc1ccccc1N[C@H](C)C(=O)Nc1ccccc1 ZINC000217699419 CH For-Sale Unstable LPL 44 35 COc1ccc(-n2nc(C(=O)O)cc2O)c(OC)c1 ZINC000217699474 CD In-Stock Unstable AKR1C2 40 33 COc1ccc(-n2nc(C(=O)O)cc2O)c(OC)c1 ZINC000217699474 CD In-Stock Unstable RPA1 68 48 C[C@](O)(CNC(=O)/C=C\c1cccc(F)c1)CC(=O)O ZINC000217699498 CD For-Sale Unstable HDAC8 40 35 C[C@](O)(CNC(=O)/C=C\c1cccc(F)c1)CC(=O)O ZINC000217699498 CD For-Sale Unstable MMP2 15 43 C[C@](O)(CNC(=O)/C=C\c1cccc(F)c1)CC(=O)O ZINC000217699498 CD For-Sale Unstable MMP9 0 45 C[C@](O)(CNC(=O)/C=C\c1cccc(F)c1)CC(=O)O ZINC000217699498 CD For-Sale Unstable MMP1 0 48 CSc1ccccc1N[C@@H](C)C(=O)NC1CCCC1 ZINC000217699524 CG For-Sale Unstable EPHX2 16 40 COC(=O)C[C@@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(OC)cc1 ZINC000217699587 FG In-Stock Unstable KCNA5 32 41 COC(=O)C[C@@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(OC)cc1 ZINC000217699587 FG In-Stock Unstable HDAC2 17 40 COc1ccc(OC)c(-n2nc(C(=O)O)cc2O)c1 ZINC000217699588 CD In-Stock Unstable AKR1C2 45 33 COc1ccc(OC)c(-n2nc(C(=O)O)cc2O)c1 ZINC000217699588 CD In-Stock Unstable RPA1 68 48 C[C@@](O)(CNC(=O)/C=C\c1cccc(F)c1)CC(=O)O ZINC000217699591 CD For-Sale Unstable HDAC8 40 35 C[C@@](O)(CNC(=O)/C=C\c1cccc(F)c1)CC(=O)O ZINC000217699591 CD For-Sale Unstable MMP2 15 43 C[C@@](O)(CNC(=O)/C=C\c1cccc(F)c1)CC(=O)O ZINC000217699591 CD For-Sale Unstable MMP9 0 45 C[C@@](O)(CNC(=O)/C=C\c1cccc(F)c1)CC(=O)O ZINC000217699591 CD For-Sale Unstable MMP1 0 48 CSc1ccccc1N[C@H](C)C(=O)NC1CCCC1 ZINC000217699614 CG For-Sale Unstable EPHX2 16 40 COC(=O)C[C@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(OC)cc1 ZINC000217699666 FG In-Stock Unstable KCNA5 32 41 COC(=O)C[C@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(OC)cc1 ZINC000217699666 FG In-Stock Unstable HDAC2 17 40 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NC(C)(C)C ZINC000217699702 DD In-Stock Unstable NEU3 0 42 c1ccc(CN2CC[C@H](c3ccccc3)[C@H](COc3ccc4c(c3)OCO4)C2)cc1 ZINC000217699719 HK For-Sale Unstable DRD4 26 40 c1ccc(CN2CC[C@H](c3ccccc3)[C@H](COc3ccc4c(c3)OCO4)C2)cc1 ZINC000217699719 HK For-Sale Unstable EDNRA 43 39 c1ccc(CN2CC[C@H](c3ccccc3)[C@H](COc3ccc4c(c3)OCO4)C2)cc1 ZINC000217699719 HK For-Sale Unstable SIGMAR1 38 46 c1ccc(CN2CC[C@H](c3ccccc3)[C@H](COc3ccc4c(c3)OCO4)C2)cc1 ZINC000217699719 HK For-Sale Unstable MCHR1 26 41 Cc1ccc(NC(=O)N/C=C/c2ccccc2C)nc1 ZINC000217699737 CG For-Sale Unstable LUCI_LUCLA 39 40 CSc1ccccc1N[C@@H](C)C(=O)N1CCCCC1 ZINC000217699741 CG For-Sale Unstable KCNQ2 57 37 CSc1ccccc1N[C@@H](C)C(=O)N1CCCCC1 ZINC000217699741 CG For-Sale Unstable DPP7 66 40 O=C(NCC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)c1ccccc1 ZINC000217699787 FD In-Stock Unstable CHRNA4 32 56 O=C(NCC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)c1ccccc1 ZINC000217699787 FD In-Stock Unstable PREP 25 44 O=C(NCC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)c1ccccc1 ZINC000217699787 FD In-Stock Unstable FAP 0 47 CCCNS(=O)(=O)c1ccc(NCC)c(C(=O)O)c1 ZINC000217699816 CD In-Stock Unstable CASP3 16 43 CSc1ccccc1N[C@H](C)C(=O)N1CCCCC1 ZINC000217699832 CG For-Sale Unstable KCNQ2 57 37 CSc1ccccc1N[C@H](C)C(=O)N1CCCCC1 ZINC000217699832 CG For-Sale Unstable DPP7 66 40 Cc1cc(S(=O)(=O)N2CCOCC2)ccc1/C=C\C(=O)O ZINC000217699842 DD For-Sale Unstable LPL 38 42 Cc1cc(S(=O)(=O)N2CCOCC2)ccc1/C=C\C(=O)O ZINC000217699842 DD For-Sale Unstable CASP3 0 48 Cc1cc(S(=O)(=O)N2CCOCC2)ccc1/C=C\C(=O)O ZINC000217699842 DD For-Sale Unstable AKR1C3 49 37 Cc1cc(S(=O)(=O)N2CCOCC2)ccc1/C=C\C(=O)O ZINC000217699842 DD For-Sale Unstable LIPG 15 42 CCCCCCCCOc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)cc1 ZINC000217699892 KK In-Stock Unstable ALOX5 0 55 CCCCCCCCOc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)cc1 ZINC000217699892 KK In-Stock Unstable AKR1B1 22 49 CCCCCCCCOc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)cc1 ZINC000217699892 KK In-Stock Unstable CYP1A1 29 42 O=C(/C=C/c1ccccc1)NCCSC1CCOCC1 ZINC000217699925 CF In-Stock Unstable IMA1 0 43 COC(=O)[C@@H](O)CNC(=O)COc1cccc([N+](=O)[O-])c1 ZINC000217699931 CB On-Demand Unstable CACNA1C 57 39 COC(=O)[C@@H](O)CNC(=O)COc1cccc([N+](=O)[O-])c1 ZINC000217699931 CB On-Demand Unstable CACNA1D 93 41 COC(=O)[C@@H](O)CNC(=O)COc1cccc([N+](=O)[O-])c1 ZINC000217699931 CB On-Demand Unstable ACR 22 44 Cc1ccc([N+](=O)[O-])cc1-n1nc(C(=O)O)cc1O ZINC000217699940 CD In-Stock Unstable RPA1 55 34 O=C(O)/C=C\c1cccc(S(=O)(=O)NC2CCCC2)c1 ZINC000217699941 CE For-Sale Unstable HDAC8 17 51 O=C(O)/C=C\c1cccc(S(=O)(=O)NC2CCCC2)c1 ZINC000217699941 CE For-Sale Unstable SFRP1 130 38 O=C(O)/C=C\c1cccc(S(=O)(=O)NC2CCCC2)c1 ZINC000217699941 CE For-Sale Unstable WNT3 87 38 CSc1ccccc1N[C@@H](C)C(=O)N1CCCC1 ZINC000217699946 CF For-Sale Unstable KCNQ2 65 38 CSc1ccccc1N[C@@H](C)C(=O)N1CCCC1 ZINC000217699946 CF For-Sale Unstable DPP7 57 38 CCCCCCCCOc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)cc1 ZINC000217699962 KK In-Stock Unstable ALOX5 0 55 CCCCCCCCOc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)cc1 ZINC000217699962 KK In-Stock Unstable AKR1B1 22 49 CCCCCCCCOc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)cc1 ZINC000217699962 KK In-Stock Unstable CYP1A1 29 42 COC(=O)[C@H](O)CNC(=O)COc1cccc([N+](=O)[O-])c1 ZINC000217700008 CB On-Demand Unstable CACNA1C 57 39 COC(=O)[C@H](O)CNC(=O)COc1cccc([N+](=O)[O-])c1 ZINC000217700008 CB On-Demand Unstable CACNA1D 93 41 COC(=O)[C@H](O)CNC(=O)COc1cccc([N+](=O)[O-])c1 ZINC000217700008 CB On-Demand Unstable ACR 22 44 Cc1cc(S(=O)(=O)NC2CCCC2)ccc1/C=C\C(=O)O ZINC000217700037 DE For-Sale Unstable LEF 32 40 Cc1cc(S(=O)(=O)NC2CCCC2)ccc1/C=C\C(=O)O ZINC000217700037 DE For-Sale Unstable SFRP1 113 34 Cc1cc(S(=O)(=O)NC2CCCC2)ccc1/C=C\C(=O)O ZINC000217700037 DE For-Sale Unstable WNT3 79 33 CSc1ccccc1N[C@H](C)C(=O)N1CCCC1 ZINC000217700040 CF For-Sale Unstable KCNQ2 65 38 CSc1ccccc1N[C@H](C)C(=O)N1CCCC1 ZINC000217700040 CF For-Sale Unstable DPP7 57 38 CCC(CC)(CNCc1ccccc1F)NC(=O)OC(C)(C)C ZINC000217700055 DH On-Demand Unstable PAPA1_CARPA 25 44 CCNc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O ZINC000217700056 EF In-Stock Unstable BDKRB1 17 41 CCNc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O ZINC000217700056 EF In-Stock Unstable MMP12 44 37 CCNc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O ZINC000217700056 EF In-Stock Unstable ADAMTS4 41 32 CCNc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O ZINC000217700056 EF In-Stock Unstable LEF 33 41 COc1ccc([C@@H]2CC(=O)Oc3c2c(=O)oc2ccccc32)c2ccccc12 ZINC000217700077 FI In-Stock Unstable NQO1 22 41 Cc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)cn1 ZINC000217700089 CH For-Sale Unstable LUCI_LUCLA 39 42 Cc1ccc(/C=C\C(=O)O)cc1S(=O)(=O)NC1CCCC1 ZINC000217700125 DE For-Sale Unstable CCR8 73 38 Cc1ccc(/C=C\C(=O)O)cc1S(=O)(=O)NC1CCCC1 ZINC000217700125 DE For-Sale Unstable SFRP1 118 35 Cc1ccc(/C=C\C(=O)O)cc1S(=O)(=O)NC1CCCC1 ZINC000217700125 DE For-Sale Unstable WNT3 83 35 Cc1ccc(/C=C\C(=O)O)cc1S(=O)(=O)NC1CCCC1 ZINC000217700125 DE For-Sale Unstable BRD4 24 52 O=C(NCCSC1CCOCC1)c1ccc(Cl)s1 ZINC000217700133 DG In-Stock Unstable F10 23 44 CCNc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O ZINC000217700144 EF In-Stock Unstable BDKRB1 17 41 CCNc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O ZINC000217700144 EF In-Stock Unstable MMP12 44 37 CCNc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O ZINC000217700144 EF In-Stock Unstable ADAMTS4 41 32 CCNc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O ZINC000217700144 EF In-Stock Unstable LEF 33 41 O=C(NCc1cccnc1)[C@@H]1[C@H]2C=C[C@@]3(CN(CCc4ccccc4)C(=O)[C@H]13)O2 ZINC000217700149 GD In-Stock Unstable NAMPT 46 38 COc1ccc([C@H]2CC(=O)Oc3c2c(=O)oc2ccccc32)c2ccccc12 ZINC000217700167 FI In-Stock Unstable NQO1 30 41 Cc1ccccc1/C=C/NC(=O)Nc1cc(Cl)ccn1 ZINC000217700199 CH For-Sale Unstable TYK2 48 34 O=C(O)/C=C\c1cccc(S(=O)(=O)Nc2ccncc2)c1 ZINC000217700213 DD For-Sale Anodyne HDAC8 17 64 O=C(O)/C=C\c1cccc(S(=O)(=O)Nc2ccncc2)c1 ZINC000217700213 DD For-Sale Anodyne HDAC1 0 64 O=C(O)/C=C\c1cccc(S(=O)(=O)Nc2ccncc2)c1 ZINC000217700213 DD For-Sale Anodyne RHOA 0 42 C[C@](O)(CNC(=O)/C=C\c1ccc(F)c(Cl)c1)CC(=O)O ZINC000217700219 DD For-Sale Unstable PYGL 27 50 C[C@](O)(CNC(=O)/C=C\c1ccc(F)c(Cl)c1)CC(=O)O ZINC000217700219 DD For-Sale Unstable HPSE 32 41 C[C@](O)(CNC(=O)/C=C\c1ccc(F)c(Cl)c1)CC(=O)O ZINC000217700219 DD For-Sale Unstable HD1B 0 40 O=C(NCc1cccnc1)[C@H]1[C@H]2C=C[C@@]3(CN(CCc4ccccc4)C(=O)[C@H]13)O2 ZINC000217700223 GD In-Stock Unstable NAMPT 46 38 CC[C@H](C(=O)NCCSC1CCOCC1)c1ccccc1 ZINC000217700246 DG In-Stock Unstable KCNQ2 42 42 O=C(O)c1cc(O)n(-c2ccc3c(c2)OCO3)n1 ZINC000217700268 BD In-Stock Unstable DHRS9 0 40 O=C(O)c1cc(O)n(-c2ccc3c(c2)OCO3)n1 ZINC000217700268 BD In-Stock Unstable RPA1 75 42 C[C@@](O)(CNC(=O)/C=C\c1ccc(F)c(Cl)c1)CC(=O)O ZINC000217700295 DD For-Sale Unstable PYGL 27 50 C[C@@](O)(CNC(=O)/C=C\c1ccc(F)c(Cl)c1)CC(=O)O ZINC000217700295 DD For-Sale Unstable HPSE 32 41 C[C@@](O)(CNC(=O)/C=C\c1ccc(F)c(Cl)c1)CC(=O)O ZINC000217700295 DD For-Sale Unstable HD1B 0 40 CCCC[C@@H](CN)N1C[C@H](C)O[C@@H](C)C1 ZINC000217700297 BD For-Sale Unstable ZM.86993 0 44 CC[C@@H](C(=O)O)[C@@H](C)NC(=O)OC(C)(C)C ZINC000217700310 BE For-Sale Unstable PAPA1_CARPA 36 43 CC[C@@H](C(=O)O)[C@@H](C)NC(=O)OC(C)(C)C ZINC000217700310 BE For-Sale Unstable CTSK 33 54 CC[C@@H](C(=O)O)[C@@H](C)NC(=O)OC(C)(C)C ZINC000217700310 BE For-Sale Unstable PGA5 23 41 CC[C@@H](C(=O)O)[C@@H](C)NC(=O)OC(C)(C)C ZINC000217700310 BE For-Sale Unstable POLG_HCV1 23 40 CC[C@@H](C(=O)O)[C@@H](C)NC(=O)OC(C)(C)C ZINC000217700310 BE For-Sale Unstable FPR1 45 38 CC[C@@H](C(=O)O)[C@@H](C)NC(=O)OC(C)(C)C ZINC000217700310 BE For-Sale Unstable POL 0 50 CC[C@@H](C(=O)NCCSC1CCOCC1)c1ccccc1 ZINC000217700331 DG In-Stock Unstable KCNQ2 42 42 CCCCNS(=O)(=O)c1ccc(NCC)c(C(=O)O)c1 ZINC000217700391 DD In-Stock Unstable CASP3 16 46 CCCCNS(=O)(=O)c1ccc(NCC)c(C(=O)O)c1 ZINC000217700391 DD In-Stock Unstable BDKRB1 0 43 CCCC[C@H](CN)N1C[C@H](C)O[C@@H](C)C1 ZINC000217700393 BD For-Sale Unstable ZM.86993 0 44 Cc1ccccc1/C=C/NC(=O)NCCCc1ccccc1 ZINC000217700437 CH For-Sale Unstable MTNR1A 27 44 Cc1ccccc1/C=C/NC(=O)NCCCc1ccccc1 ZINC000217700437 CH For-Sale Unstable MTNR1B 39 44 Cc1ccccc1/C=C/NC(=O)NCCCc1ccccc1 ZINC000217700437 CH For-Sale Unstable FAAH 18 43 Cc1ccccc1/C=C/NC(=O)NCCCc1ccccc1 ZINC000217700437 CH For-Sale Unstable SCN5A 0 43 Cc1ccccc1/C=C/NC(=O)NCCCc1ccccc1 ZINC000217700437 CH For-Sale Unstable AMP1_PLAFQ 26 45 CN(C)c1cccc(C(=O)NCCSC2CCOCC2)c1 ZINC000217700443 DE In-Stock Unstable DRD4 40 31 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cnn(C)c2)CC(=O)O4)cc1O ZINC000217700470 IG In-Stock Unstable AKR1B1 0 46 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cnn(C)c2)CC(=O)O4)cc1O ZINC000217700470 IG In-Stock Unstable CYP1B1 42 46 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cnn(C)c2)CC(=O)O4)cc1O ZINC000217700470 IG In-Stock Unstable CYP1A1 34 46 O=C(O)c1cc(O)n(-c2ccc(OCc3ccccc3)cc2)n1 ZINC000217700519 DF In-Stock Unstable MAOB 29 41 O=C(O)c1cc(O)n(-c2ccc(OCc3ccccc3)cc2)n1 ZINC000217700519 DF In-Stock Unstable PTGER2 24 40 O=C(O)c1cc(O)n(-c2ccc(OCc3ccccc3)cc2)n1 ZINC000217700519 DF In-Stock Unstable KCNH2 18 41 O=C(O)c1cc(O)n(-c2ccc(OCc3ccccc3)cc2)n1 ZINC000217700519 DF In-Stock Unstable LTA4H 28 43 O=C(O)c1cc(O)n(-c2ccc(OCc3ccccc3)cc2)n1 ZINC000217700519 DF In-Stock Unstable EDNRA 0 52 O=C(O)c1cc(O)n(-c2ccc(OCc3ccccc3)cc2)n1 ZINC000217700519 DF In-Stock Unstable PTGER1 51 38 O=C(O)c1cc(O)n(-c2ccc(OCc3ccccc3)cc2)n1 ZINC000217700519 DF In-Stock Unstable PTGER4 0 41 O=C(O)c1cc(O)n(-c2ccc(OCc3ccccc3)cc2)n1 ZINC000217700519 DF In-Stock Unstable HRAS 40 31 O=C(O)c1cc(O)n(-c2ccc(OCc3ccccc3)cc2)n1 ZINC000217700519 DF In-Stock Unstable ADAM17 21 41 O=C(O)c1cc(O)n(-c2ccc(OCc3ccccc3)cc2)n1 ZINC000217700519 DF In-Stock Unstable POBA 0 45 O=C(O)c1cc(O)n(-c2ccc(OCc3ccccc3)cc2)n1 ZINC000217700519 DF In-Stock Unstable FFAR1 44 46 O=C(O)c1cc(O)n(-c2ccc(OCc3ccccc3)cc2)n1 ZINC000217700519 DF In-Stock Unstable RPA1 83 39 O=C(O)c1cc(O)n(-c2ccc(OCc3ccccc3)cc2)n1 ZINC000217700519 DF In-Stock Unstable SLC16A3 0 40 O=C(Cc1ccc2c(c1)OCO2)N1CCCn2nc([C@@H](O)CO)cc2C1 ZINC000217700543 FC In-Stock Unstable SSTR3 43 29 Cc1ccccc1/C=C/NC(=O)NCCCCc1ccccc1 ZINC000217700555 DI For-Sale Unstable SCN2A 22 40 Cc1ccccc1/C=C/NC(=O)NCCCCc1ccccc1 ZINC000217700555 DI For-Sale Unstable MTNR1A 24 43 Cc1ccccc1/C=C/NC(=O)NCCCCc1ccccc1 ZINC000217700555 DI For-Sale Unstable MTNR1B 36 43 Cc1ccccc1/C=C/NC(=O)NCCCCc1ccccc1 ZINC000217700555 DI For-Sale Unstable FAAH 38 43 Cc1ccccc1/C=C/NC(=O)NCCCCc1ccccc1 ZINC000217700555 DI For-Sale Unstable SCN5A 0 44 Cc1ccccc1/C=C/NC(=O)NCCCCc1ccccc1 ZINC000217700555 DI For-Sale Unstable CES1 41 35 Cc1ccccc1/C=C/NC(=O)NCCCCc1ccccc1 ZINC000217700555 DI For-Sale Unstable AMP1_PLAFQ 26 46 Cc1ccccc1/C=C/NC(=O)NCCCCc1ccccc1 ZINC000217700555 DI For-Sale Unstable HDA106 0 40 Cc1ccccc1/C=C/NC(=O)NCCCCc1ccccc1 ZINC000217700555 DI For-Sale Unstable ACAT 0 44 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cnn(C)c2)CC(=O)O4)cc1O ZINC000217700571 IG In-Stock Unstable AKR1B1 0 46 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cnn(C)c2)CC(=O)O4)cc1O ZINC000217700571 IG In-Stock Unstable CYP1B1 42 46 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cnn(C)c2)CC(=O)O4)cc1O ZINC000217700571 IG In-Stock Unstable CYP1A1 34 46 O=C(O)/C=C\c1ccc(C(=O)NC2CCCCC2)c(F)c1 ZINC000217700588 CF For-Sale Unstable CNR1 20 43 O=C(O)/C=C\c1ccc(C(=O)NC2CCCCC2)c(F)c1 ZINC000217700588 CF For-Sale Unstable CNR2 28 43 CCc1cccc(C)c1-n1nc(C(=O)O)cc1O ZINC000217700616 BE In-Stock Unstable RPA1 67 41 O=C(Cc1ccccc1Cl)NCCSC1CCOCC1 ZINC000217700689 DF In-Stock Unstable P2RX7 19 40 COC(=O)[C@@H](O)CNC(=O)c1cc(Cl)ccc1OC ZINC000217700701 CC On-Demand Unstable COLA 43 33 COC(=O)[C@@H](O)CNC(=O)c1cc(Cl)ccc1OC ZINC000217700701 CC On-Demand Unstable CPT1A 43 30 COC(=O)[C@@H](O)CNC(=O)c1cc(Cl)ccc1OC ZINC000217700701 CC On-Demand Unstable KCNMA1 24 49 CCOc1ccc(-n2nc(C(=O)O)cc2O)cc1 ZINC000217700742 BD In-Stock Unstable CACNA2D1 59 38 CCOc1ccc(-n2nc(C(=O)O)cc2O)cc1 ZINC000217700742 BD In-Stock Unstable PLA2G4B 48 35 CCOc1ccc(-n2nc(C(=O)O)cc2O)cc1 ZINC000217700742 BD In-Stock Unstable CACNA2D2 59 38 CCOc1ccc(-n2nc(C(=O)O)cc2O)cc1 ZINC000217700742 BD In-Stock Unstable RPA1 78 43 COC(=O)[C@H](O)CNC(=O)c1cc(Cl)ccc1OC ZINC000217700789 CC On-Demand Unstable COLA 43 33 COC(=O)[C@H](O)CNC(=O)c1cc(Cl)ccc1OC ZINC000217700789 CC On-Demand Unstable CPT1A 43 30 COC(=O)[C@H](O)CNC(=O)c1cc(Cl)ccc1OC ZINC000217700789 CC On-Demand Unstable KCNMA1 24 49 O=C(NCCSC1CCOCC1)c1ccc(F)cc1Cl ZINC000217700816 DG In-Stock Unstable P2RX7 37 43 O=C(NCCSC1CCOCC1)c1ccc(F)cc1Cl ZINC000217700816 DG In-Stock Unstable PYGL 22 42 O=C(NCCSC1CCOCC1)c1ccc(F)cc1Cl ZINC000217700816 DG In-Stock Unstable SLC6A9 22 41 O=C(O)c1cc(C(=O)O)cc(-n2nc(C(=O)O)cc2O)c1 ZINC000217700852 CC In-Stock Anodyne RPA1 74 42 CC[C@H](CCO)N[C@@H]1CC[C@@H](NC(=O)OC(C)(C)C)C1 ZINC000217700863 CE For-Sale Unstable CTSK 15 41 O=C(NCCSC1CCOCC1)c1nc2ccccc2s1 ZINC000217700924 DF In-Stock Unstable TPSAB1 19 40 O=C(NCCSC1CCOCC1)c1nc2ccccc2s1 ZINC000217700924 DF In-Stock Unstable TMPRSS6 55 31 C[C@@H]1CN(c2ccccc2)CCN1C(=O)Cc1cnccn1 ZINC000217700945 CD In-Stock Unstable SLC6A7 0 40 NS(=O)(=O)c1ccc(-n2nc(C(=O)O)cc2O)cc1 ZINC000217700982 CB In-Stock Unstable CA2 92 45 NS(=O)(=O)c1ccc(-n2nc(C(=O)O)cc2O)cc1 ZINC000217700982 CB In-Stock Unstable PTGS2 35 44 NS(=O)(=O)c1ccc(-n2nc(C(=O)O)cc2O)cc1 ZINC000217700982 CB In-Stock Unstable CA6 23 45 NS(=O)(=O)c1ccc(-n2nc(C(=O)O)cc2O)cc1 ZINC000217700982 CB In-Stock Unstable CA1 77 48 NS(=O)(=O)c1ccc(-n2nc(C(=O)O)cc2O)cc1 ZINC000217700982 CB In-Stock Unstable CA7 48 45 NS(=O)(=O)c1ccc(-n2nc(C(=O)O)cc2O)cc1 ZINC000217700982 CB In-Stock Unstable CA5B 48 36 NS(=O)(=O)c1ccc(-n2nc(C(=O)O)cc2O)cc1 ZINC000217700982 CB In-Stock Unstable CA4 80 44 NS(=O)(=O)c1ccc(-n2nc(C(=O)O)cc2O)cc1 ZINC000217700982 CB In-Stock Unstable CA5A 56 36 NS(=O)(=O)c1ccc(-n2nc(C(=O)O)cc2O)cc1 ZINC000217700982 CB In-Stock Unstable CA12 58 45 NS(=O)(=O)c1ccc(-n2nc(C(=O)O)cc2O)cc1 ZINC000217700982 CB In-Stock Unstable CA9 64 41 NS(=O)(=O)c1ccc(-n2nc(C(=O)O)cc2O)cc1 ZINC000217700982 CB In-Stock Unstable CAH_METTE 42 34 NS(=O)(=O)c1ccc(-n2nc(C(=O)O)cc2O)cc1 ZINC000217700982 CB In-Stock Unstable NCE103 28 45 NS(=O)(=O)c1ccc(-n2nc(C(=O)O)cc2O)cc1 ZINC000217700982 CB In-Stock Unstable MTCA1 44 39 NS(=O)(=O)c1ccc(-n2nc(C(=O)O)cc2O)cc1 ZINC000217700982 CB In-Stock Unstable P96878_MYCTU 58 39 NS(=O)(=O)c1ccc(-n2nc(C(=O)O)cc2O)cc1 ZINC000217700982 CB In-Stock Unstable CA 0 45 NS(=O)(=O)c1ccc(-n2nc(C(=O)O)cc2O)cc1 ZINC000217700982 CB In-Stock Unstable RPA1 75 43 NS(=O)(=O)c1ccc(-n2nc(C(=O)O)cc2O)cc1 ZINC000217700982 CB In-Stock Unstable Q5TU56_ANOGA 0 45 O=C(O)/C=C\CN1CCc2ccccc2CC1 ZINC000217700983 BD For-Sale Unstable CHRNA6 0 46 O=C(O)/C=C\CN1CCc2ccccc2CC1 ZINC000217700983 BD For-Sale Unstable NOD2 40 33 Cc1ccccc1/C=C/NC(=O)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217701011 GF For-Sale Unstable TGM2 71 42 Cc1ccccc1/C=C/NC(=O)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217701011 GF For-Sale Unstable F13A1 90 42 Cc1ccccc1/C=C/NC(=O)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217701011 GF For-Sale Unstable AKR1C3 43 36 Cc1ccc(/C=C\C(=O)NC[C@](C)(O)CC(=O)O)cc1Cl ZINC000217701015 DE For-Sale Unstable PYGL 29 54 O=C(O)/C=C\c1ccc(C(=O)Nc2cccnc2)cc1 ZINC000217701019 CE For-Sale Anodyne TBXAS1 23 54 O=C(O)/C=C\c1ccc(C(=O)Nc2cccnc2)cc1 ZINC000217701019 CE For-Sale Anodyne TRPV1 15 55 O=C(O)/C=C\c1ccc(C(=O)Nc2cccnc2)cc1 ZINC000217701019 CE For-Sale Anodyne HDAC1 16 50 O=C(O)/C=C\c1ccc(C(=O)Nc2cccnc2)cc1 ZINC000217701019 CE For-Sale Anodyne RPS6KA3 29 42 O=C(O)/C=C\c1ccc(C(=O)Nc2cccnc2)cc1 ZINC000217701019 CE For-Sale Anodyne NAMPT 33 66 O=C(O)/C=C\c1ccc(C(=O)Nc2cccnc2)cc1 ZINC000217701019 CE For-Sale Anodyne KCNK3 73 44 C=CCOc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OC ZINC000217701022 KI In-Stock Unstable ALOX5 0 42 C=CCOc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OC ZINC000217701022 KI In-Stock Unstable AKR1B1 0 42 C=CCOc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OC ZINC000217701022 KI In-Stock Unstable CYP1B1 46 41 C=CCOc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OC ZINC000217701022 KI In-Stock Unstable CYP1A1 46 41 C=CCOc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OC ZINC000217701022 KI In-Stock Unstable ABCB1A 24 46 CC[C@H](CCO)N[C@H]1CC[C@@H](NC(=O)OC(C)(C)C)C1 ZINC000217701032 CE For-Sale Unstable CTSK 15 41 C[C@H]1CN(c2ccccc2)CCN1C(=O)Cc1cnccn1 ZINC000217701040 CD In-Stock Unstable SLC6A7 0 40 CC[C@H](C(=O)O)N(C)C(=O)/C=C\c1cc(Br)ccc1OC ZINC000217701046 FF For-Sale Unstable TNFRSF1A 15 51 COC(=O)[C@@H](O)CNC(=O)c1cc(SC)ccc1[N+](=O)[O-] ZINC000217701061 DC On-Demand Unstable GSTM2 55 36 C=CCOc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OC ZINC000217701102 KI In-Stock Unstable ALOX5 0 42 C=CCOc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OC ZINC000217701102 KI In-Stock Unstable AKR1B1 0 42 C=CCOc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OC ZINC000217701102 KI In-Stock Unstable CYP1B1 46 41 C=CCOc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OC ZINC000217701102 KI In-Stock Unstable CYP1A1 46 41 C=CCOc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OC ZINC000217701102 KI In-Stock Unstable ABCB1A 24 46 Cc1ccc(/C=C\C(=O)NC[C@@](C)(O)CC(=O)O)cc1Cl ZINC000217701104 DE For-Sale Unstable PYGL 29 54 CSc1cccc(-n2nc(C(=O)O)cc2O)c1 ZINC000217701114 CD In-Stock Unstable RPA1 77 48 Cc1ccc(S(=O)(=O)N2CCN(C(=O)N/C=C/c3ccccc3C)CC2)cc1 ZINC000217701126 GF For-Sale Unstable TGM2 70 43 Cc1ccc(S(=O)(=O)N2CCN(C(=O)N/C=C/c3ccccc3C)CC2)cc1 ZINC000217701126 GF For-Sale Unstable F13A1 89 43 NC[C@@H]1CC[C@@H]1N1CCc2ccccc2C1 ZINC000217701132 BD For-Sale Unstable CHRNA6 0 41 CC[C@@H](C(=O)O)N(C)C(=O)/C=C\c1cc(Br)ccc1OC ZINC000217701135 FF For-Sale Unstable TNFRSF1A 15 51 COC(=O)[C@H](O)CNC(=O)c1cc(SC)ccc1[N+](=O)[O-] ZINC000217701142 DC On-Demand Unstable GSTM2 55 36 CN(c1ncccc1C(=O)Nc1c(N)ncnc1Cl)S(C)(=O)=O ZINC000217701177 FC For-Sale Unstable G2YM83_BOTF4 68 34 Cc1cc(NC(=O)c2ccc(/C=C\C(=O)O)cc2)on1 ZINC000217701188 CE For-Sale Unstable RPS6KA3 15 43 NC[C@@H]1CC[C@H]1N1CCc2ccccc2C1 ZINC000217701214 BD For-Sale Unstable CHRNA6 0 41 Cc1cccc(C)c1-n1nc(C(=O)O)cc1O ZINC000217701223 BD In-Stock Unstable RPA1 75 47 COc1ccc(/C=C\C(=O)NC[C@](C)(O)CC(=O)O)cc1 ZINC000217701227 CD For-Sale Unstable PTGS2 0 46 COc1ccc(/C=C\C(=O)NC[C@](C)(O)CC(=O)O)cc1 ZINC000217701227 CD For-Sale Unstable HDAC8 15 53 COc1ccc(/C=C\C(=O)NC[C@](C)(O)CC(=O)O)cc1 ZINC000217701227 CD For-Sale Unstable MMP2 17 50 COc1ccc(/C=C\C(=O)NC[C@](C)(O)CC(=O)O)cc1 ZINC000217701227 CD For-Sale Unstable HDAC1 24 44 COc1ccc(/C=C\C(=O)NC[C@](C)(O)CC(=O)O)cc1 ZINC000217701227 CD For-Sale Unstable HDAC6 15 53 COc1ccc(/C=C\C(=O)NC[C@](C)(O)CC(=O)O)cc1 ZINC000217701227 CD For-Sale Unstable MMP9 15 50 COc1ccc(/C=C\C(=O)NC[C@](C)(O)CC(=O)O)cc1 ZINC000217701227 CD For-Sale Unstable GPR183 0 41 COc1ccc(CCC(=O)NCCSC2CCOCC2)cc1 ZINC000217701272 DF In-Stock Unstable MTNR1A 45 36 COc1ccc(/C=C\C(=O)NC[C@@](C)(O)CC(=O)O)cc1 ZINC000217701309 CD For-Sale Unstable PTGS2 0 46 COc1ccc(/C=C\C(=O)NC[C@@](C)(O)CC(=O)O)cc1 ZINC000217701309 CD For-Sale Unstable HDAC8 15 53 COc1ccc(/C=C\C(=O)NC[C@@](C)(O)CC(=O)O)cc1 ZINC000217701309 CD For-Sale Unstable MMP2 17 50 COc1ccc(/C=C\C(=O)NC[C@@](C)(O)CC(=O)O)cc1 ZINC000217701309 CD For-Sale Unstable HDAC1 24 44 COc1ccc(/C=C\C(=O)NC[C@@](C)(O)CC(=O)O)cc1 ZINC000217701309 CD For-Sale Unstable HDAC6 15 53 COc1ccc(/C=C\C(=O)NC[C@@](C)(O)CC(=O)O)cc1 ZINC000217701309 CD For-Sale Unstable MMP9 15 50 COc1ccc(/C=C\C(=O)NC[C@@](C)(O)CC(=O)O)cc1 ZINC000217701309 CD For-Sale Unstable GPR183 0 41 COc1ccc(C(=O)NC[C@@](C)(O)CSC)c(F)c1 ZINC000217701342 CD On-Demand Unstable AKR1C2 43 37 COc1ccc(C(=O)NC[C@](C)(O)CSC)c(F)c1 ZINC000217701432 CD On-Demand Unstable AKR1C2 43 37 C[C@](O)(CNC(=O)/C=C\c1ccccc1F)CC(=O)O ZINC000217701445 CD For-Sale Unstable KCNQ2 40 36 O=C(O)c1cc(O)n(-c2cccc3ccccc23)n1 ZINC000217701449 CE In-Stock Anodyne NTSR2 20 40 O=C(O)c1cc(O)n(-c2cccc3ccccc23)n1 ZINC000217701449 CE In-Stock Anodyne RPA1 70 40 C[C@@](O)(CNC(=O)/C=C\c1ccccc1F)CC(=O)O ZINC000217701533 CD For-Sale Unstable KCNQ2 40 36 CCOCCCNS(=O)(=O)c1ccc(NC)c(C(=O)O)c1 ZINC000217701549 DD In-Stock Unstable CASP3 16 41 CSC[C@@](C)(O)CNC(=O)c1cc2ccccc2s1 ZINC000217701558 CF In-Stock Unstable PIN1 29 42 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(O)c(OC)c2)CC(=O)O4)cc1O ZINC000217701580 JI In-Stock Unstable ALOX5 0 52 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(O)c(OC)c2)CC(=O)O4)cc1O ZINC000217701580 JI In-Stock Unstable AKR1B1 25 55 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(O)c(OC)c2)CC(=O)O4)cc1O ZINC000217701580 JI In-Stock Unstable CYP1B1 70 39 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(O)c(OC)c2)CC(=O)O4)cc1O ZINC000217701580 JI In-Stock Unstable CYP1A1 53 50 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(O)c(OC)c2)CC(=O)O4)cc1O ZINC000217701580 JI In-Stock Unstable CYP1A2 42 43 O=C(NCCSC1CCOCC1)c1cccc(C(F)(F)F)c1 ZINC000217701602 EG In-Stock Unstable CCR2 79 47 O=C(NCCSC1CCOCC1)c1cccc(C(F)(F)F)c1 ZINC000217701602 EG In-Stock Unstable GPR52 0 42 CSC[C@](C)(O)CNC(=O)c1cc2ccccc2s1 ZINC000217701631 CF In-Stock Unstable PIN1 29 42 CCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCC ZINC000217701668 CD In-Stock Unstable NEU3 0 40 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(O)c(OC)c2)CC(=O)O4)cc1O ZINC000217701677 JI In-Stock Unstable ALOX5 0 52 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(O)c(OC)c2)CC(=O)O4)cc1O ZINC000217701677 JI In-Stock Unstable AKR1B1 25 55 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(O)c(OC)c2)CC(=O)O4)cc1O ZINC000217701677 JI In-Stock Unstable CYP1B1 70 39 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(O)c(OC)c2)CC(=O)O4)cc1O ZINC000217701677 JI In-Stock Unstable CYP1A1 53 50 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(O)c(OC)c2)CC(=O)O4)cc1O ZINC000217701677 JI In-Stock Unstable CYP1A2 42 43 O=C(NCCSC1CCOCC1)c1ccccc1C(F)(F)F ZINC000217701712 EG In-Stock Unstable RBP4 40 32 CSc1ccccc1N[C@@H](C)C(=O)NC1CCCCC1 ZINC000217701732 CH For-Sale Unstable EPHX2 23 42 CCOc1ccccc1/C=C\C(=O)N(C)[C@@H](CC)C(=O)O ZINC000217701754 CE For-Sale Unstable PTGER2 32 42 CCOc1ccccc1/C=C\C(=O)N(C)[C@@H](CC)C(=O)O ZINC000217701754 CE For-Sale Unstable PTGER4 17 42 CN1CCCN(S(=O)(=O)c2cccc(C(=O)N3CC[C@@H](CN)C3)c2)CC1 ZINC000217701773 GC In-Stock Unstable ST14 78 33 CN1CCCN(S(=O)(=O)c2cccc(C(=O)N3CC[C@@H](CN)C3)c2)CC1 ZINC000217701773 GC In-Stock Unstable AKR1C3 66 41 CN1CCCN(S(=O)(=O)c2cccc(C(=O)N3CC[C@@H](CN)C3)c2)CC1 ZINC000217701773 GC In-Stock Unstable TMPRSS6 53 33 CCCNS(=O)(=O)c1cc(C(=O)O)ccc1NC ZINC000217701774 CD In-Stock Unstable NEU3 0 40 C=C(C)COc1ccc([C@@H]2CC(=O)Oc3ccc4c(c32)OC(=C(C)C)C4=O)cc1OC ZINC000217701797 HJ In-Stock Unstable MT-ND4 41 32 CSc1ccccc1N[C@H](C)C(=O)NC1CCCCC1 ZINC000217701810 CH For-Sale Unstable EPHX2 23 42 CCOc1ccccc1/C=C\C(=O)N(C)[C@H](CC)C(=O)O ZINC000217701843 CE For-Sale Unstable PTGER2 32 42 CCOc1ccccc1/C=C\C(=O)N(C)[C@H](CC)C(=O)O ZINC000217701843 CE For-Sale Unstable PTGER4 17 42 COC(=O)[C@@H](O)CNC(=O)COc1ccccc1 ZINC000217701864 CB On-Demand Unstable ADRB3 27 41 COC(=O)[C@@H](O)CNC(=O)COc1ccccc1 ZINC000217701864 CB On-Demand Unstable PLA2G4B 56 35 COC(=O)[C@@H](O)CNC(=O)COc1ccccc1 ZINC000217701864 CB On-Demand Unstable PDS 40 37 C=C(C)COc1ccc([C@H]2CC(=O)Oc3ccc4c(c32)OC(=C(C)C)C4=O)cc1OC ZINC000217701878 HJ In-Stock Unstable MT-ND4 41 32 O=C(O)c1cc(O)n(-c2c(Cl)cccc2Cl)n1 ZINC000217701905 CF In-Stock Anodyne RPA1 90 44 O=C(/C=C/c1ccc2c(c1)OCO2)NCCSC1CCOCC1 ZINC000217701936 EE In-Stock Unstable PYGL 0 43 O=C(/C=C/c1ccc2c(c1)OCO2)NCCSC1CCOCC1 ZINC000217701936 EE In-Stock Unstable DYRK2 45 33 CCOC(=O)[C@@H](S[C@@H](C)CC)c1ccccc1 ZINC000217701942 CH For-Sale Unstable CAPN2 21 40 CCOC(=O)[C@@H](S[C@@H](C)CC)c1ccccc1 ZINC000217701942 CH For-Sale Unstable METAP2 0 41 COC(=O)[C@H](O)CNC(=O)COc1ccccc1 ZINC000217701944 CB On-Demand Unstable ADRB3 27 41 COC(=O)[C@H](O)CNC(=O)COc1ccccc1 ZINC000217701944 CB On-Demand Unstable PLA2G4B 56 35 COC(=O)[C@H](O)CNC(=O)COc1ccccc1 ZINC000217701944 CB On-Demand Unstable PDS 40 37 Cc1ccccc1/C=C/NC(=O)NC1CCN(C(=O)OC(C)(C)C)CC1 ZINC000217701956 FH For-Sale Unstable CCR8 55 35 Cc1ccccc1/C=C/NC(=O)NC1CCN(C(=O)OC(C)(C)C)CC1 ZINC000217701956 FH For-Sale Unstable GPR119 38 42 CCN(CCOC)C(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217702001 CD For-Sale Unstable ACKR3 49 34 CNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217702019 EE In-Stock Unstable CCR8 74 42 CNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217702019 EE In-Stock Unstable SFRP1 95 35 CNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217702019 EE In-Stock Unstable WNT3 77 35 CCOC(=O)[C@H](S[C@@H](C)CC)c1ccccc1 ZINC000217702023 CH For-Sale Unstable CAPN2 21 40 CCOC(=O)[C@H](S[C@@H](C)CC)c1ccccc1 ZINC000217702023 CH For-Sale Unstable METAP2 0 41 COc1cccc(/C=C\C(=O)NC[C@](C)(O)CC(=O)O)c1 ZINC000217702058 CD For-Sale Unstable MTNR1A 49 40 COc1cccc(/C=C\C(=O)NC[C@](C)(O)CC(=O)O)c1 ZINC000217702058 CD For-Sale Unstable MTNR1B 52 40 COc1cccc(/C=C\C(=O)NC[C@](C)(O)CC(=O)O)c1 ZINC000217702058 CD For-Sale Unstable MMP2 16 45 COC(=O)[C@@H](O)CNC(=O)c1cc(O)nc2ccccc12 ZINC000217702077 CC On-Demand Unstable TACR3 48 42 COc1ccccc1/C=C/NC(=O)Nc1ccc(OC)c(OC)c1 ZINC000217702089 EH For-Sale Unstable CYP1B1 34 40 COc1ccccc1/C=C/NC(=O)Nc1ccc(OC)c(OC)c1 ZINC000217702089 EH For-Sale Unstable CYP1A1 25 49 COc1ccccc1/C=C/NC(=O)Nc1ccc(OC)c(OC)c1 ZINC000217702089 EH For-Sale Unstable PDGFRA 44 36 COc1ccccc1/C=C/NC(=O)Nc1ccc(OC)c(OC)c1 ZINC000217702089 EH For-Sale Unstable IMPDH2 0 48 COc1ccccc1/C=C/NC(=O)Nc1ccc(OC)c(OC)c1 ZINC000217702089 EH For-Sale Unstable ENPP1 73 36 COc1ccccc1/C=C/NC(=O)Nc1ccc(OC)c(OC)c1 ZINC000217702089 EH For-Sale Unstable KCNK3 40 41 COc1ccccc1/C=C/NC(=O)Nc1ccc(OC)c(OC)c1 ZINC000217702089 EH For-Sale Unstable KCNK9 34 41 O=C(O)/C=C\c1cccc(C(=O)N2CCCC[C@@H]2CO)c1 ZINC000217702096 CD For-Sale Unstable HCRTR1 15 42 O=C(O)/C=C\c1cccc(C(=O)N2CCCC[C@@H]2CO)c1 ZINC000217702096 CD For-Sale Unstable PREP 41 44 CCOC(=O)[C@@H](S[C@H](C)CC)c1ccccc1 ZINC000217702109 CH For-Sale Unstable CAPN2 21 40 CCOC(=O)[C@@H](S[C@H](C)CC)c1ccccc1 ZINC000217702109 CH For-Sale Unstable METAP2 0 41 COc1cccc(/C=C\C(=O)NC[C@@](C)(O)CC(=O)O)c1 ZINC000217702129 CD For-Sale Unstable MTNR1A 49 40 COc1cccc(/C=C\C(=O)NC[C@@](C)(O)CC(=O)O)c1 ZINC000217702129 CD For-Sale Unstable MTNR1B 52 40 COc1cccc(/C=C\C(=O)NC[C@@](C)(O)CC(=O)O)c1 ZINC000217702129 CD For-Sale Unstable MMP2 16 45 C[C@H]1CCCC[C@H]1N[C@H](C)Cc1cccc(Cl)c1 ZINC000217702141 CI For-Sale Unstable CACNA1D 0 40 COC(=O)[C@H](O)CNC(=O)c1cc(O)nc2ccccc12 ZINC000217702158 CC On-Demand Unstable TACR3 48 42 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NC1CCCCC1 ZINC000217702161 EE In-Stock Unstable CCR8 87 48 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NC1CCCCC1 ZINC000217702161 EE In-Stock Unstable SFRP1 104 37 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NC1CCCCC1 ZINC000217702161 EE In-Stock Unstable WNT3 82 36 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NC1CCCCC1 ZINC000217702161 EE In-Stock Unstable BRD4 23 41 O=C(O)/C=C\c1cccc(C(=O)N2CCCC[C@H]2CO)c1 ZINC000217702180 CD For-Sale Unstable HCRTR1 15 42 O=C(O)/C=C\c1cccc(C(=O)N2CCCC[C@H]2CO)c1 ZINC000217702180 CD For-Sale Unstable PREP 41 44 COc1ccc([C@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1O ZINC000217702186 KH In-Stock Unstable CYP1B1 63 42 COc1ccc([C@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1O ZINC000217702186 KH In-Stock Unstable CYP1A1 49 42 COc1ccc([C@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1O ZINC000217702186 KH In-Stock Unstable CYP1A2 41 42 COc1ccc([C@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1O ZINC000217702186 KH In-Stock Unstable RORC 55 39 CCOC(=O)[C@H](S[C@H](C)CC)c1ccccc1 ZINC000217702194 CH For-Sale Unstable CAPN2 21 40 CCOC(=O)[C@H](S[C@H](C)CC)c1ccccc1 ZINC000217702194 CH For-Sale Unstable METAP2 0 41 COc1ccccc1/C=C/NC(=O)NCCCN1CCCC1=O ZINC000217702203 DD For-Sale Unstable DRD2 31 46 COc1ccccc1/C=C/NC(=O)NCCCN1CCCC1=O ZINC000217702203 DD For-Sale Unstable ADRA1D 23 41 COc1ccccc1/C=C/NC(=O)NCCCN1CCCC1=O ZINC000217702203 DD For-Sale Unstable ADRA1A 23 49 COc1ccccc1/C=C/NC(=O)NCCCN1CCCC1=O ZINC000217702203 DD For-Sale Unstable ADRA1B 15 40 COc1ccccc1/C=C/NC(=O)NCCCN1CCCC1=O ZINC000217702203 DD For-Sale Unstable DRD3 42 46 COc1ccccc1/C=C/NC(=O)NCCCN1CCCC1=O ZINC000217702203 DD For-Sale Unstable TYRO3 27 47 C[C@H]1CCCC[C@@H]1N[C@H](C)Cc1cccc(Cl)c1 ZINC000217702228 CI For-Sale Unstable CACNA1D 0 40 COC(=O)[C@@H](O)CNC(=O)Cc1cccc(OC)c1 ZINC000217702264 CB On-Demand Unstable DRD4 45 35 COC(=O)[C@@H](O)CNC(=O)Cc1cccc(OC)c1 ZINC000217702264 CB On-Demand Unstable ANPEP 25 46 COC(=O)[C@@H](O)CNC(=O)Cc1cccc(OC)c1 ZINC000217702264 CB On-Demand Unstable NQO2 23 40 COC(=O)[C@@H](O)CNC(=O)Cc1cccc(OC)c1 ZINC000217702264 CB On-Demand Unstable TRPV1 30 42 COC(=O)[C@@H](O)CNC(=O)Cc1cccc(OC)c1 ZINC000217702264 CB On-Demand Unstable MTNR1A 64 49 COC(=O)[C@@H](O)CNC(=O)Cc1cccc(OC)c1 ZINC000217702264 CB On-Demand Unstable MTNR1B 59 49 COC(=O)[C@@H](O)CNC(=O)Cc1cccc(OC)c1 ZINC000217702264 CB On-Demand Unstable ROCK2 43 37 COC(=O)[C@@H](O)CNC(=O)Cc1cccc(OC)c1 ZINC000217702264 CB On-Demand Unstable HSD17B2 25 41 COC(=O)[C@@H](O)CNC(=O)Cc1cccc(OC)c1 ZINC000217702264 CB On-Demand Unstable NCE103 20 51 COc1ccc([C@@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1O ZINC000217702265 KH In-Stock Unstable CYP1B1 63 42 COc1ccc([C@@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1O ZINC000217702265 KH In-Stock Unstable CYP1A1 49 42 COc1ccc([C@@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1O ZINC000217702265 KH In-Stock Unstable CYP1A2 41 42 COc1ccc([C@@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1O ZINC000217702265 KH In-Stock Unstable RORC 55 39 COc1ccccc1/C=C/NC(=O)Nc1ccc(Br)cc1 ZINC000217702297 EI For-Sale Unstable EPHX1 0 40 C[C@@H](CCN(C)C)NC(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217702304 CD For-Sale Unstable UTS2 41 33 COC(=O)[C@H](O)CNC(=O)Cc1cccc(OC)c1 ZINC000217702338 CB On-Demand Unstable DRD4 45 35 COC(=O)[C@H](O)CNC(=O)Cc1cccc(OC)c1 ZINC000217702338 CB On-Demand Unstable ANPEP 25 46 COC(=O)[C@H](O)CNC(=O)Cc1cccc(OC)c1 ZINC000217702338 CB On-Demand Unstable NQO2 23 40 COC(=O)[C@H](O)CNC(=O)Cc1cccc(OC)c1 ZINC000217702338 CB On-Demand Unstable TRPV1 30 42 COC(=O)[C@H](O)CNC(=O)Cc1cccc(OC)c1 ZINC000217702338 CB On-Demand Unstable MTNR1A 64 49 COC(=O)[C@H](O)CNC(=O)Cc1cccc(OC)c1 ZINC000217702338 CB On-Demand Unstable MTNR1B 59 49 COC(=O)[C@H](O)CNC(=O)Cc1cccc(OC)c1 ZINC000217702338 CB On-Demand Unstable ROCK2 43 37 COC(=O)[C@H](O)CNC(=O)Cc1cccc(OC)c1 ZINC000217702338 CB On-Demand Unstable HSD17B2 25 41 COC(=O)[C@H](O)CNC(=O)Cc1cccc(OC)c1 ZINC000217702338 CB On-Demand Unstable NCE103 20 51 CCOc1ccc(CC(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc1 ZINC000217702382 FE In-Stock Unstable CHRNA4 31 48 C[C@H](CCN(C)C)NC(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217702386 CD For-Sale Unstable UTS2 41 33 COc1ccccc1/C=C/NC(=O)Nc1cccc(C(=O)O)c1 ZINC000217702401 DG For-Sale Unstable PPIA 26 46 COc1ccccc1/C=C/NC(=O)Nc1cccc(C(=O)O)c1 ZINC000217702401 DG For-Sale Unstable CCKAR 25 42 COc1ccccc1/C=C/NC(=O)Nc1cccc(C(=O)O)c1 ZINC000217702401 DG For-Sale Unstable LTB4R 15 40 COc1ccccc1/C=C/NC(=O)Nc1cccc(C(=O)O)c1 ZINC000217702401 DG For-Sale Unstable CCKBR 23 42 COc1ccccc1/C=C/NC(=O)Nc1cccc(C(=O)O)c1 ZINC000217702401 DG For-Sale Unstable IMPDH2 0 42 COc1ccccc1/C=C/NC(=O)Nc1cccc(C(=O)O)c1 ZINC000217702401 DG For-Sale Unstable AKR1C3 48 49 COc1ccccc1/C=C/NC(=O)Nc1cccc(C(=O)O)c1 ZINC000217702401 DG For-Sale Unstable SMO 15 49 COc1ccccc1/C=C/NC(=O)Nc1cccc(C(=O)O)c1 ZINC000217702401 DG For-Sale Unstable KCNK3 115 49 COc1ccccc1/C=C/NC(=O)Nc1cccc(C(=O)O)c1 ZINC000217702401 DG For-Sale Unstable KCNK9 82 45 CNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217702449 GD In-Stock Unstable TBXA2R 55 43 CNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217702449 GD In-Stock Unstable TBXAS1 27 47 CNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217702449 GD In-Stock Unstable IAP 0 47 CNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217702449 GD In-Stock Unstable AKR1C3 18 48 CNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217702449 GD In-Stock Unstable SCMU_MYCTU 0 43 C[C@@H](CCN(C)C)NC(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217702488 CD For-Sale Unstable UTS2 80 44 COc1ccc2c(O)c(C(=O)N3CCc4cc(OC)c(OC)cc4C3)cnc2c1 ZINC000217702492 GG In-Stock Unstable PDGFRB 42 36 COc1ccc2c(O)c(C(=O)N3CCc4cc(OC)c(OC)cc4C3)cnc2c1 ZINC000217702492 GG In-Stock Unstable ABCB1B 59 35 COc1ccc2c(O)c(C(=O)N3CCc4cc(OC)c(OC)cc4C3)cnc2c1 ZINC000217702492 GG In-Stock Unstable ABCB1 26 51 COc1ccc2c(O)c(C(=O)N3CCc4cc(OC)c(OC)cc4C3)cnc2c1 ZINC000217702492 GG In-Stock Unstable CSF1R 47 39 COc1ccccc1/C=C/NC(=O)Nc1ccccc1[N+](=O)[O-] ZINC000217702506 DG For-Sale Unstable TLR4 17 45 C[C@H](CCN(C)C)NC(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217702558 CD For-Sale Unstable UTS2 80 44 C[C@H]1CCC[C@H](C)C1N[C@H](C)Cc1cccc(Cl)c1 ZINC000217702567 CJ For-Sale Unstable CACNA1D 28 41 CCCCCNS(=O)(=O)c1ccc(NC)c(C(=O)O)c1 ZINC000217702576 DD In-Stock Unstable CASP3 17 46 CSC[C@@](C)(O)CNC(=O)/C=C/c1ccc(F)c(Cl)c1 ZINC000217702586 DF On-Demand Unstable PYGL 25 46 CCOC(=O)[C@@H](SC1CCCCC1)c1ccccc1 ZINC000217702625 CI On-Demand Unstable CHRM1 18 40 CCOC(=O)[C@@H](SC1CCCCC1)c1ccccc1 ZINC000217702625 CI On-Demand Unstable AMY2 54 38 CN(CC1CCOCC1)C(=O)c1ccc2[nH]c(=O)c(=O)[nH]c2c1 ZINC000217702633 DC In-Stock Unstable WNT3A 40 34 COc1ccccc1/C=C/NC(=O)Nc1cccc(O)c1 ZINC000217702637 CG For-Sale Unstable IMPDH2 0 42 COc1ccccc1/C=C/NC(=O)Nc1cccc(O)c1 ZINC000217702637 CG For-Sale Unstable KCNK3 76 45 COc1ccccc1/C=C/NC(=O)Nc1cccc(O)c1 ZINC000217702637 CG For-Sale Unstable KCNK9 64 45 C[C@H]1CCC[C@@H](C)C1N[C@H](C)Cc1cccc(Cl)c1 ZINC000217702641 CJ For-Sale Unstable CACNA1D 28 41 CSC[C@](C)(O)CNC(=O)/C=C/c1ccc(F)c(Cl)c1 ZINC000217702645 DF On-Demand Unstable PYGL 25 46 CCCCCN[C@@H](CC)CCO ZINC000217702654 AD For-Sale Unstable Q6UB75_PIG 0 44 CCOC(=O)[C@H](SC1CCCCC1)c1ccccc1 ZINC000217702692 CI On-Demand Unstable CHRM1 18 40 CCOC(=O)[C@H](SC1CCCCC1)c1ccccc1 ZINC000217702692 CI On-Demand Unstable AMY2 54 38 COC(=O)[C@@H](O)CNC(=O)CCc1cccnc1 ZINC000217702707 CB On-Demand Unstable TBXAS1 33 43 COC(=O)[C@@H](O)CNC(=O)CCc1cccnc1 ZINC000217702707 CB On-Demand Unstable PTAFR 36 41 COC(=O)[C@@H](O)CNC(=O)CCc1cccnc1 ZINC000217702707 CB On-Demand Unstable C3AR1 42 39 COC(=O)[C@@H](O)CNC(=O)CCc1cccnc1 ZINC000217702707 CB On-Demand Unstable NAMPT 23 45 CCCCCN[C@H](CC)CCO ZINC000217702724 AD For-Sale Unstable Q6UB75_PIG 0 44 COc1ccccc1/C=C/NC(=O)Nc1ccc(C)cc1 ZINC000217702736 CH For-Sale Unstable PDGFRA 40 34 COc1ccccc1/C=C/NC(=O)Nc1ccc(C)cc1 ZINC000217702736 CH For-Sale Unstable KCNK3 39 40 COc1ccccc1/C=C/NC(=O)Nc1ccc(C)cc1 ZINC000217702736 CH For-Sale Unstable KCNK9 38 40 CC(C)[C@H]1CC[C@H](C)C[C@H]1N[C@H](C)Cc1cccc(Cl)c1 ZINC000217702753 DK For-Sale Unstable TRPM8 18 55 COC(=O)[C@H](O)CNC(=O)CCc1cccnc1 ZINC000217702785 CB For-Sale Unstable TBXAS1 44 40 COC(=O)[C@H](O)CNC(=O)CCc1cccnc1 ZINC000217702785 CB For-Sale Unstable PTAFR 36 42 COC(=O)[C@H](O)CNC(=O)CCc1cccnc1 ZINC000217702785 CB For-Sale Unstable KCNA5 15 48 COC(=O)[C@H](O)CNC(=O)CCc1cccnc1 ZINC000217702785 CB For-Sale Unstable NAMPT 28 45 COc1cccc(C(=O)NCCC(=O)NC2Cc3ccccc3C2)c1 ZINC000217702824 EE In-Stock Unstable DRD2 16 50 COc1cccc(C(=O)NCCC(=O)NC2Cc3ccccc3C2)c1 ZINC000217702824 EE In-Stock Unstable DRD4 63 50 COc1cccc(C(=O)NCCC(=O)NC2Cc3ccccc3C2)c1 ZINC000217702824 EE In-Stock Unstable DRD3 22 48 COc1cccc(C(=O)NCCC(=O)NC2Cc3ccccc3C2)c1 ZINC000217702824 EE In-Stock Unstable MTNR1A 58 44 COc1cccc(C(=O)NCCC(=O)NC2Cc3ccccc3C2)c1 ZINC000217702824 EE In-Stock Unstable MTNR1B 52 43 COc1cccc(C(=O)NCCC(=O)NC2Cc3ccccc3C2)c1 ZINC000217702824 EE In-Stock Unstable MCHR1 18 46 COc1cccc(C(=O)NCCC(=O)NC2Cc3ccccc3C2)c1 ZINC000217702824 EE In-Stock Unstable LGALS1 0 42 COc1cccc(C(=O)NCCC(=O)NC2Cc3ccccc3C2)c1 ZINC000217702824 EE In-Stock Unstable LGALS9 0 42 COc1cccc(C(=O)NCCC(=O)NC2Cc3ccccc3C2)c1 ZINC000217702824 EE In-Stock Unstable ALPHA-1A 0 40 Cc1c(-n2nc(C(=O)O)cc2O)cccc1[N+](=O)[O-] ZINC000217702825 CD In-Stock Unstable RPA1 64 39 CCCCN[C@@H](CC)CCO ZINC000217702838 AD On-Demand Unstable Q6UB75_PIG 0 41 CC(C)[C@H]1CC[C@H](C)C[C@@H]1N[C@@H](C)Cc1cccc(Cl)c1 ZINC000217702842 DK For-Sale Unstable TRPM8 18 55 COc1ccccc1/C=C/NC(=O)NCCC(=O)O ZINC000217702851 CD For-Sale Unstable MTNR1B 23 42 O=C(NCCc1ccc(Cl)cc1Cl)c1ccc(Cl)cc1 ZINC000217702873 EJ For-Sale Unstable CNR1 47 52 O=C(NCCc1ccc(Cl)cc1Cl)c1ccc(Cl)cc1 ZINC000217702873 EJ For-Sale Unstable F10 22 45 O=C(NCCc1ccc(Cl)cc1Cl)c1ccc(Cl)cc1 ZINC000217702873 EJ For-Sale Unstable CNR2 20 47 O=C(NCCc1ccc(Cl)cc1Cl)c1ccc(Cl)cc1 ZINC000217702873 EJ For-Sale Unstable MC4R 22 52 O=C(NCCc1ccc(Cl)cc1Cl)c1ccc(Cl)cc1 ZINC000217702873 EJ For-Sale Unstable P2RX7 37 43 O=C(NCCc1ccc(Cl)cc1Cl)c1ccc(Cl)cc1 ZINC000217702873 EJ For-Sale Unstable MC5R 29 54 O=C(NCCc1ccc(Cl)cc1Cl)c1ccc(Cl)cc1 ZINC000217702873 EJ For-Sale Unstable EPHX2 21 52 O=C(NCCc1ccc(Cl)cc1Cl)c1ccc(Cl)cc1 ZINC000217702873 EJ For-Sale Unstable MC1R 26 54 O=C(NCCc1ccc(Cl)cc1Cl)c1ccc(Cl)cc1 ZINC000217702873 EJ For-Sale Unstable SCN10A 36 40 O=C(NCCc1ccc(Cl)cc1Cl)c1ccc(Cl)cc1 ZINC000217702873 EJ For-Sale Unstable PTGDR 23 41 O=C(NCCc1ccc(Cl)cc1Cl)c1ccc(Cl)cc1 ZINC000217702873 EJ For-Sale Unstable ALPL 61 41 O=C(NCCc1ccc(Cl)cc1Cl)c1ccc(Cl)cc1 ZINC000217702873 EJ For-Sale Unstable CXCR3 25 47 O=C(NCCc1ccc(Cl)cc1Cl)c1ccc(Cl)cc1 ZINC000217702873 EJ For-Sale Unstable PTGDR2 15 43 O=C(NCCc1ccc(Cl)cc1Cl)c1ccc(Cl)cc1 ZINC000217702873 EJ For-Sale Unstable UTS2 44 35 O=C(NCCc1ccc(Cl)cc1Cl)c1ccc(Cl)cc1 ZINC000217702873 EJ For-Sale Unstable MAPT 18 42 Cc1onc(-c2ccccc2Cl)c1C(=O)NCCSC1CCOCC1 ZINC000217702909 GH In-Stock Unstable GHSR 0 50 Cc1onc(-c2ccccc2Cl)c1C(=O)NCCSC1CCOCC1 ZINC000217702909 GH In-Stock Unstable GPBAR1 39 47 CC(C)[C@H]1CC[C@H](C)C[C@@H]1N[C@H](C)Cc1cccc(Cl)c1 ZINC000217702925 DK For-Sale Unstable TRPM8 18 55 CCCCN[C@H](CC)CCO ZINC000217702935 AD On-Demand Unstable Q6UB75_PIG 0 41 O=C(O)c1cc(O)n(-c2ccc(Br)cc2F)n1 ZINC000217702944 DE In-Stock Anodyne RPA1 66 39 O=C(CCCn1nnc(-c2ccc(F)cc2)n1)N[C@@H]1CCS(=O)(=O)C1 ZINC000217702948 FC In-Stock Unstable SCARB1 39 42 COc1ccccc1/C=C/NC(=O)Nc1ccc(N)cc1 ZINC000217702965 CG For-Sale Unstable CA12 15 42 COc1ccccc1/C=C/NC(=O)Nc1ccc(N)cc1 ZINC000217702965 CG For-Sale Unstable PDGFRA 43 36 COc1ccccc1/C=C/NC(=O)Nc1ccc(N)cc1 ZINC000217702965 CG For-Sale Unstable P96878_MYCTU 16 43 COc1ccc(N2C(=O)[C@H]3[C@H]4C[C@@H]([C@@H]5ON=C(c6ccc(Cl)cc6Cl)[C@@H]45)[C@H]3C2=O)cc1 ZINC000217702985 JI In-Stock Unstable DPP4 0 45 COc1ccc(N2C(=O)[C@H]3[C@H]4C[C@@H]([C@@H]5ON=C(c6ccc(Cl)cc6Cl)[C@@H]45)[C@H]3C2=O)cc1 ZINC000217702985 JI In-Stock Unstable DPP8 32 45 COc1ccc(N2C(=O)[C@H]3[C@H]4C[C@@H]([C@@H]5ON=C(c6ccc(Cl)cc6Cl)[C@@H]45)[C@H]3C2=O)cc1 ZINC000217702985 JI In-Stock Unstable DPP9 44 45 O=C(CCCn1nnc(-c2ccc(F)cc2)n1)N[C@H]1CCS(=O)(=O)C1 ZINC000217703029 FC In-Stock Unstable SCARB1 39 42 O=C(NCCSC1CCOCC1)c1cc(C2CC2)on1 ZINC000217703030 CE In-Stock Unstable S1PR3 0 50 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NCC ZINC000217703076 CD In-Stock Unstable NEU3 0 43 c1cc(CN[C@@H]2CCN3CCC[C@@H]23)c2c(c1)OCCCO2 ZINC000217703095 CE For-Sale Unstable HTR1B 15 40 O=C(NCCSC1CCOCC1)c1ccc(OC(F)(F)F)cc1 ZINC000217703145 EG In-Stock Unstable GCGR 39 42 O=C(NCCSC1CCOCC1)c1ccc(OC(F)(F)F)cc1 ZINC000217703145 EG In-Stock Unstable TRPV1 0 52 O=C(NCCSC1CCOCC1)c1ccc(OC(F)(F)F)cc1 ZINC000217703145 EG In-Stock Unstable GIPR 47 38 CCN(CC)S(=O)(=O)c1ccc(/C=C\C(=O)O)cc1Cl ZINC000217703171 DE For-Sale Unstable NR0B2 0 44 c1cc(CN[C@H]2CCN3CCC[C@@H]23)c2c(c1)OCCCO2 ZINC000217703174 CE For-Sale Unstable HTR1B 15 40 COc1ccccc1/C=C/NC(=O)Nc1ccc(NC(C)=O)cc1 ZINC000217703194 EG For-Sale Unstable CYP1B1 17 41 COc1ccccc1/C=C/NC(=O)Nc1ccc(NC(C)=O)cc1 ZINC000217703194 EG For-Sale Unstable MTNR1B 16 46 COc1ccccc1/C=C/NC(=O)Nc1ccc(NC(C)=O)cc1 ZINC000217703194 EG For-Sale Unstable CYP1A1 15 41 COc1ccccc1/C=C/NC(=O)Nc1ccc(NC(C)=O)cc1 ZINC000217703194 EG For-Sale Unstable PDGFRA 40 35 COc1ccccc1/C=C/NC(=O)Nc1ccc(NC(C)=O)cc1 ZINC000217703194 EG For-Sale Unstable IMPDH2 0 43 COc1ccccc1/C=C/NC(=O)Nc1ccc(NC(C)=O)cc1 ZINC000217703194 EG For-Sale Unstable TLR4 15 44 CNc1ccc(C(=O)O)cc1S(=O)(=O)NCCc1ccc(OC)c(OC)c1 ZINC000217703200 GD In-Stock Unstable TBXA2R 43 38 CNc1ccc(C(=O)O)cc1S(=O)(=O)NCCc1ccc(OC)c(OC)c1 ZINC000217703200 GD In-Stock Unstable PTGDR 25 45 CNc1ccc(C(=O)O)cc1S(=O)(=O)NCCc1ccc(OC)c(OC)c1 ZINC000217703200 GD In-Stock Unstable MT-ND1 25 40 CNc1ccc(C(=O)O)cc1S(=O)(=O)NCCc1ccc(OC)c(OC)c1 ZINC000217703200 GD In-Stock Unstable AKR1C3 17 48 CNc1ccc(C(=O)O)cc1S(=O)(=O)NCCc1ccc(OC)c(OC)c1 ZINC000217703200 GD In-Stock Unstable SCMU_MYCTU 0 50 COc1ccccc1/C=C/NC(=O)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217703288 EF For-Sale Unstable LPL 41 32 COc1ccccc1/C=C/NC(=O)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217703288 EF For-Sale Unstable CA1 48 37 COc1ccccc1/C=C/NC(=O)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217703288 EF For-Sale Unstable P96878_MYCTU 45 37 COC(=O)c1coc(CCNC(=O)OC(C)(C)C)c1 ZINC000217703298 CE In-Stock Unstable NQO2 23 42 O=C(O)c1cc(O)n(-c2ccc3c(c2)OCCO3)n1 ZINC000217703325 CD In-Stock Unstable DHRS9 0 46 O=C(O)c1cc(O)n(-c2ccc3c(c2)OCCO3)n1 ZINC000217703325 CD In-Stock Unstable RPA1 75 42 CCC(CC)NS(=O)(=O)c1ccc(/C=C\C(=O)O)cc1Cl ZINC000217703331 EF For-Sale Unstable NR0B2 0 42 CCOC(=O)[C@@H](SC1CCCC1)c1ccccc1 ZINC000217703362 CH On-Demand Unstable CHRM1 15 40 CCOC(=O)[C@@H](SC1CCCC1)c1ccccc1 ZINC000217703362 CH On-Demand Unstable SLC6A3 15 40 CCOC(=O)[C@@H](SC1CCCC1)c1ccccc1 ZINC000217703362 CH On-Demand Unstable AMY2 51 36 CN1CCN([C@@H]2CCN(C(=O)c3ccsc3)C2)CC1 ZINC000217703387 CD In-Stock Unstable L3MBTL1 0 53 CN1CCN([C@@H]2CCN(C(=O)c3ccsc3)C2)CC1 ZINC000217703387 CD In-Stock Unstable L3MBTL3 85 53 CN1CCN([C@@H]2CCN(C(=O)c3ccsc3)C2)CC1 ZINC000217703387 CD In-Stock Unstable MBTD1 0 43 COc1ccccc1/C=C/NC(=O)Nc1cccc(S(=O)(=O)O)c1 ZINC000217703398 EF For-Sale Unstable KCNK3 47 42 COc1ccccc1/C=C/NC(=O)Nc1cccc(S(=O)(=O)O)c1 ZINC000217703398 EF For-Sale Unstable KCNK9 52 42 C[C@H]1C[C@H]1c1ccc(CN[C@H](C)Cc2cccc(Cl)c2)o1 ZINC000217703418 DJ For-Sale Unstable LMGT2 0 40 CCC(CC)NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217703421 CE For-Sale Unstable HDAC8 22 48 CCOC(=O)[C@H](SC1CCCC1)c1ccccc1 ZINC000217703441 CH On-Demand Unstable CHRM1 15 40 CCOC(=O)[C@H](SC1CCCC1)c1ccccc1 ZINC000217703441 CH On-Demand Unstable SLC6A3 15 40 CCOC(=O)[C@H](SC1CCCC1)c1ccccc1 ZINC000217703441 CH On-Demand Unstable AMY2 51 36 CCOc1ccccc1-n1nc(C(=O)O)cc1O ZINC000217703454 BD In-Stock Unstable HIF1A 18 41 CCOc1ccccc1-n1nc(C(=O)O)cc1O ZINC000217703454 BD In-Stock Unstable CTSA 42 39 CCOc1ccccc1-n1nc(C(=O)O)cc1O ZINC000217703454 BD In-Stock Unstable HCN1 42 32 CCOc1ccccc1-n1nc(C(=O)O)cc1O ZINC000217703454 BD In-Stock Unstable HCN4 42 32 CCOc1ccccc1-n1nc(C(=O)O)cc1O ZINC000217703454 BD In-Stock Unstable RPA1 65 39 CN1CCN([C@H]2CCN(C(=O)c3ccsc3)C2)CC1 ZINC000217703463 CD In-Stock Unstable L3MBTL1 0 53 CN1CCN([C@H]2CCN(C(=O)c3ccsc3)C2)CC1 ZINC000217703463 CD In-Stock Unstable L3MBTL3 85 53 CN1CCN([C@H]2CCN(C(=O)c3ccsc3)C2)CC1 ZINC000217703463 CD In-Stock Unstable MBTD1 0 43 C[C@H]1C[C@@H]1c1ccc(CN[C@H](C)Cc2cccc(Cl)c2)o1 ZINC000217703491 DJ For-Sale Unstable LMGT2 0 40 CCC(CC)NS(=O)(=O)c1ccc(/C=C\C(=O)O)c(C)c1 ZINC000217703510 DF For-Sale Unstable LEF 63 44 CC(C)C[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(Cc2ccc3c(c2)OCO3)C1=O ZINC000217703529 GC In-Stock Unstable NPY1R 23 41 CC(C)C[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(Cc2ccc3c(c2)OCO3)C1=O ZINC000217703529 GC In-Stock Unstable NOS2 45 34 CC(C)C[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(Cc2ccc3c(c2)OCO3)C1=O ZINC000217703529 GC In-Stock Unstable SSTR3 97 33 CC(C)C[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(Cc2ccc3c(c2)OCO3)C1=O ZINC000217703529 GC In-Stock Unstable MCHR1 22 40 CNc1ccc(C(=O)O)cc1S(=O)(=O)NC1CCCCCC1 ZINC000217703581 EE In-Stock Unstable CCR8 84 50 CNc1ccc(C(=O)O)cc1S(=O)(=O)NC1CCCCCC1 ZINC000217703581 EE In-Stock Unstable SFRP1 105 38 CNc1ccc(C(=O)O)cc1S(=O)(=O)NC1CCCCCC1 ZINC000217703581 EE In-Stock Unstable WNT3 82 37 CNc1ccc(C(=O)O)cc1S(=O)(=O)NC1CCCCCC1 ZINC000217703581 EE In-Stock Unstable BRD4 25 41 Cc1csc(NS(=O)(=O)c2cccc(/C=C\C(=O)O)c2)n1 ZINC000217703597 DE For-Sale Unstable HDAC8 43 48 Cc1csc(NS(=O)(=O)c2cccc(/C=C\C(=O)O)c2)n1 ZINC000217703597 DE For-Sale Unstable HDAC1 15 48 Cc1csc(NS(=O)(=O)c2cccc(/C=C\C(=O)O)c2)n1 ZINC000217703597 DE For-Sale Unstable HDAC6 19 48 CCOC(=O)[C@@H](SCC(C)C)c1ccccc1 ZINC000217703606 CH On-Demand Unstable CAPN2 53 34 CCCNC(=O)N/C=C/c1ccccc1OC ZINC000217703610 BE For-Sale Unstable DRD3 18 42 CCCNC(=O)N/C=C/c1ccccc1OC ZINC000217703610 BE For-Sale Unstable CYP1B1 19 40 CCCNC(=O)N/C=C/c1ccccc1OC ZINC000217703610 BE For-Sale Unstable MTNR1A 19 51 CCCNC(=O)N/C=C/c1ccccc1OC ZINC000217703610 BE For-Sale Unstable MTNR1B 23 47 CCCNC(=O)N/C=C/c1ccccc1OC ZINC000217703610 BE For-Sale Unstable TLR4 19 45 O=C(NCCc1cc(C(=O)O)co1)OCc1ccccc1 ZINC000217703639 CE In-Stock Unstable TYR 37 40 O=C(NCCc1cc(C(=O)O)co1)OCc1ccccc1 ZINC000217703639 CE In-Stock Unstable PAPA1_CARPA 41 32 O=C(NCCc1cc(C(=O)O)co1)OCc1ccccc1 ZINC000217703639 CE In-Stock Unstable CAPNS1 52 35 O=C(NCCc1cc(C(=O)O)co1)OCc1ccccc1 ZINC000217703639 CE In-Stock Unstable CAPN1 53 37 O=C(NCCc1cc(C(=O)O)co1)OCc1ccccc1 ZINC000217703639 CE In-Stock Unstable CAPN2 90 37 O=C(NCCc1cc(C(=O)O)co1)OCc1ccccc1 ZINC000217703639 CE In-Stock Unstable NPR 62 37 CCOC(=O)c1c[nH]c(=O)c2c1OC(=O)C[C@@H]2c1cccc(O)c1 ZINC000217703648 ED In-Stock Unstable KIF11 0 43 Clc1cccc(CN[C@@H]2CCN3CCC[C@@H]23)c1Cl ZINC000217703649 CG For-Sale Unstable P2RX7 18 44 COC(=O)[C@@H](O)CNC(=O)c1ccoc1 ZINC000217703656 BB On-Demand Unstable ITGAV 39 48 COC(=O)[C@@H](O)CNC(=O)c1ccoc1 ZINC000217703656 BB On-Demand Unstable ITGA2 0 45 CCOC(=O)[C@H](SCC(C)C)c1ccccc1 ZINC000217703680 CH On-Demand Unstable CAPN2 53 34 CCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NC ZINC000217703688 CD In-Stock Unstable PLA2G4B 40 34 COc1ccccc1/C=C/NC(=O)Nc1ccc(C(C)C)cc1 ZINC000217703722 DJ For-Sale Unstable CA1 18 42 COc1ccccc1/C=C/NC(=O)Nc1ccc(C(C)C)cc1 ZINC000217703722 DJ For-Sale Unstable PDGFRA 42 35 Clc1cccc(CN[C@H]2CCN3CCC[C@@H]23)c1Cl ZINC000217703725 CG For-Sale Unstable P2RX7 18 44 CC(C)(C)OC(=O)N[C@@H](C[C@H](F)C(N)=O)C(=O)O ZINC000217703727 CC For-Sale Unstable PAPA1_CARPA 38 42 CC(C)(C)OC(=O)N[C@@H](C[C@H](F)C(N)=O)C(=O)O ZINC000217703727 CC For-Sale Unstable CTSK 18 45 CC(C)(C)OC(=O)N[C@@H](C[C@H](F)C(N)=O)C(=O)O ZINC000217703727 CC For-Sale Unstable POLG_HCV1 26 44 CC(C)(C)OC(=O)N[C@@H](C[C@H](F)C(N)=O)C(=O)O ZINC000217703727 CC For-Sale Unstable FPR1 51 40 CCOC(=O)c1c[nH]c(=O)c2c1OC(=O)C[C@H]2c1cccc(O)c1 ZINC000217703740 ED In-Stock Unstable KIF11 0 43 COC(=O)[C@H](O)CNC(=O)c1ccoc1 ZINC000217703748 BB On-Demand Unstable ITGAV 39 48 COC(=O)[C@H](O)CNC(=O)c1ccoc1 ZINC000217703748 BB On-Demand Unstable ITGA2 0 45 COC(=O)c1coc(CCNC(=O)OCc2ccccc2)c1 ZINC000217703754 DF In-Stock Unstable CTSB 36 40 COC(=O)c1coc(CCNC(=O)OCc2ccccc2)c1 ZINC000217703754 DF In-Stock Unstable PAPA1_CARPA 43 33 COC(=O)c1coc(CCNC(=O)OCc2ccccc2)c1 ZINC000217703754 DF In-Stock Unstable CTSK 20 40 COC(=O)c1coc(CCNC(=O)OCc2ccccc2)c1 ZINC000217703754 DF In-Stock Unstable CAPNS1 55 36 COC(=O)c1coc(CCNC(=O)OCc2ccccc2)c1 ZINC000217703754 DF In-Stock Unstable CAPN1 59 38 COC(=O)c1coc(CCNC(=O)OCc2ccccc2)c1 ZINC000217703754 DF In-Stock Unstable CAPN2 95 38 COC(=O)c1coc(CCNC(=O)OCc2ccccc2)c1 ZINC000217703754 DF In-Stock Unstable POL 0 40 COC(=O)c1coc(CCNC(=O)OCc2ccccc2)c1 ZINC000217703754 DF In-Stock Unstable NPR 63 38 O=C(NCc1ccccc1)N1C[C@@H]2CC[C@H](C1)O2 ZINC000217703796 BD On-Demand Unstable PREP 16 43 O=C(NCc1ccccc1)N1C[C@@H]2CC[C@H](C1)O2 ZINC000217703796 BD On-Demand Unstable TPSAB1 18 42 O=C(NCc1ccccc1)N1C[C@@H]2CC[C@H](C1)O2 ZINC000217703796 BD On-Demand Unstable NPSR1 30 49 O=C(NCc1ccccc1)N1C[C@@H]2CC[C@H](C1)O2 ZINC000217703796 BD On-Demand Unstable NAMPT 32 45 CNc1ccc(C(=O)O)cc1S(=O)(=O)NC1CCCC1 ZINC000217703797 CD In-Stock Unstable CCR8 85 48 CNc1ccc(C(=O)O)cc1S(=O)(=O)NC1CCCC1 ZINC000217703797 CD In-Stock Unstable SFRP1 106 39 CNc1ccc(C(=O)O)cc1S(=O)(=O)NC1CCCC1 ZINC000217703797 CD In-Stock Unstable WNT3 83 37 CNc1ccc(C(=O)O)cc1S(=O)(=O)NC1CCCC1 ZINC000217703797 CD In-Stock Unstable BRD4 26 42 CC(C)(C)OC(=O)N[C@H](C[C@H](F)C(N)=O)C(=O)O ZINC000217703808 CC For-Sale Unstable PAPA1_CARPA 38 42 CC(C)(C)OC(=O)N[C@H](C[C@H](F)C(N)=O)C(=O)O ZINC000217703808 CC For-Sale Unstable CTSK 18 45 CC(C)(C)OC(=O)N[C@H](C[C@H](F)C(N)=O)C(=O)O ZINC000217703808 CC For-Sale Unstable POLG_HCV1 26 44 CC(C)(C)OC(=O)N[C@H](C[C@H](F)C(N)=O)C(=O)O ZINC000217703808 CC For-Sale Unstable FPR1 51 40 CC[C@H](C(=O)O)N(C)C(=O)/C=C\c1ccc(Cl)c(Cl)c1 ZINC000217703821 DG For-Sale Unstable PYGL 0 45 COc1ccccc1/C=C/NC(=O)Nc1ccccc1OC ZINC000217703825 CG For-Sale Unstable CYP1B1 22 41 COc1ccccc1/C=C/NC(=O)Nc1ccccc1OC ZINC000217703825 CG For-Sale Unstable TLR4 19 47 CCC[C@@H]1CC[C@@H](NC)[C@@H](CCCc2ccccc2)C1 ZINC000217703844 CJ For-Sale Unstable SLC18A2 32 41 CC(C)(C)OC(=O)N[C@H](C[C@@H](F)C(N)=O)C(=O)O ZINC000217703899 CC For-Sale Unstable PAPA1_CARPA 38 42 CC(C)(C)OC(=O)N[C@H](C[C@@H](F)C(N)=O)C(=O)O ZINC000217703899 CC For-Sale Unstable CTSK 18 45 CC(C)(C)OC(=O)N[C@H](C[C@@H](F)C(N)=O)C(=O)O ZINC000217703899 CC For-Sale Unstable POLG_HCV1 26 44 CC(C)(C)OC(=O)N[C@H](C[C@@H](F)C(N)=O)C(=O)O ZINC000217703899 CC For-Sale Unstable FPR1 51 40 CNc1ccc(C(=O)O)cc1S(=O)(=O)NCCc1ccc(OC)cc1 ZINC000217703914 FD In-Stock Unstable TBXA2R 45 45 CNc1ccc(C(=O)O)cc1S(=O)(=O)NCCc1ccc(OC)cc1 ZINC000217703914 FD In-Stock Unstable TBXAS1 15 42 CNc1ccc(C(=O)O)cc1S(=O)(=O)NCCc1ccc(OC)cc1 ZINC000217703914 FD In-Stock Unstable MMP13 22 40 CNc1ccc(C(=O)O)cc1S(=O)(=O)NCCc1ccc(OC)cc1 ZINC000217703914 FD In-Stock Unstable CA9 17 41 CNc1ccc(C(=O)O)cc1S(=O)(=O)NCCc1ccc(OC)cc1 ZINC000217703914 FD In-Stock Unstable AKR1C3 36 52 CC[C@@H](C(=O)O)N(C)C(=O)/C=C\c1ccc(Cl)c(Cl)c1 ZINC000217703918 DG For-Sale Unstable PYGL 0 45 CCC[C@H]1CC[C@@H](NC)[C@@H](CCCc2ccccc2)C1 ZINC000217703930 CJ For-Sale Unstable SLC18A2 32 41 CCC[C@@H]1CC[C@H](NC)[C@@H](CCCc2ccccc2)C1 ZINC000217704027 CJ For-Sale Unstable SLC18A2 32 41 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NC ZINC000217704030 DD In-Stock Unstable PLA2G4B 43 36 CCN(CC(C)C)C(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217704033 CF For-Sale Unstable OPRM1 0 42 CCN(CC(C)C)C(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217704033 CF For-Sale Unstable OPRD1 30 43 CCN(CC(C)C)C(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217704033 CF For-Sale Unstable MLYCD 17 44 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217704044 EJ For-Sale Unstable GRM4 35 46 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217704044 EJ For-Sale Unstable PDGFRA 43 35 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217704044 EJ For-Sale Unstable IMPDH2 0 46 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217704044 EJ For-Sale Unstable IMDH_CRYPV 46 41 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217704044 EJ For-Sale Unstable BLM 0 40 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217704044 EJ For-Sale Unstable P95276_MYCTO 0 45 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217704044 EJ For-Sale Unstable CYSP_PLAFA 42 34 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217704044 EJ For-Sale Unstable PPX1 0 41 CCC[C@H]1CC[C@H](NC)[C@@H](CCCc2ccccc2)C1 ZINC000217704105 CJ For-Sale Unstable SLC18A2 32 41 O=C(CCc1ccc(Cl)c(C(F)(F)F)c1)NCCSC1CCOCC1 ZINC000217704125 GI In-Stock Unstable LUXR 40 36 CCN(CC(C)C)C(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217704128 CF For-Sale Unstable OPRM1 0 40 CCN(CC(C)C)C(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217704128 CF For-Sale Unstable OPRD1 29 40 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NCCO ZINC000217704154 CC In-Stock Unstable NEU3 0 40 COc1ccccc1/C=C/NC(=O)Nc1ccc(C)c(Cl)c1 ZINC000217704169 DI For-Sale Unstable GRM4 22 42 COc1ccccc1/C=C/NC(=O)Nc1ccc(C)c(Cl)c1 ZINC000217704169 DI For-Sale Unstable IMPDH2 0 42 COc1ccccc1/C=C/NC(=O)Nc1ccc(C)c(Cl)c1 ZINC000217704169 DI For-Sale Unstable KCNK3 43 37 COc1cc2c(cc1OC)[C@@H](c1cccnc1)N(C(=O)c1cc[nH]n1)CC2 ZINC000217704170 FF In-Stock Unstable MTNR1B 20 40 O=C(Cl)/C=C/c1cccc(OCc2ccc(Cl)cc2)c1 ZINC000217704206 DJ In-Stock Unstable MAOB 53 42 O=C(Cl)/C=C/c1cccc(OCc2ccc(Cl)cc2)c1 ZINC000217704206 DJ In-Stock Unstable PTGER2 0 42 O=C(Cl)/C=C/c1cccc(OCc2ccc(Cl)cc2)c1 ZINC000217704206 DJ In-Stock Unstable PTPN2 0 40 O=C(Cl)/C=C/c1cccc(OCc2ccc(Cl)cc2)c1 ZINC000217704206 DJ In-Stock Unstable CDC25B 0 42 O=C(Cl)/C=C/c1cccc(OCc2ccc(Cl)cc2)c1 ZINC000217704206 DJ In-Stock Unstable NR1H4 67 36 O=C(Cl)/C=C/c1cccc(OCc2ccc(Cl)cc2)c1 ZINC000217704206 DJ In-Stock Unstable ACR 20 40 O=C(Cl)/C=C/c1cccc(OCc2ccc(Cl)cc2)c1 ZINC000217704206 DJ In-Stock Unstable FFAR1 41 40 O=C(Cl)/C=C/c1cccc(OCc2ccc(Cl)cc2)c1 ZINC000217704206 DJ In-Stock Unstable AKR1C3 26 45 O=C(Cl)/C=C/c1cccc(OCc2ccc(Cl)cc2)c1 ZINC000217704206 DJ In-Stock Unstable GPR18 0 44 COc1cc2c(cc1OC)[C@H](c1cccnc1)N(C(=O)c1cc[nH]n1)CC2 ZINC000217704240 FF In-Stock Unstable MTNR1B 20 40 O=C(O)c1cc(O)n(-c2ccc(Oc3ccccc3)cc2)n1 ZINC000217704265 CG In-Stock Anodyne SRD5A2 0 43 O=C(O)c1cc(O)n(-c2ccc(Oc3ccccc3)cc2)n1 ZINC000217704265 CG In-Stock Anodyne FAAH 17 48 O=C(O)c1cc(O)n(-c2ccc(Oc3ccccc3)cc2)n1 ZINC000217704265 CG In-Stock Anodyne SCN4A 34 43 O=C(O)c1cc(O)n(-c2ccc(Oc3ccccc3)cc2)n1 ZINC000217704265 CG In-Stock Anodyne RPA1 82 56 COc1ccccc1/C=C/NC(=O)Nc1c(C)cccc1C(C)C ZINC000217704269 DJ For-Sale Unstable SOAT1 60 45 COc1ccccc1/C=C/NC(=O)Nc1c(C)cccc1C(C)C ZINC000217704269 DJ For-Sale Unstable ACAT 0 45 COc1ccccc1/C=C/NC(=O)Nc1c(C)cccc1C(C)C ZINC000217704269 DJ For-Sale Unstable KCNK3 31 42 COc1ccccc1/C=C/NC(=O)Nc1c(C)cccc1C(C)C ZINC000217704269 DJ For-Sale Unstable KCNK9 28 42 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccc2)c1 ZINC000217704306 CG For-Sale Anodyne EPHX1 0 40 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccc2)c1 ZINC000217704306 CG For-Sale Anodyne MAOB 0 53 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccc2)c1 ZINC000217704306 CG For-Sale Anodyne TRYP_PIG 15 44 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccc2)c1 ZINC000217704306 CG For-Sale Anodyne HDAC8 31 68 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccc2)c1 ZINC000217704306 CG For-Sale Anodyne PRNP 29 49 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccc2)c1 ZINC000217704306 CG For-Sale Anodyne F3 18 44 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccc2)c1 ZINC000217704306 CG For-Sale Anodyne MMP2 15 55 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccc2)c1 ZINC000217704306 CG For-Sale Anodyne HDAC1 21 47 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccc2)c1 ZINC000217704306 CG For-Sale Anodyne HDAC2 16 46 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccc2)c1 ZINC000217704306 CG For-Sale Anodyne HDAC6 28 68 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccc2)c1 ZINC000217704306 CG For-Sale Anodyne MMP9 0 55 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccc2)c1 ZINC000217704306 CG For-Sale Anodyne MMP1 25 48 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccc2)c1 ZINC000217704306 CG For-Sale Anodyne TAAR1 40 49 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccc2)c1 ZINC000217704306 CG For-Sale Anodyne AKR1C3 56 43 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccc2)c1 ZINC000217704306 CG For-Sale Anodyne RHOA 0 50 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccc2)c1 ZINC000217704306 CG For-Sale Anodyne PARP14 0 45 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccc2)c1 ZINC000217704306 CG For-Sale Anodyne PARP15 0 40 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccc2)c1 ZINC000217704306 CG For-Sale Anodyne KCNK3 141 54 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccc2)c1 ZINC000217704306 CG For-Sale Anodyne KCNK9 89 54 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccc2)c1 ZINC000217704306 CG For-Sale Anodyne PARP10 0 45 O=C(O)/C=C\c1cccc(C(=O)Nc2ccccc2)c1 ZINC000217704306 CG For-Sale Anodyne A0A060INS8_CAPHI 0 41 Cc1cccc(/C=C\C(=O)NC[C@](C)(O)CC(=O)O)c1 ZINC000217704308 CD For-Sale Unstable HDAC8 56 37 Cc1cccc(/C=C\C(=O)NC[C@](C)(O)CC(=O)O)c1 ZINC000217704308 CD For-Sale Unstable MMP2 16 45 Cc1cccc(/C=C\C(=O)NC[C@](C)(O)CC(=O)O)c1 ZINC000217704308 CD For-Sale Unstable MMP9 0 45 Cc1cccc(/C=C\C(=O)NC[C@](C)(O)CC(=O)O)c1 ZINC000217704308 CD For-Sale Unstable MMP1 0 45 O=C(Cl)/C=C/c1cccc(OCc2ccc(Cl)cc2Cl)c1 ZINC000217704313 EK In-Stock Unstable PTGER1 15 42 O=C(Cl)/C=C/c1cccc(OCc2ccc(Cl)cc2Cl)c1 ZINC000217704313 EK In-Stock Unstable CDC25B 0 42 O=C(Cl)/C=C/c1cccc(OCc2ccc(Cl)cc2Cl)c1 ZINC000217704313 EK In-Stock Unstable NR1H4 43 36 O=C(Cl)/C=C/c1cccc(OCc2ccc(Cl)cc2Cl)c1 ZINC000217704313 EK In-Stock Unstable TUBA4A 0 40 O=C(Cl)/C=C/c1cccc(OCc2ccc(Cl)cc2Cl)c1 ZINC000217704313 EK In-Stock Unstable GPR18 0 46 COc1cccc(Oc2ccc([N+](=O)[O-])c(Br)c2)c1 ZINC000217704335 DI For-Sale Unstable TAAR1 23 49 COc1cccc(Oc2ccc([N+](=O)[O-])c(Br)c2)c1 ZINC000217704335 DI For-Sale Unstable AKR1C2 19 43 CSC[C@@](C)(O)CNC(=O)c1ccc(SC)c([N+](=O)[O-])c1 ZINC000217704339 EE On-Demand Unstable GSTM2 46 36 CCCCCNS(=O)(=O)c1ccc(NCC)c(C(=O)O)c1 ZINC000217704371 DE In-Stock Unstable CASP3 22 48 CCCCCNS(=O)(=O)c1ccc(NCC)c(C(=O)O)c1 ZINC000217704371 DE In-Stock Unstable BDKRB1 0 43 COc1ccccc1/C=C/NC(=O)Nc1ccccc1C(F)(F)F ZINC000217704379 EJ For-Sale Unstable P2RY1 16 40 O=C(O)/C=C\c1ccc(F)c(C(=O)Nc2ccccc2)c1 ZINC000217704396 CG For-Sale Anodyne MAOB 0 45 O=C(O)/C=C\c1ccc(F)c(C(=O)Nc2ccccc2)c1 ZINC000217704396 CG For-Sale Anodyne MMP2 0 48 O=C(O)/C=C\c1ccc(F)c(C(=O)Nc2ccccc2)c1 ZINC000217704396 CG For-Sale Anodyne MMP9 0 48 O=C(O)/C=C\c1ccc(F)c(C(=O)Nc2ccccc2)c1 ZINC000217704396 CG For-Sale Anodyne MMP1 24 48 O=C(O)/C=C\c1ccc(F)c(C(=O)Nc2ccccc2)c1 ZINC000217704396 CG For-Sale Anodyne SMO 16 46 O=C(O)/C=C\c1ccc(F)c(C(=O)Nc2ccccc2)c1 ZINC000217704396 CG For-Sale Anodyne RHOA 0 44 O=C(O)/C=C\c1ccc(F)c(C(=O)Nc2ccccc2)c1 ZINC000217704396 CG For-Sale Anodyne KCNK3 93 38 O=C(O)/C=C\c1ccc(F)c(C(=O)Nc2ccccc2)c1 ZINC000217704396 CG For-Sale Anodyne KCNK9 73 35 Cc1cccc(/C=C\C(=O)NC[C@@](C)(O)CC(=O)O)c1 ZINC000217704403 CD For-Sale Unstable HDAC8 56 37 Cc1cccc(/C=C\C(=O)NC[C@@](C)(O)CC(=O)O)c1 ZINC000217704403 CD For-Sale Unstable MMP2 16 45 Cc1cccc(/C=C\C(=O)NC[C@@](C)(O)CC(=O)O)c1 ZINC000217704403 CD For-Sale Unstable MMP9 0 45 Cc1cccc(/C=C\C(=O)NC[C@@](C)(O)CC(=O)O)c1 ZINC000217704403 CD For-Sale Unstable MMP1 0 45 CSC[C@](C)(O)CNC(=O)c1ccc(SC)c([N+](=O)[O-])c1 ZINC000217704433 EE On-Demand Unstable GSTM2 46 36 O=C(Cl)/C=C/c1cccc(OCc2ccc(Cl)c(Cl)c2)c1 ZINC000217704434 EK In-Stock Unstable MAOB 39 45 O=C(Cl)/C=C/c1cccc(OCc2ccc(Cl)c(Cl)c2)c1 ZINC000217704434 EK In-Stock Unstable CYSLTR1 20 45 O=C(Cl)/C=C/c1cccc(OCc2ccc(Cl)c(Cl)c2)c1 ZINC000217704434 EK In-Stock Unstable CDC25B 0 41 O=C(Cl)/C=C/c1cccc(OCc2ccc(Cl)c(Cl)c2)c1 ZINC000217704434 EK In-Stock Unstable NR1H4 64 36 O=C(Cl)/C=C/c1cccc(OCc2ccc(Cl)c(Cl)c2)c1 ZINC000217704434 EK In-Stock Unstable FFAR1 40 41 O=C(Cl)/C=C/c1cccc(OCc2ccc(Cl)c(Cl)c2)c1 ZINC000217704434 EK In-Stock Unstable GPR18 0 46 Nc1cc([N+](=O)[O-])ccc1C(=O)OCCC1CC1 ZINC000217704449 CE On-Demand Unstable CACNA1C 49 38 Nc1cc([N+](=O)[O-])ccc1C(=O)OCCC1CC1 ZINC000217704449 CE On-Demand Unstable CACNA1D 77 38 Nc1cc([N+](=O)[O-])ccc1C(=O)OCCC1CC1 ZINC000217704449 CE On-Demand Unstable SLC27A4 44 34 CCNc1ccc(S(=O)(=O)N[C@@H](C)CC)cc1C(=O)O ZINC000217704483 DD In-Stock Unstable MMP12 49 37 CCNc1ccc(S(=O)(=O)N[C@@H](C)CC)cc1C(=O)O ZINC000217704483 DD In-Stock Unstable ADAMTS4 41 33 CCNc1ccc(S(=O)(=O)N[C@@H](C)CC)cc1C(=O)O ZINC000217704483 DD In-Stock Unstable LEF 53 39 O=C(O)/C=C\c1ccc(C(=O)Nc2ccccc2)c(F)c1 ZINC000217704486 CG For-Sale Anodyne MAOB 0 45 O=C(O)/C=C\c1ccc(C(=O)Nc2ccccc2)c(F)c1 ZINC000217704486 CG For-Sale Anodyne MMP2 0 48 O=C(O)/C=C\c1ccc(C(=O)Nc2ccccc2)c(F)c1 ZINC000217704486 CG For-Sale Anodyne MMP9 0 48 O=C(O)/C=C\c1ccc(C(=O)Nc2ccccc2)c(F)c1 ZINC000217704486 CG For-Sale Anodyne MMP1 24 48 O=C(O)/C=C\c1ccc(C(=O)Nc2ccccc2)c(F)c1 ZINC000217704486 CG For-Sale Anodyne SMO 16 46 O=C(O)/C=C\c1ccc(C(=O)Nc2ccccc2)c(F)c1 ZINC000217704486 CG For-Sale Anodyne RHOA 0 44 O=C(O)/C=C\c1ccc(C(=O)Nc2ccccc2)c(F)c1 ZINC000217704486 CG For-Sale Anodyne KCNK3 93 38 O=C(O)/C=C\c1ccc(C(=O)Nc2ccccc2)c(F)c1 ZINC000217704486 CG For-Sale Anodyne KCNK9 68 35 COc1ccccc1/C=C/NC(=O)Nc1ccc(C(=O)O)cc1 ZINC000217704492 DG For-Sale Unstable PPIA 22 41 COc1ccccc1/C=C/NC(=O)Nc1ccc(C(=O)O)cc1 ZINC000217704492 DG For-Sale Unstable ACR 24 42 COc1ccccc1/C=C/NC(=O)Nc1ccc(C(=O)O)cc1 ZINC000217704492 DG For-Sale Unstable PDGFRA 43 38 C[C@](O)(CNC(=O)/C=C\c1ccc(Cl)cc1)CC(=O)O ZINC000217704515 CD For-Sale Unstable PYGL 0 44 C[C@](O)(CNC(=O)/C=C\c1ccc(Cl)cc1)CC(=O)O ZINC000217704515 CD For-Sale Unstable HDAC8 0 45 C[C@](O)(CNC(=O)/C=C\c1ccc(Cl)cc1)CC(=O)O ZINC000217704515 CD For-Sale Unstable MMP2 15 46 C[C@](O)(CNC(=O)/C=C\c1ccc(Cl)cc1)CC(=O)O ZINC000217704515 CD For-Sale Unstable HDAC1 0 40 C[C@](O)(CNC(=O)/C=C\c1ccc(Cl)cc1)CC(=O)O ZINC000217704515 CD For-Sale Unstable MMP1 0 46 O=C(Cl)/C=C/c1cccc(OCc2ccc(F)cc2Cl)c1 ZINC000217704551 EJ In-Stock Unstable CDC25B 21 40 O=C(Cl)/C=C/c1cccc(OCc2ccc(F)cc2Cl)c1 ZINC000217704551 EJ In-Stock Unstable NR1H4 41 35 CCNc1ccc(S(=O)(=O)N[C@H](C)CC)cc1C(=O)O ZINC000217704560 DD In-Stock Unstable MMP12 49 37 CCNc1ccc(S(=O)(=O)N[C@H](C)CC)cc1C(=O)O ZINC000217704560 DD In-Stock Unstable ADAMTS4 41 33 CCNc1ccc(S(=O)(=O)N[C@H](C)CC)cc1C(=O)O ZINC000217704560 DD In-Stock Unstable LEF 53 39 O=C(O)/C=C\c1cccc(C(=O)Nc2cccnc2)c1 ZINC000217704578 CE For-Sale Anodyne TBXAS1 33 45 O=C(O)/C=C\c1cccc(C(=O)Nc2cccnc2)c1 ZINC000217704578 CE For-Sale Anodyne RPS6KA3 32 43 O=C(O)/C=C\c1cccc(C(=O)Nc2cccnc2)c1 ZINC000217704578 CE For-Sale Anodyne CSF1R 22 53 O=C(O)/C=C\c1cccc(C(=O)Nc2cccnc2)c1 ZINC000217704578 CE For-Sale Anodyne NAMPT 24 58 O=C(O)/C=C\c1cccc(C(=O)Nc2cccnc2)c1 ZINC000217704578 CE For-Sale Anodyne KCNK3 107 48 O=C(O)/C=C\c1cccc(C(=O)Nc2cccnc2)c1 ZINC000217704578 CE For-Sale Anodyne KCNK9 52 43 C[C@@](O)(CNC(=O)/C=C\c1ccc(Cl)cc1)CC(=O)O ZINC000217704609 CD For-Sale Unstable PYGL 0 44 C[C@@](O)(CNC(=O)/C=C\c1ccc(Cl)cc1)CC(=O)O ZINC000217704609 CD For-Sale Unstable HDAC8 0 45 C[C@@](O)(CNC(=O)/C=C\c1ccc(Cl)cc1)CC(=O)O ZINC000217704609 CD For-Sale Unstable MMP2 15 46 C[C@@](O)(CNC(=O)/C=C\c1ccc(Cl)cc1)CC(=O)O ZINC000217704609 CD For-Sale Unstable HDAC1 0 40 C[C@@](O)(CNC(=O)/C=C\c1ccc(Cl)cc1)CC(=O)O ZINC000217704609 CD For-Sale Unstable MMP1 0 46 COc1ccccc1/C=C/NC(=O)Nc1cccc(Cl)c1C ZINC000217704618 DI For-Sale Unstable CXCL8 40 32 COC(=O)[C@@H](O)CNC(=O)[C@@H](C)Oc1cccc(F)c1 ZINC000217704641 CC On-Demand Unstable MTNR1A 17 43 COC(=O)[C@@H](O)CNC(=O)[C@@H](C)Oc1cccc(F)c1 ZINC000217704641 CC On-Demand Unstable MTNR1B 19 43 O=C(Cl)/C=C/c1cccc(OCc2ccc(Br)cc2)c1 ZINC000217704661 FJ In-Stock Unstable MAOB 34 51 O=C(Cl)/C=C/c1cccc(OCc2ccc(Br)cc2)c1 ZINC000217704661 FJ In-Stock Unstable FFAR1 23 43 O=C(O)/C=C\c1ccc(F)c(C(=O)Nc2cccnc2)c1 ZINC000217704662 CF For-Sale Anodyne NAMPT 20 46 COc1ccccc1CCNC(=O)c1ccncc1Cl ZINC000217704684 CF On-Demand Unstable DRD2 16 41 COc1ccccc1CCNC(=O)c1ccncc1Cl ZINC000217704684 CF On-Demand Unstable P2RX7 15 50 COc1ccccc1CCNC(=O)c1ccncc1Cl ZINC000217704684 CF On-Demand Unstable PDE4D 19 40 COC(=O)[C@H](O)CNC(=O)[C@@H](C)Oc1cccc(F)c1 ZINC000217704726 CC On-Demand Unstable MTNR1A 17 43 COC(=O)[C@H](O)CNC(=O)[C@@H](C)Oc1cccc(F)c1 ZINC000217704726 CC On-Demand Unstable MTNR1B 19 43 CCOC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217704734 EH For-Sale Unstable PPIA 23 48 CCOC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217704734 EH For-Sale Unstable ACR 72 48 O=C(O)/C=C\c1ccc(C(=O)Nc2cccnc2)c(F)c1 ZINC000217704745 CF For-Sale Anodyne NAMPT 20 45 Cc1nc2ccc(C(=O)NCCSC3CCOCC3)cc2s1 ZINC000217704776 EG In-Stock Unstable LCK 27 43 Cc1nc2ccc(C(=O)NCCSC3CCOCC3)cc2s1 ZINC000217704776 EG In-Stock Unstable NMT1 28 49 O=C(Cl)/C=C/c1cccc(OCc2cccc(Br)c2)c1 ZINC000217704788 FJ In-Stock Unstable MAOB 50 56 O=C(Cl)/C=C/c1cccc(OCc2cccc(Br)c2)c1 ZINC000217704788 FJ In-Stock Unstable HCAR2 0 46 O=C(Cl)/C=C/c1cccc(OCc2cccc(Br)c2)c1 ZINC000217704788 FJ In-Stock Unstable FFAR1 29 49 O=C(O)c1cc(O)n(-c2cc(Cl)ccc2Oc2ccccc2)n1 ZINC000217704792 EH In-Stock Anodyne PTGER1 43 39 O=C(O)c1cc(O)n(-c2cc(Cl)ccc2Oc2ccccc2)n1 ZINC000217704792 EH In-Stock Anodyne TTR 0 41 O=C(O)c1cc(O)n(-c2cc(Cl)ccc2Oc2ccccc2)n1 ZINC000217704792 EH In-Stock Anodyne ENR 0 49 O=C(O)c1cc(O)n(-c2cc(Cl)ccc2Oc2ccccc2)n1 ZINC000217704792 EH In-Stock Anodyne RPA1 70 43 COC(=O)[C@@H](O)CNC(=O)[C@H](C)Oc1cccc(F)c1 ZINC000217704821 CC On-Demand Unstable MTNR1A 17 43 COC(=O)[C@@H](O)CNC(=O)[C@H](C)Oc1cccc(F)c1 ZINC000217704821 CC On-Demand Unstable MTNR1B 19 43 Cc1cc(NC(=O)c2cccc(/C=C\C(=O)O)c2)on1 ZINC000217704843 CE For-Sale Unstable HDAC8 29 44 Cc1cc(NC(=O)c2cccc(/C=C\C(=O)O)c2)on1 ZINC000217704843 CE For-Sale Unstable KCNK3 87 38 Cc1cc(NC(=O)c2cccc(/C=C\C(=O)O)c2)on1 ZINC000217704843 CE For-Sale Unstable KCNK9 48 38 COc1ccccc1/C=C/NC(=O)Nc1ccccc1Cl ZINC000217704849 DI For-Sale Unstable CXCL8 42 35 O=C(NCCSC1CCOCC1)c1ccc(-c2cccs2)cc1 ZINC000217704885 EI In-Stock Unstable HDAC1 0 43 Nc1ccc(-n2nc(C(=O)O)cc2O)cc1 ZINC000217704892 BC In-Stock Unstable RPA1 77 40 O=C(Cl)/C=C/c1cccc(OCc2ccccc2Cl)c1 ZINC000217704897 DJ In-Stock Unstable CYSLTR1 16 42 O=C(Cl)/C=C/c1cccc(OCc2ccccc2Cl)c1 ZINC000217704897 DJ In-Stock Unstable FABP4 19 44 O=C(Cl)/C=C/c1cccc(OCc2ccccc2Cl)c1 ZINC000217704897 DJ In-Stock Unstable CDC25B 0 41 O=C(Cl)/C=C/c1cccc(OCc2ccccc2Cl)c1 ZINC000217704897 DJ In-Stock Unstable NR1H4 51 36 O=C(Cl)/C=C/c1cccc(OCc2ccccc2Cl)c1 ZINC000217704897 DJ In-Stock Unstable FABP5 30 44 O=C(Cl)/C=C/c1cccc(OCc2ccccc2Cl)c1 ZINC000217704897 DJ In-Stock Unstable GPR18 0 45 COC(=O)[C@H](O)CNC(=O)[C@H](C)Oc1cccc(F)c1 ZINC000217704901 CC On-Demand Unstable MTNR1A 17 43 COC(=O)[C@H](O)CNC(=O)[C@H](C)Oc1cccc(F)c1 ZINC000217704901 CC On-Demand Unstable MTNR1B 19 43 CSC1C[C@@H]2CC[C@H](C1)N2C(=O)c1cc(-c2ccc(F)cc2)n[nH]1 ZINC000217704972 EH In-Stock Unstable TACR3 16 44 COc1ccccc1/C=C/NC(=O)Nc1ccccc1C(C)C ZINC000217704980 DJ For-Sale Unstable SOAT1 23 41 COc1ccccc1/C=C/NC(=O)Nc1ccccc1C(C)C ZINC000217704980 DJ For-Sale Unstable KCNK3 31 43 COc1ccccc1/C=C/NC(=O)Nc1ccccc1C(C)C ZINC000217704980 DJ For-Sale Unstable KCNK9 28 43 CNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217704987 ED In-Stock Unstable CA2 32 48 CNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217704987 ED In-Stock Unstable TBXA2R 59 48 CNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217704987 ED In-Stock Unstable TBXAS1 40 46 CNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217704987 ED In-Stock Unstable CA1 26 43 CNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217704987 ED In-Stock Unstable CA7 23 42 CNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217704987 ED In-Stock Unstable CA5B 43 41 CNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217704987 ED In-Stock Unstable CA4 30 48 CNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217704987 ED In-Stock Unstable CA5A 44 41 CNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217704987 ED In-Stock Unstable ALOX15 53 35 CNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217704987 ED In-Stock Unstable CA12 16 42 CNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217704987 ED In-Stock Unstable TPSAB1 15 40 CNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217704987 ED In-Stock Unstable AKR1C3 28 60 CNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217704987 ED In-Stock Unstable A6YCJ1_9METZ 15 42 O=C(Cl)c1ccc(OCc2ccccc2)c(Br)c1 ZINC000217705010 EI In-Stock Unstable THRA 17 49 O=C(Cl)c1ccc(OCc2ccccc2)c(Br)c1 ZINC000217705010 EI In-Stock Unstable PTGER2 41 43 O=C(Cl)c1ccc(OCc2ccccc2)c(Br)c1 ZINC000217705010 EI In-Stock Unstable PPIA 45 36 O=C(Cl)c1ccc(OCc2ccccc2)c(Br)c1 ZINC000217705010 EI In-Stock Unstable PTGER1 62 41 O=C(Cl)c1ccc(OCc2ccccc2)c(Br)c1 ZINC000217705010 EI In-Stock Unstable PTGER4 31 43 O=C(Cl)c1ccc(OCc2ccccc2)c(Br)c1 ZINC000217705010 EI In-Stock Unstable ACR 46 55 O=C(Cl)c1ccc(OCc2ccccc2)c(Br)c1 ZINC000217705010 EI In-Stock Unstable POBA 0 45 O=C(Cl)c1ccc(OCc2ccccc2)c(Br)c1 ZINC000217705010 EI In-Stock Unstable KLK_PIG 54 56 CCc1ccc(CNC(=O)c2ccncc2Cl)cc1 ZINC000217705028 CG For-Sale Unstable UL54 42 33 CCc1ccc(CNC(=O)c2ccncc2Cl)cc1 ZINC000217705028 CG For-Sale Unstable NAMPT 88 39 COc1ccccc1/C=C/NC(=O)Nc1cccc(Cl)c1Cl ZINC000217705095 EJ For-Sale Unstable CXCL8 41 31 COc1ccccc1/C=C/NC(=O)Nc1cccc(Cl)c1Cl ZINC000217705095 EJ For-Sale Unstable CYSP_PLAFA 36 41 COc1ccc(CNC(=O)CN2C(=O)c3ccccc3N3C(=O)c4c(ccc(OC)c4OC)[C@H]23)cc1 ZINC000217705104 JG In-Stock Unstable TSHR 50 33 COc1ccc(CNC(=O)CN2C(=O)c3ccccc3N3C(=O)c4c(ccc(OC)c4OC)[C@H]23)cc1 ZINC000217705104 JG In-Stock Unstable SCN9A 0 43 Cn1nc(-c2ccccc2)cc1C(=O)NCCSC1CCOCC1 ZINC000217705109 EF In-Stock Unstable INHA 54 34 Cn1nc(-c2ccccc2)cc1C(=O)NCCSC1CCOCC1 ZINC000217705109 EF In-Stock Unstable CTSV 44 31 CC[C@H](C(=O)O)N(C)C(=O)/C=C\c1ccc(O)cc1 ZINC000217705158 CD For-Sale Unstable F3 26 45 CC[C@H](C(=O)O)N(C)C(=O)/C=C\c1ccc(O)cc1 ZINC000217705158 CD For-Sale Unstable SSSIM 15 46 CC[C@H](C(=O)O)N(C)C(=O)/C=C\c1ccc(O)cc1 ZINC000217705158 CD For-Sale Unstable AKR1B10 21 41 CSC[C@@](C)(O)CNC(=O)Cc1c[nH]c2ccccc12 ZINC000217705191 CD On-Demand Unstable MC4R 25 41 CSC[C@@](C)(O)CNC(=O)Cc1c[nH]c2ccccc12 ZINC000217705191 CD On-Demand Unstable CCKAR 74 39 CSC[C@@](C)(O)CNC(=O)Cc1c[nH]c2ccccc12 ZINC000217705191 CD On-Demand Unstable BRS3 23 43 CSC[C@@](C)(O)CNC(=O)Cc1c[nH]c2ccccc12 ZINC000217705191 CD On-Demand Unstable NMBR 67 32 CSC[C@@](C)(O)CNC(=O)Cc1c[nH]c2ccccc12 ZINC000217705191 CD On-Demand Unstable MMP14 69 36 CSC[C@@](C)(O)CNC(=O)Cc1c[nH]c2ccccc12 ZINC000217705191 CD On-Demand Unstable GRPR 52 33 CSC[C@@](C)(O)CNC(=O)Cc1c[nH]c2ccccc12 ZINC000217705191 CD On-Demand Unstable ECE1 42 37 CSC[C@@](C)(O)CNC(=O)Cc1c[nH]c2ccccc12 ZINC000217705191 CD On-Demand Unstable MMP11 53 32 CSC[C@@](C)(O)CNC(=O)Cc1c[nH]c2ccccc12 ZINC000217705191 CD On-Demand Unstable CCKBR 61 40 CSC[C@@](C)(O)CNC(=O)Cc1c[nH]c2ccccc12 ZINC000217705191 CD On-Demand Unstable GHSR 49 39 CSC[C@@](C)(O)CNC(=O)Cc1c[nH]c2ccccc12 ZINC000217705191 CD On-Demand Unstable SLC15A2 0 40 CSC[C@@](C)(O)CNC(=O)Cc1c[nH]c2ccccc12 ZINC000217705191 CD On-Demand Unstable KISS1R 40 31 COc1ccc(CNC(=O)CN2C(=O)c3ccccc3N3C(=O)c4c(ccc(OC)c4OC)[C@@H]23)cc1 ZINC000217705199 JG In-Stock Unstable TSHR 50 33 COc1ccc(CNC(=O)CN2C(=O)c3ccccc3N3C(=O)c4c(ccc(OC)c4OC)[C@@H]23)cc1 ZINC000217705199 JG In-Stock Unstable SCN9A 0 43 COc1ccccc1/C=C/NC(=O)Nc1cc(Cl)ccc1Cl ZINC000217705209 EJ For-Sale Unstable PYGL 15 43 COc1ccccc1/C=C/NC(=O)Nc1cc(Cl)ccc1Cl ZINC000217705209 EJ For-Sale Unstable S1PR4 15 42 COc1ccccc1/C=C/NC(=O)Nc1cc(Cl)ccc1Cl ZINC000217705209 EJ For-Sale Unstable RBP4 15 40 COc1ccccc1/C=C/NC(=O)Nc1cc(Cl)ccc1Cl ZINC000217705209 EJ For-Sale Unstable CYSP_PLAFA 45 38 CC[C@@H](C(=O)O)N(C)C(=O)/C=C\c1ccc(O)cc1 ZINC000217705232 CD For-Sale Unstable F3 26 45 CC[C@@H](C(=O)O)N(C)C(=O)/C=C\c1ccc(O)cc1 ZINC000217705232 CD For-Sale Unstable SSSIM 15 46 CC[C@@H](C(=O)O)N(C)C(=O)/C=C\c1ccc(O)cc1 ZINC000217705232 CD For-Sale Unstable AKR1B10 21 41 CSC[C@](C)(O)CNC(=O)Cc1c[nH]c2ccccc12 ZINC000217705271 CD On-Demand Unstable CCKAR 74 39 CSC[C@](C)(O)CNC(=O)Cc1c[nH]c2ccccc12 ZINC000217705271 CD On-Demand Unstable BRS3 23 43 CSC[C@](C)(O)CNC(=O)Cc1c[nH]c2ccccc12 ZINC000217705271 CD On-Demand Unstable NMBR 67 32 CSC[C@](C)(O)CNC(=O)Cc1c[nH]c2ccccc12 ZINC000217705271 CD On-Demand Unstable GRPR 52 33 CSC[C@](C)(O)CNC(=O)Cc1c[nH]c2ccccc12 ZINC000217705271 CD On-Demand Unstable ECE1 42 37 CSC[C@](C)(O)CNC(=O)Cc1c[nH]c2ccccc12 ZINC000217705271 CD On-Demand Unstable MMP11 53 32 CSC[C@](C)(O)CNC(=O)Cc1c[nH]c2ccccc12 ZINC000217705271 CD On-Demand Unstable CCKBR 61 40 CSC[C@](C)(O)CNC(=O)Cc1c[nH]c2ccccc12 ZINC000217705271 CD On-Demand Unstable GHSR 49 39 CSC[C@](C)(O)CNC(=O)Cc1c[nH]c2ccccc12 ZINC000217705271 CD On-Demand Unstable KISS1R 40 31 Cc1ccc(S(N)(=O)=O)cc1C(=O)OCCC1CC1 ZINC000217705281 CD On-Demand Unstable CA2 77 45 Cc1ccc(S(N)(=O)=O)cc1C(=O)OCCC1CC1 ZINC000217705281 CD On-Demand Unstable CA1 64 40 Cc1ccc(S(N)(=O)=O)cc1C(=O)OCCC1CC1 ZINC000217705281 CD On-Demand Unstable CA7 59 38 Cc1ccc(S(N)(=O)=O)cc1C(=O)OCCC1CC1 ZINC000217705281 CD On-Demand Unstable CA4 71 40 Cc1ccc(S(N)(=O)=O)cc1C(=O)OCCC1CC1 ZINC000217705281 CD On-Demand Unstable CA12 40 38 Cc1ccc(S(N)(=O)=O)cc1C(=O)OCCC1CC1 ZINC000217705281 CD On-Demand Unstable CA9 42 39 Cc1ccc(S(N)(=O)=O)cc1C(=O)OCCC1CC1 ZINC000217705281 CD On-Demand Unstable CYNT 40 38 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(Cl)c(Cl)c1 ZINC000217705310 FK In-Stock Unstable CYP1A1 18 41 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(Cl)c(Cl)c1 ZINC000217705310 FK In-Stock Unstable TUBB1 55 39 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(Cl)c(Cl)c1 ZINC000217705310 FK In-Stock Unstable AKR1C3 32 46 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(Cl)c(Cl)c1 ZINC000217705310 FK In-Stock Unstable ABCG2 19 45 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(Cl)c(Cl)c1 ZINC000217705310 FK In-Stock Unstable CYSP_PLAFA 50 43 COc1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1Cl ZINC000217705319 EI For-Sale Unstable GCGR 0 42 COc1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1Cl ZINC000217705319 EI For-Sale Unstable GRM4 24 52 COc1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1Cl ZINC000217705319 EI For-Sale Unstable IMPDH2 0 44 COc1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1Cl ZINC000217705319 EI For-Sale Unstable CYSP_PLAFA 43 36 C[C@@H](Cc1cnnn1Cc1ccccc1)C(=O)O ZINC000217705327 BD For-Sale Unstable MME 52 37 C[C@@H](Cc1cnnn1Cc1ccccc1)C(=O)O ZINC000217705327 BD For-Sale Unstable CYSP_TRYCR 45 33 C[C@@H](Cc1cnnn1Cc1ccccc1)C(=O)O ZINC000217705327 BD For-Sale Unstable CPA1 52 36 C[C@@H](Cc1cnnn1Cc1ccccc1)C(=O)O ZINC000217705327 BD For-Sale Unstable CAPNS1 45 32 C[C@@H](Cc1cnnn1Cc1ccccc1)C(=O)O ZINC000217705327 BD For-Sale Unstable ACE2 49 36 C[C@@H](Cc1cnnn1Cc1ccccc1)C(=O)O ZINC000217705327 BD For-Sale Unstable FPR1 50 38 Cn1cc(CC(=O)NCCSC2CCOCC2)c2ccccc21 ZINC000217705331 EF In-Stock Unstable CNR1 0 41 c1ccc2cc(CN[C@@H]3CCN4CCC[C@@H]34)ccc2c1 ZINC000217705372 CG For-Sale Unstable SSTR3 17 44 CCCN(CC1CC1)C(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217705402 CG For-Sale Unstable OXTR 0 40 CCCN(CC1CC1)C(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217705402 CG For-Sale Unstable OPRD1 15 49 CCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCC ZINC000217705407 DD In-Stock Unstable PLA2G4B 40 34 C[C@H](Cc1cnnn1Cc1ccccc1)C(=O)O ZINC000217705413 BD For-Sale Unstable MME 52 37 C[C@H](Cc1cnnn1Cc1ccccc1)C(=O)O ZINC000217705413 BD For-Sale Unstable CYSP_TRYCR 45 33 C[C@H](Cc1cnnn1Cc1ccccc1)C(=O)O ZINC000217705413 BD For-Sale Unstable CPA1 52 36 C[C@H](Cc1cnnn1Cc1ccccc1)C(=O)O ZINC000217705413 BD For-Sale Unstable CAPNS1 45 32 C[C@H](Cc1cnnn1Cc1ccccc1)C(=O)O ZINC000217705413 BD For-Sale Unstable ACE2 49 36 C[C@H](Cc1cnnn1Cc1ccccc1)C(=O)O ZINC000217705413 BD For-Sale Unstable FPR1 50 38 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(Cl)cc1 ZINC000217705414 EJ In-Stock Unstable PTGER2 0 45 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(Cl)cc1 ZINC000217705414 EJ In-Stock Unstable PTGER1 48 38 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(Cl)cc1 ZINC000217705414 EJ In-Stock Unstable KCNA3 0 48 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(Cl)cc1 ZINC000217705414 EJ In-Stock Unstable CCR5 22 41 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(Cl)cc1 ZINC000217705414 EJ In-Stock Unstable TNFRSF1A 15 48 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(Cl)cc1 ZINC000217705414 EJ In-Stock Unstable CYP1A1 31 40 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(Cl)cc1 ZINC000217705414 EJ In-Stock Unstable MMP12 0 52 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(Cl)cc1 ZINC000217705414 EJ In-Stock Unstable TUBB1 61 40 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(Cl)cc1 ZINC000217705414 EJ In-Stock Unstable AKR1C3 35 55 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(Cl)cc1 ZINC000217705414 EJ In-Stock Unstable ABCG2 19 46 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(Cl)cc1 ZINC000217705414 EJ In-Stock Unstable NFE2L2 0 42 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(Cl)cc1 ZINC000217705414 EJ In-Stock Unstable CYSP_PLAFA 46 42 COc1ccccc1/C=C/NC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217705431 EJ For-Sale Unstable PPIA 16 45 COc1ccccc1/C=C/NC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217705431 EJ For-Sale Unstable KIT 17 47 COc1ccccc1/C=C/NC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217705431 EJ For-Sale Unstable RAF1 28 40 COc1ccccc1/C=C/NC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217705431 EJ For-Sale Unstable KDR 24 41 COc1ccccc1/C=C/NC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217705431 EJ For-Sale Unstable EPHX2 15 44 COc1ccccc1/C=C/NC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217705431 EJ For-Sale Unstable IMPDH2 0 42 COc1ccccc1/C=C/NC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217705431 EJ For-Sale Unstable TEK 36 41 COc1ccccc1/C=C/NC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217705431 EJ For-Sale Unstable KCNK3 73 44 COc1ccccc1/C=C/NC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217705431 EJ For-Sale Unstable KCNK9 61 43 c1ccc2cc(CN[C@H]3CCN4CCC[C@@H]34)ccc2c1 ZINC000217705452 CG For-Sale Unstable SSTR3 17 44 CCCN(CC1CC1)C(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217705475 CG For-Sale Unstable OPRD1 15 46 CCCN(CC1CC1)C(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217705475 CG For-Sale Unstable ACKR3 44 33 CNc1ccc(C(=O)O)cc1S(=O)(=O)NC1CCCCC1 ZINC000217705485 DE In-Stock Unstable CCR8 84 50 CNc1ccc(C(=O)O)cc1S(=O)(=O)NC1CCCCC1 ZINC000217705485 DE In-Stock Unstable SFRP1 105 38 CNc1ccc(C(=O)O)cc1S(=O)(=O)NC1CCCCC1 ZINC000217705485 DE In-Stock Unstable WNT3 82 37 CNc1ccc(C(=O)O)cc1S(=O)(=O)NC1CCCCC1 ZINC000217705485 DE In-Stock Unstable BRD4 25 41 C[C@@H](Cc1ncnn1Cc1ccccc1)C(=O)O ZINC000217705509 BD For-Sale Unstable MME 52 37 C[C@@H](Cc1ncnn1Cc1ccccc1)C(=O)O ZINC000217705509 BD For-Sale Unstable CPA1 49 36 C[C@@H](Cc1ncnn1Cc1ccccc1)C(=O)O ZINC000217705509 BD For-Sale Unstable CAPNS1 44 32 C[C@@H](Cc1ncnn1Cc1ccccc1)C(=O)O ZINC000217705509 BD For-Sale Unstable CAPN2 53 32 C[C@@H](Cc1ncnn1Cc1ccccc1)C(=O)O ZINC000217705509 BD For-Sale Unstable ACE2 49 36 C[C@@H](Cc1ncnn1Cc1ccccc1)C(=O)O ZINC000217705509 BD For-Sale Unstable FPR1 49 35 COC(=O)COc1cccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c1 ZINC000217705523 KH In-Stock Unstable AKR1B1 0 41 COC(=O)COc1cccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c1 ZINC000217705523 KH In-Stock Unstable CYP1A1 32 41 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(Br)cc1 ZINC000217705524 GJ In-Stock Unstable PTGER2 0 44 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(Br)cc1 ZINC000217705524 GJ In-Stock Unstable CCR5 25 42 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(Br)cc1 ZINC000217705524 GJ In-Stock Unstable TNFRSF1A 16 47 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(Br)cc1 ZINC000217705524 GJ In-Stock Unstable CYP1A1 19 42 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(Br)cc1 ZINC000217705524 GJ In-Stock Unstable MMP12 0 52 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(Br)cc1 ZINC000217705524 GJ In-Stock Unstable TUBB1 60 39 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(Br)cc1 ZINC000217705524 GJ In-Stock Unstable AKR1C3 34 45 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(Br)cc1 ZINC000217705524 GJ In-Stock Unstable ABCG2 29 45 C/C=C/C=C\C(=O)NC[C@](C)(O)CC(=O)O ZINC000217705558 BC For-Sale Unstable CNR2 15 57 C[C@H](Cc1ncnn1Cc1ccccc1)C(=O)O ZINC000217705586 BD For-Sale Unstable MME 52 37 C[C@H](Cc1ncnn1Cc1ccccc1)C(=O)O ZINC000217705586 BD For-Sale Unstable CPA1 49 36 C[C@H](Cc1ncnn1Cc1ccccc1)C(=O)O ZINC000217705586 BD For-Sale Unstable CAPNS1 44 32 C[C@H](Cc1ncnn1Cc1ccccc1)C(=O)O ZINC000217705586 BD For-Sale Unstable CAPN2 53 32 C[C@H](Cc1ncnn1Cc1ccccc1)C(=O)O ZINC000217705586 BD For-Sale Unstable ACE2 49 36 C[C@H](Cc1ncnn1Cc1ccccc1)C(=O)O ZINC000217705586 BD For-Sale Unstable FPR1 49 35 COC(=O)COc1cccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c1 ZINC000217705597 KH In-Stock Unstable AKR1B1 0 41 COC(=O)COc1cccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c1 ZINC000217705597 KH In-Stock Unstable CYP1A1 32 41 CSC[C@@](C)(O)CNC(=O)c1cccc(C)c1C ZINC000217705618 CE On-Demand Unstable ECR 29 45 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(F)cc1 ZINC000217705630 DI In-Stock Unstable PTGER2 24 44 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(F)cc1 ZINC000217705630 DI In-Stock Unstable TNFRSF1A 15 47 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(F)cc1 ZINC000217705630 DI In-Stock Unstable CYP1A1 22 42 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(F)cc1 ZINC000217705630 DI In-Stock Unstable TUBB1 62 39 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(F)cc1 ZINC000217705630 DI In-Stock Unstable AKR1C3 36 55 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(F)cc1 ZINC000217705630 DI In-Stock Unstable ENPP2 35 47 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(F)cc1 ZINC000217705630 DI In-Stock Unstable ABCG2 20 45 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(F)cc1 ZINC000217705630 DI In-Stock Unstable NFE2L2 0 44 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(F)cc1 ZINC000217705630 DI In-Stock Unstable CYSP_PLAFA 40 39 CC[C@H](C(=O)O)N(C)C(=O)/C=C\c1ccc(OC)c(F)c1 ZINC000217705656 CE For-Sale Unstable TUBB1 43 44 COC(=O)[C@@H](O)CNC(=O)[C@@H](C)Oc1ccccc1 ZINC000217705669 CC On-Demand Unstable NPR 41 32 COC(=O)[C@@H](O)CNC(=O)[C@@H](C)Oc1ccccc1 ZINC000217705669 CC On-Demand Unstable AMP1_PLAFQ 42 33 CSC[C@](C)(O)CNC(=O)c1cccc(C)c1C ZINC000217705690 CE On-Demand Unstable ECR 29 45 CCNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217705705 CD In-Stock Unstable CCR8 83 38 CCNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217705705 CD In-Stock Unstable SFRP1 101 37 CCNc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)O ZINC000217705705 CD In-Stock Unstable WNT3 79 37 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](C)C(=O)Nc3cccc(-c4nc[nH]n4)c3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217705714 KI In-Stock Unstable TUBA1A 17 62 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](C)C(=O)Nc3cccc(-c4nc[nH]n4)c3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217705714 KI In-Stock Unstable TPPP 0 57 CC[C@@H](C(=O)O)N(C)C(=O)/C=C\c1ccc(OC)c(F)c1 ZINC000217705740 CE For-Sale Unstable TUBB1 43 44 COC(=O)[C@H](O)CNC(=O)[C@@H](C)Oc1ccccc1 ZINC000217705745 CC On-Demand Unstable NPR 41 32 COC(=O)[C@H](O)CNC(=O)[C@@H](C)Oc1ccccc1 ZINC000217705745 CC On-Demand Unstable AMP1_PLAFQ 42 33 COc1cc(N)c(Cl)cc1C(=O)OCCC1CC1 ZINC000217705746 CF On-Demand Unstable HTR3A 38 61 COc1cc(N)c(Cl)cc1C(=O)OCCC1CC1 ZINC000217705746 CF On-Demand Unstable HTR4 146 69 COc1ccc(-c2cccnc2C=O)cc1 ZINC000217705747 BF For-Sale Unstable LUCI_PHOPE 40 38 Clc1ccccc1CN[C@@H]1CCN2CCC[C@@H]12 ZINC000217705748 CF For-Sale Unstable SLC6A1 0 47 Clc1ccccc1CN[C@@H]1CCN2CCC[C@@H]12 ZINC000217705748 CF For-Sale Unstable SLC18A3 45 35 COc1ccccc1/C=C/NC(=O)Nc1ccc(O)cc1 ZINC000217705755 CG For-Sale Unstable PDGFRA 40 34 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1cnn(CC(N)=O)c1 ZINC000217705757 CE For-Sale Unstable TRPM8 16 43 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(Cl)cc1Cl ZINC000217705761 FK In-Stock Unstable PTGER1 32 42 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(Cl)cc1Cl ZINC000217705761 FK In-Stock Unstable CYP1A1 15 40 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(Cl)cc1Cl ZINC000217705761 FK In-Stock Unstable TUBB1 51 38 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(Cl)cc1Cl ZINC000217705761 FK In-Stock Unstable AKR1C3 28 41 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(Cl)cc1Cl ZINC000217705761 FK In-Stock Unstable ABCG2 17 45 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(Cl)cc1Cl ZINC000217705761 FK In-Stock Unstable NFE2L2 0 40 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc(Cl)cc1Cl ZINC000217705761 FK In-Stock Unstable CYSP_PLAFA 43 42 C/C(=C/C(=O)O)CN1CCc2ccccc2CC1 ZINC000217705790 BE For-Sale Unstable CHRNA6 0 44 C/C(=C/C(=O)O)CN1CCc2ccccc2CC1 ZINC000217705790 BE For-Sale Unstable MTNR1B 28 43 C/C(=C/C(=O)O)CN1CCc2ccccc2CC1 ZINC000217705790 BE For-Sale Unstable NOD2 41 34 COc1cccc2c1C[C@H](N)CCC2 ZINC000217705825 AD For-Sale Unstable HTR1A 25 85 COc1cccc2c1C[C@H](N)CCC2 ZINC000217705825 AD For-Sale Unstable AADAT 19 44 Clc1ccccc1CN[C@H]1CCN2CCC[C@@H]12 ZINC000217705827 CF For-Sale Unstable SLC6A1 0 47 Clc1ccccc1CN[C@H]1CCN2CCC[C@@H]12 ZINC000217705827 CF For-Sale Unstable SLC18A3 45 35 COC(=O)[C@@H](O)CNC(=O)[C@H](C)Oc1ccccc1 ZINC000217705844 CC On-Demand Unstable NPR 41 32 COC(=O)[C@@H](O)CNC(=O)[C@H](C)Oc1ccccc1 ZINC000217705844 CC On-Demand Unstable AMP1_PLAFQ 42 33 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1cnn(CC(N)=O)c1 ZINC000217705849 CE For-Sale Unstable TRPM8 16 43 C[C@@H](CCN(C)C)NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217705856 CD For-Sale Unstable UTS2 80 46 COc1ccccc1/C=C/NC(=O)Nc1cc(Cl)ccc1OC ZINC000217705869 EI For-Sale Unstable CPT1A 43 30 COc1ccccc1/C=C/NC(=O)Nc1cc(Cl)ccc1OC ZINC000217705869 EI For-Sale Unstable RBP4 25 46 COc1ccccc1/C=C/NC(=O)Nc1cc(Cl)ccc1OC ZINC000217705869 EI For-Sale Unstable CYSP_PLAFA 46 39 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc([N+](=O)[O-])cc1 ZINC000217705870 EH In-Stock Unstable ACR 29 46 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc([N+](=O)[O-])cc1 ZINC000217705870 EH In-Stock Unstable AKR1C3 32 42 COc1ccc(/C=C/C(=O)Cl)cc1OCc1ccc([N+](=O)[O-])cc1 ZINC000217705870 EH In-Stock Unstable ABCG2 22 42 COC(=O)[C@H]1[C@@H](C(=O)O)CCC[C@H]1C ZINC000217705871 BD For-Sale Unstable PPM1B 0 46 COC(=O)[C@H]1[C@@H](C(=O)O)CCC[C@H]1C ZINC000217705871 BD For-Sale Unstable PPP1CC 0 46 O=C(Cc1c(F)cccc1Cl)NCCSC1CCOCC1 ZINC000217705893 EG In-Stock Unstable P2RX7 23 46 COc1cccc2c1C[C@@H](N)CCC2 ZINC000217705910 AD For-Sale Unstable HTR1A 25 85 COc1cccc2c1C[C@@H](N)CCC2 ZINC000217705910 AD For-Sale Unstable AADAT 19 44 COc1ccc2[nH]c3c(c2c1)CN(C(=O)[C@H]1CC(=O)N(CC(C)C)C1)CC3 ZINC000217705914 FF In-Stock Unstable MAPKAPK2 20 43 COC(=O)[C@H](O)CNC(=O)[C@H](C)Oc1ccccc1 ZINC000217705928 CC On-Demand Unstable NPR 41 32 COC(=O)[C@H](O)CNC(=O)[C@H](C)Oc1ccccc1 ZINC000217705928 CC On-Demand Unstable AMP1_PLAFQ 42 33 C[C@H](CCN(C)C)NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217705931 CD For-Sale Unstable UTS2 80 46 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1cnn(CC(N)=O)c1 ZINC000217705933 CE For-Sale Unstable TRPM8 16 43 c1ccc2c(CN[C@@H]3CCN4CCC[C@@H]34)cccc2c1 ZINC000217705940 CG For-Sale Unstable KCNB1 0 42 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NCCc1ccc(OC)cc1 ZINC000217705948 GE In-Stock Unstable TBXA2R 38 45 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NCCc1ccc(OC)cc1 ZINC000217705948 GE In-Stock Unstable TBXAS1 15 41 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NCCc1ccc(OC)cc1 ZINC000217705948 GE In-Stock Unstable MMP13 23 40 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NCCc1ccc(OC)cc1 ZINC000217705948 GE In-Stock Unstable PTGDR 28 40 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NCCc1ccc(OC)cc1 ZINC000217705948 GE In-Stock Unstable CA9 17 40 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NCCc1ccc(OC)cc1 ZINC000217705948 GE In-Stock Unstable AKR1C3 30 51 COC(=O)[C@@H]1[C@H](C)CCC[C@H]1C(=O)O ZINC000217705951 BD For-Sale Unstable Q8AWE3_CHICK 19 46 CCCCc1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217705979 DJ For-Sale Unstable INHA 51 37 CCCCc1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217705979 DJ For-Sale Unstable MTNR1B 16 44 CCCCc1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217705979 DJ For-Sale Unstable CFTR 44 36 CCCCc1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217705979 DJ For-Sale Unstable ACAT 0 46 O=C(OCCC1CC1)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217705993 CG On-Demand Unstable APLNR 0 44 COc1ccc(/C=C/C(=O)Cl)cc1OCc1cccc2ccccc12 ZINC000217705997 FK In-Stock Unstable TSHR 54 34 COc1ccc(/C=C/C(=O)Cl)cc1OCc1cccc2ccccc12 ZINC000217705997 FK In-Stock Unstable PTGER2 15 45 COc1ccc(/C=C/C(=O)Cl)cc1OCc1cccc2ccccc12 ZINC000217705997 FK In-Stock Unstable PTGER4 23 45 COc1ccc(/C=C/C(=O)Cl)cc1OCc1cccc2ccccc12 ZINC000217705997 FK In-Stock Unstable CYP1B1 24 40 COc1ccc(/C=C/C(=O)Cl)cc1OCc1cccc2ccccc12 ZINC000217705997 FK In-Stock Unstable KCNA3 0 42 COc1ccc(/C=C/C(=O)Cl)cc1OCc1cccc2ccccc12 ZINC000217705997 FK In-Stock Unstable TNFRSF1A 23 40 COc1ccc(/C=C/C(=O)Cl)cc1OCc1cccc2ccccc12 ZINC000217705997 FK In-Stock Unstable MTNR1A 30 40 COc1ccc(/C=C/C(=O)Cl)cc1OCc1cccc2ccccc12 ZINC000217705997 FK In-Stock Unstable MTNR1B 28 40 COc1ccc(/C=C/C(=O)Cl)cc1OCc1cccc2ccccc12 ZINC000217705997 FK In-Stock Unstable CYP1A1 24 40 COc1ccc(/C=C/C(=O)Cl)cc1OCc1cccc2ccccc12 ZINC000217705997 FK In-Stock Unstable TUBB1 52 40 COc1ccc(/C=C/C(=O)Cl)cc1OCc1cccc2ccccc12 ZINC000217705997 FK In-Stock Unstable AKR1C3 30 45 COc1ccc(/C=C/C(=O)Cl)cc1OCc1cccc2ccccc12 ZINC000217705997 FK In-Stock Unstable PTPA 0 48 COc1ccc(/C=C/C(=O)Cl)cc1OCc1cccc2ccccc12 ZINC000217705997 FK In-Stock Unstable ABCG2 26 53 COc1ccc(/C=C/C(=O)Cl)cc1OCc1cccc2ccccc12 ZINC000217705997 FK In-Stock Unstable PDEB1 0 47 COc1ccc(/C=C/C(=O)Cl)cc1OCc1cccc2ccccc12 ZINC000217705997 FK In-Stock Unstable CYSP_PLAFA 43 46 O=C(O)/C=C\c1ccc(C(=O)N2CCC[C@H](O)C2)cc1 ZINC000217706011 CD For-Sale Unstable GRM3 15 52 O=C(O)/C=C\c1ccc(C(=O)N2CCC[C@H](O)C2)cc1 ZINC000217706011 CD For-Sale Unstable L3MBTL3 70 42 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1cnn(CC(N)=O)c1 ZINC000217706016 CE For-Sale Unstable TRPM8 16 43 COC(=O)[C@@H]1[C@@H](C)CCC[C@H]1C(=O)O ZINC000217706033 BD For-Sale Unstable Q8AWE3_CHICK 19 46 c1ccc2c(CN[C@H]3CCN4CCC[C@@H]34)cccc2c1 ZINC000217706035 CG For-Sale Unstable KCNB1 0 42 CN(Cc1ccc2ncccc2c1)C(=O)Cc1ccc(O)c(Cl)c1 ZINC000217706048 EH In-Stock Unstable NCE103 28 41 CN(Cc1ccc2ncccc2c1)C(=O)Cc1ccc(O)c(Cl)c1 ZINC000217706048 EH In-Stock Unstable CAN2 0 42 COC(=O)[C@@H](O)CNC(=O)CNC(=O)c1cccc(Br)c1 ZINC000217706056 FB On-Demand Unstable DRD4 40 31 COC(=O)[C@@H](O)CNC(=O)CNC(=O)c1cccc(Br)c1 ZINC000217706056 FB On-Demand Unstable CCR2 41 41 COc1ccccc1-n1nc(C(=O)O)cc1O ZINC000217706087 BD In-Stock Unstable HTR1A 41 40 COc1ccccc1-n1nc(C(=O)O)cc1O ZINC000217706087 BD In-Stock Unstable TACR3 20 41 COc1ccccc1-n1nc(C(=O)O)cc1O ZINC000217706087 BD In-Stock Unstable ALS 47 37 COc1ccccc1-n1nc(C(=O)O)cc1O ZINC000217706087 BD In-Stock Unstable RPA1 71 47 COc1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217706095 CG For-Sale Unstable CYP1B1 41 48 COc1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217706095 CG For-Sale Unstable CA1 49 42 COc1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217706095 CG For-Sale Unstable MTNR1A 16 47 COc1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217706095 CG For-Sale Unstable MTNR1B 23 47 COc1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217706095 CG For-Sale Unstable CA12 22 44 COc1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217706095 CG For-Sale Unstable PDGFRA 54 40 COc1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217706095 CG For-Sale Unstable IMPDH2 0 42 COc1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217706095 CG For-Sale Unstable CA9 23 44 COc1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217706095 CG For-Sale Unstable Q8MMZ8_EIMTE 0 42 COc1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217706095 CG For-Sale Unstable AKR1C3 15 40 CCOc1cc(C(=O)Cl)ccc1OCc1ccc(Cl)cc1Cl ZINC000217706100 FK In-Stock Unstable PTGER1 66 46 CCOc1cc(C(=O)Cl)ccc1OCc1ccc(Cl)cc1Cl ZINC000217706100 FK In-Stock Unstable TTR 0 40 CC(=O)NCC1CCN(C(=O)c2ccncc2Cl)CC1 ZINC000217706101 CD On-Demand Unstable CACNA1I 45 34 O=C(O)/C=C\c1ccc(C(=O)N2CCC[C@@H](O)C2)cc1 ZINC000217706105 CD For-Sale Unstable GRM3 15 52 O=C(O)/C=C\c1ccc(C(=O)N2CCC[C@@H](O)C2)cc1 ZINC000217706105 CD For-Sale Unstable L3MBTL3 70 42 C[C@](O)(CNC(=O)/C=C\c1cccc(Br)c1)CC(=O)O ZINC000217706138 ED For-Sale Unstable HDAC8 57 38 C[C@](O)(CNC(=O)/C=C\c1cccc(Br)c1)CC(=O)O ZINC000217706138 ED For-Sale Unstable HDAC6 36 40 C[C@](O)(CNC(=O)/C=C\c1cccc(Br)c1)CC(=O)O ZINC000217706138 ED For-Sale Unstable HPSE 15 40 CCNc1ccc(S(=O)(=O)NCCOC)cc1C(=O)O ZINC000217706203 DC In-Stock Unstable BDKRB1 0 44 CCCOc1ccc(N2C[C@H](C(=O)Cl)CC2=O)cc1 ZINC000217706207 CF In-Stock Unstable PLA2G4B 49 30 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)cc1Cl ZINC000217706210 EJ For-Sale Unstable PYGL 23 48 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)cc1Cl ZINC000217706210 EJ For-Sale Unstable CYSP_PLAFA 41 41 C[C@@](O)(CNC(=O)/C=C\c1cccc(Br)c1)CC(=O)O ZINC000217706216 ED For-Sale Unstable HDAC8 57 38 C[C@@](O)(CNC(=O)/C=C\c1cccc(Br)c1)CC(=O)O ZINC000217706216 ED For-Sale Unstable HDAC6 36 40 C[C@@](O)(CNC(=O)/C=C\c1cccc(Br)c1)CC(=O)O ZINC000217706216 ED For-Sale Unstable HPSE 15 40 O=C(OCCC1CC1)c1cc([N+](=O)[O-])ccc1Cl ZINC000217706226 CG On-Demand Unstable CACNA1C 49 38 O=C(OCCC1CC1)c1cc([N+](=O)[O-])ccc1Cl ZINC000217706226 CG On-Demand Unstable CACNA1D 77 38 O=C(OCCC1CC1)c1cc([N+](=O)[O-])ccc1Cl ZINC000217706226 CG On-Demand Unstable SLC27A4 50 34 COC(=O)[C@@H](O)CNC(=O)c1cc([N+](=O)[O-])ccc1C ZINC000217706238 CC On-Demand Unstable CACNA1C 57 37 COC(=O)[C@@H](O)CNC(=O)c1cc([N+](=O)[O-])ccc1C ZINC000217706238 CC On-Demand Unstable CACNA1D 86 37 CCNc1ccc(S(=O)(=O)NCCCOC(C)C)cc1C(=O)O ZINC000217706301 ED In-Stock Unstable CASP3 16 42 CCCOc1ccc(N2C[C@@H](C(=O)Cl)CC2=O)cc1 ZINC000217706310 CF In-Stock Unstable PLA2G4B 49 30 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)Nc3ccc(O)cc3)[C@H]21 ZINC000217706317 JG In-Stock Unstable TSHR 66 36 COC(=O)[C@H](O)CNC(=O)c1cc([N+](=O)[O-])ccc1C ZINC000217706318 CC On-Demand Unstable CACNA1C 57 37 COC(=O)[C@H](O)CNC(=O)c1cc([N+](=O)[O-])ccc1C ZINC000217706318 CC On-Demand Unstable CACNA1D 86 37 COc1ccccc1/C=C/NC(=O)NCCc1ccc(O)cc1 ZINC000217706338 DF For-Sale Unstable SLC6A5 21 41 COc1ccccc1/C=C/NC(=O)NCCc1ccc(O)cc1 ZINC000217706338 DF For-Sale Unstable AKR1B10 41 45 O=C(O)c1cc(O)n(-c2cc(Cl)c(Cl)cc2Cl)n1 ZINC000217706404 DG In-Stock Anodyne RPA1 89 43 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)Nc3ccc(O)cc3)[C@@H]21 ZINC000217706407 JG In-Stock Unstable TSHR 66 36 O=C(Cl)/C=C/c1cccc(OCc2cccc3ccccc23)c1 ZINC000217706429 DK In-Stock Unstable CYSLTR1 21 44 O=C(Cl)/C=C/c1cccc(OCc2cccc3ccccc23)c1 ZINC000217706429 DK In-Stock Unstable UL80 15 42 O=C(Cl)/C=C/c1cccc(OCc2cccc3ccccc23)c1 ZINC000217706429 DK In-Stock Unstable CDC25B 0 41 O=C(Cl)/C=C/c1cccc(OCc2cccc3ccccc23)c1 ZINC000217706429 DK In-Stock Unstable 17HSDCL 0 41 COc1ccccc1/C=C/NC(=O)NC(C)C ZINC000217706444 BE For-Sale Unstable CYP1B1 19 41 COc1ccccc1/C=C/NC(=O)NC(C)C ZINC000217706444 BE For-Sale Unstable TLR4 19 47 COC(=O)[C@@H](O)CNC(=O)CCCOc1ccccc1 ZINC000217706449 CC On-Demand Unstable LTA4H 35 42 COC(=O)[C@@H](O)CNC(=O)CCCOc1ccccc1 ZINC000217706449 CC On-Demand Unstable PLA2G4B 59 35 O=C(NCCSC1CCOCC1)c1cccc(Cl)c1 ZINC000217706451 CF In-Stock Unstable DRD4 44 36 CCNc1ccc(S(=O)(=O)NCCC2=CCCCC2)cc1C(=O)O ZINC000217706515 FF In-Stock Unstable TBXA2R 41 34 COC(=O)[C@H](O)CNC(=O)CCCOc1ccccc1 ZINC000217706531 CC On-Demand Unstable LTA4H 35 42 COC(=O)[C@H](O)CNC(=O)CCCOc1ccccc1 ZINC000217706531 CC On-Demand Unstable PLA2G4B 59 35 O=C(Cl)c1ccc(OCc2ccc(F)cc2Cl)c(Cl)c1 ZINC000217706540 EK In-Stock Unstable PTGER1 32 48 O=C(Cl)c1ccc(OCc2ccc(F)cc2Cl)c(Cl)c1 ZINC000217706540 EK In-Stock Unstable P2RX7 48 34 COc1ccccc1/C=C/NC(=O)N(Cc1ccccc1)C(C)C ZINC000217706550 DI For-Sale Unstable PTGES 0 43 Clc1ccc(CN[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217706577 CF For-Sale Unstable SLC18A3 17 43 CNc1ccc(C(=O)O)cc1S(=O)(=O)NCCO ZINC000217706617 CB In-Stock Unstable NEU3 0 40 Clc1ccc(CN[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217706643 CF For-Sale Unstable SLC18A3 17 43 O=C(Cl)c1ccc(OCc2ccc(F)cc2)c(Cl)c1 ZINC000217706656 CI In-Stock Unstable PTGER2 0 40 O=C(Cl)c1ccc(OCc2ccc(F)cc2)c(Cl)c1 ZINC000217706656 CI In-Stock Unstable PTGER1 58 44 O=C(Cl)c1ccc(OCc2ccc(F)cc2)c(Cl)c1 ZINC000217706656 CI In-Stock Unstable ACR 37 40 O=C(Cl)c1ccc(OCc2ccc(F)cc2)c(Cl)c1 ZINC000217706656 CI In-Stock Unstable ADCYAP1R1 57 35 O=C(Cl)c1ccc(OCc2ccc(F)cc2)c(Cl)c1 ZINC000217706656 CI In-Stock Unstable KLK_PIG 48 41 CCCCCNS(=O)(=O)c1cc(C(=O)O)ccc1NCC ZINC000217706729 DE In-Stock Unstable PLA2G4B 43 36 Cn1c(=O)n(CCC(=O)N2CCCN(S(=O)(=O)c3ccc(F)cc3)CC2)c2ccccc21 ZINC000217706757 JD On-Demand Unstable ADORA2B 16 40 Cn1c(=O)n(CCC(=O)N2CCCN(S(=O)(=O)c3ccc(F)cc3)CC2)c2ccccc21 ZINC000217706757 JD On-Demand Unstable TGM2 56 38 Cn1c(=O)n(CCC(=O)N2CCCN(S(=O)(=O)c3ccc(F)cc3)CC2)c2ccccc21 ZINC000217706757 JD On-Demand Unstable F13A1 75 41 Cc1c(C(=O)NC[C@@H]2CCCN3CCCC[C@H]23)oc2ccccc12 ZINC000217706759 EH In-Stock Unstable NMT_PLAF7 0 40 Cc1ccccc1COc1ccc(C(=O)Cl)cc1Cl ZINC000217706772 CJ In-Stock Unstable FABP5 28 40 C/C(C(=O)O)=C(/C)C(=O)N1CCc2ccccc2CC1 ZINC000217706824 CE For-Sale Unstable DRD1 20 40 C/C(C(=O)O)=C(/C)C(=O)N1CCc2ccccc2CC1 ZINC000217706824 CE For-Sale Unstable DRD5 42 40 CCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217706841 HE In-Stock Unstable TBXA2R 51 40 CCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217706841 HE In-Stock Unstable TBXAS1 17 44 CCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217706841 HE In-Stock Unstable IAP 0 46 CCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217706841 HE In-Stock Unstable AKR1C3 15 46 CCNc1ccc(S(=O)(=O)NCCc2ccc(OC)c(OC)c2)cc1C(=O)O ZINC000217706841 HE In-Stock Unstable SCMU_MYCTU 0 44 Cc1cc(C)nc(NCCCC(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)n1 ZINC000217706876 GE In-Stock Unstable CHRNA4 29 52 O=[N+]([O-])c1ccc(NCc2cnn(-c3ccccc3)c2)cc1C(F)(F)F ZINC000217706879 FI On-Demand Unstable SERPINE1 23 40 Cc1ccc(COc2ccc(C(=O)Cl)cc2Cl)cc1 ZINC000217706905 CJ In-Stock Unstable PTGER1 43 42 Cc1ccc(COc2ccc(C(=O)Cl)cc2Cl)cc1 ZINC000217706905 CJ In-Stock Unstable PPARD 15 41 Cc1ccc(COc2ccc(C(=O)Cl)cc2Cl)cc1 ZINC000217706905 CJ In-Stock Unstable ACR 40 40 Cc1ccc(COc2ccc(C(=O)Cl)cc2Cl)cc1 ZINC000217706905 CJ In-Stock Unstable KLK_PIG 48 41 CCOc1cc(C(=O)NCCSC2CCOCC2)cc(OCC)c1OCC ZINC000217706913 GH In-Stock Unstable CACNA1I 47 34 O=C(O)/C=C\c1ccccc1CCCBr ZINC000217706917 CG For-Sale Unstable PTGER2 15 53 O=C(O)/C=C\c1ccccc1CCCBr ZINC000217706917 CG For-Sale Unstable PTGER3 21 55 Cc1ccc(/C=C\C(=O)NC[C@](C)(O)CC(=O)O)cc1 ZINC000217706986 CD For-Sale Unstable HDAC8 0 41 Cc1ccc(/C=C\C(=O)NC[C@](C)(O)CC(=O)O)cc1 ZINC000217706986 CD For-Sale Unstable MMP2 15 47 Cc1ccc(/C=C\C(=O)NC[C@](C)(O)CC(=O)O)cc1 ZINC000217706986 CD For-Sale Unstable HDAC1 16 41 O=C(O)/C=C/c1ccccc1CCCBr ZINC000217706998 CG For-Sale Unstable PTGER2 20 53 O=C(O)/C=C/c1ccccc1CCCBr ZINC000217706998 CG For-Sale Unstable PTGER4 22 45 O=C(O)/C=C/c1ccccc1CCCBr ZINC000217706998 CG For-Sale Unstable PTGER3 23 55 O=C(O)/C=C/c1ccccc1CCCBr ZINC000217706998 CG For-Sale Unstable PTGDR 19 50 O=C(Cl)c1ccc(OCc2cccc(F)c2)c(Cl)c1 ZINC000217707007 CI In-Stock Unstable EGFR 61 48 O=C(Cl)c1ccc(OCc2cccc(F)c2)c(Cl)c1 ZINC000217707007 CI In-Stock Unstable MAOB 23 44 O=C(Cl)c1ccc(OCc2cccc(F)c2)c(Cl)c1 ZINC000217707007 CI In-Stock Unstable ERBB2 74 48 O=C(Cl)c1ccc(OCc2cccc(F)c2)c(Cl)c1 ZINC000217707007 CI In-Stock Unstable PTGER1 70 39 O=C(Cl)c1ccc(OCc2cccc(F)c2)c(Cl)c1 ZINC000217707007 CI In-Stock Unstable ACR 32 40 O=C(Cl)c1ccc(OCc2cccc(F)c2)c(Cl)c1 ZINC000217707007 CI In-Stock Unstable AKR1C3 16 43 O=C(Cl)c1ccc(OCc2cccc(F)c2)c(Cl)c1 ZINC000217707007 CI In-Stock Unstable ADCYAP1R1 44 37 O=C(Cl)c1ccc(OCc2cccc(F)c2)c(Cl)c1 ZINC000217707007 CI In-Stock Unstable KLK_PIG 45 39 O=C(O)/C=C\c1cccc(S(=O)(=O)N2CCNC(=O)C2)c1 ZINC000217707021 DB For-Sale Unstable AKR1C3 67 41 CCOC(=O)C1CCN(C(=O)N/C=C/c2ccccc2OC)CC1 ZINC000217707036 EF For-Sale Unstable FDFT1 0 42 Cc1ccc(/C=C\C(=O)NC[C@@](C)(O)CC(=O)O)cc1 ZINC000217707075 CD For-Sale Unstable HDAC8 0 41 Cc1ccc(/C=C\C(=O)NC[C@@](C)(O)CC(=O)O)cc1 ZINC000217707075 CD For-Sale Unstable MMP2 15 47 Cc1ccc(/C=C\C(=O)NC[C@@](C)(O)CC(=O)O)cc1 ZINC000217707075 CD For-Sale Unstable HDAC1 16 41 O=C(Cl)c1ccc(OCc2ccccc2F)c(Cl)c1 ZINC000217707127 CI In-Stock Unstable PTGER1 63 48 O=C(Cl)c1ccc(OCc2ccccc2F)c(Cl)c1 ZINC000217707127 CI In-Stock Unstable FABP4 18 40 O=C(Cl)c1ccc(OCc2ccccc2F)c(Cl)c1 ZINC000217707127 CI In-Stock Unstable FABP5 28 40 COc1ccccc1/C=C/NC(=O)NC1CCCCC1 ZINC000217707143 CG For-Sale Unstable FAAH 16 41 COc1ccccc1/C=C/NC(=O)NC1CCCCC1 ZINC000217707143 CG For-Sale Unstable EPHX2 28 46 Cc1cc(NS(=O)(=O)c2cccc(/C=C\C(=O)O)c2)no1 ZINC000217707184 DD For-Sale Unstable PPIA 22 50 Cc1cc(NS(=O)(=O)c2cccc(/C=C\C(=O)O)c2)no1 ZINC000217707184 DD For-Sale Unstable HDAC8 34 50 Cc1cc(NS(=O)(=O)c2cccc(/C=C\C(=O)O)c2)no1 ZINC000217707184 DD For-Sale Unstable PFK 0 46 COc1ccc(CN[C@@H]2CCN3CCC[C@@H]23)cc1OC ZINC000217707197 CE For-Sale Unstable MT-ND1 18 40 O=C(Cl)c1ccc(OCc2ccccc2Cl)c(Cl)c1 ZINC000217707231 DJ In-Stock Unstable PTGER1 50 46 O=C(Cl)c1ccc(OCc2ccccc2Cl)c(Cl)c1 ZINC000217707231 DJ In-Stock Unstable FABP4 19 52 O=C(Cl)c1ccc(OCc2ccccc2Cl)c(Cl)c1 ZINC000217707231 DJ In-Stock Unstable FABP5 36 52 CCNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217707267 EE In-Stock Unstable CCR8 82 42 CCNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217707267 EE In-Stock Unstable SFRP1 101 36 CCNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217707267 EE In-Stock Unstable WNT3 80 36 COc1ccc(CN[C@H]2CCN3CCC[C@@H]23)cc1OC ZINC000217707289 CE For-Sale Unstable MT-ND1 18 40 CSCC[C@@H](CO)NC(=O)c1cc(CC(C)C)nc2ccccc12 ZINC000217707340 EG In-Stock Unstable TACR2 0 40 CSCC[C@@H](CO)NC(=O)c1cc(CC(C)C)nc2ccccc12 ZINC000217707340 EG In-Stock Unstable TACR3 37 43 O=C(Cl)c1ccc(OCc2ccc(Cl)cc2Cl)c(Cl)c1 ZINC000217707346 FK In-Stock Unstable PTGER1 63 49 O=C(Cl)c1ccc(OCc2ccc(Cl)cc2Cl)c(Cl)c1 ZINC000217707346 FK In-Stock Unstable S1PR4 25 42 COc1ccccc1/C=C/NC(=O)N1CCC(C(=O)O)CC1 ZINC000217707370 DE For-Sale Unstable SLC6A1 48 39 COc1ccccc1/C=C/NC(=O)N1CCC(C(=O)O)CC1 ZINC000217707370 DE For-Sale Unstable ITGAL 35 48 Nc1cc(C(F)(F)F)ccc1C(=O)OCCC1CC1 ZINC000217707375 CG On-Demand Unstable LIPG 54 50 COc1ccc(CN[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217707405 BE For-Sale Unstable SIGMAR1 20 49 C[C@H](NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1)C1CC1 ZINC000217707450 CD For-Sale Unstable HDAC8 30 48 C[C@H](NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1)C1CC1 ZINC000217707450 CD For-Sale Unstable LEF 21 42 O=C(Cl)c1ccc(OCc2ccc(Cl)cc2)c(Cl)c1 ZINC000217707464 DJ In-Stock Unstable PTGER1 74 46 O=C(Cl)c1ccc(OCc2ccc(Cl)cc2)c(Cl)c1 ZINC000217707464 DJ In-Stock Unstable CCR5 21 43 O=C(Cl)c1ccc(OCc2ccc(Cl)cc2)c(Cl)c1 ZINC000217707464 DJ In-Stock Unstable ACR 39 44 O=C(Cl)c1ccc(OCc2ccc(Cl)cc2)c(Cl)c1 ZINC000217707464 DJ In-Stock Unstable TTR 0 40 O=C(Cl)c1ccc(OCc2ccc(Cl)cc2)c(Cl)c1 ZINC000217707464 DJ In-Stock Unstable KLK_PIG 50 43 Cc1nc(CCNC(=O)c2ccncc2Cl)no1 ZINC000217707490 CD For-Sale Unstable F9 27 40 COc1ccc(CN[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217707491 BE For-Sale Unstable SIGMAR1 20 49 COc1ccccc1/C=C/NC(=O)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217707494 IJ For-Sale Unstable NMUR2 0 45 COc1ccccc1/C=C/NC(=O)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217707494 IJ For-Sale Unstable NMUR1 0 45 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NCCc1ccccc1 ZINC000217707499 EE In-Stock Unstable TBXA2R 44 38 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NCCc1ccccc1 ZINC000217707499 EE In-Stock Unstable AKR1C3 22 58 CCCCCCCC/C=C\C=C/C(=O)NCC(C)C ZINC000217707539 CJ Annotated Unstable CNR1 17 59 CCCCCCCC/C=C\C=C/C(=O)NCC(C)C ZINC000217707539 CJ Annotated Unstable PPARA 0 65 CCCCCCCC/C=C\C=C/C(=O)NCC(C)C ZINC000217707539 CJ Annotated Unstable CNR2 0 63 CCCCCCCC/C=C\C=C/C(=O)NCC(C)C ZINC000217707539 CJ Annotated Unstable FABP4 15 41 CCCCCCCC/C=C\C=C/C(=O)NCC(C)C ZINC000217707539 CJ Annotated Unstable FAAH 33 44 CCCCCCCC/C=C\C=C/C(=O)NCC(C)C ZINC000217707539 CJ Annotated Unstable EPHX2 0 40 CCCCCCCC/C=C\C=C/C(=O)NCC(C)C ZINC000217707539 CJ Annotated Unstable Q6UB75_PIG 0 41 CCCCCCCC/C=C\C=C/C(=O)NCC(C)C ZINC000217707539 CJ Annotated Unstable FABP3 32 41 C[C@@H](NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1)C1CC1 ZINC000217707551 CD For-Sale Unstable HDAC8 30 48 C[C@@H](NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1)C1CC1 ZINC000217707551 CD For-Sale Unstable LEF 21 42 O=C(Cl)c1ccc2oc(-c3ccccc3Br)nc2c1 ZINC000217707579 EJ In-Stock Reactive HPSE 58 34 O=C(Cl)c1ccc2oc(-c3ccccc3Br)nc2c1 ZINC000217707579 EJ In-Stock Reactive AGPAT2 38 40 COc1ccccc1/C=C\C(=O)NC[C@](C)(O)CC(=O)O ZINC000217707589 CD For-Sale Unstable DRD3 16 49 O=C(NCCSC1CCOCC1)Nc1ccccc1 ZINC000217707590 CF In-Stock Unstable ACAT 0 40 O=C(NCCSC1CCOCC1)Nc1ccccc1 ZINC000217707590 CF In-Stock Unstable P95276_MYCTO 0 41 COc1ccc(Cl)cc1-n1nc(C(=O)O)cc1O ZINC000217707600 CD In-Stock Unstable PTGER1 44 36 COc1ccc(Cl)cc1-n1nc(C(=O)O)cc1O ZINC000217707600 CD In-Stock Unstable CPT1A 59 34 COc1ccc(Cl)cc1-n1nc(C(=O)O)cc1O ZINC000217707600 CD In-Stock Unstable CPT2 43 33 COc1ccc(Cl)cc1-n1nc(C(=O)O)cc1O ZINC000217707600 CD In-Stock Unstable CPT1B 45 33 COc1ccc(Cl)cc1-n1nc(C(=O)O)cc1O ZINC000217707600 CD In-Stock Unstable RPA1 73 45 COc1ccc(CN[C@@H]2CCN3CCC[C@@H]23)c(OC)c1 ZINC000217707606 CE For-Sale Unstable TACR1 21 44 COc1ccccc1/C=C/NC(=O)NCC(C)C ZINC000217707623 BF For-Sale Unstable TLR4 15 44 Cc1cc(S(=O)(=O)N[C@@H](C)C2CC2)ccc1/C=C\C(=O)O ZINC000217707629 DE For-Sale Unstable LEF 37 47 CCCCCCCC/C=C/C=C\C(=O)NCC(C)C ZINC000217707635 CJ Annotated Unstable CNR1 17 59 CCCCCCCC/C=C/C=C\C(=O)NCC(C)C ZINC000217707635 CJ Annotated Unstable PPARA 0 65 CCCCCCCC/C=C/C=C\C(=O)NCC(C)C ZINC000217707635 CJ Annotated Unstable CNR2 0 63 CCCCCCCC/C=C/C=C\C(=O)NCC(C)C ZINC000217707635 CJ Annotated Unstable FABP4 15 41 CCCCCCCC/C=C/C=C\C(=O)NCC(C)C ZINC000217707635 CJ Annotated Unstable FAAH 33 44 CCCCCCCC/C=C/C=C\C(=O)NCC(C)C ZINC000217707635 CJ Annotated Unstable EPHX2 0 40 CCCCCCCC/C=C/C=C\C(=O)NCC(C)C ZINC000217707635 CJ Annotated Unstable Q6UB75_PIG 0 41 CCCCCCCC/C=C/C=C\C(=O)NCC(C)C ZINC000217707635 CJ Annotated Unstable FABP3 32 41 COc1ccccc1/C=C\C(=O)NC[C@@](C)(O)CC(=O)O ZINC000217707675 CD For-Sale Unstable DRD3 16 49 COc1ccc(CN[C@H]2CCN3CCC[C@@H]23)c(OC)c1 ZINC000217707677 CE For-Sale Unstable TACR1 21 44 COc1c(Cl)cc(-c2nc3cc(C(=O)Cl)ccc3o2)cc1Cl ZINC000217707684 FK In-Stock Unstable CETP 0 42 COc1c(Cl)cc(-c2nc3cc(C(=O)Cl)ccc3o2)cc1Cl ZINC000217707684 FK In-Stock Unstable HPSE 58 40 COc1c(Cl)cc(-c2nc3cc(C(=O)Cl)ccc3o2)cc1Cl ZINC000217707684 FK In-Stock Unstable AGPAT2 38 42 O=C(NCCSC1CCOCC1)Nc1ccc(F)cc1 ZINC000217707715 CF In-Stock Unstable CCR3 26 42 O=C(NCC1CCCCCC1)c1ccc2nc[nH]c2c1 ZINC000217707717 CG For-Sale Unstable HTR4 19 42 O=C(NCC1CCCCCC1)c1ccc2nc[nH]c2c1 ZINC000217707717 CG For-Sale Unstable GRIN2B 21 44 O=C(NCC1CCCCCC1)c1ccc2nc[nH]c2c1 ZINC000217707717 CG For-Sale Unstable CACNA1I 63 40 CCCCCCCC/C=C\C=C\C(=O)NCC(C)C ZINC000217707720 CJ Annotated Unstable CNR1 17 59 CCCCCCCC/C=C\C=C\C(=O)NCC(C)C ZINC000217707720 CJ Annotated Unstable PPARA 0 65 CCCCCCCC/C=C\C=C\C(=O)NCC(C)C ZINC000217707720 CJ Annotated Unstable CNR2 0 63 CCCCCCCC/C=C\C=C\C(=O)NCC(C)C ZINC000217707720 CJ Annotated Unstable FABP4 15 41 CCCCCCCC/C=C\C=C\C(=O)NCC(C)C ZINC000217707720 CJ Annotated Unstable FAAH 33 44 CCCCCCCC/C=C\C=C\C(=O)NCC(C)C ZINC000217707720 CJ Annotated Unstable EPHX2 0 40 CCCCCCCC/C=C\C=C\C(=O)NCC(C)C ZINC000217707720 CJ Annotated Unstable Q6UB75_PIG 0 41 CCCCCCCC/C=C\C=C\C(=O)NCC(C)C ZINC000217707720 CJ Annotated Unstable FABP3 32 41 Cc1cc(S(=O)(=O)N[C@H](C)C2CC2)ccc1/C=C\C(=O)O ZINC000217707721 DE For-Sale Unstable LEF 37 47 COCCNC(=O)N/C=C/c1ccccc1OC ZINC000217707747 CD For-Sale Unstable DRD3 24 41 COCCNC(=O)N/C=C/c1ccccc1OC ZINC000217707747 CD For-Sale Unstable TLR4 15 44 CCCN(CC)CCN[C@@H]1CCc2cc(O)ccc21 ZINC000217707787 CF For-Sale Unstable DRD2 15 44 CCCN(CC)CCN[C@@H]1CCc2cc(O)ccc21 ZINC000217707787 CF For-Sale Unstable DRD3 16 44 CCCN(CC)CCN[C@@H]1CCc2cc(O)ccc21 ZINC000217707787 CF For-Sale Unstable STS 49 34 O=C(Cl)c1ccc2oc(-c3cc(Br)ccc3Cl)nc2c1 ZINC000217707793 FK In-Stock Reactive HPSE 57 39 O=C(Cl)c1ccc2oc(-c3cc(Br)ccc3Cl)nc2c1 ZINC000217707793 FK In-Stock Reactive AGPAT2 48 47 O=C(Cl)c1ccc2oc(-c3cc(Br)ccc3Cl)nc2c1 ZINC000217707793 FK In-Stock Reactive PIM3 0 40 CCCCNC(=O)N/C=C/c1ccccc1OC ZINC000217707859 BF For-Sale Unstable DRD2 17 45 CCCCNC(=O)N/C=C/c1ccccc1OC ZINC000217707859 BF For-Sale Unstable DRD3 30 45 CCCCNC(=O)N/C=C/c1ccccc1OC ZINC000217707859 BF For-Sale Unstable MTNR1A 20 49 CCCCNC(=O)N/C=C/c1ccccc1OC ZINC000217707859 BF For-Sale Unstable MTNR1B 30 45 CCCCNC(=O)N/C=C/c1ccccc1OC ZINC000217707859 BF For-Sale Unstable ACAT 0 51 CCCN(CC)CCN[C@H]1CCc2cc(O)ccc21 ZINC000217707872 CF For-Sale Unstable DRD2 15 44 CCCN(CC)CCN[C@H]1CCc2cc(O)ccc21 ZINC000217707872 CF For-Sale Unstable DRD3 16 44 CCCN(CC)CCN[C@H]1CCc2cc(O)ccc21 ZINC000217707872 CF For-Sale Unstable STS 49 34 COc1cc2c(c(OC)c1OC)-c1ccc(NCCCCCC(=O)Nc3nnn[nH]3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217707873 KF In-Stock Unstable TUBA1A 17 61 COc1cc2c(c(OC)c1OC)-c1ccc(NCCCCCC(=O)Nc3nnn[nH]3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217707873 KF In-Stock Unstable TPPP 0 58 CCOc1cc(C(=O)Cl)cc(Cl)c1OCc1cccc(F)c1 ZINC000217707905 EJ In-Stock Unstable EGFR 43 38 CCOc1cc(C(=O)Cl)cc(Cl)c1OCc1cccc(F)c1 ZINC000217707905 EJ In-Stock Unstable MAOB 22 40 CCOc1cc(C(=O)Cl)cc(Cl)c1OCc1cccc(F)c1 ZINC000217707905 EJ In-Stock Unstable ERBB2 55 40 CCOc1cc(C(=O)Cl)cc(Cl)c1OCc1cccc(F)c1 ZINC000217707905 EJ In-Stock Unstable ADCYAP1R1 49 35 CCNc1ccc(C(=O)O)cc1S(=O)(=O)N[C@@H](C)CC ZINC000217707922 DD In-Stock Unstable NEU3 0 40 CCOCCCNC(=O)N/C=C/c1ccccc1OC ZINC000217707975 CE For-Sale Unstable DRD3 25 42 CCOCCCNC(=O)N/C=C/c1ccccc1OC ZINC000217707975 CE For-Sale Unstable MTNR1B 15 42 Clc1ccc(CN[C@@H]2CCN3CCC[C@@H]23)cc1Cl ZINC000217707984 CG For-Sale Unstable OPRK1 26 47 Clc1ccc(CN[C@@H]2CCN3CCC[C@@H]23)cc1Cl ZINC000217707984 CG For-Sale Unstable SIGMAR1 17 64 Clc1ccc(CN[C@@H]2CCN3CCC[C@@H]23)cc1Cl ZINC000217707984 CG For-Sale Unstable SSTR3 21 48 Clc1ccc(CN[C@@H]2CCN3CCC[C@@H]23)cc1Cl ZINC000217707984 CG For-Sale Unstable KCNB1 0 43 O=C(NCCN1CCSCC1)c1ccncc1Cl ZINC000217707987 CD On-Demand Unstable DRD4 46 37 O=C(NCCN1CCSCC1)c1ccncc1Cl ZINC000217707987 CD On-Demand Unstable PLD2 46 34 CCNc1ccc(C(=O)O)cc1S(=O)(=O)N[C@H](C)CC ZINC000217707996 DD In-Stock Unstable NEU3 0 40 COc1cc([C@H](CC(=O)NCCc2ccc(O)c(O)c2)c2c(O)nc3ccccn3c2=O)ccc1OC(C)C ZINC000217707997 KG In-Stock Unstable CAN2 0 40 CCOc1cc(C(=O)Cl)cc(Br)c1OCc1ccccc1F ZINC000217708012 GJ In-Stock Unstable THRB 15 41 Clc1ccc(CN[C@H]2CCN3CCC[C@@H]23)cc1Cl ZINC000217708055 CG For-Sale Unstable OPRK1 26 47 Clc1ccc(CN[C@H]2CCN3CCC[C@@H]23)cc1Cl ZINC000217708055 CG For-Sale Unstable SIGMAR1 17 64 Clc1ccc(CN[C@H]2CCN3CCC[C@@H]23)cc1Cl ZINC000217708055 CG For-Sale Unstable SSTR3 21 48 Clc1ccc(CN[C@H]2CCN3CCC[C@@H]23)cc1Cl ZINC000217708055 CG For-Sale Unstable KCNB1 0 43 COc1cc([C@@H](CC(=O)NCCc2ccc(O)c(O)c2)c2c(O)nc3ccccn3c2=O)ccc1OC(C)C ZINC000217708072 KG In-Stock Unstable CAN2 0 40 CCNc1ccc(S(=O)(=O)NCCCOC)cc1C(=O)O ZINC000217708103 DD In-Stock Unstable CASP3 18 41 CCNc1ccc(S(=O)(=O)NCCCOC)cc1C(=O)O ZINC000217708103 DD In-Stock Unstable BDKRB1 0 45 CCOc1cc(C(=O)Cl)cc(Br)c1OCc1ccccc1 ZINC000217708122 FJ In-Stock Unstable THRA 35 53 CCOc1cc(C(=O)Cl)cc(Br)c1OCc1ccccc1 ZINC000217708122 FJ In-Stock Unstable PPIA 42 36 CCOc1cc(C(=O)Cl)cc(Br)c1OCc1ccccc1 ZINC000217708122 FJ In-Stock Unstable PTGER1 55 36 CCOc1cc(C(=O)Cl)cc(Br)c1OCc1ccccc1 ZINC000217708122 FJ In-Stock Unstable THRB 31 53 CC[C@H](C(=O)O)N(C)C(=O)/C=C\c1ccc(Cl)cc1Cl ZINC000217708184 DG For-Sale Unstable BOTA 26 47 COC(=O)[C@@H](O)CNC(=O)COc1ccc([N+](=O)[O-])cc1 ZINC000217708194 CB On-Demand Unstable CACNA1D 47 33 O=C(NCCSC1CCOCC1)NC1CCCCC1 ZINC000217708197 CF In-Stock Unstable EPHX2 15 47 CNc1ccc(C(=O)O)cc1S(N)(=O)=O ZINC000217708214 BC In-Stock Unstable CA2 58 43 CNc1ccc(C(=O)O)cc1S(N)(=O)=O ZINC000217708214 BC In-Stock Unstable CA6 28 46 CNc1ccc(C(=O)O)cc1S(N)(=O)=O ZINC000217708214 BC In-Stock Unstable CA1 54 46 CNc1ccc(C(=O)O)cc1S(N)(=O)=O ZINC000217708214 BC In-Stock Unstable CA4 56 46 CCOc1cc(C(=O)Cl)cc(Cl)c1OCc1ccccc1 ZINC000217708231 EJ In-Stock Unstable THRA 15 42 CCOc1cc(C(=O)Cl)cc(Cl)c1OCc1ccccc1 ZINC000217708231 EJ In-Stock Unstable MAOB 19 44 CCOc1cc(C(=O)Cl)cc(Cl)c1OCc1ccccc1 ZINC000217708231 EJ In-Stock Unstable PPIA 42 37 CCOc1cc(C(=O)Cl)cc(Cl)c1OCc1ccccc1 ZINC000217708231 EJ In-Stock Unstable PTGER1 60 41 CCOc1cc(C(=O)Cl)cc(Cl)c1OCc1ccccc1 ZINC000217708231 EJ In-Stock Unstable ADCYAP1R1 38 42 CC[C@@H](C(=O)O)N(C)C(=O)/C=C\c1ccc(Cl)cc1Cl ZINC000217708278 DG For-Sale Unstable BOTA 26 47 COC(=O)[C@H](O)CNC(=O)COc1ccc([N+](=O)[O-])cc1 ZINC000217708281 CB On-Demand Unstable CACNA1D 47 33 O=C(NCCSC1CCOCC1)Nc1ccccc1Cl ZINC000217708297 DG In-Stock Unstable CXCL8 43 35 CN1CCC[C@@H]1CNC(=O)c1ccncc1Cl ZINC000217708298 CD On-Demand Unstable DRD2 31 41 CN1CCC[C@@H]1CNC(=O)c1ccncc1Cl ZINC000217708298 CD On-Demand Unstable PREP 32 54 CN1CCC[C@@H]1CNC(=O)c1ccncc1Cl ZINC000217708298 CD On-Demand Unstable CHRNA10 51 42 CN1CCC[C@@H]1CNC(=O)c1ccncc1Cl ZINC000217708298 CD On-Demand Unstable CACNA1I 48 32 CN1CCC[C@@H]1CNC(=O)c1ccncc1Cl ZINC000217708298 CD On-Demand Unstable FAP 0 54 COc1ccccc1/C=C/NC(=O)N1CCCc2ccccc21 ZINC000217708307 DH For-Sale Unstable DRD2 20 40 COc1ccccc1/C=C/NC(=O)N1CCCc2ccccc21 ZINC000217708307 DH For-Sale Unstable AVPR2 43 45 COc1ccccc1/C=C/NC(=O)N1CCCc2ccccc21 ZINC000217708307 DH For-Sale Unstable DRD3 27 40 CC(=O)c1cccc(-n2nc(C(=O)O)cc2O)c1 ZINC000217708329 BD In-Stock Unstable RPA1 79 49 CCOc1cc(C(=O)Cl)cc(Cl)c1OCc1ccccc1C ZINC000217708331 EK In-Stock Unstable FABP4 15 40 CCOc1cc(C(=O)Cl)cc(Cl)c1OCc1ccccc1C ZINC000217708331 EK In-Stock Unstable FABP5 28 40 COc1ccc(C(=O)N2CCC[C@@H]2c2ccccn2)cc1N1CCOCC1 ZINC000217708352 FF In-Stock Unstable CPT1A 54 36 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)Nc1nc(-c3ccccn3)cs1)C(=O)OC2 ZINC000217708365 JK In-Stock Unstable IMPDH1 0 58 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)Nc1nc(-c3ccccn3)cs1)C(=O)OC2 ZINC000217708365 JK In-Stock Unstable NPY5R 0 40 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)Nc1nc(-c3ccccn3)cs1)C(=O)OC2 ZINC000217708365 JK In-Stock Unstable IMPDH2 0 58 CN(C(=O)OC(C)(C)C)[C@@H](CC#N)C(F)(F)F ZINC000217708371 CF For-Sale Unstable PAPA1_CARPA 43 34 CN1CCC[C@H]1CNC(=O)c1ccncc1Cl ZINC000217708377 CD On-Demand Unstable DRD2 31 41 CN1CCC[C@H]1CNC(=O)c1ccncc1Cl ZINC000217708377 CD On-Demand Unstable PREP 32 54 CN1CCC[C@H]1CNC(=O)c1ccncc1Cl ZINC000217708377 CD On-Demand Unstable CHRNA10 51 42 CN1CCC[C@H]1CNC(=O)c1ccncc1Cl ZINC000217708377 CD On-Demand Unstable CACNA1I 48 32 CN1CCC[C@H]1CNC(=O)c1ccncc1Cl ZINC000217708377 CD On-Demand Unstable FAP 0 54 O=C(NCCSC1CCOCC1)NC12CC3CC(CC(C3)C1)C2 ZINC000217708404 EG In-Stock Unstable EPHX2 92 56 O=C(NCCSC1CCOCC1)NC12CC3CC(CC(C3)C1)C2 ZINC000217708404 EG In-Stock Unstable P95276_MYCTO 0 40 COc1ccc(C(=O)N2CCC[C@H]2c2ccccn2)cc1N1CCOCC1 ZINC000217708423 FF In-Stock Unstable CPT1A 54 36 COc1ccccc1/C=C/NC(=O)NCCc1ccccc1 ZINC000217708425 CG For-Sale Unstable PTGER2 0 42 COc1ccccc1/C=C/NC(=O)NCCc1ccccc1 ZINC000217708425 CG For-Sale Unstable MTNR1A 33 45 COc1ccccc1/C=C/NC(=O)NCCc1ccccc1 ZINC000217708425 CG For-Sale Unstable MTNR1B 33 42 COc1ccccc1/C=C/NC(=O)NCCc1ccccc1 ZINC000217708425 CG For-Sale Unstable AKR1B10 37 43 CCOc1cc(C(=O)Cl)cc(Br)c1OCc1ccccc1C ZINC000217708448 GK In-Stock Unstable THRB 19 56 COc1ccc(C(=O)NCCN(C)C)cc1/C=C\C(=O)O ZINC000217708456 CD For-Sale Unstable DRD4 40 30 CN(C(=O)OC(C)(C)C)[C@H](CC#N)C(F)(F)F ZINC000217708458 CF For-Sale Unstable PAPA1_CARPA 43 34 COc1ccc(NC(=O)CCN2C(=O)c3ccccc3N3C(=O)c4c(ccc(OC)c4OC)[C@H]23)cn1 ZINC000217708487 JG In-Stock Unstable TSHR 42 32 COc1ccc(NC(=O)CCN2C(=O)c3ccccc3N3C(=O)c4c(ccc(OC)c4OC)[C@H]23)cn1 ZINC000217708487 JG In-Stock Unstable ENPP1 55 32 COc1ccccc1/C=C/NC(=O)NC1CCCC1 ZINC000217708545 CF For-Sale Unstable EPHX2 24 44 CCOc1cc(C(=O)Cl)cc(Br)c1OCc1ccc(C)cc1 ZINC000217708558 GK In-Stock Unstable THRA 19 55 CCOc1cc(C(=O)Cl)cc(Br)c1OCc1ccc(C)cc1 ZINC000217708558 GK In-Stock Unstable THRB 22 55 CSC1C[C@@H]2CC[C@H](C1)N2C(=O)CNC(=O)OCc1ccccc1 ZINC000217708563 EF For-Sale Unstable ACE 19 40 CSC1C[C@@H]2CC[C@H](C1)N2C(=O)CNC(=O)OCc1ccccc1 ZINC000217708563 EF For-Sale Unstable CTSB 35 46 CSC1C[C@@H]2CC[C@H](C1)N2C(=O)CNC(=O)OCc1ccccc1 ZINC000217708563 EF For-Sale Unstable PAPA1_CARPA 44 37 CSC1C[C@@H]2CC[C@H](C1)N2C(=O)CNC(=O)OCc1ccccc1 ZINC000217708563 EF For-Sale Unstable CYSP_TRYCR 46 39 CSC1C[C@@H]2CC[C@H](C1)N2C(=O)CNC(=O)OCc1ccccc1 ZINC000217708563 EF For-Sale Unstable CTSK 21 40 CSC1C[C@@H]2CC[C@H](C1)N2C(=O)CNC(=O)OCc1ccccc1 ZINC000217708563 EF For-Sale Unstable PREP 19 51 CSC1C[C@@H]2CC[C@H](C1)N2C(=O)CNC(=O)OCc1ccccc1 ZINC000217708563 EF For-Sale Unstable CAPNS1 51 32 CSC1C[C@@H]2CC[C@H](C1)N2C(=O)CNC(=O)OCc1ccccc1 ZINC000217708563 EF For-Sale Unstable CAPN1 52 35 CSC1C[C@@H]2CC[C@H](C1)N2C(=O)CNC(=O)OCc1ccccc1 ZINC000217708563 EF For-Sale Unstable CAPN2 83 35 CSC1C[C@@H]2CC[C@H](C1)N2C(=O)CNC(=O)OCc1ccccc1 ZINC000217708563 EF For-Sale Unstable NPR 61 37 CSC1C[C@@H]2CC[C@H](C1)N2C(=O)CNC(=O)OCc1ccccc1 ZINC000217708563 EF For-Sale Unstable SLC12A5 42 33 CCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217708565 DE In-Stock Unstable CCR8 83 41 CCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217708565 DE In-Stock Unstable SFRP1 101 37 CCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217708565 DE In-Stock Unstable WNT3 81 36 CCNc1ccc(S(=O)(=O)NC2CCCC2)cc1C(=O)O ZINC000217708565 DE In-Stock Unstable MGAT2 0 42 COc1ccc(NC(=O)CCN2C(=O)c3ccccc3N3C(=O)c4c(ccc(OC)c4OC)[C@@H]23)cn1 ZINC000217708574 JG In-Stock Unstable TSHR 42 32 COc1ccc(NC(=O)CCN2C(=O)c3ccccc3N3C(=O)c4c(ccc(OC)c4OC)[C@@H]23)cn1 ZINC000217708574 JG In-Stock Unstable ENPP1 55 32 COc1cccc(CN[C@@H]2CCN3CCC[C@@H]23)c1 ZINC000217708595 BE For-Sale Unstable VACHT_TETCF 0 40 COc1cccc(CN[C@@H]2CCN3CCC[C@@H]23)c1 ZINC000217708595 BE For-Sale Unstable SIGMAR1 20 49 COc1cccc(CN[C@@H]2CCN3CCC[C@@H]23)c1 ZINC000217708595 BE For-Sale Unstable CHRNA10 55 45 O=C(/C=C\c1cc(Cl)cc(Cl)c1)NCC1CC(O)C1 ZINC000217708602 DF For-Sale Unstable CACNA1I 58 37 Cc1cccc(NC(=O)NCCSC2CCOCC2)c1 ZINC000217708603 CG In-Stock Unstable CCKAR 30 45 Cc1cccc(NC(=O)NCCSC2CCOCC2)c1 ZINC000217708603 CG In-Stock Unstable CCKBR 31 40 Cc1cccc(NC(=O)NCCSC2CCOCC2)c1 ZINC000217708603 CG In-Stock Unstable ACAT 0 45 Cc1cccc(NC(=O)NCCSC2CCOCC2)c1 ZINC000217708603 CG In-Stock Unstable KCNK3 42 37 Cc1cccc(NC(=O)NCCSC2CCOCC2)c1 ZINC000217708603 CG In-Stock Unstable KCNK9 41 37 O=C(O)/C=C\c1ccc(C(=O)NCc2ccccc2)s1 ZINC000217708619 CF For-Sale Unstable PTGER2 26 42 O=C(O)/C=C\c1ccc(C(=O)NCc2ccccc2)s1 ZINC000217708619 CF For-Sale Unstable HDAC1 21 56 COc1ccccc1/C=C/NC(=O)NCc1ccccc1Cl ZINC000217708660 DH For-Sale Unstable PTGER3 17 44 COc1ccccc1/C=C/NC(=O)NCc1ccccc1Cl ZINC000217708660 DH For-Sale Unstable P2RX7 29 40 COc1cccc(CN[C@H]2CCN3CCC[C@@H]23)c1 ZINC000217708674 BE For-Sale Unstable VACHT_TETCF 0 40 COc1cccc(CN[C@H]2CCN3CCC[C@@H]23)c1 ZINC000217708674 BE For-Sale Unstable SIGMAR1 20 49 COc1cccc(CN[C@H]2CCN3CCC[C@@H]23)c1 ZINC000217708674 BE For-Sale Unstable CHRNA10 55 45 CNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217708678 DE In-Stock Unstable CA2 22 42 CNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217708678 DE In-Stock Unstable LPL 33 44 CNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217708678 DE In-Stock Unstable CA1 18 50 CNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217708678 DE In-Stock Unstable CA4 38 42 CNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217708678 DE In-Stock Unstable GRM4 23 48 CNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217708678 DE In-Stock Unstable PRTN3 53 36 CNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217708678 DE In-Stock Unstable AKR1C3 45 42 CNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217708678 DE In-Stock Unstable AKR1C2 65 38 CNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217708678 DE In-Stock Unstable LIMK2 56 43 CNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217708678 DE In-Stock Unstable UQCRB 0 42 CNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217708678 DE In-Stock Unstable MGAT2 0 41 O=C(O)/C=C\c1cccc(C(=O)NCc2ccccc2)c1 ZINC000217708704 CF For-Sale Unstable PTGER2 34 42 O=C(O)/C=C\c1cccc(C(=O)NCc2ccccc2)c1 ZINC000217708704 CF For-Sale Unstable PTGER4 0 42 O=C(O)/C=C\c1cccc(C(=O)NCc2ccccc2)c1 ZINC000217708704 CF For-Sale Unstable HDAC8 39 50 O=C(O)/C=C\c1cccc(C(=O)NCc2ccccc2)c1 ZINC000217708704 CF For-Sale Unstable HDAC1 28 47 O=C(O)/C=C\c1cccc(C(=O)NCc2ccccc2)c1 ZINC000217708704 CF For-Sale Unstable HDAC6 30 61 O=C(O)/C=C\c1cccc(C(=O)NCc2ccccc2)c1 ZINC000217708704 CF For-Sale Unstable KCNK3 42 35 O=C(O)/C=C\c1cccc(C(=O)NCc2ccccc2)c1 ZINC000217708704 CF For-Sale Unstable PDS 51 34 O=C(/C=C\c1ccc(Br)cc1)NCC1CC(O)C1 ZINC000217708713 DE For-Sale Unstable HDAC8 26 41 O=C(/C=C\c1ccc(Br)cc1)NCC1CC(O)C1 ZINC000217708713 DE For-Sale Unstable HDAC2 15 41 O=C(/C=C\c1ccc(Br)cc1)NCC1CC(O)C1 ZINC000217708713 DE For-Sale Unstable HDAC6 15 41 O=C(/C=C\c1ccc(Br)cc1)NCC1CC(O)C1 ZINC000217708713 DE For-Sale Unstable IMA1 0 43 Cn1c(C2CCN(C(=O)COC[C@@H]3CCCCO3)CC2)nc2ccccc21 ZINC000217708764 FF In-Stock Unstable SMO 53 45 Cn1c(C2CCN(C(=O)COC[C@@H]3CCCCO3)CC2)nc2ccccc21 ZINC000217708764 FF In-Stock Unstable ETHR 51 33 COc1ccccc1/C=C/NC(=O)NCCc1ccc(OC)c(OC)c1 ZINC000217708776 FG For-Sale Unstable PTGER4 0 40 COc1ccccc1/C=C/NC(=O)NCCc1ccc(OC)c(OC)c1 ZINC000217708776 FG For-Sale Unstable CYP1B1 19 45 COc1ccccc1/C=C/NC(=O)NCCc1ccc(OC)c(OC)c1 ZINC000217708776 FG For-Sale Unstable MTNR1A 27 45 COc1ccccc1/C=C/NC(=O)NCCc1ccc(OC)c(OC)c1 ZINC000217708776 FG For-Sale Unstable MTNR1B 29 47 COc1ccccc1/C=C/NC(=O)NCCc1ccc(OC)c(OC)c1 ZINC000217708776 FG For-Sale Unstable CYP1A1 18 45 COc1ccccc1/C=C/NC(=O)NCCc1ccc(OC)c(OC)c1 ZINC000217708776 FG For-Sale Unstable ABCB1 0 41 COc1ccccc1/C=C/NC(=O)NCCc1ccc(OC)c(OC)c1 ZINC000217708776 FG For-Sale Unstable ABCG2 23 45 FC(F)(F)c1cccc(CN[C@@H]2CCN3CCC[C@@H]23)c1 ZINC000217708781 CG For-Sale Unstable TACR1 24 42 FC(F)(F)c1cccc(CN[C@@H]2CCN3CCC[C@@H]23)c1 ZINC000217708781 CG For-Sale Unstable CCR2 36 41 CCOc1cc(C(=O)Cl)cc(Cl)c1OCc1ccc(Cl)cc1 ZINC000217708791 FK In-Stock Unstable PTGER1 40 35 COC(=O)[C@@H](O)CNC(=O)c1ccc2c(c1)OCO2 ZINC000217708798 CB On-Demand Unstable EDNRB 42 38 COC(=O)[C@@H](O)CNC(=O)c1ccc2c(c1)OCO2 ZINC000217708798 CB On-Demand Unstable BMP1 44 42 COC(=O)[C@@H](O)CNC(=O)c1ccc2c(c1)OCO2 ZINC000217708798 CB On-Demand Unstable F3 74 35 CO[C@@H]1O[C@H](CO)[C@H](O)[C@@H](O)[C@@H]1N=[N+]=[N-] ZINC000217708815 BA In-Stock Unstable FIMH 50 39 CC(C)(F)CCS(=O)(=O)c1ccc(N)cc1 ZINC000217708834 BE For-Sale Unstable DYR_PNECA 17 42 CC(C)(F)CCS(=O)(=O)c1ccc(N)cc1 ZINC000217708834 BE For-Sale Unstable CYNT 19 42 Cn1c(C2CCN(C(=O)COC[C@H]3CCCCO3)CC2)nc2ccccc21 ZINC000217708843 FF In-Stock Unstable SMO 53 45 Cn1c(C2CCN(C(=O)COC[C@H]3CCCCO3)CC2)nc2ccccc21 ZINC000217708843 FF In-Stock Unstable ETHR 51 33 FC(F)(F)c1cccc(CN[C@H]2CCN3CCC[C@@H]23)c1 ZINC000217708847 CG For-Sale Unstable TACR1 24 42 FC(F)(F)c1cccc(CN[C@H]2CCN3CCC[C@@H]23)c1 ZINC000217708847 CG For-Sale Unstable CCR2 36 41 COC(=O)[C@H](O)CNC(=O)c1ccc2c(c1)OCO2 ZINC000217708878 CB On-Demand Unstable EDNRB 42 38 COC(=O)[C@H](O)CNC(=O)c1ccc2c(c1)OCO2 ZINC000217708878 CB On-Demand Unstable BMP1 44 42 COC(=O)[C@H](O)CNC(=O)c1ccc2c(c1)OCO2 ZINC000217708878 CB On-Demand Unstable F3 74 35 COCCCNC(=O)N/C=C/c1ccccc1OC ZINC000217708881 CE For-Sale Unstable DRD2 19 44 COCCCNC(=O)N/C=C/c1ccccc1OC ZINC000217708881 CE For-Sale Unstable DRD3 34 44 CNc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O ZINC000217708897 EE In-Stock Unstable KCNA5 23 43 CNc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O ZINC000217708897 EE In-Stock Unstable MMP12 50 39 CNc1ccc(S(=O)(=O)N[C@@H](C)c2ccccc2)cc1C(=O)O ZINC000217708897 EE In-Stock Unstable LEF 36 43 CO[C@@H]1O[C@H](CO)[C@H](O)[C@H](O)[C@@H]1N=[N+]=[N-] ZINC000217708898 BA In-Stock Unstable FIMH 50 39 CCOc1cc(C(=O)Cl)cc(Br)c1OCc1ccc(Cl)cc1 ZINC000217708909 HK In-Stock Unstable THRA 19 43 CCOc1cc(C(=O)Cl)cc(Br)c1OCc1ccc(Cl)cc1 ZINC000217708909 HK In-Stock Unstable THRB 21 43 CCOc1cc(C(=O)Cl)cc(Br)c1OCc1ccc(Cl)cc1 ZINC000217708909 HK In-Stock Unstable CCR5 19 40 CCOc1ccccc1CN[C@@H]1CCN2CCC[C@@H]12 ZINC000217708960 CE For-Sale Unstable TACR3 24 40 CCOc1ccccc1CN[C@@H]1CCN2CCC[C@@H]12 ZINC000217708960 CE For-Sale Unstable HCN1 47 36 CCOc1ccccc1CN[C@@H]1CCN2CCC[C@@H]12 ZINC000217708960 CE For-Sale Unstable HCN4 45 36 Cc1cnn(CCNC(=O)c2ccncc2Cl)c1 ZINC000217708967 CD On-Demand Unstable DRD4 40 31 CNc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O ZINC000217708969 EE In-Stock Unstable KCNA5 23 43 CNc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O ZINC000217708969 EE In-Stock Unstable MMP12 50 39 CNc1ccc(S(=O)(=O)N[C@H](C)c2ccccc2)cc1C(=O)O ZINC000217708969 EE In-Stock Unstable LEF 36 43 COc1ccc(CCN2C[C@H](C(=O)NC[C@@H]3CCCN4CCCC[C@H]34)CC2=O)cc1OC ZINC000217709002 IE In-Stock Unstable FKBP1A 41 39 CCCCOCCCNC(=O)N/C=C/c1ccccc1OC ZINC000217709006 DG For-Sale Unstable DRD3 23 42 CCCCOCCCNC(=O)N/C=C/c1ccccc1OC ZINC000217709006 DG For-Sale Unstable MTNR1A 18 45 CCCCOCCCNC(=O)N/C=C/c1ccccc1OC ZINC000217709006 DG For-Sale Unstable MTNR1B 20 41 CCCCOCCCNC(=O)N/C=C/c1ccccc1OC ZINC000217709006 DG For-Sale Unstable ACAT 0 47 O=C(NCCSC1CCOCC1)Nc1ccccc1C(F)(F)F ZINC000217709029 EH In-Stock Unstable RBP4 41 33 CCOc1ccccc1CN[C@H]1CCN2CCC[C@@H]12 ZINC000217709043 CE For-Sale Unstable HCN1 47 36 CCOc1ccccc1CN[C@H]1CCN2CCC[C@@H]12 ZINC000217709043 CE For-Sale Unstable HCN4 45 36 COc1ccc(CCN2C[C@@H](C(=O)NC[C@@H]3CCCN4CCCC[C@H]34)CC2=O)cc1OC ZINC000217709072 IE In-Stock Unstable FKBP1A 41 39 CCNc1ccc(S(=O)(=O)NC(C)C)cc1C(=O)O ZINC000217709104 CD In-Stock Unstable MMP12 49 37 CCNc1ccc(S(=O)(=O)NC(C)C)cc1C(=O)O ZINC000217709104 CD In-Stock Unstable ADAMTS4 43 33 CCNc1ccc(S(=O)(=O)NC(C)C)cc1C(=O)O ZINC000217709104 CD In-Stock Unstable LEF 53 36 CCOc1cc(C(=O)Cl)cc(Cl)c1OCc1ccc(Cl)cc1Cl ZINC000217709120 GK In-Stock Unstable PTGER1 19 40 COc1ccccc1/C=C/NC(=O)NCc1cccnc1 ZINC000217709121 CF For-Sale Unstable PTAFR 41 48 COc1ccccc1/C=C/NC(=O)NCc1cccnc1 ZINC000217709121 CF For-Sale Unstable NAMPT 64 48 O=S(=O)(NCCSC1CCOCC1)c1cccnc1 ZINC000217709142 DD In-Stock Unstable TBXA2R 21 49 CCOc1ccc(CN[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217709166 CE For-Sale Unstable HRH3 19 42 CCOc1ccc(CN[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217709166 CE For-Sale Unstable CHRNA10 40 35 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC(F)F)cc1 ZINC000217709188 CC On-Demand Unstable GCGR 16 41 CNc1ccc(S(=O)(=O)NCCO)cc1C(=O)O ZINC000217709208 CB In-Stock Unstable TBXA2R 48 35 CNc1ccc(S(=O)(=O)NCCO)cc1C(=O)O ZINC000217709208 CB In-Stock Unstable CASP3 0 41 CNc1ccc(S(=O)(=O)NCCO)cc1C(=O)O ZINC000217709208 CB In-Stock Unstable CHUK 19 41 CNc1ccc(S(=O)(=O)NCCO)cc1C(=O)O ZINC000217709208 CB In-Stock Unstable AKR1C3 25 40 COc1ccccc1/C=C/NC(=O)NC(C)(C)C ZINC000217709233 BF For-Sale Unstable CYP1B1 19 41 COc1ccccc1/C=C/NC(=O)NC(C)(C)C ZINC000217709233 BF For-Sale Unstable TLR4 20 47 CCOc1cc(C(=O)Cl)cc(Cl)c1OCc1ccccc1Cl ZINC000217709234 FK In-Stock Unstable FABP4 19 50 CCOc1cc(C(=O)Cl)cc(Cl)c1OCc1ccccc1Cl ZINC000217709234 FK In-Stock Unstable FABP5 36 50 CCOc1ccc(CN[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217709255 CE For-Sale Unstable HRH3 19 42 CCOc1ccc(CN[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217709255 CE For-Sale Unstable CHRNA10 40 35 COC(=O)[C@H](O)CNC(=O)c1ccc(OC(F)F)cc1 ZINC000217709272 CC On-Demand Unstable GCGR 16 41 C[C@H](F)CS(=O)(=O)c1ccc(CCN)cc1 ZINC000217709287 BD For-Sale Unstable CA1 17 53 C[C@H](F)CS(=O)(=O)c1ccc(CCN)cc1 ZINC000217709287 BD For-Sale Unstable CAH_METTE 15 53 C[C@H](F)CS(=O)(=O)c1ccc(CCN)cc1 ZINC000217709287 BD For-Sale Unstable TAAR1 18 41 CCCCN(CCO)C(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217709315 CE For-Sale Unstable PLM2_PLAFA 66 37 COC(=O)c1ccccc1S(=O)(=O)NC1CCC(C)CC1 ZINC000217709329 DE On-Demand Unstable CCR8 86 38 COC(=O)c1ccccc1S(=O)(=O)NC1CCC(C)CC1 ZINC000217709329 DE On-Demand Unstable SFRP1 87 34 COC(=O)c1ccccc1S(=O)(=O)NC1CCC(C)CC1 ZINC000217709329 DE On-Demand Unstable WNT3 50 31 CCOc1cc(C(=O)Cl)cc(Br)c1OCc1ccccc1Cl ZINC000217709343 HK In-Stock Unstable THRB 18 42 CCOc1cc(C(=O)Cl)cc(Br)c1OCc1ccccc1Cl ZINC000217709343 HK In-Stock Unstable FABP4 15 47 CCOc1cc(C(=O)Cl)cc(Br)c1OCc1ccccc1Cl ZINC000217709343 HK In-Stock Unstable FABP5 34 47 C[C@@H](F)CS(=O)(=O)c1ccc(CCN)cc1 ZINC000217709364 BD For-Sale Unstable CA1 17 53 C[C@@H](F)CS(=O)(=O)c1ccc(CCN)cc1 ZINC000217709364 BD For-Sale Unstable CAH_METTE 15 53 C[C@@H](F)CS(=O)(=O)c1ccc(CCN)cc1 ZINC000217709364 BD For-Sale Unstable TAAR1 18 41 COc1ccccc1/C=C/NC(=O)N1CCC(Cc2ccccc2)CC1 ZINC000217709366 FI For-Sale Unstable CHRM2 16 40 COc1ccccc1/C=C/NC(=O)N1CCC(Cc2ccccc2)CC1 ZINC000217709366 FI For-Sale Unstable HTR1A 26 43 COc1ccccc1/C=C/NC(=O)N1CCC(Cc2ccccc2)CC1 ZINC000217709366 FI For-Sale Unstable DRD2 27 43 COc1ccccc1/C=C/NC(=O)N1CCC(Cc2ccccc2)CC1 ZINC000217709366 FI For-Sale Unstable ACHE 22 43 COc1ccccc1/C=C/NC(=O)N1CCC(Cc2ccccc2)CC1 ZINC000217709366 FI For-Sale Unstable DRD3 24 40 COc1ccccc1/C=C/NC(=O)N1CCC(Cc2ccccc2)CC1 ZINC000217709366 FI For-Sale Unstable GRIN2B 91 47 COc1ccccc1/C=C/NC(=O)N1CCC(Cc2ccccc2)CC1 ZINC000217709366 FI For-Sale Unstable SIGMAR1 28 43 COc1ccccc1/C=C/NC(=O)N1CCC(Cc2ccccc2)CC1 ZINC000217709366 FI For-Sale Unstable CCR3 56 46 COc1ccccc1/C=C/NC(=O)N1CCC(Cc2ccccc2)CC1 ZINC000217709366 FI For-Sale Unstable CCR8 24 40 COc1ccccc1/C=C/NC(=O)N1CCC(Cc2ccccc2)CC1 ZINC000217709366 FI For-Sale Unstable TLR4 19 42 COc1ccccc1/C=C/NC(=O)N1CCC(Cc2ccccc2)CC1 ZINC000217709366 FI For-Sale Unstable ACKR3 40 33 COc1ccccc1CN[C@@H]1CCN2CCC[C@@H]12 ZINC000217709369 BE For-Sale Unstable TACR1 35 41 COc1ccccc1CN[C@@H]1CCN2CCC[C@@H]12 ZINC000217709369 BE For-Sale Unstable SIGMAR1 15 47 COc1ccccc1CN[C@@H]1CCN2CCC[C@@H]12 ZINC000217709369 BE For-Sale Unstable TACR3 0 52 CCCCN(CCO)C(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217709386 CE For-Sale Unstable TSPO 15 40 COc1ccccc1CN[C@H]1CCN2CCC[C@@H]12 ZINC000217709465 BE For-Sale Unstable TACR1 35 41 COc1ccccc1CN[C@H]1CCN2CCC[C@@H]12 ZINC000217709465 BE For-Sale Unstable SIGMAR1 15 47 COc1ccccc1CN[C@H]1CCN2CCC[C@@H]12 ZINC000217709465 BE For-Sale Unstable TACR3 0 52 COc1ccccc1/C=C/NC(=O)N(C)C1CCN(C)CC1 ZINC000217709501 DE For-Sale Unstable ACKR3 64 33 COc1ccc2c(c1OC)C(=O)O[C@@H]2Nc1ccc(C(=O)NCCC(=O)O)cc1 ZINC000217709510 HE In-Stock Unstable GCGR 52 34 Cc1ccc(-n2cnnc2SCC(=O)Nc2nc(-c3ccccc3)cs2)cc1C ZINC000217709538 HJ On-Demand Unstable HDAC9 15 43 Cc1ccc(-n2cnnc2SCC(=O)Nc2nc(-c3ccccc3)cs2)cc1C ZINC000217709538 HJ On-Demand Unstable TRPA1 21 47 CNc1ccc(C(=O)O)cc1S(=O)(=O)NCc1ccccc1 ZINC000217709574 DD In-Stock Unstable AKR1C3 28 43 Cc1nc(CNC(=O)c2cccc(/C=C\C(=O)O)c2)cs1 ZINC000217709576 DE For-Sale Unstable HDAC8 36 40 Cc1nc(CNC(=O)c2cccc(/C=C\C(=O)O)c2)cs1 ZINC000217709576 DE For-Sale Unstable HDAC6 22 40 Cc1ccc(C(=O)OCCC2CC2)cc1S(N)(=O)=O ZINC000217709585 CD On-Demand Unstable CA2 20 42 Cc1ccc(C(=O)OCCC2CC2)cc1S(N)(=O)=O ZINC000217709585 CD On-Demand Unstable CA1 16 42 COc1ccc2c(c1OC)C(=O)O[C@H]2Nc1ccc(C(=O)NCCC(=O)O)cc1 ZINC000217709600 HE In-Stock Unstable GCGR 52 34 COc1ccc(CCNC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217709607 EG For-Sale Unstable PTGER4 0 42 COc1ccc(CCNC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217709607 EG For-Sale Unstable CYP1B1 33 44 COc1ccc(CCNC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217709607 EG For-Sale Unstable MTNR1A 80 46 COc1ccc(CCNC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217709607 EG For-Sale Unstable MTNR1B 72 46 COc1ccc(CCNC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217709607 EG For-Sale Unstable CA9 18 45 COc1ccc(CCNC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217709607 EG For-Sale Unstable ABCG2 26 41 CCNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217709668 EF In-Stock Unstable CCR8 82 42 CCNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217709668 EF In-Stock Unstable SFRP1 101 36 CCNc1ccc(S(=O)(=O)NC2CCCCCC2)cc1C(=O)O ZINC000217709668 EF In-Stock Unstable WNT3 80 36 COC(=O)c1ccccc1S(=O)(=O)N[C@@H]1CCOC1=O ZINC000217709681 CC For-Sale Unstable LUXR 68 39 COC(=O)c1ccccc1S(=O)(=O)N[C@@H]1CCOC1=O ZINC000217709681 CC For-Sale Unstable TRAR 83 39 COC(=O)c1ccccc1S(=O)(=O)N[C@@H]1CCOC1=O ZINC000217709681 CC For-Sale Unstable LASR 57 39 Cc1ccc(NC(=O)c2cc(-c3ccc(Cl)cc3)on2)c(Cl)c1 ZINC000217709700 EK On-Demand Unstable F10 17 43 Cc1ccc(NC(=O)c2cc(-c3ccc(Cl)cc3)on2)c(Cl)c1 ZINC000217709700 EK On-Demand Unstable S1PR4 27 41 Cc1ccc(NC(=O)c2cc(-c3ccc(Cl)cc3)on2)c(Cl)c1 ZINC000217709700 EK On-Demand Unstable SCN10A 56 44 COc1ccccc1/C=C/NC(=O)NC[C@@H]1CCCO1 ZINC000217709744 CE For-Sale Unstable OXTR 27 48 COc1ccccc1/C=C/NC(=O)NC[C@@H]1CCCO1 ZINC000217709744 CE For-Sale Unstable AVPR1A 17 48 COc1ccccc1/C=C/NC(=O)NC[C@@H]1CCCO1 ZINC000217709744 CE For-Sale Unstable ACKR3 46 31 CC[C@H](C(=O)O)N(C)C(=O)/C=C\c1ccc2c(c1)CCO2 ZINC000217709750 CD For-Sale Unstable GPR183 0 42 COc1ccc(N2C[C@]34C=C[C@@H](O3)[C@@H](C(=O)NCCCc3ccccc3)[C@H]4C2=O)cc1 ZINC000217709760 HF In-Stock Unstable SCN2A 15 42 COC(=O)c1ccccc1S(=O)(=O)N[C@H]1CCOC1=O ZINC000217709769 CC On-Demand Unstable LUXR 68 39 COC(=O)c1ccccc1S(=O)(=O)N[C@H]1CCOC1=O ZINC000217709769 CC On-Demand Unstable TRAR 83 39 COC(=O)c1ccccc1S(=O)(=O)N[C@H]1CCOC1=O ZINC000217709769 CC On-Demand Unstable LASR 57 39 CCNc1ccc(S(=O)(=O)NCCCOCC)cc1C(=O)O ZINC000217709781 ED In-Stock Unstable CASP3 15 43 CCOc1cc(CN[C@@H]2CCN3CCC[C@@H]23)ccc1O ZINC000217709791 CE For-Sale Unstable SSTR5 61 44 O=S(=O)(NCCSC1CCOCC1)c1cccc(Cl)c1 ZINC000217709807 EF In-Stock Unstable TBXA2R 17 40 O=S(=O)(NCCSC1CCOCC1)c1cccc(Cl)c1 ZINC000217709807 EF In-Stock Unstable FBP1 20 40 O=C(Nc1ccc(Br)cc1F)c1cc(-c2ccc(Cl)cc2)on1 ZINC000217709812 GK On-Demand Anodyne GPR35 47 37 C[C@H](F)CS(=O)(=O)c1cccc(CCN)c1 ZINC000217709817 BD For-Sale Unstable TAAR1 16 44 COc1ccc(S(N)(=O)=O)cc1C(=O)OCCC1CC1 ZINC000217709818 CD On-Demand Unstable CA2 52 50 COc1ccc(S(N)(=O)=O)cc1C(=O)OCCC1CC1 ZINC000217709818 CD On-Demand Unstable HTR4 53 40 COc1ccc(S(N)(=O)=O)cc1C(=O)OCCC1CC1 ZINC000217709818 CD On-Demand Unstable CA1 46 44 COc1ccc(S(N)(=O)=O)cc1C(=O)OCCC1CC1 ZINC000217709818 CD On-Demand Unstable CA7 50 50 COc1ccc(S(N)(=O)=O)cc1C(=O)OCCC1CC1 ZINC000217709818 CD On-Demand Unstable CA4 38 50 COc1ccc(S(N)(=O)=O)cc1C(=O)OCCC1CC1 ZINC000217709818 CD On-Demand Unstable CA14 34 44 COc1ccc(S(N)(=O)=O)cc1C(=O)OCCC1CC1 ZINC000217709818 CD On-Demand Unstable CA12 33 50 COc1ccc(S(N)(=O)=O)cc1C(=O)OCCC1CC1 ZINC000217709818 CD On-Demand Unstable CA9 35 50 COc1ccc(S(N)(=O)=O)cc1C(=O)OCCC1CC1 ZINC000217709818 CD On-Demand Unstable CYNT 28 50 COc1ccc(S(N)(=O)=O)cc1C(=O)OCCC1CC1 ZINC000217709818 CD On-Demand Unstable NCE103 18 50 COc1ccc(S(N)(=O)=O)cc1C(=O)OCCC1CC1 ZINC000217709818 CD On-Demand Unstable CA15 17 50 COc1ccc(S(N)(=O)=O)cc1C(=O)OCCC1CC1 ZINC000217709818 CD On-Demand Unstable CA 0 50 COc1ccc(S(N)(=O)=O)cc1C(=O)OCCC1CC1 ZINC000217709818 CD On-Demand Unstable Q5TU56_ANOGA 0 50 COc1ccccc1/C=C/NC(=O)NC[C@H]1CCCO1 ZINC000217709832 CE For-Sale Unstable OXTR 27 48 COc1ccccc1/C=C/NC(=O)NC[C@H]1CCCO1 ZINC000217709832 CE For-Sale Unstable AVPR1A 17 48 COc1ccccc1/C=C/NC(=O)NC[C@H]1CCCO1 ZINC000217709832 CE For-Sale Unstable ACKR3 46 31 COc1ccc(N2C[C@]34C=C[C@@H](O3)[C@H](C(=O)NCCCc3ccccc3)[C@H]4C2=O)cc1 ZINC000217709852 HF In-Stock Unstable SCN2A 15 42 O=C(O)/C=C\c1cccc(C(=O)N2CCC[C@H](O)C2)c1 ZINC000217709868 CD For-Sale Unstable PREP 32 41 O=C(O)/C=C\c1cccc(C(=O)N2CCC[C@H](O)C2)c1 ZINC000217709868 CD For-Sale Unstable L3MBTL3 41 40 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NCCc1ccc(OC)c(OC)c1 ZINC000217709890 HE In-Stock Unstable PTGDR 28 44 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NCCc1ccc(OC)c(OC)c1 ZINC000217709890 HE In-Stock Unstable MT-ND1 24 41 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NCCc1ccc(OC)c(OC)c1 ZINC000217709890 HE In-Stock Unstable AKR1C3 17 47 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NCCc1ccc(OC)c(OC)c1 ZINC000217709890 HE In-Stock Unstable SCMU_MYCTU 0 49 CCOc1cc(CN[C@H]2CCN3CCC[C@@H]23)ccc1O ZINC000217709892 CE For-Sale Unstable SSTR5 61 44 C[C@@H](F)CS(=O)(=O)c1cccc(CCN)c1 ZINC000217709895 BD For-Sale Unstable TAAR1 16 44 O=C(Nc1ccc(Cl)cc1F)c1cc(-c2ccc(Cl)cc2)on1 ZINC000217709925 FK On-Demand Anodyne F10 32 41 COc1ccccc1/C=C/NC(=O)NCc1ccc(Cl)cc1 ZINC000217709949 DH For-Sale Unstable CYSP_PLAFA 37 40 O=C(O)/C=C\c1cccc(C(=O)N2CCC[C@@H](O)C2)c1 ZINC000217709959 CD For-Sale Unstable PREP 32 41 O=C(O)/C=C\c1cccc(C(=O)N2CCC[C@@H](O)C2)c1 ZINC000217709959 CD For-Sale Unstable RHOA 0 40 O=C(O)/C=C\c1cccc(C(=O)N2CCC[C@@H](O)C2)c1 ZINC000217709959 CD For-Sale Unstable L3MBTL1 0 40 O=C(O)/C=C\c1cccc(C(=O)N2CCC[C@@H](O)C2)c1 ZINC000217709959 CD For-Sale Unstable L3MBTL3 41 40 O=C(Cl)c1ccc(OCc2ccccc2)c(I)c1 ZINC000217709984 FI In-Stock Unstable SRD5A2 0 43 O=C(Cl)c1ccc(OCc2ccccc2)c(I)c1 ZINC000217709984 FI In-Stock Unstable PTGER2 42 46 O=C(Cl)c1ccc(OCc2ccccc2)c(I)c1 ZINC000217709984 FI In-Stock Unstable PPIA 45 36 O=C(Cl)c1ccc(OCc2ccccc2)c(I)c1 ZINC000217709984 FI In-Stock Unstable PTGER1 79 48 O=C(Cl)c1ccc(OCc2ccccc2)c(I)c1 ZINC000217709984 FI In-Stock Unstable PTGER4 31 46 O=C(Cl)c1ccc(OCc2ccccc2)c(I)c1 ZINC000217709984 FI In-Stock Unstable PTGER3 15 40 O=C(Cl)c1ccc(OCc2ccccc2)c(I)c1 ZINC000217709984 FI In-Stock Unstable ACR 65 56 O=C(Cl)c1ccc(OCc2ccccc2)c(I)c1 ZINC000217709984 FI In-Stock Unstable POBA 0 45 O=C(Cl)c1ccc(OCc2ccccc2)c(I)c1 ZINC000217709984 FI In-Stock Unstable FFAR1 17 40 O=C(Cl)c1ccc(OCc2ccccc2)c(I)c1 ZINC000217709984 FI In-Stock Unstable AKR1C3 23 40 O=C(Cl)c1ccc(OCc2ccccc2)c(I)c1 ZINC000217709984 FI In-Stock Unstable PDEC 0 40 O=C(Cl)c1ccc(OCc2ccccc2)c(I)c1 ZINC000217709984 FI In-Stock Unstable KLK_PIG 67 56 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](CC(C)C)C(=O)N3CCN(CCc4ccccn4)CC3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217710013 KI In-Stock Unstable TUBA1A 16 56 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](CC(C)C)C(=O)N3CCN(CCc4ccccn4)CC3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217710013 KI In-Stock Unstable TPPP 0 53 Cc1ccc(F)cc1NC(=O)c1cc(-c2ccc(Cl)cc2)on1 ZINC000217710025 EJ On-Demand Unstable MAPK11 24 41 Cc1ccc(F)cc1NC(=O)c1cc(-c2ccc(Cl)cc2)on1 ZINC000217710025 EJ On-Demand Unstable PLA2G7 22 42 Cc1ccc(F)cc1NC(=O)c1cc(-c2ccc(Cl)cc2)on1 ZINC000217710025 EJ On-Demand Unstable MAPK14 19 41 Cc1ccccc1COc1ccc(C(=O)Cl)cc1I ZINC000217710079 GJ In-Stock Unstable ACR 33 42 Cc1ccccc1COc1ccc(C(=O)Cl)cc1I ZINC000217710079 GJ In-Stock Unstable KLK_PIG 42 42 COc1cc(C(=O)O)c(-n2nc(C(=O)O)cc2O)cc1OC ZINC000217710118 DC In-Stock Unstable RPA1 57 38 Cc1ccc(COc2ccc(C(=O)Cl)cc2I)cc1 ZINC000217710184 GJ In-Stock Unstable PTGER1 41 38 Cc1ccc(COc2ccc(C(=O)Cl)cc2I)cc1 ZINC000217710184 GJ In-Stock Unstable ACR 57 57 Cc1ccc(COc2ccc(C(=O)Cl)cc2I)cc1 ZINC000217710184 GJ In-Stock Unstable KLK_PIG 64 57 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NC1CCCC1 ZINC000217710213 DE In-Stock Unstable CCR8 87 46 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NC1CCCC1 ZINC000217710213 DE In-Stock Unstable SFRP1 105 38 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NC1CCCC1 ZINC000217710213 DE In-Stock Unstable WNT3 82 37 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NC1CCCC1 ZINC000217710213 DE In-Stock Unstable BRD4 24 41 CCCCCCC(=O)N1CCN(CC#N)CC1 ZINC000217710257 BD On-Demand Unstable GNAI1 0 50 CCCCCCC(=O)N1CCN(CC#N)CC1 ZINC000217710257 BD On-Demand Unstable GNAI3 0 48 CCCCCCC(=O)N1CCN(CC#N)CC1 ZINC000217710257 BD On-Demand Unstable GNAO1 0 48 CCCCCCC(=O)N1CCN(CC#N)CC1 ZINC000217710257 BD On-Demand Unstable CQSS 53 33 Cc1ccc(-n2cnnc2SCC(=O)Nc2nc(-c3ccccn3)cs2)cc1C ZINC000217710288 HI On-Demand Unstable NPY5R 15 40 O=C(Cl)c1ccc(OCc2ccc(F)cc2)c(I)c1 ZINC000217710300 GI In-Stock Unstable PTGER1 38 41 O=C(Cl)c1ccc(OCc2ccc(F)cc2)c(I)c1 ZINC000217710300 GI In-Stock Unstable ACR 57 57 O=C(Cl)c1ccc(OCc2ccc(F)cc2)c(I)c1 ZINC000217710300 GI In-Stock Unstable ENPP2 22 40 O=C(Cl)c1ccc(OCc2ccc(F)cc2)c(I)c1 ZINC000217710300 GI In-Stock Unstable KLK_PIG 64 57 COc1ccc(CNC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217710371 DG For-Sale Unstable ANPEP 23 44 COc1ccc(CNC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217710371 DG For-Sale Unstable PTGER4 0 43 COc1ccc(CNC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217710371 DG For-Sale Unstable CYP1B1 37 46 COc1ccc(CNC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217710371 DG For-Sale Unstable MTNR1A 29 50 COc1ccc(CNC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217710371 DG For-Sale Unstable MTNR1B 26 50 COc1ccc(CNC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217710371 DG For-Sale Unstable CA9 16 43 COc1ccc(CNC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217710371 DG For-Sale Unstable U38 0 44 COc1ccc(CNC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217710371 DG For-Sale Unstable KCNJ2 0 42 O=C(Cl)c1ccc(OCc2cccc(F)c2)c(I)c1 ZINC000217710399 GI In-Stock Unstable EGFR 41 38 O=C(Cl)c1ccc(OCc2cccc(F)c2)c(I)c1 ZINC000217710399 GI In-Stock Unstable ERBB2 51 38 O=C(Cl)c1ccc(OCc2cccc(F)c2)c(I)c1 ZINC000217710399 GI In-Stock Unstable PTGER1 54 38 O=C(Cl)c1ccc(OCc2cccc(F)c2)c(I)c1 ZINC000217710399 GI In-Stock Unstable ACR 52 47 O=C(Cl)c1ccc(OCc2cccc(F)c2)c(I)c1 ZINC000217710399 GI In-Stock Unstable AKR1C3 18 44 O=C(Cl)c1ccc(OCc2cccc(F)c2)c(I)c1 ZINC000217710399 GI In-Stock Unstable KLK_PIG 60 57 Cc1cc(Br)ccc1NC(=O)c1cc(-c2ccc(Cl)cc2)on1 ZINC000217710406 GK On-Demand Unstable PRS 49 35 Cc1cc(Br)ccc1NC(=O)c1cc(-c2ccc(Cl)cc2)on1 ZINC000217710406 GK On-Demand Unstable SCN10A 33 40 O=C(O)/C=C\c1ccc(C(=O)N2CCN(C3CC3)CC2)s1 ZINC000217710433 DD For-Sale Unstable L3MBTL1 0 55 O=C(O)/C=C\c1ccc(C(=O)N2CCN(C3CC3)CC2)s1 ZINC000217710433 DD For-Sale Unstable L3MBTL3 81 55 COc1ccccc1/C=C/NC(=O)N1CCN(C(C)=O)CC1 ZINC000217710465 DD For-Sale Unstable DRD3 16 40 O=C(COCC(F)(F)C(F)F)N1CCC[C@@H]1c1ccccn1 ZINC000217710474 DF In-Stock Unstable CPT1A 109 44 O=S(=O)(NCCSC1CCOCC1)c1ccc2c(c1)CCCC2 ZINC000217710476 FF In-Stock Unstable TBXA2R 15 42 CCc1nc(=O)n(-c2cccnc2)[nH]1 ZINC000217710487 AC For-Sale Unstable CYP2A6 20 40 N#CCN1CCN(C(=O)c2cc(Cl)ccn2)CC1 ZINC000217710496 CD For-Sale Unstable ALPL 16 40 O=C(Nc1ccc(N2CCOCC2)cc1N1CCOCC1)c1cc(-c2ccc(Cl)cc2)on1 ZINC000217710513 JH On-Demand Unstable F10 24 48 O=C(Nc1ccc(N2CCOCC2)cc1N1CCOCC1)c1cc(-c2ccc(Cl)cc2)on1 ZINC000217710513 JH On-Demand Unstable PRKDC 15 46 O=C(Nc1ccc(N2CCOCC2)cc1N1CCOCC1)c1cc(-c2ccc(Cl)cc2)on1 ZINC000217710513 JH On-Demand Unstable PIK3CA 15 43 O=C(Nc1ccc(N2CCOCC2)cc1N1CCOCC1)c1cc(-c2ccc(Cl)cc2)on1 ZINC000217710513 JH On-Demand Unstable PRNP 44 36 O=C(Nc1ccc(N2CCOCC2)cc1N1CCOCC1)c1cc(-c2ccc(Cl)cc2)on1 ZINC000217710513 JH On-Demand Unstable MAPKAPK2 30 63 O=C(Nc1ccc(N2CCOCC2)cc1N1CCOCC1)c1cc(-c2ccc(Cl)cc2)on1 ZINC000217710513 JH On-Demand Unstable MTOR 21 43 O=C(Nc1ccc(N2CCOCC2)cc1N1CCOCC1)c1cc(-c2ccc(Cl)cc2)on1 ZINC000217710513 JH On-Demand Unstable SCN10A 34 42 O=C(Nc1ccc(N2CCOCC2)cc1N1CCOCC1)c1cc(-c2ccc(Cl)cc2)on1 ZINC000217710513 JH On-Demand Unstable CSF1R 21 40 O=C(Nc1ccc(N2CCOCC2)cc1N1CCOCC1)c1cc(-c2ccc(Cl)cc2)on1 ZINC000217710513 JH On-Demand Unstable CHEK1 0 48 O=C(Nc1ccc(N2CCOCC2)cc1N1CCOCC1)c1cc(-c2ccc(Cl)cc2)on1 ZINC000217710513 JH On-Demand Unstable AKR1C3 30 45 O=C(Nc1ccc(N2CCOCC2)cc1N1CCOCC1)c1cc(-c2ccc(Cl)cc2)on1 ZINC000217710513 JH On-Demand Unstable DGAT1 15 42 O=C(Cl)c1ccc(OCc2ccccc2F)c(I)c1 ZINC000217710515 GI In-Stock Unstable PTGER1 46 45 O=C(Cl)c1ccc(OCc2ccccc2F)c(I)c1 ZINC000217710515 GI In-Stock Unstable ACR 33 42 O=C(Cl)c1ccc(OCc2ccccc2F)c(I)c1 ZINC000217710515 GI In-Stock Unstable KLK_PIG 42 42 CCOc1ccc(CC(=O)NC[C@@H](O)C(=O)OC)cc1 ZINC000217710532 CC On-Demand Unstable CA9 24 41 C[C@@H]1CN(C(=O)OC(C)(C)C)CC=C1c1ccc2c(c1)N1C(=NNC(=O)[C@H]1C)CO2 ZINC000217710538 HF In-Stock Unstable PRKCQ 23 47 COCC(=O)N[C@@H]1CCCc2c1[nH]c1ccc(OC)cc21 ZINC000217710556 CE In-Stock Unstable MTR1B_CHICK 0 40 COCC(=O)N[C@@H]1CCCc2c1[nH]c1ccc(OC)cc21 ZINC000217710556 CE In-Stock Unstable MAPKAPK2 29 53 COCC(=O)N[C@@H]1CCCc2c1[nH]c1ccc(OC)cc21 ZINC000217710556 CE In-Stock Unstable MTNR1A 47 41 COCC(=O)N[C@@H]1CCCc2c1[nH]c1ccc(OC)cc21 ZINC000217710556 CE In-Stock Unstable MTNR1B 43 40 COCC(=O)N[C@@H]1CCCc2c1[nH]c1ccc(OC)cc21 ZINC000217710556 CE In-Stock Unstable S1PR1 22 40 CCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217710558 GE In-Stock Unstable CA2 21 41 CCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217710558 GE In-Stock Unstable TBXA2R 53 46 CCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217710558 GE In-Stock Unstable TBXAS1 18 43 CCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217710558 GE In-Stock Unstable BMP1 57 38 CCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217710558 GE In-Stock Unstable CA1 18 46 CCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217710558 GE In-Stock Unstable MMP13 47 39 CCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217710558 GE In-Stock Unstable MMP3 43 37 CCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217710558 GE In-Stock Unstable MMP14 15 41 CCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217710558 GE In-Stock Unstable ALOX15 52 41 CCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217710558 GE In-Stock Unstable CA12 15 41 CCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217710558 GE In-Stock Unstable PTGDR 27 41 CCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217710558 GE In-Stock Unstable CA9 26 44 CCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217710558 GE In-Stock Unstable MMP1 50 38 CCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217710558 GE In-Stock Unstable AKR1C3 31 50 CCNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217710558 GE In-Stock Unstable AKR1C2 52 38 O=C(COCC(F)(F)C(F)F)N1CCC[C@H]1c1ccccn1 ZINC000217710566 DF In-Stock Unstable CPT1A 109 44 COc1ccccc1/C=C/NC(=O)NCc1ccc2c(c1)OCO2 ZINC000217710568 EF For-Sale Unstable PDE5A 34 40 COc1ccccc1/C=C/NC(=O)NCc1ccc2c(c1)OCO2 ZINC000217710568 EF For-Sale Unstable EDNRB 66 40 COc1ccccc1/C=C/NC(=O)NCc1ccc2c(c1)OCO2 ZINC000217710568 EF For-Sale Unstable BMP1 52 41 COc1ccccc1/C=C/NC(=O)NCc1ccc2c(c1)OCO2 ZINC000217710568 EF For-Sale Unstable SCN9A 27 41 COc1ccccc1/C=C/NC(=O)NCc1ccc2c(c1)OCO2 ZINC000217710568 EF For-Sale Unstable NOS2 90 34 COc1ccccc1/C=C/NC(=O)NCc1ccc2c(c1)OCO2 ZINC000217710568 EF For-Sale Unstable Q9XSW7_PIG 0 41 Fc1ccc(CN[C@@H]2CCN3CCC[C@@H]23)cc1F ZINC000217710589 CE For-Sale Unstable SSTR3 17 42 CCOc1ccc(CC(=O)NC[C@H](O)C(=O)OC)cc1 ZINC000217710611 CC On-Demand Unstable CA9 24 41 C[C@H]1CN(C(=O)OC(C)(C)C)CC=C1c1ccc2c(c1)N1C(=NNC(=O)[C@H]1C)CO2 ZINC000217710621 HF In-Stock Unstable PRKCQ 23 47 O=C(Cl)c1ccc(OCc2ccccc2Cl)c(I)c1 ZINC000217710633 HJ In-Stock Unstable PTGER1 39 44 O=C(Cl)c1ccc(OCc2ccccc2Cl)c(I)c1 ZINC000217710633 HJ In-Stock Unstable FABP4 18 49 O=C(Cl)c1ccc(OCc2ccccc2Cl)c(I)c1 ZINC000217710633 HJ In-Stock Unstable ACR 39 43 O=C(Cl)c1ccc(OCc2ccccc2Cl)c(I)c1 ZINC000217710633 HJ In-Stock Unstable FABP5 33 49 O=C(Cl)c1ccc(OCc2ccccc2Cl)c(I)c1 ZINC000217710633 HJ In-Stock Unstable KLK_PIG 53 43 COCC(=O)N[C@H]1CCCc2c1[nH]c1ccc(OC)cc21 ZINC000217710639 CE In-Stock Unstable MTR1B_CHICK 0 40 COCC(=O)N[C@H]1CCCc2c1[nH]c1ccc(OC)cc21 ZINC000217710639 CE In-Stock Unstable MAPKAPK2 29 53 COCC(=O)N[C@H]1CCCc2c1[nH]c1ccc(OC)cc21 ZINC000217710639 CE In-Stock Unstable MTNR1A 47 41 COCC(=O)N[C@H]1CCCc2c1[nH]c1ccc(OC)cc21 ZINC000217710639 CE In-Stock Unstable MTNR1B 43 40 COCC(=O)N[C@H]1CCCc2c1[nH]c1ccc(OC)cc21 ZINC000217710639 CE In-Stock Unstable S1PR1 22 40 Fc1ccc(CN[C@H]2CCN3CCC[C@@H]23)cc1F ZINC000217710679 CE For-Sale Unstable SSTR3 17 42 CCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217710683 DF In-Stock Unstable CA2 23 40 CCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217710683 DF In-Stock Unstable ADRB1 0 47 CCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217710683 DF In-Stock Unstable ADRB3 15 44 CCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217710683 DF In-Stock Unstable LPL 31 42 CCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217710683 DF In-Stock Unstable CA1 19 47 CCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217710683 DF In-Stock Unstable CA4 33 40 CCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217710683 DF In-Stock Unstable PRTN3 56 37 CCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217710683 DF In-Stock Unstable MTNN 41 35 CCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217710683 DF In-Stock Unstable AKR1C3 44 40 CCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217710683 DF In-Stock Unstable LIPG 15 42 CCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217710683 DF In-Stock Unstable AKR1C2 55 36 CCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217710683 DF In-Stock Unstable LIMK2 58 46 CCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217710683 DF In-Stock Unstable MGAT2 0 41 CCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217710683 DF In-Stock Unstable MGAT3 0 41 CCNc1ccc(S(=O)(=O)Nc2ccccc2)cc1C(=O)O ZINC000217710683 DF In-Stock Unstable MGAT1 56 41 COc1ccccc1/C=C/NC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217710685 EE For-Sale Unstable CA2 88 59 COc1ccccc1/C=C/NC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217710685 EE For-Sale Unstable CA1 92 63 COc1ccccc1/C=C/NC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217710685 EE For-Sale Unstable CA7 42 45 COc1ccccc1/C=C/NC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217710685 EE For-Sale Unstable CA5B 40 45 COc1ccccc1/C=C/NC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217710685 EE For-Sale Unstable CA4 54 52 COc1ccccc1/C=C/NC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217710685 EE For-Sale Unstable CA5A 45 45 COc1ccccc1/C=C/NC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217710685 EE For-Sale Unstable CA14 38 45 COc1ccccc1/C=C/NC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217710685 EE For-Sale Unstable CA12 84 59 COc1ccccc1/C=C/NC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217710685 EE For-Sale Unstable CA9 89 46 COc1ccccc1/C=C/NC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217710685 EE For-Sale Unstable UREA_CANEN 29 47 COc1ccccc1/C=C/NC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217710685 EE For-Sale Unstable IDO1 0 42 COc1ccccc1/C=C/NC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217710685 EE For-Sale Unstable NCE103 46 44 COc1ccccc1/C=C/NC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217710685 EE For-Sale Unstable MTCA1 60 63 COc1ccccc1/C=C/NC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217710685 EE For-Sale Unstable P96878_MYCTU 75 63 C[C@]1(C(=O)O)[C@H]2CCN(Cc3ccccc3)C[C@@H]21 ZINC000217710721 BE For-Sale Unstable CHRM2 32 43 C[C@]1(C(=O)O)[C@H]2CCN(Cc3ccccc3)C[C@@H]21 ZINC000217710721 BE For-Sale Unstable DRD2 28 46 C[C@]1(C(=O)O)[C@H]2CCN(Cc3ccccc3)C[C@@H]21 ZINC000217710721 BE For-Sale Unstable DRD4 74 46 C[C@]1(C(=O)O)[C@H]2CCN(Cc3ccccc3)C[C@@H]21 ZINC000217710721 BE For-Sale Unstable ACHE 51 49 C[C@]1(C(=O)O)[C@H]2CCN(Cc3ccccc3)C[C@@H]21 ZINC000217710721 BE For-Sale Unstable SLC6A1 40 32 C[C@]1(C(=O)O)[C@H]2CCN(Cc3ccccc3)C[C@@H]21 ZINC000217710721 BE For-Sale Unstable OPRM1 20 43 C[C@]1(C(=O)O)[C@H]2CCN(Cc3ccccc3)C[C@@H]21 ZINC000217710721 BE For-Sale Unstable DRD3 24 44 C[C@]1(C(=O)O)[C@H]2CCN(Cc3ccccc3)C[C@@H]21 ZINC000217710721 BE For-Sale Unstable OPRD1 15 40 C[C@]1(C(=O)O)[C@H]2CCN(Cc3ccccc3)C[C@@H]21 ZINC000217710721 BE For-Sale Unstable OPRK1 24 43 C[C@]1(C(=O)O)[C@H]2CCN(Cc3ccccc3)C[C@@H]21 ZINC000217710721 BE For-Sale Unstable CHRM3 34 48 C[C@]1(C(=O)O)[C@H]2CCN(Cc3ccccc3)C[C@@H]21 ZINC000217710721 BE For-Sale Unstable HRH3 17 45 C[C@]1(C(=O)O)[C@H]2CCN(Cc3ccccc3)C[C@@H]21 ZINC000217710721 BE For-Sale Unstable SIGMAR1 96 48 C[C@]1(C(=O)O)[C@H]2CCN(Cc3ccccc3)C[C@@H]21 ZINC000217710721 BE For-Sale Unstable CCR3 42 40 C[C@]1(C(=O)O)[C@H]2CCN(Cc3ccccc3)C[C@@H]21 ZINC000217710721 BE For-Sale Unstable CCR5 46 39 C[C@]1(C(=O)O)[C@H]2CCN(Cc3ccccc3)C[C@@H]21 ZINC000217710721 BE For-Sale Unstable SLC18A3 34 44 C[C@]1(C(=O)O)[C@H]2CCN(Cc3ccccc3)C[C@@H]21 ZINC000217710721 BE For-Sale Unstable MCHR1 24 44 C[C@]1(C(=O)O)[C@H]2CCN(Cc3ccccc3)C[C@@H]21 ZINC000217710721 BE For-Sale Unstable CACNA1G 21 42 C[C@]1(C(=O)O)[C@H]2CCN(Cc3ccccc3)C[C@@H]21 ZINC000217710721 BE For-Sale Unstable BIRC2 28 40 C[C@]1(C(=O)O)[C@H]2CCN(Cc3ccccc3)C[C@@H]21 ZINC000217710721 BE For-Sale Unstable NPFFR1 46 33 COC(=O)[C@@H](O)CNC(=O)c1ccc(CNC(C)=O)cc1 ZINC000217710725 CB On-Demand Unstable CA2 21 42 O=C(Cl)c1ccc(OCc2ccc(Cl)cc2Cl)c(I)c1 ZINC000217710751 IK In-Stock Unstable PTGER1 54 46 O=C(Cl)c1ccc(OCc2ccc(Cl)cc2Cl)c(I)c1 ZINC000217710751 IK In-Stock Unstable ACR 33 42 O=C(Cl)c1ccc(OCc2ccc(Cl)cc2Cl)c(I)c1 ZINC000217710751 IK In-Stock Unstable KLK_PIG 51 42 CC[C@@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1NC ZINC000217710793 CD In-Stock Unstable NEU3 0 40 COc1ccccc1/C=C/NC(=O)NCc1ccccc1 ZINC000217710797 CG For-Sale Unstable PTGER2 27 41 COc1ccccc1/C=C/NC(=O)NCc1ccccc1 ZINC000217710797 CG For-Sale Unstable PTGER4 0 41 COc1ccccc1/C=C/NC(=O)NCc1ccccc1 ZINC000217710797 CG For-Sale Unstable KCNA3 42 40 COc1ccccc1/C=C/NC(=O)NCc1ccccc1 ZINC000217710797 CG For-Sale Unstable TLR4 19 44 COc1ccccc1/C=C/NC(=O)NCc1ccccc1 ZINC000217710797 CG For-Sale Unstable AKR1B10 33 40 COc1ccccc1/C=C/NC(=O)NCc1ccccc1 ZINC000217710797 CG For-Sale Unstable PDS 49 37 COC(=O)[C@H](O)CNC(=O)c1ccc(CNC(C)=O)cc1 ZINC000217710803 CB On-Demand Unstable CA2 21 42 COc1ccc(C(=O)OCCC2CC2)cc1S(N)(=O)=O ZINC000217710813 CD On-Demand Unstable CA2 15 40 CSC[C@@](C)(O)CNC(=O)c1cc(C2CC2)on1 ZINC000217710836 CD On-Demand Unstable S1PR3 0 43 CC[C@H](C)NS(=O)(=O)c1cc(C(=O)O)ccc1NC ZINC000217710876 CD In-Stock Unstable NEU3 0 40 O=C(Cl)c1ccc(OCc2ccc(Cl)cc2)c(I)c1 ZINC000217710884 HJ In-Stock Unstable PTGER1 64 44 O=C(Cl)c1ccc(OCc2ccc(Cl)cc2)c(I)c1 ZINC000217710884 HJ In-Stock Unstable CCR5 20 41 O=C(Cl)c1ccc(OCc2ccc(Cl)cc2)c(I)c1 ZINC000217710884 HJ In-Stock Unstable ACR 62 59 O=C(Cl)c1ccc(OCc2ccc(Cl)cc2)c(I)c1 ZINC000217710884 HJ In-Stock Unstable KLK_PIG 66 59 C[C@@]1(C(=O)O)[C@H]2CN(Cc3ccccc3)CC[C@H]21 ZINC000217710889 BE For-Sale Unstable CHRM2 32 43 C[C@@]1(C(=O)O)[C@H]2CN(Cc3ccccc3)CC[C@H]21 ZINC000217710889 BE For-Sale Unstable DRD2 28 46 C[C@@]1(C(=O)O)[C@H]2CN(Cc3ccccc3)CC[C@H]21 ZINC000217710889 BE For-Sale Unstable DRD4 74 46 C[C@@]1(C(=O)O)[C@H]2CN(Cc3ccccc3)CC[C@H]21 ZINC000217710889 BE For-Sale Unstable ACHE 51 49 C[C@@]1(C(=O)O)[C@H]2CN(Cc3ccccc3)CC[C@H]21 ZINC000217710889 BE For-Sale Unstable SLC6A1 40 32 C[C@@]1(C(=O)O)[C@H]2CN(Cc3ccccc3)CC[C@H]21 ZINC000217710889 BE For-Sale Unstable OPRM1 20 43 C[C@@]1(C(=O)O)[C@H]2CN(Cc3ccccc3)CC[C@H]21 ZINC000217710889 BE For-Sale Unstable DRD3 24 44 C[C@@]1(C(=O)O)[C@H]2CN(Cc3ccccc3)CC[C@H]21 ZINC000217710889 BE For-Sale Unstable OPRD1 15 40 C[C@@]1(C(=O)O)[C@H]2CN(Cc3ccccc3)CC[C@H]21 ZINC000217710889 BE For-Sale Unstable OPRK1 24 43 C[C@@]1(C(=O)O)[C@H]2CN(Cc3ccccc3)CC[C@H]21 ZINC000217710889 BE For-Sale Unstable CHRM3 34 48 C[C@@]1(C(=O)O)[C@H]2CN(Cc3ccccc3)CC[C@H]21 ZINC000217710889 BE For-Sale Unstable HRH3 17 45 C[C@@]1(C(=O)O)[C@H]2CN(Cc3ccccc3)CC[C@H]21 ZINC000217710889 BE For-Sale Unstable SIGMAR1 96 48 C[C@@]1(C(=O)O)[C@H]2CN(Cc3ccccc3)CC[C@H]21 ZINC000217710889 BE For-Sale Unstable CCR3 42 40 C[C@@]1(C(=O)O)[C@H]2CN(Cc3ccccc3)CC[C@H]21 ZINC000217710889 BE For-Sale Unstable CCR5 46 39 C[C@@]1(C(=O)O)[C@H]2CN(Cc3ccccc3)CC[C@H]21 ZINC000217710889 BE For-Sale Unstable SLC18A3 34 44 C[C@@]1(C(=O)O)[C@H]2CN(Cc3ccccc3)CC[C@H]21 ZINC000217710889 BE For-Sale Unstable MCHR1 24 44 C[C@@]1(C(=O)O)[C@H]2CN(Cc3ccccc3)CC[C@H]21 ZINC000217710889 BE For-Sale Unstable CACNA1G 21 42 C[C@@]1(C(=O)O)[C@H]2CN(Cc3ccccc3)CC[C@H]21 ZINC000217710889 BE For-Sale Unstable BIRC2 28 40 C[C@@]1(C(=O)O)[C@H]2CN(Cc3ccccc3)CC[C@H]21 ZINC000217710889 BE For-Sale Unstable NPFFR1 46 33 COc1ccccc1/C=C/NC(=O)N[C@@H](C)C12CC3CC(CC(C3)C1)C2 ZINC000217710896 FJ For-Sale Unstable EPHX2 16 42 CSC[C@](C)(O)CNC(=O)c1cc(C2CC2)on1 ZINC000217710912 CD On-Demand Unstable S1PR3 0 43 O=S(=O)(NCCSC1CCOCC1)c1ccc(OC(F)(F)F)cc1 ZINC000217710924 GF In-Stock Unstable MMP13 21 41 O=S(=O)(NCCSC1CCOCC1)c1ccc(OC(F)(F)F)cc1 ZINC000217710924 GF In-Stock Unstable MMP2 31 41 O=S(=O)(NCCSC1CCOCC1)c1ccc(OC(F)(F)F)cc1 ZINC000217710924 GF In-Stock Unstable MMP9 25 41 COC(=O)[C@@H](O)CNC(=O)c1cccc(S(C)(=O)=O)c1 ZINC000217710927 DB On-Demand Unstable DRD4 41 32 COC(=O)[C@@H](O)CNC(=O)c1cccc(S(C)(=O)=O)c1 ZINC000217710927 DB On-Demand Unstable ITGAV 54 38 Cc1cc(NS(=O)(=O)c2cccc(/C=C\C(=O)O)c2)on1 ZINC000217710955 DD For-Sale Unstable HDAC8 29 49 COc1ccccc1/C=C/NC(=O)N[C@H](C)C12CC3CC(CC(C3)C1)C2 ZINC000217710970 FJ For-Sale Unstable EPHX2 16 42 O=C(Cl)c1ccc(OCc2ccc(F)cc2Cl)c(I)c1 ZINC000217710984 IK In-Stock Unstable PTGER1 25 46 O=C(Cl)c1ccc(OCc2ccc(F)cc2Cl)c(I)c1 ZINC000217710984 IK In-Stock Unstable ACR 31 40 O=C(Cl)c1ccc(OCc2ccc(F)cc2Cl)c(I)c1 ZINC000217710984 IK In-Stock Unstable KLK_PIG 39 40 O=C(NCCc1nc2cc(Cl)ccc2[nH]1)[C@@H]1CC[C@H](O)CC1 ZINC000217710990 DE In-Stock Unstable F9 30 57 O=C(NCCc1nc2cc(Cl)ccc2[nH]1)[C@@H]1CC[C@H](O)CC1 ZINC000217710990 DE In-Stock Unstable CYSP_TRYCR 0 49 O=C(NCCc1nc2cc(Cl)ccc2[nH]1)[C@@H]1CC[C@H](O)CC1 ZINC000217710990 DE In-Stock Unstable PYGL 46 36 COC(=O)[C@H](O)CNC(=O)c1cccc(S(C)(=O)=O)c1 ZINC000217711008 DB On-Demand Unstable DRD4 41 32 COC(=O)[C@H](O)CNC(=O)c1cccc(S(C)(=O)=O)c1 ZINC000217711008 DB On-Demand Unstable ITGAV 54 38 CCCCCNS(=O)(=O)c1ccc(/C=C\C(=O)O)cc1Cl ZINC000217711050 EF For-Sale Unstable PYGL 0 44 CCCCCNS(=O)(=O)c1ccc(/C=C\C(=O)O)cc1Cl ZINC000217711050 EF For-Sale Unstable NR0B2 0 40 COc1ccccc1/C=C/NC(=O)Nc1cccc2c(O)cccc12 ZINC000217711078 EI For-Sale Unstable GCGR 0 43 COc1ccccc1/C=C/NC(=O)Nc1cccc2c(O)cccc12 ZINC000217711078 EI For-Sale Unstable ESR2 0 42 CC1=C(C)CN(C(=O)OCc2ccccc2)CC1 ZINC000217711081 BG For-Sale Unstable CHRM1 17 43 CC1=C(C)CN(C(=O)OCc2ccccc2)CC1 ZINC000217711081 BG For-Sale Unstable FABI 46 33 CC1=C(C)CN(C(=O)OCc2ccccc2)CC1 ZINC000217711081 BG For-Sale Unstable CELA1 20 43 CC1=C(C)CN(C(=O)OCc2ccccc2)CC1 ZINC000217711081 BG For-Sale Unstable CHRM4 16 43 CC1=C(C)CN(C(=O)OCc2ccccc2)CC1 ZINC000217711081 BG For-Sale Unstable CHRM5 33 43 CC1=C(C)CN(C(=O)OCc2ccccc2)CC1 ZINC000217711081 BG For-Sale Unstable GRIN2B 27 45 CC1=C(C)CN(C(=O)OCc2ccccc2)CC1 ZINC000217711081 BG For-Sale Unstable ELANE 15 40 CC1=C(C)CN(C(=O)OCc2ccccc2)CC1 ZINC000217711081 BG For-Sale Unstable PREP 36 48 CC1=C(C)CN(C(=O)OCc2ccccc2)CC1 ZINC000217711081 BG For-Sale Unstable CAPNS1 48 34 CC1=C(C)CN(C(=O)OCc2ccccc2)CC1 ZINC000217711081 BG For-Sale Unstable CAPN1 42 35 CC1=C(C)CN(C(=O)OCc2ccccc2)CC1 ZINC000217711081 BG For-Sale Unstable CAPN2 71 34 CC1=C(C)CN(C(=O)OCc2ccccc2)CC1 ZINC000217711081 BG For-Sale Unstable TGM2 44 41 CC1=C(C)CN(C(=O)OCc2ccccc2)CC1 ZINC000217711081 BG For-Sale Unstable F13A1 45 41 CC1=C(C)CN(C(=O)OCc2ccccc2)CC1 ZINC000217711081 BG For-Sale Unstable Q6PRC7_IXORI 36 40 CC1=C(C)CN(C(=O)OCc2ccccc2)CC1 ZINC000217711081 BG For-Sale Unstable SLC12A5 81 43 CCOc1cc(C(=O)Cl)cc(I)c1OCc1ccc(F)cc1Cl ZINC000217711093 JK In-Stock Unstable P2RX7 41 37 COC(=O)[C@@H](O)CNC(=O)Cc1cc(Cl)ccc1OC ZINC000217711123 DC On-Demand Unstable TRPV1 30 40 COC(=O)[C@@H](O)CNC(=O)Cc1cc(Cl)ccc1OC ZINC000217711123 DC On-Demand Unstable COLA 41 39 COC(=O)[C@@H](O)CNC(=O)Cc1cc(Cl)ccc1OC ZINC000217711123 DC On-Demand Unstable CPT1B 43 36 CCCCCNS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217711130 CE For-Sale Unstable HDAC8 18 46 CCCCCNS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217711130 CE For-Sale Unstable FBP1 29 41 CCCCCNS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217711130 CE For-Sale Unstable HDAC9 15 46 CCCCCNS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217711130 CE For-Sale Unstable HDAC7 25 46 CCCCCNS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217711130 CE For-Sale Unstable AKR1C3 25 45 COc1ccc(-c2ccc(S(=O)(=O)NCCSC3CCOCC3)cc2)cc1 ZINC000217711151 HH In-Stock Unstable AVPR1B 22 43 COc1ccc(-c2ccc(S(=O)(=O)NCCSC3CCOCC3)cc2)cc1 ZINC000217711151 HH In-Stock Unstable MMP13 40 43 COc1ccc(-c2ccc(S(=O)(=O)NCCSC3CCOCC3)cc2)cc1 ZINC000217711151 HH In-Stock Unstable MMP2 30 43 COc1ccc(-c2ccc(S(=O)(=O)NCCSC3CCOCC3)cc2)cc1 ZINC000217711151 HH In-Stock Unstable MMP3 27 43 COc1ccc(-c2ccc(S(=O)(=O)NCCSC3CCOCC3)cc2)cc1 ZINC000217711151 HH In-Stock Unstable MMP8 20 43 COc1ccc(-c2ccc(S(=O)(=O)NCCSC3CCOCC3)cc2)cc1 ZINC000217711151 HH In-Stock Unstable ALOX15 33 44 COc1ccc(-c2ccc(S(=O)(=O)NCCSC3CCOCC3)cc2)cc1 ZINC000217711151 HH In-Stock Unstable MMP9 25 43 COc1ccc(-c2ccc(S(=O)(=O)NCCSC3CCOCC3)cc2)cc1 ZINC000217711151 HH In-Stock Unstable MMP1 22 41 COc1ccc(-c2ccc(S(=O)(=O)NCCSC3CCOCC3)cc2)cc1 ZINC000217711151 HH In-Stock Unstable FFAR4 18 40 COc1ccc(-c2coc3ccc(OCC(=O)N4CCn5c4nc4ccccc45)cc23)cc1 ZINC000217711167 IJ In-Stock Unstable ALDH2 84 37 O=C(O)c1cc(O)n(-c2ccccc2Sc2ccccc2)n1 ZINC000217711191 DG In-Stock Anodyne RPA1 66 37 CC1=CCN(C(=O)OCc2ccccc2)[C@H](C)C1 ZINC000217711215 BG For-Sale Unstable CELA1 20 45 CC1=CCN(C(=O)OCc2ccccc2)[C@H](C)C1 ZINC000217711215 BG For-Sale Unstable ELANE 18 41 CC1=CCN(C(=O)OCc2ccccc2)[C@H](C)C1 ZINC000217711215 BG For-Sale Unstable PAPA1_CARPA 41 33 CC1=CCN(C(=O)OCc2ccccc2)[C@H](C)C1 ZINC000217711215 BG For-Sale Unstable PREP 36 48 CC1=CCN(C(=O)OCc2ccccc2)[C@H](C)C1 ZINC000217711215 BG For-Sale Unstable CAPN2 42 33 CC1=CCN(C(=O)OCc2ccccc2)[C@H](C)C1 ZINC000217711215 BG For-Sale Unstable KLK5 40 38 CC1=CCN(C(=O)OCc2ccccc2)[C@H](C)C1 ZINC000217711215 BG For-Sale Unstable NAAA 43 40 CC1=CCN(C(=O)OCc2ccccc2)[C@H](C)C1 ZINC000217711215 BG For-Sale Unstable SLC12A5 61 38 CCOc1cc(C(=O)Cl)cc(Br)c1OCc1ccc(F)cc1Cl ZINC000217711219 HK In-Stock Unstable P2RX7 40 37 COC(=O)[C@H](O)CNC(=O)Cc1cc(Cl)ccc1OC ZINC000217711228 DC On-Demand Unstable TRPV1 30 40 COC(=O)[C@H](O)CNC(=O)Cc1cc(Cl)ccc1OC ZINC000217711228 DC On-Demand Unstable COLA 41 39 COC(=O)[C@H](O)CNC(=O)Cc1cc(Cl)ccc1OC ZINC000217711228 DC On-Demand Unstable CPT1B 43 36 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCCC(=O)NCCc3c[nH]cn3)[C@H]21 ZINC000217711275 JF In-Stock Unstable HRH3 33 45 C[C@@H]1CCCCN1CCCNS(=O)(=O)CCCO ZINC000217711287 CC For-Sale Unstable HRH3 25 46 COc1ccccc1/C=C/NC(=O)N1CCOCC1 ZINC000217711297 CD For-Sale Unstable ITGAL 38 47 CC1=CCN(C(=O)OCc2ccccc2)[C@@H](C)C1 ZINC000217711303 BG For-Sale Unstable CELA1 20 45 CC1=CCN(C(=O)OCc2ccccc2)[C@@H](C)C1 ZINC000217711303 BG For-Sale Unstable ELANE 18 41 CC1=CCN(C(=O)OCc2ccccc2)[C@@H](C)C1 ZINC000217711303 BG For-Sale Unstable PAPA1_CARPA 41 33 CC1=CCN(C(=O)OCc2ccccc2)[C@@H](C)C1 ZINC000217711303 BG For-Sale Unstable PREP 36 48 CC1=CCN(C(=O)OCc2ccccc2)[C@@H](C)C1 ZINC000217711303 BG For-Sale Unstable CAPN2 42 33 CC1=CCN(C(=O)OCc2ccccc2)[C@@H](C)C1 ZINC000217711303 BG For-Sale Unstable KLK5 40 38 CC1=CCN(C(=O)OCc2ccccc2)[C@@H](C)C1 ZINC000217711303 BG For-Sale Unstable NAAA 43 40 CC1=CCN(C(=O)OCc2ccccc2)[C@@H](C)C1 ZINC000217711303 BG For-Sale Unstable SLC12A5 61 38 CCOc1cc(C(=O)Cl)cc(Cl)c1OCc1ccc(F)cc1Cl ZINC000217711318 GK In-Stock Unstable P2RX7 49 39 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCCC(=O)NCCc3c[nH]cn3)[C@@H]21 ZINC000217711349 JF In-Stock Unstable HRH3 33 45 C[C@H]1CCCCN1CCCNS(=O)(=O)CCCO ZINC000217711370 CC For-Sale Unstable HRH3 25 46 Cn1cc(NS(=O)(=O)c2cccc(/C=C\C(=O)O)c2)cn1 ZINC000217711386 DD For-Sale Unstable HDAC8 60 60 Cn1cc(NS(=O)(=O)c2cccc(/C=C\C(=O)O)c2)cn1 ZINC000217711386 DD For-Sale Unstable HDAC1 35 60 Cn1cc(NS(=O)(=O)c2cccc(/C=C\C(=O)O)c2)cn1 ZINC000217711386 DD For-Sale Unstable HDAC6 32 60 CC1=CC[C@@H](C)N(C(=O)OCc2ccccc2)C1 ZINC000217711409 BG For-Sale Unstable CELA1 21 44 CC1=CC[C@@H](C)N(C(=O)OCc2ccccc2)C1 ZINC000217711409 BG For-Sale Unstable ELANE 29 41 CC1=CC[C@@H](C)N(C(=O)OCc2ccccc2)C1 ZINC000217711409 BG For-Sale Unstable PAPA1_CARPA 41 32 CC1=CC[C@@H](C)N(C(=O)OCc2ccccc2)C1 ZINC000217711409 BG For-Sale Unstable PREP 34 46 CC1=CC[C@@H](C)N(C(=O)OCc2ccccc2)C1 ZINC000217711409 BG For-Sale Unstable CAPNS1 46 31 CC1=CC[C@@H](C)N(C(=O)OCc2ccccc2)C1 ZINC000217711409 BG For-Sale Unstable LGMN 51 34 CC1=CC[C@@H](C)N(C(=O)OCc2ccccc2)C1 ZINC000217711409 BG For-Sale Unstable CAPN2 44 34 CC1=CC[C@@H](C)N(C(=O)OCc2ccccc2)C1 ZINC000217711409 BG For-Sale Unstable ACE2 18 40 CC1=CC[C@@H](C)N(C(=O)OCc2ccccc2)C1 ZINC000217711409 BG For-Sale Unstable NAAA 41 40 CC1=CC[C@@H](C)N(C(=O)OCc2ccccc2)C1 ZINC000217711409 BG For-Sale Unstable SLC12A5 65 37 COc1ccccc1/C=C/NC(=O)NCC(=O)O ZINC000217711412 CD For-Sale Unstable CYP1B1 22 40 COc1ccccc1/C=C/NC(=O)NCC(=O)O ZINC000217711412 CD For-Sale Unstable TLR4 19 45 O=C(OCCC1CC1)c1cc(Cl)nc2ccccc12 ZINC000217711473 CH On-Demand Unstable HTR4 15 45 O=C(OCCC1CC1)c1cc(Cl)nc2ccccc12 ZINC000217711473 CH On-Demand Unstable ACACB 27 43 CC1=CC[C@H](C)N(C(=O)OCc2ccccc2)C1 ZINC000217711478 BG For-Sale Unstable CELA1 21 44 CC1=CC[C@H](C)N(C(=O)OCc2ccccc2)C1 ZINC000217711478 BG For-Sale Unstable ELANE 29 41 CC1=CC[C@H](C)N(C(=O)OCc2ccccc2)C1 ZINC000217711478 BG For-Sale Unstable PAPA1_CARPA 41 32 CC1=CC[C@H](C)N(C(=O)OCc2ccccc2)C1 ZINC000217711478 BG For-Sale Unstable PREP 34 46 CC1=CC[C@H](C)N(C(=O)OCc2ccccc2)C1 ZINC000217711478 BG For-Sale Unstable CAPNS1 46 31 CC1=CC[C@H](C)N(C(=O)OCc2ccccc2)C1 ZINC000217711478 BG For-Sale Unstable LGMN 51 34 CC1=CC[C@H](C)N(C(=O)OCc2ccccc2)C1 ZINC000217711478 BG For-Sale Unstable CAPN2 44 34 CC1=CC[C@H](C)N(C(=O)OCc2ccccc2)C1 ZINC000217711478 BG For-Sale Unstable ACE2 18 40 CC1=CC[C@H](C)N(C(=O)OCc2ccccc2)C1 ZINC000217711478 BG For-Sale Unstable NAAA 41 40 CC1=CC[C@H](C)N(C(=O)OCc2ccccc2)C1 ZINC000217711478 BG For-Sale Unstable SLC12A5 65 37 O=C(O)c1cc(O)n(-c2ccccc2Oc2ccccc2)n1 ZINC000217711511 CG In-Stock Anodyne RPA1 67 40 COc1ccccc1/C=C/NC(=O)N(CCO)CCO ZINC000217711519 CC For-Sale Unstable TLR4 15 44 COC(=O)[C@@H](O)CNC(=O)c1cc(OC)cc(OC)c1 ZINC000217711524 CB On-Demand Unstable DRD4 43 34 CCOc1cc(C(=O)Cl)cc(Br)c1OCc1ccc(F)cc1 ZINC000217711547 GJ In-Stock Unstable THRA 18 43 CCOc1cc(C(=O)Cl)cc(Br)c1OCc1ccc(F)cc1 ZINC000217711547 GJ In-Stock Unstable THRB 21 43 CCN(C(=O)c1ccc(OC)c(/C=C\C(=O)O)c1)C1CC1 ZINC000217711550 CE For-Sale Unstable ACKR3 40 33 COC(=O)[C@H](O)CNC(=O)c1cc(OC)cc(OC)c1 ZINC000217711627 CB On-Demand Unstable DRD4 43 34 CCNc1ccc(S(=O)(=O)NCC)cc1C(=O)O ZINC000217711630 CD In-Stock Unstable CA1 16 42 CSC1C[C@@H]2CC[C@H](C1)N2C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217711659 EJ In-Stock Unstable EPHX2 36 43 CSC1C[C@@H]2CC[C@H](C1)N2C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217711659 EJ In-Stock Unstable TRPM8 56 39 CN(C)[C@@H]1[C@H]2CC[C@@H]1CN(C(=O)c1ccc(-c3cccc(F)c3)cc1)C2 ZINC000217711758 FH In-Stock Unstable L3MBTL3 32 40 CN(C)[C@@H]1[C@H]2CC[C@@H]1CN(C(=O)c1ccc(-c3cccc(F)c3)cc1)C2 ZINC000217711758 FH In-Stock Unstable SLC6A7 0 45 c1ccc(C2CCC(N[C@@H]3CCN4CCC[C@@H]34)CC2)cc1 ZINC000217711772 CH For-Sale Unstable SLC18A3 82 51 CCOc1cc(C(=O)Cl)cc(I)c1OCc1cccc(F)c1 ZINC000217711774 IJ In-Stock Unstable MAOB 15 48 CCOc1cc(C(=O)Cl)cc(I)c1OCc1cccc(F)c1 ZINC000217711774 IJ In-Stock Unstable ACR 16 43 CSC[C@@](C)(O)CNC(=O)c1ccc(CNC(N)=O)cc1 ZINC000217711827 DC On-Demand Unstable CYNT 19 45 COc1ccccc1/C=C/NC(=O)NCCCCCC(=O)O ZINC000217711830 DF For-Sale Unstable DRD2 18 44 COc1ccccc1/C=C/NC(=O)NCCCCCC(=O)O ZINC000217711830 DF For-Sale Unstable DRD3 31 44 COc1ccccc1/C=C/NC(=O)NCCCCCC(=O)O ZINC000217711830 DF For-Sale Unstable HDAC5 17 43 COc1ccccc1/C=C/NC(=O)NCCCCCC(=O)O ZINC000217711830 DF For-Sale Unstable EPHX2 21 40 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NC1CC1 ZINC000217711844 CD In-Stock Unstable NEU3 0 40 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NC1CC1 ZINC000217711844 CD In-Stock Unstable CCR8 87 43 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NC1CC1 ZINC000217711844 CD In-Stock Unstable SFRP1 106 39 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NC1CC1 ZINC000217711844 CD In-Stock Unstable WNT3 81 38 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccncc2)CC(=O)O4)cc1O ZINC000217711847 IH In-Stock Unstable AKR1B1 0 48 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccncc2)CC(=O)O4)cc1O ZINC000217711847 IH In-Stock Unstable CYP1B1 57 36 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccncc2)CC(=O)O4)cc1O ZINC000217711847 IH In-Stock Unstable CYP1A1 41 48 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccncc2)CC(=O)O4)cc1O ZINC000217711847 IH In-Stock Unstable CYP1A2 32 40 c1ccc(C2CCC(N[C@H]3CCN4CCC[C@@H]34)CC2)cc1 ZINC000217711854 CH For-Sale Unstable SLC18A3 82 51 Cc1ncsc1CCN(C)C(=O)[C@@H]1CCCCN1C(=O)c1ccccc1 ZINC000217711881 FG In-Stock Unstable COLA 62 46 Cc1ncsc1CCN(C)C(=O)[C@@H]1CCCCN1C(=O)c1ccccc1 ZINC000217711881 FG In-Stock Unstable CPT1A 60 35 Cc1ncsc1CCN(C)C(=O)[C@@H]1CCCCN1C(=O)c1ccccc1 ZINC000217711881 FG In-Stock Unstable PREP 50 38 CCOc1cc(C(=O)Cl)cc(Br)c1OCc1cccc(F)c1 ZINC000217711889 GJ In-Stock Unstable THRA 19 44 CCOc1cc(C(=O)Cl)cc(Br)c1OCc1cccc(F)c1 ZINC000217711889 GJ In-Stock Unstable MAOB 17 48 CCOc1cc(C(=O)Cl)cc(Br)c1OCc1cccc(F)c1 ZINC000217711889 GJ In-Stock Unstable THRB 20 43 CSC[C@](C)(O)CNC(=O)c1ccc(CNC(N)=O)cc1 ZINC000217711914 DC On-Demand Unstable CYNT 19 45 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccncc2)CC(=O)O4)cc1O ZINC000217711923 IH In-Stock Unstable AKR1B1 0 48 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccncc2)CC(=O)O4)cc1O ZINC000217711923 IH In-Stock Unstable CYP1B1 57 36 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccncc2)CC(=O)O4)cc1O ZINC000217711923 IH In-Stock Unstable CYP1A1 41 48 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccncc2)CC(=O)O4)cc1O ZINC000217711923 IH In-Stock Unstable CYP1A2 32 40 COC(=O)[C@@H](O)CNC(=O)CSCc1ccc(Cl)cc1 ZINC000217711930 DD On-Demand Unstable LTA4H 27 41 CNc1ccc(S(=O)(=O)N[C@@H](C)COC)cc1C(=O)O ZINC000217711955 DC In-Stock Unstable MMP12 50 37 Cc1ncsc1CCN(C)C(=O)[C@H]1CCCCN1C(=O)c1ccccc1 ZINC000217711962 FG In-Stock Unstable COLA 62 46 Cc1ncsc1CCN(C)C(=O)[C@H]1CCCCN1C(=O)c1ccccc1 ZINC000217711962 FG In-Stock Unstable CPT1A 60 35 Cc1ncsc1CCN(C)C(=O)[C@H]1CCCCN1C(=O)c1ccccc1 ZINC000217711962 FG In-Stock Unstable PREP 50 38 COc1ccc2ccc(OC)c(C(=O)Cl)c2c1 ZINC000217711996 CG In-Stock Unstable PTGS2 44 45 COc1ccc2ccc(OC)c(C(=O)Cl)c2c1 ZINC000217711996 CG In-Stock Unstable CYP1B1 45 38 COc1ccc2ccc(OC)c(C(=O)Cl)c2c1 ZINC000217711996 CG In-Stock Unstable NQO2 33 43 COc1ccc2ccc(OC)c(C(=O)Cl)c2c1 ZINC000217711996 CG In-Stock Unstable CA7 0 45 COc1ccc2ccc(OC)c(C(=O)Cl)c2c1 ZINC000217711996 CG In-Stock Unstable CYP11B2 18 40 COc1ccc2ccc(OC)c(C(=O)Cl)c2c1 ZINC000217711996 CG In-Stock Unstable MTNR1A 109 51 COc1ccc2ccc(OC)c(C(=O)Cl)c2c1 ZINC000217711996 CG In-Stock Unstable MTNR1B 93 51 COc1ccc2ccc(OC)c(C(=O)Cl)c2c1 ZINC000217711996 CG In-Stock Unstable TUBB2B 42 39 COc1ccc2ccc(OC)c(C(=O)Cl)c2c1 ZINC000217711996 CG In-Stock Unstable TUBB1 41 39 COc1ccc2ccc(OC)c(C(=O)Cl)c2c1 ZINC000217711996 CG In-Stock Unstable AKR1C3 35 40 COc1ccc2ccc(OC)c(C(=O)Cl)c2c1 ZINC000217711996 CG In-Stock Unstable ABCG2 38 41 COc1ccc2ccc(OC)c(C(=O)Cl)c2c1 ZINC000217711996 CG In-Stock Unstable AKR1C2 42 36 COC(=O)[C@H](O)CNC(=O)CSCc1ccc(Cl)cc1 ZINC000217712016 DD On-Demand Unstable LTA4H 27 41 CNc1ccc(S(=O)(=O)N[C@H](C)COC)cc1C(=O)O ZINC000217712040 DC In-Stock Unstable MMP12 50 37 COc1ccccc1/C=C/NC(=O)NCCCC(=O)O ZINC000217712109 CD For-Sale Unstable DRD3 26 44 Cn1cnnc1SCCNC(=O)[C@H]1CCCC[C@H]1C(=O)N1CCCC1 ZINC000217712111 FD In-Stock Unstable CTSK 18 46 COC(=O)[C@@H](O)CNC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217712129 CB On-Demand Unstable DRD4 43 34 COC(=O)[C@@H](O)CNC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217712129 CB On-Demand Unstable CACNA1C 62 42 COC(=O)[C@@H](O)CNC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217712129 CB On-Demand Unstable CACNA1D 97 42 COC(=O)[C@@H](O)CNC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217712129 CB On-Demand Unstable PYGL 22 40 COC(=O)[C@@H](O)CNC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217712129 CB On-Demand Unstable UREA_CANEN 20 45 Cc1cc2ncc3c(n2n1)CCN(S(=O)(=O)c1ccccc1C(F)(F)F)C3 ZINC000217712139 GF In-Stock Unstable AKR1C3 41 35 O=C(NC[C@@H]1CCCN2CCCC[C@H]12)[C@@H]1CC(=O)N(c2ccc(F)cc2)C1 ZINC000217712148 FF In-Stock Unstable VACHT_TETCF 0 41 O=C(O)c1cc(O)n(-c2ccc(I)cc2)n1 ZINC000217712155 ED In-Stock Anodyne RPA1 82 48 CCOc1cc(C(=O)Cl)cc(I)c1OCc1ccccc1 ZINC000217712198 HJ In-Stock Unstable PPIA 42 36 CCOc1cc(C(=O)Cl)cc(I)c1OCc1ccccc1 ZINC000217712198 HJ In-Stock Unstable PTGER1 50 36 CCOc1cc(C(=O)Cl)cc(I)c1OCc1ccccc1 ZINC000217712198 HJ In-Stock Unstable ACR 20 41 COC(=O)[C@H](O)CNC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217712211 CB On-Demand Unstable DRD4 43 34 COC(=O)[C@H](O)CNC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217712211 CB On-Demand Unstable CACNA1C 62 42 COC(=O)[C@H](O)CNC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217712211 CB On-Demand Unstable CACNA1D 97 42 COC(=O)[C@H](O)CNC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217712211 CB On-Demand Unstable PYGL 22 40 COC(=O)[C@H](O)CNC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217712211 CB On-Demand Unstable UREA_CANEN 20 45 COc1ccc(B2OC(C)(C)C(C)(C)O2)cc1S(=O)(=O)NC1CC1 ZINC000217712213 FD For-Sale Unstable ADRA1D 23 40 COc1ccc(B2OC(C)(C)C(C)(C)O2)cc1S(=O)(=O)NC1CC1 ZINC000217712213 FD For-Sale Unstable ADRA1A 16 40 COc1ccc(B2OC(C)(C)C(C)(C)O2)cc1S(=O)(=O)NC1CC1 ZINC000217712213 FD For-Sale Unstable ADRA1B 28 40 COc1ccc(B2OC(C)(C)C(C)(C)O2)cc1S(=O)(=O)NC1CC1 ZINC000217712213 FD For-Sale Unstable BRD4 15 48 COc1ccccc1/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O ZINC000217712220 DE For-Sale Unstable ACE 17 40 COc1ccccc1/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O ZINC000217712220 DE For-Sale Unstable FOLH1 22 48 COc1ccccc1/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O ZINC000217712220 DE For-Sale Unstable MME 39 43 COc1ccccc1/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O ZINC000217712220 DE For-Sale Unstable ANPEP 45 51 COc1ccccc1/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O ZINC000217712220 DE For-Sale Unstable RNPEP 23 40 COc1ccccc1/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O ZINC000217712220 DE For-Sale Unstable PAPA1_CARPA 44 32 COc1ccccc1/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O ZINC000217712220 DE For-Sale Unstable CAPNS1 57 35 COc1ccccc1/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O ZINC000217712220 DE For-Sale Unstable CAPN1 62 43 COc1ccccc1/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O ZINC000217712220 DE For-Sale Unstable CAPN2 67 36 COc1ccccc1/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O ZINC000217712220 DE For-Sale Unstable LAP3 15 40 COc1ccccc1/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O ZINC000217712220 DE For-Sale Unstable FPR1 84 42 COc1ccccc1/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O ZINC000217712220 DE For-Sale Unstable NPR 74 36 COc1ccccc1/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O ZINC000217712220 DE For-Sale Unstable AMP1_PLAFQ 20 40 COc1ccccc1/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O ZINC000217712220 DE For-Sale Unstable Q9N6S8_PLAFA 47 31 O=C(NC[C@@H]1CCCN2CCCC[C@H]12)[C@H]1CC(=O)N(c2ccc(F)cc2)C1 ZINC000217712227 FF In-Stock Unstable VACHT_TETCF 0 41 CNc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217712270 DE In-Stock Unstable LPL 38 41 CNc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217712270 DE In-Stock Unstable AKR1C3 60 42 CNc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217712270 DE In-Stock Unstable LIPG 15 41 CNc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217712270 DE In-Stock Unstable LIMK2 49 40 N#CCN1CCN(C(=O)c2cnn3ccccc23)CC1 ZINC000217712292 CC On-Demand Unstable EPHB3 30 42 Cc1ccc(NC(=O)[C@@H](c2ccccc2)N(C)Cc2nc3ccsc3c(=O)[nH]2)cc1 ZINC000217712296 HI On-Demand Unstable KIF11 15 41 O=C(NCC[C@@H]1CCCN2CCCC[C@H]12)[C@H](O)c1ccccc1 ZINC000217712302 DE In-Stock Unstable SLC6A1 48 38 COc1ccccc1/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O ZINC000217712316 DE For-Sale Unstable ACE 17 40 COc1ccccc1/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O ZINC000217712316 DE For-Sale Unstable FOLH1 22 48 COc1ccccc1/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O ZINC000217712316 DE For-Sale Unstable MME 39 43 COc1ccccc1/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O ZINC000217712316 DE For-Sale Unstable ANPEP 45 51 COc1ccccc1/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O ZINC000217712316 DE For-Sale Unstable RNPEP 23 40 COc1ccccc1/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O ZINC000217712316 DE For-Sale Unstable PAPA1_CARPA 44 32 COc1ccccc1/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O ZINC000217712316 DE For-Sale Unstable CAPNS1 57 35 COc1ccccc1/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O ZINC000217712316 DE For-Sale Unstable CAPN1 62 43 COc1ccccc1/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O ZINC000217712316 DE For-Sale Unstable CAPN2 67 36 COc1ccccc1/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O ZINC000217712316 DE For-Sale Unstable LAP3 15 40 COc1ccccc1/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O ZINC000217712316 DE For-Sale Unstable FPR1 84 42 COc1ccccc1/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O ZINC000217712316 DE For-Sale Unstable NPR 74 36 COc1ccccc1/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O ZINC000217712316 DE For-Sale Unstable AMP1_PLAFQ 20 40 COc1ccccc1/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O ZINC000217712316 DE For-Sale Unstable Q9N6S8_PLAFA 47 31 COC(=O)[C@@H](O)CNC(=O)c1cccnc1OC ZINC000217712326 CB On-Demand Unstable G2YM83_BOTF4 50 30 CC(C)[C@H]1CC[C@H](C)C[C@H]1N[C@H](C)Cc1ccc(Br)cc1 ZINC000217712365 FK For-Sale Unstable TRPM8 16 42 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccnc2)CC(=O)O4)cc1O ZINC000217712366 IH In-Stock Unstable AKR1B1 0 45 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccnc2)CC(=O)O4)cc1O ZINC000217712366 IH In-Stock Unstable CYP1B1 49 34 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccnc2)CC(=O)O4)cc1O ZINC000217712366 IH In-Stock Unstable CYP1A1 34 45 Cc1ccc(NC(=O)[C@H](c2ccccc2)N(C)Cc2nc3ccsc3c(=O)[nH]2)cc1 ZINC000217712391 HI On-Demand Unstable KIF11 15 41 CNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217712392 FD In-Stock Unstable CA2 25 43 CNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217712392 FD In-Stock Unstable TBXA2R 56 48 CNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217712392 FD In-Stock Unstable TBXAS1 31 46 CNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217712392 FD In-Stock Unstable BMP1 71 39 CNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217712392 FD In-Stock Unstable CA1 26 48 CNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217712392 FD In-Stock Unstable MMP13 64 43 CNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217712392 FD In-Stock Unstable ADAM17 41 38 CNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217712392 FD In-Stock Unstable ALOX15B 0 40 CNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217712392 FD In-Stock Unstable CA4 15 43 CNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217712392 FD In-Stock Unstable MMP2 38 43 CNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217712392 FD In-Stock Unstable MMP3 52 38 CNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217712392 FD In-Stock Unstable MMP8 30 43 CNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217712392 FD In-Stock Unstable MMP14 19 43 CNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217712392 FD In-Stock Unstable ALOX15 51 40 CNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217712392 FD In-Stock Unstable MMP9 56 43 CNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217712392 FD In-Stock Unstable MMP12 30 43 CNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217712392 FD In-Stock Unstable CA12 19 46 CNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217712392 FD In-Stock Unstable PTGDR 22 40 CNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217712392 FD In-Stock Unstable MMP7 40 38 CNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217712392 FD In-Stock Unstable IAP 0 46 CNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217712392 FD In-Stock Unstable CA9 24 46 CNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217712392 FD In-Stock Unstable MMP1 58 39 CNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217712392 FD In-Stock Unstable AKR1C3 32 52 CNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217712392 FD In-Stock Unstable AKR1C2 53 40 CNc1ccc(S(=O)(=O)NCCc2ccc(OC)cc2)cc1C(=O)O ZINC000217712392 FD In-Stock Unstable A6YCJ1_9METZ 15 41 COC(=O)[C@H](O)CNC(=O)c1cccnc1OC ZINC000217712409 CB On-Demand Unstable G2YM83_BOTF4 50 30 NS(=O)(=O)c1ccc(F)c(C(=O)OCCC2CC2)c1 ZINC000217712413 CD On-Demand Unstable CA2 59 42 NS(=O)(=O)c1ccc(F)c(C(=O)OCCC2CC2)c1 ZINC000217712413 CD On-Demand Unstable CA1 52 42 NS(=O)(=O)c1ccc(F)c(C(=O)OCCC2CC2)c1 ZINC000217712413 CD On-Demand Unstable CA7 48 39 NS(=O)(=O)c1ccc(F)c(C(=O)OCCC2CC2)c1 ZINC000217712413 CD On-Demand Unstable CA4 55 42 NS(=O)(=O)c1ccc(F)c(C(=O)OCCC2CC2)c1 ZINC000217712413 CD On-Demand Unstable CA12 33 41 NS(=O)(=O)c1ccc(F)c(C(=O)OCCC2CC2)c1 ZINC000217712413 CD On-Demand Unstable CA9 32 42 COc1ccccc1/C=C/NC(=O)N[C@@H](CCSC)C(=O)O ZINC000217712422 DE For-Sale Unstable FOLH1 20 41 COc1ccccc1/C=C/NC(=O)N[C@@H](CCSC)C(=O)O ZINC000217712422 DE For-Sale Unstable NAALAD2 42 35 COc1ccccc1/C=C/NC(=O)N[C@@H](CCSC)C(=O)O ZINC000217712422 DE For-Sale Unstable PAM 0 41 COc1ccccc1/C=C/NC(=O)N[C@@H](CCSC)C(=O)O ZINC000217712422 DE For-Sale Unstable FPR1 43 43 COc1ccccc1/C=C/NC(=O)N[C@@H](CCSC)C(=O)O ZINC000217712422 DE For-Sale Unstable FPRL2 0 40 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccnc2)CC(=O)O4)cc1O ZINC000217712455 IH In-Stock Unstable AKR1B1 0 45 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccnc2)CC(=O)O4)cc1O ZINC000217712455 IH In-Stock Unstable CYP1B1 49 34 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccnc2)CC(=O)O4)cc1O ZINC000217712455 IH In-Stock Unstable CYP1A1 34 45 CC(C)[C@H]1CC[C@H](C)C[C@@H]1N[C@@H](C)Cc1ccc(Br)cc1 ZINC000217712457 FK For-Sale Unstable TRPM8 16 42 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable HTR1A 49 43 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable DRD2 54 46 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable FKBP1A 42 41 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable DRD1 22 41 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable ACHE 29 42 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable HRH2 53 44 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable ADRA1D 57 40 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable HTR2A 45 42 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable HTR2C 34 41 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable SLC6A1 49 36 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable ADRA1A 70 40 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable HRH1 18 42 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable ADRA1B 54 40 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable DRD3 76 46 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable OPRL1 18 45 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable HTR4 32 51 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable CHRM4 15 42 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable CHRM3 15 42 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable DRD5 26 41 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable LTA4H 35 43 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable HTR7 35 40 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable HRH3 78 48 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable SIGMAR1 66 51 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable KLK3 44 33 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable CTSB 56 42 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable PAPA1_CARPA 52 34 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable CYSP_TRYCR 48 41 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable CTSK 36 43 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable CTSL 43 40 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable BCHE 31 43 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable CCR3 25 46 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable KCNA3 15 40 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable SCN2A 23 48 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable CHRNA7 34 53 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable PREP 42 52 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable CAPNS1 66 36 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable EBP 15 45 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable HNMT 93 38 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable ABCB1 23 45 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable CTSS 18 43 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable CAPN1 77 50 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable CAPN2 130 58 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable TGM2 45 50 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable DPP7 42 39 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable NPR 76 45 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable F13A1 32 40 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable NPFFR1 57 36 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable SLC12A5 70 39 O=C(NCCCN1CCCCC1)OCc1ccccc1 ZINC000217712490 CF For-Sale Unstable TMPRSS11D 22 40 CCNc1ccc(S(=O)(=O)NC[C@@H]2CCCO2)cc1C(=O)O ZINC000217712491 ED In-Stock Unstable BDKRB1 23 44 COC(=O)c1ccccc1S(=O)(=O)NCCNC(C)=O ZINC000217712498 DB On-Demand Unstable MTNR1A 42 34 COC(=O)c1ccccc1S(=O)(=O)NCCNC(C)=O ZINC000217712498 DB On-Demand Unstable PRTN3 46 34 CCCC#C/C=C\C(=O)OC ZINC000217712500 AD Annotated Unstable HCAR2 0 41 COc1ccccc1/C=C/NC(=O)N[C@H](CCSC)C(=O)O ZINC000217712508 DE For-Sale Unstable FOLH1 20 41 COc1ccccc1/C=C/NC(=O)N[C@H](CCSC)C(=O)O ZINC000217712508 DE For-Sale Unstable NAALAD2 42 35 COc1ccccc1/C=C/NC(=O)N[C@H](CCSC)C(=O)O ZINC000217712508 DE For-Sale Unstable PAM 0 41 COc1ccccc1/C=C/NC(=O)N[C@H](CCSC)C(=O)O ZINC000217712508 DE For-Sale Unstable FPR1 43 43 COc1ccccc1/C=C/NC(=O)N[C@H](CCSC)C(=O)O ZINC000217712508 DE For-Sale Unstable FPRL2 0 40 CC(C)[C@H]1CC[C@H](C)C[C@@H]1N[C@H](C)Cc1ccc(Br)cc1 ZINC000217712552 FK For-Sale Unstable TRPM8 16 42 COc1ccc(C(=O)NCC2CC2)cc1/C=C\C(=O)O ZINC000217712557 CD For-Sale Unstable GRIN2B 17 40 COc1ccc(C(=O)NCC2CC2)cc1/C=C\C(=O)O ZINC000217712557 CD For-Sale Unstable CACNA1I 58 38 COc1ccc(C(=O)NCC2CC2)cc1/C=C\C(=O)O ZINC000217712557 CD For-Sale Unstable HSPB1 0 46 COc1ccc(C(=O)NCC2CC2)cc1/C=C\C(=O)O ZINC000217712557 CD For-Sale Unstable PFG6PD 0 40 CCNc1ccc(S(=O)(=O)NC[C@H]2CCCO2)cc1C(=O)O ZINC000217712569 ED In-Stock Unstable BDKRB1 23 44 CCCC#C/C=C/C(=O)OC ZINC000217712589 AD Annotated Unstable HCAR2 0 41 COc1ccccc1/C=C/NC(=O)N[C@@H](C)c1ccc(OC)c(OC)c1 ZINC000217712616 FH For-Sale Unstable KCNQ2 49 38 CNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217712655 DE In-Stock Unstable CCR8 74 42 CNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217712655 DE In-Stock Unstable SFRP1 95 35 CNc1ccc(S(=O)(=O)NC2CCCCC2)cc1C(=O)O ZINC000217712655 DE In-Stock Unstable WNT3 77 35 CSC[C@@](C)(O)CNC(=O)/C=C/c1ccc(C)c(Cl)c1 ZINC000217712684 DF On-Demand Unstable PYGL 28 50 COc1ccccc1/C=C/NC(=O)N[C@H](C)c1ccc(OC)c(OC)c1 ZINC000217712704 FH For-Sale Unstable KCNQ2 49 38 COC(=O)[C@@H](NC(=O)CCn1cc(C(C)=O)c2ccccc21)C(C)C ZINC000217712714 EF In-Stock Unstable CNR1 30 49 COC(=O)[C@@H](NC(=O)CCn1cc(C(C)=O)c2ccccc21)C(C)C ZINC000217712714 EF In-Stock Unstable CNR2 24 49 CSC[C@](C)(O)CNC(=O)/C=C/c1ccc(C)c(Cl)c1 ZINC000217712781 DF On-Demand Unstable PYGL 28 50 CCOc1cc(C(=O)Cl)cc(I)c1OCc1ccccc1Cl ZINC000217712783 JK In-Stock Unstable FABP4 18 47 CCOc1cc(C(=O)Cl)cc(I)c1OCc1ccccc1Cl ZINC000217712783 JK In-Stock Unstable FABP5 34 47 COc1ccc([C@@H](C)NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217712825 EH For-Sale Unstable CYP1B1 33 44 COc1ccc([C@@H](C)NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217712825 EH For-Sale Unstable ACACA 48 42 COc1ccc([C@@H](C)NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217712825 EH For-Sale Unstable ACACB 17 42 COC(OC)[C@H](C)NC(=O)/C=C\C(=O)O ZINC000217712829 BB For-Sale Unstable HCAR2 30 43 NS(=O)(=O)c1ccc(Cl)c(C(=O)OCCC2CC2)c1 ZINC000217712876 DD On-Demand Unstable CA2 69 46 NS(=O)(=O)c1ccc(Cl)c(C(=O)OCCC2CC2)c1 ZINC000217712876 DD On-Demand Unstable CA1 62 46 NS(=O)(=O)c1ccc(Cl)c(C(=O)OCCC2CC2)c1 ZINC000217712876 DD On-Demand Unstable CA7 61 42 NS(=O)(=O)c1ccc(Cl)c(C(=O)OCCC2CC2)c1 ZINC000217712876 DD On-Demand Unstable CA13 29 40 NS(=O)(=O)c1ccc(Cl)c(C(=O)OCCC2CC2)c1 ZINC000217712876 DD On-Demand Unstable CA5B 33 42 NS(=O)(=O)c1ccc(Cl)c(C(=O)OCCC2CC2)c1 ZINC000217712876 DD On-Demand Unstable CA4 62 46 NS(=O)(=O)c1ccc(Cl)c(C(=O)OCCC2CC2)c1 ZINC000217712876 DD On-Demand Unstable CA5A 38 42 NS(=O)(=O)c1ccc(Cl)c(C(=O)OCCC2CC2)c1 ZINC000217712876 DD On-Demand Unstable CA14 34 40 NS(=O)(=O)c1ccc(Cl)c(C(=O)OCCC2CC2)c1 ZINC000217712876 DD On-Demand Unstable CA12 39 42 NS(=O)(=O)c1ccc(Cl)c(C(=O)OCCC2CC2)c1 ZINC000217712876 DD On-Demand Unstable CA9 40 46 NS(=O)(=O)c1ccc(Cl)c(C(=O)OCCC2CC2)c1 ZINC000217712876 DD On-Demand Unstable CAH_METTE 48 40 NS(=O)(=O)c1ccc(Cl)c(C(=O)OCCC2CC2)c1 ZINC000217712876 DD On-Demand Unstable CYNT 33 40 NS(=O)(=O)c1ccc(Cl)c(C(=O)OCCC2CC2)c1 ZINC000217712876 DD On-Demand Unstable NCE103 27 40 NS(=O)(=O)c1ccc(Cl)c(C(=O)OCCC2CC2)c1 ZINC000217712876 DD On-Demand Unstable CA15 24 40 NS(=O)(=O)c1ccc(Cl)c(C(=O)OCCC2CC2)c1 ZINC000217712876 DD On-Demand Unstable CA 0 40 NS(=O)(=O)c1ccc(Cl)c(C(=O)OCCC2CC2)c1 ZINC000217712876 DD On-Demand Unstable A6YCJ1_9METZ 26 40 O=C(O)c1cc(O)n(-c2ccccc2C(=O)O)n1 ZINC000217712885 BC In-Stock Anodyne BCL2 0 40 O=C(O)c1cc(O)n(-c2ccccc2C(=O)O)n1 ZINC000217712885 BC In-Stock Anodyne RPA1 72 40 O=C(Cl)c1ccc2oc(-c3cccc(F)c3)nc2c1 ZINC000217712889 CI In-Stock Reactive CETP 0 45 O=C(Cl)c1ccc2oc(-c3cccc(F)c3)nc2c1 ZINC000217712889 CI In-Stock Reactive HPSE 72 49 COc1ccc([C@H](C)NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217712904 EH For-Sale Unstable CYP1B1 33 44 COc1ccc([C@H](C)NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217712904 EH For-Sale Unstable ACACA 48 42 COc1ccc([C@H](C)NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217712904 EH For-Sale Unstable ACACB 17 42 COC(OC)[C@@H](C)NC(=O)/C=C\C(=O)O ZINC000217712906 BB For-Sale Unstable HCAR2 30 43 O=C(Cl)c1ccc2oc(-c3cccc(Cl)c3)nc2c1 ZINC000217712989 CJ In-Stock Reactive CETP 0 47 O=C(Cl)c1ccc2oc(-c3cccc(Cl)c3)nc2c1 ZINC000217712989 CJ In-Stock Reactive HPSE 64 50 O=C(Cl)c1ccc2oc(-c3cccc(Cl)c3)nc2c1 ZINC000217712989 CJ In-Stock Reactive IMDH_CRYPV 30 44 NS(=O)(=O)c1ccc(CCC(=O)OCCC2CC2)cc1 ZINC000217712999 CD On-Demand Unstable CA2 119 55 NS(=O)(=O)c1ccc(CCC(=O)OCCC2CC2)cc1 ZINC000217712999 CD On-Demand Unstable CA6 22 45 NS(=O)(=O)c1ccc(CCC(=O)OCCC2CC2)cc1 ZINC000217712999 CD On-Demand Unstable CA1 102 48 NS(=O)(=O)c1ccc(CCC(=O)OCCC2CC2)cc1 ZINC000217712999 CD On-Demand Unstable CA7 81 48 NS(=O)(=O)c1ccc(CCC(=O)OCCC2CC2)cc1 ZINC000217712999 CD On-Demand Unstable CA13 26 45 NS(=O)(=O)c1ccc(CCC(=O)OCCC2CC2)cc1 ZINC000217712999 CD On-Demand Unstable CA5B 50 40 NS(=O)(=O)c1ccc(CCC(=O)OCCC2CC2)cc1 ZINC000217712999 CD On-Demand Unstable CA4 81 50 NS(=O)(=O)c1ccc(CCC(=O)OCCC2CC2)cc1 ZINC000217712999 CD On-Demand Unstable CA5A 52 40 NS(=O)(=O)c1ccc(CCC(=O)OCCC2CC2)cc1 ZINC000217712999 CD On-Demand Unstable CA14 60 43 NS(=O)(=O)c1ccc(CCC(=O)OCCC2CC2)cc1 ZINC000217712999 CD On-Demand Unstable CA12 81 48 NS(=O)(=O)c1ccc(CCC(=O)OCCC2CC2)cc1 ZINC000217712999 CD On-Demand Unstable CA9 89 48 NS(=O)(=O)c1ccc(CCC(=O)OCCC2CC2)cc1 ZINC000217712999 CD On-Demand Unstable CAH_METTE 25 45 NS(=O)(=O)c1ccc(CCC(=O)OCCC2CC2)cc1 ZINC000217712999 CD On-Demand Unstable CYNT 34 43 NS(=O)(=O)c1ccc(CCC(=O)OCCC2CC2)cc1 ZINC000217712999 CD On-Demand Unstable NCE103 25 55 NS(=O)(=O)c1ccc(CCC(=O)OCCC2CC2)cc1 ZINC000217712999 CD On-Demand Unstable CA15 17 45 NS(=O)(=O)c1ccc(CCC(=O)OCCC2CC2)cc1 ZINC000217712999 CD On-Demand Unstable MTCA1 40 37 NS(=O)(=O)c1ccc(CCC(=O)OCCC2CC2)cc1 ZINC000217712999 CD On-Demand Unstable P96878_MYCTU 49 39 NS(=O)(=O)c1ccc(CCC(=O)OCCC2CC2)cc1 ZINC000217712999 CD On-Demand Unstable CA 0 55 NS(=O)(=O)c1ccc(CCC(=O)OCCC2CC2)cc1 ZINC000217712999 CD On-Demand Unstable A6YCJ1_9METZ 24 45 NS(=O)(=O)c1ccc(CCC(=O)OCCC2CC2)cc1 ZINC000217712999 CD On-Demand Unstable Q5TU56_ANOGA 0 45 CC(C)c1cc(C(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)[nH]n1 ZINC000217713032 ED In-Stock Unstable CHRNA4 29 46 CCOc1ccccc1C(=O)N1CC(n2ccnn2)C1 ZINC000217713052 CD In-Stock Unstable HCN1 46 36 CCOc1ccccc1C(=O)N1CC(n2ccnn2)C1 ZINC000217713052 CD In-Stock Unstable HCN4 46 36 COC(=O)[C@@H](O)CNC(=O)[C@@H](OC)c1ccccc1 ZINC000217713056 CC On-Demand Unstable CAPN2 43 34 O=C(Cl)c1ccc2oc(-c3cccc(Br)c3)nc2c1 ZINC000217713086 EJ In-Stock Reactive HPSE 61 41 COc1ccc(OC)c(C(=O)NC[C@@](C)(O)CSC)c1 ZINC000217713092 CD On-Demand Unstable MT-ND1 23 41 COc1ccc(OC)c(C(=O)NC[C@@](C)(O)CSC)c1 ZINC000217713092 CD On-Demand Unstable AKR1C2 45 35 CNc1ccc(S(=O)(=O)NCCCOC)cc1C(=O)O ZINC000217713102 DC In-Stock Unstable CASP3 24 41 CNc1ccc(S(=O)(=O)NCCCOC)cc1C(=O)O ZINC000217713102 DC In-Stock Unstable BDKRB1 0 42 O=C(/C=C\c1cccc([N+](=O)[O-])c1)NCC1CC(O)C1 ZINC000217713116 CD For-Sale Unstable CACNA1C 47 37 O=C(/C=C\c1cccc([N+](=O)[O-])c1)NCC1CC(O)C1 ZINC000217713116 CD For-Sale Unstable CACNA1D 77 37 O=C(/C=C\c1cccc([N+](=O)[O-])c1)NCC1CC(O)C1 ZINC000217713116 CD For-Sale Unstable TRPM8 0 54 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)Nc1ccncc1)C(=O)OC2 ZINC000217713138 HH In-Stock Unstable IMPDH1 0 63 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)Nc1ccncc1)C(=O)OC2 ZINC000217713138 HH In-Stock Unstable IMPDH2 0 63 CCOC(=O)c1ccc(N2C(=O)[C@H]3[C@H]4C[C@@H]([C@@H]5ON=C(c6ccc(Cl)cc6Cl)[C@@H]45)[C@H]3C2=O)cc1 ZINC000217713140 JI In-Stock Unstable DPP8 61 35 CCOC(=O)c1ccc(N2C(=O)[C@H]3[C@H]4C[C@@H]([C@@H]5ON=C(c6ccc(Cl)cc6Cl)[C@@H]45)[C@H]3C2=O)cc1 ZINC000217713140 JI In-Stock Unstable DPP9 59 35 COC(=O)[C@H](O)CNC(=O)[C@@H](OC)c1ccccc1 ZINC000217713149 CC On-Demand Unstable CAPN2 43 34 O=[N+]([O-])c1ccc(CNC[C@@H](O)CCc2ccccc2)cc1 ZINC000217713159 DF On-Demand Unstable CCR3 21 46 O=C(Cl)c1ccc2oc(-c3cccc(I)c3)nc2c1 ZINC000217713179 GI In-Stock Reactive HPSE 51 39 COc1ccc(OC)c(C(=O)NC[C@](C)(O)CSC)c1 ZINC000217713195 CD On-Demand Unstable MT-ND1 23 41 COc1ccc(OC)c(C(=O)NC[C@](C)(O)CSC)c1 ZINC000217713195 CD On-Demand Unstable AKR1C2 45 35 COc1cc(-n2nc(C(=O)O)cc2O)c(OC)cc1Cl ZINC000217713214 CD In-Stock Unstable RPA1 69 38 COC(=O)[C@@H](O)CNC(=O)[C@H](OC)c1ccccc1 ZINC000217713245 CC On-Demand Unstable CAPN2 43 34 O=[N+]([O-])c1ccc(CNC[C@H](O)CCc2ccccc2)cc1 ZINC000217713253 DF On-Demand Unstable CCR3 21 46 O=C(c1ccc(-n2cccc2)cc1)N1CC(n2ccnn2)C1 ZINC000217713271 CD In-Stock Unstable SLC6A7 0 50 N#Cc1ccccc1-c1ccc(C(=O)Cl)o1 ZINC000217713312 BG In-Stock Reactive MAP 0 46 N#Cc1ccccc1-c1ccc(C(=O)Cl)o1 ZINC000217713312 BG In-Stock Reactive SLC9A1 15 40 COC(=O)[C@H](O)CNC(=O)[C@H](OC)c1ccccc1 ZINC000217713330 CC On-Demand Unstable CAPN2 43 34 COc1ccc(/C=C\C(=O)NCC2CC(O)C2)cc1 ZINC000217713345 CD On-Demand Unstable PTGS2 0 46 COc1ccc(/C=C\C(=O)NCC2CC(O)C2)cc1 ZINC000217713345 CD On-Demand Unstable HDAC8 27 57 COc1ccc(/C=C\C(=O)NCC2CC(O)C2)cc1 ZINC000217713345 CD On-Demand Unstable MMP2 23 49 COc1ccc(/C=C\C(=O)NCC2CC(O)C2)cc1 ZINC000217713345 CD On-Demand Unstable HDAC1 30 47 COc1ccc(/C=C\C(=O)NCC2CC(O)C2)cc1 ZINC000217713345 CD On-Demand Unstable HDAC4 0 47 COc1ccc(/C=C\C(=O)NCC2CC(O)C2)cc1 ZINC000217713345 CD On-Demand Unstable HDAC6 20 57 COc1ccc(/C=C\C(=O)NCC2CC(O)C2)cc1 ZINC000217713345 CD On-Demand Unstable MMP9 27 49 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NCc1ccccc1 ZINC000217713358 EE In-Stock Unstable AKR1C3 24 42 NCc1nc2cccc(N)c2n1Cc1ccccc1 ZINC000217713388 CE For-Sale Unstable TLR7 64 47 N#Cc1ccc(-c2ccc(C(=O)Cl)o2)cc1 ZINC000217713419 BG In-Stock Reactive MAPKAPK2 30 41 N#Cc1ccc(-c2ccc(C(=O)Cl)o2)cc1 ZINC000217713419 BG In-Stock Reactive SCN10A 27 52 CCc1ccc([C@@H](C)NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217713433 DI For-Sale Unstable KCNQ2 44 33 COC(=O)[C@@H](O)CNC(=O)CNC(=O)c1ccccc1 ZINC000217713441 CB On-Demand Unstable CA2 28 44 COC(=O)[C@@H](O)CNC(=O)CNC(=O)c1ccccc1 ZINC000217713441 CB On-Demand Unstable ITGAV 44 40 CNc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O ZINC000217713467 CC In-Stock Unstable TBXA2R 41 33 CNc1ccc(S(=O)(=O)NCCCO)cc1C(=O)O ZINC000217713467 CC In-Stock Unstable CASP3 22 43 NCc1nc2ccc(N)cc2n1Cc1ccccc1 ZINC000217713485 CE For-Sale Unstable ALOX5AP 23 40 NCc1nc2ccc(N)cc2n1Cc1ccccc1 ZINC000217713485 CE For-Sale Unstable AGTR1B 15 51 NCc1nc2ccc(N)cc2n1Cc1ccccc1 ZINC000217713485 CE For-Sale Unstable PDE6D 40 35 NCc1nc2ccc(N)cc2n1Cc1ccccc1 ZINC000217713485 CE For-Sale Unstable TLR7 48 41 CCc1ccc([C@H](C)NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217713517 DI For-Sale Unstable KCNQ2 44 33 O=C(Cl)c1ccc2oc(-c3cncc(Br)c3)nc2c1 ZINC000217713524 EI In-Stock Reactive HPSE 47 34 COC(=O)[C@H](O)CNC(=O)CNC(=O)c1ccccc1 ZINC000217713525 CB On-Demand Unstable CA2 28 44 COC(=O)[C@H](O)CNC(=O)CNC(=O)c1ccccc1 ZINC000217713525 CB On-Demand Unstable ITGAV 44 40 Cc1cccc(/C=C\C(=O)NCC2CC(O)C2)c1 ZINC000217713560 BD For-Sale Unstable HDAC8 61 39 Cc1cccc(/C=C\C(=O)NCC2CC(O)C2)c1 ZINC000217713560 BD For-Sale Unstable MMP2 0 45 Cc1cccc(/C=C\C(=O)NCC2CC(O)C2)c1 ZINC000217713560 BD For-Sale Unstable HDAC6 41 39 Cc1cccc(/C=C\C(=O)NCC2CC(O)C2)c1 ZINC000217713560 BD For-Sale Unstable MMP9 0 45 Cc1cccc(/C=C\C(=O)NCC2CC(O)C2)c1 ZINC000217713560 BD For-Sale Unstable MMP1 0 45 Cc1cccc(/C=C\C(=O)NCC2CC(O)C2)c1 ZINC000217713560 BD For-Sale Unstable IMA1 0 42 CCCCCCCN[C@@H](CC)CCO ZINC000217713564 BF For-Sale Unstable CQSS 40 31 CNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217713569 DD In-Stock Unstable CA2 27 46 CNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217713569 DD In-Stock Unstable GNRHR 18 43 CNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217713569 DD In-Stock Unstable CASP3 22 44 CNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217713569 DD In-Stock Unstable CA1 25 40 CNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217713569 DD In-Stock Unstable CA5B 27 40 CNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217713569 DD In-Stock Unstable CA4 24 46 CNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217713569 DD In-Stock Unstable CA5A 31 40 CNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217713569 DD In-Stock Unstable CASP6 19 44 CNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217713569 DD In-Stock Unstable AKR1C3 32 43 CNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217713569 DD In-Stock Unstable NAMPT 27 40 CC[C@@H](C)[C@@H](C)NC(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217713575 CF For-Sale Unstable CTRB1 34 40 CC[C@@H](C)[C@@H](C)NC(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217713575 CF For-Sale Unstable CELA2A 19 40 NCc1nc2c(N)cccc2n1Cc1ccccc1 ZINC000217713591 CE For-Sale Unstable TLR7 57 41 CN(CCC(=O)Nc1sc2c(c1C#N)CCCCC2)Cc1nc2ccsc2c(=O)[nH]1 ZINC000217713618 IH On-Demand Unstable MAPK10 17 44 CN(CCC(=O)Nc1sc2c(c1C#N)CCCCC2)Cc1nc2ccsc2c(=O)[nH]1 ZINC000217713618 IH On-Demand Unstable VIPR1 32 49 COc1ccccc1/C=C/NC(=O)N[C@@H](C)c1ccc2c(c1)CCCC2 ZINC000217713629 FJ For-Sale Unstable KCNQ2 47 37 CCCCCCCN[C@H](CC)CCO ZINC000217713648 BF For-Sale Unstable CQSS 40 31 Nc1ncnc2c1nc(S)n2CC(=O)O ZINC000217713650 BB In-Stock Unstable AHCY 77 40 Nc1ncnc2c1nc(S)n2CC(=O)O ZINC000217713650 BB In-Stock Unstable OXGR1 99 37 Nc1ncnc2c1nc(S)n2CC(=O)O ZINC000217713650 BB In-Stock Unstable HSP90B1 73 37 COC(=O)[C@@H](O)CNC(=O)c1ccccc1OC ZINC000217713655 CB On-Demand Unstable KCNA3 45 61 COC(=O)[C@@H](O)CNC(=O)c1ccccc1OC ZINC000217713655 CB On-Demand Unstable ITGAV 17 41 COC(=O)[C@@H](O)CNC(=O)c1ccccc1OC ZINC000217713655 CB On-Demand Unstable HCN1 68 44 COC(=O)[C@@H](O)CNC(=O)c1ccccc1OC ZINC000217713655 CB On-Demand Unstable HCN4 54 44 COC(=O)[C@@H](O)CNC(=O)c1ccccc1OC ZINC000217713655 CB On-Demand Unstable KCNK3 65 49 COC(=O)[C@@H](O)CNC(=O)c1ccccc1OC ZINC000217713655 CB On-Demand Unstable KCNK9 54 49 O=C(/C=C\c1ccc(F)c(Cl)c1)NCC1CC(O)C1 ZINC000217713658 CE For-Sale Unstable PYGL 28 48 O=C(/C=C\c1ccc(F)c(Cl)c1)NCC1CC(O)C1 ZINC000217713658 CE For-Sale Unstable HDAC8 20 40 CC[C@H](C)[C@@H](C)NC(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217713665 CF For-Sale Unstable CTRB1 34 40 CC[C@H](C)[C@@H](C)NC(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217713665 CF For-Sale Unstable CELA2A 19 40 CNc1ccc(C(=O)O)cc1S(=O)(=O)NCCc1ccccc1 ZINC000217713676 ED In-Stock Unstable TBXA2R 47 41 CNc1ccc(C(=O)O)cc1S(=O)(=O)NCCc1ccccc1 ZINC000217713676 ED In-Stock Unstable AKR1C3 25 60 NCc1cccc2nc(N)n(Cc3ccccc3)c12 ZINC000217713700 CE For-Sale Unstable TLR7 58 43 O=C(N[C@@H]1CCN2CCC[C@@H]12)c1ccc(CCl)cc1 ZINC000217713709 CE For-Sale Unstable SSTR3 30 42 O=C(N[C@@H]1CCN2CCC[C@@H]12)c1ccc(CCl)cc1 ZINC000217713709 CE For-Sale Unstable L3MBTL3 49 37 CCCCOc1ccc(NC(=O)N2[C@H]3CC[C@H]2CC(SC)C3)cc1 ZINC000217713722 EJ In-Stock Unstable PLA2G4B 65 35 CCCCOc1ccc(NC(=O)N2[C@H]3CC[C@H]2CC(SC)C3)cc1 ZINC000217713722 EJ In-Stock Unstable FAAH 24 42 COc1ccccc1/C=C/NC(=O)N[C@H](C)c1ccc2c(c1)CCCC2 ZINC000217713723 FJ For-Sale Unstable KCNQ2 47 37 COC(=O)[C@H](O)CNC(=O)c1ccccc1OC ZINC000217713735 CB On-Demand Unstable KCNA3 45 61 COC(=O)[C@H](O)CNC(=O)c1ccccc1OC ZINC000217713735 CB On-Demand Unstable ITGAV 17 41 COC(=O)[C@H](O)CNC(=O)c1ccccc1OC ZINC000217713735 CB On-Demand Unstable HCN1 68 44 COC(=O)[C@H](O)CNC(=O)c1ccccc1OC ZINC000217713735 CB On-Demand Unstable HCN4 54 44 COC(=O)[C@H](O)CNC(=O)c1ccccc1OC ZINC000217713735 CB On-Demand Unstable KCNK3 65 49 COC(=O)[C@H](O)CNC(=O)c1ccccc1OC ZINC000217713735 CB On-Demand Unstable KCNK9 54 49 CC[C@@H](C)[C@@H](C)NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217713746 CF For-Sale Unstable AGTR2 16 41 CC[C@@H](C)[C@@H](C)NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217713746 CF For-Sale Unstable HDAC8 18 43 CC[C@@H](C)[C@@H](C)NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217713746 CF For-Sale Unstable CTRB1 29 40 CC[C@@H](C)[C@@H](C)NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217713746 CF For-Sale Unstable NR1H4 49 36 CC[C@@H](C)[C@@H](C)NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217713746 CF For-Sale Unstable CELA2A 15 40 CC[C@@H](C)[C@@H](C)NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217713746 CF For-Sale Unstable KCNK3 47 35 Nc1ccc(OCC(=O)O)c(-c2nc3ccccc3[nH]2)c1 ZINC000217713749 CE In-Stock Unstable FABP4 25 41 Nc1ccc(OCC(=O)O)c(-c2nc3ccccc3[nH]2)c1 ZINC000217713749 CE In-Stock Unstable FGFR1 23 41 Nc1ccc(OCC(=O)O)c(-c2nc3ccccc3[nH]2)c1 ZINC000217713749 CE In-Stock Unstable FLT1 0 41 Nc1ccc(OCC(=O)O)c(-c2nc3ccccc3[nH]2)c1 ZINC000217713749 CE In-Stock Unstable PTGDR2 25 44 CNc1ccc(S(=O)(=O)NCCCOC(C)C)cc1C(=O)O ZINC000217713776 ED In-Stock Unstable CASP3 16 42 O=C(N[C@H]1CCN2CCC[C@@H]12)c1ccc(CCl)cc1 ZINC000217713799 CE For-Sale Unstable SSTR3 30 42 O=C(N[C@H]1CCN2CCC[C@@H]12)c1ccc(CCl)cc1 ZINC000217713799 CE For-Sale Unstable L3MBTL3 49 37 NCc1ccc2nc(N)n(Cc3ccccc3)c2c1 ZINC000217713808 CE For-Sale Unstable ALOX5AP 27 40 NCc1ccc2nc(N)n(Cc3ccccc3)c2c1 ZINC000217713808 CE For-Sale Unstable TLR7 48 41 CC[C@H](C)[C@@H](C)NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217713833 CF For-Sale Unstable AGTR2 16 41 CC[C@H](C)[C@@H](C)NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217713833 CF For-Sale Unstable HDAC8 18 43 CC[C@H](C)[C@@H](C)NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217713833 CF For-Sale Unstable CTRB1 29 40 CC[C@H](C)[C@@H](C)NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217713833 CF For-Sale Unstable NR1H4 49 36 CC[C@H](C)[C@@H](C)NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217713833 CF For-Sale Unstable CELA2A 15 40 CC[C@H](C)[C@@H](C)NC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217713833 CF For-Sale Unstable KCNK3 47 35 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NC1CCCCCC1 ZINC000217713867 EF In-Stock Unstable CCR8 87 48 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NC1CCCCCC1 ZINC000217713867 EF In-Stock Unstable SFRP1 104 37 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NC1CCCCCC1 ZINC000217713867 EF In-Stock Unstable WNT3 82 36 CCNc1ccc(C(=O)O)cc1S(=O)(=O)NC1CCCCCC1 ZINC000217713867 EF In-Stock Unstable BRD4 23 41 C=CCCCNC(=O)c1ccc(Br)cc1 ZINC000217713903 CG On-Demand Unstable FOLH1 21 43 NCc1ccc2c(c1)nc(N)n2Cc1ccccc1 ZINC000217713907 CE For-Sale Unstable ALOX5AP 22 42 NCc1ccc2c(c1)nc(N)n2Cc1ccccc1 ZINC000217713907 CE For-Sale Unstable TLR7 46 41 CN(C(=O)Cc1ccccc1)[C@H](CO)c1ccccc1 ZINC000217713918 CE For-Sale Unstable OPRK1 35 64 CN(C(=O)Cc1ccccc1)[C@H](CO)c1ccccc1 ZINC000217713918 CE For-Sale Unstable CPA1 26 41 CN(C(=O)Cc1ccccc1)[C@H](CO)c1ccccc1 ZINC000217713918 CE For-Sale Unstable CCR5 20 44 CN(C(=O)Cc1ccccc1)[C@H](CO)c1ccccc1 ZINC000217713918 CE For-Sale Unstable NPY5R 30 40 O=C(/C=C\c1ccccc1)OCCNC(=O)c1ccccc1 ZINC000217713929 CF On-Demand Unstable HDAC8 15 43 O=C(/C=C\c1ccccc1)OCCNC(=O)c1ccccc1 ZINC000217713929 CF On-Demand Unstable CTRB1 21 41 O=C(/C=C\c1ccccc1)OCCNC(=O)c1ccccc1 ZINC000217713929 CF On-Demand Unstable F3 18 42 O=C(/C=C\c1ccccc1)OCCNC(=O)c1ccccc1 ZINC000217713929 CF On-Demand Unstable MMP2 15 44 O=C(/C=C\c1ccccc1)OCCNC(=O)c1ccccc1 ZINC000217713929 CF On-Demand Unstable HCAR2 28 41 O=C(/C=C\c1ccccc1)OCCNC(=O)c1ccccc1 ZINC000217713929 CF On-Demand Unstable AKR1B10 39 50 C[C@@H](C(=O)Nc1ccc(OCc2ccccc2)cc1)N(C)Cc1nc2ccsc2c(=O)[nH]1 ZINC000217713931 II On-Demand Unstable TSHR 43 33 C[C@@H](C(=O)Nc1ccc(OCc2ccccc2)cc1)N(C)Cc1nc2ccsc2c(=O)[nH]1 ZINC000217713931 II On-Demand Unstable LTA4H 18 40 O=C(N[C@@H]1CCN2CCC[C@@H]12)c1cccc(CCl)c1 ZINC000217713934 CE For-Sale Unstable DRD4 16 42 O=C(N[C@@H]1CCN2CCC[C@@H]12)c1cccc(CCl)c1 ZINC000217713934 CE For-Sale Unstable SIGMAR1 18 45 O=C(N[C@@H]1CCN2CCC[C@@H]12)c1cccc(CCl)c1 ZINC000217713934 CE For-Sale Unstable CHRNA7 23 40 CCCCCCOc1ccc2c(c1)NCCC2 ZINC000217713960 BI For-Sale Unstable THRA 41 40 CCCCCCOc1ccc2c(c1)NCCC2 ZINC000217713960 BI For-Sale Unstable THRB 28 40 CCCCCCOc1ccc2c(c1)NCCC2 ZINC000217713960 BI For-Sale Unstable PLA2G4B 85 38 COc1ccccc1/C=C/NC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217713963 FK For-Sale Unstable EPHX1 0 47 COc1ccccc1/C=C/NC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217713963 FK For-Sale Unstable LTA4H 33 40 COc1ccccc1/C=C/NC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217713963 FK For-Sale Unstable CYP1B1 25 42 COc1ccccc1/C=C/NC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217713963 FK For-Sale Unstable CA1 45 45 COc1ccccc1/C=C/NC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217713963 FK For-Sale Unstable RAF1 39 47 COc1ccccc1/C=C/NC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217713963 FK For-Sale Unstable KDR 26 44 COc1ccccc1/C=C/NC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217713963 FK For-Sale Unstable MTNR1B 20 45 COc1ccccc1/C=C/NC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217713963 FK For-Sale Unstable NPY5R 27 41 COc1ccccc1/C=C/NC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217713963 FK For-Sale Unstable CA12 17 45 COc1ccccc1/C=C/NC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217713963 FK For-Sale Unstable PDGFRA 56 44 COc1ccccc1/C=C/NC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217713963 FK For-Sale Unstable CA9 17 45 COc1ccccc1/C=C/NC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217713963 FK For-Sale Unstable Q8MMZ8_EIMTE 42 47 O=C(NCc1ccco1)c1ccc(NC(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc1 ZINC000217713975 IG In-Stock Unstable CHRNA4 27 43 NCc1cccc2c1nc(N)n2Cc1ccccc1 ZINC000217714019 CE For-Sale Unstable TLR7 43 43 O=C(N[C@H]1CCN2CCC[C@@H]12)c1cccc(CCl)c1 ZINC000217714023 CE For-Sale Unstable DRD4 16 42 O=C(N[C@H]1CCN2CCC[C@@H]12)c1cccc(CCl)c1 ZINC000217714023 CE For-Sale Unstable SIGMAR1 18 45 O=C(N[C@H]1CCN2CCC[C@@H]12)c1cccc(CCl)c1 ZINC000217714023 CE For-Sale Unstable CHRNA7 23 40 C[C@H](C(=O)Nc1ccc(OCc2ccccc2)cc1)N(C)Cc1nc2ccsc2c(=O)[nH]1 ZINC000217714032 II On-Demand Unstable TSHR 43 33 C[C@H](C(=O)Nc1ccc(OCc2ccccc2)cc1)N(C)Cc1nc2ccsc2c(=O)[nH]1 ZINC000217714032 II On-Demand Unstable LTA4H 18 40 O=S(=O)(c1ccccc1Cl)N1CC(n2ccnn2)C1 ZINC000217714033 CD In-Stock Unstable CCR1 15 41 COc1ccccc1/C=C/NC(=O)Nc1cc(Cl)ccc1C ZINC000217714070 DI For-Sale Unstable S1PR4 23 41 CCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217714089 EE In-Stock Unstable CA2 21 44 CCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217714089 EE In-Stock Unstable GNRHR 18 44 CCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217714089 EE In-Stock Unstable CASP3 21 43 CCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217714089 EE In-Stock Unstable CA4 17 44 CCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217714089 EE In-Stock Unstable CASP6 19 43 CCNc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)O ZINC000217714089 EE In-Stock Unstable AKR1C3 22 42 CC[C@@H](CCO)N[C@@H](C)C(=O)O ZINC000217714165 AC For-Sale Unstable BHMT2 44 28 O=C(N[C@@H]1CCN2CCC[C@@H]12)[C@H](Cl)c1ccccc1 ZINC000217714170 CE For-Sale Unstable SLC18A3 64 36 COc1ccc(OC)c(NC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217714174 EH For-Sale Unstable CYP1B1 57 52 COc1ccc(OC)c(NC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217714174 EH For-Sale Unstable MTNR1A 30 51 COc1ccc(OC)c(NC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217714174 EH For-Sale Unstable MTNR1B 31 51 COc1ccc(OC)c(NC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217714174 EH For-Sale Unstable CYP1A1 40 43 COc1ccc(OC)c(NC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217714174 EH For-Sale Unstable ABCG2 23 44 COc1ccc(OC)c(NC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217714174 EH For-Sale Unstable AKR1C2 50 34 COc1ccc(OC)c(NC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217714174 EH For-Sale Unstable CYSP_PLAFA 40 40 C[C@@H](C(=O)NC(c1ccccc1)c1ccccc1)N(C)Cc1nc2ccsc2c(=O)[nH]1 ZINC000217714175 IH On-Demand Unstable PARP3 21 42 NC(=O)c1ccc(-n2nc(C(=O)O)cc2O)cc1 ZINC000217714196 BC In-Stock Unstable RPA1 84 44 C[C@@H](CN1CCCC1)NC(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217714203 DE For-Sale Unstable P2RX3 28 42 C[C@@H](CN1CCCC1)NC(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217714203 DE For-Sale Unstable PLD1 45 35 O=C(N[C@@H]1CCN2CCC[C@@H]12)[C@@H](Cl)c1ccccc1 ZINC000217714235 CE For-Sale Unstable SLC18A3 64 36 CSC1C[C@@H]2CC[C@H](C1)N2C(=O)NCc1ccc(Cl)cc1 ZINC000217714247 DH In-Stock Unstable SLC6A1 54 47 CSC1C[C@@H]2CC[C@H](C1)N2C(=O)NCc1ccc(Cl)cc1 ZINC000217714247 DH In-Stock Unstable SLC6A3 24 45 CSC1C[C@@H]2CC[C@H](C1)N2C(=O)NCc1ccc(Cl)cc1 ZINC000217714247 DH In-Stock Unstable P2RX7 24 46 COc1ccccc1CCN1[C@H]2CC[C@H]1CC(=O)C2 ZINC000217714250 CE For-Sale Unstable HTR1A 41 44 COc1ccccc1CCN1[C@H]2CC[C@H]1CC(=O)C2 ZINC000217714250 CE For-Sale Unstable DRD2 26 41 COc1ccccc1CCN1[C@H]2CC[C@H]1CC(=O)C2 ZINC000217714250 CE For-Sale Unstable SLC18A2 26 45 COc1ccccc1CCN1[C@H]2CC[C@H]1CC(=O)C2 ZINC000217714250 CE For-Sale Unstable MBTPS1 51 35 CN(C[C@@H]1CCCN1C)c1ccc(F)cc1CBr ZINC000217714254 DG For-Sale Unstable CHRNA10 73 46 CN(C[C@@H]1CCCN1C)c1ccc(F)cc1CBr ZINC000217714254 DG For-Sale Unstable ACKR3 60 35 CC[C@H](CCO)N[C@@H](C)C(=O)O ZINC000217714259 AC For-Sale Unstable BHMT2 44 28 C[C@H](C(=O)NC(c1ccccc1)c1ccccc1)N(C)Cc1nc2ccsc2c(=O)[nH]1 ZINC000217714261 IH On-Demand Unstable PARP3 21 42 Nc1ccc([N+](=O)[O-])cc1C(=O)OCCC1CC1 ZINC000217714264 CE On-Demand Unstable CACNA1C 54 39 Nc1ccc([N+](=O)[O-])cc1C(=O)OCCC1CC1 ZINC000217714264 CE On-Demand Unstable CACNA1D 83 39 Nc1ccc([N+](=O)[O-])cc1C(=O)OCCC1CC1 ZINC000217714264 CE On-Demand Unstable SLC27A4 45 34 CCc1cccc(C)c1NC(=O)N/C=C/c1ccccc1OC ZINC000217714283 DI For-Sale Unstable ACAT 0 43 CC(=O)Nc1ccc(CN[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217714287 CD For-Sale Unstable SSTR3 18 40 COC(=O)[C@@H](O)CNC(=O)c1cc(Br)ccc1O ZINC000217714289 DC On-Demand Unstable PYK 75 38 C[C@H](CN1CCCC1)NC(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217714290 DE For-Sale Unstable P2RX3 28 42 C[C@H](CN1CCCC1)NC(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217714290 DE For-Sale Unstable PLD1 45 35 CCNc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217714308 DF In-Stock Unstable LPL 37 40 CCNc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217714308 DF In-Stock Unstable NEU3 0 40 CCNc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217714308 DF In-Stock Unstable AKR1C3 54 40 CCNc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccccc1 ZINC000217714308 DF In-Stock Unstable LIMK2 52 44 O=C(N[C@H]1CCN2CCC[C@@H]12)[C@H](Cl)c1ccccc1 ZINC000217714319 CE For-Sale Unstable SLC18A3 64 36 CC[C@@H](CCO)N[C@H](C)C(=O)O ZINC000217714324 AC For-Sale Unstable BHMT2 44 28 CN(C[C@H]1CCCN1C)c1ccc(F)cc1CBr ZINC000217714335 DG For-Sale Unstable CHRNA10 73 46 CN(C[C@H]1CCCN1C)c1ccc(F)cc1CBr ZINC000217714335 DG For-Sale Unstable ACKR3 60 35 CC(=O)Nc1ccc(CN[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217714366 CD For-Sale Unstable SSTR3 18 40 COC(=O)[C@H](O)CNC(=O)c1cc(Br)ccc1O ZINC000217714373 DC For-Sale Unstable PYK 93 38 CSC[C@@](C)(O)CNC(=O)c1ccc(S(C)(=O)=O)cc1 ZINC000217714376 DC On-Demand Unstable CA2 22 41 CSC[C@@](C)(O)CNC(=O)c1ccc(S(C)(=O)=O)cc1 ZINC000217714376 DC On-Demand Unstable PTGS2 17 40 CSC[C@@](C)(O)CNC(=O)c1ccc(S(C)(=O)=O)cc1 ZINC000217714376 DC On-Demand Unstable LOX1.1 48 40 CSC[C@@](C)(O)CNC(=O)c1ccc(S(C)(=O)=O)cc1 ZINC000217714376 DC On-Demand Unstable O49150_SOLTU 56 40 CSC[C@@](C)(O)CNC(=O)c1ccc(S(C)(=O)=O)cc1 ZINC000217714376 DC On-Demand Unstable CYNT 26 41 CN(CCC(=O)Nc1sc2c(c1C#N)CCCC2)Cc1nc2ccsc2c(=O)[nH]1 ZINC000217714378 IG On-Demand Unstable MAPK10 18 44 CN(CCC(=O)Nc1sc2c(c1C#N)CCCC2)Cc1nc2ccsc2c(=O)[nH]1 ZINC000217714378 IG On-Demand Unstable VIPR1 32 50 O=C(O)/C=C\c1ccc(C(=O)Nc2nc3c(s2)CCC3)s1 ZINC000217714392 DG For-Sale Unstable SLC27A1 32 43 COc1ccccc1/C=C/NC(=O)Nc1c(C)cc(C)cc1C ZINC000217714394 DI For-Sale Unstable CYP1B1 19 40 COc1ccccc1/C=C/NC(=O)Nc1c(C)cc(C)cc1C ZINC000217714394 DI For-Sale Unstable PYGL 41 40 O=C(N[C@H]1CCN2CCC[C@@H]12)[C@@H](Cl)c1ccccc1 ZINC000217714416 CE For-Sale Unstable SLC18A3 64 36 CC[C@H](CCO)N[C@H](C)C(=O)O ZINC000217714418 AC For-Sale Unstable BHMT2 44 28 COc1ccc(C)cc1-n1nc(C(=O)O)cc1O ZINC000217714428 BD In-Stock Unstable RPA1 66 40 CN(C[C@@H]1CCCN1C)c1c(F)cc(CBr)cc1F ZINC000217714436 EG For-Sale Unstable CHRNA10 70 43 CN(C[C@@H]1CCCN1C)c1c(F)cc(CBr)cc1F ZINC000217714436 EG For-Sale Unstable ACKR3 63 32 CSC[C@](C)(O)CNC(=O)c1ccc(S(C)(=O)=O)cc1 ZINC000217714463 DC On-Demand Unstable CA2 22 41 CSC[C@](C)(O)CNC(=O)c1ccc(S(C)(=O)=O)cc1 ZINC000217714463 DC On-Demand Unstable PTGS2 17 40 CSC[C@](C)(O)CNC(=O)c1ccc(S(C)(=O)=O)cc1 ZINC000217714463 DC On-Demand Unstable LOX1.1 48 40 CSC[C@](C)(O)CNC(=O)c1ccc(S(C)(=O)=O)cc1 ZINC000217714463 DC On-Demand Unstable O49150_SOLTU 56 40 CSC[C@](C)(O)CNC(=O)c1ccc(S(C)(=O)=O)cc1 ZINC000217714463 DC On-Demand Unstable CYNT 26 41 Clc1ccc(CN[C@@H]2CCN3CCC[C@@H]23)c(Cl)c1 ZINC000217714468 CG For-Sale Unstable P2RX7 29 45 Clc1ccc(CN[C@@H]2CCN3CCC[C@@H]23)c(Cl)c1 ZINC000217714468 CG For-Sale Unstable EPHX2 15 46 C[C@@H](Cn1ccnc1)NC(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217714477 DD For-Sale Unstable TBXAS1 52 46 COc1cccc(CCN2[C@H]3CC[C@H]2CC(=O)C3)c1 ZINC000217714504 CE For-Sale Unstable DRD4 40 31 COc1cccc(CCN2[C@H]3CC[C@H]2CC(=O)C3)c1 ZINC000217714504 CE For-Sale Unstable SLC18A2 36 47 COc1cccc(CCN2[C@H]3CC[C@H]2CC(=O)C3)c1 ZINC000217714504 CE For-Sale Unstable KCNH2 25 43 COc1cccc(CCN2[C@H]3CC[C@H]2CC(=O)C3)c1 ZINC000217714504 CE For-Sale Unstable SIGMAR1 24 57 COc1cccc(CCN2[C@H]3CC[C@H]2CC(=O)C3)c1 ZINC000217714504 CE For-Sale Unstable MTNR1A 15 42 COc1cccc(CCN2[C@H]3CC[C@H]2CC(=O)C3)c1 ZINC000217714504 CE For-Sale Unstable MTNR1B 16 42 COc1cccc(CCN2[C@H]3CC[C@H]2CC(=O)C3)c1 ZINC000217714504 CE For-Sale Unstable Q8WSF8_APLCA 15 41 NS(=O)(=O)c1cc(C(=O)OCCC2CC2)ccc1Cl ZINC000217714505 DD On-Demand Unstable CA2 29 49 NS(=O)(=O)c1cc(C(=O)OCCC2CC2)ccc1Cl ZINC000217714505 DD On-Demand Unstable CA6 33 44 NS(=O)(=O)c1cc(C(=O)OCCC2CC2)ccc1Cl ZINC000217714505 DD On-Demand Unstable CA1 28 49 NS(=O)(=O)c1cc(C(=O)OCCC2CC2)ccc1Cl ZINC000217714505 DD On-Demand Unstable CA7 28 49 NS(=O)(=O)c1cc(C(=O)OCCC2CC2)ccc1Cl ZINC000217714505 DD On-Demand Unstable CA13 47 49 NS(=O)(=O)c1cc(C(=O)OCCC2CC2)ccc1Cl ZINC000217714505 DD On-Demand Unstable CA4 29 49 NS(=O)(=O)c1cc(C(=O)OCCC2CC2)ccc1Cl ZINC000217714505 DD On-Demand Unstable CA12 15 41 Cc1nc2ccc(C(=O)NC[C@@H]3CCCN4CCCC[C@H]34)cc2nc1C ZINC000217714511 FG In-Stock Unstable CACNA1I 48 35 CN(C[C@H]1CCCN1C)c1c(F)cc(CBr)cc1F ZINC000217714520 EG For-Sale Unstable CHRNA10 70 43 CN(C[C@H]1CCCN1C)c1c(F)cc(CBr)cc1F ZINC000217714520 EG For-Sale Unstable ACKR3 63 32 C[C@@H]1CCCCN1CCCNS(=O)(=O)CCCCO ZINC000217714531 CC For-Sale Unstable HRH3 21 43 O=C(O)c1cc(O)n(-c2ccc(Cl)c(C(F)(F)F)c2)n1 ZINC000217714550 DF In-Stock Anodyne RPA1 102 50 Clc1ccc(CN[C@H]2CCN3CCC[C@@H]23)c(Cl)c1 ZINC000217714560 CG For-Sale Unstable P2RX7 29 45 Clc1ccc(CN[C@H]2CCN3CCC[C@@H]23)c(Cl)c1 ZINC000217714560 CG For-Sale Unstable EPHX2 15 46 C[C@H](Cn1ccnc1)NC(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217714561 DD For-Sale Unstable TBXAS1 52 46 CCOc1ccc(C(=O)NC[C@@](C)(O)CSC)cc1OC ZINC000217714595 DD On-Demand Unstable MT-ND1 24 40 COc1ccccc1/C=C/NC(=O)Nc1ccc(F)cc1 ZINC000217714617 CH For-Sale Unstable KDR 15 41 COc1ccccc1/C=C/NC(=O)Nc1ccc(F)cc1 ZINC000217714617 CH For-Sale Unstable PDGFRA 42 41 COc1ccccc1/C=C/NC(=O)Nc1ccc(F)cc1 ZINC000217714617 CH For-Sale Unstable TLR4 17 43 C[C@H]1CCCCN1CCCNS(=O)(=O)CCCCO ZINC000217714622 CC For-Sale Unstable HRH3 21 43 CN(C[C@@H]1CCCN1C)c1cccc(Cl)c1CBr ZINC000217714636 EH For-Sale Unstable CHRNA10 71 43 O=C(O)/C=C\c1ccc(C(=O)NCCn2cccn2)cc1 ZINC000217714642 CD For-Sale Unstable CYP24A1 31 41 O=C(O)/C=C\c1ccc(C(=O)NCCn2cccn2)cc1 ZINC000217714642 CD For-Sale Unstable CYP27B1 39 41 CCNc1ccc(S(=O)(=O)NCC(C)C)cc1C(=O)O ZINC000217714651 DD In-Stock Unstable CASP3 17 40 CCNc1ccc(S(=O)(=O)NCC(C)C)cc1C(=O)O ZINC000217714651 DD In-Stock Unstable BDKRB1 0 42 CCNc1ccc(S(=O)(=O)NCC(C)C)cc1C(=O)O ZINC000217714651 DD In-Stock Unstable MTNN 41 33 C=CCCCNC(=O)/C=C\c1ccccc1 ZINC000217714665 BF On-Demand Unstable DRD3 15 47 C=CCCCNC(=O)/C=C\c1ccccc1 ZINC000217714665 BF On-Demand Unstable HDAC8 48 39 C=CCCCNC(=O)/C=C\c1ccccc1 ZINC000217714665 BF On-Demand Unstable F3 19 46 C=CCCCNC(=O)/C=C\c1ccccc1 ZINC000217714665 BF On-Demand Unstable MMP2 23 63 C=CCCCNC(=O)/C=C\c1ccccc1 ZINC000217714665 BF On-Demand Unstable HDAC1 24 50 C=CCCCNC(=O)/C=C\c1ccccc1 ZINC000217714665 BF On-Demand Unstable HDAC2 23 50 C=CCCCNC(=O)/C=C\c1ccccc1 ZINC000217714665 BF On-Demand Unstable HDAC3 19 50 C=CCCCNC(=O)/C=C\c1ccccc1 ZINC000217714665 BF On-Demand Unstable HDAC4 16 50 C=CCCCNC(=O)/C=C\c1ccccc1 ZINC000217714665 BF On-Demand Unstable HDAC6 35 54 C=CCCCNC(=O)/C=C\c1ccccc1 ZINC000217714665 BF On-Demand Unstable MMP9 20 63 C=CCCCNC(=O)/C=C\c1ccccc1 ZINC000217714665 BF On-Demand Unstable HDAC9 39 50 C=CCCCNC(=O)/C=C\c1ccccc1 ZINC000217714665 BF On-Demand Unstable HDAC7 47 50 O=C(/C=C\c1ccc2c(c1)OCO2)NCC1CC(O)C1 ZINC000217714675 CD On-Demand Unstable HDAC1 0 51 O=C(/C=C\c1ccc2c(c1)OCO2)NCC1CC(O)C1 ZINC000217714675 CD On-Demand Unstable DYRK1A 18 40 O=C(/C=C\c1ccc2c(c1)OCO2)NCC1CC(O)C1 ZINC000217714675 CD On-Demand Unstable CLK1 31 40 O=C(/C=C\c1ccc2c(c1)OCO2)NCC1CC(O)C1 ZINC000217714675 CD On-Demand Unstable CLK3 30 40 O=C(/C=C\c1ccc2c(c1)OCO2)NCC1CC(O)C1 ZINC000217714675 CD On-Demand Unstable DYRK2 63 40 CCOc1ccc(C(=O)NC[C@](C)(O)CSC)cc1OC ZINC000217714677 DD On-Demand Unstable MT-ND1 24 40 COC(=O)[C@@H](O)CNC(=O)c1ccc(OC)c([N+](=O)[O-])c1 ZINC000217714684 CB On-Demand Unstable TAAR1 18 41 O=C(/C=C/c1ccccc1)N1CC(N2C(=O)CCC2=O)C1 ZINC000217714704 CD In-Stock Unstable GPR183 0 41 CN(C[C@H]1CCCN1C)c1cccc(Cl)c1CBr ZINC000217714713 EH For-Sale Unstable CHRNA10 71 43 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217714724 EI For-Sale Unstable TAAR1 22 48 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217714724 EI For-Sale Unstable IMDH_CRYPV 35 45 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217714724 EI For-Sale Unstable BLM 0 44 O=C(O)/C=C\c1cccc(C(=O)NCCn2cccn2)c1 ZINC000217714725 CD For-Sale Unstable DRD4 42 32 O=C(O)/C=C\c1cccc(C(=O)NCCn2cccn2)c1 ZINC000217714725 CD For-Sale Unstable HDAC8 28 40 O=C(O)/C=C\c1cccc(C(=O)NCCn2cccn2)c1 ZINC000217714725 CD For-Sale Unstable HDAC6 15 40 C=CCCCNC(=O)/C=C/c1ccccc1 ZINC000217714753 BF On-Demand Unstable DRD3 15 47 C=CCCCNC(=O)/C=C/c1ccccc1 ZINC000217714753 BF On-Demand Unstable HDAC8 48 39 C=CCCCNC(=O)/C=C/c1ccccc1 ZINC000217714753 BF On-Demand Unstable F3 19 46 C=CCCCNC(=O)/C=C/c1ccccc1 ZINC000217714753 BF On-Demand Unstable MMP2 23 63 C=CCCCNC(=O)/C=C/c1ccccc1 ZINC000217714753 BF On-Demand Unstable HDAC1 24 50 C=CCCCNC(=O)/C=C/c1ccccc1 ZINC000217714753 BF On-Demand Unstable HDAC2 23 50 C=CCCCNC(=O)/C=C/c1ccccc1 ZINC000217714753 BF On-Demand Unstable HDAC3 19 50 C=CCCCNC(=O)/C=C/c1ccccc1 ZINC000217714753 BF On-Demand Unstable HDAC4 16 50 C=CCCCNC(=O)/C=C/c1ccccc1 ZINC000217714753 BF On-Demand Unstable HDAC6 35 54 C=CCCCNC(=O)/C=C/c1ccccc1 ZINC000217714753 BF On-Demand Unstable MMP9 20 63 C=CCCCNC(=O)/C=C/c1ccccc1 ZINC000217714753 BF On-Demand Unstable HDAC9 39 50 C=CCCCNC(=O)/C=C/c1ccccc1 ZINC000217714753 BF On-Demand Unstable HDAC7 47 50 COC(=O)[C@H](O)CNC(=O)c1ccc(OC)c([N+](=O)[O-])c1 ZINC000217714763 CB On-Demand Unstable TAAR1 18 41 Cc1cccc(CC(=O)N2CC(N3C(=O)CCC3=O)C2)c1 ZINC000217714817 CC In-Stock Unstable GPR183 0 42 Cc1cc(CBr)cnc1N(C)C[C@@H]1CCCN1C ZINC000217714821 DF For-Sale Unstable CHRNA10 55 35 COc1ccccc1/C=C/NC(=O)Nc1ccc([N+](=O)[O-])cc1OC ZINC000217714825 EG For-Sale Unstable EPHX1 0 56 COc1ccccc1/C=C/NC(=O)Nc1ccc([N+](=O)[O-])cc1OC ZINC000217714825 EG For-Sale Unstable CACNA1D 45 32 COc1ccccc1/C=C/NC(=O)Nc1ccc([N+](=O)[O-])cc1OC ZINC000217714825 EG For-Sale Unstable KCNMA1 25 56 O=C(O)/C=C\c1ccc(C(=O)NCCn2ccnc2)s1 ZINC000217714842 CD For-Sale Unstable TBXAS1 61 59 CCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217714874 EE In-Stock Unstable CA2 26 46 CCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217714874 EE In-Stock Unstable TBXA2R 55 44 CCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217714874 EE In-Stock Unstable CA1 22 41 CCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217714874 EE In-Stock Unstable CA7 19 40 CCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217714874 EE In-Stock Unstable CA4 20 46 CCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217714874 EE In-Stock Unstable ALOX15 50 36 CCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217714874 EE In-Stock Unstable AKR1C3 19 57 CCNc1ccc(S(=O)(=O)NCCc2ccccc2)cc1C(=O)O ZINC000217714874 EE In-Stock Unstable A6YCJ1_9METZ 15 40 Cc1cc(CBr)cnc1N(C)C[C@H]1CCCN1C ZINC000217714902 DF For-Sale Unstable CHRNA10 55 35 COc1ccccc1/C=C/NC(=O)Nc1ccc([N+](=O)[O-])cc1 ZINC000217714935 DG For-Sale Unstable NMBR 56 36 COc1ccccc1/C=C/NC(=O)Nc1ccc([N+](=O)[O-])cc1 ZINC000217714935 DG For-Sale Unstable KCNMA1 19 41 O=C(COc1ccccc1)N1CC(N2C(=O)CCC2=O)C1 ZINC000217714937 CC In-Stock Unstable COLA 136 41 O=C(COc1ccccc1)N1CC(N2C(=O)CCC2=O)C1 ZINC000217714937 CC In-Stock Unstable CPT1A 112 41 O=C(COc1ccccc1)N1CC(N2C(=O)CCC2=O)C1 ZINC000217714937 CC In-Stock Unstable CPT2 47 38 O=C(COc1ccccc1)N1CC(N2C(=O)CCC2=O)C1 ZINC000217714937 CC In-Stock Unstable GPR183 0 43 CSC[C@@](C)(O)CNC(=O)CCc1c[nH]c2ccccc12 ZINC000217714982 DE On-Demand Unstable ACHE 29 44 CSC[C@@](C)(O)CNC(=O)CCc1c[nH]c2ccccc12 ZINC000217714982 DE On-Demand Unstable EDNRA 0 40 CSC[C@@](C)(O)CNC(=O)CCc1c[nH]c2ccccc12 ZINC000217714982 DE On-Demand Unstable MC4R 37 41 CSC[C@@](C)(O)CNC(=O)CCc1c[nH]c2ccccc12 ZINC000217714982 DE On-Demand Unstable TACR2 0 40 CSC[C@@](C)(O)CNC(=O)CCc1c[nH]c2ccccc12 ZINC000217714982 DE On-Demand Unstable CCKAR 68 40 CSC[C@@](C)(O)CNC(=O)CCc1c[nH]c2ccccc12 ZINC000217714982 DE On-Demand Unstable BRS3 22 41 CSC[C@@](C)(O)CNC(=O)CCc1c[nH]c2ccccc12 ZINC000217714982 DE On-Demand Unstable NMBR 62 32 CSC[C@@](C)(O)CNC(=O)CCc1c[nH]c2ccccc12 ZINC000217714982 DE On-Demand Unstable MC5R 35 43 CSC[C@@](C)(O)CNC(=O)CCc1c[nH]c2ccccc12 ZINC000217714982 DE On-Demand Unstable MMP14 54 35 CSC[C@@](C)(O)CNC(=O)CCc1c[nH]c2ccccc12 ZINC000217714982 DE On-Demand Unstable GRPR 50 31 CSC[C@@](C)(O)CNC(=O)CCc1c[nH]c2ccccc12 ZINC000217714982 DE On-Demand Unstable CCKBR 50 38 CSC[C@@](C)(O)CNC(=O)CCc1c[nH]c2ccccc12 ZINC000217714982 DE On-Demand Unstable GHSR 52 38 COc1ccccc1/C=C/NC(=O)Nc1cccc([N+](=O)[O-])c1 ZINC000217715033 DG For-Sale Unstable CACNA1C 42 34 COc1ccccc1/C=C/NC(=O)Nc1cccc([N+](=O)[O-])c1 ZINC000217715033 DG For-Sale Unstable PPIA 25 46 COc1ccccc1/C=C/NC(=O)Nc1cccc([N+](=O)[O-])c1 ZINC000217715033 DG For-Sale Unstable CACNA1D 72 34 COc1ccccc1/C=C/NC(=O)Nc1cccc([N+](=O)[O-])c1 ZINC000217715033 DG For-Sale Unstable KCNMA1 19 41 COc1ccccc1/C=C/NC(=O)Nc1cccc([N+](=O)[O-])c1 ZINC000217715033 DG For-Sale Unstable TAAR1 25 52 COc1ccccc1/C=C/NC(=O)Nc1cccc([N+](=O)[O-])c1 ZINC000217715033 DG For-Sale Unstable ABCG2 17 41 COc1ccccc1/C=C/NC(=O)Nc1cccc([N+](=O)[O-])c1 ZINC000217715033 DG For-Sale Unstable DDX3X 0 51 COc1ccccc1/C=C/NC(=O)Nc1cccc([N+](=O)[O-])c1 ZINC000217715033 DG For-Sale Unstable TRPM8 0 50 COc1ccccc1/C=C/NC(=O)Nc1cccc([N+](=O)[O-])c1 ZINC000217715033 DG For-Sale Unstable KCNK3 46 41 COc1ccccc1/C=C/NC(=O)Nc1cccc([N+](=O)[O-])c1 ZINC000217715033 DG For-Sale Unstable KCNK9 51 41 O=C(Cc1ccc(F)cc1)N1CC(N2C(=O)CCC2=O)C1 ZINC000217715042 CC In-Stock Unstable MLNR 26 40 CSC[C@](C)(O)CNC(=O)CCc1c[nH]c2ccccc12 ZINC000217715063 DE On-Demand Unstable ACHE 29 44 CSC[C@](C)(O)CNC(=O)CCc1c[nH]c2ccccc12 ZINC000217715063 DE On-Demand Unstable EDNRA 0 40 CSC[C@](C)(O)CNC(=O)CCc1c[nH]c2ccccc12 ZINC000217715063 DE On-Demand Unstable MC4R 37 41 CSC[C@](C)(O)CNC(=O)CCc1c[nH]c2ccccc12 ZINC000217715063 DE On-Demand Unstable TACR2 0 40 CSC[C@](C)(O)CNC(=O)CCc1c[nH]c2ccccc12 ZINC000217715063 DE On-Demand Unstable CCKAR 68 40 CSC[C@](C)(O)CNC(=O)CCc1c[nH]c2ccccc12 ZINC000217715063 DE On-Demand Unstable BRS3 22 41 CSC[C@](C)(O)CNC(=O)CCc1c[nH]c2ccccc12 ZINC000217715063 DE On-Demand Unstable NMBR 62 32 CSC[C@](C)(O)CNC(=O)CCc1c[nH]c2ccccc12 ZINC000217715063 DE On-Demand Unstable MC5R 35 43 CSC[C@](C)(O)CNC(=O)CCc1c[nH]c2ccccc12 ZINC000217715063 DE On-Demand Unstable MMP14 54 35 CSC[C@](C)(O)CNC(=O)CCc1c[nH]c2ccccc12 ZINC000217715063 DE On-Demand Unstable GRPR 50 31 CSC[C@](C)(O)CNC(=O)CCc1c[nH]c2ccccc12 ZINC000217715063 DE On-Demand Unstable CCKBR 50 38 CSC[C@](C)(O)CNC(=O)CCc1c[nH]c2ccccc12 ZINC000217715063 DE On-Demand Unstable GHSR 52 38 C[C@@H]1CCCCN1S(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217715123 DE For-Sale Unstable AKR1C3 55 43 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1OC ZINC000217715133 JI In-Stock Unstable AKR1B1 22 48 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1OC ZINC000217715133 JI In-Stock Unstable CYP1B1 76 44 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1OC ZINC000217715133 JI In-Stock Unstable CYP1A1 56 44 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1OC ZINC000217715133 JI In-Stock Unstable CYP1A2 47 52 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1OC ZINC000217715133 JI In-Stock Unstable ABCG2 0 43 COc1ccccc1/C=C/NC(=O)Nc1cc([N+](=O)[O-])ccc1Cl ZINC000217715137 EI For-Sale Unstable KCNMA1 22 46 CSc1ncccc1C(=O)N1CCC[C@@H]1c1nc(C)n[nH]1 ZINC000217715147 DE In-Stock Unstable COLA 78 42 CSc1ncccc1C(=O)N1CCC[C@@H]1c1nc(C)n[nH]1 ZINC000217715147 DE In-Stock Unstable CPT1A 72 42 CSc1ncccc1C(=O)N1CCC[C@@H]1c1nc(C)n[nH]1 ZINC000217715147 DE In-Stock Unstable HCRTR2 42 38 CC[C@@H](Oc1ccccc1)C(=O)NC[C@@](C)(O)CSC ZINC000217715175 CE For-Sale Unstable PDS 67 38 C[C@H]1CCCCN1S(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217715207 DE For-Sale Unstable AKR1C3 55 43 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1OC ZINC000217715218 JI In-Stock Unstable AKR1B1 22 48 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1OC ZINC000217715218 JI In-Stock Unstable CYP1B1 76 44 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1OC ZINC000217715218 JI In-Stock Unstable CYP1A1 56 44 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1OC ZINC000217715218 JI In-Stock Unstable CYP1A2 47 52 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1OC ZINC000217715218 JI In-Stock Unstable ABCG2 0 43 CSc1ncccc1C(=O)N1CCC[C@H]1c1nc(C)n[nH]1 ZINC000217715229 DE In-Stock Unstable COLA 78 42 CSc1ncccc1C(=O)N1CCC[C@H]1c1nc(C)n[nH]1 ZINC000217715229 DE In-Stock Unstable CPT1A 72 42 CSc1ncccc1C(=O)N1CCC[C@H]1c1nc(C)n[nH]1 ZINC000217715229 DE In-Stock Unstable HCRTR2 42 38 COc1ccccc1/C=C/NC(=O)NCCCCl ZINC000217715244 CF For-Sale Unstable DRD2 17 45 COc1ccccc1/C=C/NC(=O)NCCCCl ZINC000217715244 CF For-Sale Unstable DRD3 30 45 COc1ccccc1/C=C/NC(=O)NCCCCl ZINC000217715244 CF For-Sale Unstable MTNR1B 18 42 COc1ccccc1/C=C/NC(=O)NCCCCl ZINC000217715244 CF For-Sale Unstable ACAT 0 43 CC[C@H](Oc1ccccc1)C(=O)NC[C@@](C)(O)CSC ZINC000217715249 CE For-Sale Unstable PDS 67 38 NC(=O)COc1ccc(CN[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217715281 CC For-Sale Unstable HRH3 17 40 C[C@H]1CC[C@@](C)(CC(=O)O)C1(C)C ZINC000217715291 AF In-Stock Unstable CACNA2D1 54 39 O=C(O)[C@@H]1CCCN(C[C@@H]2CCCCO2)C1 ZINC000217715306 BD On-Demand Unstable SLC6A1 135 43 CC[C@@H](Oc1ccccc1)C(=O)NC[C@](C)(O)CSC ZINC000217715326 CE For-Sale Unstable PDS 67 38 COc1ccccc1/C=C/NC(=O)NCCCl ZINC000217715358 CE For-Sale Unstable DRD3 19 42 COc1ccccc1/C=C/NC(=O)NCCCl ZINC000217715358 CE For-Sale Unstable CYP1B1 19 40 COc1ccccc1/C=C/NC(=O)NCCCl ZINC000217715358 CE For-Sale Unstable TLR4 19 45 NC(=O)COc1ccc(CN[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217715367 CC For-Sale Unstable HRH3 17 40 O=C1Cc2cc(C(=O)NCC(F)F)ccc2N1 ZINC000217715375 BD For-Sale Unstable HDAC9 25 48 COC(=O)c1ccc(C(=O)N2CC(N3C(=O)CCC3=O)C2)cc1 ZINC000217715387 DC In-Stock Unstable AVPR1A 25 45 COC(=O)c1ccc(C(=O)N2CC(N3C(=O)CCC3=O)C2)cc1 ZINC000217715387 DC In-Stock Unstable L3MBTL1 0 40 COC(=O)c1ccc(C(=O)N2CC(N3C(=O)CCC3=O)C2)cc1 ZINC000217715387 DC In-Stock Unstable L3MBTL3 44 40 COC(=O)c1ccc(C(=O)N2CC(N3C(=O)CCC3=O)C2)cc1 ZINC000217715387 DC In-Stock Unstable GPR183 0 41 CC[C@H](Oc1ccccc1)C(=O)NC[C@](C)(O)CSC ZINC000217715403 CE For-Sale Unstable PDS 67 38 O=C(O)[C@@H]1CCCN(C[C@@H]2COc3ccccc3O2)C1 ZINC000217715422 CD On-Demand Unstable HTR1A 15 54 O=C(O)[C@@H]1CCCN(C[C@@H]2COc3ccccc3O2)C1 ZINC000217715422 CD On-Demand Unstable SLC6A1 189 49 O=C(O)[C@@H]1CCCN(C[C@@H]2COc3ccccc3O2)C1 ZINC000217715422 CD On-Demand Unstable ADRA2B 27 48 O=C(O)[C@@H]1CCCN(C[C@@H]2COc3ccccc3O2)C1 ZINC000217715422 CD On-Demand Unstable ADRA2C 16 45 CN(C)CCNS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217715457 CC For-Sale Unstable AKR1C3 26 45 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccc(F)cc2)CC1 ZINC000217715468 FG For-Sale Unstable HTR1A 24 42 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccc(F)cc2)CC1 ZINC000217715468 FG For-Sale Unstable DRD2 19 40 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccc(F)cc2)CC1 ZINC000217715468 FG For-Sale Unstable DRD3 27 40 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccc(F)cc2)CC1 ZINC000217715468 FG For-Sale Unstable SSTR1 21 40 COC(=O)C[C@H](CC(C)C)c1c(O)c2ccccc2oc1=O ZINC000217715469 DG In-Stock Unstable CYP2C9 17 40 COC(=O)C[C@H](CC(C)C)c1c(O)c2ccccc2oc1=O ZINC000217715469 DG In-Stock Unstable NQO1 50 38 C[C@H]1CCC[C@@H](C)N1CC(=O)NCCc1nc2cc(Cl)ccc2[nH]1 ZINC000217715476 EG In-Stock Unstable F9 29 52 C[C@H]1CCC[C@@H](C)N1CC(=O)NCCc1nc2cc(Cl)ccc2[nH]1 ZINC000217715476 EG In-Stock Unstable CYSP_TRYCR 0 50 C[C@H]1CCC[C@@H](C)N1CC(=O)NCCc1nc2cc(Cl)ccc2[nH]1 ZINC000217715476 EG In-Stock Unstable PYGL 42 37 CCOC(=O)c1ccc(NC(=O)COc2ccccc2C(=O)O)cc1 ZINC000217715485 EF In-Stock Unstable PPIA 18 50 CCOC(=O)c1ccc(NC(=O)COc2ccccc2C(=O)O)cc1 ZINC000217715485 EF In-Stock Unstable CETP 0 46 CCOC(=O)c1ccc(NC(=O)COc2ccccc2C(=O)O)cc1 ZINC000217715485 EF In-Stock Unstable GUAB 0 44 CCOC(=O)c1ccc(NC(=O)COc2ccccc2C(=O)O)cc1 ZINC000217715485 EF In-Stock Unstable ACR 59 40 CCOC(=O)c1ccc(NC(=O)COc2ccccc2C(=O)O)cc1 ZINC000217715485 EF In-Stock Unstable AKR1C2 45 38 CCOC(=O)c1ccc(NC(=O)COc2ccccc2C(=O)O)cc1 ZINC000217715485 EF In-Stock Unstable HCN1 42 31 CCOC(=O)c1ccc(NC(=O)COc2ccccc2C(=O)O)cc1 ZINC000217715485 EF In-Stock Unstable NOD2 18 43 CCOC(=O)c1ccc(NC(=O)COc2ccccc2C(=O)O)cc1 ZINC000217715485 EF In-Stock Unstable SENP1 0 40 CCOC(=O)c1ccc(NC(=O)COc2ccccc2C(=O)O)cc1 ZINC000217715485 EF In-Stock Unstable SLC27A1 18 44 CCOC(=O)c1ccc(NC(=O)COc2ccccc2C(=O)O)cc1 ZINC000217715485 EF In-Stock Unstable KCNK3 33 40 CCOC(=O)c1ccc(NC(=O)COc2ccccc2C(=O)O)cc1 ZINC000217715485 EF In-Stock Unstable KCNK9 29 40 CCOc1ccc(CC(=O)N2CC(N3C(=O)CCC3=O)C2)cc1 ZINC000217715499 DC In-Stock Unstable AVPR1A 20 46 COC(=O)C[C@@H](CC(C)C)c1c(O)c2ccccc2oc1=O ZINC000217715550 DG In-Stock Unstable CYP2C9 17 40 COC(=O)C[C@@H](CC(C)C)c1c(O)c2ccccc2oc1=O ZINC000217715550 DG In-Stock Unstable NQO1 50 38 COc1ccccc1/C=C/NC(=O)Nc1ccccc1O ZINC000217715589 CG For-Sale Unstable TLR4 15 44 NS(=O)(=O)c1ccc(NC(=O)COc2ccccc2C(=O)O)cc1 ZINC000217715595 FD In-Stock Unstable CA2 163 58 NS(=O)(=O)c1ccc(NC(=O)COc2ccccc2C(=O)O)cc1 ZINC000217715595 FD In-Stock Unstable PPIA 31 48 NS(=O)(=O)c1ccc(NC(=O)COc2ccccc2C(=O)O)cc1 ZINC000217715595 FD In-Stock Unstable LTA4H 23 44 NS(=O)(=O)c1ccc(NC(=O)COc2ccccc2C(=O)O)cc1 ZINC000217715595 FD In-Stock Unstable CA1 148 58 NS(=O)(=O)c1ccc(NC(=O)COc2ccccc2C(=O)O)cc1 ZINC000217715595 FD In-Stock Unstable CA7 71 58 NS(=O)(=O)c1ccc(NC(=O)COc2ccccc2C(=O)O)cc1 ZINC000217715595 FD In-Stock Unstable CETP 0 43 NS(=O)(=O)c1ccc(NC(=O)COc2ccccc2C(=O)O)cc1 ZINC000217715595 FD In-Stock Unstable CA13 22 46 NS(=O)(=O)c1ccc(NC(=O)COc2ccccc2C(=O)O)cc1 ZINC000217715595 FD In-Stock Unstable CA5B 77 58 NS(=O)(=O)c1ccc(NC(=O)COc2ccccc2C(=O)O)cc1 ZINC000217715595 FD In-Stock Unstable CA4 135 55 NS(=O)(=O)c1ccc(NC(=O)COc2ccccc2C(=O)O)cc1 ZINC000217715595 FD In-Stock Unstable CA5A 83 58 NS(=O)(=O)c1ccc(NC(=O)COc2ccccc2C(=O)O)cc1 ZINC000217715595 FD In-Stock Unstable CA14 50 58 NS(=O)(=O)c1ccc(NC(=O)COc2ccccc2C(=O)O)cc1 ZINC000217715595 FD In-Stock Unstable CA12 103 58 NS(=O)(=O)c1ccc(NC(=O)COc2ccccc2C(=O)O)cc1 ZINC000217715595 FD In-Stock Unstable CA9 113 51 NS(=O)(=O)c1ccc(NC(=O)COc2ccccc2C(=O)O)cc1 ZINC000217715595 FD In-Stock Unstable F13A1 60 35 NS(=O)(=O)c1ccc(NC(=O)COc2ccccc2C(=O)O)cc1 ZINC000217715595 FD In-Stock Unstable UREA_CANEN 27 45 NS(=O)(=O)c1ccc(NC(=O)COc2ccccc2C(=O)O)cc1 ZINC000217715595 FD In-Stock Unstable NCE103 56 46 NS(=O)(=O)c1ccc(NC(=O)COc2ccccc2C(=O)O)cc1 ZINC000217715595 FD In-Stock Unstable MTCA1 56 52 NS(=O)(=O)c1ccc(NC(=O)COc2ccccc2C(=O)O)cc1 ZINC000217715595 FD In-Stock Unstable P96878_MYCTU 71 52 NS(=O)(=O)c1ccc(NC(=O)COc2ccccc2C(=O)O)cc1 ZINC000217715595 FD In-Stock Unstable NAMPT 17 50 O=C1CCC(=O)N1C1CN(C(=O)C23CC4CC(CC(C4)C2)C3)C1 ZINC000217715603 DD In-Stock Unstable GRM1 18 42 COc1cc([C@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)ccc1O ZINC000217715656 KH In-Stock Unstable CYP1B1 53 39 COc1cc([C@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)ccc1O ZINC000217715656 KH In-Stock Unstable CYP1A1 44 39 COc1cc([C@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)ccc1O ZINC000217715656 KH In-Stock Unstable RORC 54 38 COC(=O)[C@@H](O)CNC(=O)CNC(=O)c1cccc(F)c1 ZINC000217715664 CB On-Demand Unstable DRD4 40 31 COC(=O)[C@@H](O)CNC(=O)CNC(=O)c1cccc(F)c1 ZINC000217715664 CB On-Demand Unstable CCR2 57 45 COC(=O)[C@@H](O)CNC(=O)CNC(=O)c1cccc(F)c1 ZINC000217715664 CB On-Demand Unstable KCNK3 19 40 CCOc1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217715700 DH For-Sale Unstable TSHR 42 33 CCOc1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217715700 DH For-Sale Unstable CA1 43 44 CCOc1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217715700 DH For-Sale Unstable PRNP 15 52 CCOc1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217715700 DH For-Sale Unstable MTNR1B 20 45 CCOc1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217715700 DH For-Sale Unstable CA12 16 44 CCOc1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217715700 DH For-Sale Unstable PDGFRA 46 38 CCOc1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217715700 DH For-Sale Unstable CA9 16 44 CCOc1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217715700 DH For-Sale Unstable KCNK3 42 40 CCOc1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217715700 DH For-Sale Unstable KCNK9 32 40 O=C(c1ccccc1C(F)(F)F)N1CC(N2C(=O)CCC2=O)C1 ZINC000217715706 ED In-Stock Unstable P2RX7 47 41 O=C(c1ccccc1C(F)(F)F)N1CC(N2C(=O)CCC2=O)C1 ZINC000217715706 ED In-Stock Unstable RBP4 69 39 O=C(c1ccccc1C(F)(F)F)N1CC(N2C(=O)CCC2=O)C1 ZINC000217715706 ED In-Stock Unstable SCD1 17 41 COc1ccc(C(=O)O)c(OCC(=O)Nc2ccccc2Cl)c1 ZINC000217715718 EG In-Stock Unstable PYGL 22 43 COc1ccc(C(=O)O)c(OCC(=O)Nc2ccccc2Cl)c1 ZINC000217715718 EG In-Stock Unstable PYGM 26 47 COc1ccc(C(=O)O)c(OCC(=O)Nc2ccccc2Cl)c1 ZINC000217715718 EG In-Stock Unstable HCAR2 23 48 COc1ccc(C(=O)O)c(OCC(=O)Nc2ccccc2Cl)c1 ZINC000217715718 EG In-Stock Unstable EPHB3 43 44 COc1ccc(C(=O)O)c(OCC(=O)Nc2ccccc2Cl)c1 ZINC000217715718 EG In-Stock Unstable AKR1C3 39 47 COc1ccc(C(=O)O)c(OCC(=O)Nc2ccccc2Cl)c1 ZINC000217715718 EG In-Stock Unstable AKR1C2 87 47 COc1ccc(C(=O)O)c(OCC(=O)Nc2ccccc2Cl)c1 ZINC000217715718 EG In-Stock Unstable ISPD 0 41 COc1cc([C@@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)ccc1O ZINC000217715724 KH In-Stock Unstable CYP1B1 53 39 COc1cc([C@@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)ccc1O ZINC000217715724 KH In-Stock Unstable CYP1A1 44 39 COc1cc([C@@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)ccc1O ZINC000217715724 KH In-Stock Unstable RORC 54 38 COC(=O)[C@H](O)CNC(=O)CNC(=O)c1cccc(F)c1 ZINC000217715764 CB On-Demand Unstable DRD4 40 31 COC(=O)[C@H](O)CNC(=O)CNC(=O)c1cccc(F)c1 ZINC000217715764 CB On-Demand Unstable CCR2 57 45 COC(=O)[C@H](O)CNC(=O)CNC(=O)c1cccc(F)c1 ZINC000217715764 CB On-Demand Unstable KCNK3 19 40 COc1ccc(/C=C\C(=O)NCC2CC(O)C2)cc1F ZINC000217715774 CD For-Sale Unstable MMP2 0 43 COc1ccc(/C=C\C(=O)NCC2CC(O)C2)cc1F ZINC000217715774 CD For-Sale Unstable HDAC1 0 41 COc1ccc(/C=C\C(=O)NCC2CC(O)C2)cc1F ZINC000217715774 CD For-Sale Unstable TUBB1 47 45 CCCCOC(=O)c1ccccc1NC(=O)N/C=C/c1ccccc1OC ZINC000217715800 FI For-Sale Unstable ACAT 0 42 CCC[C@@H](C)NS(=O)(=O)c1ccc(/C=C\C(=O)O)cc1Cl ZINC000217715809 EF For-Sale Unstable NR0B2 0 40 COc1ccc(CC(=O)N2CC(N3C(=O)CCC3=O)C2)cc1OC ZINC000217715826 EC In-Stock Unstable OPRK1 0 40 COc1ccc(CC(=O)N2CC(N3C(=O)CCC3=O)C2)cc1OC ZINC000217715826 EC In-Stock Unstable P2RX7 0 42 O=C(Cn1cnc2sccc2c1=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217715837 GD In-Stock Unstable CHRNA4 27 43 CN(C[C@@H]1CCCN1C)c1ccc(CBr)cc1Cl ZINC000217715838 EH For-Sale Unstable CHRNA10 69 43 CCOC(=O)c1ccc(NC(=O)COc2cc(OC)ccc2C(=O)O)cc1 ZINC000217715862 FF In-Stock Unstable SENP1 0 42 O=C(/C=C\c1ccccc1F)NCC1CC(O)C1 ZINC000217715880 BD On-Demand Unstable KCNQ2 41 39 O=C(Nc1cc(Cl)c(O)c(Cl)c1)c1cc(Cl)ccc1I ZINC000217715883 IK On-Demand Anodyne KCNMA1 28 49 O=C(Nc1cc(Cl)c(O)c(Cl)c1)c1cc(Cl)ccc1I ZINC000217715883 IK On-Demand Anodyne Q25615_ONCVO 94 50 CCC[C@H](C)NS(=O)(=O)c1ccc(/C=C\C(=O)O)cc1Cl ZINC000217715903 EF For-Sale Unstable NR0B2 0 40 COc1ccccc1/C=C/NC(=O)Nc1ccc(C(C)=O)cc1 ZINC000217715918 DH For-Sale Unstable PRNP 16 41 COc1ccccc1/C=C/NC(=O)Nc1ccc(C(C)=O)cc1 ZINC000217715918 DH For-Sale Unstable ACR 26 42 COc1ccccc1/C=C/NC(=O)Nc1ccc(C(C)=O)cc1 ZINC000217715918 DH For-Sale Unstable PDGFRA 43 35 CN(C[C@H]1CCCN1C)c1ccc(CBr)cc1Cl ZINC000217715928 EH For-Sale Unstable CHRNA10 69 43 CSC[C@@](C)(O)CNC(=O)Cc1cccc(C(F)(F)F)c1 ZINC000217715952 DE On-Demand Unstable CSNK1D 27 43 CSC[C@@](C)(O)CNC(=O)Cc1cccc(C(F)(F)F)c1 ZINC000217715952 DE On-Demand Unstable CCR2 59 36 CSC[C@@](C)(O)CNC(=O)Cc1cccc(C(F)(F)F)c1 ZINC000217715952 DE On-Demand Unstable PDS 43 38 COc1ccc(C(=O)O)c(OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217715976 GD In-Stock Unstable CA2 134 59 COc1ccc(C(=O)O)c(OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217715976 GD In-Stock Unstable LTA4H 19 42 COc1ccc(C(=O)O)c(OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217715976 GD In-Stock Unstable CA1 125 59 COc1ccc(C(=O)O)c(OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217715976 GD In-Stock Unstable CA7 66 46 COc1ccc(C(=O)O)c(OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217715976 GD In-Stock Unstable CETP 0 40 COc1ccc(C(=O)O)c(OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217715976 GD In-Stock Unstable CA13 15 40 COc1ccc(C(=O)O)c(OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217715976 GD In-Stock Unstable CA5B 56 46 COc1ccc(C(=O)O)c(OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217715976 GD In-Stock Unstable CA4 107 47 COc1ccc(C(=O)O)c(OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217715976 GD In-Stock Unstable CA5A 64 46 COc1ccc(C(=O)O)c(OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217715976 GD In-Stock Unstable CA14 58 40 COc1ccc(C(=O)O)c(OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217715976 GD In-Stock Unstable MTNR1A 21 45 COc1ccc(C(=O)O)c(OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217715976 GD In-Stock Unstable MTNR1B 25 45 COc1ccc(C(=O)O)c(OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217715976 GD In-Stock Unstable CA12 88 59 COc1ccc(C(=O)O)c(OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217715976 GD In-Stock Unstable CA9 103 59 COc1ccc(C(=O)O)c(OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217715976 GD In-Stock Unstable AKR1C3 23 43 COc1ccc(C(=O)O)c(OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217715976 GD In-Stock Unstable UREA_CANEN 28 47 COc1ccc(C(=O)O)c(OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217715976 GD In-Stock Unstable NCE103 46 37 COc1ccc(C(=O)O)c(OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217715976 GD In-Stock Unstable AKR1C2 60 43 COc1ccc(C(=O)O)c(OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217715976 GD In-Stock Unstable MTCA1 56 52 COc1ccc(C(=O)O)c(OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217715976 GD In-Stock Unstable P96878_MYCTU 68 52 O=C(O)/C=C\c1cccc(S(=O)(=O)Nc2cn[nH]c2)c1 ZINC000217715991 CD For-Sale Anodyne HDAC8 23 59 O=C(O)/C=C\c1cccc(S(=O)(=O)Nc2cn[nH]c2)c1 ZINC000217715991 CD For-Sale Anodyne HDAC1 0 59 O=C(c1ccc(-c2ccsc2)cc1)N1CC(N2C(=O)CCC2=O)C1 ZINC000217716029 EE In-Stock Unstable AVPR1A 21 40 O=C(Nc1cc(Cl)c(O)c(Cl)c1)c1ccc(F)cc1I ZINC000217716030 IJ On-Demand Anodyne GRM4 25 46 O=C(Nc1cc(Cl)c(O)c(Cl)c1)c1ccc(F)cc1I ZINC000217716030 IJ On-Demand Anodyne Q25615_ONCVO 87 51 CSC[C@](C)(O)CNC(=O)Cc1cccc(C(F)(F)F)c1 ZINC000217716032 DE On-Demand Unstable CSNK1D 27 43 CSC[C@](C)(O)CNC(=O)Cc1cccc(C(F)(F)F)c1 ZINC000217716032 DE On-Demand Unstable CCR2 59 36 CSC[C@](C)(O)CNC(=O)Cc1cccc(C(F)(F)F)c1 ZINC000217716032 DE On-Demand Unstable PDS 43 38 Cc1cc(CBr)ccc1N(C)C[C@@H]1CCCN1C ZINC000217716038 DG For-Sale Unstable CHRNA10 67 38 COc1ccccc1/C=C/NC(=O)Nc1cccc(C(C)=O)c1 ZINC000217716039 DH For-Sale Unstable CYP1B1 20 41 COc1ccccc1/C=C/NC(=O)Nc1cccc(C(C)=O)c1 ZINC000217716039 DH For-Sale Unstable CCR3 23 43 COc1ccccc1/C=C/NC(=O)Nc1cccc(C(C)=O)c1 ZINC000217716039 DH For-Sale Unstable CYP1A1 17 41 COc1ccccc1/C=C/NC(=O)Nc1cccc(C(C)=O)c1 ZINC000217716039 DH For-Sale Unstable AKR1C3 31 45 COc1ccccc1/C=C/NC(=O)Nc1cccc(C(C)=O)c1 ZINC000217716039 DH For-Sale Unstable KCNK3 110 46 COc1ccccc1/C=C/NC(=O)Nc1cccc(C(C)=O)c1 ZINC000217716039 DH For-Sale Unstable KCNK9 79 45 CC(C)Cc1cc(C(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)[nH]n1 ZINC000217716062 EE In-Stock Unstable CHRNA4 30 47 COc1ccc(C(=O)O)c(OCC(=O)Nc2cccc(C(C)=O)c2)c1 ZINC000217716080 EF In-Stock Unstable CETP 0 42 COc1ccc(C(=O)O)c(OCC(=O)Nc2cccc(C(C)=O)c2)c1 ZINC000217716080 EF In-Stock Unstable MTNR1A 37 41 COc1ccc(C(=O)O)c(OCC(=O)Nc2cccc(C(C)=O)c2)c1 ZINC000217716080 EF In-Stock Unstable MTNR1B 38 45 COc1ccc(C(=O)O)c(OCC(=O)Nc2cccc(C(C)=O)c2)c1 ZINC000217716080 EF In-Stock Unstable MCHR1 17 42 COc1ccc(C(=O)O)c(OCC(=O)Nc2cccc(C(C)=O)c2)c1 ZINC000217716080 EF In-Stock Unstable HIF1A 25 47 COc1ccc(C(=O)O)c(OCC(=O)Nc2cccc(C(C)=O)c2)c1 ZINC000217716080 EF In-Stock Unstable AKR1C3 62 48 COc1ccc(C(=O)O)c(OCC(=O)Nc2cccc(C(C)=O)c2)c1 ZINC000217716080 EF In-Stock Unstable AKR1C2 78 48 COc1ccc(C(=O)O)c(OCC(=O)Nc2cccc(C(C)=O)c2)c1 ZINC000217716080 EF In-Stock Unstable ISPD 0 40 COc1ccc(C(=O)O)c(OCC(=O)Nc2cccc(C(C)=O)c2)c1 ZINC000217716080 EF In-Stock Unstable KCNK3 67 41 COc1ccc(C(=O)O)c(OCC(=O)Nc2cccc(C(C)=O)c2)c1 ZINC000217716080 EF In-Stock Unstable KCNK9 65 37 COc1ccc(C(=O)O)c(OCC(=O)Nc2cccc(C(C)=O)c2)c1 ZINC000217716080 EF In-Stock Unstable PARP10 0 41 Cc1cc(CBr)ccc1N(C)C[C@H]1CCCN1C ZINC000217716130 DG For-Sale Unstable CHRNA10 67 38 COc1ccc(C(=O)NCC(F)F)c(F)c1 ZINC000217716155 BD On-Demand Unstable MTNR1A 54 42 COc1ccc(C(=O)NCC(F)F)c(F)c1 ZINC000217716155 BD On-Demand Unstable MTNR1B 48 42 COc1ccc(C(=O)NCC(F)F)c(F)c1 ZINC000217716155 BD On-Demand Unstable U38 0 40 COc1ccc(C(=O)NCC(F)F)c(F)c1 ZINC000217716155 BD On-Demand Unstable AKR1C2 52 38 COc1ccc(C(=O)NCC(F)F)c(F)c1 ZINC000217716155 BD On-Demand Unstable GPR35 20 41 CSC[C@@](C)(O)CNC(=O)/C=C/c1cccc(Cl)c1 ZINC000217716157 CF On-Demand Unstable TUBA4A 0 42 CN(Cc1cccs1)C(=O)c1cccc(Br)n1 ZINC000217716160 DG On-Demand Unstable HCAR3 15 40 CCOc1cc([C@@H]2CC(=O)Oc3c(C(C)=O)c(O)c4c(C)cc(=O)oc4c32)ccc1O ZINC000217716163 HH In-Stock Unstable NTBBF1.1 0 40 O=C(COc1ccc(Cl)cc1C(=O)O)Nc1ccccc1Cl ZINC000217716212 EH In-Stock Unstable PTGER1 52 42 O=C(COc1ccc(Cl)cc1C(=O)O)Nc1ccccc1Cl ZINC000217716212 EH In-Stock Unstable CXCL8 24 40 O=C(COc1ccc(Cl)cc1C(=O)O)Nc1ccccc1Cl ZINC000217716212 EH In-Stock Unstable CETP 0 44 O=C(COc1ccc(Cl)cc1C(=O)O)Nc1ccccc1Cl ZINC000217716212 EH In-Stock Unstable HCAR2 28 42 O=C(COc1ccc(Cl)cc1C(=O)O)Nc1ccccc1Cl ZINC000217716212 EH In-Stock Unstable FABH 0 41 O=C(COc1ccc(Cl)cc1C(=O)O)Nc1ccccc1Cl ZINC000217716212 EH In-Stock Unstable PTGDR2 36 46 O=C(COc1ccc(Cl)cc1C(=O)O)Nc1ccccc1Cl ZINC000217716212 EH In-Stock Unstable FEN1 0 40 O=C(COc1ccc(Cl)cc1C(=O)O)Nc1ccccc1Cl ZINC000217716212 EH In-Stock Unstable ACPS 0 41 O=C(COc1ccc(Cl)cc1C(=O)O)Nc1ccccc1Cl ZINC000217716212 EH In-Stock Unstable EPHB3 44 35 O=C(COc1ccc(Cl)cc1C(=O)O)Nc1ccccc1Cl ZINC000217716212 EH In-Stock Unstable AKR1C3 21 42 O=C(COc1ccc(Cl)cc1C(=O)O)Nc1ccccc1Cl ZINC000217716212 EH In-Stock Unstable AKR1C2 53 45 CN(C[C@@H]1CCCN1C)c1ccccc1CBr ZINC000217716235 CG For-Sale Unstable CHRNA10 73 47 CSC[C@](C)(O)CNC(=O)/C=C/c1cccc(Cl)c1 ZINC000217716238 CF On-Demand Unstable TUBA4A 0 42 CCOc1cc([C@H]2CC(=O)Oc3c(C(C)=O)c(O)c4c(C)cc(=O)oc4c32)ccc1O ZINC000217716248 HH In-Stock Unstable NTBBF1.1 0 40 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable ACE 37 45 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable PPARA 17 42 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable MME 94 44 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable LTA4H 19 40 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable ANPEP 79 34 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable CASP3 18 42 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable BMP1 23 40 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable KLK3 79 37 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable CTSB 71 51 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable PAPA1_CARPA 80 42 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable CYSP_TRYCR 59 40 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable CTSK 44 50 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable CTSL 49 43 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable CPA1 45 35 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable CAPNS1 73 42 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable MMP3 15 45 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable HDAC2 19 40 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable MMP11 50 32 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable CTSS 21 50 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable CAPN1 98 46 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable CASP1 25 45 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable CAPN2 143 48 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable CASP6 23 40 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable CASP9 29 40 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable TGM2 24 40 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable LAP3 60 42 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable TPSAB1 40 36 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable FPR1 47 33 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable NPR 96 48 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable AMP1_PLAFQ 46 36 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable NAAA 30 41 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable PSMB5 38 40 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable NPFFR1 44 31 CO[C@@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716277 CD For-Sale Unstable PDS 44 33 CN(C[C@H]1CCCN1C)c1ccccc1CBr ZINC000217716319 CG For-Sale Unstable CHRNA10 73 47 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable ACE 37 45 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable PPARA 17 42 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable MME 94 44 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable LTA4H 19 40 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable ANPEP 79 34 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable CASP3 18 42 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable BMP1 23 40 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable KLK3 79 37 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable CTSB 71 51 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable PAPA1_CARPA 80 42 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable CYSP_TRYCR 59 40 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable CTSK 44 50 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable CTSL 49 43 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable CPA1 45 35 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable CAPNS1 73 42 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable MMP3 15 45 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable HDAC2 19 40 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable MMP11 50 32 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable CTSS 21 50 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable CAPN1 98 46 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable CASP1 25 45 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable CAPN2 143 48 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable CASP6 23 40 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable CASP9 29 40 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable TGM2 24 40 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable LAP3 60 42 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable TPSAB1 40 36 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable FPR1 47 33 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable NPR 96 48 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable AMP1_PLAFQ 46 36 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable NAAA 30 41 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable PSMB5 38 40 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable NPFFR1 44 31 CO[C@H](CCNC(=O)OCc1ccccc1)C(=O)O ZINC000217716345 CD For-Sale Unstable PDS 44 33 CCCN(CC)C(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217716350 CF For-Sale Unstable ACKR3 44 34 COC(=O)C[C@H](C1=Cc2ccccc2OC1)c1c(O)c2ccccc2oc1=O ZINC000217716357 GH In-Stock Unstable NQO1 35 47 CCOC(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716367 GG In-Stock Unstable HTR2A 19 41 CCOC(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716367 GG In-Stock Unstable P2RY12 22 43 CCOC(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716367 GG In-Stock Unstable PTGER1 50 43 CCOC(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716367 GG In-Stock Unstable CETP 0 45 CCOC(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716367 GG In-Stock Unstable COLA 69 38 CCOC(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716367 GG In-Stock Unstable CPT1A 65 38 CCOC(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716367 GG In-Stock Unstable CPT2 48 37 CCOC(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716367 GG In-Stock Unstable F3 62 34 CCOC(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716367 GG In-Stock Unstable ACR 55 38 CCOC(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716367 GG In-Stock Unstable CPT1B 47 35 CCOC(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716367 GG In-Stock Unstable AGPAT2 80 41 CCOC(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716367 GG In-Stock Unstable MCHR2 35 42 CCOC(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716367 GG In-Stock Unstable AKR1C3 23 40 CCOC(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716367 GG In-Stock Unstable AKR1C2 45 35 CCOC(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716367 GG In-Stock Unstable SENP1 0 43 CCOC(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716367 GG In-Stock Unstable PSBA 0 47 CC[C@@H](CCO)NCCCc1ccccc1 ZINC000217716398 BE For-Sale Unstable SIGMAR1 16 56 CC[C@@H](CCO)NCCCc1ccccc1 ZINC000217716398 BE For-Sale Unstable AMP1_PLAFQ 26 40 COc1ccccc1/C=C/NC(=O)Nc1ccc(C)cc1C ZINC000217716405 CI For-Sale Unstable EPHX1 0 43 COc1ccccc1/C=C/NC(=O)Nc1ccc(C)cc1C ZINC000217716405 CI For-Sale Unstable KCNK3 37 40 COc1ccccc1/C=C/NC(=O)Nc1ccc(C)cc1C ZINC000217716405 CI For-Sale Unstable KCNK9 41 40 CCC(C)(C)NC(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217716426 CF For-Sale Unstable COLA 0 42 CCC(C)(C)NC(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217716426 CF For-Sale Unstable CPT1A 17 42 COC(=O)C[C@@H](C1=Cc2ccccc2OC1)c1c(O)c2ccccc2oc1=O ZINC000217716451 GH In-Stock Unstable NQO1 35 47 CN(C[C@@H]1CCCN1C)c1ccc(CBr)cn1 ZINC000217716453 CF For-Sale Unstable CHRNA10 62 38 Cc1cc(C(=O)Nc2ccc(Cl)nc2)c(C)nn1 ZINC000217716454 CE On-Demand Unstable JUN 22 42 Cc1cc(C(=O)Nc2ccc(Cl)nc2)c(C)nn1 ZINC000217716454 CE On-Demand Unstable CSF1R 23 40 Cc1cc(C(=O)Nc2ccc(Cl)nc2)c(C)nn1 ZINC000217716454 CE On-Demand Unstable SHH 41 38 CC[C@H](C(=O)O)N(C)C/C=C\c1ccccc1 ZINC000217716472 BE On-Demand Unstable NA 0 40 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716477 GD In-Stock Unstable CA2 110 45 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716477 GD In-Stock Unstable PTGER1 39 40 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716477 GD In-Stock Unstable CA1 95 45 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716477 GD In-Stock Unstable CA7 53 47 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716477 GD In-Stock Unstable CETP 0 42 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716477 GD In-Stock Unstable COLA 66 37 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716477 GD In-Stock Unstable CPT1A 61 37 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716477 GD In-Stock Unstable CPT2 46 35 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716477 GD In-Stock Unstable CA5B 62 47 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716477 GD In-Stock Unstable CA4 100 43 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716477 GD In-Stock Unstable CA5A 71 47 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716477 GD In-Stock Unstable CA14 43 39 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716477 GD In-Stock Unstable CA12 73 50 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716477 GD In-Stock Unstable CPT1B 48 34 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716477 GD In-Stock Unstable AGPAT2 47 33 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716477 GD In-Stock Unstable CA9 84 45 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716477 GD In-Stock Unstable PTGDR2 32 43 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716477 GD In-Stock Unstable UREA_CANEN 26 42 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716477 GD In-Stock Unstable NCE103 44 39 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716477 GD In-Stock Unstable MTCA1 39 40 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)cc1 ZINC000217716477 GD In-Stock Unstable P96878_MYCTU 57 50 CC[C@H](CCO)NCCCc1ccccc1 ZINC000217716487 BE For-Sale Unstable SIGMAR1 16 56 CC[C@H](CCO)NCCCc1ccccc1 ZINC000217716487 BE For-Sale Unstable AMP1_PLAFQ 26 40 COc1ccccc1/C=C/NC(=O)Nc1cc(C)ccc1OC ZINC000217716517 DH For-Sale Unstable CYP1B1 18 41 COc1ccccc1/C=C/NC(=O)Nc1cc(C)ccc1OC ZINC000217716517 DH For-Sale Unstable CYP1A1 15 41 COc1ccccc1/C=C/NC(=O)Nc1cc(C)ccc1OC ZINC000217716517 DH For-Sale Unstable KCNK3 38 40 COc1ccccc1/C=C/NC(=O)Nc1cc(C)ccc1OC ZINC000217716517 DH For-Sale Unstable KCNK9 41 40 CN(C[C@H]1CCCN1C)c1ccc(CBr)cn1 ZINC000217716538 CF For-Sale Unstable CHRNA10 62 38 CC[C@@H](C(=O)O)N(C)C/C=C\c1ccccc1 ZINC000217716554 BE On-Demand Unstable NA 0 40 CC(=O)c1cccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)c1 ZINC000217716564 EG In-Stock Unstable HTR2A 20 42 CC(=O)c1cccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)c1 ZINC000217716564 EG In-Stock Unstable PTGER1 51 46 CC(=O)c1cccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)c1 ZINC000217716564 EG In-Stock Unstable CETP 0 42 CC(=O)c1cccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)c1 ZINC000217716564 EG In-Stock Unstable COLA 62 38 CC(=O)c1cccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)c1 ZINC000217716564 EG In-Stock Unstable CPT1A 59 38 CC(=O)c1cccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)c1 ZINC000217716564 EG In-Stock Unstable CPT2 44 34 CC(=O)c1cccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)c1 ZINC000217716564 EG In-Stock Unstable GUAB 0 41 CC(=O)c1cccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)c1 ZINC000217716564 EG In-Stock Unstable CPT1B 40 37 CC(=O)c1cccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)c1 ZINC000217716564 EG In-Stock Unstable AGPAT2 41 34 CC(=O)c1cccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)c1 ZINC000217716564 EG In-Stock Unstable MCHR2 35 43 CC(=O)c1cccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)c1 ZINC000217716564 EG In-Stock Unstable AKR1C3 57 48 CC(=O)c1cccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)c1 ZINC000217716564 EG In-Stock Unstable AKR1C2 50 39 CC(=O)c1cccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)c1 ZINC000217716564 EG In-Stock Unstable IMDH_CRYPV 15 41 CC(=O)c1cccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)c1 ZINC000217716564 EG In-Stock Unstable PSBA 0 41 CC(=O)c1cccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)c1 ZINC000217716564 EG In-Stock Unstable KCNK3 67 40 CC(=O)c1cccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)c1 ZINC000217716564 EG In-Stock Unstable KCNK9 63 38 CC(=O)c1cccc(NC(=O)COc2ccc(Cl)cc2C(=O)O)c1 ZINC000217716564 EG In-Stock Unstable PARP10 0 41 O=C(Cc1c(F)cccc1Cl)N1CC(N2C(=O)CCC2=O)C1 ZINC000217716573 DD In-Stock Unstable P2RX7 18 43 CN1CCN(C(=O)c2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217716584 CD For-Sale Unstable INHA 19 41 CN1CCN(C(=O)c2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217716584 CD For-Sale Unstable HRH4 28 40 CCOc1ccccc1NC(=O)N1[C@H]2CC[C@H]1CC(SC)C2 ZINC000217716593 DH In-Stock Unstable HCN1 49 36 CCOc1ccccc1NC(=O)N1[C@H]2CC[C@H]1CC(SC)C2 ZINC000217716593 DH In-Stock Unstable HCN4 43 36 CN(C[C@@H]1CCCN1C)c1ccc(CBr)cc1F ZINC000217716630 DG For-Sale Unstable HRH1 29 41 CN(C[C@@H]1CCCN1C)c1ccc(CBr)cc1F ZINC000217716630 DG For-Sale Unstable CHRNA10 71 43 COc1ccccc1/C=C/NC(=O)Nc1cccc(C)c1 ZINC000217716641 CH For-Sale Unstable KIT 22 41 COc1ccccc1/C=C/NC(=O)Nc1cccc(C)c1 ZINC000217716641 CH For-Sale Unstable CCKAR 25 47 COc1ccccc1/C=C/NC(=O)Nc1cccc(C)c1 ZINC000217716641 CH For-Sale Unstable KDR 22 43 COc1ccccc1/C=C/NC(=O)Nc1cccc(C)c1 ZINC000217716641 CH For-Sale Unstable PDGFRA 23 43 COc1ccccc1/C=C/NC(=O)Nc1cccc(C)c1 ZINC000217716641 CH For-Sale Unstable KCNK3 113 51 COc1ccccc1/C=C/NC(=O)Nc1cccc(C)c1 ZINC000217716641 CH For-Sale Unstable KCNK9 89 51 CN1CCN(C(=O)c2cc(/C=C\C(=O)O)ccc2F)CC1 ZINC000217716685 CD For-Sale Unstable HRH4 30 46 CN1CCN(C(=O)c2cc(/C=C\C(=O)O)ccc2F)CC1 ZINC000217716685 CD For-Sale Unstable PARP1 52 40 CN(C[C@H]1CCCN1C)c1ccc(CBr)cc1F ZINC000217716721 DG For-Sale Unstable HRH1 29 41 CN(C[C@H]1CCCN1C)c1ccc(CBr)cc1F ZINC000217716721 DG For-Sale Unstable CHRNA10 71 43 O=C(/C=C\c1ccc([N+](=O)[O-])cc1)NCC1CC(O)C1 ZINC000217716732 CD On-Demand Unstable HDAC8 0 49 O=C(/C=C\c1ccc([N+](=O)[O-])cc1)NCC1CC(O)C1 ZINC000217716732 CD On-Demand Unstable HDAC1 0 49 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217716765 FK For-Sale Unstable GUAB 0 45 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217716765 FK For-Sale Unstable RAF1 40 48 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217716765 FK For-Sale Unstable Q8MMZ8_EIMTE 63 48 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217716765 FK For-Sale Unstable BRAF 15 40 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217716765 FK For-Sale Unstable PTPA 0 43 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217716765 FK For-Sale Unstable IMDH_CRYPV 42 48 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217716765 FK For-Sale Unstable BLM 0 43 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217716765 FK For-Sale Unstable KCNK3 43 37 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217716765 FK For-Sale Unstable KCNK9 41 37 COC(=O)C[C@H](c1cc2cc3c(cc2[nH]c1=O)OCO3)c1c(O)c2ccccc2oc1=O ZINC000217716778 IF In-Stock Unstable NQO1 26 44 Cc1nn(C)c(N(C)C[C@@H]2CCCN2C)c1CBr ZINC000217716812 DE For-Sale Unstable CHRNA10 45 31 CN1CCN(C(=O)c2ccc(/C=C\C(=O)O)cc2F)CC1 ZINC000217716822 CD For-Sale Unstable HRH4 28 43 CCOC(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716827 GH In-Stock Unstable DHODH 22 40 CCOC(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716827 GH In-Stock Unstable P2RY12 29 42 CCOC(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716827 GH In-Stock Unstable PPIA 17 47 CCOC(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716827 GH In-Stock Unstable LTA4H 42 39 CCOC(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716827 GH In-Stock Unstable NPR1 40 30 CCOC(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716827 GH In-Stock Unstable ADORA2A 0 45 CCOC(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716827 GH In-Stock Unstable ADORA2B 41 36 CCOC(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716827 GH In-Stock Unstable CA1 36 44 CCOC(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716827 GH In-Stock Unstable CETP 0 43 CCOC(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716827 GH In-Stock Unstable GUAB 0 46 CCOC(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716827 GH In-Stock Unstable PRNP 34 49 CCOC(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716827 GH In-Stock Unstable F3 44 34 CCOC(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716827 GH In-Stock Unstable ACR 73 39 CCOC(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716827 GH In-Stock Unstable CA9 15 48 CCOC(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716827 GH In-Stock Unstable DHOD 0 41 CCOC(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716827 GH In-Stock Unstable AKR1C2 42 35 CCOC(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716827 GH In-Stock Unstable NOD1 16 40 CCOC(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716827 GH In-Stock Unstable NOD2 33 40 CCCN(CC)CCNCCCc1ccccc1 ZINC000217716828 BF For-Sale Unstable SIGMAR1 25 59 CCCN(CC)CCNCCCc1ccccc1 ZINC000217716828 BF For-Sale Unstable S1PR2 21 40 COC(=O)C[C@@H](c1cc2cc3c(cc2[nH]c1=O)OCO3)c1c(O)c2ccccc2oc1=O ZINC000217716838 IF In-Stock Unstable NQO1 26 44 Cc1nn(C)c(N(C)C[C@H]2CCCN2C)c1CBr ZINC000217716896 DE For-Sale Unstable CHRNA10 45 31 NS(=O)(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716914 HE In-Stock Unstable CA2 151 53 NS(=O)(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716914 HE In-Stock Unstable PPIA 16 45 NS(=O)(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716914 HE In-Stock Unstable LTA4H 35 45 NS(=O)(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716914 HE In-Stock Unstable CA1 141 53 NS(=O)(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716914 HE In-Stock Unstable CA7 66 53 NS(=O)(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716914 HE In-Stock Unstable CETP 0 42 NS(=O)(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716914 HE In-Stock Unstable GUAB 0 48 NS(=O)(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716914 HE In-Stock Unstable CA13 17 43 NS(=O)(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716914 HE In-Stock Unstable CA5B 74 53 NS(=O)(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716914 HE In-Stock Unstable CA4 124 48 NS(=O)(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716914 HE In-Stock Unstable CA5A 80 53 NS(=O)(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716914 HE In-Stock Unstable CA14 49 53 NS(=O)(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716914 HE In-Stock Unstable CA12 99 53 NS(=O)(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716914 HE In-Stock Unstable CA9 113 51 NS(=O)(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716914 HE In-Stock Unstable F13A1 47 36 NS(=O)(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716914 HE In-Stock Unstable NCE103 49 43 NS(=O)(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716914 HE In-Stock Unstable MTCA1 55 51 NS(=O)(=O)c1ccc(NC(=O)COc2cc3ccccc3cc2C(=O)O)cc1 ZINC000217716914 HE In-Stock Unstable P96878_MYCTU 70 51 CCCN(CC)CCNCc1ccc(O)c(OCC)c1 ZINC000217716922 CF On-Demand Unstable SLC6A13 0 42 CSc1cccc(NC(=O)c2ccc(/C=C\C(=O)O)s2)c1 ZINC000217716995 DH For-Sale Unstable KCNK3 80 36 CSc1cccc(NC(=O)c2ccc(/C=C\C(=O)O)s2)c1 ZINC000217716995 DH For-Sale Unstable KCNK9 42 36 COc1ccccc1/C=C/NC(=O)Nc1ccc(N)c(Cl)c1 ZINC000217716999 DH For-Sale Unstable GRM4 19 41 C[C@@H](N[C@@H]1CCN2CCC[C@@H]12)c1ccc(Br)cc1 ZINC000217717011 DG For-Sale Unstable SDH1 0 43 O=C(Nc1ccc(Cl)cc1Cl)N(Cc1cccs1)Cc1cccs1 ZINC000217717012 GK On-Demand Unstable CA5B 30 48 O=C(Nc1ccc(Cl)cc1Cl)N(Cc1cccs1)Cc1cccs1 ZINC000217717012 GK On-Demand Unstable CA5A 35 48 O=C(COc1c(C(=O)O)ccc2ccccc12)Nc1ccccc1Cl ZINC000217717055 FI In-Stock Unstable HCAR2 33 40 O=C(COc1c(C(=O)O)ccc2ccccc12)Nc1ccccc1Cl ZINC000217717055 FI In-Stock Unstable EPHB3 47 34 O=C(Nc1ccc(Cl)c(Cl)c1)N1CC(N2C(=O)CCC2=O)C1 ZINC000217717056 EE In-Stock Unstable P95276_MYCTO 0 42 O=C(Nc1ccc(Cl)c(Cl)c1)N1CC(N2C(=O)CCC2=O)C1 ZINC000217717056 EE In-Stock Unstable PPX1 0 41 C[C@H](N[C@@H]1CCN2CCC[C@@H]12)c1ccc(Br)cc1 ZINC000217717092 DG For-Sale Unstable SDH1 0 43 O=C(Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1)c1ccccc1I ZINC000217717139 II On-Demand Bother GRM4 16 41 O=C(Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1)c1ccccc1I ZINC000217717139 II On-Demand Bother Q25615_ONCVO 52 37 O=C(Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1)c1ccccc1I ZINC000217717139 II On-Demand Bother KCNK3 56 41 O=C(Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1)c1ccccc1I ZINC000217717139 II On-Demand Bother KCNK9 51 40 CCCCOc1ccc(NC(=O)N2CC(N3C(=O)CCC3=O)C2)cc1 ZINC000217717168 EE In-Stock Unstable AVPR1A 21 47 CCCCOc1ccc(NC(=O)N2CC(N3C(=O)CCC3=O)C2)cc1 ZINC000217717168 EE In-Stock Unstable MMP13 25 41 CCCCOc1ccc(NC(=O)N2CC(N3C(=O)CCC3=O)C2)cc1 ZINC000217717168 EE In-Stock Unstable MMP3 18 41 CCCCOc1ccc(NC(=O)N2CC(N3C(=O)CCC3=O)C2)cc1 ZINC000217717168 EE In-Stock Unstable PLA2G4B 61 33 CCCCOc1ccc(NC(=O)N2CC(N3C(=O)CCC3=O)C2)cc1 ZINC000217717168 EE In-Stock Unstable FAAH 21 43 C[C@@H](N[C@H]1CCN2CCC[C@@H]12)c1ccc(Br)cc1 ZINC000217717173 DG For-Sale Unstable SDH1 0 43 CN(C[C@@H]1CCCN1C)c1ncc(CBr)cn1 ZINC000217717195 CD For-Sale Unstable CHRNA10 61 38 COC(=O)c1ccccc1S(=O)(=O)NC[C@@H]1CCCO1 ZINC000217717199 CC On-Demand Unstable OXTR 24 41 COC(=O)c1ccccc1S(=O)(=O)NC[C@@H]1CCCO1 ZINC000217717199 CC On-Demand Unstable NPY2R 48 36 COC(=O)c1ccccc1S(=O)(=O)NC[C@@H]1CCCO1 ZINC000217717199 CC On-Demand Unstable TNK2 54 38 CCOC(=O)c1ccc(NC(=O)COc2c(C(=O)O)ccc3ccccc23)cc1 ZINC000217717202 GH In-Stock Unstable P2RY12 23 40 CCOC(=O)c1ccc(NC(=O)COc2c(C(=O)O)ccc3ccccc23)cc1 ZINC000217717202 GH In-Stock Unstable GUAB 0 44 CCOC(=O)c1ccc(NC(=O)COc2c(C(=O)O)ccc3ccccc23)cc1 ZINC000217717202 GH In-Stock Unstable ACR 59 39 CCOC(=O)c1ccc(NC(=O)COc2c(C(=O)O)ccc3ccccc23)cc1 ZINC000217717202 GH In-Stock Unstable NOD2 17 40 COc1ccccc1/C=C/NC(=O)Nc1cccc(Cl)c1 ZINC000217717251 DI For-Sale Unstable PPIA 28 43 COc1ccccc1/C=C/NC(=O)Nc1cccc(Cl)c1 ZINC000217717251 DI For-Sale Unstable PTGER3 22 42 COc1ccccc1/C=C/NC(=O)Nc1cccc(Cl)c1 ZINC000217717251 DI For-Sale Unstable CPT1A 43 30 COc1ccccc1/C=C/NC(=O)Nc1cccc(Cl)c1 ZINC000217717251 DI For-Sale Unstable GRM4 18 40 COc1ccccc1/C=C/NC(=O)Nc1cccc(Cl)c1 ZINC000217717251 DI For-Sale Unstable PDGFRA 17 44 COc1ccccc1/C=C/NC(=O)Nc1cccc(Cl)c1 ZINC000217717251 DI For-Sale Unstable IMPDH2 0 42 COc1ccccc1/C=C/NC(=O)Nc1cccc(Cl)c1 ZINC000217717251 DI For-Sale Unstable IMDH_CRYPV 22 40 COc1ccccc1/C=C/NC(=O)Nc1cccc(Cl)c1 ZINC000217717251 DI For-Sale Unstable KCNK3 77 44 COc1ccccc1/C=C/NC(=O)Nc1cccc(Cl)c1 ZINC000217717251 DI For-Sale Unstable KCNK9 69 44 COc1ccccc1/C=C/NC(=O)Nc1cccc(Cl)c1 ZINC000217717251 DI For-Sale Unstable CYSP_PLAFA 43 36 Cc1ccccc1C(=O)Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1 ZINC000217717263 DI On-Demand Unstable GRM4 21 42 Cc1ccccc1C(=O)Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1 ZINC000217717263 DI On-Demand Unstable MTTP 64 38 Cc1ccccc1C(=O)Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1 ZINC000217717263 DI On-Demand Unstable KCNMA1 25 47 Cc1ccccc1C(=O)Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1 ZINC000217717263 DI On-Demand Unstable SHH 29 41 Cc1ccccc1C(=O)Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1 ZINC000217717263 DI On-Demand Unstable SMO 22 41 Cc1ccccc1C(=O)Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1 ZINC000217717263 DI On-Demand Unstable KCNK3 59 48 Cc1ccccc1C(=O)Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1 ZINC000217717263 DI On-Demand Unstable KCNK9 70 45 O=C(O)[C@H]1CCCN1P(=O)(O)O ZINC000217717267 AB For-Sale Unstable ACE 29 45 O=C(O)[C@H]1CCCN1P(=O)(O)O ZINC000217717267 AB For-Sale Unstable MVD 15 48 O=C(NCc1ccc(Cl)cc1)N1CC(N2C(=O)CCC2=O)C1 ZINC000217717269 DD In-Stock Unstable SLC6A1 27 44 C[C@H](N[C@H]1CCN2CCC[C@@H]12)c1ccc(Br)cc1 ZINC000217717275 DG For-Sale Unstable SDH1 0 43 CN(C[C@H]1CCCN1C)c1ncc(CBr)cn1 ZINC000217717286 CD For-Sale Unstable CHRNA10 61 38 COC(=O)c1ccccc1S(=O)(=O)NC[C@H]1CCCO1 ZINC000217717294 CC On-Demand Unstable OXTR 24 41 COC(=O)c1ccccc1S(=O)(=O)NC[C@H]1CCCO1 ZINC000217717294 CC On-Demand Unstable NPY2R 48 36 COC(=O)c1ccccc1S(=O)(=O)NC[C@H]1CCCO1 ZINC000217717294 CC On-Demand Unstable TNK2 54 38 NS(=O)(=O)c1ccc(NC(=O)COc2c(C(=O)O)ccc3ccccc23)cc1 ZINC000217717318 HE In-Stock Unstable CA2 134 53 NS(=O)(=O)c1ccc(NC(=O)COc2c(C(=O)O)ccc3ccccc23)cc1 ZINC000217717318 HE In-Stock Unstable CA1 123 53 NS(=O)(=O)c1ccc(NC(=O)COc2c(C(=O)O)ccc3ccccc23)cc1 ZINC000217717318 HE In-Stock Unstable CA7 55 53 NS(=O)(=O)c1ccc(NC(=O)COc2c(C(=O)O)ccc3ccccc23)cc1 ZINC000217717318 HE In-Stock Unstable GUAB 0 45 NS(=O)(=O)c1ccc(NC(=O)COc2c(C(=O)O)ccc3ccccc23)cc1 ZINC000217717318 HE In-Stock Unstable CA13 17 43 NS(=O)(=O)c1ccc(NC(=O)COc2c(C(=O)O)ccc3ccccc23)cc1 ZINC000217717318 HE In-Stock Unstable CA5B 73 53 NS(=O)(=O)c1ccc(NC(=O)COc2c(C(=O)O)ccc3ccccc23)cc1 ZINC000217717318 HE In-Stock Unstable CA4 110 48 NS(=O)(=O)c1ccc(NC(=O)COc2c(C(=O)O)ccc3ccccc23)cc1 ZINC000217717318 HE In-Stock Unstable CA5A 83 53 NS(=O)(=O)c1ccc(NC(=O)COc2c(C(=O)O)ccc3ccccc23)cc1 ZINC000217717318 HE In-Stock Unstable CA14 45 53 NS(=O)(=O)c1ccc(NC(=O)COc2c(C(=O)O)ccc3ccccc23)cc1 ZINC000217717318 HE In-Stock Unstable CA12 86 53 NS(=O)(=O)c1ccc(NC(=O)COc2c(C(=O)O)ccc3ccccc23)cc1 ZINC000217717318 HE In-Stock Unstable CA9 93 47 NS(=O)(=O)c1ccc(NC(=O)COc2c(C(=O)O)ccc3ccccc23)cc1 ZINC000217717318 HE In-Stock Unstable F13A1 43 37 NS(=O)(=O)c1ccc(NC(=O)COc2c(C(=O)O)ccc3ccccc23)cc1 ZINC000217717318 HE In-Stock Unstable NCE103 38 43 NS(=O)(=O)c1ccc(NC(=O)COc2c(C(=O)O)ccc3ccccc23)cc1 ZINC000217717318 HE In-Stock Unstable MT-CO2 45 33 NS(=O)(=O)c1ccc(NC(=O)COc2c(C(=O)O)ccc3ccccc23)cc1 ZINC000217717318 HE In-Stock Unstable MTCA1 53 48 NS(=O)(=O)c1ccc(NC(=O)COc2c(C(=O)O)ccc3ccccc23)cc1 ZINC000217717318 HE In-Stock Unstable P96878_MYCTU 66 48 O=C(O)[C@@H]1CCCN1P(=O)(O)O ZINC000217717328 AB For-Sale Unstable ACE 29 45 O=C(O)[C@@H]1CCCN1P(=O)(O)O ZINC000217717328 AB For-Sale Unstable MVD 15 48 O=C(Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1)c1cccc(Cl)c1Cl ZINC000217717356 GK On-Demand Bother GRM4 31 40 O=C(Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1)c1cccc(Cl)c1Cl ZINC000217717356 GK On-Demand Bother TAAR1 45 40 O=C(Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1)c1cccc(Cl)c1Cl ZINC000217717356 GK On-Demand Bother NR2E3 62 33 O=C(Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1)c1cccc(Cl)c1Cl ZINC000217717356 GK On-Demand Bother SHH 38 40 O=C(Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1)c1cccc(Cl)c1Cl ZINC000217717356 GK On-Demand Bother SMO 29 41 O=C(Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1)c1cccc(Cl)c1Cl ZINC000217717356 GK On-Demand Bother KCNK3 53 44 O=C(Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1)c1cccc(Cl)c1Cl ZINC000217717356 GK On-Demand Bother KCNK9 46 39 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)cc1 ZINC000217717366 DI For-Sale Unstable EPHX1 0 40 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)cc1 ZINC000217717366 DI For-Sale Unstable HTR2A 20 41 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)cc1 ZINC000217717366 DI For-Sale Unstable KDR 21 40 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)cc1 ZINC000217717366 DI For-Sale Unstable PDGFRA 42 40 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)cc1 ZINC000217717366 DI For-Sale Unstable CYSP_PLAFA 38 41 CN1CCC[C@H](NC(=O)c2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217717376 CD For-Sale Unstable SLC6A5 33 42 COc1ccc(CNC(=O)N2CC(N3C(=O)CCC3=O)C2)cc1OC ZINC000217717378 EC In-Stock Unstable TRPV1 0 40 COc1ccc(CNC(=O)N2CC(N3C(=O)CCC3=O)C2)cc1OC ZINC000217717378 EC In-Stock Unstable MT-ND1 24 42 O=C(NCc1ccc(O)cc1)c1cccc(Br)n1 ZINC000217717397 DE On-Demand Unstable Q76353_9HIV1 0 40 O=C(NCc1ccc(O)cc1)c1cccc(Br)n1 ZINC000217717397 DE On-Demand Unstable USP9X 0 41 Cc1cc(N(C)C[C@@H]2CCCN2C)ccc1CBr ZINC000217717405 DG For-Sale Unstable CHRNA10 60 37 CC(=O)c1cccc(NC(=O)COc2c(C(=O)O)ccc3ccccc23)c1 ZINC000217717432 FH In-Stock Unstable CETP 23 40 CC(=O)c1cccc(NC(=O)COc2c(C(=O)O)ccc3ccccc23)c1 ZINC000217717432 FH In-Stock Unstable GUAB 0 43 CC(=O)c1cccc(NC(=O)COc2c(C(=O)O)ccc3ccccc23)c1 ZINC000217717432 FH In-Stock Unstable CAPN2 0 43 CC(=O)c1cccc(NC(=O)COc2c(C(=O)O)ccc3ccccc23)c1 ZINC000217717432 FH In-Stock Unstable AKR1C3 51 48 CC(=O)c1cccc(NC(=O)COc2c(C(=O)O)ccc3ccccc23)c1 ZINC000217717432 FH In-Stock Unstable AKR1C2 45 36 CC(=O)c1cccc(NC(=O)COc2c(C(=O)O)ccc3ccccc23)c1 ZINC000217717432 FH In-Stock Unstable MT-CO1 0 40 CC(=O)c1cccc(NC(=O)COc2c(C(=O)O)ccc3ccccc23)c1 ZINC000217717432 FH In-Stock Unstable MT-CO2 49 40 CC(=O)c1cccc(NC(=O)COc2c(C(=O)O)ccc3ccccc23)c1 ZINC000217717432 FH In-Stock Unstable KCNK3 76 36 CC(=O)c1cccc(NC(=O)COc2c(C(=O)O)ccc3ccccc23)c1 ZINC000217717432 FH In-Stock Unstable KCNK9 62 35 CC(=O)c1cccc(NC(=O)COc2c(C(=O)O)ccc3ccccc23)c1 ZINC000217717432 FH In-Stock Unstable PARP10 0 41 Cc1cc(N(C)C[C@H]2CCCN2C)ccc1CBr ZINC000217717481 DG For-Sale Unstable CHRNA10 60 37 CN1CCC[C@H](NC(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217717494 CD For-Sale Unstable DRD4 18 41 CN1CCC[C@H](NC(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217717494 CD For-Sale Unstable HDAC8 41 44 CN1CCC[C@H](NC(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217717494 CD For-Sale Unstable HDAC1 19 44 CN1CCC[C@H](NC(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217717494 CD For-Sale Unstable HDAC6 23 44 Cc1onc(-c2c(F)cccc2Cl)c1C(=O)Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1 ZINC000217717560 IK On-Demand Unstable GHSR 16 51 Cc1onc(-c2c(F)cccc2Cl)c1C(=O)Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1 ZINC000217717560 IK On-Demand Unstable TYK2 50 35 Cc1onc(-c2c(F)cccc2Cl)c1C(=O)Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1 ZINC000217717560 IK On-Demand Unstable TAAR1 42 39 Cc1onc(-c2c(F)cccc2Cl)c1C(=O)Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1 ZINC000217717560 IK On-Demand Unstable GPBAR1 27 46 O=C(COc1ccc(Br)cc1C(=O)O)NCc1ccccc1 ZINC000217717574 FF In-Stock Unstable PRS 55 40 O=C(COc1ccc(Br)cc1C(=O)O)NCc1ccccc1 ZINC000217717574 FF In-Stock Unstable AMP1_PLAFQ 42 36 O=C(COc1ccc(Br)cc1C(=O)O)NCc1ccccc1 ZINC000217717574 FF In-Stock Unstable NCEH1 28 46 O=C(COc1ccc(Br)cc1C(=O)O)NCc1ccccc1 ZINC000217717574 FF In-Stock Unstable PDS 46 42 COc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccccc2)CC1 ZINC000217717580 FG For-Sale Unstable HTR1A 46 45 COc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccccc2)CC1 ZINC000217717580 FG For-Sale Unstable DRD2 59 45 COc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccccc2)CC1 ZINC000217717580 FG For-Sale Unstable DRD4 65 42 COc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccccc2)CC1 ZINC000217717580 FG For-Sale Unstable ACHE 37 42 COc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccccc2)CC1 ZINC000217717580 FG For-Sale Unstable DRD3 58 42 COc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccccc2)CC1 ZINC000217717580 FG For-Sale Unstable HTR7 35 42 COc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccccc2)CC1 ZINC000217717580 FG For-Sale Unstable SIGMAR1 55 47 COc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccccc2)CC1 ZINC000217717580 FG For-Sale Unstable CCR3 17 41 COc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccccc2)CC1 ZINC000217717580 FG For-Sale Unstable FAAH 29 52 COc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccccc2)CC1 ZINC000217717580 FG For-Sale Unstable MGLL 0 40 COc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccccc2)CC1 ZINC000217717580 FG For-Sale Unstable CCR8 41 45 CC[C@@H](C)[C@@H](C)NC(=O)c1cc(/C=C\C(=O)O)ccc1F ZINC000217717583 CG For-Sale Unstable AKR1C3 40 39 CN(C[C@@H]1CCCN1C)c1cc(Br)ccc1CBr ZINC000217717594 GH For-Sale Unstable CHRNA10 67 39 O=C(N[C@@H]1CCN(C2CC2)C1)c1cccc(Br)n1 ZINC000217717649 DD On-Demand Unstable SLC6A5 20 41 CC[C@H](C)[C@@H](C)NC(=O)c1cc(/C=C\C(=O)O)ccc1F ZINC000217717664 CG For-Sale Unstable AKR1C3 40 39 O=C(Cc1cccc(F)c1)Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1 ZINC000217717670 EH On-Demand Unstable AR 19 59 COC(=O)c1ccccc1S(=O)(=O)N[C@@H]1CCS(=O)(=O)C1 ZINC000217717671 EB On-Demand Unstable CCR8 72 35 O=C(/C=C\c1ccc(F)cc1)NCC1CC(O)C1 ZINC000217717676 BD For-Sale Unstable HDAC4 0 40 O=C(/C=C\c1ccc(F)cc1)NCC1CC(O)C1 ZINC000217717676 BD For-Sale Unstable IMA1 0 43 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)Nc3ccc4[nH]cnc4c3)[C@H]21 ZINC000217717677 JH In-Stock Unstable TSHR 50 34 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)Nc3ccc4[nH]cnc4c3)[C@H]21 ZINC000217717677 JH In-Stock Unstable ENPP1 69 35 CN(C[C@H]1CCCN1C)c1cc(Br)ccc1CBr ZINC000217717685 GH For-Sale Unstable CHRNA10 67 39 COc1ccccc1/C=C/NC(=O)N1CCN(C)CC1 ZINC000217717690 CD For-Sale Unstable HTR1A 17 48 COc1ccccc1/C=C/NC(=O)N1CCN(C)CC1 ZINC000217717690 CD For-Sale Unstable DRD2 15 42 COc1ccccc1/C=C/NC(=O)N1CCN(C)CC1 ZINC000217717690 CD For-Sale Unstable DRD3 22 42 COc1ccccc1/C=C/NC(=O)N1CCN(C)CC1 ZINC000217717690 CD For-Sale Unstable HTR7 16 43 O=C(N[C@H]1CCN(C2CC2)C1)c1cccc(Br)n1 ZINC000217717730 DD On-Demand Unstable SLC6A5 20 41 COC(=O)c1ccccc1S(=O)(=O)N[C@H]1CCS(=O)(=O)C1 ZINC000217717759 EB On-Demand Unstable CCR8 72 35 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)Nc3ccc4[nH]cnc4c3)[C@@H]21 ZINC000217717767 JH In-Stock Unstable TSHR 50 34 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)Nc3ccc4[nH]cnc4c3)[C@@H]21 ZINC000217717767 JH In-Stock Unstable ENPP1 69 35 COc1ccc(CCC(=O)Nc2ccc([N+](=O)[O-])c(C(F)(F)F)c2)cc1OC ZINC000217717781 GI On-Demand Unstable ENPP1 69 33 CN(C[C@@H]1CCCN1C)c1ccc(CBr)cc1 ZINC000217717788 CG For-Sale Unstable CHRNA10 63 39 COc1ccccc1/C=C/NC(=O)N1CCCCC1 ZINC000217717802 CF For-Sale Unstable DRD3 17 40 Cc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217717804 FG In-Stock Unstable ADORA2B 26 43 Cc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217717804 FG In-Stock Unstable PRS 65 37 Cc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217717804 FG In-Stock Unstable CETP 0 56 Cc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217717804 FG In-Stock Unstable AKR1C3 27 43 Cc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217717804 FG In-Stock Unstable AKR1C2 53 40 CN(C[C@H]1CCCN1C)c1ccc(CBr)cc1 ZINC000217717888 CG For-Sale Unstable CHRNA10 63 39 O=C(Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1)c1ccccc1OC(F)F ZINC000217717891 GI On-Demand Bother KCNK3 59 47 O=C(Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1)c1ccccc1OC(F)F ZINC000217717891 GI On-Demand Bother KCNK9 61 47 COc1ccccc1/C=C/NC(=O)NC1CCCCCCCCCCC1 ZINC000217717902 FK For-Sale Unstable FAAH 16 41 COc1ccccc1/C=C/NC(=O)NC1CCCCCCCCCCC1 ZINC000217717902 FK For-Sale Unstable EPHX2 28 46 Cc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1C ZINC000217717907 GH In-Stock Unstable CETP 0 49 Cc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1C ZINC000217717907 GH In-Stock Unstable MCHR1 18 40 Cc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1C ZINC000217717907 GH In-Stock Unstable MCHR2 39 40 Cc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1C ZINC000217717907 GH In-Stock Unstable AKR1C3 25 42 Cc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1C ZINC000217717907 GH In-Stock Unstable AKR1C2 42 42 Cc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1C ZINC000217717907 GH In-Stock Unstable ENPP1 58 37 CCC[C@@H]1CC[C@@H](NCC)[C@@H](CCOc2ccccc2)C1 ZINC000217717964 CJ For-Sale Unstable GRIN2B 15 40 O=C(NCc1cccc(CO)c1)c1cccc(Br)n1 ZINC000217717979 DE On-Demand Unstable MMP13 17 46 O=C(NCc1cccc(CO)c1)c1cccc(Br)n1 ZINC000217717979 DE On-Demand Unstable USP9X 0 50 COc1cc(C(=O)Nc2ccc([N+](=O)[O-])c(C(F)(F)F)c2)cc(OC)c1Br ZINC000217717995 IJ On-Demand Unstable TAAR1 48 46 COc1cc(C(=O)Nc2ccc([N+](=O)[O-])c(C(F)(F)F)c2)cc(OC)c1Br ZINC000217717995 IJ On-Demand Unstable KCNK3 49 35 COc1cc(C(=O)Nc2ccc([N+](=O)[O-])c(C(F)(F)F)c2)cc(OC)c1Br ZINC000217717995 IJ On-Demand Unstable KCNK9 45 35 COc1ccccc1/C=C/NC(=O)NCCN1CCOCC1 ZINC000217718014 DD For-Sale Unstable HTR1A 55 47 COc1ccccc1/C=C/NC(=O)NCCN1CCOCC1 ZINC000217718014 DD For-Sale Unstable DRD2 42 48 COc1ccccc1/C=C/NC(=O)NCCN1CCOCC1 ZINC000217718014 DD For-Sale Unstable CNR1 0 45 COc1ccccc1/C=C/NC(=O)NCCN1CCOCC1 ZINC000217718014 DD For-Sale Unstable DRD4 48 37 COc1ccccc1/C=C/NC(=O)NCCN1CCOCC1 ZINC000217718014 DD For-Sale Unstable HTR2A 23 41 COc1ccccc1/C=C/NC(=O)NCCN1CCOCC1 ZINC000217718014 DD For-Sale Unstable DRD3 58 48 COc1ccccc1/C=C/NC(=O)NCCN1CCOCC1 ZINC000217718014 DD For-Sale Unstable ITGAL 22 42 COc1ccccc1/C=C/NC(=O)NCCN1CCOCC1 ZINC000217718014 DD For-Sale Unstable CNR2 17 44 COc1ccccc1/C=C/NC(=O)NCCN1CCOCC1 ZINC000217718014 DD For-Sale Unstable CASR 40 39 COc1ccccc1/C=C/NC(=O)NCCN1CCOCC1 ZINC000217718014 DD For-Sale Unstable EPHX2 22 45 COc1ccccc1/C=C/NC(=O)NCCN1CCOCC1 ZINC000217718014 DD For-Sale Unstable ACKR3 22 41 Cc1cc(C)cc(NC(=O)COc2ccc(Br)cc2C(=O)O)c1 ZINC000217718033 GH In-Stock Unstable PRS 55 34 Cc1cc(C)cc(NC(=O)COc2ccc(Br)cc2C(=O)O)c1 ZINC000217718033 GH In-Stock Unstable CETP 0 52 Cc1cc(C)cc(NC(=O)COc2ccc(Br)cc2C(=O)O)c1 ZINC000217718033 GH In-Stock Unstable AKR1C2 42 38 CCC[C@H]1CC[C@@H](NCC)[C@@H](CCOc2ccccc2)C1 ZINC000217718054 CJ For-Sale Unstable GRIN2B 15 40 COC(=O)c1cc(N)c2nccnc2c1 ZINC000217718061 BC In-Stock Unstable KDM5C 0 40 Cc1cccc(N2CCN(CC(=O)N[C@@H]3CCOC3)CC2)c1 ZINC000217718062 DD In-Stock Unstable HTR1A 21 48 Cc1cccc(N2CCN(CC(=O)N[C@@H]3CCOC3)CC2)c1 ZINC000217718062 DD In-Stock Unstable DRD4 24 51 Cc1cccc(N2CCN(CC(=O)N[C@@H]3CCOC3)CC2)c1 ZINC000217718062 DD In-Stock Unstable HTR2A 17 48 CCC[C@@H]1CC[C@H](NCC)[C@@H](CCOc2ccccc2)C1 ZINC000217718129 CJ For-Sale Unstable GRIN2B 15 40 O=C(COc1ccc(Br)cc1C(=O)O)Nc1ccccc1F ZINC000217718141 FG In-Stock Unstable CETP 0 40 O=C(COc1ccc(Br)cc1C(=O)O)Nc1ccccc1F ZINC000217718141 FG In-Stock Unstable FABH 0 40 O=C(COc1ccc(Br)cc1C(=O)O)Nc1ccccc1F ZINC000217718141 FG In-Stock Unstable AKR1C2 47 36 Cc1cccc(N2CCN(CC(=O)N[C@H]3CCOC3)CC2)c1 ZINC000217718155 DD In-Stock Unstable HTR1A 21 48 Cc1cccc(N2CCN(CC(=O)N[C@H]3CCOC3)CC2)c1 ZINC000217718155 DD In-Stock Unstable DRD4 24 51 Cc1cccc(N2CCN(CC(=O)N[C@H]3CCOC3)CC2)c1 ZINC000217718155 DD In-Stock Unstable HTR2A 17 48 COC(=O)c1cc([N+](=O)[O-])c2nccnc2c1 ZINC000217718188 BD In-Stock Unstable TRXR2 0 45 CN(Cc1cnn(C)c1)C(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217718218 DD For-Sale Unstable HSD17B2 21 42 CCC[C@H]1CC[C@H](NCC)[C@@H](CCOc2ccccc2)C1 ZINC000217718226 CJ For-Sale Unstable GRIN2B 15 40 COc1ccccc1/C=C/NC(=O)N1CCN(CCN)CC1 ZINC000217718252 DC For-Sale Unstable HTR1A 61 40 COc1ccccc1/C=C/NC(=O)N1CCN(CCN)CC1 ZINC000217718252 DC For-Sale Unstable DRD2 43 47 COc1ccccc1/C=C/NC(=O)N1CCN(CCN)CC1 ZINC000217718252 DC For-Sale Unstable DRD4 41 33 COc1ccccc1/C=C/NC(=O)N1CCN(CCN)CC1 ZINC000217718252 DC For-Sale Unstable DRD3 57 47 COc1ccccc1/C=C/NC(=O)N1CCN(CCN)CC1 ZINC000217718252 DC For-Sale Unstable HTR4 21 40 COc1ccccc1/C=C/NC(=O)N1CCN(CCN)CC1 ZINC000217718252 DC For-Sale Unstable HTR7 43 39 O=C(COc1ccc(Br)cc1C(=O)O)Nc1ccccc1Cl ZINC000217718257 GH In-Stock Unstable CETP 0 40 O=C(COc1ccc(Br)cc1C(=O)O)Nc1ccccc1Cl ZINC000217718257 GH In-Stock Unstable EPHB3 44 37 O=C(COc1ccc(Br)cc1C(=O)O)Nc1ccccc1Cl ZINC000217718257 GH In-Stock Unstable AKR1C2 54 38 O=C(O)c1cc([N+](=O)[O-])c2nccnc2c1 ZINC000217718289 BD In-Stock Bother TPMT 0 44 O=C(O)c1cc([N+](=O)[O-])c2nccnc2c1 ZINC000217718289 BD In-Stock Bother TRXR2 0 50 COc1ccccc1/C=C/NC(=O)NCCN1CCNCC1 ZINC000217718352 DC For-Sale Unstable HTR1A 52 47 COc1ccccc1/C=C/NC(=O)NCCN1CCNCC1 ZINC000217718352 DC For-Sale Unstable DRD2 41 48 COc1ccccc1/C=C/NC(=O)NCCN1CCNCC1 ZINC000217718352 DC For-Sale Unstable DRD4 46 36 COc1ccccc1/C=C/NC(=O)NCCN1CCNCC1 ZINC000217718352 DC For-Sale Unstable HTR2A 22 42 COc1ccccc1/C=C/NC(=O)NCCN1CCNCC1 ZINC000217718352 DC For-Sale Unstable DRD3 59 48 COc1ccccc1/C=C/NC(=O)NCCN1CCNCC1 ZINC000217718352 DC For-Sale Unstable HTR4 22 46 O=C(COc1ccc(Br)cc1C(=O)O)Nc1cccc(Cl)c1 ZINC000217718357 GH In-Stock Unstable PPIA 15 40 O=C(COc1ccc(Br)cc1C(=O)O)Nc1cccc(Cl)c1 ZINC000217718357 GH In-Stock Unstable CETP 0 42 O=C(COc1ccc(Br)cc1C(=O)O)Nc1cccc(Cl)c1 ZINC000217718357 GH In-Stock Unstable PTPN22 24 42 O=C(COc1ccc(Br)cc1C(=O)O)Nc1cccc(Cl)c1 ZINC000217718357 GH In-Stock Unstable PTGDR2 23 46 O=C(COc1ccc(Br)cc1C(=O)O)Nc1cccc(Cl)c1 ZINC000217718357 GH In-Stock Unstable AKR1C3 26 46 O=C(COc1ccc(Br)cc1C(=O)O)Nc1cccc(Cl)c1 ZINC000217718357 GH In-Stock Unstable AKR1C2 45 46 O=C(COc1ccc(Br)cc1C(=O)O)Nc1cccc(Cl)c1 ZINC000217718357 GH In-Stock Unstable PSBA 0 42 CN(C[C@@H]1CCCN1C)c1cc(Cl)ccc1CBr ZINC000217718392 EH For-Sale Unstable NOS3 16 42 CN(C[C@@H]1CCCN1C)c1cc(Cl)ccc1CBr ZINC000217718392 EH For-Sale Unstable CHRNA10 70 46 Cc1ccccc1CC(=O)Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1 ZINC000217718432 EI On-Demand Unstable COLA 89 36 Cc1ccccc1CC(=O)Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1 ZINC000217718432 EI On-Demand Unstable ECE1 17 40 Cc1ccccc1CC(=O)Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1 ZINC000217718432 EI On-Demand Unstable IMDH_CRYPV 28 41 O=C(COc1ccc(Br)cc1C(=O)O)Nc1ccc(Cl)cc1 ZINC000217718478 GH In-Stock Unstable PTGER1 40 39 O=C(COc1ccc(Br)cc1C(=O)O)Nc1ccc(Cl)cc1 ZINC000217718478 GH In-Stock Unstable CETP 0 46 O=C(COc1ccc(Br)cc1C(=O)O)Nc1ccc(Cl)cc1 ZINC000217718478 GH In-Stock Unstable CCR5 20 40 O=C(COc1ccc(Br)cc1C(=O)O)Nc1ccc(Cl)cc1 ZINC000217718478 GH In-Stock Unstable COLA 41 36 O=C(COc1ccc(Br)cc1C(=O)O)Nc1ccc(Cl)cc1 ZINC000217718478 GH In-Stock Unstable CPT1A 41 36 O=C(COc1ccc(Br)cc1C(=O)O)Nc1ccc(Cl)cc1 ZINC000217718478 GH In-Stock Unstable CPT2 42 32 O=C(COc1ccc(Br)cc1C(=O)O)Nc1ccc(Cl)cc1 ZINC000217718478 GH In-Stock Unstable GUAB 0 50 O=C(COc1ccc(Br)cc1C(=O)O)Nc1ccc(Cl)cc1 ZINC000217718478 GH In-Stock Unstable AGPAT2 38 40 O=C(COc1ccc(Br)cc1C(=O)O)Nc1ccc(Cl)cc1 ZINC000217718478 GH In-Stock Unstable MCHR2 21 40 O=C(COc1ccc(Br)cc1C(=O)O)Nc1ccc(Cl)cc1 ZINC000217718478 GH In-Stock Unstable PTGDR2 24 46 O=C(COc1ccc(Br)cc1C(=O)O)Nc1ccc(Cl)cc1 ZINC000217718478 GH In-Stock Unstable AKR1C3 19 40 O=C(COc1ccc(Br)cc1C(=O)O)Nc1ccc(Cl)cc1 ZINC000217718478 GH In-Stock Unstable AKR1C2 41 43 O=C(COc1ccc(Br)cc1C(=O)O)Nc1ccc(Cl)cc1 ZINC000217718478 GH In-Stock Unstable SENP1 0 41 O=C(COc1ccc(Br)cc1C(=O)O)Nc1ccc(Cl)cc1 ZINC000217718478 GH In-Stock Unstable PSBA 0 42 O=C(NC[C@@H]1CCCN2CCCC[C@H]12)C1CCN(c2ncccn2)CC1 ZINC000217718479 FE In-Stock Unstable GPBAR1 0 44 CN(C[C@H]1CCCN1C)c1cc(Cl)ccc1CBr ZINC000217718490 EH For-Sale Unstable NOS3 16 42 CN(C[C@H]1CCCN1C)c1cc(Cl)ccc1CBr ZINC000217718490 EH For-Sale Unstable CHRNA10 70 46 O=C(NC[C@@H](O)c1ccsc1)c1cccc(Br)n1 ZINC000217718524 EE On-Demand Unstable SCD 0 43 O=C(Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1)c1ccc2c(c1)OCCCO2 ZINC000217718559 GI On-Demand Unstable PLK1 16 44 O=C(Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1)c1ccc2c(c1)OCCCO2 ZINC000217718559 GI On-Demand Unstable TAAR1 44 39 O=C(COc1ccc(Br)cc1C(=O)O)Nc1ccc(Br)cc1 ZINC000217718572 IH In-Stock Unstable PRS 62 38 O=C(COc1ccc(Br)cc1C(=O)O)Nc1ccc(Br)cc1 ZINC000217718572 IH In-Stock Unstable CETP 0 49 O=C(COc1ccc(Br)cc1C(=O)O)Nc1ccc(Br)cc1 ZINC000217718572 IH In-Stock Unstable AKR1C3 23 44 O=C(COc1ccc(Br)cc1C(=O)O)Nc1ccc(Br)cc1 ZINC000217718572 IH In-Stock Unstable AKR1C2 51 44 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCc1cccnc1 ZINC000217718590 IG In-Stock Unstable SCN9A 0 44 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCc1cccnc1 ZINC000217718590 IG In-Stock Unstable NAMPT 45 36 O=C(O)/C=C\c1ccc(C(=O)NCCn2ccnc2)cc1 ZINC000217718592 CD For-Sale Unstable TBXAS1 68 61 O=C(O)/C=C\c1ccc(C(=O)NCCn2ccnc2)cc1 ZINC000217718592 CD For-Sale Unstable CYP24A1 55 47 O=C(O)/C=C\c1ccc(C(=O)NCCn2ccnc2)cc1 ZINC000217718592 CD For-Sale Unstable CYP27B1 74 47 COc1ccccc1/C=C/NC(=O)NCc1ccncc1 ZINC000217718604 CF For-Sale Unstable ROCK2 22 42 O=C(NC[C@H](O)c1ccsc1)c1cccc(Br)n1 ZINC000217718612 EE On-Demand Unstable SCD 0 43 CN(C[C@@H]1CCCN1C)c1ccc(Cl)cc1CBr ZINC000217718625 EH For-Sale Unstable NOS2 17 44 CN(C[C@@H]1CCCN1C)c1ccc(Cl)cc1CBr ZINC000217718625 EH For-Sale Unstable NOS3 19 44 CN(C[C@@H]1CCCN1C)c1ccc(Cl)cc1CBr ZINC000217718625 EH For-Sale Unstable CHRNA10 70 49 O=C(Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1)c1ccc(F)c(F)c1 ZINC000217718665 EI On-Demand Bother TAAR1 54 50 O=C(Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1)c1ccc(F)c(F)c1 ZINC000217718665 EI On-Demand Bother KCNK3 40 38 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCc1cccnc1 ZINC000217718677 IG In-Stock Unstable SCN9A 0 44 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCc1cccnc1 ZINC000217718677 IG In-Stock Unstable NAMPT 45 36 O=C(COc1ccc(Br)cc1C(=O)O)Nc1cc(Cl)cc(Cl)c1 ZINC000217718688 HI In-Stock Unstable CETP 0 42 O=C(COc1ccc(Br)cc1C(=O)O)Nc1cc(Cl)cc(Cl)c1 ZINC000217718688 HI In-Stock Unstable PTGDR2 16 49 CN(C[C@H]1CCCN1C)c1ccc(Cl)cc1CBr ZINC000217718708 EH For-Sale Unstable NOS2 17 44 CN(C[C@H]1CCCN1C)c1ccc(Cl)cc1CBr ZINC000217718708 EH For-Sale Unstable NOS3 19 44 CN(C[C@H]1CCCN1C)c1ccc(Cl)cc1CBr ZINC000217718708 EH For-Sale Unstable CHRNA10 70 49 O=C(O)/C=C\c1cccc(C(=O)NCCn2ccnc2)c1 ZINC000217718718 CD For-Sale Unstable DRD4 41 31 O=C(O)/C=C\c1cccc(C(=O)NCCn2ccnc2)c1 ZINC000217718718 CD For-Sale Unstable TBXAS1 65 62 O=C(O)/C=C\c1cccc(C(=O)NCCn2ccnc2)c1 ZINC000217718718 CD For-Sale Unstable CYP24A1 56 41 O=C(O)/C=C\c1cccc(C(=O)NCCn2ccnc2)c1 ZINC000217718718 CD For-Sale Unstable CYP27B1 76 41 C[C@H](O)[C@H](NC(=O)c1ccc(F)c(Br)c1)C(=O)O ZINC000217718730 DD For-Sale Unstable CA2 21 54 C[C@H](O)[C@H](NC(=O)c1ccc(F)c(Br)c1)C(=O)O ZINC000217718730 DD For-Sale Unstable CA4 16 56 Cc1cc(N2C[C@]34C=C[C@@H](O3)[C@@H](C(=O)Nc3ccc(OC(F)(F)F)cc3)[C@H]4C2=O)no1 ZINC000217718755 IF In-Stock Unstable P2RY1 53 32 Cc1cc(N2C[C@]34C=C[C@@H](O3)[C@@H](C(=O)Nc3ccc(OC(F)(F)F)cc3)[C@H]4C2=O)no1 ZINC000217718755 IF In-Stock Unstable EPHX2 48 44 O=C(C[C@@H]1C=CCC1)Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1 ZINC000217718774 DH On-Demand Unstable AADAC 0 54 CCOc1ccc(/C=C\C(=O)NCC2CC(O)C2)cc1 ZINC000217718794 CD For-Sale Unstable HDAC8 22 42 CCOc1ccc(/C=C\C(=O)NCC2CC(O)C2)cc1 ZINC000217718794 CD For-Sale Unstable IMA1 0 40 CS(=O)(=O)CCNS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217718802 EC For-Sale Unstable HDAC8 15 47 CS(=O)(=O)CCNS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217718802 EC For-Sale Unstable AKR1C3 38 45 O=C(COc1ccc(Br)cc1C(=O)O)Nc1cccc(C(F)(F)F)c1 ZINC000217718810 HI In-Stock Unstable UL80 21 41 O=C(COc1ccc(Br)cc1C(=O)O)Nc1cccc(C(F)(F)F)c1 ZINC000217718810 HI In-Stock Unstable CETP 0 42 O=C(COc1ccc(Br)cc1C(=O)O)Nc1cccc(C(F)(F)F)c1 ZINC000217718810 HI In-Stock Unstable KDR 19 41 O=C(COc1ccc(Br)cc1C(=O)O)Nc1cccc(C(F)(F)F)c1 ZINC000217718810 HI In-Stock Unstable AKR1C3 26 47 O=C(COc1ccc(Br)cc1C(=O)O)Nc1cccc(C(F)(F)F)c1 ZINC000217718810 HI In-Stock Unstable AKR1C2 31 49 O=C(COc1ccc(Br)cc1C(=O)O)Nc1cccc(C(F)(F)F)c1 ZINC000217718810 HI In-Stock Unstable TRPM4 0 49 O=C(COc1ccc(Br)cc1C(=O)O)Nc1cccc(C(F)(F)F)c1 ZINC000217718810 HI In-Stock Unstable KCNK3 43 38 O=C(COc1ccc(Br)cc1C(=O)O)Nc1cccc(C(F)(F)F)c1 ZINC000217718810 HI In-Stock Unstable PDS 39 40 CCCCCCCCCC(=O)C(C)(C)CN ZINC000217718820 BH For-Sale Unstable FABP2 0 46 CCCCCCCCCC(=O)C(C)(C)CN ZINC000217718820 BH For-Sale Unstable FABP4 16 46 CCCCCCCCCC(=O)C(C)(C)CN ZINC000217718820 BH For-Sale Unstable FAAH 25 55 CCCCCCCCCC(=O)C(C)(C)CN ZINC000217718820 BH For-Sale Unstable CES2 57 55 CCCCCCCCCC(=O)C(C)(C)CN ZINC000217718820 BH For-Sale Unstable CES1 47 55 CCCCCCCCCC(=O)C(C)(C)CN ZINC000217718820 BH For-Sale Unstable EST1_PIG 81 55 CCCCCCCCCC(=O)C(C)(C)CN ZINC000217718820 BH For-Sale Unstable CES2C 64 40 CCCCCCCCCC(=O)C(C)(C)CN ZINC000217718820 BH For-Sale Unstable JHE 0 55 CCCCCCCCCC(=O)C(C)(C)CN ZINC000217718820 BH For-Sale Unstable FABP5 15 46 CCCCCCCCCC(=O)C(C)(C)CN ZINC000217718820 BH For-Sale Unstable SLC22A20 0 46 CCCCCCCCCC(=O)C(C)(C)CN ZINC000217718820 BH For-Sale Unstable Q9GPG0_MANSE 0 55 CCCCCCCCCC(=O)C(C)(C)CN ZINC000217718820 BH For-Sale Unstable CQSS 67 42 C[C@H](O)[C@@H](NC(=O)c1ccc(F)c(Br)c1)C(=O)O ZINC000217718832 DD For-Sale Unstable CA2 21 54 C[C@H](O)[C@@H](NC(=O)c1ccc(F)c(Br)c1)C(=O)O ZINC000217718832 DD For-Sale Unstable CA4 16 56 COc1ccccc1/C=C/NC(=O)NCCCN1CCOCC1 ZINC000217718838 DD For-Sale Unstable HTR1A 69 46 COc1ccccc1/C=C/NC(=O)NCCCN1CCOCC1 ZINC000217718838 DD For-Sale Unstable DRD2 55 54 COc1ccccc1/C=C/NC(=O)NCCCN1CCOCC1 ZINC000217718838 DD For-Sale Unstable CNR1 0 43 COc1ccccc1/C=C/NC(=O)NCCCN1CCOCC1 ZINC000217718838 DD For-Sale Unstable DRD1 23 43 COc1ccccc1/C=C/NC(=O)NCCCN1CCOCC1 ZINC000217718838 DD For-Sale Unstable DRD4 41 32 COc1ccccc1/C=C/NC(=O)NCCCN1CCOCC1 ZINC000217718838 DD For-Sale Unstable ADRA1D 47 43 COc1ccccc1/C=C/NC(=O)NCCCN1CCOCC1 ZINC000217718838 DD For-Sale Unstable HTR2A 36 43 COc1ccccc1/C=C/NC(=O)NCCCN1CCOCC1 ZINC000217718838 DD For-Sale Unstable HTR2C 24 40 COc1ccccc1/C=C/NC(=O)NCCCN1CCOCC1 ZINC000217718838 DD For-Sale Unstable ADRA1A 60 42 COc1ccccc1/C=C/NC(=O)NCCCN1CCOCC1 ZINC000217718838 DD For-Sale Unstable ADRA1B 39 43 COc1ccccc1/C=C/NC(=O)NCCCN1CCOCC1 ZINC000217718838 DD For-Sale Unstable DRD3 82 54 COc1ccccc1/C=C/NC(=O)NCCCN1CCOCC1 ZINC000217718838 DD For-Sale Unstable HTR7 49 39 COc1ccccc1/C=C/NC(=O)NCCCN1CCOCC1 ZINC000217718838 DD For-Sale Unstable TACR2 29 45 COc1ccccc1/C=C/NC(=O)NCCCN1CCOCC1 ZINC000217718838 DD For-Sale Unstable CCR3 26 43 COc1ccccc1/C=C/NC(=O)NCCCN1CCOCC1 ZINC000217718838 DD For-Sale Unstable EPHX2 23 42 COc1ccccc1/C=C/NC(=O)NCCCN1CCOCC1 ZINC000217718838 DD For-Sale Unstable AP2S1 0 40 COc1ccccc1/C=C/NC(=O)NCCCN1CCOCC1 ZINC000217718838 DD For-Sale Unstable ALPHA-1A 0 41 COc1ccccc1/C=C/NC(=O)NCCCN1CCOCC1 ZINC000217718838 DD For-Sale Unstable ACKR3 22 44 Cc1cc(N2C[C@]34C=C[C@@H](O3)[C@H](C(=O)Nc3ccc(OC(F)(F)F)cc3)[C@H]4C2=O)no1 ZINC000217718846 IF In-Stock Unstable P2RY1 53 32 Cc1cc(N2C[C@]34C=C[C@@H](O3)[C@H](C(=O)Nc3ccc(OC(F)(F)F)cc3)[C@H]4C2=O)no1 ZINC000217718846 IF In-Stock Unstable EPHX2 48 44 O=C(C[C@H]1C=CCC1)Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1 ZINC000217718856 DH On-Demand Unstable AADAC 0 54 COc1ccc(S(=O)(=O)NC(C)C)cc1/C=C\C(=O)O ZINC000217718888 CD For-Sale Unstable MMP13 34 42 COc1ccc(S(=O)(=O)NC(C)C)cc1/C=C\C(=O)O ZINC000217718888 CD For-Sale Unstable MMP2 24 42 COc1ccc(S(=O)(=O)NC(C)C)cc1/C=C\C(=O)O ZINC000217718888 CD For-Sale Unstable MMP12 74 42 COc1ccc(S(=O)(=O)NC(C)C)cc1/C=C\C(=O)O ZINC000217718888 CD For-Sale Unstable MMP7 16 42 COc1ccc(S(=O)(=O)NC(C)C)cc1/C=C\C(=O)O ZINC000217718888 CD For-Sale Unstable ADAMTS4 51 34 COc1ccc(S(=O)(=O)NC(C)C)cc1/C=C\C(=O)O ZINC000217718888 CD For-Sale Unstable LEF 27 42 C[C@@H](O)[C@@H](NC(=O)c1ccc(F)c(Br)c1)C(=O)O ZINC000217718909 DD For-Sale Unstable CA2 21 54 C[C@@H](O)[C@@H](NC(=O)c1ccc(F)c(Br)c1)C(=O)O ZINC000217718909 DD For-Sale Unstable CA4 16 56 O=C1[C@H]2[C@@H]3C=C[C@@H](C3)[C@H]2C(=O)N1c1cccc(I)c1 ZINC000217718912 FF For-Sale Unstable AR 15 63 O=C1[C@H]2[C@@H]3C=C[C@@H](C3)[C@H]2C(=O)N1c1cccc(I)c1 ZINC000217718912 FF For-Sale Unstable WNT3 28 44 COc1cccc(NC(=O)COc2ccc(Br)cc2C(=O)O)c1 ZINC000217718914 GG In-Stock Unstable PDGFRB 19 45 COc1cccc(NC(=O)COc2ccc(Br)cc2C(=O)O)c1 ZINC000217718914 GG In-Stock Unstable CETP 0 47 COc1cccc(NC(=O)COc2ccc(Br)cc2C(=O)O)c1 ZINC000217718914 GG In-Stock Unstable MTNR1A 37 49 COc1cccc(NC(=O)COc2ccc(Br)cc2C(=O)O)c1 ZINC000217718914 GG In-Stock Unstable MTNR1B 43 49 COc1cccc(NC(=O)COc2ccc(Br)cc2C(=O)O)c1 ZINC000217718914 GG In-Stock Unstable FPR2 21 40 COc1cccc(NC(=O)COc2ccc(Br)cc2C(=O)O)c1 ZINC000217718914 GG In-Stock Unstable TAAR1 33 44 COc1cccc(NC(=O)COc2ccc(Br)cc2C(=O)O)c1 ZINC000217718914 GG In-Stock Unstable AKR1C3 46 50 COc1cccc(NC(=O)COc2ccc(Br)cc2C(=O)O)c1 ZINC000217718914 GG In-Stock Unstable AKR1C2 78 46 COc1cccc(NC(=O)COc2ccc(Br)cc2C(=O)O)c1 ZINC000217718914 GG In-Stock Unstable ENPP1 46 34 COc1cccc(NC(=O)COc2ccc(Br)cc2C(=O)O)c1 ZINC000217718914 GG In-Stock Unstable KCNK3 53 42 COc1cccc(NC(=O)COc2ccc(Br)cc2C(=O)O)c1 ZINC000217718914 GG In-Stock Unstable KCNK9 45 42 COc1ccc(NC(=O)ON=C(C)C)c(OC)c1 ZINC000217718916 CF For-Sale Unstable CYP1B1 37 56 COc1ccc(NC(=O)ON=C(C)C)c(OC)c1 ZINC000217718916 CF For-Sale Unstable MTNR1A 37 42 COc1ccc(NC(=O)ON=C(C)C)c(OC)c1 ZINC000217718916 CF For-Sale Unstable MTNR1B 35 42 COc1ccc(NC(=O)ON=C(C)C)c(OC)c1 ZINC000217718916 CF For-Sale Unstable AKR1C2 50 35 COC(=O)c1cc(Cl)c2nccnc2c1 ZINC000217718933 BE In-Stock Unstable KDM5C 0 40 O=C(Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1)c1cc(F)ccc1Br ZINC000217718966 HJ On-Demand Bother TAAR1 35 40 O=C1[C@H]2[C@@H]3C=C[C@H](C3)[C@H]2C(=O)N1c1cccc(I)c1 ZINC000217718989 FF For-Sale Unstable AR 15 63 O=C1[C@H]2[C@@H]3C=C[C@H](C3)[C@H]2C(=O)N1c1cccc(I)c1 ZINC000217718989 FF For-Sale Unstable WNT3 28 44 CC(C)[C@@H]1C[C@@]1(CCC#N)NC(=O)OC(C)(C)C ZINC000217719007 CG For-Sale Unstable PAPA1_CARPA 43 35 CCCN(CC)CCNCc1cc(OC)c(O)c(OC)c1 ZINC000217719009 CE On-Demand Unstable SLC6A13 0 42 COc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217719016 GG In-Stock Unstable ADORA2B 40 43 COc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217719016 GG In-Stock Unstable PRS 41 33 COc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217719016 GG In-Stock Unstable CETP 0 49 COc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217719016 GG In-Stock Unstable MTNR1A 25 41 COc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217719016 GG In-Stock Unstable MTNR1B 22 45 COc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217719016 GG In-Stock Unstable CA9 17 40 COc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217719016 GG In-Stock Unstable AKR1C3 36 52 COc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217719016 GG In-Stock Unstable AKR1C2 74 52 COc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217719016 GG In-Stock Unstable ENPP1 58 37 COc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217719016 GG In-Stock Unstable PSBA 0 40 COc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217719016 GG In-Stock Unstable FAS 29 42 O=C(Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1)c1cc(Cl)ccc1F ZINC000217719063 FJ On-Demand Bother GRM4 15 46 O=C1[C@H]2[C@@H]3C=C[C@H](C3)[C@@H]2C(=O)N1c1cccc(I)c1 ZINC000217719070 FF For-Sale Unstable AR 15 63 O=C1[C@H]2[C@@H]3C=C[C@H](C3)[C@@H]2C(=O)N1c1cccc(I)c1 ZINC000217719070 FF For-Sale Unstable WNT3 28 44 COc1ccccc1/C=C/NC(=O)N(C)Cc1ccccc1 ZINC000217719080 CH For-Sale Unstable PTGER2 24 41 COc1ccccc1/C=C/NC(=O)N(C)Cc1ccccc1 ZINC000217719080 CH For-Sale Unstable PTGES 0 40 COc1ccccc1/C=C/NC(=O)N(C)Cc1ccccc1 ZINC000217719080 CH For-Sale Unstable LIMK2 20 44 COc1ccccc1/C=C/NC(=O)N(C)Cc1ccccc1 ZINC000217719080 CH For-Sale Unstable AKR1B10 32 42 CC(C)[C@H]1C[C@@]1(CCC#N)NC(=O)OC(C)(C)C ZINC000217719091 CG For-Sale Unstable PAPA1_CARPA 43 35 CCOc1ccccc1NC(=O)COc1ccc(Br)cc1C(=O)O ZINC000217719109 GH In-Stock Unstable CETP 0 43 CCOc1ccccc1NC(=O)COc1ccc(Br)cc1C(=O)O ZINC000217719109 GH In-Stock Unstable AGPAT2 22 40 CCOc1ccccc1NC(=O)COc1ccc(Br)cc1C(=O)O ZINC000217719109 GH In-Stock Unstable AKR1C2 44 35 CCOc1ccccc1NC(=O)COc1ccc(Br)cc1C(=O)O ZINC000217719109 GH In-Stock Unstable HCN1 41 32 CCOc1ccccc1NC(=O)COc1ccc(Br)cc1C(=O)O ZINC000217719109 GH In-Stock Unstable HCN4 41 32 CCOc1ccccc1NC(=O)COc1ccc(Br)cc1C(=O)O ZINC000217719109 GH In-Stock Unstable KCNK3 26 40 CCOc1ccccc1NC(=O)COc1ccc(Br)cc1C(=O)O ZINC000217719109 GH In-Stock Unstable KCNK9 20 40 CC(C)[C@@H]1C[C@]1(CCC#N)NC(=O)OC(C)(C)C ZINC000217719173 CG For-Sale Unstable PAPA1_CARPA 43 35 CCC[C@@H](C)NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217719191 CE For-Sale Unstable HDAC8 16 45 CCC[C@@H](C)NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217719191 CE For-Sale Unstable LEF 17 44 CCOc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217719200 GH In-Stock Unstable ADORA2B 43 42 CCOc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217719200 GH In-Stock Unstable CETP 0 46 CCOc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217719200 GH In-Stock Unstable AGPAT2 27 40 CCOc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217719200 GH In-Stock Unstable AKR1C3 26 43 CCOc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217719200 GH In-Stock Unstable AKR1C2 52 43 Cc1ccc(N2C(=O)[C@H]3[C@@H]4C=C[C@@H](C4)[C@H]3C2=O)c(Br)c1 ZINC000217719224 EG For-Sale Unstable WNT3 21 40 Cc1ccc(C)n1CC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217719229 ED In-Stock Unstable CHRNA4 33 55 CC(C)[C@H]1C[C@]1(CCC#N)NC(=O)OC(C)(C)C ZINC000217719249 CG For-Sale Unstable PAPA1_CARPA 43 35 CCC[C@H](C)NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217719272 CE For-Sale Unstable HDAC8 16 45 CCC[C@H](C)NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217719272 CE For-Sale Unstable LEF 17 44 O=C(COc1ccc(Br)cc1C(=O)O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217719296 IJ In-Stock Unstable LTA4H 51 47 O=C(COc1ccc(Br)cc1C(=O)O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217719296 IJ In-Stock Unstable CA1 28 42 O=C(COc1ccc(Br)cc1C(=O)O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217719296 IJ In-Stock Unstable CETP 0 48 O=C(COc1ccc(Br)cc1C(=O)O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217719296 IJ In-Stock Unstable GUAB 0 53 O=C(COc1ccc(Br)cc1C(=O)O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217719296 IJ In-Stock Unstable FABH 0 41 O=C(COc1ccc(Br)cc1C(=O)O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217719296 IJ In-Stock Unstable MCHR1 20 42 O=C(COc1ccc(Br)cc1C(=O)O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217719296 IJ In-Stock Unstable AKR1C3 28 40 O=C(COc1ccc(Br)cc1C(=O)O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217719296 IJ In-Stock Unstable AKR1C2 64 40 Cc1ccc(N2C(=O)[C@H]3[C@@H]4C=C[C@H](C4)[C@H]3C2=O)c(Br)c1 ZINC000217719311 EG For-Sale Unstable WNT3 21 40 COc1ccccc1/C=C/NC(=O)Nc1nc(C)cs1 ZINC000217719328 CG For-Sale Unstable GCK 20 53 CC[C@@H](CCO)NCc1cncn1C1CC1 ZINC000217719343 BD For-Sale Unstable CAMC 0 45 CCC[C@@H](C)NS(=O)(=O)c1ccc(/C=C\C(=O)O)c(C)c1 ZINC000217719345 DF For-Sale Unstable LEF 62 42 Cc1ccc(N2C(=O)[C@H]3[C@@H]4C=C[C@H](C4)[C@@H]3C2=O)c(Br)c1 ZINC000217719397 EG For-Sale Unstable WNT3 21 40 CC[C@@H](C)[C@@H](N)C(=O)N[C@@H]1CCC[C@@H](O)C1 ZINC000217719413 BC For-Sale Unstable TPP2 39 41 CC[C@H](CCO)NCc1cncn1C1CC1 ZINC000217719415 BD For-Sale Unstable CAMC 0 45 COc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)c(OC)c1 ZINC000217719418 HG In-Stock Unstable AKR1C3 27 49 COc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)c(OC)c1 ZINC000217719418 HG In-Stock Unstable AKR1C2 64 49 COc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)c(OC)c1 ZINC000217719418 HG In-Stock Unstable GPR35 46 36 COc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)c(OC)c1 ZINC000217719418 HG In-Stock Unstable FAS 46 45 CCC[C@H](C)NS(=O)(=O)c1ccc(/C=C\C(=O)O)c(C)c1 ZINC000217719435 DF For-Sale Unstable LEF 62 42 Cc1cc(NC(=O)C2CCN(S(=O)(=O)c3c(C)c(C)cc(C)c3C)CC2)n(-c2ccccn2)n1 ZINC000217719481 JH On-Demand Unstable EPHX2 44 46 CC[C@H](C)[C@@H](N)C(=O)N[C@@H]1CCC[C@@H](O)C1 ZINC000217719531 BC For-Sale Unstable TPP2 39 41 COc1ccc(C)cc1NC(=O)COc1ccc(Br)cc1C(=O)O ZINC000217719533 GG In-Stock Unstable CETP 0 41 COc1ccc(C)cc1NC(=O)COc1ccc(Br)cc1C(=O)O ZINC000217719533 GG In-Stock Unstable AKR1C2 50 39 COc1cccc(NC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217719537 CG For-Sale Unstable PDGFRB 15 40 COc1cccc(NC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217719537 CG For-Sale Unstable CYP1B1 48 49 COc1cccc(NC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217719537 CG For-Sale Unstable KDR 17 44 COc1cccc(NC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217719537 CG For-Sale Unstable MTNR1A 29 47 COc1cccc(NC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217719537 CG For-Sale Unstable MTNR1B 35 47 COc1cccc(NC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217719537 CG For-Sale Unstable CYP1A1 37 41 COc1cccc(NC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217719537 CG For-Sale Unstable FLT4 18 40 COc1cccc(NC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217719537 CG For-Sale Unstable PDGFRA 36 44 COc1cccc(NC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217719537 CG For-Sale Unstable IMPDH2 0 43 COc1cccc(NC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217719537 CG For-Sale Unstable Q8MMZ8_EIMTE 0 48 COc1cccc(NC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217719537 CG For-Sale Unstable TAAR1 33 44 COc1cccc(NC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217719537 CG For-Sale Unstable AKR1C3 25 42 COc1cccc(NC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217719537 CG For-Sale Unstable KCNK3 94 49 COc1cccc(NC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217719537 CG For-Sale Unstable KCNK9 78 46 N#Cc1cccc(N2C(=O)[C@H]3[C@@H]4C=C[C@@H](C4)[C@H]3C2=O)c1 ZINC000217719543 CD For-Sale Unstable AR 19 59 N#Cc1cccc(N2C(=O)[C@H]3[C@@H]4C=C[C@@H](C4)[C@H]3C2=O)c1 ZINC000217719543 CD For-Sale Unstable WNT3 26 40 CC[C@@H](CCO)NCc1cn(CCO)nn1 ZINC000217719555 BB For-Sale Unstable GBA 15 40 CC[C@@H](C)[C@H](N)C(=O)N[C@@H]1CCC[C@@H](O)C1 ZINC000217719614 BC For-Sale Unstable TPP2 39 41 N#Cc1cccc(N2C(=O)[C@H]3[C@@H]4C=C[C@H](C4)[C@H]3C2=O)c1 ZINC000217719618 CD For-Sale Unstable AR 19 59 N#Cc1cccc(N2C(=O)[C@H]3[C@@H]4C=C[C@H](C4)[C@H]3C2=O)c1 ZINC000217719618 CD For-Sale Unstable WNT3 26 40 CC[C@H](CCO)NCc1cn(CCO)nn1 ZINC000217719641 BB For-Sale Unstable GBA 15 40 COc1ccccc1/C=C/NC(=O)Nc1cc(Cl)ccc1O ZINC000217719652 DH For-Sale Unstable KCNMA1 39 46 COc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1Cl ZINC000217719653 HH In-Stock Unstable HTR2A 17 42 COc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1Cl ZINC000217719653 HH In-Stock Unstable CYSP_TRYCR 0 43 COc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1Cl ZINC000217719653 HH In-Stock Unstable CETP 0 43 COc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1Cl ZINC000217719653 HH In-Stock Unstable COLA 45 37 COc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1Cl ZINC000217719653 HH In-Stock Unstable CPT1A 44 37 COc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1Cl ZINC000217719653 HH In-Stock Unstable CPT2 44 37 COc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1Cl ZINC000217719653 HH In-Stock Unstable GRM4 20 47 COc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1Cl ZINC000217719653 HH In-Stock Unstable MCHR2 34 42 COc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1Cl ZINC000217719653 HH In-Stock Unstable AKR1C3 25 41 COc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1Cl ZINC000217719653 HH In-Stock Unstable AKR1C2 49 41 COc1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1Cl ZINC000217719653 HH In-Stock Unstable ENPP1 72 38 Cc1cc(NC(=O)C2CCN(S(=O)(=O)c3ccc(Cl)cc3)CC2)n(-c2ccccn2)n1 ZINC000217719697 JG On-Demand Unstable GRM4 21 47 Cc1cc(NC(=O)C2CCN(S(=O)(=O)c3ccc(Cl)cc3)CC2)n(-c2ccccn2)n1 ZINC000217719697 JG On-Demand Unstable EPHX2 43 44 Cc1cc(NC(=O)C2CCN(S(=O)(=O)c3ccc(Cl)cc3)CC2)n(-c2ccccn2)n1 ZINC000217719697 JG On-Demand Unstable TGM2 31 42 Cc1cc(NC(=O)C2CCN(S(=O)(=O)c3ccc(Cl)cc3)CC2)n(-c2ccccn2)n1 ZINC000217719697 JG On-Demand Unstable TYK2 43 34 Cc1cc(NC(=O)C2CCN(S(=O)(=O)c3ccc(Cl)cc3)CC2)n(-c2ccccn2)n1 ZINC000217719697 JG On-Demand Unstable F13A1 30 42 N#Cc1cccc(N2C(=O)[C@H]3[C@@H]4C=C[C@H](C4)[C@@H]3C2=O)c1 ZINC000217719713 CD For-Sale Unstable AR 19 59 N#Cc1cccc(N2C(=O)[C@H]3[C@@H]4C=C[C@H](C4)[C@@H]3C2=O)c1 ZINC000217719713 CD For-Sale Unstable WNT3 26 40 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](CC(C)C)C(=O)Nc3nnn[nH]3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217719741 KF In-Stock Unstable TUBA1A 17 62 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](CC(C)C)C(=O)Nc3nnn[nH]3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217719741 KF In-Stock Unstable TPPP 0 58 COC(=O)c1ccccc1NC(=O)COc1ccc(Br)cc1C(=O)O ZINC000217719754 HF In-Stock Unstable CETP 0 43 COC(=O)c1ccccc1NC(=O)COc1ccc(Br)cc1C(=O)O ZINC000217719754 HF In-Stock Unstable HCAR2 39 41 COC(=O)c1ccccc1NC(=O)COc1ccc(Br)cc1C(=O)O ZINC000217719754 HF In-Stock Unstable FABH 0 41 COC(=O)c1ccccc1NC(=O)COc1ccc(Br)cc1C(=O)O ZINC000217719754 HF In-Stock Unstable AKR1C3 25 40 COC(=O)c1ccccc1NC(=O)COc1ccc(Br)cc1C(=O)O ZINC000217719754 HF In-Stock Unstable AKR1C2 64 40 COC(=O)c1ccccc1NC(=O)COc1ccc(Br)cc1C(=O)O ZINC000217719754 HF In-Stock Unstable FAS 80 53 CCOc1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1OCC ZINC000217719757 FI For-Sale Unstable IMPDH2 0 44 CCOc1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1OCC ZINC000217719757 FI For-Sale Unstable ENPP1 62 33 CCOc1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1OCC ZINC000217719757 FI For-Sale Unstable KCNK3 48 46 CCOc1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1OCC ZINC000217719757 FI For-Sale Unstable KCNK9 37 46 O=C(O)/C=C\c1cccc(S(=O)(=O)N2CCSCC2)c1 ZINC000217719777 DD For-Sale Unstable AKR1C3 64 41 CN1CCC(N2CCN(C(=O)c3ccncc3O)CC2)CC1 ZINC000217719805 DC In-Stock Unstable L3MBTL1 0 55 CN1CCC(N2CCN(C(=O)c3ccncc3O)CC2)CC1 ZINC000217719805 DC In-Stock Unstable L3MBTL3 75 55 CN1CCC(N2CCN(C(=O)c3ccncc3O)CC2)CC1 ZINC000217719805 DC In-Stock Unstable MBTD1 0 42 CN1CCC(N2CCN(C(=O)c3ccncc3O)CC2)CC1 ZINC000217719805 DC In-Stock Unstable TP53BP1 0 45 Cc1ccc(S(=O)(=O)N(C)c2ccc(C(=O)Nc3cc(C)nn3-c3ccccn3)cc2)cc1 ZINC000217719810 JH On-Demand Unstable SLC11A2 47 35 Cc1cc(S(=O)(=O)N2CCSCC2)ccc1/C=C\C(=O)O ZINC000217719850 ED For-Sale Unstable AKR1C3 46 35 COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc(OC)c1O ZINC000217719854 JI In-Stock Unstable AKR1B1 26 53 COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc(OC)c1O ZINC000217719854 JI In-Stock Unstable CYP1B1 77 41 COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc(OC)c1O ZINC000217719854 JI In-Stock Unstable CYP1A1 57 44 COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc(OC)c1O ZINC000217719854 JI In-Stock Unstable CYP1A2 46 51 COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc(OC)c1O ZINC000217719854 JI In-Stock Unstable ABCG2 0 40 COc1ccccc1/C=C/NC(=O)Nc1nccs1 ZINC000217719871 CF For-Sale Unstable MAP1 128 48 COC(=O)c1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217719878 HF In-Stock Unstable CETP 0 46 COC(=O)c1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217719878 HF In-Stock Unstable ACR 55 38 COC(=O)c1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217719878 HF In-Stock Unstable AKR1C3 32 43 COC(=O)c1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217719878 HF In-Stock Unstable AKR1C2 45 43 CCCN(C)C(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217719937 CE For-Sale Unstable CYSP_PLAFA 41 35 COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc(OC)c1O ZINC000217719941 JI In-Stock Unstable AKR1B1 26 53 COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc(OC)c1O ZINC000217719941 JI In-Stock Unstable CYP1B1 77 41 COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc(OC)c1O ZINC000217719941 JI In-Stock Unstable CYP1A1 57 44 COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc(OC)c1O ZINC000217719941 JI In-Stock Unstable CYP1A2 46 51 COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc(OC)c1O ZINC000217719941 JI In-Stock Unstable ABCG2 0 40 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217719977 ID In-Stock Unstable CA2 132 49 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217719977 ID In-Stock Unstable CA1 123 48 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217719977 ID In-Stock Unstable CA7 58 48 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217719977 ID In-Stock Unstable CETP 0 43 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217719977 ID In-Stock Unstable CA5B 62 48 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217719977 ID In-Stock Unstable CA4 114 49 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217719977 ID In-Stock Unstable CA5A 71 48 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217719977 ID In-Stock Unstable CA14 44 39 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217719977 ID In-Stock Unstable CA12 85 51 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217719977 ID In-Stock Unstable CA9 92 48 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217719977 ID In-Stock Unstable MTCA1 54 51 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(Br)cc2C(=O)O)cc1 ZINC000217719977 ID In-Stock Unstable P96878_MYCTU 69 51 COc1ccccc1/C=C/NC(=O)Nc1cccc(SC)c1 ZINC000217719978 DI For-Sale Unstable CYP1B1 25 45 COc1ccccc1/C=C/NC(=O)Nc1cccc(SC)c1 ZINC000217719978 DI For-Sale Unstable KCNK3 60 42 COc1ccccc1/C=C/NC(=O)Nc1cccc(SC)c1 ZINC000217719978 DI For-Sale Unstable KCNK9 61 42 CC(=O)c1cccc(NC(=O)COc2ccc(Br)cc2C(=O)O)c1 ZINC000217720072 GG In-Stock Unstable EGFR 37 41 CC(=O)c1cccc(NC(=O)COc2ccc(Br)cc2C(=O)O)c1 ZINC000217720072 GG In-Stock Unstable CETP 0 43 CC(=O)c1cccc(NC(=O)COc2ccc(Br)cc2C(=O)O)c1 ZINC000217720072 GG In-Stock Unstable HIF1A 20 43 CC(=O)c1cccc(NC(=O)COc2ccc(Br)cc2C(=O)O)c1 ZINC000217720072 GG In-Stock Unstable AKR1C3 55 49 CC(=O)c1cccc(NC(=O)COc2ccc(Br)cc2C(=O)O)c1 ZINC000217720072 GG In-Stock Unstable AKR1C2 52 48 CC(=O)c1cccc(NC(=O)COc2ccc(Br)cc2C(=O)O)c1 ZINC000217720072 GG In-Stock Unstable KCNK3 69 34 CC(=O)c1cccc(NC(=O)COc2ccc(Br)cc2C(=O)O)c1 ZINC000217720072 GG In-Stock Unstable KCNK9 67 37 CC(=O)c1cccc(NC(=O)COc2ccc(Br)cc2C(=O)O)c1 ZINC000217720072 GG In-Stock Unstable PARP10 0 42 COc1ccccc1/C=C/NC(=O)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217720083 JG For-Sale Unstable LPL 48 42 COc1ccccc1/C=C/NC(=O)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217720083 JG For-Sale Unstable LIPG 19 42 O=C(NCc1nc(-c2cnccn2)n[nH]1)c1ccccc1N1CCOCC1 ZINC000217720147 FD In-Stock Unstable STAT6 52 35 CCOc1ccc([C@@H](C)N[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217720168 CF For-Sale Unstable ACACA 25 41 Cc1cccc(C(=O)O)c1OCC(=O)NCc1ccccc1 ZINC000217720185 CE In-Stock Unstable PTGER2 0 45 Cc1cccc(C(=O)O)c1OCC(=O)NCc1ccccc1 ZINC000217720185 CE In-Stock Unstable FABP4 42 36 Cc1cccc(C(=O)O)c1OCC(=O)NCc1ccccc1 ZINC000217720185 CE In-Stock Unstable AMP1_PLAFQ 44 35 Cc1cccc(C(=O)O)c1OCC(=O)NCc1ccccc1 ZINC000217720185 CE In-Stock Unstable MCL1 47 33 Cc1cccc(C(=O)O)c1OCC(=O)NCc1ccccc1 ZINC000217720185 CE In-Stock Unstable AKR1C2 21 40 Cc1cccc(C(=O)O)c1OCC(=O)NCc1ccccc1 ZINC000217720185 CE In-Stock Unstable PDS 46 39 COc1ccccc1/C=C/NC(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000217720187 FD For-Sale Unstable CA2 104 53 COc1ccccc1/C=C/NC(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000217720187 FD For-Sale Unstable CA1 90 53 COc1ccccc1/C=C/NC(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000217720187 FD For-Sale Unstable CA7 56 51 COc1ccccc1/C=C/NC(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000217720187 FD For-Sale Unstable CA5B 53 51 COc1ccccc1/C=C/NC(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000217720187 FD For-Sale Unstable CA4 63 52 COc1ccccc1/C=C/NC(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000217720187 FD For-Sale Unstable CA5A 56 51 COc1ccccc1/C=C/NC(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000217720187 FD For-Sale Unstable CA14 47 49 COc1ccccc1/C=C/NC(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000217720187 FD For-Sale Unstable CA12 74 53 COc1ccccc1/C=C/NC(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000217720187 FD For-Sale Unstable CA9 81 53 COc1ccccc1/C=C/NC(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000217720187 FD For-Sale Unstable CYNT 24 43 COc1ccccc1/C=C/NC(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000217720187 FD For-Sale Unstable MTCA1 40 49 COc1ccccc1/C=C/NC(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000217720187 FD For-Sale Unstable P96878_MYCTU 51 49 CCOc1ccc([C@H](C)N[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217720247 CF For-Sale Unstable ACACA 25 41 COc1ccccc1/C=C/NC(=O)Nc1cccnc1Cl ZINC000217720291 DH For-Sale Unstable G2YM83_BOTF4 52 33 Cc1cccc(C(=O)O)c1OCC(=O)NCCc1ccccc1 ZINC000217720295 DE In-Stock Unstable CYSP_TRYCR 0 41 Cc1cccc(C(=O)O)c1OCC(=O)NCCc1ccccc1 ZINC000217720295 DE In-Stock Unstable CA5B 15 40 Cc1cccc(C(=O)O)c1OCC(=O)NCCc1ccccc1 ZINC000217720295 DE In-Stock Unstable NCE103 20 40 Cc1cccc(C(=O)O)c1OCC(=O)NCCc1ccccc1 ZINC000217720295 DE In-Stock Unstable O60989_PLAVI 0 40 Cc1cccc(C(=O)O)c1OCC(=O)NCCc1ccccc1 ZINC000217720295 DE In-Stock Unstable CAN2 0 40 CCOc1ccc([C@@H](C)N[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217720336 CF For-Sale Unstable ACACA 25 41 COC(=O)C[C@H](c1c(O)c2ccccc2oc1=O)c1cc2ccccc2n(C)c1=O ZINC000217720342 HG In-Stock Unstable NQO1 42 48 CCO[C@@H]1C[C@@H](NC(=O)Oc2ccccc2)C1(C)C ZINC000217720350 CF For-Sale Unstable TIMP3 57 33 CCO[C@@H]1C[C@@H](NC(=O)Oc2ccccc2)C1(C)C ZINC000217720350 CF For-Sale Unstable FAAH 25 40 COCCNC(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217720363 CD For-Sale Unstable DRD4 42 32 COCCNC(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217720363 CD For-Sale Unstable TNFRSF1A 28 45 COCCNC(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217720363 CD For-Sale Unstable ABCG2 15 47 O=C(/C=C\c1cccc(F)c1)NCC1CC(O)C1 ZINC000217720373 BD On-Demand Unstable HDAC8 51 37 O=C(/C=C\c1cccc(F)c1)NCC1CC(O)C1 ZINC000217720373 BD On-Demand Unstable MMP2 0 46 O=C(/C=C\c1cccc(F)c1)NCC1CC(O)C1 ZINC000217720373 BD On-Demand Unstable IMPDH2 0 44 O=C(/C=C\c1cccc(F)c1)NCC1CC(O)C1 ZINC000217720373 BD On-Demand Unstable MMP1 0 46 O=C(/C=C\c1cccc(F)c1)NCC1CC(O)C1 ZINC000217720373 BD On-Demand Unstable IMA1 0 44 CC[C@H](C(=O)O)N(C)C[C@@H](O)c1ccccc1 ZINC000217720379 BD On-Demand Unstable AOC3 32 53 O=C(NCC1C[C@@H]2CC[C@H](C1)N2)Nc1ccccc1 ZINC000217720383 CE For-Sale Unstable CCR3 34 43 O=C(NCC1C[C@@H]2CC[C@H](C1)N2)Nc1ccccc1 ZINC000217720383 CE For-Sale Unstable EPHX2 23 44 O=C(NCC1C[C@@H]2CC[C@H](C1)N2)Nc1ccccc1 ZINC000217720383 CE For-Sale Unstable NAMPT 17 43 CCC[C@@H]1CC[C@@H](NCC)[C@@H](CCCc2ccccc2)C1 ZINC000217720390 CK For-Sale Unstable SLC18A2 32 40 COc1ccccc1/C=C/NC(=O)N1C[C@@H](C)C[C@@H](C)C1 ZINC000217720395 CG For-Sale Unstable RORC 27 42 CCOc1ccc([C@H](C)N[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217720403 CF For-Sale Unstable ACACA 25 41 Cc1cccc(NC(=O)COc2c(C)cccc2C(=O)O)c1 ZINC000217720415 CG In-Stock Unstable CCKAR 22 40 Cc1cccc(NC(=O)COc2c(C)cccc2C(=O)O)c1 ZINC000217720415 CG In-Stock Unstable CETP 30 42 Cc1cccc(NC(=O)COc2c(C)cccc2C(=O)O)c1 ZINC000217720415 CG In-Stock Unstable F2R 0 46 Cc1cccc(NC(=O)COc2c(C)cccc2C(=O)O)c1 ZINC000217720415 CG In-Stock Unstable AKR1C3 26 48 Cc1cccc(NC(=O)COc2c(C)cccc2C(=O)O)c1 ZINC000217720415 CG In-Stock Unstable AKR1C2 41 48 Cc1cccc(NC(=O)COc2c(C)cccc2C(=O)O)c1 ZINC000217720415 CG In-Stock Unstable KCNK3 70 41 Cc1cccc(NC(=O)COc2c(C)cccc2C(=O)O)c1 ZINC000217720415 CG In-Stock Unstable KCNK9 81 44 COC(=O)C[C@@H](c1c(O)c2ccccc2oc1=O)c1cc2ccccc2n(C)c1=O ZINC000217720424 HG In-Stock Unstable NQO1 42 48 CCO[C@H]1C[C@@H](NC(=O)Oc2ccccc2)C1(C)C ZINC000217720450 CF For-Sale Unstable TIMP3 57 33 CCO[C@H]1C[C@@H](NC(=O)Oc2ccccc2)C1(C)C ZINC000217720450 CF For-Sale Unstable FAAH 25 40 CN(C(=O)c1ccc(/C=C\C(=O)O)s1)c1ccccc1 ZINC000217720452 CG For-Sale Unstable HSD17B2 48 49 CC[C@@H](C(=O)O)N(C)C[C@@H](O)c1ccccc1 ZINC000217720455 BD On-Demand Unstable AOC3 32 53 COc1ccc2c(c1)[C@@]1(C(=O)N2)[C@H](C(=O)c2ccc3c(c2)OCO3)[C@@H](c2ccc(F)cc2)CN1C ZINC000217720461 JH In-Stock Unstable EDNRB 67 39 COc1ccc2c(c1)[C@@]1(C(=O)N2)[C@H](C(=O)c2ccc3c(c2)OCO3)[C@@H](c2ccc(F)cc2)CN1C ZINC000217720461 JH In-Stock Unstable EDNRA 59 40 CCC[C@H]1CC[C@@H](NCC)[C@@H](CCCc2ccccc2)C1 ZINC000217720473 CK For-Sale Unstable SLC18A2 32 40 COc1ccccc1/C=C/NC(=O)N1C[C@H](C)C[C@@H](C)C1 ZINC000217720487 CG For-Sale Unstable RORC 27 42 Cc1ccc(NC(=O)COc2c(C)cccc2C(=O)O)cc1 ZINC000217720523 CG In-Stock Unstable CETP 50 46 Cc1ccc(NC(=O)COc2c(C)cccc2C(=O)O)cc1 ZINC000217720523 CG In-Stock Unstable AKR1C3 16 43 COc1ccc(C(=O)N(C)C(C)C)cc1/C=C\C(=O)O ZINC000217720529 CE For-Sale Unstable TNFRSF1A 28 42 CCO[C@@H]1C[C@H](NC(=O)Oc2ccccc2)C1(C)C ZINC000217720535 CF For-Sale Unstable TIMP3 57 33 CCO[C@@H]1C[C@H](NC(=O)Oc2ccccc2)C1(C)C ZINC000217720535 CF For-Sale Unstable FAAH 25 40 O=C1C[C@@H](c2cccc(O)c2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217720544 HI In-Stock Unstable AKR1B1 0 46 O=C1C[C@@H](c2cccc(O)c2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217720544 HI In-Stock Unstable CYP1B1 25 41 O=C1C[C@@H](c2cccc(O)c2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217720544 HI In-Stock Unstable CYP1A1 27 41 O=C1C[C@@H](c2cccc(O)c2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217720544 HI In-Stock Unstable CYP1A2 19 41 CCC[C@@H]1CC[C@H](NCC)[C@@H](CCCc2ccccc2)C1 ZINC000217720551 CK For-Sale Unstable SLC18A2 32 40 COc1ccccc1/C=C/NC(=O)N1C[C@@H](C)C[C@H](C)C1 ZINC000217720572 CG For-Sale Unstable RORC 27 42 CCO[C@H]1C[C@H](NC(=O)Oc2ccccc2)C1(C)C ZINC000217720605 CF For-Sale Unstable TIMP3 57 33 CCO[C@H]1C[C@H](NC(=O)Oc2ccccc2)C1(C)C ZINC000217720605 CF For-Sale Unstable FAAH 25 40 O=C(/C=C\c1ccc(Cl)cc1Cl)NCC1CC(O)C1 ZINC000217720612 DF For-Sale Unstable BOTA 35 60 NCCc1cc(Br)c(Cl)cc1F ZINC000217720621 CF For-Sale Unstable TAAR1 22 41 O=S(=O)(c1cccc2cnccc12)N1CCC(CCc2ccccc2)CC1 ZINC000217720623 GI On-Demand Unstable ROCK2 16 55 Cc1ccc2c(C(N)=O)n[nH]c2c1 ZINC000217720626 AC In-Stock Unstable ITK 29 44 CCC[C@H]1CC[C@H](NCC)[C@@H](CCCc2ccccc2)C1 ZINC000217720628 CK For-Sale Unstable SLC18A2 32 40 O=C1C[C@H](c2cccc(O)c2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217720631 HI In-Stock Unstable AKR1B1 0 46 O=C1C[C@H](c2cccc(O)c2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217720631 HI In-Stock Unstable CYP1B1 25 41 O=C1C[C@H](c2cccc(O)c2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217720631 HI In-Stock Unstable CYP1A1 27 41 O=C1C[C@H](c2cccc(O)c2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217720631 HI In-Stock Unstable CYP1A2 19 41 CCN1CC[C@H](CNC(=O)c2ccc(/C=C\C(=O)O)s2)C1 ZINC000217720633 DD For-Sale Unstable HTR4 47 35 CCN1CC[C@H](CNC(=O)c2ccc(/C=C\C(=O)O)s2)C1 ZINC000217720633 DD For-Sale Unstable CACNA1I 60 36 Cc1ccc(NC(=O)COc2c(C)cccc2C(=O)O)cc1C ZINC000217720635 DG In-Stock Unstable CETP 0 40 Cc1ccc(NC(=O)COc2c(C)cccc2C(=O)O)cc1C ZINC000217720635 DG In-Stock Unstable KCNK3 42 35 Cc1ccc(NC(=O)COc2c(C)cccc2C(=O)O)cc1C ZINC000217720635 DG In-Stock Unstable KCNK9 45 35 CCCN(CC)CCNCc1cccc(OCC#N)c1 ZINC000217720666 CE For-Sale Unstable SQLE 72 34 NCCc1cc(Cl)c(Br)cc1F ZINC000217720732 CF For-Sale Unstable TAAR1 20 41 CN1CC[C@H](CNC(=O)c2ccc(/C=C\C(=O)O)s2)C1 ZINC000217720736 CD For-Sale Unstable CACNA1I 54 36 COc1ccc(CCN2C(=O)N[C@@H](CC(=O)Nc3ccc4c(ccn4C)c3)C2=O)cc1OC ZINC000217720745 JF In-Stock Unstable ENPP1 74 35 Cc1cc(C)cc(NC(=O)COc2c(C)cccc2C(=O)O)c1 ZINC000217720762 DG In-Stock Unstable CETP 0 41 Cc1cc(C)cc(NC(=O)COc2c(C)cccc2C(=O)O)c1 ZINC000217720762 DG In-Stock Unstable AKR1C3 19 40 Cc1cc(C)cc(NC(=O)COc2c(C)cccc2C(=O)O)c1 ZINC000217720762 DG In-Stock Unstable AKR1C2 28 40 COc1ccccc1/C=C/NC(=O)Nc1ccccc1F ZINC000217720807 CH For-Sale Unstable TLR4 17 43 CN1CC[C@H](CNC(=O)c2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217720839 CD For-Sale Unstable CACNA1I 79 43 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccccc1F ZINC000217720868 DF In-Stock Unstable AKR1C3 15 43 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccccc1F ZINC000217720868 DF In-Stock Unstable AKR1C2 40 43 COc1ccccc1/C=C/NC(=O)N(C)c1ccccc1 ZINC000217720928 CH For-Sale Unstable TLR4 19 44 COc1ccc(C(=O)N2CC[C@@H](C)C2)cc1/C=C\C(=O)O ZINC000217720930 CE For-Sale Unstable L3MBTL3 50 34 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(F)cc1 ZINC000217720973 DF In-Stock Unstable CETP 0 45 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(F)cc1 ZINC000217720973 DF In-Stock Unstable GUAB 0 43 Cc1cc(C(C)(C)C)cc(C)c1S(=O)(=O)N1CCC[C@@H](O)C1 ZINC000217720974 EF On-Demand Unstable EPHX2 25 41 Cc1cc(C(C)(C)C)cc(C)c1S(=O)(=O)N1CCC[C@@H](O)C1 ZINC000217720974 EF On-Demand Unstable AKR1C3 22 50 COc1ccc(C(=O)N2CC[C@H](C)C2)cc1/C=C\C(=O)O ZINC000217721027 CE For-Sale Unstable L3MBTL3 50 34 Cc1cc(C(C)(C)C)cc(C)c1S(=O)(=O)N1CCC[C@H](O)C1 ZINC000217721045 EF On-Demand Unstable EPHX2 25 41 Cc1cc(C(C)(C)C)cc(C)c1S(=O)(=O)N1CCC[C@H](O)C1 ZINC000217721045 EF On-Demand Unstable AKR1C3 22 50 COc1ccccc1/C=C/NC(=O)N1CCCC1 ZINC000217721048 BE For-Sale Unstable DRD3 17 41 COc1ccccc1/C=C/NC(=O)N1CCCC1 ZINC000217721048 BE For-Sale Unstable TLR4 16 44 O=C1C/C(=C/c2ccc([N+](=O)[O-])cc2)C(=O)N1 ZINC000217721079 BD For-Sale Unstable RASGRP3 0 40 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccccc1Cl ZINC000217721084 DG In-Stock Unstable CXCL8 45 36 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccccc1Cl ZINC000217721084 DG In-Stock Unstable FABP2 0 42 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccccc1Cl ZINC000217721084 DG In-Stock Unstable HCAR2 32 41 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccccc1Cl ZINC000217721084 DG In-Stock Unstable EPHB3 41 34 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccccc1Cl ZINC000217721084 DG In-Stock Unstable AKR1C3 17 43 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccccc1Cl ZINC000217721084 DG In-Stock Unstable AKR1C2 44 43 O=C(COCc1ccccc1)NC[C@@H](c1ccccc1)N1CCCCC1 ZINC000217721099 FH In-Stock Unstable TACR1 15 44 O=C(COCc1ccccc1)NC[C@@H](c1ccccc1)N1CCCCC1 ZINC000217721099 FH In-Stock Unstable CCR3 29 40 CC(C)c1ccc(/C=C\C(=O)NCC2CC(O)C2)cc1 ZINC000217721110 CF For-Sale Unstable HDAC4 0 43 COc1ccccc1/C=C/NC(=O)N1CCCCCC1 ZINC000217721123 CG For-Sale Unstable DRD3 17 40 N[C@@H](Cc1cc(Oc2ccccc2)ccc1[N+](=O)[O-])C(=O)O ZINC000217721165 DE For-Sale Unstable THRA 19 41 N[C@@H](Cc1cc(Oc2ccccc2)ccc1[N+](=O)[O-])C(=O)O ZINC000217721165 DE For-Sale Unstable LTA4H 20 43 N[C@@H](Cc1cc(Oc2ccccc2)ccc1[N+](=O)[O-])C(=O)O ZINC000217721165 DE For-Sale Unstable COLA 72 34 Cc1cccc(C(=O)O)c1OCC(=O)Nc1cccc(Cl)c1 ZINC000217721183 DG In-Stock Unstable CETP 0 43 Cc1cccc(C(=O)O)c1OCC(=O)Nc1cccc(Cl)c1 ZINC000217721183 DG In-Stock Unstable F2R 0 44 Cc1cccc(C(=O)O)c1OCC(=O)Nc1cccc(Cl)c1 ZINC000217721183 DG In-Stock Unstable PTPN22 27 42 Cc1cccc(C(=O)O)c1OCC(=O)Nc1cccc(Cl)c1 ZINC000217721183 DG In-Stock Unstable MCHR1 16 41 Cc1cccc(C(=O)O)c1OCC(=O)Nc1cccc(Cl)c1 ZINC000217721183 DG In-Stock Unstable MCHR2 39 41 Cc1cccc(C(=O)O)c1OCC(=O)Nc1cccc(Cl)c1 ZINC000217721183 DG In-Stock Unstable AKR1C3 27 46 Cc1cccc(C(=O)O)c1OCC(=O)Nc1cccc(Cl)c1 ZINC000217721183 DG In-Stock Unstable AKR1C2 41 46 Cc1cccc(C(=O)O)c1OCC(=O)Nc1cccc(Cl)c1 ZINC000217721183 DG In-Stock Unstable IMDH_CRYPV 15 42 Cc1cccc(C(=O)O)c1OCC(=O)Nc1cccc(Cl)c1 ZINC000217721183 DG In-Stock Unstable PSBA 0 43 Cc1cccc(C(=O)O)c1OCC(=O)Nc1cccc(Cl)c1 ZINC000217721183 DG In-Stock Unstable KCNK3 56 40 Cc1cccc(C(=O)O)c1OCC(=O)Nc1cccc(Cl)c1 ZINC000217721183 DG In-Stock Unstable KCNK9 63 39 O=C(COCc1ccccc1)NC[C@H](c1ccccc1)N1CCCCC1 ZINC000217721186 FH In-Stock Unstable TACR1 15 44 O=C(COCc1ccccc1)NC[C@H](c1ccccc1)N1CCCCC1 ZINC000217721186 FH In-Stock Unstable CCR3 29 40 COc1ccccc1/C=C/NC(=O)NC[C@@H](C)O ZINC000217721240 CD For-Sale Unstable TLR4 15 44 CC[C@H](NC(=O)c1cccc(/C=C\C(=O)O)c1)C(C)C ZINC000217721283 CF For-Sale Unstable HDAC8 16 43 O=[N+]([O-])c1ccc(Oc2ccccc2)cc1CBr ZINC000217721284 DI For-Sale Unstable COLA 60 32 O=[N+]([O-])c1ccc(Oc2ccccc2)cc1CBr ZINC000217721284 DI For-Sale Unstable PQSD 0 40 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(Cl)cc1 ZINC000217721289 DG In-Stock Unstable CETP 0 45 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(Cl)cc1 ZINC000217721289 DG In-Stock Unstable GUAB 0 41 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(Cl)cc1 ZINC000217721289 DG In-Stock Unstable MCHR2 38 41 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(Cl)cc1 ZINC000217721289 DG In-Stock Unstable AKR1C2 37 42 COc1ccccc1/C=C/NC(=O)NC[C@H](C)O ZINC000217721307 CD For-Sale Unstable TLR4 15 44 COc1ccnc(CNC(=O)c2sccc2Cl)c1 ZINC000217721363 CF In-Stock Unstable MAP 0 53 CC[C@@H](NC(=O)c1cccc(/C=C\C(=O)O)c1)C(C)C ZINC000217721381 CF For-Sale Unstable HDAC8 16 43 CCNC(=O)N/C=C/c1ccccc1OC ZINC000217721391 BD For-Sale Unstable CYP1B1 23 42 Cc1cn(-c2cccnc2)c(=O)[nH]1 ZINC000217721431 AC For-Sale Unstable CYP2A6 29 53 CC[C@@H](N[C@@H]1CCN2CCC[C@@H]12)c1ccccc1O ZINC000217721432 CF For-Sale Unstable SLC18A3 42 35 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(Br)cc1 ZINC000217721452 FG In-Stock Unstable PRS 50 34 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(Br)cc1 ZINC000217721452 FG In-Stock Unstable CETP 0 45 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(Br)cc1 ZINC000217721452 FG In-Stock Unstable IMDH_CRYPV 15 40 CC[C@H](N[C@@H]1CCN2CCC[C@@H]12)c1ccccc1O ZINC000217721506 CF For-Sale Unstable SLC18A3 42 35 Cc1ccc(NC(=O)COc2c(C)cccc2C(=O)O)cc1Cl ZINC000217721532 EH In-Stock Unstable AVPR2 21 40 Cc1ccc(NC(=O)COc2c(C)cccc2C(=O)O)cc1Cl ZINC000217721532 EH In-Stock Unstable CETP 0 41 Cc1ccc(NC(=O)COc2c(C)cccc2C(=O)O)cc1Cl ZINC000217721532 EH In-Stock Unstable GRM4 22 40 Cc1ccc(NC(=O)COc2c(C)cccc2C(=O)O)cc1Cl ZINC000217721532 EH In-Stock Unstable MCHR1 16 40 Cc1ccc(NC(=O)COc2c(C)cccc2C(=O)O)cc1Cl ZINC000217721532 EH In-Stock Unstable MCHR2 41 42 COCCCNS(=O)(=O)c1ccccc1C(=O)OC ZINC000217721555 CC On-Demand Unstable PRTN3 44 32 CC[C@@H](N[C@H]1CCN2CCC[C@@H]12)c1ccccc1O ZINC000217721577 CF For-Sale Unstable SLC18A3 42 35 CCCCCNC(=O)N/C=C/c1ccccc1OC ZINC000217721595 CG For-Sale Unstable DRD2 18 47 CCCCCNC(=O)N/C=C/c1ccccc1OC ZINC000217721595 CG For-Sale Unstable DRD3 33 47 CCCCCNC(=O)N/C=C/c1ccccc1OC ZINC000217721595 CG For-Sale Unstable MTNR1A 18 48 CCCCCNC(=O)N/C=C/c1ccccc1OC ZINC000217721595 CG For-Sale Unstable MTNR1B 23 44 CCCCCNC(=O)N/C=C/c1ccccc1OC ZINC000217721595 CG For-Sale Unstable EPHX2 28 40 CCCCCNC(=O)N/C=C/c1ccccc1OC ZINC000217721595 CG For-Sale Unstable ASAH1 71 33 CCCCCNC(=O)N/C=C/c1ccccc1OC ZINC000217721595 CG For-Sale Unstable ACAT 0 56 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217721639 FI In-Stock Unstable AVPR2 17 40 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217721639 FI In-Stock Unstable CETP 0 43 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217721639 FI In-Stock Unstable GRM4 38 42 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217721639 FI In-Stock Unstable SLC1A2 23 40 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217721639 FI In-Stock Unstable MCHR1 23 43 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217721639 FI In-Stock Unstable MCHR2 42 43 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217721639 FI In-Stock Unstable IMDH_CRYPV 59 42 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217721639 FI In-Stock Unstable KCNK3 41 36 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217721639 FI In-Stock Unstable PPX1 0 40 CC[C@H](N[C@H]1CCN2CCC[C@@H]12)c1ccccc1O ZINC000217721665 CF For-Sale Unstable SLC18A3 42 35 CN1CC[C@H](NC(=O)c2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217721681 CD For-Sale Unstable DRD4 15 46 CN1CC[C@H](NC(=O)c2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217721681 CD For-Sale Unstable UTS2R 20 40 CN1CC[C@H](NC(=O)c2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217721681 CD For-Sale Unstable SLC6A5 35 45 COc1ccccc1/C=C/NC(=O)Nc1ccccc1 ZINC000217721719 CG For-Sale Unstable EPHX1 0 44 COc1ccccc1/C=C/NC(=O)Nc1ccccc1 ZINC000217721719 CG For-Sale Unstable CYP1B1 22 41 COc1ccccc1/C=C/NC(=O)Nc1ccccc1 ZINC000217721719 CG For-Sale Unstable TLR4 20 47 COc1ccccc1/C=C/NC(=O)Nc1ccccc1 ZINC000217721719 CG For-Sale Unstable P95276_MYCTO 0 44 COc1ccccc1/C=C/NC(=O)Nc1ccccc1 ZINC000217721719 CG For-Sale Unstable KCNK3 41 43 COc1ccccc1/C=C/NC(=O)Nc1ccccc1 ZINC000217721719 CG For-Sale Unstable KCNK9 35 41 Cc1cccc(C(=O)O)c1OCC(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000217721739 FI In-Stock Unstable CETP 0 42 Cc1cccc(C(=O)O)c1OCC(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000217721739 FI In-Stock Unstable MCHR1 18 40 COc1ccc([C@@H]2CC(=O)Oc3ccc4c(c32)OC(C)(C)CC4=O)cc1OC ZINC000217721768 GH In-Stock Unstable MT-ND4 50 31 CCOc1ccccc1[C@@H](C)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217721771 CF For-Sale Unstable HCN1 53 36 CCOc1ccccc1[C@@H](C)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217721771 CF For-Sale Unstable HCN4 46 36 COC(=O)c1ccccc1S(=O)(=O)NCC1CCCCC1 ZINC000217721811 DE On-Demand Unstable NPY1R 0 41 COC(=O)c1ccccc1S(=O)(=O)NCC1CCCCC1 ZINC000217721811 DE On-Demand Unstable NPY2R 119 42 COC(=O)c1ccccc1S(=O)(=O)NCC1CCCCC1 ZINC000217721811 DE On-Demand Unstable AMY2 42 29 COC(=O)c1ccccc1S(=O)(=O)NCC1CCCCC1 ZINC000217721811 DE On-Demand Unstable NPY5R 41 42 COC(=O)c1ccccc1S(=O)(=O)NCC1CCCCC1 ZINC000217721811 DE On-Demand Unstable PRTN3 43 31 CN1CC[C@H](NC(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217721814 CD For-Sale Unstable DRD4 22 45 CN1CC[C@H](NC(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217721814 CD For-Sale Unstable HDAC8 32 40 CN1CC[C@H](NC(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217721814 CD For-Sale Unstable UTS2R 19 40 CN1CC[C@H](NC(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217721814 CD For-Sale Unstable HDAC6 18 40 CN1CC[C@H](NC(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217721814 CD For-Sale Unstable SLC6A5 21 40 CCOC(=O)[C@@H]1CCCN(C(=O)N/C=C/c2ccccc2OC)C1 ZINC000217721824 EF For-Sale Unstable SLC6A1 57 38 CCOC(=O)[C@@H]1CCCN(C(=O)N/C=C/c2ccccc2OC)C1 ZINC000217721824 EF For-Sale Unstable FDFT1 26 45 Cc1cccc(C(=O)O)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217721851 FH In-Stock Unstable LCK 32 41 Cc1cccc(C(=O)O)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217721851 FH In-Stock Unstable UL80 23 41 Cc1cccc(C(=O)O)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217721851 FH In-Stock Unstable CETP 0 44 Cc1cccc(C(=O)O)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217721851 FH In-Stock Unstable KDR 17 43 Cc1cccc(C(=O)O)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217721851 FH In-Stock Unstable SLC1A1 21 43 Cc1cccc(C(=O)O)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217721851 FH In-Stock Unstable SLC1A3 19 43 Cc1cccc(C(=O)O)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217721851 FH In-Stock Unstable SLC1A2 33 43 Cc1cccc(C(=O)O)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217721851 FH In-Stock Unstable TEK 24 41 Cc1cccc(C(=O)O)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217721851 FH In-Stock Unstable MCHR1 21 44 Cc1cccc(C(=O)O)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217721851 FH In-Stock Unstable BTK 24 42 Cc1cccc(C(=O)O)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217721851 FH In-Stock Unstable AKR1C3 27 47 Cc1cccc(C(=O)O)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217721851 FH In-Stock Unstable AKR1C2 27 49 Cc1cccc(C(=O)O)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217721851 FH In-Stock Unstable TRPM4 0 49 Cc1cccc(C(=O)O)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217721851 FH In-Stock Unstable KCNK3 56 42 Cc1cccc(C(=O)O)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217721851 FH In-Stock Unstable KCNK9 60 38 Cc1cccc(C(=O)O)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217721851 FH In-Stock Unstable PDS 40 40 COc1ccc([C@H]2CC(=O)Oc3ccc4c(c32)OC(C)(C)CC4=O)cc1OC ZINC000217721855 GH In-Stock Unstable MT-ND4 50 31 CCOc1ccccc1[C@H](C)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217721857 CF For-Sale Unstable HCN1 53 36 CCOc1ccccc1[C@H](C)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217721857 CF For-Sale Unstable HCN4 46 36 CC(C)(C)OC(=O)C[C@H](N)C(=O)Nc1ccc(OCCNC(=O)OC(C)(C)C)cc1 ZINC000217721882 HF For-Sale Unstable LTA4H 20 42 CCOC(=O)[C@H]1CCCN(C(=O)N/C=C/c2ccccc2OC)C1 ZINC000217721901 EF For-Sale Unstable SLC6A1 57 38 CCOC(=O)[C@H]1CCCN(C(=O)N/C=C/c2ccccc2OC)C1 ZINC000217721901 EF For-Sale Unstable FDFT1 26 45 O=C(/C=C\c1cc(Cl)ccc1Cl)NCC1CC(O)C1 ZINC000217721930 DF For-Sale Unstable BOTA 25 47 CCOc1ccccc1[C@@H](C)N[C@H]1CCN2CCC[C@@H]12 ZINC000217721931 CF For-Sale Unstable HCN1 53 36 CCOc1ccccc1[C@@H](C)N[C@H]1CCN2CCC[C@@H]12 ZINC000217721931 CF For-Sale Unstable HCN4 46 36 COc1ccccc1NC(=O)COc1c(C)cccc1C(=O)O ZINC000217721955 DF In-Stock Unstable CETP 0 41 COc1ccccc1NC(=O)COc1c(C)cccc1C(=O)O ZINC000217721955 DF In-Stock Unstable AKR1C3 19 42 COc1ccccc1NC(=O)COc1c(C)cccc1C(=O)O ZINC000217721955 DF In-Stock Unstable AKR1C2 47 42 COc1ccccc1NC(=O)COc1c(C)cccc1C(=O)O ZINC000217721955 DF In-Stock Unstable KCNK3 45 39 CC[C@@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc([N+](=O)[O-])cc1 ZINC000217721989 HH On-Demand Unstable COLA 80 43 CC[C@@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc([N+](=O)[O-])cc1 ZINC000217721989 HH On-Demand Unstable MMP2 22 41 CC[C@@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc([N+](=O)[O-])cc1 ZINC000217721989 HH On-Demand Unstable MMP8 42 41 CC[C@@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc([N+](=O)[O-])cc1 ZINC000217721989 HH On-Demand Unstable MMP9 22 41 CC[C@@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc([N+](=O)[O-])cc1 ZINC000217721989 HH On-Demand Unstable MMP1 34 41 COc1ccccc1/C=C/NC(=O)Nc1ccc(CC(=O)O)cc1 ZINC000217722001 EG For-Sale Unstable TSHR 47 32 CCOc1ccccc1[C@H](C)N[C@H]1CCN2CCC[C@@H]12 ZINC000217722019 CF For-Sale Unstable HCN1 53 36 CCOc1ccccc1[C@H](C)N[C@H]1CCN2CCC[C@@H]12 ZINC000217722019 CF For-Sale Unstable HCN4 46 36 O=C(/C=C\c1ccccc1Cl)NCC1CC(O)C1 ZINC000217722027 CE On-Demand Unstable KCNQ2 21 41 O=C(/C=C\c1ccccc1Cl)NCC1CC(O)C1 ZINC000217722027 CE On-Demand Unstable BOTA 27 42 CC(C)[C@@H](NC(=O)CN1CCC[C@@H](CO)C1)c1cccs1 ZINC000217722061 DE For-Sale Unstable BIRC2 43 36 CC[C@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc([N+](=O)[O-])cc1 ZINC000217722072 HH On-Demand Unstable COLA 80 43 CC[C@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc([N+](=O)[O-])cc1 ZINC000217722072 HH On-Demand Unstable MMP2 22 41 CC[C@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc([N+](=O)[O-])cc1 ZINC000217722072 HH On-Demand Unstable MMP8 42 41 CC[C@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc([N+](=O)[O-])cc1 ZINC000217722072 HH On-Demand Unstable MMP9 22 41 CC[C@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc([N+](=O)[O-])cc1 ZINC000217722072 HH On-Demand Unstable MMP1 34 41 COc1cccc(NC(=O)COc2c(C)cccc2C(=O)O)c1 ZINC000217722073 DF In-Stock Unstable PDGFRB 18 42 COc1cccc(NC(=O)COc2c(C)cccc2C(=O)O)c1 ZINC000217722073 DF In-Stock Unstable CETP 0 43 COc1cccc(NC(=O)COc2c(C)cccc2C(=O)O)c1 ZINC000217722073 DF In-Stock Unstable MTNR1A 32 48 COc1cccc(NC(=O)COc2c(C)cccc2C(=O)O)c1 ZINC000217722073 DF In-Stock Unstable MTNR1B 32 47 COc1cccc(NC(=O)COc2c(C)cccc2C(=O)O)c1 ZINC000217722073 DF In-Stock Unstable FPR2 21 40 COc1cccc(NC(=O)COc2c(C)cccc2C(=O)O)c1 ZINC000217722073 DF In-Stock Unstable AKR1C3 37 51 COc1cccc(NC(=O)COc2c(C)cccc2C(=O)O)c1 ZINC000217722073 DF In-Stock Unstable AKR1C2 74 43 COc1cccc(NC(=O)COc2c(C)cccc2C(=O)O)c1 ZINC000217722073 DF In-Stock Unstable KCNK3 59 40 COc1cccc(NC(=O)COc2c(C)cccc2C(=O)O)c1 ZINC000217722073 DF In-Stock Unstable KCNK9 63 40 COc1ccccc1/C=C/NC(=O)Nc1c(F)cccc1F ZINC000217722127 DH For-Sale Unstable TLR4 17 43 CC(C)[C@H](NC(=O)CN1CCC[C@@H](CO)C1)c1cccs1 ZINC000217722136 DE For-Sale Unstable BIRC2 43 36 COc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)Nc1cccc(C(C)=O)c1)C(=O)OC2 ZINC000217722154 II In-Stock Unstable IMPDH1 0 71 COc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)Nc1cccc(C(C)=O)c1)C(=O)OC2 ZINC000217722154 II In-Stock Unstable IMPDH2 0 71 COc1ccc(NC(=O)COc2c(C)cccc2C(=O)O)cc1 ZINC000217722181 DF In-Stock Unstable CETP 0 46 COc1ccc(NC(=O)COc2c(C)cccc2C(=O)O)cc1 ZINC000217722181 DF In-Stock Unstable GUAB 0 43 COc1ccc(NC(=O)COc2c(C)cccc2C(=O)O)cc1 ZINC000217722181 DF In-Stock Unstable MTNR1A 34 44 COc1ccc(NC(=O)COc2c(C)cccc2C(=O)O)cc1 ZINC000217722181 DF In-Stock Unstable MTNR1B 32 48 COc1ccc(NC(=O)COc2c(C)cccc2C(=O)O)cc1 ZINC000217722181 DF In-Stock Unstable CA9 15 40 COc1ccc(NC(=O)COc2c(C)cccc2C(=O)O)cc1 ZINC000217722181 DF In-Stock Unstable AKR1C3 28 41 COc1ccc(NC(=O)COc2c(C)cccc2C(=O)O)cc1 ZINC000217722181 DF In-Stock Unstable AKR1C2 68 47 COc1ccc(NC(=O)COc2c(C)cccc2C(=O)O)cc1 ZINC000217722181 DF In-Stock Unstable IMDH_CRYPV 26 40 O=c1oc2c(O)nncc2n1Cc1ccccc1 ZINC000217722228 BD In-Stock Unstable MIF 19 46 Cc1ccc([C@@H](C)NC(=O)c2ccc(/C=C\C(=O)O)s2)s1 ZINC000217722242 DH For-Sale Unstable UL26 19 41 Cc1ccc([C@@H](C)NC(=O)c2ccc(/C=C\C(=O)O)s2)s1 ZINC000217722242 DH For-Sale Unstable SCAF_EBVB9 25 41 COc1cc(C)c(F)c(CS(=O)(=O)Cl)c1 ZINC000217722287 CE For-Sale Unstable FFAR4 17 40 CCOc1ccccc1NC(=O)COc1c(C)cccc1C(=O)O ZINC000217722310 EG In-Stock Unstable AKR1C2 29 41 CCOc1ccccc1NC(=O)COc1c(C)cccc1C(=O)O ZINC000217722310 EG In-Stock Unstable HCN1 41 32 CCOc1ccccc1NC(=O)COc1c(C)cccc1C(=O)O ZINC000217722310 EG In-Stock Unstable HCN4 41 32 CCOc1ccccc1NC(=O)COc1c(C)cccc1C(=O)O ZINC000217722310 EG In-Stock Unstable KCNK3 38 40 CCOc1ccccc1NC(=O)COc1c(C)cccc1C(=O)O ZINC000217722310 EG In-Stock Unstable KCNK9 33 40 Cc1ccc([C@H](C)NC(=O)c2ccc(/C=C\C(=O)O)s2)s1 ZINC000217722353 DH For-Sale Unstable UL26 19 41 Cc1ccc([C@H](C)NC(=O)c2ccc(/C=C\C(=O)O)s2)s1 ZINC000217722353 DH For-Sale Unstable SCAF_EBVB9 25 41 CCc1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217722356 CI For-Sale Unstable MTNR1B 15 46 CCc1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217722356 CI For-Sale Unstable ACR 19 43 CC[C@@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1cc([N+](=O)[O-])ccc1C ZINC000217722364 IH On-Demand Unstable COLA 52 36 O=C(Nc1ccc(C(=O)O)cc1)OCCCc1ccccc1 ZINC000217722374 CH For-Sale Unstable FKBP1A 37 51 O=C(Nc1ccc(C(=O)O)cc1)OCCCc1ccccc1 ZINC000217722374 CH For-Sale Unstable LTA4H 48 47 O=C(Nc1ccc(C(=O)O)cc1)OCCCc1ccccc1 ZINC000217722374 CH For-Sale Unstable CA1 18 40 O=C(Nc1ccc(C(=O)O)cc1)OCCCc1ccccc1 ZINC000217722374 CH For-Sale Unstable HRH3 17 52 O=C(Nc1ccc(C(=O)O)cc1)OCCCc1ccccc1 ZINC000217722374 CH For-Sale Unstable CTSK 15 47 O=C(Nc1ccc(C(=O)O)cc1)OCCCc1ccccc1 ZINC000217722374 CH For-Sale Unstable S1PR4 19 42 O=C(Nc1ccc(C(=O)O)cc1)OCCCc1ccccc1 ZINC000217722374 CH For-Sale Unstable HDAC8 15 44 O=C(Nc1ccc(C(=O)O)cc1)OCCCc1ccccc1 ZINC000217722374 CH For-Sale Unstable S1PR3 18 42 O=C(Nc1ccc(C(=O)O)cc1)OCCCc1ccccc1 ZINC000217722374 CH For-Sale Unstable PLA2G4B 34 48 O=C(Nc1ccc(C(=O)O)cc1)OCCCc1ccccc1 ZINC000217722374 CH For-Sale Unstable HDAC2 17 40 O=C(Nc1ccc(C(=O)O)cc1)OCCCc1ccccc1 ZINC000217722374 CH For-Sale Unstable FAAH 46 40 O=C(Nc1ccc(C(=O)O)cc1)OCCCc1ccccc1 ZINC000217722374 CH For-Sale Unstable S1PR1 15 42 O=C(Nc1ccc(C(=O)O)cc1)OCCCc1ccccc1 ZINC000217722374 CH For-Sale Unstable SPHK1 23 45 O=C(Nc1ccc(C(=O)O)cc1)OCCCc1ccccc1 ZINC000217722374 CH For-Sale Unstable S1PR5 21 42 O=C(Nc1ccc(C(=O)O)cc1)OCCCc1ccccc1 ZINC000217722374 CH For-Sale Unstable ACR 54 40 O=C(Nc1ccc(C(=O)O)cc1)OCCCc1ccccc1 ZINC000217722374 CH For-Sale Unstable NAAA 49 48 O=C(Nc1ccc(C(=O)O)cc1)OCCCc1ccccc1 ZINC000217722374 CH For-Sale Unstable NCE103 23 40 O=C(Nc1ccc(C(=O)O)cc1)OCCCc1ccccc1 ZINC000217722374 CH For-Sale Unstable AKR1B10 21 42 CCOc1ccc(NC(=O)COc2c(C)cccc2C(=O)O)cc1 ZINC000217722427 EG In-Stock Unstable ADORA2B 42 36 CCOc1ccc(NC(=O)COc2c(C)cccc2C(=O)O)cc1 ZINC000217722427 EG In-Stock Unstable CETP 0 41 CCOc1ccc(NC(=O)COc2c(C)cccc2C(=O)O)cc1 ZINC000217722427 EG In-Stock Unstable PLA2G4B 45 33 CCOc1ccc(NC(=O)COc2c(C)cccc2C(=O)O)cc1 ZINC000217722427 EG In-Stock Unstable P4HTM 0 45 CCOc1ccc(NC(=O)COc2c(C)cccc2C(=O)O)cc1 ZINC000217722427 EG In-Stock Unstable NR5A1 16 41 CC[C@@H]1CCCN1S(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217722434 DE For-Sale Unstable CASP3 98 39 CC[C@@H]1CCCN1S(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217722434 DE For-Sale Unstable CASP7 111 40 CC[C@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1cc([N+](=O)[O-])ccc1C ZINC000217722436 IH On-Demand Unstable COLA 52 36 COC(=O)C[C@@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(O)c(OC)c1 ZINC000217722446 GF In-Stock Unstable PNLIP 0 42 COC(=O)C[C@@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(O)c(OC)c1 ZINC000217722446 GF In-Stock Unstable FOLH1 0 40 COC(=O)C[C@@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(O)c(OC)c1 ZINC000217722446 GF In-Stock Unstable TNF 22 42 COC(=O)C[C@@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(O)c(OC)c1 ZINC000217722446 GF In-Stock Unstable N1L 0 43 COC(=O)C[C@@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(O)c(OC)c1 ZINC000217722446 GF In-Stock Unstable SLC22A3 0 40 COC(=O)C[C@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(O)c(OC)c1 ZINC000217722521 GF In-Stock Unstable PNLIP 0 42 COC(=O)C[C@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(O)c(OC)c1 ZINC000217722521 GF In-Stock Unstable FOLH1 0 40 COC(=O)C[C@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(O)c(OC)c1 ZINC000217722521 GF In-Stock Unstable TNF 22 42 COC(=O)C[C@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(O)c(OC)c1 ZINC000217722521 GF In-Stock Unstable N1L 0 43 COC(=O)C[C@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(O)c(OC)c1 ZINC000217722521 GF In-Stock Unstable SLC22A3 0 40 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccccn1 ZINC000217722526 CD For-Sale Unstable GRM4 44 38 CC[C@H]1CCCN1S(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217722529 DE For-Sale Unstable CASP3 98 39 CC[C@H]1CCCN1S(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217722529 DE For-Sale Unstable CASP7 111 40 CC[C@@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc(OC)cc1 ZINC000217722533 HH On-Demand Unstable BMP1 118 46 CC[C@@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc(OC)cc1 ZINC000217722533 HH On-Demand Unstable MMP13 54 47 CC[C@@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc(OC)cc1 ZINC000217722533 HH On-Demand Unstable ADAM17 27 40 CC[C@@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc(OC)cc1 ZINC000217722533 HH On-Demand Unstable COLA 20 40 CC[C@@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc(OC)cc1 ZINC000217722533 HH On-Demand Unstable MMP16 0 41 CC[C@@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc(OC)cc1 ZINC000217722533 HH On-Demand Unstable MMP2 38 47 CC[C@@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc(OC)cc1 ZINC000217722533 HH On-Demand Unstable MMP3 39 47 CC[C@@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc(OC)cc1 ZINC000217722533 HH On-Demand Unstable MMP8 42 45 CC[C@@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc(OC)cc1 ZINC000217722533 HH On-Demand Unstable MMP14 16 45 CC[C@@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc(OC)cc1 ZINC000217722533 HH On-Demand Unstable MMP9 50 47 CC[C@@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc(OC)cc1 ZINC000217722533 HH On-Demand Unstable MMP12 34 45 CC[C@@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc(OC)cc1 ZINC000217722533 HH On-Demand Unstable MMP7 15 42 CC[C@@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc(OC)cc1 ZINC000217722533 HH On-Demand Unstable MMP1 40 47 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217722543 GJ In-Stock Unstable LTA4H 56 45 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217722543 GJ In-Stock Unstable CA1 34 42 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217722543 GJ In-Stock Unstable ACOX1 27 41 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217722543 GJ In-Stock Unstable CETP 0 43 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217722543 GJ In-Stock Unstable SCN2A 15 43 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217722543 GJ In-Stock Unstable GUAB 0 42 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217722543 GJ In-Stock Unstable MTNR1A 16 46 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217722543 GJ In-Stock Unstable MTNR1B 15 50 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217722543 GJ In-Stock Unstable NPY5R 0 43 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217722543 GJ In-Stock Unstable PDGFRA 31 40 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217722543 GJ In-Stock Unstable FABH 0 40 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217722543 GJ In-Stock Unstable AKR1C2 48 38 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217722543 GJ In-Stock Unstable PFKFB3 40 33 COc1ccccc1/C=C/NC(=O)NC1CC(C)(C)NC(C)(C)C1 ZINC000217722594 EG For-Sale Unstable EZH2 61 44 CC(C)n1cnnc1-c1cccnc1 ZINC000217722601 AD For-Sale Unstable CYP2A6 52 41 CC[C@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc(OC)cc1 ZINC000217722613 HH On-Demand Unstable BMP1 118 46 CC[C@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc(OC)cc1 ZINC000217722613 HH On-Demand Unstable MMP13 54 47 CC[C@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc(OC)cc1 ZINC000217722613 HH On-Demand Unstable ADAM17 27 40 CC[C@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc(OC)cc1 ZINC000217722613 HH On-Demand Unstable COLA 20 40 CC[C@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc(OC)cc1 ZINC000217722613 HH On-Demand Unstable MMP16 0 41 CC[C@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc(OC)cc1 ZINC000217722613 HH On-Demand Unstable MMP2 38 47 CC[C@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc(OC)cc1 ZINC000217722613 HH On-Demand Unstable MMP3 39 47 CC[C@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc(OC)cc1 ZINC000217722613 HH On-Demand Unstable MMP8 42 45 CC[C@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc(OC)cc1 ZINC000217722613 HH On-Demand Unstable MMP14 16 45 CC[C@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc(OC)cc1 ZINC000217722613 HH On-Demand Unstable MMP9 50 47 CC[C@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc(OC)cc1 ZINC000217722613 HH On-Demand Unstable MMP12 34 45 CC[C@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc(OC)cc1 ZINC000217722613 HH On-Demand Unstable MMP7 15 42 CC[C@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc(OC)cc1 ZINC000217722613 HH On-Demand Unstable MMP1 40 47 O=C(NC[C@H]1CCCN1c1nccs1)c1ccccn1 ZINC000217722615 CD For-Sale Unstable GRM4 44 38 CCN1CCC[C@@H]1CN(C)c1ccc(Cl)cc1CBr ZINC000217722616 EI For-Sale Unstable NOS2 16 40 CCN1CCC[C@@H]1CN(C)c1ccc(Cl)cc1CBr ZINC000217722616 EI For-Sale Unstable NOS3 18 40 COc1ccc(NC(=O)COc2c(C)cccc2C(=O)O)c(OC)c1 ZINC000217722654 EF In-Stock Unstable DHODH 15 41 COc1ccc(NC(=O)COc2c(C)cccc2C(=O)O)c(OC)c1 ZINC000217722654 EF In-Stock Unstable AKR1C3 26 41 COc1ccc(NC(=O)COc2c(C)cccc2C(=O)O)c(OC)c1 ZINC000217722654 EF In-Stock Unstable AKR1C2 64 41 CCN1CCC[C@H]1CN(C)c1ccc(Cl)cc1CBr ZINC000217722692 EI For-Sale Unstable NOS2 16 40 CCN1CCC[C@H]1CN(C)c1ccc(Cl)cc1CBr ZINC000217722692 EI For-Sale Unstable NOS3 18 40 COc1ccccc1/C=C/NC(=O)Nc1cc(C)ccc1O ZINC000217722723 CH For-Sale Unstable KCNMA1 24 47 C[C@@H]1CCCN1S(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217722798 CD For-Sale Unstable CASP3 41 35 C[C@@H]1CCCN1S(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217722798 CD For-Sale Unstable HDAC8 30 40 C[C@@H]1CCCN1S(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217722798 CD For-Sale Unstable CASP7 51 34 C[C@@H]1CCCN1S(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217722798 CD For-Sale Unstable AKR1C3 47 42 COc1ccccc1/C=C/NC(=O)N1CCN(CCO)CC1 ZINC000217722842 DC For-Sale Unstable HTR1A 68 41 COc1ccccc1/C=C/NC(=O)N1CCN(CCO)CC1 ZINC000217722842 DC For-Sale Unstable DRD2 47 48 COc1ccccc1/C=C/NC(=O)N1CCN(CCO)CC1 ZINC000217722842 DC For-Sale Unstable DRD4 40 31 COc1ccccc1/C=C/NC(=O)N1CCN(CCO)CC1 ZINC000217722842 DC For-Sale Unstable DRD3 59 48 COc1ccccc1/C=C/NC(=O)N1CCN(CCO)CC1 ZINC000217722842 DC For-Sale Unstable HTR7 50 39 COc1ccc(NC(=O)COc2c(C)cccc2C(=O)O)cc1Cl ZINC000217722852 EG In-Stock Unstable CETP 0 41 COc1ccc(NC(=O)COc2c(C)cccc2C(=O)O)cc1Cl ZINC000217722852 EG In-Stock Unstable GRM4 21 47 COc1ccc(NC(=O)COc2c(C)cccc2C(=O)O)cc1Cl ZINC000217722852 EG In-Stock Unstable MCHR2 41 44 COc1ccc(NC(=O)COc2c(C)cccc2C(=O)O)cc1Cl ZINC000217722852 EG In-Stock Unstable AKR1C2 46 34 COc1ccc(NC(=O)COc2c(C)cccc2C(=O)O)cc1Cl ZINC000217722852 EG In-Stock Unstable ENPP1 58 35 COc1ccc(NC(=O)COc2c(C)cccc2C(=O)O)cc1Cl ZINC000217722852 EG In-Stock Unstable KCNK3 44 38 CC[C@@H](N[C@@H]1CCN2CCC[C@@H]12)c1ccc(OC)cc1 ZINC000217722856 CF For-Sale Unstable CHRM2 22 41 O=C(c1ccc(F)cc1Cl)N1CC(N2C(=O)[C@H]3CC=CC[C@H]3C2=O)C1 ZINC000217722875 FE In-Stock Unstable P2RX7 22 51 C[C@H]1CCCN1S(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217722885 CD For-Sale Unstable CASP3 41 35 C[C@H]1CCCN1S(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217722885 CD For-Sale Unstable HDAC8 30 40 C[C@H]1CCCN1S(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217722885 CD For-Sale Unstable CASP7 51 34 C[C@H]1CCCN1S(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217722885 CD For-Sale Unstable AKR1C3 47 42 Cc1ccccc1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217722930 DF For-Sale Unstable AVPR2 27 42 Cc1ccccc1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217722930 DF For-Sale Unstable HCRTR1 33 40 Cc1ccccc1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217722930 DF For-Sale Unstable HCRTR2 16 40 Cc1ccccc1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217722930 DF For-Sale Unstable CCR8 50 33 CC[C@H](N[C@@H]1CCN2CCC[C@@H]12)c1ccc(OC)cc1 ZINC000217722941 CF For-Sale Unstable CHRM2 22 41 COc1ccccc1/C=C/NC(=O)N1CCC[C@@H](C)C1 ZINC000217722946 CG For-Sale Unstable RORC 38 41 COc1ccccc1/C=C/NC(=O)N1CCC[C@@H](C)C1 ZINC000217722946 CG For-Sale Unstable ACKR3 62 32 COC(=O)c1ccccc1NC(=O)COc1c(C)cccc1C(=O)O ZINC000217722951 EE In-Stock Unstable HCAR2 36 40 COC(=O)c1ccccc1NC(=O)COc1c(C)cccc1C(=O)O ZINC000217722951 EE In-Stock Unstable AKR1C3 16 43 COC(=O)c1ccccc1NC(=O)COc1c(C)cccc1C(=O)O ZINC000217722951 EE In-Stock Unstable AKR1C2 43 43 COC(=O)c1ccccc1NC(=O)COc1c(C)cccc1C(=O)O ZINC000217722951 EE In-Stock Unstable FAS 49 52 O=C(c1ccc(F)cc1Cl)N1CC(N2C(=O)[C@H]3CC=CC[C@@H]3C2=O)C1 ZINC000217722960 FE In-Stock Unstable P2RX7 22 51 Cc1ccccc1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217723018 DF For-Sale Unstable AVPR2 27 42 Cc1ccccc1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217723018 DF For-Sale Unstable HCRTR1 33 40 Cc1ccccc1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217723018 DF For-Sale Unstable HCRTR2 16 40 Cc1ccccc1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217723018 DF For-Sale Unstable CCR8 50 33 CC[C@@H](N[C@H]1CCN2CCC[C@@H]12)c1ccc(OC)cc1 ZINC000217723022 CF For-Sale Unstable CHRM2 22 41 COc1ccccc1/C=C/NC(=O)N1CCC[C@H](C)C1 ZINC000217723037 CG For-Sale Unstable RORC 38 41 COc1ccccc1/C=C/NC(=O)N1CCC[C@H](C)C1 ZINC000217723037 CG For-Sale Unstable ACKR3 62 32 O=C(c1ccc(F)cc1Cl)N1CC(N2C(=O)[C@@H]3CC=CC[C@H]3C2=O)C1 ZINC000217723047 FE In-Stock Unstable P2RX7 26 51 COC(=O)c1ccc(NC(=O)COc2c(C)cccc2C(=O)O)cc1 ZINC000217723070 EE In-Stock Unstable CETP 0 48 COC(=O)c1ccc(NC(=O)COc2c(C)cccc2C(=O)O)cc1 ZINC000217723070 EE In-Stock Unstable ACR 60 42 CC[C@H](N[C@H]1CCN2CCC[C@@H]12)c1ccc(OC)cc1 ZINC000217723108 CF For-Sale Unstable CHRM2 22 41 COC[C@H](C)NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217723137 CD For-Sale Unstable HDAC8 15 45 COC[C@H](C)NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217723137 CD For-Sale Unstable LEF 18 41 COc1ccccc1/C=C/NC(=O)Nc1ccc(C)c(C)c1 ZINC000217723142 CI For-Sale Unstable GRM4 15 43 COc1ccccc1/C=C/NC(=O)Nc1ccc(C)c(C)c1 ZINC000217723142 CI For-Sale Unstable IMPDH2 0 45 COc1ccccc1/C=C/NC(=O)Nc1ccc(C)c(C)c1 ZINC000217723142 CI For-Sale Unstable KCNK3 44 42 COc1ccccc1/C=C/NC(=O)Nc1ccc(C)c(C)c1 ZINC000217723142 CI For-Sale Unstable KCNK9 47 40 CCOC(=O)CN1CCN(c2ccc(Br)cc2)CC1 ZINC000217723152 EE On-Demand Unstable CCR1 22 43 CCOC(=O)c1ccc(NC(=O)COc2c(C)cccc2C(=O)O)cc1 ZINC000217723172 FF In-Stock Unstable CETP 0 42 CCCOc1ccc([C@@H](C)N[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217723218 CG For-Sale Unstable ACACA 41 47 CCCOc1ccc([C@@H](C)N[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217723218 CG For-Sale Unstable ACACB 22 47 COC[C@@H](C)NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217723224 CD For-Sale Unstable HDAC8 15 45 COC[C@@H](C)NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217723224 CD For-Sale Unstable LEF 18 41 CCN(Cc1ccccc1)C(=O)N/C=C/c1ccccc1OC ZINC000217723264 DH For-Sale Unstable PTGES 20 42 O=C(/C=C\c1cccnc1)Nc1cc(C(=O)O)ccn1 ZINC000217723268 CD For-Sale Anodyne TBXAS1 16 40 O=C(/C=C\c1cccnc1)Nc1cc(C(=O)O)ccn1 ZINC000217723268 CD For-Sale Anodyne MMP2 18 41 O=C(/C=C\c1cccnc1)Nc1cc(C(=O)O)ccn1 ZINC000217723268 CD For-Sale Anodyne MMP9 15 41 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217723278 FD In-Stock Unstable CA2 115 48 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217723278 FD In-Stock Unstable CA1 99 48 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217723278 FD In-Stock Unstable CA7 54 50 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217723278 FD In-Stock Unstable CETP 0 40 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217723278 FD In-Stock Unstable CA5B 66 50 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217723278 FD In-Stock Unstable CA4 97 48 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217723278 FD In-Stock Unstable CA5A 77 50 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217723278 FD In-Stock Unstable CA14 43 41 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217723278 FD In-Stock Unstable CA12 76 47 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217723278 FD In-Stock Unstable CA9 91 45 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217723278 FD In-Stock Unstable TTK 21 41 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217723278 FD In-Stock Unstable UREA_CANEN 27 44 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217723278 FD In-Stock Unstable NCE103 48 40 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217723278 FD In-Stock Unstable MTCA1 41 45 Cc1cccc(C(=O)O)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217723278 FD In-Stock Unstable P96878_MYCTU 57 45 COC[C@H](C)NS(=O)(=O)c1ccc(/C=C\C(=O)O)c(C)c1 ZINC000217723306 DD For-Sale Unstable LEF 60 41 CCCOc1ccc([C@H](C)N[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217723317 CG For-Sale Unstable ACACA 41 47 CCCOc1ccc([C@H](C)N[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217723317 CG For-Sale Unstable ACACB 22 47 Cc1cc(C)cc(S(=O)(=O)Nc2cccnc2Cl)c1 ZINC000217723321 CG For-Sale Unstable PIK3CA 21 41 Cc1cc(C)cc(S(=O)(=O)Nc2cccnc2Cl)c1 ZINC000217723321 CG For-Sale Unstable GRM4 19 41 Cc1cc(C)cc(S(=O)(=O)Nc2cccnc2Cl)c1 ZINC000217723321 CG For-Sale Unstable CCR2 0 43 Cc1cc(C)cc(S(=O)(=O)Nc2cccnc2Cl)c1 ZINC000217723321 CG For-Sale Unstable NFKBIA 0 41 Cc1cc(C)cc(S(=O)(=O)Nc2cccnc2Cl)c1 ZINC000217723321 CG For-Sale Unstable C0L093_TOBAC 49 36 Cc1cc(C)cc(S(=O)(=O)Nc2cccnc2Cl)c1 ZINC000217723321 CG For-Sale Unstable G2YM83_BOTF4 44 32 COc1ccc(N2C[C@]34C=C[C@@H](O3)[C@@H](C(=O)Nc3nccs3)[C@H]4C2=O)cc1 ZINC000217723325 GE In-Stock Unstable MAP1 59 37 COc1ccc(/C=C(\CO)CCO)cc1 ZINC000217723337 BD For-Sale Unstable CYP1B1 25 41 COc1ccc(/C=C(\CO)CCO)cc1 ZINC000217723337 BD For-Sale Unstable CYP1A1 21 41 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccccc1F ZINC000217723358 DF For-Sale Unstable MAP1 15 40 CC(=O)c1cccc(NC(=O)COc2c(C)cccc2C(=O)O)c1 ZINC000217723388 EF In-Stock Unstable CETP 0 43 CC(=O)c1cccc(NC(=O)COc2c(C)cccc2C(=O)O)c1 ZINC000217723388 EF In-Stock Unstable F2R 0 44 CC(=O)c1cccc(NC(=O)COc2c(C)cccc2C(=O)O)c1 ZINC000217723388 EF In-Stock Unstable HIF1A 16 44 CC(=O)c1cccc(NC(=O)COc2c(C)cccc2C(=O)O)c1 ZINC000217723388 EF In-Stock Unstable AKR1C3 52 50 CC(=O)c1cccc(NC(=O)COc2c(C)cccc2C(=O)O)c1 ZINC000217723388 EF In-Stock Unstable AKR1C2 46 36 CC(=O)c1cccc(NC(=O)COc2c(C)cccc2C(=O)O)c1 ZINC000217723388 EF In-Stock Unstable KCNK3 86 45 CC(=O)c1cccc(NC(=O)COc2c(C)cccc2C(=O)O)c1 ZINC000217723388 EF In-Stock Unstable KCNK9 79 40 CC(=O)c1cccc(NC(=O)COc2c(C)cccc2C(=O)O)c1 ZINC000217723388 EF In-Stock Unstable PARP10 0 42 COC[C@@H](C)NS(=O)(=O)c1ccc(/C=C\C(=O)O)c(C)c1 ZINC000217723394 DD For-Sale Unstable LEF 60 41 COC(=O)[C@@H](O)CNC(=O)CCn1cncn1 ZINC000217723403 BA For-Sale Unstable HIS3 79 38 CCCOc1ccc([C@@H](C)N[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217723409 CG For-Sale Unstable ACACA 41 47 CCCOc1ccc([C@@H](C)N[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217723409 CG For-Sale Unstable ACACB 22 47 COc1ccc(N2C[C@]34C=C[C@@H](O3)[C@H](C(=O)Nc3nccs3)[C@H]4C2=O)cc1 ZINC000217723417 GE In-Stock Unstable MAP1 59 37 Cc1ccc(/C=C\C(=O)NCC2CC(O)C2)cc1Cl ZINC000217723434 CF For-Sale Unstable PYGL 0 51 Cc1ccc(/C=C\C(=O)NCC2CC(O)C2)cc1Cl ZINC000217723434 CF For-Sale Unstable CCR2 0 42 O=C(NC[C@H]1CCCN1c1nccs1)c1ccccc1F ZINC000217723446 DF For-Sale Unstable MAP1 15 40 COC(=O)[C@H](O)CNC(=O)CCn1cncn1 ZINC000217723473 BA For-Sale Unstable HIS3 79 38 Cc1ccc(/C=C\C(=O)O)cc1S(=O)(=O)N1CCSCC1 ZINC000217723476 ED For-Sale Unstable CNR2 0 48 CCCOc1ccc([C@H](C)N[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217723499 CG For-Sale Unstable ACACA 41 47 CCCOc1ccc([C@H](C)N[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217723499 CG For-Sale Unstable ACACB 22 47 O=C(COc1cc(Cl)ccc1C(=O)O)Nc1ccccc1Cl ZINC000217723528 EH In-Stock Unstable KCNQ2 28 40 O=C(COc1cc(Cl)ccc1C(=O)O)Nc1ccccc1Cl ZINC000217723528 EH In-Stock Unstable CETP 0 44 O=C(COc1cc(Cl)ccc1C(=O)O)Nc1ccccc1Cl ZINC000217723528 EH In-Stock Unstable PYGL 24 40 O=C(COc1cc(Cl)ccc1C(=O)O)Nc1ccccc1Cl ZINC000217723528 EH In-Stock Unstable PYGM 25 43 O=C(COc1cc(Cl)ccc1C(=O)O)Nc1ccccc1Cl ZINC000217723528 EH In-Stock Unstable HCAR2 27 40 O=C(COc1cc(Cl)ccc1C(=O)O)Nc1ccccc1Cl ZINC000217723528 EH In-Stock Unstable POBA 0 40 O=C(COc1cc(Cl)ccc1C(=O)O)Nc1ccccc1Cl ZINC000217723528 EH In-Stock Unstable PTGDR2 26 43 O=C(COc1cc(Cl)ccc1C(=O)O)Nc1ccccc1Cl ZINC000217723528 EH In-Stock Unstable EPHB3 41 33 O=C(COc1cc(Cl)ccc1C(=O)O)Nc1ccccc1Cl ZINC000217723528 EH In-Stock Unstable AKR1C3 18 42 O=C(COc1cc(Cl)ccc1C(=O)O)Nc1ccccc1Cl ZINC000217723528 EH In-Stock Unstable AKR1C2 41 42 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccc(F)cc1 ZINC000217723568 DF For-Sale Unstable HCRTR1 19 45 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccc(F)cc1 ZINC000217723568 DF For-Sale Unstable PLA2G4A 40 32 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccc(F)cc1 ZINC000217723568 DF For-Sale Unstable HCRTR2 15 45 CC[C@@H]1CCCCN1C(=O)N/C=C/c1ccccc1OC ZINC000217723584 CH For-Sale Unstable FKBP1A 47 36 CC[C@@H]1CCCCN1C(=O)N/C=C/c1ccccc1OC ZINC000217723584 CH For-Sale Unstable ACKR3 65 34 O=C(NC[C@H]1CCCN1c1nccs1)c1ccc(F)cc1 ZINC000217723643 DF For-Sale Unstable HCRTR1 19 45 O=C(NC[C@H]1CCCN1c1nccs1)c1ccc(F)cc1 ZINC000217723643 DF For-Sale Unstable PLA2G4A 40 32 O=C(NC[C@H]1CCCN1c1nccs1)c1ccc(F)cc1 ZINC000217723643 DF For-Sale Unstable HCRTR2 15 45 O=C(O)/C=C\c1ccc(S(=O)(=O)NCC2CCC2)c(Cl)c1 ZINC000217723656 EF For-Sale Unstable NPY1R 40 31 COCc1n[nH]c(-c2ccc(NC(=O)CCCC[C@@H]3CCSS3)cc2)n1 ZINC000217723663 GI In-Stock Unstable PTPN2 0 55 CC[C@H]1CCCCN1C(=O)N/C=C/c1ccccc1OC ZINC000217723669 CH For-Sale Unstable FKBP1A 47 36 CC[C@H]1CCCCN1C(=O)N/C=C/c1ccccc1OC ZINC000217723669 CH For-Sale Unstable ACKR3 65 34 CCCCCCCCNC[C@@H](O)CCC ZINC000217723670 BG For-Sale Unstable S1PR3 18 41 CCCCCCCCNC[C@@H](O)CCC ZINC000217723670 BG For-Sale Unstable S1PR2 44 41 CCCCCCCCNC[C@@H](O)CCC ZINC000217723670 BG For-Sale Unstable Q8WS26_TRYCR 45 52 CCCCCCCCNC[C@@H](O)CCC ZINC000217723670 BG For-Sale Unstable CQSS 45 38 CCOC(=O)c1ccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)cc1 ZINC000217723682 GG In-Stock Unstable P2RY12 22 43 CCOC(=O)c1ccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)cc1 ZINC000217723682 GG In-Stock Unstable ADORA2B 21 43 CCOC(=O)c1ccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)cc1 ZINC000217723682 GG In-Stock Unstable CETP 0 43 CCOC(=O)c1ccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)cc1 ZINC000217723682 GG In-Stock Unstable COLA 62 36 CCOC(=O)c1ccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)cc1 ZINC000217723682 GG In-Stock Unstable CPT1A 60 36 CCOC(=O)c1ccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)cc1 ZINC000217723682 GG In-Stock Unstable CPT2 46 35 CCOC(=O)c1ccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)cc1 ZINC000217723682 GG In-Stock Unstable ACR 60 40 CCOC(=O)c1ccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)cc1 ZINC000217723682 GG In-Stock Unstable CPT1B 45 34 CCOC(=O)c1ccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)cc1 ZINC000217723682 GG In-Stock Unstable MCHR1 16 41 CCOC(=O)c1ccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)cc1 ZINC000217723682 GG In-Stock Unstable MCHR2 35 40 CCOC(=O)c1ccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)cc1 ZINC000217723682 GG In-Stock Unstable SENP1 0 42 CCOC(=O)c1ccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)cc1 ZINC000217723682 GG In-Stock Unstable PSBA 0 42 COc1cc(Br)ccc1C(=O)N1CC[C@H]2CC[C@@H](C1)N2C ZINC000217723705 FF On-Demand Unstable L3MBTL3 42 35 COCc1n[nH]c(-c2ccc(NC(=O)CCCC[C@H]3CCSS3)cc2)n1 ZINC000217723754 GI In-Stock Unstable PTPN2 0 55 CN(C(=O)c1ccc(/C=C\C(=O)O)cc1)C1CCCC1 ZINC000217723760 CF For-Sale Unstable ACE 43 40 CCCCCCCCNC[C@H](O)CCC ZINC000217723763 BG For-Sale Unstable S1PR3 18 41 CCCCCCCCNC[C@H](O)CCC ZINC000217723763 BG For-Sale Unstable S1PR2 44 41 CCCCCCCCNC[C@H](O)CCC ZINC000217723763 BG For-Sale Unstable Q8WS26_TRYCR 45 52 CCCCCCCCNC[C@H](O)CCC ZINC000217723763 BG For-Sale Unstable CQSS 45 38 COc1ccccc1/C=C/NC(=O)N(Cc1ccccc1)Cc1ccccc1 ZINC000217723772 FK For-Sale Unstable PTGER2 23 40 COc1ccccc1/C=C/NC(=O)N(Cc1ccccc1)Cc1ccccc1 ZINC000217723772 FK For-Sale Unstable PTGES 25 42 COc1ccccc1/C=C/NC(=O)N(Cc1ccccc1)Cc1ccccc1 ZINC000217723772 FK For-Sale Unstable LIMK2 18 41 COc1ccccc1/C=C/NC(=O)N(Cc1ccccc1)Cc1ccccc1 ZINC000217723772 FK For-Sale Unstable AKR1B10 29 41 NCc1ccc(C(=O)N[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217723781 CD For-Sale Unstable SSTR3 28 42 NCc1ccc(C(=O)N[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217723781 CD For-Sale Unstable PLAU 15 41 NCc1ccc(C(=O)N[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217723781 CD For-Sale Unstable L3MBTL3 53 35 NS(=O)(=O)c1ccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)cc1 ZINC000217723811 GD In-Stock Unstable CA2 106 45 NS(=O)(=O)c1ccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)cc1 ZINC000217723811 GD In-Stock Unstable CA1 94 45 NS(=O)(=O)c1ccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)cc1 ZINC000217723811 GD In-Stock Unstable CA7 53 47 NS(=O)(=O)c1ccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)cc1 ZINC000217723811 GD In-Stock Unstable CETP 0 42 NS(=O)(=O)c1ccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)cc1 ZINC000217723811 GD In-Stock Unstable COLA 57 35 NS(=O)(=O)c1ccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)cc1 ZINC000217723811 GD In-Stock Unstable CPT1A 59 35 NS(=O)(=O)c1ccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)cc1 ZINC000217723811 GD In-Stock Unstable CPT2 45 33 NS(=O)(=O)c1ccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)cc1 ZINC000217723811 GD In-Stock Unstable CA5B 62 47 NS(=O)(=O)c1ccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)cc1 ZINC000217723811 GD In-Stock Unstable CA4 95 43 NS(=O)(=O)c1ccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)cc1 ZINC000217723811 GD In-Stock Unstable CA5A 71 47 NS(=O)(=O)c1ccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)cc1 ZINC000217723811 GD In-Stock Unstable CA14 43 39 NS(=O)(=O)c1ccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)cc1 ZINC000217723811 GD In-Stock Unstable CA12 78 50 NS(=O)(=O)c1ccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)cc1 ZINC000217723811 GD In-Stock Unstable CPT1B 42 33 NS(=O)(=O)c1ccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)cc1 ZINC000217723811 GD In-Stock Unstable CA9 91 45 NS(=O)(=O)c1ccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)cc1 ZINC000217723811 GD In-Stock Unstable UREA_CANEN 26 42 NS(=O)(=O)c1ccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)cc1 ZINC000217723811 GD In-Stock Unstable NCE103 43 42 NS(=O)(=O)c1ccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)cc1 ZINC000217723811 GD In-Stock Unstable PFK 0 41 NS(=O)(=O)c1ccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)cc1 ZINC000217723811 GD In-Stock Unstable MTCA1 40 43 NS(=O)(=O)c1ccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)cc1 ZINC000217723811 GD In-Stock Unstable P96878_MYCTU 57 50 CCCN(C(=O)c1ccc(/C=C\C(=O)O)cc1)C1CC1 ZINC000217723843 CF For-Sale Unstable MBTPS1 62 35 C=C(C)C(=O)N(CCO)Cc1ccccc1 ZINC000217723846 BD For-Sale Unstable LIMK2 42 48 NCc1ccc(C(=O)N[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217723855 CD For-Sale Unstable SSTR3 28 42 NCc1ccc(C(=O)N[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217723855 CD For-Sale Unstable PLAU 15 41 NCc1ccc(C(=O)N[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217723855 CD For-Sale Unstable L3MBTL3 53 35 COC(=O)C1CC2(C1)NC(=O)NC2=O ZINC000217723873 AB In-Stock Unstable PYGB 43 32 COc1ccccc1/C=C/NC(=O)N(CCO)Cc1ccccc1 ZINC000217723906 EF For-Sale Unstable PTGES 0 41 CCCN(C(=O)c1cccc(/C=C\C(=O)O)c1)C1CC1 ZINC000217723923 CF For-Sale Unstable ACE 32 41 CC(=O)c1cccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)c1 ZINC000217723926 EG In-Stock Unstable PTGER1 31 42 CC(=O)c1cccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)c1 ZINC000217723926 EG In-Stock Unstable CETP 0 41 CC(=O)c1cccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)c1 ZINC000217723926 EG In-Stock Unstable COLA 41 36 CC(=O)c1cccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)c1 ZINC000217723926 EG In-Stock Unstable CPT1A 44 31 CC(=O)c1cccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)c1 ZINC000217723926 EG In-Stock Unstable GUAB 0 41 CC(=O)c1cccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)c1 ZINC000217723926 EG In-Stock Unstable PTPN22 23 41 CC(=O)c1cccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)c1 ZINC000217723926 EG In-Stock Unstable MCHR1 17 40 CC(=O)c1cccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)c1 ZINC000217723926 EG In-Stock Unstable MCHR2 39 41 CC(=O)c1cccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)c1 ZINC000217723926 EG In-Stock Unstable HIF1A 23 44 CC(=O)c1cccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)c1 ZINC000217723926 EG In-Stock Unstable AKR1C3 53 45 CC(=O)c1cccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)c1 ZINC000217723926 EG In-Stock Unstable AKR1C2 52 44 CC(=O)c1cccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)c1 ZINC000217723926 EG In-Stock Unstable IMDH_CRYPV 15 41 CC(=O)c1cccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)c1 ZINC000217723926 EG In-Stock Unstable KCNK3 67 42 CC(=O)c1cccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)c1 ZINC000217723926 EG In-Stock Unstable KCNK9 63 40 CC(=O)c1cccc(NC(=O)COc2cc(Cl)ccc2C(=O)O)c1 ZINC000217723926 EG In-Stock Unstable PARP10 0 41 C[C@@H](N[C@@H]1CCN2CCC[C@@H]12)c1cccc(Cl)c1 ZINC000217723982 CG For-Sale Unstable OPRL1 0 40 O=C(/C=C/c1ccc2c(c1)OCO2)N1CC(N2C(=O)[C@H]3CC=CC[C@H]3C2=O)C1 ZINC000217724006 GD In-Stock Unstable DYRK2 46 31 COc1ccc(C(=O)Nc2nccs2)cc1/C=C\C(=O)O ZINC000217724007 DF For-Sale Unstable MAP1 133 44 COc1ccc(C(=O)Nc2nccs2)cc1/C=C\C(=O)O ZINC000217724007 DF For-Sale Unstable CPT1A 29 42 COc1ccc(C(=O)Nc2nccs2)cc1/C=C\C(=O)O ZINC000217724007 DF For-Sale Unstable TNFRSF1A 29 41 COc1ccc(C(=O)Nc2nccs2)cc1/C=C\C(=O)O ZINC000217724007 DF For-Sale Unstable MAPKAPK2 15 41 COc1ccc(NC(=O)N/C=C/c2ccccc2OC)c(OC)c1 ZINC000217724022 EH For-Sale Unstable CYP1B1 50 55 COc1ccc(NC(=O)N/C=C/c2ccccc2OC)c(OC)c1 ZINC000217724022 EH For-Sale Unstable MTNR1A 28 47 COc1ccc(NC(=O)N/C=C/c2ccccc2OC)c(OC)c1 ZINC000217724022 EH For-Sale Unstable MTNR1B 27 47 COc1ccc(NC(=O)N/C=C/c2ccccc2OC)c(OC)c1 ZINC000217724022 EH For-Sale Unstable CYP1A1 42 43 COc1ccc(NC(=O)N/C=C/c2ccccc2OC)c(OC)c1 ZINC000217724022 EH For-Sale Unstable ABCG2 17 40 COc1ccc(NC(=O)N/C=C/c2ccccc2OC)c(OC)c1 ZINC000217724022 EH For-Sale Unstable AKR1C2 48 33 CC(C)CCNC(=O)CN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12 ZINC000217724039 GF In-Stock Unstable PSMB5 15 41 C[C@H](N[C@@H]1CCN2CCC[C@@H]12)c1cccc(Cl)c1 ZINC000217724057 CG For-Sale Unstable OPRL1 0 40 Cc1ccc(C(=O)O)c(OCC(=O)Nc2ccccc2Cl)c1 ZINC000217724064 DG In-Stock Unstable CXCL8 42 35 Cc1ccc(C(=O)O)c(OCC(=O)Nc2ccccc2Cl)c1 ZINC000217724064 DG In-Stock Unstable PYGL 21 40 Cc1ccc(C(=O)O)c(OCC(=O)Nc2ccccc2Cl)c1 ZINC000217724064 DG In-Stock Unstable PYGM 23 40 Cc1ccc(C(=O)O)c(OCC(=O)Nc2ccccc2Cl)c1 ZINC000217724064 DG In-Stock Unstable EPHB3 43 40 Cc1ccc(C(=O)O)c(OCC(=O)Nc2ccccc2Cl)c1 ZINC000217724064 DG In-Stock Unstable AKR1C2 54 38 CN(C(=O)c1cccc(/C=C\C(=O)O)c1)c1ccccc1 ZINC000217724101 CG For-Sale Unstable HDAC8 18 42 CN(C(=O)c1cccc(/C=C\C(=O)O)c1)c1ccccc1 ZINC000217724101 CG For-Sale Unstable NR1H4 27 40 CN(C(=O)c1cccc(/C=C\C(=O)O)c1)c1ccccc1 ZINC000217724101 CG For-Sale Unstable TTR 0 40 CN(C(=O)c1cccc(/C=C\C(=O)O)c1)c1ccccc1 ZINC000217724101 CG For-Sale Unstable HSD17B2 30 43 CN(C(=O)c1cccc(/C=C\C(=O)O)c1)c1ccccc1 ZINC000217724101 CG For-Sale Unstable RHOA 0 40 O=C(/C=C/c1ccc2c(c1)OCO2)N1CC(N2C(=O)[C@H]3CC=CC[C@@H]3C2=O)C1 ZINC000217724116 GD In-Stock Unstable DYRK2 41 30 COc1ccccc1/C=C/NC(=O)Nc1cc(C)on1 ZINC000217724128 CF For-Sale Unstable CYP1B1 19 41 CC(C)CCNC(=O)CN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12 ZINC000217724138 GF In-Stock Unstable PSMB5 15 41 C[C@@H](N[C@H]1CCN2CCC[C@@H]12)c1cccc(Cl)c1 ZINC000217724145 CG For-Sale Unstable OPRL1 0 40 O=C(Cc1cccs1)NC[C@@H]1CCCN1c1nccs1 ZINC000217724157 DF For-Sale Unstable ADAM17 18 44 COC(=O)[C@@H](O)CNC(=O)Cc1cccs1 ZINC000217724164 BB On-Demand Unstable ADAM17 0 40 COC(=O)[C@@H](O)CNC(=O)Cc1cccs1 ZINC000217724164 BB On-Demand Unstable CA5B 38 48 COC(=O)[C@@H](O)CNC(=O)Cc1cccs1 ZINC000217724164 BB On-Demand Unstable CA5A 36 48 COC(=O)[C@@H](O)CNC(=O)Cc1cccs1 ZINC000217724164 BB On-Demand Unstable CTSC 32 44 Nc1ccc(C(=O)N[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217724166 BD For-Sale Unstable SLC18A3 27 46 Nc1ccc(C(=O)N[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217724166 BD For-Sale Unstable L3MBTL3 62 35 O=C(/C=C/c1ccc2c(c1)OCO2)N1CC(N2C(=O)[C@@H]3CC=CC[C@H]3C2=O)C1 ZINC000217724197 GD In-Stock Unstable DYRK2 46 31 CCOC(=O)c1ccc(NC(=O)COc2cc(C)ccc2C(=O)O)cc1 ZINC000217724203 FF In-Stock Unstable CETP 0 42 CN1CC[C@H](CNC(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217724211 CD For-Sale Unstable DRD4 41 31 CN1CC[C@H](CNC(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217724211 CD For-Sale Unstable HDAC8 40 40 CN1CC[C@H](CNC(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217724211 CD For-Sale Unstable HDAC1 21 40 CN1CC[C@H](CNC(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217724211 CD For-Sale Unstable HDAC6 21 40 CN1CC[C@H](CNC(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217724211 CD For-Sale Unstable CACNA1I 76 48 CN1CC[C@H](CNC(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217724211 CD For-Sale Unstable ACKR3 50 34 C[C@H](N[C@H]1CCN2CCC[C@@H]12)c1cccc(Cl)c1 ZINC000217724235 CG For-Sale Unstable OPRL1 0 40 O=C(Cc1cccs1)NC[C@H]1CCCN1c1nccs1 ZINC000217724239 DF For-Sale Unstable ADAM17 18 44 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)cc1C ZINC000217724243 DI For-Sale Unstable PYGL 15 43 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)cc1C ZINC000217724243 DI For-Sale Unstable H9CNL0_SPOEX 0 40 COC(=O)[C@H](O)CNC(=O)Cc1cccs1 ZINC000217724245 BB On-Demand Unstable ADAM17 0 40 COC(=O)[C@H](O)CNC(=O)Cc1cccs1 ZINC000217724245 BB On-Demand Unstable CA5B 38 48 COC(=O)[C@H](O)CNC(=O)Cc1cccs1 ZINC000217724245 BB On-Demand Unstable CA5A 36 48 COC(=O)[C@H](O)CNC(=O)Cc1cccs1 ZINC000217724245 BB On-Demand Unstable CTSC 32 44 Nc1ccc(C(=O)N[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217724246 BD For-Sale Unstable SLC18A3 27 46 Nc1ccc(C(=O)N[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217724246 BD For-Sale Unstable L3MBTL3 62 35 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)N1CCSCC1)C(=O)OC2 ZINC000217724253 HH In-Stock Unstable IMPDH1 0 67 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)N1CCSCC1)C(=O)OC2 ZINC000217724253 HH In-Stock Unstable IMPDH2 0 67 CC[C@@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc(C)c([N+](=O)[O-])c1 ZINC000217724276 IH On-Demand Unstable COLA 97 40 NC(=O)CCCNC(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217724297 CC For-Sale Unstable HDAC6 15 42 NC(=O)CCCNC(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217724297 CC For-Sale Unstable HDA106 0 47 Cc1ccc(C(=O)O)c(OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217724304 FD In-Stock Unstable CA2 114 45 Cc1ccc(C(=O)O)c(OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217724304 FD In-Stock Unstable CA1 100 45 Cc1ccc(C(=O)O)c(OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217724304 FD In-Stock Unstable CA7 59 47 Cc1ccc(C(=O)O)c(OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217724304 FD In-Stock Unstable CETP 0 42 Cc1ccc(C(=O)O)c(OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217724304 FD In-Stock Unstable CA5B 60 47 Cc1ccc(C(=O)O)c(OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217724304 FD In-Stock Unstable CA4 102 45 Cc1ccc(C(=O)O)c(OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217724304 FD In-Stock Unstable CA5A 69 47 Cc1ccc(C(=O)O)c(OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217724304 FD In-Stock Unstable CA14 48 44 Cc1ccc(C(=O)O)c(OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217724304 FD In-Stock Unstable CA12 79 47 Cc1ccc(C(=O)O)c(OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217724304 FD In-Stock Unstable CA9 95 47 Cc1ccc(C(=O)O)c(OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217724304 FD In-Stock Unstable UREA_CANEN 26 42 Cc1ccc(C(=O)O)c(OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217724304 FD In-Stock Unstable MTCA1 44 38 Cc1ccc(C(=O)O)c(OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217724304 FD In-Stock Unstable P96878_MYCTU 63 45 COc1ccccc1/C=C/NC(=O)NCCCO ZINC000217724345 CD For-Sale Unstable DRD2 17 45 COc1ccccc1/C=C/NC(=O)NCCCO ZINC000217724345 CD For-Sale Unstable DRD3 29 45 COc1cccc(CN[C@@H]2CCN3CCC[C@@H]23)c1OC ZINC000217724351 CE For-Sale Unstable TACR3 25 42 CC[C@H](C)N(CC(=O)Nc1cccc(C)c1C)S(=O)(=O)c1ccc(C)c([N+](=O)[O-])c1 ZINC000217724367 IH On-Demand Unstable COLA 97 40 CCOc1ccccc1/C=C\C(=O)NCC1CC(O)C1 ZINC000217724395 CD For-Sale Unstable HCN1 48 31 CCOc1ccccc1/C=C\C(=O)NCC1CC(O)C1 ZINC000217724395 CD For-Sale Unstable HCN4 41 31 C[C@@H]1CCN(C(=O)c2cc(/C=C\C(=O)O)ccc2F)C1 ZINC000217724405 CE For-Sale Unstable CCR2 49 39 CC(=O)c1cccc(NC(=O)COc2cc(C)ccc2C(=O)O)c1 ZINC000217724437 EF In-Stock Unstable CETP 0 43 CC(=O)c1cccc(NC(=O)COc2cc(C)ccc2C(=O)O)c1 ZINC000217724437 EF In-Stock Unstable PYGL 0 40 CC(=O)c1cccc(NC(=O)COc2cc(C)ccc2C(=O)O)c1 ZINC000217724437 EF In-Stock Unstable HIF1A 24 45 CC(=O)c1cccc(NC(=O)COc2cc(C)ccc2C(=O)O)c1 ZINC000217724437 EF In-Stock Unstable AKR1C3 52 46 CC(=O)c1cccc(NC(=O)COc2cc(C)ccc2C(=O)O)c1 ZINC000217724437 EF In-Stock Unstable AKR1C2 45 40 CC(=O)c1cccc(NC(=O)COc2cc(C)ccc2C(=O)O)c1 ZINC000217724437 EF In-Stock Unstable KCNK3 84 42 CC(=O)c1cccc(NC(=O)COc2cc(C)ccc2C(=O)O)c1 ZINC000217724437 EF In-Stock Unstable KCNK9 81 42 CC(=O)c1cccc(NC(=O)COc2cc(C)ccc2C(=O)O)c1 ZINC000217724437 EF In-Stock Unstable PARP10 0 42 COc1cccc(CN[C@H]2CCN3CCC[C@@H]23)c1OC ZINC000217724444 CE For-Sale Unstable TACR3 25 42 O=C(/C=C\c1ccc(Cl)cc1)Nc1cnccc1C(=O)O ZINC000217724459 DG For-Sale Anodyne LTB4R 0 52 O=C(/C=C\c1ccc(Cl)cc1)Nc1cnccc1C(=O)O ZINC000217724459 DG For-Sale Anodyne MMP2 0 50 O=C(/C=C\c1ccc(Cl)cc1)Nc1cnccc1C(=O)O ZINC000217724459 DG For-Sale Anodyne HDAC1 0 45 O=C(/C=C\c1ccc(Cl)cc1)Nc1cnccc1C(=O)O ZINC000217724459 DG For-Sale Anodyne MMP9 0 50 O=C(/C=C\c1ccc(Cl)cc1)Nc1cnccc1C(=O)O ZINC000217724459 DG For-Sale Anodyne HPSE 41 39 O=C(/C=C\c1ccc(Cl)cc1)Nc1cnccc1C(=O)O ZINC000217724459 DG For-Sale Anodyne MMP1 23 50 O=C(/C=C\c1ccc(Cl)cc1)Nc1cnccc1C(=O)O ZINC000217724459 DG For-Sale Anodyne TRPM2 0 44 CCC[C@@H](O)CNCCCSC ZINC000217724469 AD For-Sale Unstable SPPS 43 38 C[C@H]1CCN(C(=O)c2cc(/C=C\C(=O)O)ccc2F)C1 ZINC000217724491 CE For-Sale Unstable CCR2 49 39 COc1ccc(Br)c(C(=O)N2CC[C@H]3CC[C@@H](C2)N3C)c1 ZINC000217724513 FF On-Demand Unstable L3MBTL3 40 38 COC(=O)[C@H](Cc1ccccc1)NC(=O)CC/C(C)=C/Cc1c(OC)c(C)c2c(c1OC)C(=O)OC2 ZINC000217724553 JH In-Stock Unstable IMPDH1 0 89 COC(=O)[C@H](Cc1ccccc1)NC(=O)CC/C(C)=C/Cc1c(OC)c(C)c2c(c1OC)C(=O)OC2 ZINC000217724553 JH In-Stock Unstable IMPDH2 0 89 COC(=O)[C@H](Cc1ccccc1)NC(=O)CC/C(C)=C/Cc1c(OC)c(C)c2c(c1OC)C(=O)OC2 ZINC000217724553 JH In-Stock Unstable HDA106 0 45 CCC[C@H](O)CNCCCSC ZINC000217724559 AD For-Sale Unstable SPPS 43 38 C[C@@H]1CCN(C(=O)c2ccc(/C=C\C(=O)O)cc2F)C1 ZINC000217724570 CE For-Sale Unstable CCR2 61 39 COC(=O)[C@@H](O)CNC(=O)CCOc1ccccc1 ZINC000217724575 CC On-Demand Unstable LTA4H 37 43 COC(=O)[C@@H](O)CNC(=O)CCOc1ccccc1 ZINC000217724575 CC On-Demand Unstable PLA2G4B 49 33 CCOC(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724595 EF In-Stock Unstable PRSS1 16 46 CCOC(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724595 EF In-Stock Unstable SRD5A2 26 40 CCOC(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724595 EF In-Stock Unstable PPIA 16 42 CCOC(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724595 EF In-Stock Unstable ADORA2A 0 49 CCOC(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724595 EF In-Stock Unstable ADORA2B 42 38 CCOC(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724595 EF In-Stock Unstable TRY1_BOVIN 19 44 CCOC(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724595 EF In-Stock Unstable CETP 0 42 CCOC(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724595 EF In-Stock Unstable MTNR1B 20 40 CCOC(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724595 EF In-Stock Unstable PLA2G4B 62 47 CCOC(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724595 EF In-Stock Unstable P4HTM 0 41 CCOC(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724595 EF In-Stock Unstable ACR 67 46 CCOC(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724595 EF In-Stock Unstable HIF1A 25 45 CCOC(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724595 EF In-Stock Unstable AKR1C3 33 40 CCOC(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724595 EF In-Stock Unstable NOD2 17 40 CCOC(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724595 EF In-Stock Unstable SENP1 0 47 C/C=C\C(=O)Nc1cc(C(=O)O)ccn1 ZINC000217724619 BD For-Sale Unstable KDM4C 0 45 C/C=C\C(=O)Nc1cc(C(=O)O)ccn1 ZINC000217724619 BD For-Sale Unstable KDM3A 0 45 C/C=C\C(=O)Nc1cc(C(=O)O)ccn1 ZINC000217724619 BD For-Sale Unstable KDM5C 0 45 C/C=C\C(=O)Nc1cc(C(=O)O)ccn1 ZINC000217724619 BD For-Sale Unstable FTO 0 45 C[C@H]1CCN(C(=O)c2ccc(/C=C\C(=O)O)cc2F)C1 ZINC000217724633 CE For-Sale Unstable CCR2 61 39 COC(=O)[C@H](O)CNC(=O)CCOc1ccccc1 ZINC000217724651 CC On-Demand Unstable LTA4H 37 43 COC(=O)[C@H](O)CNC(=O)CCOc1ccccc1 ZINC000217724651 CC On-Demand Unstable PLA2G4B 49 33 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc(F)c2)CC(=O)O4)cc1O ZINC000217724664 II In-Stock Unstable AKR1B1 0 46 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc(F)c2)CC(=O)O4)cc1O ZINC000217724664 II In-Stock Unstable CYP1B1 76 46 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc(F)c2)CC(=O)O4)cc1O ZINC000217724664 II In-Stock Unstable CYP1A1 61 46 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc(F)c2)CC(=O)O4)cc1O ZINC000217724664 II In-Stock Unstable CYP1A2 45 46 CC(=O)Cc1oc2ccccc2c1Br ZINC000217724665 CG For-Sale Unstable CYP2C9 18 45 CC(=O)Cc1oc2ccccc2c1Br ZINC000217724665 CG For-Sale Unstable AKR1C1 15 45 CC(=O)Cc1oc2ccccc2c1Br ZINC000217724665 CG For-Sale Unstable SLC22A12 33 45 CCCCN(CCCC)C(=O)N/C=C/c1ccccc1OC ZINC000217724672 DI For-Sale Unstable ACAT 0 41 NS(=O)(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724708 FD In-Stock Unstable CA2 131 58 NS(=O)(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724708 FD In-Stock Unstable PRSS1 17 51 NS(=O)(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724708 FD In-Stock Unstable PPIA 16 40 NS(=O)(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724708 FD In-Stock Unstable F10 22 51 NS(=O)(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724708 FD In-Stock Unstable LTA4H 35 44 NS(=O)(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724708 FD In-Stock Unstable CA6 20 43 NS(=O)(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724708 FD In-Stock Unstable CA1 120 58 NS(=O)(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724708 FD In-Stock Unstable CA7 71 52 NS(=O)(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724708 FD In-Stock Unstable CA13 29 44 NS(=O)(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724708 FD In-Stock Unstable CA5B 70 52 NS(=O)(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724708 FD In-Stock Unstable CA4 116 58 NS(=O)(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724708 FD In-Stock Unstable CA5A 75 52 NS(=O)(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724708 FD In-Stock Unstable CA14 52 43 NS(=O)(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724708 FD In-Stock Unstable PLA2G4B 41 43 NS(=O)(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724708 FD In-Stock Unstable CDK1 0 40 NS(=O)(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724708 FD In-Stock Unstable CA12 82 50 NS(=O)(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724708 FD In-Stock Unstable CA9 99 53 NS(=O)(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724708 FD In-Stock Unstable F13A1 41 36 NS(=O)(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724708 FD In-Stock Unstable HIF1A 24 46 NS(=O)(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724708 FD In-Stock Unstable AKR1C3 37 42 NS(=O)(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724708 FD In-Stock Unstable UREA_CANEN 30 52 NS(=O)(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724708 FD In-Stock Unstable CYNT 41 42 NS(=O)(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724708 FD In-Stock Unstable NCE103 55 43 NS(=O)(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724708 FD In-Stock Unstable PFK 0 44 NS(=O)(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724708 FD In-Stock Unstable MTCA1 44 44 NS(=O)(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724708 FD In-Stock Unstable P96878_MYCTU 58 44 NS(=O)(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724708 FD In-Stock Unstable CA 0 43 NS(=O)(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724708 FD In-Stock Unstable SMG1 18 40 NS(=O)(=O)c1ccc(NC(=O)COc2cccc(C(=O)O)c2)cc1 ZINC000217724708 FD In-Stock Unstable Q5TU56_ANOGA 0 43 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc(F)c2)CC(=O)O4)cc1O ZINC000217724740 II In-Stock Unstable AKR1B1 0 46 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc(F)c2)CC(=O)O4)cc1O ZINC000217724740 II In-Stock Unstable CYP1B1 76 46 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc(F)c2)CC(=O)O4)cc1O ZINC000217724740 II In-Stock Unstable CYP1A1 61 46 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc(F)c2)CC(=O)O4)cc1O ZINC000217724740 II In-Stock Unstable CYP1A2 45 46 CCN(CC)CCCNC(=O)N/C=C/c1ccccc1OC ZINC000217724774 DF For-Sale Unstable ACHE 19 43 CCN(CC)CCCNC(=O)N/C=C/c1ccccc1OC ZINC000217724774 DF For-Sale Unstable DRD3 21 42 CCN(CC)CCCNC(=O)N/C=C/c1ccccc1OC ZINC000217724774 DF For-Sale Unstable BCHE 15 44 CN(Cc1nccs1)C(=O)c1cc(=O)n(-c2ccccc2)[nH]1 ZINC000217724782 DD In-Stock Unstable CTSA 50 39 COc1ccccc1/C=C/NC(=O)NCCCN(C)C ZINC000217724872 CD For-Sale Unstable DRD2 15 44 COc1ccccc1/C=C/NC(=O)NCCCN(C)C ZINC000217724872 CD For-Sale Unstable DRD3 26 44 COc1ccccc1/C=C/NC(=O)NCCCN(C)C ZINC000217724872 CD For-Sale Unstable MTNR1B 15 44 CCCCCC[C@@H](C)NC(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217724899 DH For-Sale Unstable NOD1 68 38 CCOC(=O)c1ccc(NC(=O)COc2cc(C(=O)O)ccc2[N+](=O)[O-])cc1 ZINC000217724909 GE In-Stock Unstable PPIA 15 40 CCOC(=O)c1ccc(NC(=O)COc2cc(C(=O)O)ccc2[N+](=O)[O-])cc1 ZINC000217724909 GE In-Stock Unstable GSTM2 32 42 CCOC(=O)c1ccc(NC(=O)COc2cc(C(=O)O)ccc2[N+](=O)[O-])cc1 ZINC000217724909 GE In-Stock Unstable CETP 26 43 CCOC(=O)c1ccc(NC(=O)COc2cc(C(=O)O)ccc2[N+](=O)[O-])cc1 ZINC000217724909 GE In-Stock Unstable PLA2G4B 26 43 CCOC(=O)c1ccc(NC(=O)COc2cc(C(=O)O)ccc2[N+](=O)[O-])cc1 ZINC000217724909 GE In-Stock Unstable ACR 56 33 O=C(/C=C/c1ccccc1)NC[C@@H]1CCCN1c1nccs1 ZINC000217724920 DF For-Sale Unstable HDAC8 43 36 Nc1ccc(CC(=O)N[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217724971 CD For-Sale Unstable SIGMAR1 22 56 Nc1ccc(CC(=O)N[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217724971 CD For-Sale Unstable SLC18A3 19 40 CCCCCC[C@H](C)NC(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217724988 DH For-Sale Unstable NOD1 68 38 CCCCCCNC[C@@H](O)CCC ZINC000217724993 AE For-Sale Unstable ADH1A 0 40 CCCCCCNC[C@@H](O)CCC ZINC000217724993 AE For-Sale Unstable ADH7 0 40 CCCCCCNC[C@@H](O)CCC ZINC000217724993 AE For-Sale Unstable S1PR3 18 41 CCCCCCNC[C@@H](O)CCC ZINC000217724993 AE For-Sale Unstable S1PR2 44 41 CCCCCCNC[C@@H](O)CCC ZINC000217724993 AE For-Sale Unstable ADH1B 0 40 CCCCCCNC[C@@H](O)CCC ZINC000217724993 AE For-Sale Unstable Q8WS26_TRYCR 45 52 CCCCCCNC[C@@H](O)CCC ZINC000217724993 AE For-Sale Unstable FPPS 0 52 CCCCCCNC[C@@H](O)CCC ZINC000217724993 AE For-Sale Unstable SPPS 0 52 CCCCCCNC[C@@H](O)CCC ZINC000217724993 AE For-Sale Unstable CQSS 45 38 O=C(/C=C/c1ccccc1)NC[C@H]1CCCN1c1nccs1 ZINC000217725013 DF For-Sale Unstable HDAC8 43 36 NS(=O)(=O)c1ccc(NC(=O)COc2cc(C(=O)O)ccc2[N+](=O)[O-])cc1 ZINC000217725022 GC In-Stock Unstable CA2 111 48 NS(=O)(=O)c1ccc(NC(=O)COc2cc(C(=O)O)ccc2[N+](=O)[O-])cc1 ZINC000217725022 GC In-Stock Unstable CA1 96 48 NS(=O)(=O)c1ccc(NC(=O)COc2cc(C(=O)O)ccc2[N+](=O)[O-])cc1 ZINC000217725022 GC In-Stock Unstable CA7 44 48 NS(=O)(=O)c1ccc(NC(=O)COc2cc(C(=O)O)ccc2[N+](=O)[O-])cc1 ZINC000217725022 GC In-Stock Unstable CA5B 48 45 NS(=O)(=O)c1ccc(NC(=O)COc2cc(C(=O)O)ccc2[N+](=O)[O-])cc1 ZINC000217725022 GC In-Stock Unstable CA4 94 48 NS(=O)(=O)c1ccc(NC(=O)COc2cc(C(=O)O)ccc2[N+](=O)[O-])cc1 ZINC000217725022 GC In-Stock Unstable CA5A 55 45 NS(=O)(=O)c1ccc(NC(=O)COc2cc(C(=O)O)ccc2[N+](=O)[O-])cc1 ZINC000217725022 GC In-Stock Unstable CA12 60 46 NS(=O)(=O)c1ccc(NC(=O)COc2cc(C(=O)O)ccc2[N+](=O)[O-])cc1 ZINC000217725022 GC In-Stock Unstable CA9 65 46 NS(=O)(=O)c1ccc(NC(=O)COc2cc(C(=O)O)ccc2[N+](=O)[O-])cc1 ZINC000217725022 GC In-Stock Unstable UREA_CANEN 27 41 NS(=O)(=O)c1ccc(NC(=O)COc2cc(C(=O)O)ccc2[N+](=O)[O-])cc1 ZINC000217725022 GC In-Stock Unstable CYNT 40 42 NS(=O)(=O)c1ccc(NC(=O)COc2cc(C(=O)O)ccc2[N+](=O)[O-])cc1 ZINC000217725022 GC In-Stock Unstable NCE103 22 43 NS(=O)(=O)c1ccc(NC(=O)COc2cc(C(=O)O)ccc2[N+](=O)[O-])cc1 ZINC000217725022 GC In-Stock Unstable MTCA1 50 43 NS(=O)(=O)c1ccc(NC(=O)COc2cc(C(=O)O)ccc2[N+](=O)[O-])cc1 ZINC000217725022 GC In-Stock Unstable P96878_MYCTU 64 43 Nc1ccc(CC(=O)N[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217725057 CD For-Sale Unstable SIGMAR1 22 56 Nc1ccc(CC(=O)N[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217725057 CD For-Sale Unstable SLC18A3 19 40 CCCCCCNC[C@H](O)CCC ZINC000217725077 AE For-Sale Unstable ADH1A 0 40 CCCCCCNC[C@H](O)CCC ZINC000217725077 AE For-Sale Unstable ADH7 0 40 CCCCCCNC[C@H](O)CCC ZINC000217725077 AE For-Sale Unstable S1PR3 18 41 CCCCCCNC[C@H](O)CCC ZINC000217725077 AE For-Sale Unstable S1PR2 44 41 CCCCCCNC[C@H](O)CCC ZINC000217725077 AE For-Sale Unstable ADH1B 0 40 CCCCCCNC[C@H](O)CCC ZINC000217725077 AE For-Sale Unstable Q8WS26_TRYCR 45 52 CCCCCCNC[C@H](O)CCC ZINC000217725077 AE For-Sale Unstable FPPS 0 52 CCCCCCNC[C@H](O)CCC ZINC000217725077 AE For-Sale Unstable SPPS 0 52 CCCCCCNC[C@H](O)CCC ZINC000217725077 AE For-Sale Unstable CQSS 45 38 O=C(O)/C=C\c1ccc(C(=O)NCCN2CCCCC2)s1 ZINC000217725098 DE For-Sale Unstable DRD4 41 33 O=C(O)/C=C\c1ccc(C(=O)NCCN2CCCCC2)s1 ZINC000217725098 DE For-Sale Unstable DRD3 19 41 O=C(O)/C=C\c1ccc(C(=O)NCCN2CCCCC2)s1 ZINC000217725098 DE For-Sale Unstable PLD2 45 37 C[C@@H](N[C@@H]1CCN2CCC[C@@H]12)c1cccc2ccccc12 ZINC000217725114 CH For-Sale Unstable CASR 0 48 O=C(CCc1ccccc1)NC[C@@H]1CCCN1c1nccs1 ZINC000217725117 DF For-Sale Unstable GRIN2B 17 41 O=C(CCc1ccccc1)NC[C@@H]1CCCN1c1nccs1 ZINC000217725117 DF For-Sale Unstable PREP 57 42 CC(=O)c1cccc(NC(=O)COc2cc(C(=O)O)ccc2[N+](=O)[O-])c1 ZINC000217725125 FF In-Stock Unstable AKR1C4 0 47 O=C(N[C@@H]1CCN2CCC[C@@H]12)[C@@H]1Cc2ccccc2CN1 ZINC000217725154 CD For-Sale Unstable MC4R 36 41 O=C(N[C@@H]1CCN2CCC[C@@H]12)[C@@H]1Cc2ccccc2CN1 ZINC000217725154 CD For-Sale Unstable SLC18A3 59 39 COc1ccc(Br)cc1S(=O)(=O)N1CCN(Cc2cccnc2)CC1 ZINC000217725160 IE On-Demand Unstable DRD4 15 43 O=C(CCc1ccccc1)NC[C@H]1CCCN1c1nccs1 ZINC000217725194 DF For-Sale Unstable GRIN2B 17 41 O=C(CCc1ccccc1)NC[C@H]1CCCN1c1nccs1 ZINC000217725194 DF For-Sale Unstable PREP 57 42 C[C@H](N[C@@H]1CCN2CCC[C@@H]12)c1cccc2ccccc12 ZINC000217725198 CH For-Sale Unstable CASR 0 48 CCC[C@@H](O)CN[C@@H](C)Cc1ccccc1 ZINC000217725206 BE For-Sale Unstable ADRB2 32 47 CCC[C@@H](O)CN[C@@H](C)Cc1ccccc1 ZINC000217725206 BE For-Sale Unstable ADRB1 23 47 CCC[C@@H](O)CN[C@@H](C)Cc1ccccc1 ZINC000217725206 BE For-Sale Unstable MME 65 38 CCC[C@@H](O)CN[C@@H](C)Cc1ccccc1 ZINC000217725206 BE For-Sale Unstable SCN5A 0 51 CCC[C@@H](O)CN[C@@H](C)Cc1ccccc1 ZINC000217725206 BE For-Sale Unstable LMGT2 0 41 COc1ccc(C(=O)N2CC[C@H]3CC[C@@H](C2)N3C)c(F)c1 ZINC000217725215 CE On-Demand Unstable L3MBTL3 45 35 CN1CC[C@H](NC(=O)c2ccc(/C=C\C(=O)O)cc2F)C1 ZINC000217725218 CD For-Sale Unstable HTR4 20 40 CC(C)NC(=O)COc1cc(C(=O)O)cc(C(=O)O)c1 ZINC000217725233 CC In-Stock Unstable PLA2G4B 45 35 CN1c2ccccc2C(=O)N2CCc3c(n(CCC(=O)NCc4ccccc4)c4ccccc34)[C@H]21 ZINC000217725237 JI In-Stock Unstable FABI 47 32 CN1c2ccccc2C(=O)N2CCc3c(n(CCC(=O)NCc4ccccc4)c4ccccc34)[C@H]21 ZINC000217725237 JI In-Stock Unstable HTR7 16 40 O=C(N[C@H]1CCN2CCC[C@@H]12)[C@@H]1Cc2ccccc2CN1 ZINC000217725246 CD For-Sale Unstable MC4R 36 41 O=C(N[C@H]1CCN2CCC[C@@H]12)[C@@H]1Cc2ccccc2CN1 ZINC000217725246 CD For-Sale Unstable SLC18A3 59 39 CC(=O)N1CCc2cc(S(=O)(=O)N3CCN(Cc4cccnc4)CC3)ccc21 ZINC000217725261 HD On-Demand Unstable CYP11B1 20 45 CC(=O)N1CCc2cc(S(=O)(=O)N3CCN(Cc4cccnc4)CC3)ccc21 ZINC000217725261 HD On-Demand Unstable ADORA2B 44 34 CC(=O)N1CCc2cc(S(=O)(=O)N3CCN(Cc4cccnc4)CC3)ccc21 ZINC000217725261 HD On-Demand Unstable CYP11B2 43 53 CC(=O)N1CCc2cc(S(=O)(=O)N3CCN(Cc4cccnc4)CC3)ccc21 ZINC000217725261 HD On-Demand Unstable AKR1C3 45 33 CC(=O)N1CCc2cc(S(=O)(=O)N3CCN(Cc4cccnc4)CC3)ccc21 ZINC000217725261 HD On-Demand Unstable NAMPT 58 43 C[C@@H](N[C@H]1CCN2CCC[C@@H]12)c1cccc2ccccc12 ZINC000217725265 CH For-Sale Unstable CASR 0 48 CCC[C@H](O)CN[C@@H](C)Cc1ccccc1 ZINC000217725300 BE For-Sale Unstable ADRB2 32 47 CCC[C@H](O)CN[C@@H](C)Cc1ccccc1 ZINC000217725300 BE For-Sale Unstable ADRB1 23 47 CCC[C@H](O)CN[C@@H](C)Cc1ccccc1 ZINC000217725300 BE For-Sale Unstable MME 65 38 CCC[C@H](O)CN[C@@H](C)Cc1ccccc1 ZINC000217725300 BE For-Sale Unstable SCN5A 0 51 CCC[C@H](O)CN[C@@H](C)Cc1ccccc1 ZINC000217725300 BE For-Sale Unstable LMGT2 0 41 C[C@@H]1OC(=O)[C@H](NC=O)[C@@H]1C ZINC000217725306 AB For-Sale Unstable NAAA 51 36 O=[N+]([O-])c1cc2c(cc1OC1CCC1)OCO2 ZINC000217725310 BE In-Stock Unstable TRXR2 0 45 CC[C@@H](C)NC(=O)COc1cc(C(=O)O)cc(C(=O)O)c1 ZINC000217725334 CD In-Stock Unstable PLA2G4B 42 37 COC(=O)[C@H](Cc1ccccc1)NC(=O)CCn1cc(C(C)=O)c2ccccc21 ZINC000217725346 GG In-Stock Unstable ACE 21 41 COC(=O)[C@H](Cc1ccccc1)NC(=O)CCn1cc(C(C)=O)c2ccccc21 ZINC000217725346 GG In-Stock Unstable CNR1 34 47 COC(=O)[C@H](Cc1ccccc1)NC(=O)CCn1cc(C(C)=O)c2ccccc21 ZINC000217725346 GG In-Stock Unstable MME 60 39 COC(=O)[C@H](Cc1ccccc1)NC(=O)CCn1cc(C(C)=O)c2ccccc21 ZINC000217725346 GG In-Stock Unstable ANPEP 43 31 COC(=O)[C@H](Cc1ccccc1)NC(=O)CCn1cc(C(C)=O)c2ccccc21 ZINC000217725346 GG In-Stock Unstable TACR1 28 41 COC(=O)[C@H](Cc1ccccc1)NC(=O)CCn1cc(C(C)=O)c2ccccc21 ZINC000217725346 GG In-Stock Unstable CNR2 33 47 COC(=O)[C@H](Cc1ccccc1)NC(=O)CCn1cc(C(C)=O)c2ccccc21 ZINC000217725346 GG In-Stock Unstable FCER2 40 32 COC(=O)[C@H](Cc1ccccc1)NC(=O)CCn1cc(C(C)=O)c2ccccc21 ZINC000217725346 GG In-Stock Unstable PAPA1_CARPA 52 38 COC(=O)[C@H](Cc1ccccc1)NC(=O)CCn1cc(C(C)=O)c2ccccc21 ZINC000217725346 GG In-Stock Unstable CYSP_TRYCR 50 35 COC(=O)[C@H](Cc1ccccc1)NC(=O)CCn1cc(C(C)=O)c2ccccc21 ZINC000217725346 GG In-Stock Unstable CCR3 0 41 COC(=O)[C@H](Cc1ccccc1)NC(=O)CCn1cc(C(C)=O)c2ccccc21 ZINC000217725346 GG In-Stock Unstable CAPNS1 54 38 COC(=O)[C@H](Cc1ccccc1)NC(=O)CCn1cc(C(C)=O)c2ccccc21 ZINC000217725346 GG In-Stock Unstable PAM 0 42 COC(=O)[C@H](Cc1ccccc1)NC(=O)CCn1cc(C(C)=O)c2ccccc21 ZINC000217725346 GG In-Stock Unstable CAPN1 50 44 COC(=O)[C@H](Cc1ccccc1)NC(=O)CCn1cc(C(C)=O)c2ccccc21 ZINC000217725346 GG In-Stock Unstable ACE2 49 33 COC(=O)[C@H](Cc1ccccc1)NC(=O)CCn1cc(C(C)=O)c2ccccc21 ZINC000217725346 GG In-Stock Unstable MMP1 15 41 COC(=O)[C@H](Cc1ccccc1)NC(=O)CCn1cc(C(C)=O)c2ccccc21 ZINC000217725346 GG In-Stock Unstable POL 0 41 COC(=O)[C@H](Cc1ccccc1)NC(=O)CCn1cc(C(C)=O)c2ccccc21 ZINC000217725346 GG In-Stock Unstable NPR 18 42 COC(=O)[C@H](Cc1ccccc1)NC(=O)CCn1cc(C(C)=O)c2ccccc21 ZINC000217725346 GG In-Stock Unstable HDA106 0 54 COC(=O)[C@H](Cc1ccccc1)NC(=O)CCn1cc(C(C)=O)c2ccccc21 ZINC000217725346 GG In-Stock Unstable SLC15A2 0 40 C[C@H](N[C@H]1CCN2CCC[C@@H]12)c1cccc2ccccc12 ZINC000217725351 CH For-Sale Unstable CASR 0 48 CCC[C@@H](O)CN[C@H](C)Cc1ccccc1 ZINC000217725379 BE For-Sale Unstable ADRB2 32 47 CCC[C@@H](O)CN[C@H](C)Cc1ccccc1 ZINC000217725379 BE For-Sale Unstable ADRB1 23 47 CCC[C@@H](O)CN[C@H](C)Cc1ccccc1 ZINC000217725379 BE For-Sale Unstable MME 65 38 CCC[C@@H](O)CN[C@H](C)Cc1ccccc1 ZINC000217725379 BE For-Sale Unstable SCN5A 0 51 CCC[C@@H](O)CN[C@H](C)Cc1ccccc1 ZINC000217725379 BE For-Sale Unstable LMGT2 0 41 C[C@@H]1OC(=O)[C@@H](NC=O)[C@H]1C ZINC000217725404 AB For-Sale Unstable NAAA 51 36 CN(Cc1ccoc1)C(=O)c1ccc(/C=C\C(=O)O)s1 ZINC000217725410 CF For-Sale Unstable HSD17B2 31 44 CC[C@H](C)NC(=O)COc1cc(C(=O)O)cc(C(=O)O)c1 ZINC000217725427 CD In-Stock Unstable PLA2G4B 42 37 CCC[C@H](O)CN[C@H](C)Cc1ccccc1 ZINC000217725464 BE For-Sale Unstable ADRB2 32 47 CCC[C@H](O)CN[C@H](C)Cc1ccccc1 ZINC000217725464 BE For-Sale Unstable ADRB1 23 47 CCC[C@H](O)CN[C@H](C)Cc1ccccc1 ZINC000217725464 BE For-Sale Unstable MME 65 38 CCC[C@H](O)CN[C@H](C)Cc1ccccc1 ZINC000217725464 BE For-Sale Unstable SCN5A 0 51 CCC[C@H](O)CN[C@H](C)Cc1ccccc1 ZINC000217725464 BE For-Sale Unstable LMGT2 0 41 CCOc1ccc(/C=C/C(=O)NC[C@H](O)C(=O)OC)cc1 ZINC000217725484 CC On-Demand Unstable HDAC8 16 44 CN1CCN(c2cc3c(cc2[N+](=O)[O-])OCO3)CC1 ZINC000217725531 CD In-Stock Unstable TRXR2 0 41 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)NC1CCCCC1 ZINC000217725532 DD In-Stock Unstable FAAH 23 40 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)NC1CCCCC1 ZINC000217725532 DD In-Stock Unstable EPHX2 39 43 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)NC1CCCCC1 ZINC000217725532 DD In-Stock Unstable PLAU 17 42 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)NC1CCCCC1 ZINC000217725532 DD In-Stock Unstable ST14 17 42 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)NC1CCCCC1 ZINC000217725532 DD In-Stock Unstable LUXN 0 55 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)NC1CCCCC1 ZINC000217725532 DD In-Stock Unstable ADIPOR1 0 46 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)NC1CCCCC1 ZINC000217725532 DD In-Stock Unstable ADIPOR2 0 46 COc1ccc2nc(Br)nc(C)c2c1 ZINC000217725535 CF For-Sale Unstable CYP1B1 48 38 COc1ccc2nc(Br)nc(C)c2c1 ZINC000217725535 CF For-Sale Unstable LUCI_PHOPE 30 41 O=S(=O)(NCc1csc(-c2ccccc2)n1)c1ccccc1C(F)(F)F ZINC000217725547 GI On-Demand Unstable ADAMTS5 15 41 COc1ccc(C(=O)N2CC[C@H]3CC[C@@H](C2)N3C)cc1Br ZINC000217725551 FF On-Demand Unstable L3MBTL1 0 46 COc1ccc(C(=O)N2CC[C@H]3CC[C@@H](C2)N3C)cc1Br ZINC000217725551 FF On-Demand Unstable L3MBTL3 72 43 COc1ccc(C(=O)N2CC[C@H]3CC[C@@H](C2)N3C)cc1Br ZINC000217725551 FF On-Demand Unstable MBTD1 0 46 Nc1[nH]nc(C(=O)N[C@@H](CC(=O)O)c2ccccc2)c1Cl ZINC000217725582 DD In-Stock Unstable CTSA 71 41 Cc1cc(S(=O)(=O)N2CCC[C@@H]2C)ccc1/C=C\C(=O)O ZINC000217725594 DE For-Sale Unstable CASP3 50 37 Cc1cc(S(=O)(=O)N2CCC[C@@H]2C)ccc1/C=C\C(=O)O ZINC000217725594 DE For-Sale Unstable CASP7 59 36 Cc1cc(S(=O)(=O)N2CCC[C@@H]2C)ccc1/C=C\C(=O)O ZINC000217725594 DE For-Sale Unstable AKR1C3 31 45 COC(=O)C1=C(NC(=S)N2CCN(c3c(F)cc4c(=O)c(C(=O)O)cn(C5CC5)c4c3OC)C[C@@H]2C)S[C@@H]2CCCCC[C@@H]12 ZINC000217725627 KJ In-Stock Unstable POLC 15 41 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)NCc1ccccc1 ZINC000217725628 ED In-Stock Unstable SRD5A2 28 42 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)NCc1ccccc1 ZINC000217725628 ED In-Stock Unstable GRIN2B 15 40 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)NCc1ccccc1 ZINC000217725628 ED In-Stock Unstable ADORA2B 0 45 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)NCc1ccccc1 ZINC000217725628 ED In-Stock Unstable UL80 28 44 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)NCc1ccccc1 ZINC000217725628 ED In-Stock Unstable HDAC8 20 45 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)NCc1ccccc1 ZINC000217725628 ED In-Stock Unstable PLA2G4B 54 43 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)NCc1ccccc1 ZINC000217725628 ED In-Stock Unstable AMP1_PLAFQ 46 37 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)NCc1ccccc1 ZINC000217725628 ED In-Stock Unstable NCE103 17 43 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)NCc1ccccc1 ZINC000217725628 ED In-Stock Unstable CRTM 56 36 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)NCc1ccccc1 ZINC000217725628 ED In-Stock Unstable KDM4E 22 43 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)NCc1ccccc1 ZINC000217725628 ED In-Stock Unstable PDS 65 43 COc1ccc2c(C)nc(Br)nc2c1 ZINC000217725645 CF For-Sale Unstable CYP1B1 42 36 Cc1ccc(Br)cc1S(=O)(=O)NCc1csc(-c2ccccc2)n1 ZINC000217725657 HI On-Demand Unstable ADAMTS5 17 40 Nc1[nH]nc(C(=O)N[C@H](CC(=O)O)c2ccccc2)c1Cl ZINC000217725658 DD In-Stock Unstable CTSA 71 41 Cc1ccc(/C=C\C(=O)O)cc1S(=O)(=O)N1CCC[C@@H]1C ZINC000217725684 DE For-Sale Unstable AKR1C3 0 40 COc1ccccc1/C=C/NC(=O)NCCCOC(C)C ZINC000217725685 CF For-Sale Unstable DRD3 26 42 C[C@@H]1OC(=O)[C@H](NC=O)[C@H]1C ZINC000217725693 AB For-Sale Unstable NAAA 51 36 O=C(CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)Nc1ccc2[nH]cnc2c1 ZINC000217725708 FE In-Stock Unstable PTPN2 24 58 O=C(CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)Nc1ccc2[nH]cnc2c1 ZINC000217725708 FE In-Stock Unstable PLCD1 0 41 O=C(CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)Nc1ccc2[nH]cnc2c1 ZINC000217725708 FE In-Stock Unstable AGAL_COFAR 0 47 O=C(CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)Nc1ccc2[nH]cnc2c1 ZINC000217725708 FE In-Stock Unstable CYTH3 0 41 O=C(CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)Nc1ccc2[nH]cnc2c1 ZINC000217725708 FE In-Stock Unstable HLCS 0 47 O=C(CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)Nc1ccc2[nH]cnc2c1 ZINC000217725708 FE In-Stock Unstable BIRA 0 41 O=C(COc1ccccc1)NC[C@@H]1CCCN1c1nccs1 ZINC000217725712 DE For-Sale Unstable CPT1A 95 38 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)NCCc1ccccc1 ZINC000217725730 ED In-Stock Unstable SRD5A2 24 41 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)NCCc1ccccc1 ZINC000217725730 ED In-Stock Unstable CYSP_TRYCR 0 41 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)NCCc1ccccc1 ZINC000217725730 ED In-Stock Unstable PLA2G4A 29 40 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)NCCc1ccccc1 ZINC000217725730 ED In-Stock Unstable HDAC8 22 49 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)NCCc1ccccc1 ZINC000217725730 ED In-Stock Unstable CA5B 17 44 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)NCCc1ccccc1 ZINC000217725730 ED In-Stock Unstable CA5A 15 44 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)NCCc1ccccc1 ZINC000217725730 ED In-Stock Unstable PLA2G4B 54 45 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)NCCc1ccccc1 ZINC000217725730 ED In-Stock Unstable AMP1_PLAFQ 26 40 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)NCCc1ccccc1 ZINC000217725730 ED In-Stock Unstable AKR1C3 17 43 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)NCCc1ccccc1 ZINC000217725730 ED In-Stock Unstable NCE103 26 46 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)NCCc1ccccc1 ZINC000217725730 ED In-Stock Unstable CRTM 60 41 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)NCCc1ccccc1 ZINC000217725730 ED In-Stock Unstable P96878_MYCTU 17 46 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)NCCc1ccccc1 ZINC000217725730 ED In-Stock Unstable KDM4E 26 54 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)NCCc1ccccc1 ZINC000217725730 ED In-Stock Unstable CAN2 0 46 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)NCCc1ccccc1 ZINC000217725730 ED In-Stock Unstable PDS 42 39 COc1cccc2c(C)nc(Br)nc12 ZINC000217725750 CF For-Sale Unstable ATP4A 28 47 CC1CCN(S(=O)(=O)c2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217725766 DE For-Sale Unstable EPHX2 16 42 CC1CCN(S(=O)(=O)c2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217725766 DE For-Sale Unstable AKR1C3 64 40 CNC(=O)c1cc(N[C@@H]2CCC[C@@H](C)[C@@H]2C)ccn1 ZINC000217725770 CF On-Demand Unstable RAF1 46 32 CNC(=O)c1cc(N[C@@H]2CCC[C@@H](C)[C@@H]2C)ccn1 ZINC000217725770 CF On-Demand Unstable Q8MMZ8_EIMTE 47 39 Cc1ccc(C(=O)N[C@@H]2CCN3CCC[C@@H]23)cc1N ZINC000217725771 CD For-Sale Unstable L3MBTL3 44 37 CC(=O)N1CCc2cc(S(=O)(=O)NCc3csc(-c4ccccc4)n3)ccc21 ZINC000217725772 HG On-Demand Unstable HSD17B3 45 34 CC(=O)N1CCc2cc(S(=O)(=O)NCc3csc(-c4ccccc4)n3)ccc21 ZINC000217725772 HG On-Demand Unstable ADAMTS5 25 42 CC(=O)N1CCc2cc(S(=O)(=O)NCc3csc(-c4ccccc4)n3)ccc21 ZINC000217725772 HG On-Demand Unstable LUXN 0 40 C[C@@H]1[C@@H](C)OC(=O)[C@@H]1NC=O ZINC000217725791 AB For-Sale Unstable NAAA 51 36 O=C(COc1ccccc1)NC[C@H]1CCCN1c1nccs1 ZINC000217725798 DE For-Sale Unstable CPT1A 95 38 CCc1ccc(/C=C\C(=O)NCC2CC(O)C2)cc1 ZINC000217725799 CE For-Sale Unstable HDAC8 23 43 COc1ccc([C@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1O ZINC000217725822 KH In-Stock Unstable AKR1B1 0 41 COc1ccc([C@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1O ZINC000217725822 KH In-Stock Unstable PRKDC 15 43 COc1ccc([C@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1O ZINC000217725822 KH In-Stock Unstable CYP1B1 60 39 COc1ccc([C@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1O ZINC000217725822 KH In-Stock Unstable CYP1A1 48 39 COc1ccc([C@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1O ZINC000217725822 KH In-Stock Unstable RORC 0 40 CNC(=O)c1cc(N[C@H]2CCC[C@@H](C)[C@@H]2C)ccn1 ZINC000217725840 CF For-Sale Unstable RAF1 46 32 CNC(=O)c1cc(N[C@H]2CCC[C@@H](C)[C@@H]2C)ccn1 ZINC000217725840 CF For-Sale Unstable Q8MMZ8_EIMTE 47 39 CN1CCN(S(=O)(=O)c2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217725844 DC For-Sale Unstable LPL 20 41 CN1CCN(S(=O)(=O)c2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217725844 DC For-Sale Unstable HDAC8 25 40 CN1CCN(S(=O)(=O)c2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217725844 DC For-Sale Unstable F13A1 45 37 CN1CCN(S(=O)(=O)c2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217725844 DC For-Sale Unstable AKR1C3 71 44 Cc1ccc(C(=O)N[C@H]2CCN3CCC[C@@H]23)cc1N ZINC000217725847 CD For-Sale Unstable L3MBTL3 44 37 CS(=O)(=O)OCCc1ccc(F)cc1F ZINC000217725884 BD For-Sale Unstable HTR2A 16 45 COc1ccc([C@@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1O ZINC000217725904 KH In-Stock Unstable AKR1B1 0 41 COc1ccc([C@@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1O ZINC000217725904 KH In-Stock Unstable PRKDC 15 43 COc1ccc([C@@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1O ZINC000217725904 KH In-Stock Unstable CYP1B1 60 39 COc1ccc([C@@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1O ZINC000217725904 KH In-Stock Unstable CYP1A1 48 39 COc1ccc([C@@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1O ZINC000217725904 KH In-Stock Unstable RORC 0 40 COc1ccccc1/C=C/NC(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000217725909 FK For-Sale Unstable EPHX1 0 40 COc1ccccc1/C=C/NC(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000217725909 FK For-Sale Unstable AKR1C3 27 42 COc1ccccc1/C=C/NC(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000217725909 FK For-Sale Unstable P95276_MYCTO 0 40 COc1ccccc1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217725918 DF For-Sale Unstable HTR1A 20 45 COc1ccccc1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217725918 DF For-Sale Unstable DRD2 41 43 COc1ccccc1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217725918 DF For-Sale Unstable DRD4 17 40 COc1ccccc1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217725918 DF For-Sale Unstable DRD3 26 44 COc1ccccc1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217725918 DF For-Sale Unstable KCNA3 48 38 COc1ccccc1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217725918 DF For-Sale Unstable MAP1 22 40 COc1ccccc1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217725918 DF For-Sale Unstable HCN1 80 43 COc1ccccc1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217725918 DF For-Sale Unstable HCN4 56 39 COc1ccccc1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217725918 DF For-Sale Unstable ACKR3 67 35 Cc1ccc(/C=C\C(=O)NCC2CC(O)C2)c(C)c1 ZINC000217725920 CE For-Sale Unstable BOTA 16 45 CNC(=O)c1cc(N[C@@H]2CCC[C@H](C)[C@@H]2C)ccn1 ZINC000217725929 CF On-Demand Unstable RAF1 46 32 CNC(=O)c1cc(N[C@@H]2CCC[C@H](C)[C@@H]2C)ccn1 ZINC000217725929 CF On-Demand Unstable Q8MMZ8_EIMTE 47 39 Cc1onc(-c2ccccc2Cl)c1C(=O)N1CC(N2C(=O)[C@H]3CC=CC[C@H]3C2=O)C1 ZINC000217725946 IG In-Stock Unstable GPBAR1 34 45 Cc1onc(-c2ccccc2Cl)c1C(=O)N1CC(N2C(=O)[C@H]3CC=CC[C@H]3C2=O)C1 ZINC000217725946 IG In-Stock Unstable BLAACC-4 0 45 Cc1onc(-c2ccccc2Cl)c1C(=O)N1CC(N2C(=O)[C@H]3CC=CC[C@H]3C2=O)C1 ZINC000217725946 IG In-Stock Unstable SUGE 0 45 Cc1onc(-c2ccccc2Cl)c1C(=O)N1CC(N2C(=O)[C@H]3CC=CC[C@H]3C2=O)C1 ZINC000217725946 IG In-Stock Unstable BLA_LAT-2 0 45 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccccc1 ZINC000217725960 DE In-Stock Unstable EPHX1 0 40 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccccc1 ZINC000217725960 DE In-Stock Unstable LTA4H 41 42 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccccc1 ZINC000217725960 DE In-Stock Unstable ADORA2A 0 44 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccccc1 ZINC000217725960 DE In-Stock Unstable ADORA2B 43 44 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccccc1 ZINC000217725960 DE In-Stock Unstable CETP 0 42 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccccc1 ZINC000217725960 DE In-Stock Unstable HDAC8 25 43 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccccc1 ZINC000217725960 DE In-Stock Unstable PLA2G4B 47 37 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccccc1 ZINC000217725960 DE In-Stock Unstable HIF1A 26 49 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccccc1 ZINC000217725960 DE In-Stock Unstable AKR1C3 35 40 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccccc1 ZINC000217725960 DE In-Stock Unstable PFHDAC1 0 40 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccccc1 ZINC000217725960 DE In-Stock Unstable P95276_MYCTO 0 40 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccccc1 ZINC000217725960 DE In-Stock Unstable KCNK3 44 38 N[C@@H](C(=O)N[C@@H]1CCN2CCC[C@@H]12)c1ccccc1 ZINC000217725962 CD For-Sale Unstable SLC18A3 59 36 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable ACE 74 59 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable TYR 36 45 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable OPRM1 61 45 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable OPRD1 82 45 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable FOLH1 19 56 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable MME 177 59 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable LTA4H 19 40 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable ANPEP 82 40 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable FCER2 59 38 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable RNPEP 28 40 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable CTSB 21 57 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable PAPA1_CARPA 46 33 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable CCKAR 28 41 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable NTSR1 50 34 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable CTSL 22 42 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable CPA1 72 58 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable ITGA4 46 37 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable NAALAD2 47 60 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable CAPNS1 54 39 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable MMP8 18 41 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable GRIA1 61 40 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable ECE1 66 47 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable YARS 77 44 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable CAPN1 27 47 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable MMP9 16 42 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable CASP1 16 51 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable CAPN2 29 57 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable ENPEP 24 50 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable ACE2 107 58 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable LAP3 26 40 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable MMP1 25 41 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable FPR1 78 43 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable NPPA 24 41 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable AMP1_PLAFQ 16 40 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable XIAP 24 43 O=C(O)C[C@@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217725969 CB For-Sale Unstable BLA1_STEMA 81 41 COc1ccccc1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217725991 DF For-Sale Unstable HTR1A 20 45 COc1ccccc1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217725991 DF For-Sale Unstable DRD2 41 43 COc1ccccc1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217725991 DF For-Sale Unstable DRD4 17 40 COc1ccccc1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217725991 DF For-Sale Unstable DRD3 26 44 COc1ccccc1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217725991 DF For-Sale Unstable KCNA3 48 38 COc1ccccc1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217725991 DF For-Sale Unstable MAP1 22 40 COc1ccccc1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217725991 DF For-Sale Unstable HCN1 80 43 COc1ccccc1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217725991 DF For-Sale Unstable HCN4 56 39 COc1ccccc1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217725991 DF For-Sale Unstable ACKR3 67 35 CNC(=O)c1cc(N[C@H]2CCC[C@H](C)[C@@H]2C)ccn1 ZINC000217726012 CF For-Sale Unstable RAF1 46 32 CNC(=O)c1cc(N[C@H]2CCC[C@H](C)[C@@H]2C)ccn1 ZINC000217726012 CF For-Sale Unstable Q8MMZ8_EIMTE 47 39 O=C(O)/C=C\c1cccc(S(=O)(=O)Nc2ccccn2)c1 ZINC000217726020 DD For-Sale Anodyne HDAC8 31 55 O=C(O)/C=C\c1cccc(S(=O)(=O)Nc2ccccn2)c1 ZINC000217726020 DD For-Sale Anodyne HDAC1 15 55 O=C(O)/C=C\c1cccc(S(=O)(=O)Nc2ccccn2)c1 ZINC000217726020 DD For-Sale Anodyne RHOA 0 45 Cc1onc(-c2ccccc2Cl)c1C(=O)N1CC(N2C(=O)[C@H]3CC=CC[C@@H]3C2=O)C1 ZINC000217726021 IG In-Stock Unstable GPBAR1 34 45 Cc1onc(-c2ccccc2Cl)c1C(=O)N1CC(N2C(=O)[C@H]3CC=CC[C@@H]3C2=O)C1 ZINC000217726021 IG In-Stock Unstable BLAACC-4 0 45 Cc1onc(-c2ccccc2Cl)c1C(=O)N1CC(N2C(=O)[C@H]3CC=CC[C@@H]3C2=O)C1 ZINC000217726021 IG In-Stock Unstable SUGE 0 45 Cc1onc(-c2ccccc2Cl)c1C(=O)N1CC(N2C(=O)[C@H]3CC=CC[C@@H]3C2=O)C1 ZINC000217726021 IG In-Stock Unstable BLA_LAT-2 0 45 N[C@H](C(=O)N[C@@H]1CCN2CCC[C@@H]12)c1ccccc1 ZINC000217726047 CD For-Sale Unstable SLC18A3 59 36 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable ACE 74 59 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable TYR 36 45 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable OPRM1 61 45 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable OPRD1 82 45 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable FOLH1 19 56 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable MME 177 59 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable LTA4H 19 40 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable ANPEP 82 40 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable FCER2 59 38 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable RNPEP 28 40 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable CTSB 21 57 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable PAPA1_CARPA 46 33 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable CCKAR 28 41 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable NTSR1 50 34 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable CTSL 22 42 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable CPA1 72 58 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable ITGA4 46 37 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable NAALAD2 47 60 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable CAPNS1 54 39 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable MMP8 18 41 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable GRIA1 61 40 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable ECE1 66 47 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable YARS 77 44 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable CAPN1 27 47 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable MMP9 16 42 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable CASP1 16 51 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable CAPN2 29 57 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable ENPEP 24 50 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable ACE2 107 58 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable LAP3 26 40 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable MMP1 25 41 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable FPR1 78 43 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable NPPA 24 41 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable AMP1_PLAFQ 16 40 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable XIAP 24 43 O=C(O)C[C@H](O)C(=O)N[C@H](Cc1ccc(O)cc1)C(=O)O ZINC000217726048 CB For-Sale Unstable BLA1_STEMA 81 41 Cc1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217726058 EE In-Stock Unstable CCKAR 23 44 Cc1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217726058 EE In-Stock Unstable CETP 0 43 Cc1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217726058 EE In-Stock Unstable HDAC8 16 48 Cc1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217726058 EE In-Stock Unstable PLA2G4B 41 38 Cc1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217726058 EE In-Stock Unstable SCN10A 20 41 Cc1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217726058 EE In-Stock Unstable HIF1A 26 49 Cc1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217726058 EE In-Stock Unstable AKR1C3 40 42 Cc1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217726058 EE In-Stock Unstable AKR1C2 19 42 Cc1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217726058 EE In-Stock Unstable KCNK3 91 46 Cc1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217726058 EE In-Stock Unstable KCNK9 77 45 COc1nc(Br)nc2c(C)cccc12 ZINC000217726084 CF For-Sale Unstable TNKS 29 44 Cc1onc(-c2ccccc2Cl)c1C(=O)N1CC(N2C(=O)[C@@H]3CC=CC[C@H]3C2=O)C1 ZINC000217726098 IG In-Stock Unstable GPBAR1 34 45 Cc1onc(-c2ccccc2Cl)c1C(=O)N1CC(N2C(=O)[C@@H]3CC=CC[C@H]3C2=O)C1 ZINC000217726098 IG In-Stock Unstable BLAACC-4 0 45 Cc1onc(-c2ccccc2Cl)c1C(=O)N1CC(N2C(=O)[C@@H]3CC=CC[C@H]3C2=O)C1 ZINC000217726098 IG In-Stock Unstable SUGE 0 45 Cc1onc(-c2ccccc2Cl)c1C(=O)N1CC(N2C(=O)[C@@H]3CC=CC[C@H]3C2=O)C1 ZINC000217726098 IG In-Stock Unstable BLA_LAT-2 0 45 C[C@@H]1CCCN(S(=O)(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217726099 DE For-Sale Unstable AKR1C3 59 44 C[C@@H]1CCCN(S(=O)(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217726099 DE For-Sale Unstable RAC1 0 43 C[C@@H]1CCCN(S(=O)(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217726099 DE For-Sale Unstable AKR1C1 22 43 COc1cccc(C(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217726114 DF For-Sale Unstable DRD4 53 40 COc1cccc(C(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217726114 DF For-Sale Unstable DRD3 15 41 COc1cccc(C(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217726114 DF For-Sale Unstable MTNR1B 23 40 COc1cccc(C(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217726114 DF For-Sale Unstable CHRNA10 50 42 COc1cccc(C(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217726114 DF For-Sale Unstable ACKR3 65 35 Cn1nc(-c2ccc(F)cc2)cc1C(=O)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217726115 FG In-Stock Unstable CCR3 69 33 COc1ccccc1/C=C/NC(=O)Nc1cccc(C)n1 ZINC000217726122 CG For-Sale Unstable GRM5 18 51 N[C@@H](C(=O)N[C@H]1CCN2CCC[C@@H]12)c1ccccc1 ZINC000217726127 CD For-Sale Unstable SLC18A3 59 36 CN1C[C@H](c2cccc([N+](=O)[O-])c2)[C@@H](C(=O)c2cccs2)[C@@]12C(=O)Nc1ccc(F)cc12 ZINC000217726153 JI In-Stock Unstable CACNA1D 62 35 Cc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217726170 EE In-Stock Unstable LTA4H 34 40 Cc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217726170 EE In-Stock Unstable ADORA2A 15 44 Cc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217726170 EE In-Stock Unstable ADORA2B 48 44 Cc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217726170 EE In-Stock Unstable CETP 0 48 Cc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217726170 EE In-Stock Unstable HDAC8 24 42 Cc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217726170 EE In-Stock Unstable PLA2G4B 46 35 Cc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217726170 EE In-Stock Unstable P4HTM 0 42 Cc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217726170 EE In-Stock Unstable ACR 38 41 Cc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217726170 EE In-Stock Unstable MCHR1 16 40 Cc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217726170 EE In-Stock Unstable HIF1A 24 41 Cc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217726170 EE In-Stock Unstable AKR1C3 22 42 C[C@H]1CCCN(S(=O)(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217726176 DE For-Sale Unstable AKR1C3 59 44 C[C@H]1CCCN(S(=O)(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217726176 DE For-Sale Unstable RAC1 0 43 C[C@H]1CCCN(S(=O)(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217726176 DE For-Sale Unstable AKR1C1 22 43 O=C1C[C@@H](C(=O)Nc2cc(C(=O)O)ccn2)NC(=O)N1 ZINC000217726193 CB For-Sale Unstable TYK2 57 35 COc1ccc(C(=O)OCCC2CC2)c(N)c1 ZINC000217726204 BE On-Demand Unstable HTR4 58 39 COc1ccc(C(=O)OCCC2CC2)c(N)c1 ZINC000217726204 BE On-Demand Unstable MTNR1A 41 37 COc1ccc(C(=O)OCCC2CC2)c(N)c1 ZINC000217726204 BE On-Demand Unstable AKR1C2 42 35 COc1cccc(C(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217726207 DF For-Sale Unstable DRD4 53 40 COc1cccc(C(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217726207 DF For-Sale Unstable DRD3 15 41 COc1cccc(C(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217726207 DF For-Sale Unstable MTNR1B 23 40 COc1cccc(C(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217726207 DF For-Sale Unstable CHRNA10 50 42 COc1cccc(C(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217726207 DF For-Sale Unstable ACKR3 65 35 N[C@H](C(=O)N[C@H]1CCN2CCC[C@@H]12)c1ccccc1 ZINC000217726221 CD For-Sale Unstable SLC18A3 59 36 COc1cccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c1 ZINC000217726228 JI In-Stock Unstable AKR1B1 0 46 COc1cccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c1 ZINC000217726228 JI In-Stock Unstable CYP1B1 58 37 COc1cccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c1 ZINC000217726228 JI In-Stock Unstable CYP1A1 46 46 COc1ccccc1/C=C/NC(=O)NCCCCCO ZINC000217726231 CE For-Sale Unstable DRD2 17 46 COc1ccccc1/C=C/NC(=O)NCCCCCO ZINC000217726231 CE For-Sale Unstable DRD3 33 46 Cc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1C ZINC000217726290 EF In-Stock Unstable ADORA2B 41 39 Cc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1C ZINC000217726290 EF In-Stock Unstable MCHR1 17 43 Cc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1C ZINC000217726290 EF In-Stock Unstable MCHR2 41 41 Cc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1C ZINC000217726290 EF In-Stock Unstable HIF1A 24 42 Cc1cccc2c(=O)n(C)c(Br)nc12 ZINC000217726301 CE For-Sale Unstable TNKS 34 44 Cc1cccc2c(=O)n(C)c(Br)nc12 ZINC000217726301 CE For-Sale Unstable TNKS2 22 44 COc1cccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c1 ZINC000217726303 JI In-Stock Unstable AKR1B1 0 46 COc1cccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c1 ZINC000217726303 JI In-Stock Unstable CYP1B1 58 37 COc1cccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c1 ZINC000217726303 JI In-Stock Unstable CYP1A1 46 46 Cc1cc(C)cc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217726403 EF In-Stock Unstable HIF1A 20 40 CCCCNS(=O)(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217726440 DD For-Sale Unstable LTB4R 26 41 CCCCNS(=O)(=O)c1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217726440 DD For-Sale Unstable IAP 0 43 COc1ccccc1/C=C/NC(=O)Nc1cccnc1 ZINC000217726450 CF For-Sale Unstable NAMPT 21 43 CC(=O)NCC1CCN([C@@H](C)C(=O)OC(C)(C)C)CC1 ZINC000217726486 CD On-Demand Unstable CACNA1I 48 34 CCCCNS(=O)(=O)c1ccc(/C=C\C(=O)O)cc1Cl ZINC000217726511 DF For-Sale Unstable PYGL 17 42 O=C(OCCC1CC1)c1ccc(NCCO)cc1 ZINC000217726536 BE On-Demand Unstable ACR 45 34 O=C(OCCC1CC1)c1ccc(NCCO)cc1 ZINC000217726536 BE On-Demand Unstable CNGA1 0 47 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccccc1F ZINC000217726538 EE In-Stock Unstable FABH 0 43 CCN(CC)C(=O)N/C=C/c1ccccc1OC ZINC000217726544 BF For-Sale Unstable CYP1B1 19 41 CCN(CC)C(=O)N/C=C/c1ccccc1OC ZINC000217726544 BF For-Sale Unstable TLR4 19 47 CC(=O)NCC1CCN([C@H](C)C(=O)OC(C)(C)C)CC1 ZINC000217726558 CD On-Demand Unstable CACNA1I 48 34 O=C(O)/C=C\c1cccc(S(=O)(=O)NCC2CCC2)c1 ZINC000217726609 CD For-Sale Unstable NPY2R 63 41 O=C(O)/C=C\c1cccc(S(=O)(=O)NCC2CCC2)c1 ZINC000217726609 CD For-Sale Unstable HDAC8 23 48 O=C(O)/C=C\c1cccc(S(=O)(=O)NCC2CCC2)c1 ZINC000217726609 CD For-Sale Unstable NPY5R 19 41 O=C(O)/C=C\c1cccc(S(=O)(=O)NCC2CCC2)c1 ZINC000217726609 CD For-Sale Unstable SFRP1 40 32 CC(=O)c1ccc(C(=O)Nc2ccc3nc[nH]c3c2)cc1 ZINC000217726629 CG On-Demand Unstable MAOB 17 40 CC(=O)c1ccc(C(=O)Nc2ccc3nc[nH]c3c2)cc1 ZINC000217726629 CG On-Demand Unstable PRNP 49 47 CC(=O)c1ccc(C(=O)Nc2ccc3nc[nH]c3c2)cc1 ZINC000217726629 CG On-Demand Unstable AKR1C3 18 40 CC(=O)c1ccc(C(=O)Nc2ccc3nc[nH]c3c2)cc1 ZINC000217726629 CG On-Demand Unstable KCNK3 76 40 CC(=O)c1ccc(C(=O)Nc2ccc3nc[nH]c3c2)cc1 ZINC000217726629 CG On-Demand Unstable KCNK9 41 37 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(F)cc1 ZINC000217726657 EE In-Stock Unstable ADORA2A 0 45 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(F)cc1 ZINC000217726657 EE In-Stock Unstable ADORA2B 50 45 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(F)cc1 ZINC000217726657 EE In-Stock Unstable CETP 0 46 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(F)cc1 ZINC000217726657 EE In-Stock Unstable HIF1A 24 41 CCN1Cc2ccccc2C[C@@H]1C(=O)N1CCC(c2ccnc(N)n2)CC1 ZINC000217726685 FE In-Stock Unstable PREP 31 42 CCN1Cc2ccccc2C[C@@H]1C(=O)N1CCC(c2ccnc(N)n2)CC1 ZINC000217726685 FE In-Stock Unstable ADAM9 60 34 Cc1cc(S(=O)(=O)NCC2CCC2)ccc1/C=C\C(=O)O ZINC000217726687 DE For-Sale Unstable NPY2R 46 39 Nc1cncc(C(=O)NCC2CC2)c1 ZINC000217726711 AC In-Stock Unstable GRIN2B 0 42 Nc1cncc(C(=O)NCC2CC2)c1 ZINC000217726711 AC In-Stock Unstable CACNA1I 50 41 Nc1cncc(C(=O)NCC2CC2)c1 ZINC000217726711 AC In-Stock Unstable HSPB1 0 40 COc1ccc(CN2C(=O)N[C@@H](CCC(=O)NCCc3ccc(O)cc3)C2=O)cc1OC ZINC000217726712 ID In-Stock Unstable IAP 0 40 COc1ccc(CN2C(=O)N[C@@H](CCC(=O)NCCc3ccc(O)cc3)C2=O)cc1OC ZINC000217726712 ID In-Stock Unstable CAN2 0 46 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccccc1Cl ZINC000217726779 EF In-Stock Unstable EPHB3 46 39 Cc1ccc(/C=C\C(=O)O)cc1S(=O)(=O)NCC1CCC1 ZINC000217726780 DE For-Sale Unstable NPY2R 45 33 CCN1Cc2ccccc2C[C@H]1C(=O)N1CCC(c2ccnc(N)n2)CC1 ZINC000217726791 FE In-Stock Unstable PREP 31 42 CCN1Cc2ccccc2C[C@H]1C(=O)N1CCC(c2ccnc(N)n2)CC1 ZINC000217726791 FE In-Stock Unstable ADAM9 60 34 CCC[C@@H]1CCN(C(=O)c2ccc3c(c2)CC(=O)N3)C1 ZINC000217726794 CE For-Sale Unstable L3MBTL3 49 33 CN(C(=O)c1cccc(/C=C\C(=O)O)c1)C1CCCC1 ZINC000217726860 CF For-Sale Unstable ACE 44 43 CCC[C@H]1CCN(C(=O)c2ccc3c(c2)CC(=O)N3)C1 ZINC000217726878 CE For-Sale Unstable L3MBTL3 49 33 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cccc(Cl)c1 ZINC000217726898 EF In-Stock Unstable PPIA 25 41 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cccc(Cl)c1 ZINC000217726898 EF In-Stock Unstable PTGER1 20 42 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cccc(Cl)c1 ZINC000217726898 EF In-Stock Unstable UL80 25 43 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cccc(Cl)c1 ZINC000217726898 EF In-Stock Unstable CETP 0 44 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cccc(Cl)c1 ZINC000217726898 EF In-Stock Unstable CAMK2D 16 43 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cccc(Cl)c1 ZINC000217726898 EF In-Stock Unstable PTPN22 23 43 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cccc(Cl)c1 ZINC000217726898 EF In-Stock Unstable MCHR1 19 40 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cccc(Cl)c1 ZINC000217726898 EF In-Stock Unstable HIF1A 25 49 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cccc(Cl)c1 ZINC000217726898 EF In-Stock Unstable TAAR1 19 44 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cccc(Cl)c1 ZINC000217726898 EF In-Stock Unstable AKR1C3 39 50 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cccc(Cl)c1 ZINC000217726898 EF In-Stock Unstable KCNK3 56 37 CN(C(=O)c1cc(/C=C\C(=O)O)ccc1F)C1CCCC1 ZINC000217726948 CF For-Sale Unstable ACE 45 34 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccc(Cl)cc1 ZINC000217726955 DG For-Sale Unstable CACNA1I 57 33 C=CCNC(=O)N/C=C/c1ccccc1OC ZINC000217726957 BE For-Sale Unstable KCNA3 22 42 C=CCNC(=O)N/C=C/c1ccccc1OC ZINC000217726957 BE For-Sale Unstable TLR4 15 44 COC(=O)[C@@H](O)CNC(=O)Cc1ccc(OC)c(F)c1 ZINC000217726960 CC On-Demand Unstable TRPV1 25 43 COC(=O)[C@@H](O)CNC(=O)Cc1ccc(OC)c(F)c1 ZINC000217726960 CC On-Demand Unstable CAN2 0 40 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Cl)cc1 ZINC000217727002 EF In-Stock Unstable LTA4H 27 44 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Cl)cc1 ZINC000217727002 EF In-Stock Unstable PTGER1 19 44 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Cl)cc1 ZINC000217727002 EF In-Stock Unstable ADORA2B 42 44 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Cl)cc1 ZINC000217727002 EF In-Stock Unstable CETP 0 49 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Cl)cc1 ZINC000217727002 EF In-Stock Unstable ACR 31 41 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Cl)cc1 ZINC000217727002 EF In-Stock Unstable HIF1A 24 41 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Cl)cc1 ZINC000217727002 EF In-Stock Unstable AKR1C3 20 42 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Cl)cc1 ZINC000217727002 EF In-Stock Unstable Q25615_ONCVO 31 41 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Cl)cc1 ZINC000217727002 EF In-Stock Unstable SENP1 0 41 O=C(NC[C@H]1CCCN1c1nccs1)c1ccc(Cl)cc1 ZINC000217727041 DG For-Sale Unstable CACNA1I 57 33 COC(=O)[C@H](O)CNC(=O)Cc1ccc(OC)c(F)c1 ZINC000217727043 CC On-Demand Unstable TRPV1 25 43 COC(=O)[C@H](O)CNC(=O)Cc1ccc(OC)c(F)c1 ZINC000217727043 CC On-Demand Unstable CAN2 0 40 CCC[C@@H]1CCN(C(=O)c2ccc(N)c([N+](=O)[O-])c2)C1 ZINC000217727045 CE For-Sale Unstable L3MBTL3 44 45 Nc1cc(C(=O)N[C@@H]2CCN3CCC[C@@H]23)ccc1Cl ZINC000217727098 CD For-Sale Unstable HTR3A 24 43 Nc1cc(C(=O)N[C@@H]2CCN3CCC[C@@H]23)ccc1Cl ZINC000217727098 CD For-Sale Unstable HTR4 34 43 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Br)cc1 ZINC000217727118 GF In-Stock Unstable ADORA2B 43 44 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Br)cc1 ZINC000217727118 GF In-Stock Unstable UL80 20 42 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Br)cc1 ZINC000217727118 GF In-Stock Unstable ACR 33 41 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Br)cc1 ZINC000217727118 GF In-Stock Unstable HIF1A 24 41 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Br)cc1 ZINC000217727118 GF In-Stock Unstable AKR1C3 15 42 CCC[C@H]1CCN(C(=O)c2ccc(N)c([N+](=O)[O-])c2)C1 ZINC000217727126 CE For-Sale Unstable L3MBTL3 44 45 COc1ccccc1/C=C/NC(=O)Nc1cccc(NC(C)=O)c1 ZINC000217727179 EG For-Sale Unstable CYP1B1 25 40 COc1ccccc1/C=C/NC(=O)Nc1cccc(NC(C)=O)c1 ZINC000217727179 EG For-Sale Unstable MTNR1B 15 44 COc1ccccc1/C=C/NC(=O)Nc1cccc(NC(C)=O)c1 ZINC000217727179 EG For-Sale Unstable CYP1A1 17 42 COc1ccccc1/C=C/NC(=O)Nc1cccc(NC(C)=O)c1 ZINC000217727179 EG For-Sale Unstable IMPDH2 0 43 COc1ccccc1/C=C/NC(=O)Nc1cccc(NC(C)=O)c1 ZINC000217727179 EG For-Sale Unstable KCNK3 118 49 COc1ccccc1/C=C/NC(=O)Nc1cccc(NC(C)=O)c1 ZINC000217727179 EG For-Sale Unstable KCNK9 87 49 Nc1cc(C(=O)N[C@H]2CCN3CCC[C@@H]23)ccc1Cl ZINC000217727196 CD For-Sale Unstable HTR3A 24 43 Nc1cc(C(=O)N[C@H]2CCN3CCC[C@@H]23)ccc1Cl ZINC000217727196 CD For-Sale Unstable HTR4 34 43 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)NC3CC3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217727235 JF In-Stock Unstable TUBA1A 20 75 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)NC3CC3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217727235 JF In-Stock Unstable SLC22A3 0 71 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)NC3CC3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217727235 JF In-Stock Unstable TPPP 0 71 Cc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1Cl ZINC000217727244 FG In-Stock Unstable DHODH 18 44 Cc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1Cl ZINC000217727244 FG In-Stock Unstable CETP 0 42 Cc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1Cl ZINC000217727244 FG In-Stock Unstable MCHR1 23 45 Cc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1Cl ZINC000217727244 FG In-Stock Unstable MCHR2 43 40 Cc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1Cl ZINC000217727244 FG In-Stock Unstable HIF1A 20 41 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727316 CC For-Sale Unstable F2 25 48 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727316 CC For-Sale Unstable PLG 15 40 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727316 CC For-Sale Unstable PRSS1 18 40 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727316 CC For-Sale Unstable ACE 81 44 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727316 CC For-Sale Unstable OPRM1 89 46 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727316 CC For-Sale Unstable OPRD1 80 46 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727316 CC For-Sale Unstable OPRK1 26 42 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727316 CC For-Sale Unstable MME 90 44 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727316 CC For-Sale Unstable ANPEP 63 37 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727316 CC For-Sale Unstable TACR1 19 44 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727316 CC For-Sale Unstable SIGMAR1 20 40 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727316 CC For-Sale Unstable SLC15A1 0 46 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727316 CC For-Sale Unstable DPP4 25 48 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727316 CC For-Sale Unstable SLC18A3 53 36 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727316 CC For-Sale Unstable PEPD 0 41 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727316 CC For-Sale Unstable YARS 60 40 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727316 CC For-Sale Unstable ACE2 44 35 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727316 CC For-Sale Unstable DPP7 56 39 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727316 CC For-Sale Unstable LAP3 49 38 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727316 CC For-Sale Unstable CTSC 23 42 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727316 CC For-Sale Unstable POL 0 44 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727316 CC For-Sale Unstable AMP1_PLAFQ 51 38 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727316 CC For-Sale Unstable XIAP 55 38 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727316 CC For-Sale Unstable DPP8 35 47 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727316 CC For-Sale Unstable DPP9 23 47 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727316 CC For-Sale Unstable FAP 0 42 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727316 CC For-Sale Unstable SLC15A2 0 46 O=C(O)/C=C\c1cnc(NC(=O)c2ccc(F)c(F)c2)s1 ZINC000217727327 DF For-Sale Anodyne SCD 28 43 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Cl)c(Cl)c1 ZINC000217727347 GG In-Stock Unstable CETP 0 43 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Cl)c(Cl)c1 ZINC000217727347 GG In-Stock Unstable KMO 0 40 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Cl)c(Cl)c1 ZINC000217727347 GG In-Stock Unstable MCHR1 17 42 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Cl)c(Cl)c1 ZINC000217727347 GG In-Stock Unstable HIF1A 25 42 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Cl)c(Cl)c1 ZINC000217727347 GG In-Stock Unstable SHH 23 40 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Cl)c(Cl)c1 ZINC000217727347 GG In-Stock Unstable PFK 0 43 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Cl)c(Cl)c1 ZINC000217727347 GG In-Stock Unstable P95276_MYCTO 0 43 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Cl)c(Cl)c1 ZINC000217727347 GG In-Stock Unstable PPX1 0 42 COC(=O)[C@@H](O)CNC(=O)Cn1ccc(=O)[nH]c1=O ZINC000217727371 CA For-Sale Unstable Q8II92_PLAF7 54 36 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727404 CC For-Sale Unstable F2 25 48 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727404 CC For-Sale Unstable PLG 15 40 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727404 CC For-Sale Unstable PRSS1 18 40 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727404 CC For-Sale Unstable ACE 81 44 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727404 CC For-Sale Unstable OPRM1 89 46 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727404 CC For-Sale Unstable OPRD1 80 46 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727404 CC For-Sale Unstable OPRK1 26 42 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727404 CC For-Sale Unstable MME 90 44 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727404 CC For-Sale Unstable ANPEP 63 37 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727404 CC For-Sale Unstable TACR1 19 44 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727404 CC For-Sale Unstable SIGMAR1 20 40 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727404 CC For-Sale Unstable SLC15A1 0 46 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727404 CC For-Sale Unstable DPP4 25 48 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727404 CC For-Sale Unstable SLC18A3 53 36 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727404 CC For-Sale Unstable PEPD 0 41 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727404 CC For-Sale Unstable YARS 60 40 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727404 CC For-Sale Unstable ACE2 44 35 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727404 CC For-Sale Unstable DPP7 56 39 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727404 CC For-Sale Unstable LAP3 49 38 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727404 CC For-Sale Unstable CTSC 23 42 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727404 CC For-Sale Unstable POL 0 44 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727404 CC For-Sale Unstable AMP1_PLAFQ 51 38 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727404 CC For-Sale Unstable XIAP 55 38 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727404 CC For-Sale Unstable DPP8 35 47 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727404 CC For-Sale Unstable DPP9 23 47 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727404 CC For-Sale Unstable FAP 0 42 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727404 CC For-Sale Unstable SLC15A2 0 46 CC(=O)Nc1ccc2c(O)cc(S(=O)(=O)Cl)cc2c1 ZINC000217727434 CE For-Sale Unstable CA12 15 40 CC(=O)[C@@H](NC(=O)CN1CCc2ccc(F)cc21)C(C)C ZINC000217727441 CD On-Demand Unstable ELANE 43 39 COC(=O)[C@H](O)CNC(=O)Cn1ccc(=O)[nH]c1=O ZINC000217727449 CA For-Sale Unstable Q8II92_PLAF7 54 36 Cc1ccc(/C=C\C(=O)Nc2cnccc2C(=O)O)s1 ZINC000217727450 CF For-Sale Unstable SCAF_EBVB9 19 40 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cc(Cl)cc(Cl)c1 ZINC000217727461 GG In-Stock Unstable HIF1A 19 40 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cc(Cl)cc(Cl)c1 ZINC000217727461 GG In-Stock Unstable HCAR1 0 41 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727484 CC For-Sale Unstable F2 25 48 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727484 CC For-Sale Unstable PLG 15 40 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727484 CC For-Sale Unstable PRSS1 18 40 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727484 CC For-Sale Unstable ACE 81 44 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727484 CC For-Sale Unstable OPRM1 89 46 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727484 CC For-Sale Unstable OPRD1 80 46 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727484 CC For-Sale Unstable OPRK1 26 42 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727484 CC For-Sale Unstable MME 90 44 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727484 CC For-Sale Unstable ANPEP 63 37 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727484 CC For-Sale Unstable TACR1 19 44 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727484 CC For-Sale Unstable SIGMAR1 20 40 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727484 CC For-Sale Unstable SLC15A1 0 46 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727484 CC For-Sale Unstable DPP4 25 48 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727484 CC For-Sale Unstable SLC18A3 53 36 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727484 CC For-Sale Unstable PEPD 0 41 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727484 CC For-Sale Unstable YARS 60 40 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727484 CC For-Sale Unstable ACE2 44 35 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727484 CC For-Sale Unstable DPP7 56 39 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727484 CC For-Sale Unstable LAP3 49 38 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727484 CC For-Sale Unstable CTSC 23 42 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727484 CC For-Sale Unstable POL 0 44 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727484 CC For-Sale Unstable AMP1_PLAFQ 51 38 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727484 CC For-Sale Unstable XIAP 55 38 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727484 CC For-Sale Unstable DPP8 35 47 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727484 CC For-Sale Unstable DPP9 23 47 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727484 CC For-Sale Unstable FAP 0 42 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727484 CC For-Sale Unstable SLC15A2 0 46 CC(=O)[C@H](NC(=O)CN1CCc2ccc(F)cc21)C(C)C ZINC000217727513 CD On-Demand Unstable ELANE 43 39 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727559 CC For-Sale Unstable F2 25 48 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727559 CC For-Sale Unstable PLG 15 40 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727559 CC For-Sale Unstable PRSS1 18 40 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727559 CC For-Sale Unstable ACE 81 44 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727559 CC For-Sale Unstable OPRM1 89 46 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727559 CC For-Sale Unstable OPRD1 80 46 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727559 CC For-Sale Unstable OPRK1 26 42 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727559 CC For-Sale Unstable MME 90 44 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727559 CC For-Sale Unstable ANPEP 63 37 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727559 CC For-Sale Unstable TACR1 19 44 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727559 CC For-Sale Unstable SIGMAR1 20 40 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727559 CC For-Sale Unstable SLC15A1 0 46 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727559 CC For-Sale Unstable DPP4 25 48 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727559 CC For-Sale Unstable SLC18A3 53 36 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727559 CC For-Sale Unstable PEPD 0 41 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727559 CC For-Sale Unstable YARS 60 40 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727559 CC For-Sale Unstable ACE2 44 35 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727559 CC For-Sale Unstable DPP7 56 39 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727559 CC For-Sale Unstable LAP3 49 38 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727559 CC For-Sale Unstable CTSC 23 42 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727559 CC For-Sale Unstable POL 0 44 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727559 CC For-Sale Unstable AMP1_PLAFQ 51 38 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727559 CC For-Sale Unstable XIAP 55 38 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727559 CC For-Sale Unstable DPP8 35 47 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727559 CC For-Sale Unstable DPP9 23 47 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727559 CC For-Sale Unstable FAP 0 42 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217727559 CC For-Sale Unstable SLC15A2 0 46 O=C(NC[C@@H]1CCCN1c1nccs1)c1cc2ccccc2o1 ZINC000217727566 EG For-Sale Unstable CTSV 20 40 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cccc(C(F)(F)F)c1 ZINC000217727586 GG In-Stock Unstable DHODH 0 45 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cccc(C(F)(F)F)c1 ZINC000217727586 GG In-Stock Unstable PPIA 16 44 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cccc(C(F)(F)F)c1 ZINC000217727586 GG In-Stock Unstable KIT 15 42 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cccc(C(F)(F)F)c1 ZINC000217727586 GG In-Stock Unstable UL80 32 44 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cccc(C(F)(F)F)c1 ZINC000217727586 GG In-Stock Unstable RAF1 19 42 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cccc(C(F)(F)F)c1 ZINC000217727586 GG In-Stock Unstable HDAC10 15 52 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cccc(C(F)(F)F)c1 ZINC000217727586 GG In-Stock Unstable KDR 20 45 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cccc(C(F)(F)F)c1 ZINC000217727586 GG In-Stock Unstable SLC1A1 21 41 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cccc(C(F)(F)F)c1 ZINC000217727586 GG In-Stock Unstable SLC1A3 18 41 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cccc(C(F)(F)F)c1 ZINC000217727586 GG In-Stock Unstable EPHX2 19 45 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cccc(C(F)(F)F)c1 ZINC000217727586 GG In-Stock Unstable SLC1A2 35 41 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cccc(C(F)(F)F)c1 ZINC000217727586 GG In-Stock Unstable TEK 31 41 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cccc(C(F)(F)F)c1 ZINC000217727586 GG In-Stock Unstable MCHR1 25 43 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cccc(C(F)(F)F)c1 ZINC000217727586 GG In-Stock Unstable Q8MMZ8_EIMTE 22 42 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cccc(C(F)(F)F)c1 ZINC000217727586 GG In-Stock Unstable BTK 21 43 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cccc(C(F)(F)F)c1 ZINC000217727586 GG In-Stock Unstable BRAF 38 41 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cccc(C(F)(F)F)c1 ZINC000217727586 GG In-Stock Unstable HIF1A 25 47 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cccc(C(F)(F)F)c1 ZINC000217727586 GG In-Stock Unstable AKR1C3 28 52 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cccc(C(F)(F)F)c1 ZINC000217727586 GG In-Stock Unstable TRPM4 0 45 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cccc(C(F)(F)F)c1 ZINC000217727586 GG In-Stock Unstable KCNK3 69 49 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cccc(C(F)(F)F)c1 ZINC000217727586 GG In-Stock Unstable KCNK9 46 34 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1cccc(C(F)(F)F)c1 ZINC000217727586 GG In-Stock Unstable PDS 43 43 CC(=O)NCC(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217727592 CC For-Sale Unstable PTGER2 24 40 CC(=O)NCC(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217727592 CC For-Sale Unstable NR1H4 41 37 CC(=O)NCC(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217727592 CC For-Sale Unstable HSD17B2 25 40 CC(=O)NCC(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217727592 CC For-Sale Unstable AKR1C3 30 41 O=C(NC[C@H]1CCCN1c1nccs1)c1cc2ccccc2o1 ZINC000217727648 EG For-Sale Unstable CTSV 20 40 CC[C@@H](C)[C@@H](N)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727655 BC For-Sale Unstable TPP2 41 43 Cc1nc([C@@H]2CCCN(C(=O)c3ccc(-c4ccco4)cc3)C2)no1 ZINC000217727665 EH In-Stock Unstable RHOA 0 51 COc1ccccc1NC(=O)COc1cc(C(=O)O)cc(C(=O)O)c1 ZINC000217727695 EE In-Stock Unstable P2RX7 0 41 COc1ccccc1NC(=O)COc1cc(C(=O)O)cc(C(=O)O)c1 ZINC000217727695 EE In-Stock Unstable LTB4R 18 49 COc1ccccc1NC(=O)COc1cc(C(=O)O)cc(C(=O)O)c1 ZINC000217727695 EE In-Stock Unstable MTNR1B 17 44 COc1ccccc1NC(=O)COc1cc(C(=O)O)cc(C(=O)O)c1 ZINC000217727695 EE In-Stock Unstable PLA2G4B 46 38 COc1ccccc1NC(=O)COc1cc(C(=O)O)cc(C(=O)O)c1 ZINC000217727695 EE In-Stock Unstable ACAT 0 44 COc1ccccc1NC(=O)COc1cc(C(=O)O)cc(C(=O)O)c1 ZINC000217727695 EE In-Stock Unstable KCNK3 42 36 COc1cc([C@@H]2CC(=O)Oc3ccc(C(C)=O)c(O)c32)ccc1OCCc1ccccc1 ZINC000217727726 IJ In-Stock Unstable TSHR 42 34 CC[C@H](C)[C@@H](N)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727729 BC For-Sale Unstable TPP2 41 43 Cc1nc([C@H]2CCCN(C(=O)c3ccc(-c4ccco4)cc3)C2)no1 ZINC000217727736 EH In-Stock Unstable RHOA 0 51 COC(=O)[C@@H](O)CNC(=O)c1cc2ccccc2c(=O)[nH]1 ZINC000217727748 CB On-Demand Unstable CDC25B 0 40 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccc(Cl)s1 ZINC000217727767 EG For-Sale Unstable F10 22 43 COc1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217727804 EE In-Stock Unstable DRD4 45 34 COc1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217727804 EE In-Stock Unstable PDGFRB 18 42 COc1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217727804 EE In-Stock Unstable CCR3 15 40 COc1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217727804 EE In-Stock Unstable MTNR1A 33 51 COc1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217727804 EE In-Stock Unstable MTNR1B 34 51 COc1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217727804 EE In-Stock Unstable PLA2G4B 46 40 COc1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217727804 EE In-Stock Unstable ACR 24 40 COc1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217727804 EE In-Stock Unstable MCHR1 21 43 COc1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217727804 EE In-Stock Unstable HIF1A 22 48 COc1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217727804 EE In-Stock Unstable TAAR1 37 43 COc1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217727804 EE In-Stock Unstable AKR1C3 51 48 COc1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217727804 EE In-Stock Unstable AKR1C2 54 38 COc1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217727804 EE In-Stock Unstable PSBA 0 50 COc1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217727804 EE In-Stock Unstable ISPD 0 41 COc1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217727804 EE In-Stock Unstable KCNK3 69 53 COc1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217727804 EE In-Stock Unstable KCNK9 70 38 COc1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217727804 EE In-Stock Unstable BRPF1 0 41 CC[C@@H](C)[C@H](N)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727814 BC For-Sale Unstable TPP2 41 43 COc1cc([C@H]2CC(=O)Oc3ccc(C(C)=O)c(O)c32)ccc1OCCc1ccccc1 ZINC000217727822 IJ In-Stock Unstable TSHR 42 34 COC(=O)[C@H](O)CNC(=O)c1cc2ccccc2c(=O)[nH]1 ZINC000217727826 CB On-Demand Unstable CDC25B 0 40 O=C(NC[C@H]1CCCN1c1nccs1)c1ccc(Cl)s1 ZINC000217727833 EG For-Sale Unstable F10 22 43 CC[C@H](C)[C@H](N)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217727908 BC For-Sale Unstable TPP2 41 43 O=C(O)/C=C\c1cccc(NC(=O)c2cccnc2)c1 ZINC000217727929 CE For-Sale Anodyne TBXAS1 47 45 O=C(O)/C=C\c1cccc(NC(=O)c2cccnc2)c1 ZINC000217727929 CE For-Sale Anodyne CSF1R 21 47 O=C(O)/C=C\c1cccc(NC(=O)c2cccnc2)c1 ZINC000217727929 CE For-Sale Anodyne BRAF 15 42 O=C(O)/C=C\c1cccc(NC(=O)c2cccnc2)c1 ZINC000217727929 CE For-Sale Anodyne SIRT2 17 40 O=C(O)/C=C\c1cccc(NC(=O)c2cccnc2)c1 ZINC000217727929 CE For-Sale Anodyne NAMPT 16 51 O=C(O)/C=C\c1cccc(NC(=O)c2cccnc2)c1 ZINC000217727929 CE For-Sale Anodyne KCNK3 111 51 O=C(O)/C=C\c1cccc(NC(=O)c2cccnc2)c1 ZINC000217727929 CE For-Sale Anodyne KCNK9 57 43 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217727933 EE In-Stock Unstable ADORA1 18 40 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217727933 EE In-Stock Unstable ADORA2A 22 46 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217727933 EE In-Stock Unstable ADORA2B 51 40 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217727933 EE In-Stock Unstable CETP 0 48 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217727933 EE In-Stock Unstable HDAC8 32 45 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217727933 EE In-Stock Unstable MTNR1A 35 43 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217727933 EE In-Stock Unstable MTNR1B 35 50 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217727933 EE In-Stock Unstable PLA2G4B 53 38 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217727933 EE In-Stock Unstable P4HTM 0 42 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217727933 EE In-Stock Unstable ACR 49 34 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217727933 EE In-Stock Unstable CA12 15 44 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217727933 EE In-Stock Unstable CA9 21 44 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217727933 EE In-Stock Unstable MCHR1 23 50 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217727933 EE In-Stock Unstable HIF1A 25 43 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217727933 EE In-Stock Unstable AKR1C3 37 48 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217727933 EE In-Stock Unstable AKR1C2 57 43 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217727933 EE In-Stock Unstable ENPP1 49 30 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217727933 EE In-Stock Unstable ETHR 15 49 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217727933 EE In-Stock Unstable ISPD 0 43 O=C(/C=C\c1cccnc1)Nc1cnccc1C(=O)O ZINC000217728015 CD For-Sale Anodyne MMP2 20 47 O=C(/C=C\c1cccnc1)Nc1cnccc1C(=O)O ZINC000217728015 CD For-Sale Anodyne MMP9 17 47 O=C(/C=C\c1cccnc1)Nc1cnccc1C(=O)O ZINC000217728015 CD For-Sale Anodyne MMP1 23 47 O=C(/C=C\c1cccnc1)Nc1cnccc1C(=O)O ZINC000217728015 CD For-Sale Anodyne TRPM2 0 42 O=C(O)/C=C\c1ccc(NC(=O)c2ccc[nH]2)c(F)c1 ZINC000217728019 CF For-Sale Anodyne MMP1 0 43 N[C@@H](CC(=O)N[C@@H]1CCN2CCC[C@@H]12)c1ccccc1 ZINC000217728028 CD For-Sale Unstable SIGMAR1 17 44 N[C@@H](CC(=O)N[C@@H]1CCN2CCC[C@@H]12)c1ccccc1 ZINC000217728028 CD For-Sale Unstable DPP4 15 40 N[C@@H](CC(=O)N[C@@H]1CCN2CCC[C@@H]12)c1ccccc1 ZINC000217728028 CD For-Sale Unstable SLC18A3 47 35 CCOc1ccccc1NC(=O)COc1cc(C(=O)O)cc(C(=O)O)c1 ZINC000217728044 FE In-Stock Unstable PLA2G4B 56 37 CCOc1ccccc1NC(=O)COc1cc(C(=O)O)cc(C(=O)O)c1 ZINC000217728044 FE In-Stock Unstable FABH 0 40 CCOc1ccccc1NC(=O)COc1cc(C(=O)O)cc(C(=O)O)c1 ZINC000217728044 FE In-Stock Unstable HCN1 41 31 CCOc1ccccc1NC(=O)COc1cc(C(=O)O)cc(C(=O)O)c1 ZINC000217728044 FE In-Stock Unstable HCN4 40 31 N[C@H](CC(=O)N[C@@H]1CCN2CCC[C@@H]12)c1ccccc1 ZINC000217728121 CD For-Sale Unstable SIGMAR1 17 44 N[C@H](CC(=O)N[C@@H]1CCN2CCC[C@@H]12)c1ccccc1 ZINC000217728121 CD For-Sale Unstable DPP4 15 40 N[C@H](CC(=O)N[C@@H]1CCN2CCC[C@@H]12)c1ccccc1 ZINC000217728121 CD For-Sale Unstable SLC18A3 47 35 COc1ccc(-c2coc3ccc(OC/C=C/c4ccccc4)cc23)cc1OC ZINC000217728150 GK In-Stock Unstable CYP1B1 21 40 COc1ccc(-c2coc3ccc(OC/C=C/c4ccccc4)cc23)cc1OC ZINC000217728150 GK In-Stock Unstable CYP1A1 18 40 COC(=O)[C@@H](O)CNC(=O)/C=C/c1cccc(Cl)c1 ZINC000217728156 CD On-Demand Unstable PYGL 23 43 COC(=O)[C@@H](O)CNC(=O)/C=C/c1cccc(Cl)c1 ZINC000217728156 CD On-Demand Unstable HDAC8 51 37 COC(=O)[C@@H](O)CNC(=O)/C=C/c1cccc(Cl)c1 ZINC000217728156 CD On-Demand Unstable MMP2 0 48 COC(=O)[C@@H](O)CNC(=O)/C=C/c1cccc(Cl)c1 ZINC000217728156 CD On-Demand Unstable NR1H4 41 45 COC(=O)[C@@H](O)CNC(=O)/C=C/c1cccc(Cl)c1 ZINC000217728156 CD On-Demand Unstable MMP9 0 48 COC(=O)[C@@H](O)CNC(=O)/C=C/c1cccc(Cl)c1 ZINC000217728156 CD On-Demand Unstable MMP1 0 48 COC(=O)[C@@H](O)CNC(=O)/C=C/c1cccc(Cl)c1 ZINC000217728156 CD On-Demand Unstable TUBA4A 0 42 CCOc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217728183 FE In-Stock Unstable SRD5A2 0 43 CCOc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217728183 FE In-Stock Unstable LTA4H 40 41 CCOc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217728183 FE In-Stock Unstable ADORA2A 0 46 CCOc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217728183 FE In-Stock Unstable ADORA2B 54 43 CCOc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217728183 FE In-Stock Unstable CETP 0 42 CCOc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217728183 FE In-Stock Unstable PLA2G4B 84 42 CCOc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217728183 FE In-Stock Unstable P4HTM 0 55 CCOc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217728183 FE In-Stock Unstable ACR 48 31 CCOc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217728183 FE In-Stock Unstable HIF1A 26 45 N[C@@H](CC(=O)N[C@H]1CCN2CCC[C@@H]12)c1ccccc1 ZINC000217728203 CD For-Sale Unstable SIGMAR1 17 44 N[C@@H](CC(=O)N[C@H]1CCN2CCC[C@@H]12)c1ccccc1 ZINC000217728203 CD For-Sale Unstable DPP4 15 40 N[C@@H](CC(=O)N[C@H]1CCN2CCC[C@@H]12)c1ccccc1 ZINC000217728203 CD For-Sale Unstable SLC18A3 47 35 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217728284 HH In-Stock Unstable EPHX1 0 45 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217728284 HH In-Stock Unstable SRD5A2 33 45 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217728284 HH In-Stock Unstable LTA4H 72 51 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217728284 HH In-Stock Unstable ADORA2A 0 41 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217728284 HH In-Stock Unstable ADORA2B 44 41 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217728284 HH In-Stock Unstable CA1 28 43 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217728284 HH In-Stock Unstable ACOX1 18 40 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217728284 HH In-Stock Unstable CETP 0 43 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217728284 HH In-Stock Unstable SCN2A 15 49 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217728284 HH In-Stock Unstable GUAB 0 40 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217728284 HH In-Stock Unstable RAF1 39 42 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217728284 HH In-Stock Unstable MTNR1B 15 52 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217728284 HH In-Stock Unstable PLA2G4B 47 39 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217728284 HH In-Stock Unstable NPY5R 22 40 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217728284 HH In-Stock Unstable CFTR 42 41 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217728284 HH In-Stock Unstable ACR 52 38 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217728284 HH In-Stock Unstable SLC1A2 29 40 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217728284 HH In-Stock Unstable FABH 0 43 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217728284 HH In-Stock Unstable MCHR1 26 40 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217728284 HH In-Stock Unstable Q8MMZ8_EIMTE 55 42 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217728284 HH In-Stock Unstable F13A1 22 41 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217728284 HH In-Stock Unstable HIF1A 25 45 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217728284 HH In-Stock Unstable AKR1C3 21 49 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217728284 HH In-Stock Unstable YOPH 0 42 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217728284 HH In-Stock Unstable CRTM 44 34 O=C(COc1cc(C(=O)O)cc(C(=O)O)c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217728284 HH In-Stock Unstable PFKFB3 52 38 N[C@H](CC(=O)N[C@H]1CCN2CCC[C@@H]12)c1ccccc1 ZINC000217728293 CD For-Sale Unstable SIGMAR1 17 44 N[C@H](CC(=O)N[C@H]1CCN2CCC[C@@H]12)c1ccccc1 ZINC000217728293 CD For-Sale Unstable DPP4 15 40 N[C@H](CC(=O)N[C@H]1CCN2CCC[C@@H]12)c1ccccc1 ZINC000217728293 CD For-Sale Unstable SLC18A3 47 35 COC(=O)[C@@H](O)CNC(=O)/C=C/c1cccc([N+](=O)[O-])c1 ZINC000217728358 CC On-Demand Unstable CACNA1C 57 42 COC(=O)[C@@H](O)CNC(=O)/C=C/c1cccc([N+](=O)[O-])c1 ZINC000217728358 CC On-Demand Unstable CACNA1D 92 42 COC(=O)[C@@H](O)CNC(=O)/C=C/c1cccc([N+](=O)[O-])c1 ZINC000217728358 CC On-Demand Unstable HDAC8 36 40 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c(OC)c1 ZINC000217728392 GE In-Stock Unstable CYP1B1 20 57 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c(OC)c1 ZINC000217728392 GE In-Stock Unstable LTB4R 17 40 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c(OC)c1 ZINC000217728392 GE In-Stock Unstable PLA2G4B 47 40 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c(OC)c1 ZINC000217728392 GE In-Stock Unstable AKR1C3 27 40 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c(OC)c1 ZINC000217728392 GE In-Stock Unstable AKR1C2 53 40 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c(OC)c1 ZINC000217728392 GE In-Stock Unstable FAS 19 40 CCC[C@@H]1CCN(C(=O)c2cc(Cl)ccc2Br)C1 ZINC000217728393 EI For-Sale Unstable CACNA1I 41 31 CC(C)C[C@@H](N)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217728423 BC For-Sale Unstable AMPX_VIBPR 0 41 c1ccc(CN2CC[C@H](N[C@@H]3CCN4CCC[C@@H]34)C2)cc1 ZINC000217728429 CE For-Sale Unstable DRD4 42 46 c1ccc(CN2CC[C@H](N[C@@H]3CCN4CCC[C@@H]34)C2)cc1 ZINC000217728429 CE For-Sale Unstable ACHE 29 42 c1ccc(CN2CC[C@H](N[C@@H]3CCN4CCC[C@@H]34)C2)cc1 ZINC000217728429 CE For-Sale Unstable SIGMAR1 61 45 c1ccc(CN2CC[C@H](N[C@@H]3CCN4CCC[C@@H]34)C2)cc1 ZINC000217728429 CE For-Sale Unstable CCR3 16 40 c1ccc(CN2CC[C@H](N[C@@H]3CCN4CCC[C@@H]34)C2)cc1 ZINC000217728429 CE For-Sale Unstable SLC18A3 45 46 CCC[C@H]1CCN(C(=O)c2cc(Cl)ccc2Br)C1 ZINC000217728477 EI For-Sale Unstable CACNA1I 41 31 CC(C)C[C@H](N)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217728506 BC For-Sale Unstable AMPX_VIBPR 0 41 c1ccc(CN2CC[C@@H](N[C@@H]3CCN4CCC[C@@H]34)C2)cc1 ZINC000217728510 CE For-Sale Unstable DRD4 42 46 c1ccc(CN2CC[C@@H](N[C@@H]3CCN4CCC[C@@H]34)C2)cc1 ZINC000217728510 CE For-Sale Unstable ACHE 29 42 c1ccc(CN2CC[C@@H](N[C@@H]3CCN4CCC[C@@H]34)C2)cc1 ZINC000217728510 CE For-Sale Unstable SIGMAR1 61 45 c1ccc(CN2CC[C@@H](N[C@@H]3CCN4CCC[C@@H]34)C2)cc1 ZINC000217728510 CE For-Sale Unstable CCR3 16 40 c1ccc(CN2CC[C@@H](N[C@@H]3CCN4CCC[C@@H]34)C2)cc1 ZINC000217728510 CE For-Sale Unstable SLC18A3 45 46 COc1ccccc1/C=C/NC(=O)Nc1ccccc1N1CCOCC1 ZINC000217728518 FG For-Sale Unstable DRD2 29 43 COc1ccccc1/C=C/NC(=O)Nc1ccccc1N1CCOCC1 ZINC000217728518 FG For-Sale Unstable DRD3 39 43 COc1ccccc1/C=C/NC(=O)Nc1ccccc1N1CCOCC1 ZINC000217728518 FG For-Sale Unstable KCNQ2 80 40 COc1ccccc1/C=C/NC(=O)Nc1ccccc1N1CCOCC1 ZINC000217728518 FG For-Sale Unstable BRPF1 0 45 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccc2c(c1)OCO2 ZINC000217728560 EE For-Sale Unstable NOS2 86 40 COC(=O)[C@@H](O)CNC(=O)CSc1ccncc1 ZINC000217728562 CB On-Demand Unstable FAS 48 36 CC(C)C[C@@H](N)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217728600 BC For-Sale Unstable AMPX_VIBPR 0 41 Cc1cc(NC(=O)c2sccc2C)ccc1/C=C\C(=O)O ZINC000217728608 DH For-Sale Unstable KCNK3 50 35 COc1ccccc1/C=C/NC(=O)Nc1ccc(N2CCN(C)CC2)cc1 ZINC000217728615 FG For-Sale Unstable HTR1A 28 48 COc1ccccc1/C=C/NC(=O)Nc1ccc(N2CCN(C)CC2)cc1 ZINC000217728615 FG For-Sale Unstable DRD2 22 41 COc1ccccc1/C=C/NC(=O)Nc1ccc(N2CCN(C)CC2)cc1 ZINC000217728615 FG For-Sale Unstable HTR1D 23 48 COc1ccccc1/C=C/NC(=O)Nc1ccc(N2CCN(C)CC2)cc1 ZINC000217728615 FG For-Sale Unstable HTR1B 19 48 COc1ccccc1/C=C/NC(=O)Nc1ccc(N2CCN(C)CC2)cc1 ZINC000217728615 FG For-Sale Unstable DRD3 29 41 COc1ccccc1/C=C/NC(=O)Nc1ccc(N2CCN(C)CC2)cc1 ZINC000217728615 FG For-Sale Unstable HTR7 18 40 COc1ccccc1/C=C/NC(=O)Nc1ccc(N2CCN(C)CC2)cc1 ZINC000217728615 FG For-Sale Unstable LCK 18 45 COc1ccccc1/C=C/NC(=O)Nc1ccc(N2CCN(C)CC2)cc1 ZINC000217728615 FG For-Sale Unstable PRNP 44 47 COc1ccccc1/C=C/NC(=O)Nc1ccc(N2CCN(C)CC2)cc1 ZINC000217728615 FG For-Sale Unstable JAK2 15 40 COc1ccccc1/C=C/NC(=O)Nc1ccc(N2CCN(C)CC2)cc1 ZINC000217728615 FG For-Sale Unstable MTOR 22 41 COc1ccccc1/C=C/NC(=O)Nc1ccc(N2CCN(C)CC2)cc1 ZINC000217728615 FG For-Sale Unstable FLT3 15 41 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1Cl ZINC000217728624 GF In-Stock Unstable HTR2A 15 41 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1Cl ZINC000217728624 GF In-Stock Unstable COLA 56 37 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1Cl ZINC000217728624 GF In-Stock Unstable CPT1A 53 37 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1Cl ZINC000217728624 GF In-Stock Unstable CPT2 45 34 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1Cl ZINC000217728624 GF In-Stock Unstable GRM4 17 49 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1Cl ZINC000217728624 GF In-Stock Unstable CPT1B 41 34 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1Cl ZINC000217728624 GF In-Stock Unstable MCHR1 22 41 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1Cl ZINC000217728624 GF In-Stock Unstable MCHR2 40 41 COc1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1Cl ZINC000217728624 GF In-Stock Unstable ENPP1 73 37 COC(=O)[C@H](O)CNC(=O)CSc1ccncc1 ZINC000217728635 CB On-Demand Unstable FAS 48 36 O=C(NC[C@H]1CCCN1c1nccs1)c1ccc2c(c1)OCO2 ZINC000217728637 EE For-Sale Unstable NOS2 86 40 CCCCCC/C=C\SCCCC ZINC000217728641 BK For-Sale Unstable FABP3 23 41 CC(C)C[C@H](N)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217728688 BC For-Sale Unstable AMPX_VIBPR 0 41 Cc1cc(NC(=O)CC(C)(C)C)ccc1/C=C\C(=O)O ZINC000217728695 CG For-Sale Unstable ECE1 29 42 Oc1ccc2c(oc3c(-c4ccc5c(c4)OCCO5)c4cn[nH]c4nc32)c1O ZINC000217728714 GH In-Stock Unstable HSP82 0 41 COc1ccccc1/C=C/NC(=O)Nc1ccc(N2CCCCC2)cc1 ZINC000217728730 FI For-Sale Unstable KCNQ2 16 42 COc1ccccc1/C=C/NC(=O)Nc1ccc(N2CCCCC2)cc1 ZINC000217728730 FI For-Sale Unstable PRNP 41 35 COC(=O)c1ccccc1NC(=O)COc1cc(C(=O)O)cc(C(=O)O)c1 ZINC000217728732 FD In-Stock Unstable BDKRB1 0 41 COC(=O)c1ccccc1NC(=O)COc1cc(C(=O)O)cc(C(=O)O)c1 ZINC000217728732 FD In-Stock Unstable PLA2G4B 44 34 COC(=O)c1ccccc1NC(=O)COc1cc(C(=O)O)cc(C(=O)O)c1 ZINC000217728732 FD In-Stock Unstable HCAR2 35 43 COC(=O)c1ccccc1NC(=O)COc1cc(C(=O)O)cc(C(=O)O)c1 ZINC000217728732 FD In-Stock Unstable FABH 0 43 COC(=O)c1ccccc1NC(=O)COc1cc(C(=O)O)cc(C(=O)O)c1 ZINC000217728732 FD In-Stock Unstable AKR1C2 55 37 COC(=O)c1ccccc1NC(=O)COc1cc(C(=O)O)cc(C(=O)O)c1 ZINC000217728732 FD In-Stock Unstable FAS 57 53 COC(=O)[C@@H](O)CNC(=O)COc1ccc(C)cc1 ZINC000217728735 CC On-Demand Unstable PLA2G4B 43 31 COc1ccc(CC(=O)NC[C@@H]2CCCN2c2nccs2)cc1 ZINC000217728739 EE For-Sale Unstable NOS2 28 42 CCC[C@@H]1CCN(C(=O)c2cccc(C)c2I)C1 ZINC000217728791 FH For-Sale Unstable CCR8 55 34 Cc1cc(NC(=O)Cc2cccs2)ccc1/C=C\C(=O)O ZINC000217728793 DG For-Sale Unstable CA5B 41 48 Cc1cc(NC(=O)Cc2cccs2)ccc1/C=C\C(=O)O ZINC000217728793 DG For-Sale Unstable CA5A 43 48 COC(=O)[C@H](O)CNC(=O)COc1ccc(C)cc1 ZINC000217728808 CC On-Demand Unstable PLA2G4B 43 31 COc1ccc(CC(=O)NC[C@H]2CCCN2c2nccs2)cc1 ZINC000217728829 EE For-Sale Unstable NOS2 28 42 CCC[C@H]1CCN(C(=O)c2cccc(C)c2I)C1 ZINC000217728857 FH For-Sale Unstable CCR8 55 34 COC(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217728870 FD In-Stock Unstable ADORA2A 0 42 COC(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217728870 FD In-Stock Unstable ADORA2B 44 45 COC(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217728870 FD In-Stock Unstable PLA2G4B 47 35 COC(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217728870 FD In-Stock Unstable P4HTM 0 41 COC(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217728870 FD In-Stock Unstable ACR 65 46 COC(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217728870 FD In-Stock Unstable HIF1A 24 43 COC(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217728870 FD In-Stock Unstable KDM3A 0 44 COC(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217728870 FD In-Stock Unstable KDM5C 0 44 CCOc1ccccc1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217728916 EF For-Sale Unstable HCN1 77 46 CCOc1ccccc1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217728916 EF For-Sale Unstable HCN4 66 44 Cc1ccc(/C=C\C(=O)Nc2cnccc2C(=O)O)cc1 ZINC000217728940 CF For-Sale Unstable MMP2 0 44 Cc1ccc(/C=C\C(=O)Nc2cnccc2C(=O)O)cc1 ZINC000217728940 CF For-Sale Unstable HDAC1 0 43 Cc1ccc(/C=C\C(=O)Nc2cnccc2C(=O)O)cc1 ZINC000217728940 CF For-Sale Unstable MMP9 0 49 Cc1ccc(/C=C\C(=O)Nc2cnccc2C(=O)O)cc1 ZINC000217728940 CF For-Sale Unstable MMP1 22 49 Cc1ccc(/C=C\C(=O)Nc2cnccc2C(=O)O)cc1 ZINC000217728940 CF For-Sale Unstable MCHR1 0 42 COc1ccc(Br)cc1CN[C@@H]1CCN2CCC[C@@H]12 ZINC000217728946 EF For-Sale Unstable TACR1 35 41 CCOc1ccccc1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217728987 EF For-Sale Unstable HCN1 77 46 CCOc1ccccc1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217728987 EF For-Sale Unstable HCN4 66 44 CCOC(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217728993 GE In-Stock Unstable PRSS1 0 40 CCOC(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217728993 GE In-Stock Unstable ADORA2A 0 51 CCOC(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217728993 GE In-Stock Unstable ADORA2B 45 39 CCOC(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217728993 GE In-Stock Unstable PLA2G4B 47 35 CCOC(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217728993 GE In-Stock Unstable ACR 75 40 CCOC(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217728993 GE In-Stock Unstable NOD2 17 40 Cc1cc(C(=O)N[C@@H]2CCN3CCC[C@@H]23)ccc1N ZINC000217729021 CD For-Sale Unstable L3MBTL3 47 35 C[C@@H](C(=O)OC(C)(C)C)N1CC[C@@H](N2CCCC2)C1 ZINC000217729023 CD On-Demand Unstable L3MBTL3 56 38 O=C(/C=C\c1cccc(F)c1)Nc1cnccc1C(=O)O ZINC000217729035 CF For-Sale Anodyne MMP2 0 55 O=C(/C=C\c1cccc(F)c1)Nc1cnccc1C(=O)O ZINC000217729035 CF For-Sale Anodyne MMP9 0 52 O=C(/C=C\c1cccc(F)c1)Nc1cnccc1C(=O)O ZINC000217729035 CF For-Sale Anodyne HPSE 44 36 O=C(/C=C\c1cccc(F)c1)Nc1cnccc1C(=O)O ZINC000217729035 CF For-Sale Anodyne MMP1 24 55 COc1ccc(Br)cc1CN[C@H]1CCN2CCC[C@@H]12 ZINC000217729039 EF For-Sale Unstable TACR1 35 41 COC(=O)[C@@H](O)CNC(=O)/C=C/c1ccccc1[N+](=O)[O-] ZINC000217729082 CC On-Demand Unstable COLA 62 32 COC(=O)[C@@H](O)CNC(=O)/C=C/c1ccccc1[N+](=O)[O-] ZINC000217729082 CC On-Demand Unstable TLR4 25 51 NS(=O)(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217729095 GC In-Stock Unstable CA2 166 57 NS(=O)(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217729095 GC In-Stock Unstable LTA4H 29 42 NS(=O)(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217729095 GC In-Stock Unstable CA6 25 46 NS(=O)(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217729095 GC In-Stock Unstable CA1 150 57 NS(=O)(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217729095 GC In-Stock Unstable CA7 82 52 NS(=O)(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217729095 GC In-Stock Unstable CA13 28 44 NS(=O)(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217729095 GC In-Stock Unstable CA5B 70 52 NS(=O)(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217729095 GC In-Stock Unstable CA4 135 53 NS(=O)(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217729095 GC In-Stock Unstable CA5A 75 52 NS(=O)(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217729095 GC In-Stock Unstable CA14 57 52 NS(=O)(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217729095 GC In-Stock Unstable ACR 42 31 NS(=O)(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217729095 GC In-Stock Unstable CDK1 0 40 NS(=O)(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217729095 GC In-Stock Unstable CA12 103 57 NS(=O)(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217729095 GC In-Stock Unstable CA9 115 57 NS(=O)(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217729095 GC In-Stock Unstable F13A1 42 32 NS(=O)(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217729095 GC In-Stock Unstable UREA_CANEN 28 44 NS(=O)(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217729095 GC In-Stock Unstable CYNT 44 45 NS(=O)(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217729095 GC In-Stock Unstable NCE103 63 46 NS(=O)(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217729095 GC In-Stock Unstable MTCA1 58 47 NS(=O)(=O)c1ccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)cc1 ZINC000217729095 GC In-Stock Unstable P96878_MYCTU 72 47 Cc1cc(C(=O)N[C@H]2CCN3CCC[C@@H]23)ccc1N ZINC000217729098 CD For-Sale Unstable L3MBTL3 47 35 C[C@H](C(=O)OC(C)(C)C)N1CC[C@@H](N2CCCC2)C1 ZINC000217729110 CD On-Demand Unstable L3MBTL3 56 38 COc1ccccc1/C=C/NC(=O)NCCO ZINC000217729111 BC For-Sale Unstable DRD3 19 42 COc1ccccc1/C=C/NC(=O)NCCO ZINC000217729111 BC For-Sale Unstable CYP1B1 19 40 COc1ccccc1/C=C/NC(=O)NCCO ZINC000217729111 BC For-Sale Unstable TLR4 19 45 CCCCCC(=O)N[C@@H](C)c1cccc(/C=C\C(=O)O)c1 ZINC000217729133 CH For-Sale Unstable SOAT1 32 43 CCCCCC(=O)N[C@@H](C)c1cccc(/C=C\C(=O)O)c1 ZINC000217729133 CH For-Sale Unstable AKR1C3 26 41 CCCCCC(=O)N[C@@H](C)c1cccc(/C=C\C(=O)O)c1 ZINC000217729133 CH For-Sale Unstable NOD1 79 41 CC(=O)c1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217729197 FE In-Stock Unstable ADORA2B 31 48 CC(=O)c1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217729197 FE In-Stock Unstable PLA2G4B 42 41 CC(=O)c1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217729197 FE In-Stock Unstable HIF1A 31 55 CC(=O)c1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217729197 FE In-Stock Unstable AKR1C3 55 55 CC(=O)c1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217729197 FE In-Stock Unstable KCNK3 83 38 CC(=O)c1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217729197 FE In-Stock Unstable KCNK9 67 36 CC(=O)c1cccc(NC(=O)COc2cc(C(=O)O)cc(C(=O)O)c2)c1 ZINC000217729197 FE In-Stock Unstable PARP10 0 46 COc1ccccc1/C=C/NC(=O)Nc1cccc2ccccc12 ZINC000217729200 DJ For-Sale Unstable CHAT 51 33 COc1ccccc1/C=C/NC(=O)Nc1cccc2ccccc12 ZINC000217729200 DJ For-Sale Unstable TRPV1 40 42 COc1ccccc1/C=C/NC(=O)Nc1cccc2ccccc12 ZINC000217729200 DJ For-Sale Unstable MTNR1A 18 55 COc1ccccc1/C=C/NC(=O)Nc1cccc2ccccc12 ZINC000217729200 DJ For-Sale Unstable MTNR1B 27 51 CCCCCC(=O)N[C@H](C)c1cccc(/C=C\C(=O)O)c1 ZINC000217729223 CH For-Sale Unstable SOAT1 32 43 CCCCCC(=O)N[C@H](C)c1cccc(/C=C\C(=O)O)c1 ZINC000217729223 CH For-Sale Unstable AKR1C3 26 41 CCCCCC(=O)N[C@H](C)c1cccc(/C=C\C(=O)O)c1 ZINC000217729223 CH For-Sale Unstable NOD1 79 41 COc1ccnc(CNC(=O)[C@H](CC(C)C)NC(C)=O)c1 ZINC000217729279 CD In-Stock Unstable ANPEP 38 47 COc1ccnc(CNC(=O)[C@H](CC(C)C)NC(C)=O)c1 ZINC000217729279 CD In-Stock Unstable CTSK 23 42 COc1ccnc(CNC(=O)[C@H](CC(C)C)NC(C)=O)c1 ZINC000217729279 CD In-Stock Unstable CTSL 21 43 COc1ccnc(CNC(=O)[C@H](CC(C)C)NC(C)=O)c1 ZINC000217729279 CD In-Stock Unstable CTSS 26 43 COc1ccnc(CNC(=O)[C@H](CC(C)C)NC(C)=O)c1 ZINC000217729279 CD In-Stock Unstable CAPN1 42 42 COc1ccnc(CNC(=O)[C@H](CC(C)C)NC(C)=O)c1 ZINC000217729279 CD In-Stock Unstable CAPN2 41 38 COc1ccnc(CNC(=O)[C@H](CC(C)C)NC(C)=O)c1 ZINC000217729279 CD In-Stock Unstable HPN 69 38 COC(=O)[C@@H](O)CNC(=O)Cc1ccc([N+](=O)[O-])cc1 ZINC000217729293 CB On-Demand Unstable CACNA1D 63 33 COC(=O)[C@@H](O)CNC(=O)Cc1ccc([N+](=O)[O-])cc1 ZINC000217729293 CB On-Demand Unstable CCR3 0 46 COC(=O)[C@@H](O)CNC(=O)Cc1ccc([N+](=O)[O-])cc1 ZINC000217729293 CB On-Demand Unstable MMP8 29 42 COC(=O)[C@@H](O)CNC(=O)Cc1ccc([N+](=O)[O-])cc1 ZINC000217729293 CB On-Demand Unstable MMP9 15 42 COC(=O)[C@@H](O)CNC(=O)Cc1ccc([N+](=O)[O-])cc1 ZINC000217729293 CB On-Demand Unstable MMP1 36 42 COc1cccc(CC(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217729301 EE For-Sale Unstable DRD4 40 31 COc1cccc(CC(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217729301 EE For-Sale Unstable CHRNA10 46 41 COc1cccc(CC(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217729301 EE For-Sale Unstable ACKR3 50 31 COC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217729307 EG For-Sale Unstable ACR 45 47 COC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217729307 EG For-Sale Unstable PDGFRA 48 35 COc1ccc2c(c1)O[C@H](c1ccc(OC)c(O)c1)CC2=O ZINC000217729318 DG Annotated Unstable CYP19A1 24 74 COc1ccc2c(c1)O[C@H](c1ccc(OC)c(O)c1)CC2=O ZINC000217729318 DG Annotated Unstable CYP1B1 15 63 COc1ccc2c(c1)O[C@H](c1ccc(OC)c(O)c1)CC2=O ZINC000217729318 DG Annotated Unstable HDAC2 21 40 COc1ccc2c(c1)O[C@H](c1ccc(OC)c(O)c1)CC2=O ZINC000217729318 DG Annotated Unstable MT-ND4 50 31 COc1ccc2c(c1)O[C@H](c1ccc(OC)c(O)c1)CC2=O ZINC000217729318 DG Annotated Unstable TAS2R31 0 55 O=c1cc(Cl)nc(C2CCCC2)[nH]1 ZINC000217729367 AE In-Stock Unstable ADORA1 24 42 Cc1cc(=O)oc2cc(OCC(=O)N[C@H](c3nc4ccccc4n3C)C(C)C)ccc12 ZINC000217729374 HH In-Stock Unstable MAOA 63 53 Cc1cc(=O)oc2cc(OCC(=O)N[C@H](c3nc4ccccc4n3C)C(C)C)ccc12 ZINC000217729374 HH In-Stock Unstable ACHE 19 47 Cc1cc(=O)oc2cc(OCC(=O)N[C@H](c3nc4ccccc4n3C)C(C)C)ccc12 ZINC000217729374 HH In-Stock Unstable MAOB 41 53 Cc1cc(=O)oc2cc(OCC(=O)N[C@H](c3nc4ccccc4n3C)C(C)C)ccc12 ZINC000217729374 HH In-Stock Unstable BCHE 23 47 COC(=O)[C@H](O)CNC(=O)Cc1ccc([N+](=O)[O-])cc1 ZINC000217729381 CB On-Demand Unstable CACNA1D 63 33 COC(=O)[C@H](O)CNC(=O)Cc1ccc([N+](=O)[O-])cc1 ZINC000217729381 CB On-Demand Unstable CCR3 0 46 COC(=O)[C@H](O)CNC(=O)Cc1ccc([N+](=O)[O-])cc1 ZINC000217729381 CB On-Demand Unstable MMP8 29 42 COC(=O)[C@H](O)CNC(=O)Cc1ccc([N+](=O)[O-])cc1 ZINC000217729381 CB On-Demand Unstable MMP9 15 42 COC(=O)[C@H](O)CNC(=O)Cc1ccc([N+](=O)[O-])cc1 ZINC000217729381 CB On-Demand Unstable MMP1 36 42 COc1cccc(CC(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217729388 EE For-Sale Unstable DRD4 40 31 COc1cccc(CC(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217729388 EE For-Sale Unstable CHRNA10 46 41 COc1cccc(CC(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217729388 EE For-Sale Unstable ACKR3 50 31 CCOC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729391 EF In-Stock Unstable PRSS1 0 46 CCOC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729391 EF In-Stock Unstable SRD5A2 35 48 CCOC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729391 EF In-Stock Unstable LTA4H 50 43 CCOC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729391 EF In-Stock Unstable ADORA2A 0 52 CCOC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729391 EF In-Stock Unstable RARB 25 41 CCOC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729391 EF In-Stock Unstable ADORA2B 48 43 CCOC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729391 EF In-Stock Unstable CA1 26 42 CCOC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729391 EF In-Stock Unstable CETP 0 41 CCOC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729391 EF In-Stock Unstable PLA2G4B 76 45 CCOC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729391 EF In-Stock Unstable P4HTM 0 51 CCOC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729391 EF In-Stock Unstable EPHX2 20 41 CCOC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729391 EF In-Stock Unstable ACR 82 44 CCOC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729391 EF In-Stock Unstable MCHR1 15 41 CCOC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729391 EF In-Stock Unstable MCHR2 37 41 CCOC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729391 EF In-Stock Unstable HIF1A 25 42 CCOC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729391 EF In-Stock Unstable NOD1 16 41 CCOC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729391 EF In-Stock Unstable NOD2 33 41 COc1ccccc1/C=C/NC(=O)N(Cc1ccccc1)c1ccccc1 ZINC000217729424 FK For-Sale Unstable NR1H4 37 41 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)Nc3cccc(O)c3)[C@H]21 ZINC000217729479 JH In-Stock Unstable TSHR 50 33 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729504 FD In-Stock Unstable CA2 140 60 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729504 FD In-Stock Unstable SRD5A2 27 45 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729504 FD In-Stock Unstable LTA4H 46 45 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729504 FD In-Stock Unstable ADORA2B 41 37 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729504 FD In-Stock Unstable CA6 26 55 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729504 FD In-Stock Unstable CA1 122 60 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729504 FD In-Stock Unstable CA7 73 53 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729504 FD In-Stock Unstable CA5B 69 53 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729504 FD In-Stock Unstable CA4 111 60 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729504 FD In-Stock Unstable CA5A 75 53 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729504 FD In-Stock Unstable CA14 59 46 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729504 FD In-Stock Unstable PLA2G4B 56 39 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729504 FD In-Stock Unstable P4HTM 0 43 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729504 FD In-Stock Unstable ACR 51 35 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729504 FD In-Stock Unstable CA12 95 54 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729504 FD In-Stock Unstable CA9 113 55 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729504 FD In-Stock Unstable F13A1 48 33 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729504 FD In-Stock Unstable HIF1A 24 42 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729504 FD In-Stock Unstable UREA_CANEN 27 42 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729504 FD In-Stock Unstable CYNT 46 49 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729504 FD In-Stock Unstable NCE103 61 55 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729504 FD In-Stock Unstable PFK 0 42 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729504 FD In-Stock Unstable MTCA1 46 54 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729504 FD In-Stock Unstable P96878_MYCTU 63 54 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729504 FD In-Stock Unstable CA 0 55 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2)cc1 ZINC000217729504 FD In-Stock Unstable Q5TU56_ANOGA 0 55 CCOc1ccccc1OCC(=O)NC[C@@H](O)C(=O)OC ZINC000217729518 CC On-Demand Unstable HCN1 40 32 CCOc1ccccc1OCC(=O)NC[C@@H](O)C(=O)OC ZINC000217729518 CC On-Demand Unstable HCN4 40 32 Cc1ccc(/C=C\C(=O)O)cc1NC(=O)c1ccccc1 ZINC000217729519 CG For-Sale Unstable EPHX1 0 43 Cc1ccc(/C=C\C(=O)O)cc1NC(=O)c1ccccc1 ZINC000217729519 CG For-Sale Unstable MAPK14 24 45 Cc1ccc(/C=C\C(=O)O)cc1NC(=O)c1ccccc1 ZINC000217729519 CG For-Sale Unstable HDAC8 17 41 Cc1ccc(/C=C\C(=O)O)cc1NC(=O)c1ccccc1 ZINC000217729519 CG For-Sale Unstable LDLR 0 44 Cc1ccc(/C=C\C(=O)O)cc1NC(=O)c1ccccc1 ZINC000217729519 CG For-Sale Unstable MMP2 0 47 Cc1ccc(/C=C\C(=O)O)cc1NC(=O)c1ccccc1 ZINC000217729519 CG For-Sale Unstable HDAC1 22 41 Cc1ccc(/C=C\C(=O)O)cc1NC(=O)c1ccccc1 ZINC000217729519 CG For-Sale Unstable HDAC2 17 42 Cc1ccc(/C=C\C(=O)O)cc1NC(=O)c1ccccc1 ZINC000217729519 CG For-Sale Unstable MMP9 0 47 Cc1ccc(/C=C\C(=O)O)cc1NC(=O)c1ccccc1 ZINC000217729519 CG For-Sale Unstable MMP1 0 47 Cc1ccc(/C=C\C(=O)O)cc1NC(=O)c1ccccc1 ZINC000217729519 CG For-Sale Unstable KCNK3 94 43 Cc1ccc(/C=C\C(=O)O)cc1NC(=O)c1ccccc1 ZINC000217729519 CG For-Sale Unstable KCNK9 48 43 COc1ccccc1/C=C/NC(=O)Nc1ccc2ccccc2c1 ZINC000217729531 DJ For-Sale Unstable CYP1B1 27 42 COc1ccccc1/C=C/NC(=O)Nc1ccc2ccccc2c1 ZINC000217729531 DJ For-Sale Unstable CA1 17 43 COc1ccccc1/C=C/NC(=O)Nc1ccc2ccccc2c1 ZINC000217729531 DJ For-Sale Unstable MTNR1B 15 49 COc1ccccc1/C=C/NC(=O)Nc1ccc2ccccc2c1 ZINC000217729531 DJ For-Sale Unstable PDGFRA 43 35 COc1ccccc1/C=C/NC(=O)Nc1ccc2ccccc2c1 ZINC000217729531 DJ For-Sale Unstable IMPDH2 0 44 COc1ccccc1/C=C/NC(=O)Nc1ccc2ccccc2c1 ZINC000217729531 DJ For-Sale Unstable IMDH_CRYPV 30 41 CC[C@@H](N)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217729541 BC For-Sale Unstable TPP2 50 40 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)Nc3cccc(O)c3)[C@@H]21 ZINC000217729558 JH In-Stock Unstable TSHR 50 33 COc1nccn(Cc2ccccc2)c1=O ZINC000217729578 BD For-Sale Unstable CYP11B1 30 43 COc1nccn(Cc2ccccc2)c1=O ZINC000217729578 BD For-Sale Unstable CYP11B2 32 43 O=C(c1cc2ccccc2[nH]1)N1CC(N2C(=O)[C@H]3CC=CC[C@H]3C2=O)C1 ZINC000217729587 ED In-Stock Unstable HRH4 24 52 O=C(c1cc2ccccc2[nH]1)N1CC(N2C(=O)[C@H]3CC=CC[C@H]3C2=O)C1 ZINC000217729587 ED In-Stock Unstable AKR1C3 19 48 CCOc1ccccc1OCC(=O)NC[C@H](O)C(=O)OC ZINC000217729591 CC On-Demand Unstable HCN1 40 32 CCOc1ccccc1OCC(=O)NC[C@H](O)C(=O)OC ZINC000217729591 CC On-Demand Unstable HCN4 40 32 CC[C@H](N)C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217729612 BC For-Sale Unstable TPP2 50 40 CC1(C)[C@H]2CC[C@@]1(C)[C@@H](NS(=O)(=O)c1ccccc1)C2 ZINC000217729658 CG On-Demand Unstable STS 23 40 O=C(COc1ccc(C(=O)O)cc1Cl)Nc1ccccc1Cl ZINC000217729679 EH In-Stock Unstable LTB4R 16 44 O=C(COc1ccc(C(=O)O)cc1Cl)Nc1ccccc1Cl ZINC000217729679 EH In-Stock Unstable EPHB3 42 33 O=C(c1cc2ccccc2[nH]1)N1CC(N2C(=O)[C@H]3CC=CC[C@@H]3C2=O)C1 ZINC000217729681 ED In-Stock Unstable HRH4 24 52 O=C(c1cc2ccccc2[nH]1)N1CC(N2C(=O)[C@H]3CC=CC[C@@H]3C2=O)C1 ZINC000217729681 ED In-Stock Unstable AKR1C3 19 48 CC[C@@H](N)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217729704 BC For-Sale Unstable TPP2 50 40 O=C(/C=C\c1ccc(Br)cc1)Nc1cnccc1C(=O)O ZINC000217729724 EG For-Sale Anodyne LTB4R 0 52 O=C(/C=C\c1ccc(Br)cc1)Nc1cnccc1C(=O)O ZINC000217729724 EG For-Sale Anodyne MMP2 0 43 O=C(/C=C\c1ccc(Br)cc1)Nc1cnccc1C(=O)O ZINC000217729724 EG For-Sale Anodyne HDAC1 22 43 O=C(/C=C\c1ccc(Br)cc1)Nc1cnccc1C(=O)O ZINC000217729724 EG For-Sale Anodyne MMP9 0 43 O=C(/C=C\c1ccc(Br)cc1)Nc1cnccc1C(=O)O ZINC000217729724 EG For-Sale Anodyne HPSE 34 41 O=C(/C=C\c1ccc(Br)cc1)Nc1cnccc1C(=O)O ZINC000217729724 EG For-Sale Anodyne MMP1 0 43 O=C(/C=C\c1ccc(Br)cc1)Nc1cnccc1C(=O)O ZINC000217729724 EG For-Sale Anodyne TRPM2 0 44 O=C(c1cc2ccccc2[nH]1)N1CC(N2C(=O)[C@@H]3CC=CC[C@H]3C2=O)C1 ZINC000217729758 ED In-Stock Unstable HRH4 24 52 O=C(c1cc2ccccc2[nH]1)N1CC(N2C(=O)[C@@H]3CC=CC[C@H]3C2=O)C1 ZINC000217729758 ED In-Stock Unstable AKR1C3 19 48 CCC[C@@H]1CCN(C(=O)c2ccc(OC)cc2F)C1 ZINC000217729773 CG For-Sale Unstable CHRM2 22 41 CCC[C@@H]1CCN(C(=O)c2ccc(OC)cc2F)C1 ZINC000217729773 CG For-Sale Unstable GRM3 15 51 CC[C@H](N)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217729781 BC For-Sale Unstable TPP2 50 40 C[C@H]1Cc2ccccc2N([C@H](C)C(=O)OC(C)(C)C)C1 ZINC000217729785 CG For-Sale Unstable TPP2 53 32 O=C(/C=C\c1ccc(O)cc1)Nc1cnccc1C(=O)O ZINC000217729801 CE For-Sale Anodyne F3 24 41 O=C(/C=C\c1ccc(O)cc1)Nc1cnccc1C(=O)O ZINC000217729801 CE For-Sale Anodyne MMP2 23 55 O=C(/C=C\c1ccc(O)cc1)Nc1cnccc1C(=O)O ZINC000217729801 CE For-Sale Anodyne MMP9 16 55 CCOC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)cc1 ZINC000217729833 GG In-Stock Unstable P2RY12 27 44 CCOC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)cc1 ZINC000217729833 GG In-Stock Unstable ADORA2B 16 42 CCOC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)cc1 ZINC000217729833 GG In-Stock Unstable CETP 0 40 CCOC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)cc1 ZINC000217729833 GG In-Stock Unstable ACR 63 34 CCOC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)cc1 ZINC000217729833 GG In-Stock Unstable MCHR1 15 44 CCOC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)cc1 ZINC000217729833 GG In-Stock Unstable MCHR2 40 43 CCC[C@H]1CCN(C(=O)c2ccc(OC)cc2F)C1 ZINC000217729864 CG For-Sale Unstable CHRM2 22 41 CCC[C@H]1CCN(C(=O)c2ccc(OC)cc2F)C1 ZINC000217729864 CG For-Sale Unstable GRM3 15 51 Cc1cccc(C(=O)Nc2cccc(/C=C\C(=O)O)n2)c1 ZINC000217729866 CF For-Sale Unstable GRM5 24 49 Cc1cccc(C(=O)Nc2cccc(/C=C\C(=O)O)n2)c1 ZINC000217729866 CF For-Sale Unstable KCNK3 106 50 Cc1cccc(C(=O)Nc2cccc(/C=C\C(=O)O)n2)c1 ZINC000217729866 CF For-Sale Unstable KCNK9 59 50 COc1ccccc1N1CCN(C(=O)c2cc(Cl)c[nH]c2=O)[C@@H](C)C1 ZINC000217729881 FE In-Stock Unstable HTR1A 53 40 COc1ccccc1N1CCN(C(=O)c2cc(Cl)c[nH]c2=O)[C@@H](C)C1 ZINC000217729881 FE In-Stock Unstable DRD2 43 39 COc1ccccc1N1CCN(C(=O)c2cc(Cl)c[nH]c2=O)[C@@H](C)C1 ZINC000217729881 FE In-Stock Unstable ADRA1D 46 40 COc1ccccc1N1CCN(C(=O)c2cc(Cl)c[nH]c2=O)[C@@H](C)C1 ZINC000217729881 FE In-Stock Unstable ADRA1A 38 40 COc1ccccc1N1CCN(C(=O)c2cc(Cl)c[nH]c2=O)[C@@H](C)C1 ZINC000217729881 FE In-Stock Unstable DRD3 44 37 COc1ccccc1N1CCN(C(=O)c2cc(Cl)c[nH]c2=O)[C@@H](C)C1 ZINC000217729881 FE In-Stock Unstable TACR3 26 61 O=C(/C=C\c1ccccc1Cl)Nc1cnccc1C(=O)O ZINC000217729883 DG For-Sale Anodyne BOTA 26 42 NC(=O)c1sc2ccncc2c1N ZINC000217729891 AC In-Stock Unstable EEF2K 58 39 CCCS(=O)(=O)N1CCC[C@@H]1C(=O)NC[C@@H](O)C(=O)OC ZINC000217729902 DA On-Demand Unstable TPP2 42 40 O=C1[C@@H]2[C@H](Cc3ccccc3)N[C@@H](c3ccc([N+](=O)[O-])cc3)[C@@H]2C(=O)N1c1ccccc1 ZINC000217729914 IH In-Stock Unstable H9B8T9_CAPHI 22 41 O=C1[C@@H]2[C@H](Cc3ccccc3)N[C@@H](c3ccc([N+](=O)[O-])cc3)[C@@H]2C(=O)N1c1ccccc1 ZINC000217729914 IH In-Stock Unstable A0A060INS8_CAPHI 0 41 Brc1ccc2c(ccn2-c2ccccc2OCc2ccccc2)c1 ZINC000217729929 GK For-Sale Unstable PTGER1 24 40 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)cc1 ZINC000217729941 GD In-Stock Unstable CA2 115 50 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)cc1 ZINC000217729941 GD In-Stock Unstable CA6 15 44 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)cc1 ZINC000217729941 GD In-Stock Unstable CA1 100 50 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)cc1 ZINC000217729941 GD In-Stock Unstable CA7 58 47 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)cc1 ZINC000217729941 GD In-Stock Unstable COLA 49 37 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)cc1 ZINC000217729941 GD In-Stock Unstable CPT1A 51 37 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)cc1 ZINC000217729941 GD In-Stock Unstable CA5B 62 47 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)cc1 ZINC000217729941 GD In-Stock Unstable CA4 106 50 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)cc1 ZINC000217729941 GD In-Stock Unstable CA5A 71 47 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)cc1 ZINC000217729941 GD In-Stock Unstable CA14 45 41 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)cc1 ZINC000217729941 GD In-Stock Unstable CA12 63 44 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)cc1 ZINC000217729941 GD In-Stock Unstable CA9 72 43 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)cc1 ZINC000217729941 GD In-Stock Unstable UREA_CANEN 27 42 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)cc1 ZINC000217729941 GD In-Stock Unstable CYNT 41 43 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)cc1 ZINC000217729941 GD In-Stock Unstable NCE103 33 44 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)cc1 ZINC000217729941 GD In-Stock Unstable PFK 0 45 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)cc1 ZINC000217729941 GD In-Stock Unstable MTCA1 40 40 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)cc1 ZINC000217729941 GD In-Stock Unstable P96878_MYCTU 56 44 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)cc1 ZINC000217729941 GD In-Stock Unstable CA 0 44 CCC(CC)C(=O)Nc1cc(/C=C\C(=O)O)ccc1OC ZINC000217729964 CG For-Sale Unstable TUBB1 47 38 CCC(CC)C(=O)Nc1cc(/C=C\C(=O)O)ccc1OC ZINC000217729964 CG For-Sale Unstable AKR1C3 31 42 COc1ccccc1N1CCN(C(=O)c2cc(Cl)c[nH]c2=O)[C@H](C)C1 ZINC000217729967 FE In-Stock Unstable HTR1A 53 40 COc1ccccc1N1CCN(C(=O)c2cc(Cl)c[nH]c2=O)[C@H](C)C1 ZINC000217729967 FE In-Stock Unstable DRD2 43 39 COc1ccccc1N1CCN(C(=O)c2cc(Cl)c[nH]c2=O)[C@H](C)C1 ZINC000217729967 FE In-Stock Unstable ADRA1D 46 40 COc1ccccc1N1CCN(C(=O)c2cc(Cl)c[nH]c2=O)[C@H](C)C1 ZINC000217729967 FE In-Stock Unstable ADRA1A 38 40 COc1ccccc1N1CCN(C(=O)c2cc(Cl)c[nH]c2=O)[C@H](C)C1 ZINC000217729967 FE In-Stock Unstable DRD3 44 37 COc1ccccc1N1CCN(C(=O)c2cc(Cl)c[nH]c2=O)[C@H](C)C1 ZINC000217729967 FE In-Stock Unstable TACR3 26 61 CCCS(=O)(=O)N1CCC[C@H]1C(=O)NC[C@@H](O)C(=O)OC ZINC000217729974 DA On-Demand Unstable TPP2 42 40 CCCN(CCC)C(=O)N/C=C/c1ccccc1OC ZINC000217729991 CG For-Sale Unstable TLR4 15 44 CC(=O)c1cccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)c1 ZINC000217730054 EG In-Stock Unstable CETP 0 41 CC(=O)c1cccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)c1 ZINC000217730054 EG In-Stock Unstable CPT1A 43 30 CC(=O)c1cccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)c1 ZINC000217730054 EG In-Stock Unstable NR1H4 40 40 CC(=O)c1cccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)c1 ZINC000217730054 EG In-Stock Unstable MCHR2 40 44 CC(=O)c1cccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)c1 ZINC000217730054 EG In-Stock Unstable HIF1A 17 48 CC(=O)c1cccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)c1 ZINC000217730054 EG In-Stock Unstable AKR1C3 52 52 CC(=O)c1cccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)c1 ZINC000217730054 EG In-Stock Unstable KCNK3 71 37 CC(=O)c1cccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)c1 ZINC000217730054 EG In-Stock Unstable KCNK9 57 33 CC(=O)c1cccc(NC(=O)COc2ccc(C(=O)O)cc2Cl)c1 ZINC000217730054 EG In-Stock Unstable PARP10 0 42 COc1ccc(/C=C\C(=O)O)cc1NC(=O)CC(C)(C)C ZINC000217730058 CG For-Sale Unstable MMP2 0 45 COc1ccc(/C=C\C(=O)O)cc1NC(=O)CC(C)(C)C ZINC000217730058 CG For-Sale Unstable TUBB1 47 38 CSc1ncccc1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217730059 EF For-Sale Unstable HCRTR1 28 40 CSc1ncccc1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217730059 EF For-Sale Unstable HCRTR2 25 40 CSc1ncccc1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217730130 EF For-Sale Unstable HCRTR1 28 40 CSc1ncccc1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217730130 EF For-Sale Unstable HCRTR2 25 40 COc1ccc(/C=C\C(=O)O)cc1NC(=O)CNC(C)=O ZINC000217730146 CC For-Sale Unstable TUBB1 44 38 O=C(c1ccc2cc[nH]c2c1)N1CC(N2C(=O)[C@H]3CC=CC[C@H]3C2=O)C1 ZINC000217730171 ED In-Stock Unstable GHSR 0 49 O=C(/C=C\c1ccccc1F)Nc1cc(C(=O)O)ccn1 ZINC000217730182 CF For-Sale Anodyne KCNQ2 43 40 O=C(/C=C\c1ccccc1F)Nc1cc(C(=O)O)ccn1 ZINC000217730182 CF For-Sale Anodyne MMP1 0 45 O=C(/C=C\c1ccccc1F)Nc1cc(C(=O)O)ccn1 ZINC000217730182 CF For-Sale Anodyne KDM4E 33 40 COC(=O)c1ccccc1NC(=O)COc1ccc(C(=O)O)cc1OC ZINC000217730204 FE In-Stock Unstable LTB4R 22 51 COC(=O)c1ccccc1NC(=O)COc1ccc(C(=O)O)cc1OC ZINC000217730204 FE In-Stock Unstable CPT1A 43 30 COC(=O)c1ccccc1NC(=O)COc1ccc(C(=O)O)cc1OC ZINC000217730204 FE In-Stock Unstable PLA2G4B 35 45 COC(=O)c1ccccc1NC(=O)COc1ccc(C(=O)O)cc1OC ZINC000217730204 FE In-Stock Unstable NR1H4 0 52 COC(=O)c1ccccc1NC(=O)COc1ccc(C(=O)O)cc1OC ZINC000217730204 FE In-Stock Unstable TTR 0 40 COC(=O)c1ccccc1NC(=O)COc1ccc(C(=O)O)cc1OC ZINC000217730204 FE In-Stock Unstable HCAR2 29 41 COC(=O)c1ccccc1NC(=O)COc1ccc(C(=O)O)cc1OC ZINC000217730204 FE In-Stock Unstable ABCG2 42 40 COC(=O)c1ccccc1NC(=O)COc1ccc(C(=O)O)cc1OC ZINC000217730204 FE In-Stock Unstable AKR1C2 43 37 COC(=O)c1ccccc1NC(=O)COc1ccc(C(=O)O)cc1OC ZINC000217730204 FE In-Stock Unstable KCNK3 42 36 COC(=O)c1ccccc1NC(=O)COc1ccc(C(=O)O)cc1OC ZINC000217730204 FE In-Stock Unstable FAS 51 50 COc1ccccc1/C=C/NC(=O)NCCCNC=O ZINC000217730221 CD For-Sale Unstable DRD2 16 45 COc1ccccc1/C=C/NC(=O)NCCCNC=O ZINC000217730221 CD For-Sale Unstable DRD3 32 45 COc1ccccc1/C=C/NC(=O)NCCCNC=O ZINC000217730221 CD For-Sale Unstable ACAT 0 43 COc1ccc(C(=O)Nc2ncc(/C=C\C(=O)O)s2)cc1 ZINC000217730228 DF For-Sale Unstable ADORA2B 17 40 COc1ccc(C(=O)Nc2ncc(/C=C\C(=O)O)s2)cc1 ZINC000217730228 DF For-Sale Unstable CSNK1D 18 40 COc1ccc(C(=O)Nc2ncc(/C=C\C(=O)O)s2)cc1 ZINC000217730228 DF For-Sale Unstable CSNK2A2 15 60 COc1ccc(C(=O)Nc2ncc(/C=C\C(=O)O)s2)cc1 ZINC000217730228 DF For-Sale Unstable LUCI_LUCLA 23 44 COc1ccc(C(=O)Nc2ncc(/C=C\C(=O)O)s2)cc1 ZINC000217730228 DF For-Sale Unstable SCD1 27 44 COc1ccc(C(=O)Nc2ncc(/C=C\C(=O)O)s2)cc1 ZINC000217730228 DF For-Sale Unstable SCD 32 44 O=C(c1ccc2cc[nH]c2c1)N1CC(N2C(=O)[C@H]3CC=CC[C@@H]3C2=O)C1 ZINC000217730237 ED In-Stock Unstable GHSR 0 49 CC(C)[C@@H](CO)NC(=O)[C@@H]1CC(=O)N(Cc2ccc3c(c2)OCO3)C1 ZINC000217730259 EC In-Stock Unstable NOS2 53 34 CC(C)[C@@H](CO)NC(=O)[C@@H]1CC(=O)N(Cc2ccc3c(c2)OCO3)C1 ZINC000217730259 EC In-Stock Unstable SSTR3 63 32 CCCC[C@@H](CC)C(=O)NC[C@@H](O)C(=O)OC ZINC000217730273 BC On-Demand Unstable SLC22A20 0 44 CCCC[C@@H](CC)C(=O)NC[C@@H](O)C(=O)OC ZINC000217730273 BC On-Demand Unstable CQSS 42 32 Brc1ccccc1CN[C@@H]1CCN2CCC[C@@H]12 ZINC000217730299 CF For-Sale Unstable SLC18A3 32 40 O=C(c1ccc2cc[nH]c2c1)N1CC(N2C(=O)[C@@H]3CC=CC[C@H]3C2=O)C1 ZINC000217730301 ED In-Stock Unstable GHSR 0 49 COC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2OC)cc1 ZINC000217730312 FE In-Stock Unstable CYSLTR1 0 40 COC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2OC)cc1 ZINC000217730312 FE In-Stock Unstable CETP 0 42 COC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2OC)cc1 ZINC000217730312 FE In-Stock Unstable COLA 64 40 COC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2OC)cc1 ZINC000217730312 FE In-Stock Unstable CPT1A 56 40 COC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2OC)cc1 ZINC000217730312 FE In-Stock Unstable CPT2 44 37 COC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2OC)cc1 ZINC000217730312 FE In-Stock Unstable PLA2G4B 32 48 COC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2OC)cc1 ZINC000217730312 FE In-Stock Unstable ACR 58 42 COC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2OC)cc1 ZINC000217730312 FE In-Stock Unstable CPT1B 47 37 COC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2OC)cc1 ZINC000217730312 FE In-Stock Unstable PDGFRA 55 36 COC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2OC)cc1 ZINC000217730312 FE In-Stock Unstable ENPP1 62 37 COC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2OC)cc1 ZINC000217730312 FE In-Stock Unstable KDM4C 0 46 COC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2OC)cc1 ZINC000217730312 FE In-Stock Unstable DRTS_TRYCR 38 40 COC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2OC)cc1 ZINC000217730312 FE In-Stock Unstable KDM3A 0 46 COC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2OC)cc1 ZINC000217730312 FE In-Stock Unstable GLMU 0 40 COC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2OC)cc1 ZINC000217730312 FE In-Stock Unstable KDM5C 0 46 Brc1ccc(N2C[C@@H]3C[C@H](C2)N3)cc1 ZINC000217730337 CD For-Sale Unstable CHRNA4 31 61 CC(C)[C@@H](CO)NC(=O)[C@H]1CC(=O)N(Cc2ccc3c(c2)OCO3)C1 ZINC000217730347 EC In-Stock Unstable NOS2 53 34 CC(C)[C@@H](CO)NC(=O)[C@H]1CC(=O)N(Cc2ccc3c(c2)OCO3)C1 ZINC000217730347 EC In-Stock Unstable SSTR3 63 32 CCCC[C@H](CC)C(=O)NC[C@@H](O)C(=O)OC ZINC000217730350 BC On-Demand Unstable SLC22A20 0 44 CCCC[C@H](CC)C(=O)NC[C@@H](O)C(=O)OC ZINC000217730350 BC On-Demand Unstable CQSS 42 32 O=C(/C=C\c1cccc(F)c1)Nc1cc(C(=O)O)ccn1 ZINC000217730354 CF For-Sale Anodyne HDAC8 38 43 O=C(/C=C\c1cccc(F)c1)Nc1cc(C(=O)O)ccn1 ZINC000217730354 CF For-Sale Anodyne MMP2 0 54 O=C(/C=C\c1cccc(F)c1)Nc1cc(C(=O)O)ccn1 ZINC000217730354 CF For-Sale Anodyne HDAC6 20 43 O=C(/C=C\c1cccc(F)c1)Nc1cc(C(=O)O)ccn1 ZINC000217730354 CF For-Sale Anodyne MMP9 0 51 O=C(/C=C\c1cccc(F)c1)Nc1cc(C(=O)O)ccn1 ZINC000217730354 CF For-Sale Anodyne MMP1 24 54 Brc1ccccc1CN[C@H]1CCN2CCC[C@@H]12 ZINC000217730385 CF For-Sale Unstable SLC18A3 32 40 CC1(C)[C@H]2CC[C@@]1(C)[C@@H](NS(=O)(=O)c1cccc(Br)c1)C2 ZINC000217730387 FH For-Sale Unstable STS 26 46 O=C(O)/C=C\c1cnc(NC(=O)c2cc(Cl)ccc2F)s1 ZINC000217730388 EG For-Sale Anodyne HSD17B1 0 40 CCCC[C@@H](CC)C(=O)NC[C@H](O)C(=O)OC ZINC000217730434 BC On-Demand Unstable SLC22A20 0 44 CCCC[C@@H](CC)C(=O)NC[C@H](O)C(=O)OC ZINC000217730434 BC On-Demand Unstable CQSS 42 32 O=C(/C=C\c1ccccc1Cl)Nc1cc(C(=O)O)ccn1 ZINC000217730438 DG For-Sale Anodyne PTGER2 0 40 O=C(/C=C\c1ccccc1Cl)Nc1cc(C(=O)O)ccn1 ZINC000217730438 DG For-Sale Anodyne TYK2 62 36 O=C(/C=C\c1ccccc1Cl)Nc1cc(C(=O)O)ccn1 ZINC000217730438 DG For-Sale Anodyne MMP1 0 45 CCOC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2OC)cc1 ZINC000217730448 FF In-Stock Unstable CETP 0 41 CCOC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2OC)cc1 ZINC000217730448 FF In-Stock Unstable CPT1A 43 30 COc1ccccc1/C=C/NC(=O)N1C[C@@]2(C)C[C@H]1CC(C)(C)C2 ZINC000217730524 EI For-Sale Unstable AVPR2 18 49 COc1ccccc1/C=C/NC(=O)N1C[C@@]2(C)C[C@H]1CC(C)(C)C2 ZINC000217730524 EI For-Sale Unstable AVPR1A 39 47 Cn1cc(/C=C\C(=O)Nc2cc(C(=O)O)ccn2)cn1 ZINC000217730525 CD For-Sale Unstable HDAC8 41 34 CCCC[C@H](CC)C(=O)NC[C@H](O)C(=O)OC ZINC000217730531 BC On-Demand Unstable SLC22A20 0 44 CCCC[C@H](CC)C(=O)NC[C@H](O)C(=O)OC ZINC000217730531 BC On-Demand Unstable CQSS 42 32 COc1cc(C(=O)O)ccc1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217730547 GD In-Stock Unstable CA2 145 51 COc1cc(C(=O)O)ccc1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217730547 GD In-Stock Unstable GRM3 15 40 COc1cc(C(=O)O)ccc1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217730547 GD In-Stock Unstable CA6 17 44 COc1cc(C(=O)O)ccc1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217730547 GD In-Stock Unstable CA1 130 51 COc1cc(C(=O)O)ccc1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217730547 GD In-Stock Unstable CA7 69 50 COc1cc(C(=O)O)ccc1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217730547 GD In-Stock Unstable LTB4R 15 40 COc1cc(C(=O)O)ccc1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217730547 GD In-Stock Unstable COLA 71 41 COc1cc(C(=O)O)ccc1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217730547 GD In-Stock Unstable CPT1A 72 41 COc1cc(C(=O)O)ccc1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217730547 GD In-Stock Unstable CPT2 48 38 COc1cc(C(=O)O)ccc1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217730547 GD In-Stock Unstable CA13 22 40 COc1cc(C(=O)O)ccc1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217730547 GD In-Stock Unstable CA5B 60 47 COc1cc(C(=O)O)ccc1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217730547 GD In-Stock Unstable CA4 121 50 COc1cc(C(=O)O)ccc1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217730547 GD In-Stock Unstable CA5A 69 47 COc1cc(C(=O)O)ccc1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217730547 GD In-Stock Unstable CA14 53 50 COc1cc(C(=O)O)ccc1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217730547 GD In-Stock Unstable PLA2G4B 26 44 COc1cc(C(=O)O)ccc1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217730547 GD In-Stock Unstable CA12 79 51 COc1cc(C(=O)O)ccc1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217730547 GD In-Stock Unstable CPT1B 51 38 COc1cc(C(=O)O)ccc1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217730547 GD In-Stock Unstable CA9 85 51 COc1cc(C(=O)O)ccc1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217730547 GD In-Stock Unstable UREA_CANEN 29 43 COc1cc(C(=O)O)ccc1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217730547 GD In-Stock Unstable CYNT 44 46 COc1cc(C(=O)O)ccc1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217730547 GD In-Stock Unstable NCE103 32 44 COc1cc(C(=O)O)ccc1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217730547 GD In-Stock Unstable ENPP1 72 34 COc1cc(C(=O)O)ccc1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217730547 GD In-Stock Unstable MTCA1 52 47 COc1cc(C(=O)O)ccc1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217730547 GD In-Stock Unstable P96878_MYCTU 69 47 COc1cc(C(=O)O)ccc1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217730547 GD In-Stock Unstable CA 0 44 COc1cn(CC(=O)NCCc2c[nH]c3ccc(Cl)cc23)c(C)cc1=O ZINC000217730552 FF In-Stock Unstable HTR1D 20 40 COc1cn(CC(=O)NCCc2c[nH]c3ccc(Cl)cc23)c(C)cc1=O ZINC000217730552 FF In-Stock Unstable HTR1B 29 40 COc1cn(CC(=O)NCCc2c[nH]c3ccc(Cl)cc23)c(C)cc1=O ZINC000217730552 FF In-Stock Unstable NQO2 19 43 COc1cn(CC(=O)NCCc2c[nH]c3ccc(Cl)cc23)c(C)cc1=O ZINC000217730552 FF In-Stock Unstable MTNR1A 19 50 COc1cn(CC(=O)NCCc2c[nH]c3ccc(Cl)cc23)c(C)cc1=O ZINC000217730552 FF In-Stock Unstable MAPT 19 42 Brc1cccc(N2C[C@@H]3C[C@H](C2)N3)c1 ZINC000217730633 CD For-Sale Unstable CHRNA4 25 51 O=C(Cc1ccccc1Cl)NC[C@@H]1CCCN1c1nccs1 ZINC000217730653 EG For-Sale Unstable TK 18 42 COC(=O)[C@@H](O)CNC(=O)CCSc1ccccc1 ZINC000217730660 CC On-Demand Unstable FAS 45 47 COc1ccccc1/C=C/NC(=O)Nc1cccc(N(C)C)c1 ZINC000217730725 DH For-Sale Unstable KCNK3 59 42 COc1ccccc1/C=C/NC(=O)Nc1cccc(N(C)C)c1 ZINC000217730725 DH For-Sale Unstable KCNK9 57 42 O=C(Cc1ccccc1Cl)NC[C@H]1CCCN1c1nccs1 ZINC000217730736 EG For-Sale Unstable TK 18 42 COC(=O)[C@H](O)CNC(=O)CCSc1ccccc1 ZINC000217730739 CC On-Demand Unstable FAS 45 47 COc1ccccc1/C=C/NC(=O)Nc1nc2c(s1)CN(C)CC2 ZINC000217730823 EF For-Sale Unstable F10 23 44 O=C(NC[C@@H]1CCCN1c1nccs1)c1cnc2ccccc2n1 ZINC000217730856 EE For-Sale Unstable CCR1 40 38 COc1cc(C(=O)O)cc(OC)c1OCC(=O)NC1CCCCC1 ZINC000217730861 EE In-Stock Unstable CYSLTR1 22 44 COc1cc(C(=O)O)cc(OC)c1OCC(=O)NC1CCCCC1 ZINC000217730861 EE In-Stock Unstable EPHX2 32 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)NC1CCCCC1 ZINC000217730861 EE In-Stock Unstable LUXN 0 48 Brc1ccccc1N1C[C@@H]2C[C@H](C1)N2 ZINC000217730890 CD For-Sale Unstable CHRNA4 17 45 CC[C@@H](C)N(CC(=O)Nc1cccc(C)c1C)C(=O)c1ccccc1Cl ZINC000217730912 FJ On-Demand Unstable CXCL8 43 40 CC[C@@H](C)N(CC(=O)Nc1cccc(C)c1C)C(=O)c1ccccc1Cl ZINC000217730912 FJ On-Demand Unstable ECR 49 44 O=C(NC[C@H]1CCCN1c1nccs1)c1cnc2ccccc2n1 ZINC000217730943 EE For-Sale Unstable CCR1 40 38 COc1ccccc1/C=C/NC(=O)Nc1ccc2nc[nH]c2c1 ZINC000217730952 DG For-Sale Unstable PDGFRA 43 35 COc1ccccc1/C=C/NC(=O)Nc1ccc2nc[nH]c2c1 ZINC000217730952 DG For-Sale Unstable IMPDH2 0 42 COc1cc(C(=O)O)cc(OC)c1OCC(=O)NCc1ccccc1 ZINC000217730969 EE In-Stock Unstable DRD2 15 45 COc1cc(C(=O)O)cc(OC)c1OCC(=O)NCc1ccccc1 ZINC000217730969 EE In-Stock Unstable ADORA2B 0 41 COc1cc(C(=O)O)cc(OC)c1OCC(=O)NCc1ccccc1 ZINC000217730969 EE In-Stock Unstable TRPV1 26 45 COc1cc(C(=O)O)cc(OC)c1OCC(=O)NCc1ccccc1 ZINC000217730969 EE In-Stock Unstable SIGMAR1 15 42 COc1cc(C(=O)O)cc(OC)c1OCC(=O)NCc1ccccc1 ZINC000217730969 EE In-Stock Unstable MMP13 15 45 COc1cc(C(=O)O)cc(OC)c1OCC(=O)NCc1ccccc1 ZINC000217730969 EE In-Stock Unstable LTB4R 25 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)NCc1ccccc1 ZINC000217730969 EE In-Stock Unstable HCRTR2 22 41 COc1cc(C(=O)O)cc(OC)c1OCC(=O)NCc1ccccc1 ZINC000217730969 EE In-Stock Unstable AMP1_PLAFQ 44 35 COc1cc(C(=O)O)cc(OC)c1OCC(=O)NCc1ccccc1 ZINC000217730969 EE In-Stock Unstable NCE103 16 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)NCc1ccccc1 ZINC000217730969 EE In-Stock Unstable P96878_MYCTU 16 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)NCc1ccccc1 ZINC000217730969 EE In-Stock Unstable KDM4E 21 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)NCc1ccccc1 ZINC000217730969 EE In-Stock Unstable CAN2 0 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)NCc1ccccc1 ZINC000217730969 EE In-Stock Unstable PDS 58 39 CC[C@H](C)N(CC(=O)Nc1cccc(C)c1C)C(=O)c1ccccc1Cl ZINC000217731000 FJ On-Demand Unstable CXCL8 43 40 CC[C@H](C)N(CC(=O)Nc1cccc(C)c1C)C(=O)c1ccccc1Cl ZINC000217731000 FJ On-Demand Unstable ECR 49 44 Nc1cncc(CN2CCc3ccccc3C2)c1 ZINC000217731022 BE In-Stock Unstable CHRNA6 0 44 Nc1cncc(CN2CCc3ccccc3C2)c1 ZINC000217731022 BE In-Stock Unstable NOD1 30 40 Nc1cncc(CN2CCc3ccccc3C2)c1 ZINC000217731022 BE In-Stock Unstable NOD2 45 38 COc1ccccc1CN1C(=O)N[C@@H](CCC(=O)NC[C@@H]2CCCN3CCCC[C@H]23)C1=O ZINC000217731063 IE In-Stock Unstable MBTPS1 52 37 COc1cc(C(=O)O)cc(OC)c1OCC(=O)NCCc1ccccc1 ZINC000217731087 FE In-Stock Unstable CNR2 27 43 COc1cc(C(=O)O)cc(OC)c1OCC(=O)NCCc1ccccc1 ZINC000217731087 FE In-Stock Unstable MTNR1A 44 39 COc1cc(C(=O)O)cc(OC)c1OCC(=O)NCCc1ccccc1 ZINC000217731087 FE In-Stock Unstable MTNR1B 59 45 COc1cc(C(=O)O)cc(OC)c1OCC(=O)NCCc1ccccc1 ZINC000217731087 FE In-Stock Unstable AKR1C3 24 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)NCCc1ccccc1 ZINC000217731087 FE In-Stock Unstable NCE103 29 42 COc1cc(C(=O)O)cc(OC)c1OCC(=O)NCCc1ccccc1 ZINC000217731087 FE In-Stock Unstable CRTM 40 36 COc1cc(C(=O)O)cc(OC)c1OCC(=O)NCCc1ccccc1 ZINC000217731087 FE In-Stock Unstable KDM4E 24 50 COc1cc(C(=O)O)cc(OC)c1OCC(=O)NCCc1ccccc1 ZINC000217731087 FE In-Stock Unstable CAN2 0 42 COc1ccc2c(CC(=O)NCCCC[C@H](N)C(=O)O)cc(=O)oc2c1 ZINC000217731147 FD For-Sale Unstable CYP19A1 16 42 COc1ccc2c(CC(=O)NCCCC[C@H](N)C(=O)O)cc(=O)oc2c1 ZINC000217731147 FD For-Sale Unstable MAOA 39 40 COc1ccc2c(CC(=O)NCCCC[C@H](N)C(=O)O)cc(=O)oc2c1 ZINC000217731147 FD For-Sale Unstable MAOB 30 48 COc1ccc2c(CC(=O)NCCCC[C@H](N)C(=O)O)cc(=O)oc2c1 ZINC000217731147 FD For-Sale Unstable MTNR1A 55 41 COc1ccc2c(CC(=O)NCCCC[C@H](N)C(=O)O)cc(=O)oc2c1 ZINC000217731147 FD For-Sale Unstable GRIA1 48 33 COc1ccc2c(CC(=O)NCCCC[C@H](N)C(=O)O)cc(=O)oc2c1 ZINC000217731147 FD For-Sale Unstable NOD1 54 39 C[C@@H](C(=O)OC(C)(C)C)N1CC[C@@H](N2CCCCC2)C1 ZINC000217731218 CE On-Demand Unstable L3MBTL3 55 37 O=C1CC2(CCN(C(=O)c3cc(Cl)ccc3Br)CC2)CN1 ZINC000217731225 FF On-Demand Unstable AVPR1A 19 40 COc1ccc2c(CC(=O)NCCCC[C@@H](N)C(=O)O)cc(=O)oc2c1 ZINC000217731227 FD For-Sale Unstable CYP19A1 16 42 COc1ccc2c(CC(=O)NCCCC[C@@H](N)C(=O)O)cc(=O)oc2c1 ZINC000217731227 FD For-Sale Unstable MAOA 39 40 COc1ccc2c(CC(=O)NCCCC[C@@H](N)C(=O)O)cc(=O)oc2c1 ZINC000217731227 FD For-Sale Unstable MAOB 34 48 COc1ccc2c(CC(=O)NCCCC[C@@H](N)C(=O)O)cc(=O)oc2c1 ZINC000217731227 FD For-Sale Unstable MTNR1A 66 41 COc1ccc2c(CC(=O)NCCCC[C@@H](N)C(=O)O)cc(=O)oc2c1 ZINC000217731227 FD For-Sale Unstable MTNR1B 52 39 COc1ccc2c(CC(=O)NCCCC[C@@H](N)C(=O)O)cc(=O)oc2c1 ZINC000217731227 FD For-Sale Unstable GRIA1 48 33 COc1ccc2c(CC(=O)NCCCC[C@@H](N)C(=O)O)cc(=O)oc2c1 ZINC000217731227 FD For-Sale Unstable NOD1 54 39 O=C(O)/C=C\c1ccc(NC(=O)Cc2ccsc2)c(F)c1 ZINC000217731267 DG For-Sale Unstable CA5B 17 40 O=C(O)/C=C\c1ccc(NC(=O)Cc2ccsc2)c(F)c1 ZINC000217731267 DG For-Sale Unstable CA5A 19 40 Cn1cc(/C=C\C(=O)Nc2cnccc2C(=O)O)cn1 ZINC000217731278 CD For-Sale Unstable LTB4R 18 43 C[C@H](C(=O)OC(C)(C)C)N1CC[C@@H](N2CCCCC2)C1 ZINC000217731288 CE On-Demand Unstable L3MBTL3 55 37 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccccc1 ZINC000217731304 EE In-Stock Unstable CETP 0 44 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccccc1 ZINC000217731304 EE In-Stock Unstable LTB4R 21 43 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccccc1 ZINC000217731304 EE In-Stock Unstable CPT1A 52 36 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccccc1 ZINC000217731304 EE In-Stock Unstable GUAB 0 44 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccccc1 ZINC000217731304 EE In-Stock Unstable KDR 21 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccccc1 ZINC000217731304 EE In-Stock Unstable MTNR1A 18 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccccc1 ZINC000217731304 EE In-Stock Unstable MTNR1B 25 44 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccccc1 ZINC000217731304 EE In-Stock Unstable ABCB1 0 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccccc1 ZINC000217731304 EE In-Stock Unstable PDGFRA 43 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccccc1 ZINC000217731304 EE In-Stock Unstable HIF1A 16 41 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccccc1 ZINC000217731304 EE In-Stock Unstable ENPP1 49 30 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccccc1 ZINC000217731304 EE In-Stock Unstable SMO 23 45 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccccc1 ZINC000217731304 EE In-Stock Unstable GLMU 0 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccccc1 ZINC000217731304 EE In-Stock Unstable KCNK3 57 42 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccccc1 ZINC000217731304 EE In-Stock Unstable KCNK9 58 40 c1ccc2c(c1)CCC[C@H]2N[C@@H]1CCN2CCC[C@@H]12 ZINC000217731310 CF For-Sale Unstable SLC18A3 45 34 c1ccc2c(c1)CCC[C@H]2N[C@@H]1CCN2CCC[C@@H]12 ZINC000217731310 CF For-Sale Unstable KCNN3 18 40 Cc1ccc(C(=O)Nc2ccc(/C=C\C(=O)O)cc2F)o1 ZINC000217731338 CG For-Sale Unstable HPSE 41 41 O=C1CC2(CCN(C(=O)c3cc(Cl)ccc3I)CC2)CN1 ZINC000217731344 HF On-Demand Unstable AVPR1A 0 40 Cc1ccnc(Cl)c1C(=O)NC1CC1 ZINC000217731355 BD In-Stock Unstable MAPK13 53 34 Cc1ccnc(Cl)c1C(=O)NC1CC1 ZINC000217731355 BD In-Stock Unstable TYK2 41 33 COc1ccc(OC)c([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c1 ZINC000217731369 JI In-Stock Unstable AKR1B1 0 48 COc1ccc(OC)c([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c1 ZINC000217731369 JI In-Stock Unstable CYP1B1 57 42 COc1ccc(OC)c([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c1 ZINC000217731369 JI In-Stock Unstable CYP1A1 43 48 COc1ccc(OC)c([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c1 ZINC000217731369 JI In-Stock Unstable CYP1A2 33 42 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(C)c1 ZINC000217731401 EF In-Stock Unstable CCKAR 22 42 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(C)c1 ZINC000217731401 EF In-Stock Unstable CETP 0 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(C)c1 ZINC000217731401 EF In-Stock Unstable CPT1A 43 30 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(C)c1 ZINC000217731401 EF In-Stock Unstable KDR 26 43 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(C)c1 ZINC000217731401 EF In-Stock Unstable PDGFRA 19 43 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(C)c1 ZINC000217731401 EF In-Stock Unstable HIF1A 16 42 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(C)c1 ZINC000217731401 EF In-Stock Unstable AKR1C3 39 42 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(C)c1 ZINC000217731401 EF In-Stock Unstable AKR1C2 22 42 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(C)c1 ZINC000217731401 EF In-Stock Unstable ENPP1 49 30 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(C)c1 ZINC000217731401 EF In-Stock Unstable SMO 21 44 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(C)c1 ZINC000217731401 EF In-Stock Unstable KCNK3 85 43 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(C)c1 ZINC000217731401 EF In-Stock Unstable KCNK9 85 45 c1ccc2c(c1)CCC[C@H]2N[C@H]1CCN2CCC[C@@H]12 ZINC000217731402 CF For-Sale Unstable SLC18A3 45 34 c1ccc2c(c1)CCC[C@H]2N[C@H]1CCN2CCC[C@@H]12 ZINC000217731402 CF For-Sale Unstable KCNN3 18 40 Cc1cc(NC(=O)c2snnc2C)ccc1/C=C\C(=O)O ZINC000217731418 DF For-Sale Unstable PRMT3 60 35 COc1ccccc1/C=C/NC(=O)Nc1cccc(Br)c1 ZINC000217731419 EI For-Sale Unstable IMPDH2 0 44 COc1ccccc1/C=C/NC(=O)Nc1cccc(Br)c1 ZINC000217731419 EI For-Sale Unstable KCNK3 66 44 COc1ccccc1/C=C/NC(=O)Nc1cccc(Br)c1 ZINC000217731419 EI For-Sale Unstable KCNK9 63 44 COC(=O)[C@@H](O)CNC(=O)CSc1ccc([N+](=O)[O-])cc1 ZINC000217731438 DC On-Demand Unstable FAS 45 48 COc1ccc(OC)c([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c1 ZINC000217731458 JI In-Stock Unstable AKR1B1 0 48 COc1ccc(OC)c([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c1 ZINC000217731458 JI In-Stock Unstable CYP1B1 57 42 COc1ccc(OC)c([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c1 ZINC000217731458 JI In-Stock Unstable CYP1A1 43 48 COc1ccc(OC)c([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c1 ZINC000217731458 JI In-Stock Unstable CYP1A2 33 42 O=C(NC[C@@H]1CCCN1c1nccs1)c1nc2ccccc2s1 ZINC000217731459 EG For-Sale Unstable TRY1_BOVIN 42 37 Cc1ccnc(Cl)c1C(=O)N1CCCC1 ZINC000217731465 BE In-Stock Unstable CCR5 33 40 Cc1ccnc(Cl)c1C(=O)N1CCCC1 ZINC000217731465 BE In-Stock Unstable REN 0 43 Cc1ccnc(Cl)c1C(=O)N1CCCC1 ZINC000217731465 BE In-Stock Unstable L3MBTL3 41 34 CON(C)C(=O)/C(C)=C/c1ccc(F)cc1 ZINC000217731482 BE On-Demand Unstable TLR4 20 50 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(C)cc1 ZINC000217731510 EF In-Stock Unstable CETP 0 47 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(C)cc1 ZINC000217731510 EF In-Stock Unstable LTB4R 19 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(C)cc1 ZINC000217731510 EF In-Stock Unstable CPT1A 43 30 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(C)cc1 ZINC000217731510 EF In-Stock Unstable KDR 20 41 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(C)cc1 ZINC000217731510 EF In-Stock Unstable PDGFRA 45 34 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(C)cc1 ZINC000217731510 EF In-Stock Unstable AKR1C3 19 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(C)cc1 ZINC000217731510 EF In-Stock Unstable ENPP1 56 33 COC(=O)[C@H](O)CNC(=O)CSc1ccc([N+](=O)[O-])cc1 ZINC000217731515 DC On-Demand Unstable FAS 45 48 CCN1CCN(C(=O)N/C=C/c2ccccc2OC)CC1 ZINC000217731520 CE For-Sale Unstable HTR1A 38 45 CCN1CCN(C(=O)N/C=C/c2ccccc2OC)CC1 ZINC000217731520 CE For-Sale Unstable DRD2 35 44 CCN1CCN(C(=O)N/C=C/c2ccccc2OC)CC1 ZINC000217731520 CE For-Sale Unstable DRD3 45 44 O=C(c1cccc(Cl)c1)N1CC(N2C(=O)[C@H]3CC=CC[C@H]3C2=O)C1 ZINC000217731551 EE In-Stock Unstable SLC6A7 0 42 O=C(NC[C@H]1CCCN1c1nccs1)c1nc2ccccc2s1 ZINC000217731558 EG For-Sale Unstable TRY1_BOVIN 42 37 COc1ccc([C@H](N)C(=O)O)c(OC)c1Cl ZINC000217731579 BD For-Sale Unstable CACNA2D1 19 40 Cc1cc(NC(=O)c2ccc(Cl)o2)ccc1/C=C\C(=O)O ZINC000217731604 DH For-Sale Unstable SCN10A 20 44 Cc1cc(NC(=O)c2ccc(Cl)o2)ccc1/C=C\C(=O)O ZINC000217731604 DH For-Sale Unstable KCNK3 45 33 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(C)c(C)c1 ZINC000217731613 FG In-Stock Unstable CETP 0 42 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(C)c(C)c1 ZINC000217731613 FG In-Stock Unstable MCHR1 24 43 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(C)c(C)c1 ZINC000217731613 FG In-Stock Unstable MCHR2 41 39 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(C)c(C)c1 ZINC000217731613 FG In-Stock Unstable ENPP1 72 37 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(C)c(C)c1 ZINC000217731613 FG In-Stock Unstable SMO 19 41 O=C(c1cccc(Cl)c1)N1CC(N2C(=O)[C@H]3CC=CC[C@@H]3C2=O)C1 ZINC000217731633 EE In-Stock Unstable SLC6A7 0 42 CCOc1ccc(CCNC(=O)N/C=C/c2ccccc2OC)cc1OCC ZINC000217731640 GI For-Sale Unstable SSTR5 46 36 CCOc1ccc(CCNC(=O)N/C=C/c2ccccc2OC)cc1OCC ZINC000217731640 GI For-Sale Unstable MTNR1A 22 44 CCOc1ccc(CCNC(=O)N/C=C/c2ccccc2OC)cc1OCC ZINC000217731640 GI For-Sale Unstable MTNR1B 25 41 COc1ccc([C@@H](N)C(=O)O)c(OC)c1Cl ZINC000217731650 BD For-Sale Unstable CACNA2D1 19 40 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc(OC(F)F)c2)CC(=O)O4)cc1O ZINC000217731696 JJ In-Stock Unstable AKR1B1 0 42 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc(OC(F)F)c2)CC(=O)O4)cc1O ZINC000217731696 JJ In-Stock Unstable CYP1B1 55 36 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc(OC(F)F)c2)CC(=O)O4)cc1O ZINC000217731696 JJ In-Stock Unstable CYP1A1 35 42 O=C(c1cccc(Cl)c1)N1CC(N2C(=O)[C@@H]3CC=CC[C@H]3C2=O)C1 ZINC000217731722 EE In-Stock Unstable SLC6A7 0 42 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cc(C)cc(C)c1 ZINC000217731726 FG In-Stock Unstable CETP 0 41 COc1ccc2c(c1)C[C@@H](C(=O)NCCCn1ccccc1=O)CO2 ZINC000217731757 ED In-Stock Unstable DRD4 41 34 COc1ccc2c(c1)C[C@@H](C(=O)NCCCn1ccccc1=O)CO2 ZINC000217731757 ED In-Stock Unstable MTNR1A 51 48 COc1ccc2c(c1)C[C@@H](C(=O)NCCCn1ccccc1=O)CO2 ZINC000217731757 ED In-Stock Unstable ROCK2 37 48 COc1ccc2c(c1)C[C@@H](C(=O)NCCCn1ccccc1=O)CO2 ZINC000217731757 ED In-Stock Unstable CDC42BPA 0 47 COc1ccccc1/C=C/NC(=O)Nc1ccc(C(C)(C)C)cc1 ZINC000217731766 DJ For-Sale Unstable TRPV1 21 47 COc1ccccc1/C=C/NC(=O)Nc1ccc(C(C)(C)C)cc1 ZINC000217731766 DJ For-Sale Unstable P2RY1 15 42 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc(OC(F)F)c2)CC(=O)O4)cc1O ZINC000217731778 JJ In-Stock Unstable AKR1B1 0 42 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc(OC(F)F)c2)CC(=O)O4)cc1O ZINC000217731778 JJ In-Stock Unstable CYP1B1 55 36 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc(OC(F)F)c2)CC(=O)O4)cc1O ZINC000217731778 JJ In-Stock Unstable CYP1A1 35 42 Cn1ccc(C(=O)N2CCC3(CC2)CNC(=O)C3)n1 ZINC000217731831 CC For-Sale Unstable ACACA 47 37 COc1ccc2c(c1)C[C@H](C(=O)NCCCn1ccccc1=O)CO2 ZINC000217731832 ED In-Stock Unstable DRD4 41 34 COc1ccc2c(c1)C[C@H](C(=O)NCCCn1ccccc1=O)CO2 ZINC000217731832 ED In-Stock Unstable MTNR1A 51 48 COc1ccc2c(c1)C[C@H](C(=O)NCCCn1ccccc1=O)CO2 ZINC000217731832 ED In-Stock Unstable ROCK2 37 48 COc1ccc2c(c1)C[C@H](C(=O)NCCCn1ccccc1=O)CO2 ZINC000217731832 ED In-Stock Unstable CDC42BPA 0 47 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccccc1F ZINC000217731845 EF In-Stock Unstable LTB4R 18 45 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccccc1F ZINC000217731845 EF In-Stock Unstable CPT1A 43 30 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccccc1F ZINC000217731845 EF In-Stock Unstable KDR 15 42 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccccc1F ZINC000217731845 EF In-Stock Unstable PDGFRA 24 42 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccccc1F ZINC000217731845 EF In-Stock Unstable GLMU 0 41 O=C(O)c1cnnc(N2CCNCC2)c1 ZINC000217731910 BB In-Stock Unstable PRKD1 33 40 O=C1CC2(CCN(C(=O)c3ccnc(F)c3)CC2)CN1 ZINC000217731940 CC For-Sale Unstable ACACA 63 37 O=C1CC2(CCN(C(=O)c3ccnc(F)c3)CC2)CN1 ZINC000217731940 CC For-Sale Unstable ACACB 49 34 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(F)cc1 ZINC000217731963 EF In-Stock Unstable ADORA2B 34 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(F)cc1 ZINC000217731963 EF In-Stock Unstable CETP 0 42 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(F)cc1 ZINC000217731963 EF In-Stock Unstable KDR 25 42 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(F)cc1 ZINC000217731963 EF In-Stock Unstable MET 19 41 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(F)cc1 ZINC000217731963 EF In-Stock Unstable PDGFRA 48 42 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(F)cc1 ZINC000217731963 EF In-Stock Unstable ENPP1 59 34 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(F)cc1 ZINC000217731963 EF In-Stock Unstable DRTS_TRYCR 45 32 CC(C)(C)[C@@H]1CCCC[C@@H]1NC(=O)[C@@H](Cl)c1ccccc1 ZINC000217731986 DJ For-Sale Unstable AMY2 44 31 O=C(Nc1cc(Br)cc2cc[nH]c12)C1CC1 ZINC000217732015 CG For-Sale Unstable ROCK2 15 41 O=C1[C@@H]2[C@@H](ON(c3cccc(Br)c3)[C@H]2c2ccc(Cl)cc2)C(=O)N1c1cccc(Br)c1 ZINC000217732018 KK In-Stock Anodyne ACHE 15 60 O=C(O)c1cnnc(N2CCCNCC2)c1 ZINC000217732024 BB In-Stock Unstable CHRNA4 38 43 O=C(/C=C\c1ccc(F)cc1)Nc1cc(C(=O)O)ccn1 ZINC000217732054 CF For-Sale Anodyne MAPK14 23 54 O=C(/C=C\c1ccc(F)cc1)Nc1cc(C(=O)O)ccn1 ZINC000217732054 CF For-Sale Anodyne CSNK1D 21 40 O=C(/C=C\c1ccc(F)cc1)Nc1cc(C(=O)O)ccn1 ZINC000217732054 CF For-Sale Anodyne MMP2 15 53 O=C(/C=C\c1ccc(F)cc1)Nc1cc(C(=O)O)ccn1 ZINC000217732054 CF For-Sale Anodyne HDAC1 0 40 O=C(/C=C\c1ccc(F)cc1)Nc1cc(C(=O)O)ccn1 ZINC000217732054 CF For-Sale Anodyne MMP9 0 53 O=C(/C=C\c1ccc(F)cc1)Nc1cc(C(=O)O)ccn1 ZINC000217732054 CF For-Sale Anodyne MMP1 24 53 O=C(/C=C\c1ccc(F)cc1)Nc1cc(C(=O)O)ccn1 ZINC000217732054 CF For-Sale Anodyne MCHR1 0 41 CC(C)(C)[C@H]1CCCC[C@@H]1NC(=O)[C@@H](Cl)c1ccccc1 ZINC000217732058 DJ For-Sale Unstable AMY2 44 31 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccccc1Cl ZINC000217732062 FG In-Stock Unstable LTB4R 20 45 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccccc1Cl ZINC000217732062 FG In-Stock Unstable CPT1A 46 32 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccccc1Cl ZINC000217732062 FG In-Stock Unstable EPHB3 41 37 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccccc1Cl ZINC000217732062 FG In-Stock Unstable ADCYAP1R1 37 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccccc1Cl ZINC000217732062 FG In-Stock Unstable SMO 25 44 COc1ccccc1-n1ccc2cc(Br)cc(NC(=O)C3CC3)c21 ZINC000217732134 GJ For-Sale Unstable HTR1A 21 45 CC(C)(C)[C@@H]1CCCC[C@H]1NC(=O)[C@@H](Cl)c1ccccc1 ZINC000217732149 DJ For-Sale Unstable AMY2 44 31 CCC[C@H](O)CN[C@@H]1CC[C@@H](NC(=O)OC(C)(C)C)C1 ZINC000217732152 CE For-Sale Unstable PGA5 43 40 O=C(/C=C\c1ccccc1)Nc1cc(C(=O)O)ccn1 ZINC000217732153 CE For-Sale Anodyne HDAC8 60 48 O=C(/C=C\c1ccccc1)Nc1cc(C(=O)O)ccn1 ZINC000217732153 CE For-Sale Anodyne F3 18 42 O=C(/C=C\c1ccccc1)Nc1cc(C(=O)O)ccn1 ZINC000217732153 CE For-Sale Anodyne MMP2 24 54 O=C(/C=C\c1ccccc1)Nc1cc(C(=O)O)ccn1 ZINC000217732153 CE For-Sale Anodyne HDAC1 32 40 O=C(/C=C\c1ccccc1)Nc1cc(C(=O)O)ccn1 ZINC000217732153 CE For-Sale Anodyne HDAC6 45 50 O=C(/C=C\c1ccccc1)Nc1cc(C(=O)O)ccn1 ZINC000217732153 CE For-Sale Anodyne MMP9 16 54 C[C@H]1CCC[C@H](C)N1CCNC(=O)c1cc(Cl)ccc1O ZINC000217732170 DG On-Demand Unstable KCNMA1 25 43 CC(=O)N[C@@H](C)c1cccc(/C=C\C(=O)O)c1 ZINC000217732184 BD For-Sale Unstable KCNQ2 41 35 CC(=O)N[C@@H](C)c1cccc(/C=C\C(=O)O)c1 ZINC000217732184 BD For-Sale Unstable ACACA 22 45 CC(=O)N[C@@H](C)c1cccc(/C=C\C(=O)O)c1 ZINC000217732184 BD For-Sale Unstable RHOA 0 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(Cl)c1 ZINC000217732190 FG In-Stock Unstable PPIA 24 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(Cl)c1 ZINC000217732190 FG In-Stock Unstable FDFT1 0 41 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(Cl)c1 ZINC000217732190 FG In-Stock Unstable UL80 25 44 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(Cl)c1 ZINC000217732190 FG In-Stock Unstable COLA 73 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(Cl)c1 ZINC000217732190 FG In-Stock Unstable CPT1A 67 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(Cl)c1 ZINC000217732190 FG In-Stock Unstable CPT2 45 37 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(Cl)c1 ZINC000217732190 FG In-Stock Unstable GRM4 16 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(Cl)c1 ZINC000217732190 FG In-Stock Unstable CPT1B 48 37 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(Cl)c1 ZINC000217732190 FG In-Stock Unstable PTPN22 23 41 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(Cl)c1 ZINC000217732190 FG In-Stock Unstable CSF1R 18 41 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(Cl)c1 ZINC000217732190 FG In-Stock Unstable TAAR1 23 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(Cl)c1 ZINC000217732190 FG In-Stock Unstable AKR1C3 36 46 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(Cl)c1 ZINC000217732190 FG In-Stock Unstable AKR1C2 22 43 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(Cl)c1 ZINC000217732190 FG In-Stock Unstable ENPP1 49 35 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(Cl)c1 ZINC000217732190 FG In-Stock Unstable SMO 22 43 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(Cl)c1 ZINC000217732190 FG In-Stock Unstable PSBA 0 43 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(Cl)c1 ZINC000217732190 FG In-Stock Unstable KCNK3 58 39 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(Cl)c1 ZINC000217732190 FG In-Stock Unstable KCNK9 62 39 O=C1C[C@@H](C2=Cc3ccccc3OC2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217732215 JJ In-Stock Unstable CYP1A1 21 41 C/C=C\C=C/C(=O)Nc1cc(C(=O)O)ccn1 ZINC000217732228 BD For-Sale Unstable KDM4C 0 42 C/C=C\C=C/C(=O)Nc1cc(C(=O)O)ccn1 ZINC000217732228 BD For-Sale Unstable KDM3A 0 42 C/C=C\C=C/C(=O)Nc1cc(C(=O)O)ccn1 ZINC000217732228 BD For-Sale Unstable KDM5C 0 42 C/C=C\C=C/C(=O)Nc1cc(C(=O)O)ccn1 ZINC000217732228 BD For-Sale Unstable FTO 0 41 COc1ccccc1/C=C/NC(=O)Nc1ccc2cn[nH]c2c1 ZINC000217732229 DG For-Sale Unstable ROCK1 15 40 COc1ccccc1/C=C/NC(=O)Nc1ccc2cn[nH]c2c1 ZINC000217732229 DG For-Sale Unstable IMPDH2 0 43 COc1ccccc1/C=C/NC(=O)Nc1ccc2cn[nH]c2c1 ZINC000217732229 DG For-Sale Unstable ENPP1 40 32 CC(C)Cn1c(Br)nc2ccccc21 ZINC000217732231 CG For-Sale Unstable HRH1 19 47 CC(C)Cn1c(Br)nc2ccccc21 ZINC000217732231 CG For-Sale Unstable ALOX5AP 34 42 CC(C)Cn1c(Br)nc2ccccc21 ZINC000217732231 CG For-Sale Unstable RPS6KB1 19 51 CC(C)(C)[C@H]1CCCC[C@H]1NC(=O)[C@@H](Cl)c1ccccc1 ZINC000217732232 DJ For-Sale Unstable AMY2 44 31 C[C@@H]1CCC[C@@H](C)N1CCNC(=O)c1cc(Cl)ccc1O ZINC000217732249 DG On-Demand Unstable KCNMA1 25 43 CC(=O)N[C@H](C)c1cccc(/C=C\C(=O)O)c1 ZINC000217732277 BD For-Sale Unstable KCNQ2 41 35 CC(=O)N[C@H](C)c1cccc(/C=C\C(=O)O)c1 ZINC000217732277 BD For-Sale Unstable ACACA 22 45 CC(=O)N[C@H](C)c1cccc(/C=C\C(=O)O)c1 ZINC000217732277 BD For-Sale Unstable RHOA 0 40 C/C=C/C=C\C(=O)Nc1cc(C(=O)O)ccn1 ZINC000217732289 BD For-Sale Unstable KDM4C 0 42 C/C=C/C=C\C(=O)Nc1cc(C(=O)O)ccn1 ZINC000217732289 BD For-Sale Unstable KDM3A 0 42 C/C=C/C=C\C(=O)Nc1cc(C(=O)O)ccn1 ZINC000217732289 BD For-Sale Unstable KDM5C 0 42 C/C=C/C=C\C(=O)Nc1cc(C(=O)O)ccn1 ZINC000217732289 BD For-Sale Unstable FTO 0 41 O=C1C[C@H](C2=Cc3ccccc3OC2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217732297 JJ In-Stock Unstable CYP1A1 21 41 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)cc1 ZINC000217732316 FG In-Stock Unstable HTR2A 23 41 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)cc1 ZINC000217732316 FG In-Stock Unstable PTGS2 0 41 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)cc1 ZINC000217732316 FG In-Stock Unstable LTA4H 18 41 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)cc1 ZINC000217732316 FG In-Stock Unstable PTGER1 33 48 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)cc1 ZINC000217732316 FG In-Stock Unstable CETP 0 44 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)cc1 ZINC000217732316 FG In-Stock Unstable COLA 80 47 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)cc1 ZINC000217732316 FG In-Stock Unstable CPT1A 79 47 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)cc1 ZINC000217732316 FG In-Stock Unstable CPT2 50 43 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)cc1 ZINC000217732316 FG In-Stock Unstable KDR 27 42 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)cc1 ZINC000217732316 FG In-Stock Unstable CPT1B 62 43 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)cc1 ZINC000217732316 FG In-Stock Unstable PDGFRA 45 42 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)cc1 ZINC000217732316 FG In-Stock Unstable MCHR1 24 44 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)cc1 ZINC000217732316 FG In-Stock Unstable MCHR2 39 41 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)cc1 ZINC000217732316 FG In-Stock Unstable AKR1C3 27 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)cc1 ZINC000217732316 FG In-Stock Unstable AKR1C2 28 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)cc1 ZINC000217732316 FG In-Stock Unstable ENPP1 63 37 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)cc1 ZINC000217732316 FG In-Stock Unstable SMO 17 41 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)cc1 ZINC000217732316 FG In-Stock Unstable DRTS_TRYCR 45 32 COc1ccccc1/C=C/NC(=O)Nc1ccccc1C(C)(C)C ZINC000217732340 DJ For-Sale Unstable P2RY1 22 41 CCC[C@H](O)CN[C@H]1CC[C@@H](NC(=O)OC(C)(C)C)C1 ZINC000217732341 CE For-Sale Unstable PGA5 43 40 C/C=C\C=C\C(=O)Nc1cc(C(=O)O)ccn1 ZINC000217732362 BD For-Sale Unstable KDM4C 0 42 C/C=C\C=C\C(=O)Nc1cc(C(=O)O)ccn1 ZINC000217732362 BD For-Sale Unstable KDM3A 0 42 C/C=C\C=C\C(=O)Nc1cc(C(=O)O)ccn1 ZINC000217732362 BD For-Sale Unstable KDM5C 0 42 C/C=C\C=C\C(=O)Nc1cc(C(=O)O)ccn1 ZINC000217732362 BD For-Sale Unstable FTO 0 41 Cc1ccc(/C=C\C(=O)O)cc1NC(=O)c1ccccn1 ZINC000217732367 CF For-Sale Unstable GRM4 68 47 Cc1ccc(/C=C\C(=O)O)cc1NC(=O)c1ccccn1 ZINC000217732367 CF For-Sale Unstable MMP1 0 43 Cc1ccc(/C=C\C(=O)O)cc1NC(=O)c1ccccn1 ZINC000217732367 CF For-Sale Unstable SMO 24 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Br)cc1 ZINC000217732436 HG In-Stock Unstable PDGFRB 25 42 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Br)cc1 ZINC000217732436 HG In-Stock Unstable ADORA2B 19 47 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Br)cc1 ZINC000217732436 HG In-Stock Unstable UL80 20 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Br)cc1 ZINC000217732436 HG In-Stock Unstable CETP 0 42 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Br)cc1 ZINC000217732436 HG In-Stock Unstable AKR1C3 15 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Br)cc1 ZINC000217732436 HG In-Stock Unstable AKR1C2 25 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Br)cc1 ZINC000217732436 HG In-Stock Unstable ENPP1 63 36 COc1ccccc1/C=C/NC(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000217732443 GD For-Sale Unstable CA2 101 56 COc1ccccc1/C=C/NC(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000217732443 GD For-Sale Unstable CA1 89 56 COc1ccccc1/C=C/NC(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000217732443 GD For-Sale Unstable CA7 57 53 COc1ccccc1/C=C/NC(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000217732443 GD For-Sale Unstable CA5B 51 53 COc1ccccc1/C=C/NC(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000217732443 GD For-Sale Unstable CA4 60 54 COc1ccccc1/C=C/NC(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000217732443 GD For-Sale Unstable CA5A 52 53 COc1ccccc1/C=C/NC(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000217732443 GD For-Sale Unstable CA14 46 51 COc1ccccc1/C=C/NC(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000217732443 GD For-Sale Unstable CA12 72 56 COc1ccccc1/C=C/NC(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000217732443 GD For-Sale Unstable CA9 80 56 COc1ccccc1/C=C/NC(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000217732443 GD For-Sale Unstable CYNT 26 45 COc1ccccc1/C=C/NC(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000217732443 GD For-Sale Unstable NCE103 36 51 COc1ccccc1/C=C/NC(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000217732443 GD For-Sale Unstable LIG1 0 43 COc1ccccc1/C=C/NC(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000217732443 GD For-Sale Unstable MTCA1 33 45 COc1ccccc1/C=C/NC(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000217732443 GD For-Sale Unstable P96878_MYCTU 50 45 COc1ccccc1/C=C/NC(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000217732443 GD For-Sale Unstable CAN2 0 41 COc1ccccc1/C=C/NC(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000217732443 GD For-Sale Unstable A6YCJ1_9METZ 24 47 Cc1ccc(/C=C\C(=O)O)cc1NC(=O)c1ccncc1 ZINC000217732449 CF For-Sale Unstable MAPK11 27 40 Cc1ccc(/C=C\C(=O)O)cc1NC(=O)c1ccncc1 ZINC000217732449 CF For-Sale Unstable SMO 22 41 Cc1ccc(/C=C\C(=O)O)cc1NC(=O)c1ccncc1 ZINC000217732449 CF For-Sale Unstable KCNK3 42 44 O=C(/C=C\c1ccc(O)cc1)Nc1cc(C(=O)O)ccn1 ZINC000217732452 CE For-Sale Anodyne HDAC8 31 40 O=C(/C=C\c1ccc(O)cc1)Nc1cc(C(=O)O)ccn1 ZINC000217732452 CE For-Sale Anodyne F3 26 42 O=C(/C=C\c1ccc(O)cc1)Nc1cc(C(=O)O)ccn1 ZINC000217732452 CE For-Sale Anodyne MMP2 23 52 O=C(/C=C\c1ccc(O)cc1)Nc1cc(C(=O)O)ccn1 ZINC000217732452 CE For-Sale Anodyne HDAC6 15 45 O=C(/C=C\c1ccc(O)cc1)Nc1cc(C(=O)O)ccn1 ZINC000217732452 CE For-Sale Anodyne MMP9 17 52 COc1cccc(C(=O)NC[C@@H]2CCCN2c2nccs2)c1OC ZINC000217732457 EF For-Sale Unstable DRD2 47 46 COc1cccc(C(=O)NC[C@@H]2CCCN2c2nccs2)c1OC ZINC000217732457 EF For-Sale Unstable DRD3 20 46 COc1cccc(C(=O)NC[C@@H]2CCCN2c2nccs2)c1OC ZINC000217732457 EF For-Sale Unstable HCN1 50 32 COc1cccc(C(=O)NC[C@@H]2CCCN2c2nccs2)c1OC ZINC000217732457 EF For-Sale Unstable HCN4 48 32 COc1cccc(C(=O)NC[C@@H]2CCCN2c2nccs2)c1OC ZINC000217732457 EF For-Sale Unstable ACKR3 64 34 CCOc1ccc([C@@H](C)N[C@@H]2CCC[C@@H](C)C2)cc1 ZINC000217732462 CI For-Sale Unstable ACACA 41 43 CCOc1ccc([C@@H](C)N[C@@H]2CCC[C@@H](C)C2)cc1 ZINC000217732462 CI For-Sale Unstable ACACB 20 43 CCOc1ccc([C@H](C)N[C@@H]2CCC[C@@H](C)C2)cc1 ZINC000217732521 CI For-Sale Unstable ACACA 41 43 CCOc1ccc([C@H](C)N[C@@H]2CCC[C@@H](C)C2)cc1 ZINC000217732521 CI For-Sale Unstable ACACB 20 43 Cc1ccc(/C=C\C(=O)O)cc1NC(=O)c1cccnc1 ZINC000217732539 CF For-Sale Unstable TBXAS1 39 45 Cc1ccc(/C=C\C(=O)O)cc1NC(=O)c1cccnc1 ZINC000217732539 CF For-Sale Unstable MAPK11 15 42 Cc1ccc(/C=C\C(=O)O)cc1NC(=O)c1cccnc1 ZINC000217732539 CF For-Sale Unstable MAPK14 17 42 Cc1ccc(/C=C\C(=O)O)cc1NC(=O)c1cccnc1 ZINC000217732539 CF For-Sale Unstable HDAC1 0 47 COc1cccc(C(=O)NC[C@H]2CCCN2c2nccs2)c1OC ZINC000217732542 EF For-Sale Unstable DRD2 47 46 COc1cccc(C(=O)NC[C@H]2CCCN2c2nccs2)c1OC ZINC000217732542 EF For-Sale Unstable DRD3 20 46 COc1cccc(C(=O)NC[C@H]2CCCN2c2nccs2)c1OC ZINC000217732542 EF For-Sale Unstable HCN1 50 32 COc1cccc(C(=O)NC[C@H]2CCCN2c2nccs2)c1OC ZINC000217732542 EF For-Sale Unstable HCN4 48 32 COc1cccc(C(=O)NC[C@H]2CCCN2c2nccs2)c1OC ZINC000217732542 EF For-Sale Unstable ACKR3 64 34 COc1ccccc1/C=C/NC(=O)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217732554 HK For-Sale Unstable PTPA 0 43 COc1ccccc1/C=C/NC(=O)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217732554 HK For-Sale Unstable KCNK3 49 37 COc1ccccc1/C=C/NC(=O)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217732554 HK For-Sale Unstable KCNK9 41 37 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(C)c(Cl)c1 ZINC000217732559 GG In-Stock Unstable CETP 0 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(C)c(Cl)c1 ZINC000217732559 GG In-Stock Unstable COLA 45 38 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(C)c(Cl)c1 ZINC000217732559 GG In-Stock Unstable CPT1A 46 38 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(C)c(Cl)c1 ZINC000217732559 GG In-Stock Unstable CPT2 45 36 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(C)c(Cl)c1 ZINC000217732559 GG In-Stock Unstable GRM4 19 41 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(C)c(Cl)c1 ZINC000217732559 GG In-Stock Unstable MCHR1 23 43 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(C)c(Cl)c1 ZINC000217732559 GG In-Stock Unstable MCHR2 43 43 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(C)c(Cl)c1 ZINC000217732559 GG In-Stock Unstable ENPP1 70 35 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(C)c(Cl)c1 ZINC000217732559 GG In-Stock Unstable SMO 19 41 O=C(N[C@@H]1COC2(CCNCC2)C1)c1cc(Cl)ccc1O ZINC000217732621 DD In-Stock Unstable KCNMA1 23 41 CCOc1ccc([C@@H](C)N[C@H]2CCC[C@@H](C)C2)cc1 ZINC000217732625 CI For-Sale Unstable ACACA 41 43 CCOc1ccc([C@@H](C)N[C@H]2CCC[C@@H](C)C2)cc1 ZINC000217732625 CI For-Sale Unstable ACACB 20 43 O=C(/C=C\c1ccccc1Br)Nc1cnccc1C(=O)O ZINC000217732630 EG For-Sale Anodyne LTB4R 0 45 COc1cccc(OC)c1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217732654 EF For-Sale Unstable DRD2 43 43 COc1cccc(OC)c1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217732654 EF For-Sale Unstable ACKR3 68 34 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217732665 HH In-Stock Unstable EGFR 19 42 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217732665 HH In-Stock Unstable HTR2A 17 42 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217732665 HH In-Stock Unstable COLA 52 39 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217732665 HH In-Stock Unstable CPT1A 52 39 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217732665 HH In-Stock Unstable CPT2 44 36 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217732665 HH In-Stock Unstable GRM4 23 44 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217732665 HH In-Stock Unstable PDGFRA 39 44 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217732665 HH In-Stock Unstable CSF1R 27 41 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217732665 HH In-Stock Unstable MCHR1 23 42 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217732665 HH In-Stock Unstable MCHR2 41 42 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217732665 HH In-Stock Unstable SHH 21 41 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217732665 HH In-Stock Unstable PFK 0 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217732665 HH In-Stock Unstable ENPP1 74 38 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217732665 HH In-Stock Unstable SMO 22 44 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217732665 HH In-Stock Unstable IMDH_CRYPV 43 43 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217732665 HH In-Stock Unstable P95276_MYCTO 0 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217732665 HH In-Stock Unstable PPX1 0 42 Cc1c(C(=O)N2CC(N3C(=O)[C@H]4CC=CC[C@H]4C3=O)C2)cnn1-c1ccccc1 ZINC000217732677 GD In-Stock Unstable SLC9A2 0 47 O=C(N[C@H]1COC2(CCNCC2)C1)c1cc(Cl)ccc1O ZINC000217732700 DD In-Stock Unstable KCNMA1 23 41 CCOc1ccc([C@H](C)N[C@H]2CCC[C@@H](C)C2)cc1 ZINC000217732704 CI For-Sale Unstable ACACA 41 43 CCOc1ccc([C@H](C)N[C@H]2CCC[C@@H](C)C2)cc1 ZINC000217732704 CI For-Sale Unstable ACACB 20 43 Cc1ccsc1/C=C\C(=O)Nc1cnccc1C(=O)O ZINC000217732707 CF For-Sale Unstable UL26 18 42 Cc1ccsc1/C=C\C(=O)Nc1cnccc1C(=O)O ZINC000217732707 CF For-Sale Unstable SCAF_EBVB9 15 42 CNC(=O)[C@@H]1CCCN([C@@H](C)C(=O)OC(C)(C)C)C1 ZINC000217732720 CD On-Demand Unstable SSTR2 44 38 COc1cccc(OC)c1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217732743 EF For-Sale Unstable DRD2 43 43 COc1cccc(OC)c1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217732743 EF For-Sale Unstable ACKR3 68 34 Cc1c(C(=O)N2CC(N3C(=O)[C@H]4CC=CC[C@@H]4C3=O)C2)cnn1-c1ccccc1 ZINC000217732763 GD In-Stock Unstable SLC9A2 0 47 O=C(CBr)c1ccc(OCCCO)cc1 ZINC000217732773 CE For-Sale Unstable PLA2G4B 78 42 O=C(CBr)c1ccc(OCCCO)cc1 ZINC000217732773 CE For-Sale Unstable LSS 16 46 O=C(CBr)c1ccc(OCCCO)cc1 ZINC000217732773 CE For-Sale Unstable ACR 27 42 Cc1ccc(/C=C\C(=O)Nc2cc(C(=O)O)ccn2)cc1 ZINC000217732779 CF For-Sale Unstable HDAC8 44 39 Cc1ccc(/C=C\C(=O)Nc2cc(C(=O)O)ccn2)cc1 ZINC000217732779 CF For-Sale Unstable MMP2 15 53 Cc1ccc(/C=C\C(=O)Nc2cc(C(=O)O)ccn2)cc1 ZINC000217732779 CF For-Sale Unstable MMP9 0 49 Cc1ccc(/C=C\C(=O)Nc2cc(C(=O)O)ccn2)cc1 ZINC000217732779 CF For-Sale Unstable MMP1 23 49 Cc1ccc(/C=C\C(=O)Nc2cc(C(=O)O)ccn2)cc1 ZINC000217732779 CF For-Sale Unstable MCHR1 15 42 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000217732782 HH In-Stock Unstable CPT1A 45 32 CCCCCCCCOc1ccc([C@@H]2CC(=O)Oc3cc4c(cc32)OCO4)cc1 ZINC000217732796 GK In-Stock Unstable THRA 39 41 CCCCCCCCOc1ccc([C@@H]2CC(=O)Oc3cc4c(cc32)OCO4)cc1 ZINC000217732796 GK In-Stock Unstable EDNRB 28 41 CCCCCCCCOc1ccc([C@@H]2CC(=O)Oc3cc4c(cc32)OCO4)cc1 ZINC000217732796 GK In-Stock Unstable EDNRA 32 41 CCCCCCCCOc1ccc([C@@H]2CC(=O)Oc3cc4c(cc32)OCO4)cc1 ZINC000217732796 GK In-Stock Unstable THRB 23 41 CCCCCCCCOc1ccc([C@@H]2CC(=O)Oc3cc4c(cc32)OCO4)cc1 ZINC000217732796 GK In-Stock Unstable PLA2G4B 79 34 Cc1occc1C(=O)Nc1cccc(/C=C\C(=O)O)n1 ZINC000217732797 CE For-Sale Unstable SORT1 25 40 Cc1cc(C)c(CS(=O)(=O)Cl)c(Cl)c1 ZINC000217732809 CG For-Sale Unstable RAPGEF4 51 33 Cc1c(C(=O)N2CC(N3C(=O)[C@@H]4CC=CC[C@H]4C3=O)C2)cnn1-c1ccccc1 ZINC000217732838 GD In-Stock Unstable SLC9A2 0 47 O=C(/C=C\c1ccc(Br)cc1)Nc1cc(C(=O)O)ccn1 ZINC000217732862 EG For-Sale Anodyne HDAC8 42 42 O=C(/C=C\c1ccc(Br)cc1)Nc1cc(C(=O)O)ccn1 ZINC000217732862 EG For-Sale Anodyne MMP2 0 42 O=C(/C=C\c1ccc(Br)cc1)Nc1cc(C(=O)O)ccn1 ZINC000217732862 EG For-Sale Anodyne HDAC6 26 42 O=C(/C=C\c1ccc(Br)cc1)Nc1cc(C(=O)O)ccn1 ZINC000217732862 EG For-Sale Anodyne MMP9 0 40 O=C(/C=C\c1ccc(Br)cc1)Nc1cc(C(=O)O)ccn1 ZINC000217732862 EG For-Sale Anodyne MMP1 23 40 COc1ccc(C(=O)NC[C@@H]2CCCN2c2nccs2)cc1OC ZINC000217732865 EF For-Sale Unstable SLC5A7 30 41 COc1ccc(C(=O)NC[C@@H]2CCCN2c2nccs2)cc1OC ZINC000217732865 EF For-Sale Unstable ACKR3 72 40 CCCCCCCCOc1ccc([C@H]2CC(=O)Oc3cc4c(cc32)OCO4)cc1 ZINC000217732876 GK In-Stock Unstable THRA 39 41 CCCCCCCCOc1ccc([C@H]2CC(=O)Oc3cc4c(cc32)OCO4)cc1 ZINC000217732876 GK In-Stock Unstable EDNRB 25 41 CCCCCCCCOc1ccc([C@H]2CC(=O)Oc3cc4c(cc32)OCO4)cc1 ZINC000217732876 GK In-Stock Unstable EDNRA 32 41 CCCCCCCCOc1ccc([C@H]2CC(=O)Oc3cc4c(cc32)OCO4)cc1 ZINC000217732876 GK In-Stock Unstable THRB 23 41 CCCCCCCCOc1ccc([C@H]2CC(=O)Oc3cc4c(cc32)OCO4)cc1 ZINC000217732876 GK In-Stock Unstable PLA2G4B 69 34 COc1ccccc1/C=C/NC(=O)Nc1ccc(C(N)=O)cc1 ZINC000217732886 DF For-Sale Unstable PPIA 19 42 COc1ccccc1/C=C/NC(=O)Nc1ccc(C(N)=O)cc1 ZINC000217732886 DF For-Sale Unstable ACR 40 47 COc1ccccc1/C=C/NC(=O)Nc1ccc(C(N)=O)cc1 ZINC000217732886 DF For-Sale Unstable CA12 15 41 COc1ccccc1/C=C/NC(=O)Nc1ccc(C(N)=O)cc1 ZINC000217732886 DF For-Sale Unstable PDGFRA 43 38 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217732897 GG In-Stock Unstable KIT 17 41 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217732897 GG In-Stock Unstable UL80 32 46 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217732897 GG In-Stock Unstable KDR 28 44 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217732897 GG In-Stock Unstable CSF1R 15 41 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217732897 GG In-Stock Unstable TEK 33 41 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217732897 GG In-Stock Unstable MCHR1 26 41 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217732897 GG In-Stock Unstable HIF1A 19 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217732897 GG In-Stock Unstable AKR1C3 29 48 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217732897 GG In-Stock Unstable SCD1 32 41 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217732897 GG In-Stock Unstable RIPK1 44 34 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217732897 GG In-Stock Unstable ADCYAP1R1 27 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217732897 GG In-Stock Unstable AKR1C2 16 47 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217732897 GG In-Stock Unstable ENPP1 40 31 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217732897 GG In-Stock Unstable SMO 20 42 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217732897 GG In-Stock Unstable TRPM4 0 42 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217732897 GG In-Stock Unstable KCNK3 75 45 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217732897 GG In-Stock Unstable KCNK9 62 39 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217732897 GG In-Stock Unstable PDS 40 41 COc1ccc(C(=O)NC[C@H]2CCCN2c2nccs2)cc1OC ZINC000217732958 EF For-Sale Unstable SLC5A7 30 41 COc1ccc(C(=O)NC[C@H]2CCCN2c2nccs2)cc1OC ZINC000217732958 EF For-Sale Unstable ACKR3 72 40 COc1ccc2c(c1)CCC[C@H]2N[C@@H]1CCN2CCC[C@@H]12 ZINC000217732976 CF For-Sale Unstable EBP 25 47 COc1ccccc1/C=C/NC(=O)Nc1ccc(F)c(Cl)c1 ZINC000217732998 DI For-Sale Unstable HTR2A 18 41 COc1ccccc1/C=C/NC(=O)Nc1ccc(F)c(Cl)c1 ZINC000217732998 DI For-Sale Unstable GCGR 0 40 COc1ccccc1/C=C/NC(=O)Nc1ccc(F)c(Cl)c1 ZINC000217732998 DI For-Sale Unstable PYGL 0 42 COc1ccccc1/C=C/NC(=O)Nc1ccc(F)c(Cl)c1 ZINC000217732998 DI For-Sale Unstable GRM4 24 43 COc1ccccc1/C=C/NC(=O)Nc1ccc(F)c(Cl)c1 ZINC000217732998 DI For-Sale Unstable IMPDH2 0 42 COC(=O)[C@@H](O)CNC(=O)COc1cccc(Br)c1 ZINC000217733007 EC On-Demand Unstable PDS 59 43 COc1ccccc1NC(=O)COc1c(OC)cc(C(=O)O)cc1OC ZINC000217733013 FE In-Stock Unstable CPT1A 43 30 COc1ccccc1NC(=O)COc1c(OC)cc(C(=O)O)cc1OC ZINC000217733013 FE In-Stock Unstable ABCB1 0 41 COc1ccccc1NC(=O)COc1c(OC)cc(C(=O)O)cc1OC ZINC000217733013 FE In-Stock Unstable KCNK3 43 36 O=C(/C=C\c1ccc(Cl)cc1)Nc1cc(C(=O)O)ccn1 ZINC000217733045 DG For-Sale Anodyne MMP2 15 53 O=C(/C=C\c1ccc(Cl)cc1)Nc1cc(C(=O)O)ccn1 ZINC000217733045 DG For-Sale Anodyne MMP9 0 53 O=C(/C=C\c1ccc(Cl)cc1)Nc1cc(C(=O)O)ccn1 ZINC000217733045 DG For-Sale Anodyne MMP1 24 53 CC[C@@H](C)N(CC(=O)Nc1cccc(C)c1C)C(=O)CC1CCCC1 ZINC000217733052 EI On-Demand Unstable DEF 0 41 COc1ccccc1OCC(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217733058 EE For-Sale Unstable MBTPS1 49 34 COc1ccccc1OCC(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217733058 EE For-Sale Unstable ACKR3 63 33 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(OC)c(OC)c2OC)CC(=O)O4)cc1O ZINC000217733086 KI In-Stock Unstable ALOX5 0 52 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(OC)c(OC)c2OC)CC(=O)O4)cc1O ZINC000217733086 KI In-Stock Unstable AKR1B1 23 52 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(OC)c(OC)c2OC)CC(=O)O4)cc1O ZINC000217733086 KI In-Stock Unstable CYP1B1 68 38 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(OC)c(OC)c2OC)CC(=O)O4)cc1O ZINC000217733086 KI In-Stock Unstable CYP1A1 48 48 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(OC)c(OC)c2OC)CC(=O)O4)cc1O ZINC000217733086 KI In-Stock Unstable CYP1A2 38 41 COc1ccc2c(c1)CCC[C@@H]2N[C@@H]1CCN2CCC[C@@H]12 ZINC000217733092 CF For-Sale Unstable EBP 25 47 COC(=O)[C@H](O)CNC(=O)COc1cccc(Br)c1 ZINC000217733093 EC On-Demand Unstable PDS 59 43 COc1cccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)c1 ZINC000217733101 FE In-Stock Unstable DRD4 41 31 COc1cccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)c1 ZINC000217733101 FE In-Stock Unstable PDGFRB 48 48 COc1cccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)c1 ZINC000217733101 FE In-Stock Unstable LTA4H 15 41 COc1cccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)c1 ZINC000217733101 FE In-Stock Unstable CPT1A 43 30 COc1cccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)c1 ZINC000217733101 FE In-Stock Unstable KDR 28 44 COc1cccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)c1 ZINC000217733101 FE In-Stock Unstable MTNR1A 57 50 COc1cccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)c1 ZINC000217733101 FE In-Stock Unstable MTNR1B 59 54 COc1cccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)c1 ZINC000217733101 FE In-Stock Unstable EPHX2 17 40 COc1cccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)c1 ZINC000217733101 FE In-Stock Unstable FLT4 28 48 COc1cccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)c1 ZINC000217733101 FE In-Stock Unstable PDGFRA 30 44 COc1cccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)c1 ZINC000217733101 FE In-Stock Unstable CSF1R 19 48 COc1cccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)c1 ZINC000217733101 FE In-Stock Unstable MCHR1 25 42 COc1cccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)c1 ZINC000217733101 FE In-Stock Unstable TAAR1 42 45 COc1cccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)c1 ZINC000217733101 FE In-Stock Unstable AKR1C3 50 46 COc1cccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)c1 ZINC000217733101 FE In-Stock Unstable AKR1C2 52 37 COc1cccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)c1 ZINC000217733101 FE In-Stock Unstable ENPP1 57 33 COc1cccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)c1 ZINC000217733101 FE In-Stock Unstable SMO 23 44 COc1cccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)c1 ZINC000217733101 FE In-Stock Unstable KCNK3 82 48 COc1cccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)c1 ZINC000217733101 FE In-Stock Unstable KCNK9 60 42 CCN(CC)c1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217733116 EI For-Sale Unstable MTNR1B 15 45 CCN(CC)c1ccc(NC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217733116 EI For-Sale Unstable GHSR 0 48 CN(C)C1[C@H]2CNC[C@H]1CN(Cc1ccccc1)C2 ZINC000217733131 CD For-Sale Unstable SIGMAR1 43 42 CC[C@H](C)N(CC(=O)Nc1cccc(C)c1C)C(=O)CC1CCCC1 ZINC000217733134 EI On-Demand Unstable DEF 0 41 COc1ccccc1OCC(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217733142 EE For-Sale Unstable MBTPS1 49 34 COc1ccccc1OCC(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217733142 EE For-Sale Unstable ACKR3 63 33 Cc1ccc(C=O)c(N2CCCC2)n1 ZINC000217733159 AD In-Stock Unstable NPY5R 0 40 CCOC(=O)[C@@H](CN(CC)CC)NCc1ccccc1 ZINC000217733162 CE For-Sale Unstable MME 42 34 CCOC(=O)[C@@H](CN(CC)CC)NCc1ccccc1 ZINC000217733162 CE For-Sale Unstable ANPEP 55 34 CCOC(=O)[C@@H](CN(CC)CC)NCc1ccccc1 ZINC000217733162 CE For-Sale Unstable CPA1 30 47 CCOC(=O)[C@@H](CN(CC)CC)NCc1ccccc1 ZINC000217733162 CE For-Sale Unstable CAPN2 50 35 CCOC(=O)[C@@H](CN(CC)CC)NCc1ccccc1 ZINC000217733162 CE For-Sale Unstable NPR 65 36 CCOC(=O)[C@@H](CN(CC)CC)NCc1ccccc1 ZINC000217733162 CE For-Sale Unstable PDS 49 36 O=C(O)[C@@H]1Cc2ccccc2CN1C(=O)c1cc(-n2cnnn2)ccc1O ZINC000217733165 FD In-Stock Unstable AGTR2 47 42 O=C(O)[C@@H]1Cc2ccccc2CN1C(=O)c1cc(-n2cnnn2)ccc1O ZINC000217733165 FD In-Stock Unstable CFTR 49 37 COc1ccc2c(c1)CCC[C@H]2N[C@H]1CCN2CCC[C@@H]12 ZINC000217733170 CF For-Sale Unstable EBP 25 47 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(OC)c(OC)c2OC)CC(=O)O4)cc1O ZINC000217733174 KI In-Stock Unstable ALOX5 0 52 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(OC)c(OC)c2OC)CC(=O)O4)cc1O ZINC000217733174 KI In-Stock Unstable AKR1B1 23 52 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(OC)c(OC)c2OC)CC(=O)O4)cc1O ZINC000217733174 KI In-Stock Unstable CYP1B1 68 38 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(OC)c(OC)c2OC)CC(=O)O4)cc1O ZINC000217733174 KI In-Stock Unstable CYP1A1 48 48 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(OC)c(OC)c2OC)CC(=O)O4)cc1O ZINC000217733174 KI In-Stock Unstable CYP1A2 38 41 Cc1ncccc1NC(=O)c1ccc2c(c1)CC(=O)N2 ZINC000217733197 CE For-Sale Unstable G2YM83_BOTF4 61 35 O=C(O)/C=C\c1cnc(NC(=O)Cc2ccccn2)s1 ZINC000217733210 CD For-Sale Unstable CDK5 44 45 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733215 FE In-Stock Unstable TSHR 48 34 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733215 FE In-Stock Unstable PDGFRB 57 41 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733215 FE In-Stock Unstable ADORA2A 18 40 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733215 FE In-Stock Unstable ADORA2B 44 39 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733215 FE In-Stock Unstable CETP 0 44 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733215 FE In-Stock Unstable CPT1A 43 30 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733215 FE In-Stock Unstable GUAB 0 42 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733215 FE In-Stock Unstable TNFRSF1A 19 40 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733215 FE In-Stock Unstable HDAC8 25 44 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733215 FE In-Stock Unstable KDR 42 39 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733215 FE In-Stock Unstable MTNR1A 50 44 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733215 FE In-Stock Unstable MTNR1B 47 48 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733215 FE In-Stock Unstable PLA2G4B 36 41 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733215 FE In-Stock Unstable P4HTM 0 40 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733215 FE In-Stock Unstable FLT4 33 41 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733215 FE In-Stock Unstable TUBB2B 22 41 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733215 FE In-Stock Unstable ACR 50 41 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733215 FE In-Stock Unstable CA12 17 42 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733215 FE In-Stock Unstable PDGFRA 58 43 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733215 FE In-Stock Unstable FLT3 18 41 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733215 FE In-Stock Unstable CSF1R 20 41 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733215 FE In-Stock Unstable CA9 20 42 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733215 FE In-Stock Unstable MCHR1 30 48 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733215 FE In-Stock Unstable AKR1C3 38 46 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733215 FE In-Stock Unstable AKR1C2 52 41 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733215 FE In-Stock Unstable ENPP1 72 35 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733215 FE In-Stock Unstable IMDH_CRYPV 17 40 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733215 FE In-Stock Unstable DRTS_TRYCR 45 32 COc1ccccc1/C=C/NC(=O)NCc1ccc(F)cc1 ZINC000217733224 DG For-Sale Unstable GRIN2B 0 40 COc1ccccc1/C=C/NC(=O)NCc1ccc(F)cc1 ZINC000217733224 DG For-Sale Unstable TLR4 16 42 CCOc1ccccc1C(=O)N(CC(=O)Nc1cccc(C)c1C)[C@@H](C)CC ZINC000217733240 GJ On-Demand Unstable HCN1 50 34 CCOc1ccccc1C(=O)N(CC(=O)Nc1cccc(C)c1C)[C@@H](C)CC ZINC000217733240 GJ On-Demand Unstable HCN4 41 34 CCOc1ccccc1C(=O)N(CC(=O)Nc1cccc(C)c1C)[C@@H](C)CC ZINC000217733240 GJ On-Demand Unstable KCNK3 27 40 CCOc1ccccc1C(=O)N(CC(=O)Nc1cccc(C)c1C)[C@@H](C)CC ZINC000217733240 GJ On-Demand Unstable KCNK9 25 40 O=C(O)[C@H]1Cc2ccccc2CN1C(=O)c1cc(-n2cnnn2)ccc1O ZINC000217733250 FD In-Stock Unstable AGTR2 47 42 O=C(O)[C@H]1Cc2ccccc2CN1C(=O)c1cc(-n2cnnn2)ccc1O ZINC000217733250 FD In-Stock Unstable CFTR 49 37 COc1cccc(OCC(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217733258 EE For-Sale Unstable CHRNA10 35 44 COc1ccc2c(c1)CCC[C@@H]2N[C@H]1CCN2CCC[C@@H]12 ZINC000217733264 CF For-Sale Unstable EBP 25 47 Cc1ccc(C=O)c(N2CCCCC2)n1 ZINC000217733266 BE In-Stock Unstable NPY5R 22 42 O=C(O)/C=C\c1cnc(NC(=O)Cc2ccc(Cl)cc2)s1 ZINC000217733286 DG For-Sale Unstable CSNK1D 21 42 O=C(O)/C=C\c1cnc(NC(=O)Cc2ccc(Cl)cc2)s1 ZINC000217733286 DG For-Sale Unstable CDK5 39 46 CCOc1ccccc1C(=O)N(CC(=O)Nc1cccc(C)c1C)[C@H](C)CC ZINC000217733317 GJ On-Demand Unstable HCN1 50 34 CCOc1ccccc1C(=O)N(CC(=O)Nc1cccc(C)c1C)[C@H](C)CC ZINC000217733317 GJ On-Demand Unstable HCN4 41 34 CCOc1ccccc1C(=O)N(CC(=O)Nc1cccc(C)c1C)[C@H](C)CC ZINC000217733317 GJ On-Demand Unstable KCNK3 27 40 CCOc1ccccc1C(=O)N(CC(=O)Nc1cccc(C)c1C)[C@H](C)CC ZINC000217733317 GJ On-Demand Unstable KCNK9 25 40 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccccc2OC)CC1 ZINC000217733339 FG For-Sale Unstable HTR1A 97 54 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccccc2OC)CC1 ZINC000217733339 FG For-Sale Unstable DRD2 73 54 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccccc2OC)CC1 ZINC000217733339 FG For-Sale Unstable DRD1 27 41 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccccc2OC)CC1 ZINC000217733339 FG For-Sale Unstable DRD4 40 49 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccccc2OC)CC1 ZINC000217733339 FG For-Sale Unstable ADRA1D 73 41 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccccc2OC)CC1 ZINC000217733339 FG For-Sale Unstable HTR1D 23 45 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccccc2OC)CC1 ZINC000217733339 FG For-Sale Unstable HTR1B 20 54 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccccc2OC)CC1 ZINC000217733339 FG For-Sale Unstable HTR2A 36 45 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccccc2OC)CC1 ZINC000217733339 FG For-Sale Unstable ADRA1A 66 41 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccccc2OC)CC1 ZINC000217733339 FG For-Sale Unstable ADRA1B 59 41 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccccc2OC)CC1 ZINC000217733339 FG For-Sale Unstable DRD3 77 54 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccccc2OC)CC1 ZINC000217733339 FG For-Sale Unstable HTR7 61 46 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccccc2OC)CC1 ZINC000217733339 FG For-Sale Unstable TACR3 24 46 CCOc1ccccc1NC(=O)COc1c(OC)cc(C(=O)O)cc1OC ZINC000217733341 GF In-Stock Unstable EPHX1 0 42 CCOc1ccccc1NC(=O)COc1c(OC)cc(C(=O)O)cc1OC ZINC000217733341 GF In-Stock Unstable LTB4R 16 44 CCOc1ccccc1NC(=O)COc1c(OC)cc(C(=O)O)cc1OC ZINC000217733341 GF In-Stock Unstable KCNK3 45 44 CCOc1ccccc1NC(=O)COc1c(OC)cc(C(=O)O)cc1OC ZINC000217733341 GF In-Stock Unstable KCNK9 34 44 COc1cccc(OCC(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217733342 EE For-Sale Unstable CHRNA10 35 44 Cc1ncccc1NC(=O)c1cc(Br)ccc1I ZINC000217733349 HI On-Demand Unstable G2YM83_BOTF4 70 36 O=C(O)/C=C\c1cnc(NC(=O)c2ccc(Cl)c(Cl)c2)s1 ZINC000217733368 EH For-Sale Anodyne KMO 0 46 O=C(O)/C=C\c1cnc(NC(=O)c2ccc(Cl)c(Cl)c2)s1 ZINC000217733368 EH For-Sale Anodyne SCD1 35 42 O=C(O)/C=C\c1cnc(NC(=O)c2ccc(Cl)c(Cl)c2)s1 ZINC000217733368 EH For-Sale Anodyne SCD 27 42 CCc1ccc(C(=O)Nc2ncc(/C=C\C(=O)O)s2)cc1 ZINC000217733441 DG For-Sale Unstable CDK5 22 40 CCOc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733443 GF In-Stock Unstable TSHR 54 32 CCOc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733443 GF In-Stock Unstable ADORA2B 43 38 CCOc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733443 GF In-Stock Unstable CETP 0 40 CCOc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733443 GF In-Stock Unstable PRNP 15 51 CCOc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733443 GF In-Stock Unstable MTNR1A 20 42 CCOc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733443 GF In-Stock Unstable MTNR1B 25 43 CCOc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733443 GF In-Stock Unstable PLA2G4B 49 44 CCOc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733443 GF In-Stock Unstable PDGFRA 53 37 CCOc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733443 GF In-Stock Unstable HIF1A 20 40 CCOc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217733443 GF In-Stock Unstable ENPP1 49 30 CC(C)Cc1cc(C(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)n(C)n1 ZINC000217733505 FE In-Stock Unstable CHRNA4 29 48 COC(=O)[C@H](O)CNC(=O)c1c(F)cccc1Cl ZINC000217733554 CC For-Sale Unstable PPIA 24 43 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217733560 HI In-Stock Unstable EPHX1 0 46 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217733560 HI In-Stock Unstable TSHR 56 34 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217733560 HI In-Stock Unstable SRD5A2 30 41 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217733560 HI In-Stock Unstable PDGFRB 66 46 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217733560 HI In-Stock Unstable LTA4H 62 49 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217733560 HI In-Stock Unstable CETP 0 42 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217733560 HI In-Stock Unstable CPT1A 45 32 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217733560 HI In-Stock Unstable GUAB 0 42 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217733560 HI In-Stock Unstable HDAC8 19 41 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217733560 HI In-Stock Unstable PRNP 21 42 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217733560 HI In-Stock Unstable RAF1 42 43 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217733560 HI In-Stock Unstable KDR 50 46 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217733560 HI In-Stock Unstable MTNR1A 25 56 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217733560 HI In-Stock Unstable MTNR1B 35 56 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217733560 HI In-Stock Unstable FAAH 17 41 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217733560 HI In-Stock Unstable NPY5R 26 43 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217733560 HI In-Stock Unstable MAP2K1 0 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217733560 HI In-Stock Unstable MET 26 47 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217733560 HI In-Stock Unstable FLT4 33 45 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217733560 HI In-Stock Unstable PDGFRA 62 46 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217733560 HI In-Stock Unstable FLT3 20 45 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217733560 HI In-Stock Unstable CSF1R 21 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217733560 HI In-Stock Unstable MCHR1 31 51 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217733560 HI In-Stock Unstable Q8MMZ8_EIMTE 60 43 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217733560 HI In-Stock Unstable AKR1C3 26 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217733560 HI In-Stock Unstable AKR1C2 45 36 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217733560 HI In-Stock Unstable ENPP1 56 33 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217733560 HI In-Stock Unstable PFKFB3 47 36 O=c1cc(Cl)nc(-c2ccncc2)[nH]1 ZINC000217733584 BD In-Stock Anodyne GCGR 23 45 O=c1cc(Cl)nc(-c2ccncc2)[nH]1 ZINC000217733584 BD In-Stock Anodyne RAF1 28 43 O=c1cc(Cl)nc(-c2ccncc2)[nH]1 ZINC000217733584 BD In-Stock Anodyne BRAF 22 40 COC(C)(C)C(=O)Nc1cccnc1C ZINC000217733601 BD On-Demand Unstable MAP1 15 41 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)c(OC)c1 ZINC000217733682 GE In-Stock Unstable CYP1B1 27 53 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)c(OC)c1 ZINC000217733682 GE In-Stock Unstable LTB4R 21 40 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)c(OC)c1 ZINC000217733682 GE In-Stock Unstable MTNR1A 52 33 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)c(OC)c1 ZINC000217733682 GE In-Stock Unstable MTNR1B 45 38 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)c(OC)c1 ZINC000217733682 GE In-Stock Unstable PLA2G4B 30 40 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)c(OC)c1 ZINC000217733682 GE In-Stock Unstable AKR1C3 35 40 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)c(OC)c1 ZINC000217733682 GE In-Stock Unstable AKR1C2 53 40 O=c1cc(Cl)nc(-c2cccnc2)[nH]1 ZINC000217733697 BD In-Stock Anodyne CYP11B2 26 40 COc1ccc(C(=O)Nc2cccnc2C)c(F)c1 ZINC000217733727 CF On-Demand Unstable PYGL 23 40 COc1ccc(C(=O)Nc2cccnc2C)c(F)c1 ZINC000217733727 CF On-Demand Unstable KDR 42 35 COc1ccc(C(=O)Nc2cccnc2C)c(F)c1 ZINC000217733727 CF On-Demand Unstable PYGM 23 40 COc1ccc(C(=O)Nc2cccnc2C)c(F)c1 ZINC000217733727 CF On-Demand Unstable AKR1C2 52 37 COc1ccc(C(=O)Nc2cccnc2C)c(F)c1 ZINC000217733727 CF On-Demand Unstable GPR35 29 46 COc1ccc(C(=O)Nc2cccnc2C)c(F)c1 ZINC000217733727 CF On-Demand Unstable G2YM83_BOTF4 66 34 O=C(O)/C=C\c1cccc(NC(=O)C2CCCCC2)c1 ZINC000217733731 CG For-Sale Unstable HDAC8 15 40 O=C(O)/C=C\c1cccc(NC(=O)C2CCCCC2)c1 ZINC000217733731 CG For-Sale Unstable NR1H4 24 40 O=C(O)/C=C\c1cccc(NC(=O)C2CCCCC2)c1 ZINC000217733731 CG For-Sale Unstable TYK2 48 38 O=C(O)/C=C\c1cccc(NC(=O)C2CCCCC2)c1 ZINC000217733731 CG For-Sale Unstable KCNK3 19 59 COc1ccccc1/C=C/NC(=O)NC1CCCCCC1 ZINC000217733735 CH For-Sale Unstable FAAH 16 41 COc1ccccc1/C=C/NC(=O)NC1CCCCCC1 ZINC000217733735 CH For-Sale Unstable EPHX2 28 46 COc1ccc(C)cc1NC(=O)COc1c(OC)cc(C(=O)O)cc1OC ZINC000217733796 GF In-Stock Unstable LTB4R 17 48 O=c1[nH]c(-c2ccccc2)nc(Cl)c1Br ZINC000217733822 CF In-Stock Anodyne TNKS 41 46 O=c1[nH]c(-c2ccccc2)nc(Cl)c1Br ZINC000217733822 CF In-Stock Anodyne TNKS2 33 46 COc1ccccc1/C=C/NC(=O)Nc1cc(C)ccc1C ZINC000217733840 CI For-Sale Unstable EPHX1 0 40 COc1ccccc1/C=C/NC(=O)Nc1cc(C)ccc1C ZINC000217733840 CI For-Sale Unstable KCNK3 37 40 COc1ccccc1/C=C/NC(=O)Nc1cc(C)ccc1C ZINC000217733840 CI For-Sale Unstable KCNK9 41 40 Cc1ncccc1NC(=O)c1cc(F)cc([N+](=O)[O-])c1N ZINC000217733847 CE On-Demand Unstable G2YM83_BOTF4 50 32 Cc1ccccc1/C=C\C(=O)Nc1cnccc1C(=O)O ZINC000217733855 CF For-Sale Unstable LTB4R 19 44 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1Cl ZINC000217733905 GG In-Stock Unstable HTR2A 17 44 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1Cl ZINC000217733905 GG In-Stock Unstable COLA 62 41 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1Cl ZINC000217733905 GG In-Stock Unstable CPT1A 60 41 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1Cl ZINC000217733905 GG In-Stock Unstable CPT2 47 38 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1Cl ZINC000217733905 GG In-Stock Unstable GRM4 18 50 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1Cl ZINC000217733905 GG In-Stock Unstable PDE6A 44 35 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1Cl ZINC000217733905 GG In-Stock Unstable CPT1B 44 38 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1Cl ZINC000217733905 GG In-Stock Unstable MCHR1 21 44 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1Cl ZINC000217733905 GG In-Stock Unstable MCHR2 41 44 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1Cl ZINC000217733905 GG In-Stock Unstable ENPP1 74 38 COc1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1Cl ZINC000217733905 GG In-Stock Unstable SMO 20 42 COc1ccccc1/C=C/NC(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000217733940 EJ For-Sale Unstable PDGFRA 16 40 COc1ccccc1/C=C/NC(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000217733940 EJ For-Sale Unstable CYSP_PLAFA 43 35 CCCCCNC[C@@H](O)CCC ZINC000217733942 AD For-Sale Unstable Q8WS26_TRYCR 43 48 CCCCCNC[C@@H](O)CCC ZINC000217733942 AD For-Sale Unstable FPPS 0 50 CCCCCNC[C@@H](O)CCC ZINC000217733942 AD For-Sale Unstable SPPS 0 48 CCCCCNC[C@@H](O)CCC ZINC000217733942 AD For-Sale Unstable CQSS 41 35 O=C(OCCC1CC1)c1cc([N+](=O)[O-])ccc1F ZINC000217733966 CF On-Demand Unstable CACNA1C 47 38 O=C(OCCC1CC1)c1cc([N+](=O)[O-])ccc1F ZINC000217733966 CF On-Demand Unstable CACNA1D 72 38 O=C(OCCC1CC1)c1cc([N+](=O)[O-])ccc1F ZINC000217733966 CF On-Demand Unstable SLC27A4 52 35 CN(C)CCCNC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217734009 GD In-Stock Unstable EDNRA 25 40 CN(C)CCCNC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217734009 GD In-Stock Unstable MC4R 52 37 CN(C)CCCNC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217734009 GD In-Stock Unstable TACR2 0 44 CN(C)CCCNC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217734009 GD In-Stock Unstable CCKAR 42 36 CN(C)CCCNC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217734009 GD In-Stock Unstable BRS3 21 41 CN(C)CCCNC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217734009 GD In-Stock Unstable MC3R 40 31 CN(C)CCCNC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217734009 GD In-Stock Unstable GRIA1 20 46 CN(C)CCCNC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217734009 GD In-Stock Unstable MC1R 42 35 CN(C)CCCNC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217734009 GD In-Stock Unstable MMP1 15 45 COC(=O)c1ccccc1NC(=O)COc1c(OC)cc(C(=O)O)cc1OC ZINC000217734013 GE In-Stock Unstable LTB4R 17 44 COC(=O)c1ccccc1NC(=O)COc1c(OC)cc(C(=O)O)cc1OC ZINC000217734013 GE In-Stock Unstable NR1H4 0 45 COC(=O)c1ccccc1NC(=O)COc1c(OC)cc(C(=O)O)cc1OC ZINC000217734013 GE In-Stock Unstable PTK2 21 41 COC(=O)c1ccccc1NC(=O)COc1c(OC)cc(C(=O)O)cc1OC ZINC000217734013 GE In-Stock Unstable HCAR2 36 42 COC(=O)c1ccccc1NC(=O)COc1c(OC)cc(C(=O)O)cc1OC ZINC000217734013 GE In-Stock Unstable KCNK3 43 36 COC(=O)c1ccccc1NC(=O)COc1c(OC)cc(C(=O)O)cc1OC ZINC000217734013 GE In-Stock Unstable FAS 52 51 CCCCCNC[C@H](O)CCC ZINC000217734028 AD For-Sale Unstable Q8WS26_TRYCR 43 48 CCCCCNC[C@H](O)CCC ZINC000217734028 AD For-Sale Unstable FPPS 0 50 CCCCCNC[C@H](O)CCC ZINC000217734028 AD For-Sale Unstable SPPS 0 48 CCCCCNC[C@H](O)CCC ZINC000217734028 AD For-Sale Unstable CQSS 41 35 COc1ccccc1-c1cc(C(=O)N2CC(N3C(=O)[C@H]4CC=CC[C@H]4C3=O)C2)[nH]n1 ZINC000217734029 HD In-Stock Unstable TACR3 20 44 CCOc1ccccc1NC(=O)N/C=C/c1ccccc1OC ZINC000217734050 DH For-Sale Unstable KCNK3 37 42 CCOc1ccccc1NC(=O)N/C=C/c1ccccc1OC ZINC000217734050 DH For-Sale Unstable KCNK9 28 42 COc1ccccc1-c1cc(C(=O)N2CC(N3C(=O)[C@H]4CC=CC[C@@H]4C3=O)C2)[nH]n1 ZINC000217734105 HD In-Stock Unstable TACR3 20 44 COC(=O)c1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217734115 GE In-Stock Unstable CYSLTR1 23 40 COC(=O)c1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217734115 GE In-Stock Unstable COLA 39 40 COC(=O)c1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217734115 GE In-Stock Unstable CPT1A 45 31 COC(=O)c1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217734115 GE In-Stock Unstable ACR 58 39 COC(=O)c1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217734115 GE In-Stock Unstable PDGFRA 55 36 COC(=O)c1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217734115 GE In-Stock Unstable ENPP1 50 31 COC(=O)c1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217734115 GE In-Stock Unstable DRTS_TRYCR 29 40 O=C(/C=C\c1ccccc1F)Nc1cnccc1C(=O)O ZINC000217734149 CF For-Sale Anodyne KCNQ2 44 44 CC(C)(C)C(=O)C[C@H]1SC(=O)NC1=O ZINC000217734153 BD For-Sale Unstable FFAR1 65 46 CC(C)(C)C(=O)C[C@H]1SC(=O)NC1=O ZINC000217734153 BD For-Sale Unstable CISD1 0 46 COc1ccccc1/C=C/NC(=O)Nc1cc(C)cc(C)c1 ZINC000217734169 CI For-Sale Unstable KCNK9 42 39 COc1ccc(Cl)cc1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217734196 FG For-Sale Unstable DRD2 39 41 COc1ccc(Cl)cc1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217734196 FG For-Sale Unstable DRD3 21 47 COc1ccc(Cl)cc1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217734196 FG For-Sale Unstable HTR4 30 40 COc1ccc(Cl)cc1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217734196 FG For-Sale Unstable F10 50 33 COc1ccc(Cl)cc1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217734196 FG For-Sale Unstable CACNA1I 41 32 COc1ccc(Cl)cc1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217734196 FG For-Sale Unstable ACKR3 62 31 COc1ccccc1-c1cc(C(=O)N2CC(N3C(=O)[C@@H]4CC=CC[C@H]4C3=O)C2)[nH]n1 ZINC000217734208 HD In-Stock Unstable TACR3 20 44 CC(C)(C)C(=O)C[C@@H]1SC(=O)NC1=O ZINC000217734226 BD For-Sale Unstable FFAR1 65 46 CC(C)(C)C(=O)C[C@@H]1SC(=O)NC1=O ZINC000217734226 BD For-Sale Unstable CISD1 0 46 Cc1cc(NC(=O)c2cccn2C)ccc1/C=C\C(=O)O ZINC000217734230 CF For-Sale Unstable KCNK3 67 36 COc1ccc(F)c(F)c1C(=O)NCc1nc2cc(F)ccc2[nH]1 ZINC000217734234 EF In-Stock Unstable FABK 0 43 CCOC(=O)c1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217734239 HF In-Stock Unstable CYSLTR1 23 40 CCOC(=O)c1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217734239 HF In-Stock Unstable PDGFRB 32 49 CCOC(=O)c1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217734239 HF In-Stock Unstable ADORA2B 21 42 CCOC(=O)c1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217734239 HF In-Stock Unstable CPT1A 42 29 CCOC(=O)c1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217734239 HF In-Stock Unstable CA14 0 40 CCOC(=O)c1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217734239 HF In-Stock Unstable ACR 70 42 CCOC(=O)c1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217734239 HF In-Stock Unstable PDGFRA 41 34 CCOC(=O)c1ccc(NC(=O)COc2c(OC)cc(C(=O)O)cc2OC)cc1 ZINC000217734239 HF In-Stock Unstable ENPP1 51 32 CC[C@@H](C)N(CC(=O)Nc1cccc(C)c1C)C(=O)c1cccc(C)c1 ZINC000217734241 FI On-Demand Unstable KCNK3 52 37 COc1ccc(OCCNC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217734275 EG For-Sale Unstable HRH2 18 40 COc1ccc(OCCNC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217734275 EG For-Sale Unstable CYP1B1 33 44 COc1ccc(OCCNC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217734275 EG For-Sale Unstable MTNR1A 49 46 COc1ccc(OCCNC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217734275 EG For-Sale Unstable MTNR1B 44 46 COc1ccc(Cl)cc1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217734287 FG For-Sale Unstable DRD2 39 41 COc1ccc(Cl)cc1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217734287 FG For-Sale Unstable DRD3 21 47 COc1ccc(Cl)cc1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217734287 FG For-Sale Unstable HTR4 30 40 COc1ccc(Cl)cc1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217734287 FG For-Sale Unstable F10 50 33 COc1ccc(Cl)cc1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217734287 FG For-Sale Unstable CACNA1I 41 32 COc1ccc(Cl)cc1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217734287 FG For-Sale Unstable ACKR3 62 31 COC(=O)[C@@H](O)CNC(=O)/C=C/c1ccc([N+](=O)[O-])cc1 ZINC000217734302 CC On-Demand Unstable HDAC8 16 52 Cc1cc(NC(=O)c2ccc[nH]2)ccc1/C=C\C(=O)O ZINC000217734309 CF For-Sale Unstable KCNK3 86 39 CC[C@H](C)N(CC(=O)Nc1cccc(C)c1C)C(=O)c1cccc(C)c1 ZINC000217734324 FI On-Demand Unstable KCNK3 52 37 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217734343 HD In-Stock Unstable CA2 151 52 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217734343 HD In-Stock Unstable CA6 20 42 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217734343 HD In-Stock Unstable CA1 136 52 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217734343 HD In-Stock Unstable CA7 75 51 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217734343 HD In-Stock Unstable CPT1A 45 31 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217734343 HD In-Stock Unstable CA13 25 41 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217734343 HD In-Stock Unstable CA5B 62 48 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217734343 HD In-Stock Unstable CA4 124 49 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217734343 HD In-Stock Unstable CA5A 71 48 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217734343 HD In-Stock Unstable CA14 57 51 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217734343 HD In-Stock Unstable CA12 86 52 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217734343 HD In-Stock Unstable CA9 93 52 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217734343 HD In-Stock Unstable UREA_CANEN 29 45 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217734343 HD In-Stock Unstable CYNT 43 44 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217734343 HD In-Stock Unstable NCE103 37 42 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217734343 HD In-Stock Unstable ENPP1 50 31 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217734343 HD In-Stock Unstable MTCA1 53 48 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217734343 HD In-Stock Unstable P96878_MYCTU 68 48 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000217734343 HD In-Stock Unstable CA 0 42 O=C(NC[C@@H]1CCCN1c1nccs1)c1cc(-c2ccccc2)on1 ZINC000217734403 FG For-Sale Unstable HDAC10 16 42 Cc1c[nH]c(C(=O)N2CCC(N3CCC(O)CC3)CC2)n1 ZINC000217734426 CC In-Stock Unstable L3MBTL1 0 44 Cc1c[nH]c(C(=O)N2CCC(N3CCC(O)CC3)CC2)n1 ZINC000217734426 CC In-Stock Unstable L3MBTL3 77 44 Cc1c[nH]c(C(=O)N2CCC(N3CCC(O)CC3)CC2)n1 ZINC000217734426 CC In-Stock Unstable MBTD1 0 40 Cc1c[nH]c(C(=O)N2CCC(N3CCC(O)CC3)CC2)n1 ZINC000217734426 CC In-Stock Unstable TP53BP1 0 40 Cc1c(F)cccc1NC(=O)c1ccc(F)c(Br)c1 ZINC000217734439 EI On-Demand Unstable NR1H4 0 41 Cc1c(F)cccc1NC(=O)c1ccc(F)c(Br)c1 ZINC000217734439 EI On-Demand Unstable FABH 0 42 Cc1c(F)cccc1NC(=O)c1ccc(F)c(Br)c1 ZINC000217734439 EI On-Demand Unstable TAAR1 29 57 Cc1c(F)cccc1NC(=O)c1ccc(F)c(Br)c1 ZINC000217734439 EI On-Demand Unstable KCNK3 67 40 COc1cc(C(=O)O)cc(OC)c1OCC(=O)Nc1cccc(C(C)=O)c1 ZINC000217734443 FF In-Stock Unstable PARP10 0 43 COCCCNC(=O)[C@H](CC(C)C)Nc1ccc2c(cc1=O)[C@@H](NC(C)=O)CCc1cc(OC)c(OC)c(OC)c1-2 ZINC000217734451 KH In-Stock Unstable TUBA1A 18 66 COCCCNC(=O)[C@H](CC(C)C)Nc1ccc2c(cc1=O)[C@@H](NC(C)=O)CCc1cc(OC)c(OC)c(OC)c1-2 ZINC000217734451 KH In-Stock Unstable TPPP 0 63 CCCCCNC(=O)[C@@H](C)N1CCO[C@@H](CN)C1 ZINC000217734482 CC On-Demand Unstable NOD1 53 37 O=C(NC[C@H]1CCCN1c1nccs1)c1cc(-c2ccccc2)on1 ZINC000217734501 FG For-Sale Unstable HDAC10 16 42 COc1ccccc1/C=C/NC(=O)NCCNC(C)=O ZINC000217734516 CD For-Sale Unstable DRD3 15 41 COc1ccccc1/C=C/NC(=O)NCCNC(C)=O ZINC000217734516 CD For-Sale Unstable CYP1B1 17 41 COc1ccccc1/C=C/NC(=O)NCCNC(C)=O ZINC000217734516 CD For-Sale Unstable NQO2 46 32 COc1ccccc1/C=C/NC(=O)NCCNC(C)=O ZINC000217734516 CD For-Sale Unstable MTNR1A 67 49 COc1ccccc1/C=C/NC(=O)NCCNC(C)=O ZINC000217734516 CD For-Sale Unstable MTNR1B 64 49 COc1ccccc1/C=C/NC(=O)NCCNC(C)=O ZINC000217734516 CD For-Sale Unstable CYP1A1 15 41 COc1ccccc1/C=C/NC(=O)NCCNC(C)=O ZINC000217734516 CD For-Sale Unstable TLR4 15 44 Cc1c(F)cccc1NC(=O)c1cc(Br)ccc1I ZINC000217734550 IJ On-Demand Unstable PYK 48 35 CCCCCNC(=O)[C@H](C)N1CCO[C@@H](CN)C1 ZINC000217734581 CC On-Demand Unstable NOD1 53 37 O=C(NC[C@@H]1CCCN1c1nccs1)c1cccc(C(F)(F)F)c1 ZINC000217734625 FH For-Sale Unstable CCR2 73 48 O=C(NC[C@@H]1CCCN1c1nccs1)c1cccc(C(F)(F)F)c1 ZINC000217734625 FH For-Sale Unstable CACNA1I 18 41 COC(=O)c1ccccc1NC(=O)COc1ccc(C(=O)O)cc1[N+](=O)[O-] ZINC000217734643 FE In-Stock Unstable AKR1C2 33 44 COC(=O)c1ccccc1NC(=O)COc1ccc(C(=O)O)cc1[N+](=O)[O-] ZINC000217734643 FE In-Stock Unstable FAS 46 45 O=C(NC[C@H]1CCCN1c1nccs1)c1cccc(C(F)(F)F)c1 ZINC000217734711 FH For-Sale Unstable CCR2 73 48 O=C(NC[C@H]1CCCN1c1nccs1)c1cccc(C(F)(F)F)c1 ZINC000217734711 FH For-Sale Unstable CACNA1I 18 41 COc1ccccc1/C=C/NC(=O)NC12CC3CC(CC(C3)C1)C2 ZINC000217734754 EH For-Sale Unstable CNR2 15 47 COc1ccccc1/C=C/NC(=O)NC12CC3CC(CC(C3)C1)C2 ZINC000217734754 EH For-Sale Unstable EPHX2 110 50 COC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2[N+](=O)[O-])cc1 ZINC000217734763 FE In-Stock Unstable CETP 25 40 COC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2[N+](=O)[O-])cc1 ZINC000217734763 FE In-Stock Unstable ACR 48 35 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCCC(=O)NCc3cccnc3)[C@H]21 ZINC000217734771 JG In-Stock Unstable HTR7 25 47 CC[C@@H](C)N(C)CCNCc1c[nH]c2ccccc12 ZINC000217734820 CF For-Sale Unstable HTR1D 18 40 CC[C@@H](C)N(C)CCNCc1c[nH]c2ccccc12 ZINC000217734820 CF For-Sale Unstable CTSL 22 40 CC[C@@H](C)N(C)CCNCc1c[nH]c2ccccc12 ZINC000217734820 CF For-Sale Unstable MPO 30 40 CC[C@@H](C)N(C)CCNCc1c[nH]c2ccccc12 ZINC000217734820 CF For-Sale Unstable MMP1 15 40 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCCC(=O)NCc3cccnc3)[C@@H]21 ZINC000217734857 JG In-Stock Unstable HTR7 25 47 CCOC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2[N+](=O)[O-])cc1 ZINC000217734877 GE In-Stock Unstable CETP 26 42 CCOC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2[N+](=O)[O-])cc1 ZINC000217734877 GE In-Stock Unstable PLA2G4B 27 52 CCOC(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2[N+](=O)[O-])cc1 ZINC000217734877 GE In-Stock Unstable ACR 56 32 CC[C@H](C)N(C)CCNCc1c[nH]c2ccccc12 ZINC000217734916 CF For-Sale Unstable HTR1D 18 40 CC[C@H](C)N(C)CCNCc1c[nH]c2ccccc12 ZINC000217734916 CF For-Sale Unstable CTSL 22 40 CC[C@H](C)N(C)CCNCc1c[nH]c2ccccc12 ZINC000217734916 CF For-Sale Unstable MPO 30 40 CC[C@H](C)N(C)CCNCc1c[nH]c2ccccc12 ZINC000217734916 CF For-Sale Unstable MMP1 15 40 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2[N+](=O)[O-])cc1 ZINC000217734992 GC In-Stock Unstable CA2 105 47 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2[N+](=O)[O-])cc1 ZINC000217734992 GC In-Stock Unstable CA1 88 47 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2[N+](=O)[O-])cc1 ZINC000217734992 GC In-Stock Unstable CA7 40 44 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2[N+](=O)[O-])cc1 ZINC000217734992 GC In-Stock Unstable CA5B 40 44 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2[N+](=O)[O-])cc1 ZINC000217734992 GC In-Stock Unstable CA4 89 47 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2[N+](=O)[O-])cc1 ZINC000217734992 GC In-Stock Unstable CA5A 46 44 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2[N+](=O)[O-])cc1 ZINC000217734992 GC In-Stock Unstable CA12 55 45 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2[N+](=O)[O-])cc1 ZINC000217734992 GC In-Stock Unstable CA9 57 45 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2[N+](=O)[O-])cc1 ZINC000217734992 GC In-Stock Unstable UREA_CANEN 26 40 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2[N+](=O)[O-])cc1 ZINC000217734992 GC In-Stock Unstable CYNT 35 41 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2[N+](=O)[O-])cc1 ZINC000217734992 GC In-Stock Unstable NCE103 19 42 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2[N+](=O)[O-])cc1 ZINC000217734992 GC In-Stock Unstable MTCA1 47 42 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2[N+](=O)[O-])cc1 ZINC000217734992 GC In-Stock Unstable P96878_MYCTU 61 42 NS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(=O)O)cc2[N+](=O)[O-])cc1 ZINC000217734992 GC In-Stock Unstable SCMU_MYCTU 0 41 COc1ccc(C(=O)Nc2cccc(F)c2C)c(F)c1 ZINC000217735011 CH On-Demand Unstable DRD4 40 31 COc1ccc(C(=O)Nc2cccc(F)c2C)c(F)c1 ZINC000217735011 CH On-Demand Unstable DHODH 15 45 COc1ccc(C(=O)Nc2cccc(F)c2C)c(F)c1 ZINC000217735011 CH On-Demand Unstable PYGM 16 41 COc1ccc(C(=O)Nc2cccc(F)c2C)c(F)c1 ZINC000217735011 CH On-Demand Unstable LUCI_LUCLA 16 41 COc1ccc(C(=O)Nc2cccc(F)c2C)c(F)c1 ZINC000217735011 CH On-Demand Unstable TAAR1 17 41 COc1ccc(C(=O)Nc2cccc(F)c2C)c(F)c1 ZINC000217735011 CH On-Demand Unstable AKR1C3 27 42 COc1ccc(C(=O)Nc2cccc(F)c2C)c(F)c1 ZINC000217735011 CH On-Demand Unstable AKR1C2 60 42 COc1ccc(C(=O)Nc2cccc(F)c2C)c(F)c1 ZINC000217735011 CH On-Demand Unstable GPR35 47 48 COc1ccc(C(=O)Nc2cccc(F)c2C)c(F)c1 ZINC000217735011 CH On-Demand Unstable KCNK9 40 36 COC(=O)[C@@H](O)CNC(=O)/C=C/c1ccccc1OC ZINC000217735016 CC On-Demand Unstable DRD3 15 49 O=C(NC[C@@H]1CCCN1c1nccs1)c1cc(=O)c2ccccc2o1 ZINC000217735025 FF For-Sale Unstable BCHE 26 40 CCCCC(=O)N[C@@H](C)c1cccc(/C=C\C(=O)O)c1 ZINC000217735045 CG For-Sale Unstable SOAT1 24 43 CCCCC(=O)N[C@@H](C)c1cccc(/C=C\C(=O)O)c1 ZINC000217735045 CG For-Sale Unstable AKR1C3 28 42 CCCCC(=O)N[C@@H](C)c1cccc(/C=C\C(=O)O)c1 ZINC000217735045 CG For-Sale Unstable NOD1 75 37 CCCCC(=O)N[C@@H](C)c1cccc(/C=C\C(=O)O)c1 ZINC000217735045 CG For-Sale Unstable ACER2 0 46 CCCCC(=O)N[C@@H](C)c1cccc(/C=C\C(=O)O)c1 ZINC000217735045 CG For-Sale Unstable COL4A3BP 0 40 COc1ccccc1/C=C/NC(=O)N1c2ccccc2C[C@@H]1C ZINC000217735080 DH For-Sale Unstable DRD2 19 48 COc1ccccc1/C=C/NC(=O)N1c2ccccc2C[C@@H]1C ZINC000217735080 DH For-Sale Unstable DRD4 31 42 COc1ccccc1/C=C/NC(=O)N1c2ccccc2C[C@@H]1C ZINC000217735080 DH For-Sale Unstable DRD3 21 40 COC(=O)[C@H](O)CNC(=O)/C=C/c1ccccc1OC ZINC000217735093 CC For-Sale Unstable DRD3 15 49 CC(C)NC(=O)COc1c(Br)cc(C(=O)O)cc1Br ZINC000217735099 GF In-Stock Unstable THRB 29 45 CC(C)NC(=O)COc1c(Br)cc(C(=O)O)cc1Br ZINC000217735099 GF In-Stock Unstable TPMT 0 45 CCCCC(=O)N[C@H](C)c1cccc(/C=C\C(=O)O)c1 ZINC000217735117 CG For-Sale Unstable SOAT1 24 43 CCCCC(=O)N[C@H](C)c1cccc(/C=C\C(=O)O)c1 ZINC000217735117 CG For-Sale Unstable AKR1C3 28 42 CCCCC(=O)N[C@H](C)c1cccc(/C=C\C(=O)O)c1 ZINC000217735117 CG For-Sale Unstable NOD1 75 37 CCCCC(=O)N[C@H](C)c1cccc(/C=C\C(=O)O)c1 ZINC000217735117 CG For-Sale Unstable ACER2 0 46 CCCCC(=O)N[C@H](C)c1cccc(/C=C\C(=O)O)c1 ZINC000217735117 CG For-Sale Unstable COL4A3BP 0 40 O=C(NC[C@H]1CCCN1c1nccs1)c1cc(=O)c2ccccc2o1 ZINC000217735120 FF For-Sale Unstable BCHE 26 40 Nc1cc(C(=O)OCCC2CC2)cc(C(F)(F)F)c1 ZINC000217735157 CG For-Sale Unstable LIPG 26 42 COc1ccccc1/C=C/NC(=O)N1c2ccccc2C[C@H]1C ZINC000217735164 DH For-Sale Unstable DRD2 19 48 COc1ccccc1/C=C/NC(=O)N1c2ccccc2C[C@H]1C ZINC000217735164 DH For-Sale Unstable DRD4 31 42 COc1ccccc1/C=C/NC(=O)N1c2ccccc2C[C@H]1C ZINC000217735164 DH For-Sale Unstable DRD3 21 40 CC[C@@H](C)NC(=O)COc1c(Br)cc(C(=O)O)cc1Br ZINC000217735206 HG In-Stock Unstable THRA 28 41 CC[C@@H](C)NC(=O)COc1c(Br)cc(C(=O)O)cc1Br ZINC000217735206 HG In-Stock Unstable THRB 23 43 CC[C@@H](C)NC(=O)COc1c(Br)cc(C(=O)O)cc1Br ZINC000217735206 HG In-Stock Unstable TPMT 0 43 Cn1cc(S(=O)(=O)N[C@@H]2CCN3CCC[C@@H]23)cc1C(=O)O ZINC000217735210 DC For-Sale Unstable SFRP1 76 33 Cn1cc(S(=O)(=O)N[C@@H]2CCN3CCC[C@@H]23)cc1C(=O)O ZINC000217735210 DC For-Sale Unstable WNT3 60 33 COC(=O)[C@@H](O)CNC(=O)CCOc1cccc(Br)c1 ZINC000217735224 EC On-Demand Unstable MTNR1A 24 41 COC(=O)[C@@H](O)CNC(=O)CCOc1cccc(Br)c1 ZINC000217735224 EC On-Demand Unstable MTNR1B 20 41 COC(=O)[C@@H](O)CNC(=O)CCOc1cccc(Br)c1 ZINC000217735224 EC On-Demand Unstable PDS 30 42 CC[C@@H](C)N(CC(=O)Nc1cccc(C)c1C)C(=O)Cc1cccc(F)c1 ZINC000217735235 FI On-Demand Unstable KCNQ2 19 42 Cn1cc(S(=O)(=O)N[C@H]2CCN3CCC[C@@H]23)cc1C(=O)O ZINC000217735274 DC For-Sale Unstable SFRP1 76 33 Cn1cc(S(=O)(=O)N[C@H]2CCN3CCC[C@@H]23)cc1C(=O)O ZINC000217735274 DC For-Sale Unstable WNT3 60 33 COc1ccccc1/C=C/NC(=O)NC1CC1 ZINC000217735292 BE For-Sale Unstable TLR4 15 44 O=C(O)c1cc(S(=O)(=O)N2CCCC2)c(Cl)cc1O ZINC000217735298 DD For-Sale Unstable EPHX2 20 40 O=C(O)c1cc(S(=O)(=O)N2CCCC2)c(Cl)cc1O ZINC000217735298 DD For-Sale Unstable AKR1C2 40 35 CC[C@H](C)N(CC(=O)Nc1cccc(C)c1C)C(=O)Cc1cccc(F)c1 ZINC000217735311 FI On-Demand Unstable KCNQ2 19 42 COC(=O)[C@H](O)CNC(=O)CCOc1cccc(Br)c1 ZINC000217735314 EC On-Demand Unstable MTNR1A 24 41 COC(=O)[C@H](O)CNC(=O)CCOc1cccc(Br)c1 ZINC000217735314 EC On-Demand Unstable MTNR1B 20 41 COC(=O)[C@H](O)CNC(=O)CCOc1cccc(Br)c1 ZINC000217735314 EC On-Demand Unstable PDS 30 42 O=C(/C=C\c1cccc(Br)c1)Nc1cnccc1C(=O)O ZINC000217735317 EG For-Sale Anodyne LTB4R 0 45 O=C(/C=C\c1cccc(Br)c1)Nc1cnccc1C(=O)O ZINC000217735317 EG For-Sale Anodyne HDAC8 45 41 O=C(/C=C\c1cccc(Br)c1)Nc1cnccc1C(=O)O ZINC000217735317 EG For-Sale Anodyne MMP2 0 43 O=C(/C=C\c1cccc(Br)c1)Nc1cnccc1C(=O)O ZINC000217735317 EG For-Sale Anodyne HDAC1 0 40 O=C(/C=C\c1cccc(Br)c1)Nc1cnccc1C(=O)O ZINC000217735317 EG For-Sale Anodyne HDAC6 33 41 O=C(/C=C\c1cccc(Br)c1)Nc1cnccc1C(=O)O ZINC000217735317 EG For-Sale Anodyne MMP9 0 43 O=C(/C=C\c1cccc(Br)c1)Nc1cnccc1C(=O)O ZINC000217735317 EG For-Sale Anodyne HPSE 36 44 O=C(/C=C\c1cccc(Br)c1)Nc1cnccc1C(=O)O ZINC000217735317 EG For-Sale Anodyne MMP1 22 43 CC[C@H](C)NC(=O)COc1c(Br)cc(C(=O)O)cc1Br ZINC000217735322 HG In-Stock Unstable THRA 28 41 CC[C@H](C)NC(=O)COc1c(Br)cc(C(=O)O)cc1Br ZINC000217735322 HG In-Stock Unstable THRB 23 43 CC[C@H](C)NC(=O)COc1c(Br)cc(C(=O)O)cc1Br ZINC000217735322 HG In-Stock Unstable TPMT 0 43 N#Cc1ccc(S(=O)(=O)Nc2ccccc2[N+](=O)[O-])cc1 ZINC000217735333 DE For-Sale Mild PRTN3 50 32 COC(=O)C[C@H]1c2cc3c(cc2Oc2nc4ccc(OC)cc4cc21)OCO3 ZINC000217735392 GH In-Stock Unstable EDNRB 62 40 COC(=O)C[C@H]1c2cc3c(cc2Oc2nc4ccc(OC)cc4cc21)OCO3 ZINC000217735392 GH In-Stock Unstable EDNRA 59 40 COC(=O)C[C@H]1c2cc3c(cc2Oc2nc4ccc(OC)cc4cc21)OCO3 ZINC000217735392 GH In-Stock Unstable BMP1 44 36 COc1ccccc1/C=C/NC(=O)NCc1ccccc1OC ZINC000217735398 DG For-Sale Unstable TACR1 0 41 COc1ccccc1/C=C/NC(=O)NCc1ccccc1OC ZINC000217735398 DG For-Sale Unstable TLR4 15 44 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1N[C@H](c1ccccc1)C1CC1 ZINC000217735401 CK For-Sale Unstable TRPM8 17 46 CC[C@@H](C)N(CC(=O)Nc1cccc(C)c1C)C(=O)CCc1ccc(OC)c(OC)c1 ZINC000217735427 IJ On-Demand Unstable P2RX7 0 44 O=C(COc1c(Br)cc(C(=O)O)cc1Br)NC1CCCCC1 ZINC000217735435 IH In-Stock Unstable THRA 16 44 O=C(COc1c(Br)cc(C(=O)O)cc1Br)NC1CCCCC1 ZINC000217735435 IH In-Stock Unstable THRB 19 44 O=C(COc1c(Br)cc(C(=O)O)cc1Br)NC1CCCCC1 ZINC000217735435 IH In-Stock Unstable FAAH 0 42 O=C(COc1c(Br)cc(C(=O)O)cc1Br)NC1CCCCC1 ZINC000217735435 IH In-Stock Unstable EPHX2 29 43 O=C(COc1c(Br)cc(C(=O)O)cc1Br)NC1CCCCC1 ZINC000217735435 IH In-Stock Unstable LUXN 0 46 O=C(COc1c(Br)cc(C(=O)O)cc1Br)NC1CCCCC1 ZINC000217735435 IH In-Stock Unstable ADIPOR1 0 41 O=C(COc1c(Br)cc(C(=O)O)cc1Br)NC1CCCCC1 ZINC000217735435 IH In-Stock Unstable ADIPOR2 0 41 COc1cccc2cc(C(=O)NC[C@@H]3CCCN3c3nccs3)oc12 ZINC000217735438 FG For-Sale Unstable DRD3 16 46 COc1cccc2cc(C(=O)NC[C@@H]3CCCN3c3nccs3)oc12 ZINC000217735438 FG For-Sale Unstable ACKR3 61 31 COC(=O)C[C@@H]1c2cc3c(cc2Oc2nc4ccc(OC)cc4cc21)OCO3 ZINC000217735471 GH In-Stock Unstable EDNRB 50 38 COC(=O)C[C@@H]1c2cc3c(cc2Oc2nc4ccc(OC)cc4cc21)OCO3 ZINC000217735471 GH In-Stock Unstable EDNRA 46 38 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1N[C@H](c1ccccc1)C1CC1 ZINC000217735482 CK For-Sale Unstable TRPM8 17 46 COc1ccccc1/C=C/NC(=O)N1CCN(c2ncccn2)CC1 ZINC000217735499 ED For-Sale Unstable HTR1A 27 41 COc1ccccc1/C=C/NC(=O)N1CCN(c2ncccn2)CC1 ZINC000217735499 ED For-Sale Unstable DRD2 20 41 COc1ccccc1/C=C/NC(=O)N1CCN(c2ncccn2)CC1 ZINC000217735499 ED For-Sale Unstable DRD4 17 41 COc1ccccc1/C=C/NC(=O)N1CCN(c2ncccn2)CC1 ZINC000217735499 ED For-Sale Unstable DRD3 24 40 COc1ccccc1/C=C/NC(=O)N1CCN(c2ncccn2)CC1 ZINC000217735499 ED For-Sale Unstable PDGFRB 48 39 COc1ccccc1/C=C/NC(=O)N1CCN(c2ncccn2)CC1 ZINC000217735499 ED For-Sale Unstable SLC6A7 0 45 CC[C@H](C)N(CC(=O)Nc1cccc(C)c1C)C(=O)CCc1ccc(OC)c(OC)c1 ZINC000217735513 IJ On-Demand Unstable P2RX7 0 44 COc1cccc2cc(C(=O)NC[C@H]3CCCN3c3nccs3)oc12 ZINC000217735515 FG For-Sale Unstable DRD3 16 46 COc1cccc2cc(C(=O)NC[C@H]3CCCN3c3nccs3)oc12 ZINC000217735515 FG For-Sale Unstable ACKR3 61 31 O=C(COc1c(Br)cc(C(=O)O)cc1Br)NCc1ccccc1 ZINC000217735545 IH In-Stock Unstable THRA 32 47 O=C(COc1c(Br)cc(C(=O)O)cc1Br)NCc1ccccc1 ZINC000217735545 IH In-Stock Unstable THRB 30 47 O=C(COc1c(Br)cc(C(=O)O)cc1Br)NCc1ccccc1 ZINC000217735545 IH In-Stock Unstable UL80 28 40 O=C(COc1c(Br)cc(C(=O)O)cc1Br)NCc1ccccc1 ZINC000217735545 IH In-Stock Unstable HDAC8 17 43 O=C(COc1c(Br)cc(C(=O)O)cc1Br)NCc1ccccc1 ZINC000217735545 IH In-Stock Unstable CA5B 28 42 O=C(COc1c(Br)cc(C(=O)O)cc1Br)NCc1ccccc1 ZINC000217735545 IH In-Stock Unstable CA5A 32 42 O=C(COc1c(Br)cc(C(=O)O)cc1Br)NCc1ccccc1 ZINC000217735545 IH In-Stock Unstable PTPN1 15 41 O=C(COc1c(Br)cc(C(=O)O)cc1Br)NCc1ccccc1 ZINC000217735545 IH In-Stock Unstable TPMT 0 40 O=C(COc1c(Br)cc(C(=O)O)cc1Br)NCc1ccccc1 ZINC000217735545 IH In-Stock Unstable AMP1_PLAFQ 51 38 O=C(COc1c(Br)cc(C(=O)O)cc1Br)NCc1ccccc1 ZINC000217735545 IH In-Stock Unstable KDM4E 21 41 O=C(COc1c(Br)cc(C(=O)O)cc1Br)NCc1ccccc1 ZINC000217735545 IH In-Stock Unstable PDS 66 39 O=C(Nc1ccc(Cl)c(Cl)c1)N1CC(N2C(=O)[C@H]3CC=CC[C@H]3C2=O)C1 ZINC000217735558 GG In-Stock Unstable PPX1 0 41 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1N[C@H](c1ccccc1)C1CC1 ZINC000217735572 CK For-Sale Unstable TRPM8 17 46 Cc1cccc(/C=C\C(=O)Nc2cc(C(=O)O)ccn2)c1 ZINC000217735589 CF For-Sale Unstable HDAC8 50 43 Cc1cccc(/C=C\C(=O)Nc2cc(C(=O)O)ccn2)c1 ZINC000217735589 CF For-Sale Unstable MMP2 15 47 Cc1cccc(/C=C\C(=O)Nc2cc(C(=O)O)ccn2)c1 ZINC000217735589 CF For-Sale Unstable HDAC6 30 43 Cc1cccc(/C=C\C(=O)Nc2cc(C(=O)O)ccn2)c1 ZINC000217735589 CF For-Sale Unstable MMP9 0 50 Cc1cccc(/C=C\C(=O)Nc2cc(C(=O)O)ccn2)c1 ZINC000217735589 CF For-Sale Unstable MMP1 24 50 Cc1cccc(/C=C\C(=O)Nc2cc(C(=O)O)ccn2)c1 ZINC000217735589 CF For-Sale Unstable KCNK3 48 39 COc1ccccc1/C=C/NC(=O)N1CCN(c2cccc(C)c2)CC1 ZINC000217735606 FH For-Sale Unstable GPR183 0 40 O=C(/C=C/c1ccc2c(c1)OCO2)NC[C@@H]1CCCN1c1nccs1 ZINC000217735639 FF For-Sale Unstable NOS2 91 39 O=C(Nc1ccc(Cl)c(Cl)c1)N1CC(N2C(=O)[C@H]3CC=CC[C@@H]3C2=O)C1 ZINC000217735648 GG In-Stock Unstable PPX1 0 41 O=C(COc1c(Br)cc(C(=O)O)cc1Br)NCCc1ccccc1 ZINC000217735659 JH In-Stock Unstable THRA 30 45 O=C(COc1c(Br)cc(C(=O)O)cc1Br)NCCc1ccccc1 ZINC000217735659 JH In-Stock Unstable THRB 28 45 O=C(COc1c(Br)cc(C(=O)O)cc1Br)NCCc1ccccc1 ZINC000217735659 JH In-Stock Unstable HDAC8 20 47 O=C(COc1c(Br)cc(C(=O)O)cc1Br)NCCc1ccccc1 ZINC000217735659 JH In-Stock Unstable CA5B 25 44 O=C(COc1c(Br)cc(C(=O)O)cc1Br)NCCc1ccccc1 ZINC000217735659 JH In-Stock Unstable CA5A 24 44 O=C(COc1c(Br)cc(C(=O)O)cc1Br)NCCc1ccccc1 ZINC000217735659 JH In-Stock Unstable AMP1_PLAFQ 26 40 O=C(COc1c(Br)cc(C(=O)O)cc1Br)NCCc1ccccc1 ZINC000217735659 JH In-Stock Unstable NCE103 26 46 O=C(COc1c(Br)cc(C(=O)O)cc1Br)NCCc1ccccc1 ZINC000217735659 JH In-Stock Unstable CRTM 41 36 O=C(COc1c(Br)cc(C(=O)O)cc1Br)NCCc1ccccc1 ZINC000217735659 JH In-Stock Unstable P96878_MYCTU 18 46 O=C(COc1c(Br)cc(C(=O)O)cc1Br)NCCc1ccccc1 ZINC000217735659 JH In-Stock Unstable KDM4E 24 51 O=C(COc1c(Br)cc(C(=O)O)cc1Br)NCCc1ccccc1 ZINC000217735659 JH In-Stock Unstable CAN2 0 46 CC(C)[C@H]1CC[C@H](C)C[C@@H]1N[C@H](c1ccccc1)C1CC1 ZINC000217735666 CK For-Sale Unstable TRPM8 17 46 COc1ccc2c(c1)[C@@]1(C(=O)N2)[C@H](C(=O)c2cccs2)[C@@H](c2cccc([N+](=O)[O-])c2)CN1C ZINC000217735693 JI In-Stock Unstable CACNA1C 55 37 COc1ccc2c(c1)[C@@]1(C(=O)N2)[C@H](C(=O)c2cccs2)[C@@H](c2cccc([N+](=O)[O-])c2)CN1C ZINC000217735693 JI In-Stock Unstable CACNA1D 87 37 O=C(/C=C/c1ccc2c(c1)OCO2)NC[C@H]1CCCN1c1nccs1 ZINC000217735724 FF For-Sale Unstable NOS2 91 39 O=C(Nc1ccc(Cl)c(Cl)c1)N1CC(N2C(=O)[C@@H]3CC=CC[C@H]3C2=O)C1 ZINC000217735733 GG In-Stock Unstable PPX1 0 41 CCOC(=O)N1CCC(NC(=O)N/C=C/c2ccccc2OC)CC1 ZINC000217735742 EF For-Sale Unstable CCR8 30 42 COc1cc(C[C@H](N)C(=O)O)c(O)cc1Cl ZINC000217735793 BD For-Sale Unstable HTR4 18 40 COc1cc(C[C@H](N)C(=O)O)c(O)cc1Cl ZINC000217735793 BD For-Sale Unstable TRPV1 19 41 CCOC(=O)N1CCC(NC(=O)C[C@@H]2NC(=O)c3ccccc3NC2=O)CC1 ZINC000217735807 GC In-Stock Unstable CHRM1 16 44 CCOC(=O)N1CCC(NC(=O)C[C@@H]2NC(=O)c3ccccc3NC2=O)CC1 ZINC000217735807 GC In-Stock Unstable CCR8 24 40 O=C(O)/C=C\c1cnc(NC(=O)c2cc(F)ccc2F)s1 ZINC000217735819 DF For-Sale Anodyne HSD17B1 0 40 COc1ccccc1/C=C/NC(=O)N1CCN(c2cccc(Cl)c2)CC1 ZINC000217735851 FH For-Sale Unstable DRD4 42 35 COc1ccccc1/C=C/NC(=O)N1CCN(c2cccc(Cl)c2)CC1 ZINC000217735851 FH For-Sale Unstable DRD3 30 41 COc1ccccc1/C=C/NC(=O)N1CCN(c2cccc(Cl)c2)CC1 ZINC000217735851 FH For-Sale Unstable CCKAR 0 40 Cc1cccnc1C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217735879 EG On-Demand Unstable HTR2A 18 45 Cc1cccnc1C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217735879 EG On-Demand Unstable HSD11B1 20 67 Cc1cccnc1C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217735879 EG On-Demand Unstable CCR5 20 43 Cc1cccnc1C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217735879 EG On-Demand Unstable SLC18A3 43 50 Cc1cccnc1C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217735879 EG On-Demand Unstable MLNR 17 42 Cc1cccnc1C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217735879 EG On-Demand Unstable WNT3A 48 35 Cc1cccnc1C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217735879 EG On-Demand Unstable L3MBTL3 62 35 COc1cc(C[C@@H](N)C(=O)O)c(O)cc1Cl ZINC000217735880 BD For-Sale Unstable HTR4 18 40 COc1cc(C[C@@H](N)C(=O)O)c(O)cc1Cl ZINC000217735880 BD For-Sale Unstable TRPV1 19 41 COc1cccc([C@H](O)CN2CCSC[C@@H]2C)c1 ZINC000217735901 CE For-Sale Unstable RORC 19 40 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1ccccc1 ZINC000217735904 IH In-Stock Unstable GUAB 0 48 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1ccccc1 ZINC000217735904 IH In-Stock Unstable HDAC8 19 41 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1ccccc1 ZINC000217735904 IH In-Stock Unstable HDAC3 20 41 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1ccccc1 ZINC000217735904 IH In-Stock Unstable HDAC6 15 41 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1ccccc1 ZINC000217735904 IH In-Stock Unstable TPMT 0 41 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1ccccc1 ZINC000217735904 IH In-Stock Unstable HIF1A 19 41 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1ccccc1 ZINC000217735904 IH In-Stock Unstable PFHDAC1 0 41 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1ccccc1 ZINC000217735904 IH In-Stock Unstable KCNK3 44 34 O=C(OCCC1CC1)c1cc([N+](=O)[O-])ccc1Br ZINC000217735941 DG On-Demand Unstable CACNA1C 45 38 O=C(OCCC1CC1)c1cc([N+](=O)[O-])ccc1Br ZINC000217735941 DG On-Demand Unstable CACNA1D 68 38 O=C(OCCC1CC1)c1cc([N+](=O)[O-])ccc1Br ZINC000217735941 DG On-Demand Unstable SLC27A4 44 33 CC(C)[C@@H]1CC(=O)Oc2c1c(=O)oc1ccccc21 ZINC000217735945 CF In-Stock Unstable NQO1 26 44 OC[C@H]1Cc2ccccc2CN1Cc1ccccc1 ZINC000217735949 CF For-Sale Unstable SIGMAR1 26 50 COc1ccccc1/C=C/NC(=O)Nc1ccc(-c2nc3ccc(C)cc3s2)cc1 ZINC000217735955 HK For-Sale Unstable CSNK1D 27 47 COc1ccccc1/C=C/NC(=O)Nc1ccc(-c2nc3ccc(C)cc3s2)cc1 ZINC000217735955 HK For-Sale Unstable APP 25 49 COc1ccccc1/C=C/NC(=O)Nc1ccc(-c2nc3ccc(C)cc3s2)cc1 ZINC000217735955 HK For-Sale Unstable LUCI_PHOPE 31 40 CCCCOc1ccc(C(=O)NC[C@@H]2CCCN2c2nccs2)cc1 ZINC000217735986 FH For-Sale Unstable PLA2G4B 45 34 Cc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217735987 II In-Stock Unstable THRA 18 42 Cc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217735987 II In-Stock Unstable THRB 21 42 Cc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217735987 II In-Stock Unstable CETP 0 41 Cc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217735987 II In-Stock Unstable GUAB 0 42 Cc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217735987 II In-Stock Unstable P4HTM 0 42 Cc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217735987 II In-Stock Unstable TPMT 0 41 CC(C)[C@H]1CC(=O)Oc2c1c(=O)oc1ccccc21 ZINC000217736005 CF In-Stock Unstable NQO1 26 44 COc1ccccc1/C=C/NC(=O)Nc1ccc2c(c1)OCO2 ZINC000217736055 DG For-Sale Unstable CCR2 0 45 COc1ccccc1/C=C/NC(=O)Nc1ccc2c(c1)OCO2 ZINC000217736055 DG For-Sale Unstable IMPDH2 0 45 COc1cccc(C(=O)Nc2ncc(/C=C\C(=O)O)s2)c1 ZINC000217736066 DF For-Sale Unstable DRD4 46 35 COc1cccc(C(=O)Nc2ncc(/C=C\C(=O)O)s2)c1 ZINC000217736066 DF For-Sale Unstable CSNK1D 19 43 COc1cccc(C(=O)Nc2ncc(/C=C\C(=O)O)s2)c1 ZINC000217736066 DF For-Sale Unstable GCK 22 43 COc1cccc(C(=O)Nc2ncc(/C=C\C(=O)O)s2)c1 ZINC000217736066 DF For-Sale Unstable TAAR1 31 41 COc1cccc(C(=O)Nc2ncc(/C=C\C(=O)O)s2)c1 ZINC000217736066 DF For-Sale Unstable SCD 34 46 COc1cccc(C(=O)Nc2ncc(/C=C\C(=O)O)s2)c1 ZINC000217736066 DF For-Sale Unstable KCNK3 57 49 CCCCOc1ccc(C(=O)NC[C@H]2CCCN2c2nccs2)cc1 ZINC000217736074 FH For-Sale Unstable PLA2G4B 45 34 Cc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1C ZINC000217736099 JJ In-Stock Unstable TPMT 0 40 Cc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1C ZINC000217736099 JJ In-Stock Unstable MCHR1 19 40 Cc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1C ZINC000217736099 JJ In-Stock Unstable MCHR2 40 39 Cc1cc(N2C[C@]34C=C[C@@H](O3)[C@@H](C(=O)NCc3ccc(Cl)cc3Cl)[C@H]4C2=O)no1 ZINC000217736105 IF In-Stock Unstable P2RX7 57 45 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217736129 JD In-Stock Unstable CHRNA4 26 40 CCCCOc1ccc(NC(=O)N2CC(N3C(=O)[C@H]4CC=CC[C@H]4C3=O)C2)cc1 ZINC000217736132 GG In-Stock Unstable FAAH 20 40 O=C(O)c1cc(S(=O)(=O)N[C@@H]2CCN3CCC[C@@H]23)c(Br)s1 ZINC000217736155 GD For-Sale Unstable SFRP1 57 32 O=C(O)c1cc(S(=O)(=O)N[C@@H]2CCN3CCC[C@@H]23)c(Br)s1 ZINC000217736155 GD For-Sale Unstable WNT3 50 32 O=C(O)/C=C\c1cnc(NC(=O)c2ccc([N+](=O)[O-])o2)s1 ZINC000217736165 DD For-Sale Bother DDIT3 0 44 Cc1cc(N2C[C@]34C=C[C@@H](O3)[C@H](C(=O)NCc3ccc(Cl)cc3Cl)[C@H]4C2=O)no1 ZINC000217736179 IF In-Stock Unstable P2RX7 57 45 CCCCOc1ccc(NC(=O)N2CC(N3C(=O)[C@H]4CC=CC[C@@H]4C3=O)C2)cc1 ZINC000217736214 GG In-Stock Unstable PLA2G4B 44 32 CCCCOc1ccc(NC(=O)N2CC(N3C(=O)[C@H]4CC=CC[C@@H]4C3=O)C2)cc1 ZINC000217736214 GG In-Stock Unstable FAAH 23 40 Cc1cc(C)cc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)c1 ZINC000217736224 JJ In-Stock Unstable TPMT 0 43 COc1cc(Cl)ccc1C(=O)N[C@@H](C)Cc1cccnc1 ZINC000217736231 DG In-Stock Unstable F10 40 31 COc1cc(Cl)ccc1C(=O)N[C@@H](C)Cc1cccnc1 ZINC000217736231 DG In-Stock Unstable TBXAS1 29 40 COc1cc(Cl)ccc1C(=O)N[C@@H](C)Cc1cccnc1 ZINC000217736231 DG In-Stock Unstable PTAFR 28 44 O=C(O)/C=C\c1cnc(NC(=O)CCC2CCCC2)s1 ZINC000217736246 CG For-Sale Unstable CDK5 53 45 O=C(O)c1cc(S(=O)(=O)N[C@H]2CCN3CCC[C@@H]23)c(Br)s1 ZINC000217736247 GD For-Sale Unstable SFRP1 57 32 O=C(O)c1cc(S(=O)(=O)N[C@H]2CCN3CCC[C@@H]23)c(Br)s1 ZINC000217736247 GD For-Sale Unstable WNT3 50 32 c1cc2c(cc1CN[C@@H]1CCN3CCC[C@@H]13)OCO2 ZINC000217736248 CD For-Sale Unstable NOS2 61 36 c1cc2c(cc1CN[C@@H]1CCN3CCC[C@@H]13)OCO2 ZINC000217736248 CD For-Sale Unstable SSTR3 48 30 CCCCOc1ccc(NC(=O)N2CC(N3C(=O)[C@@H]4CC=CC[C@H]4C3=O)C2)cc1 ZINC000217736301 GG In-Stock Unstable PLA2G4B 44 32 CCCCOc1ccc(NC(=O)N2CC(N3C(=O)[C@@H]4CC=CC[C@H]4C3=O)C2)cc1 ZINC000217736301 GG In-Stock Unstable FAAH 23 40 COc1ccccc1/C=C/NC(=O)Nc1cccc(F)c1 ZINC000217736305 CH For-Sale Unstable PDGFRA 26 44 COc1ccccc1/C=C/NC(=O)Nc1cccc(F)c1 ZINC000217736305 CH For-Sale Unstable TLR4 15 40 COc1ccccc1/C=C/NC(=O)Nc1cccc(F)c1 ZINC000217736305 CH For-Sale Unstable KCNK3 80 44 COc1ccccc1/C=C/NC(=O)Nc1cccc(F)c1 ZINC000217736305 CH For-Sale Unstable KCNK9 70 44 Cc1cc(C(=O)OCCC2CC2)c(N)c([N+](=O)[O-])c1 ZINC000217736311 CE On-Demand Unstable CACNA1D 43 35 COc1cc(Cl)ccc1C(=O)N[C@H](C)Cc1cccnc1 ZINC000217736324 DG In-Stock Unstable F10 40 31 COc1cc(Cl)ccc1C(=O)N[C@H](C)Cc1cccnc1 ZINC000217736324 DG In-Stock Unstable TBXAS1 29 40 COc1cc(Cl)ccc1C(=O)N[C@H](C)Cc1cccnc1 ZINC000217736324 DG In-Stock Unstable PTAFR 28 44 c1cc2c(cc1CN[C@H]1CCN3CCC[C@@H]13)OCO2 ZINC000217736328 CD For-Sale Unstable NOS2 61 36 c1cc2c(cc1CN[C@H]1CCN3CCC[C@@H]13)OCO2 ZINC000217736328 CD For-Sale Unstable SSTR3 48 30 COc1ccc(CC(=O)NC[C@@H]2CCCN2c2nccs2)cc1OC ZINC000217736408 FE For-Sale Unstable NOS2 25 44 COc1ccc(CC(=O)NC[C@@H]2CCCN2c2nccs2)cc1OC ZINC000217736408 FE For-Sale Unstable ACKR3 65 35 COc1ccccc1/C=C/NC(=O)NCCc1ccc(F)cc1 ZINC000217736411 DG For-Sale Unstable CCR3 15 42 COc1ccccc1/C=C/NC(=O)NCCc1ccc(F)cc1 ZINC000217736411 DG For-Sale Unstable MTNR1A 15 43 O=C(NCc1ccc(Cl)cc1)N1CC(N2C(=O)[C@H]3CC=CC[C@H]3C2=O)C1 ZINC000217736418 FE In-Stock Unstable SLC6A1 29 43 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1ccc(F)cc1 ZINC000217736433 II In-Stock Unstable LTA4H 16 40 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1ccc(F)cc1 ZINC000217736433 II In-Stock Unstable CETP 0 41 O=C(NCc1ccc(Cl)cc1)N1CC(N2C(=O)[C@H]3CC=CC[C@@H]3C2=O)C1 ZINC000217736498 FE In-Stock Unstable SLC6A1 29 43 COc1ccc(CC(=O)NC[C@H]2CCCN2c2nccs2)cc1OC ZINC000217736506 FE For-Sale Unstable NOS2 25 44 COc1ccc(CC(=O)NC[C@H]2CCCN2c2nccs2)cc1OC ZINC000217736506 FE For-Sale Unstable ACKR3 65 35 Cc1cc(C(=O)Nc2cccc(/C=C\C(=O)O)c2)on1 ZINC000217736508 CE For-Sale Unstable KCNK3 97 39 Cc1cc(C(=O)Nc2cccc(/C=C\C(=O)O)c2)on1 ZINC000217736508 CE For-Sale Unstable KCNK9 51 38 COc1ccccc1/C=C/NC(=O)N1CCc2ccccc21 ZINC000217736517 CG For-Sale Unstable DRD2 21 42 COc1ccccc1/C=C/NC(=O)N1CCc2ccccc21 ZINC000217736517 CG For-Sale Unstable DRD3 28 42 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1ccccc1Cl ZINC000217736542 JJ In-Stock Unstable EPHB3 47 35 O=C(/C=C\c1cccc(Cl)c1)Nc1cnccc1C(=O)O ZINC000217736565 DG For-Sale Anodyne LTB4R 0 45 O=C(/C=C\c1cccc(Cl)c1)Nc1cnccc1C(=O)O ZINC000217736565 DG For-Sale Anodyne MMP2 0 55 O=C(/C=C\c1cccc(Cl)c1)Nc1cnccc1C(=O)O ZINC000217736565 DG For-Sale Anodyne MMP9 0 52 O=C(/C=C\c1cccc(Cl)c1)Nc1cnccc1C(=O)O ZINC000217736565 DG For-Sale Anodyne HPSE 35 44 O=C(/C=C\c1cccc(Cl)c1)Nc1cnccc1C(=O)O ZINC000217736565 DG For-Sale Anodyne MMP1 24 55 O=C(/C=C\c1cccc(Cl)c1)Nc1cnccc1C(=O)O ZINC000217736565 DG For-Sale Anodyne PIM2 15 44 O=C(/C=C\c1cccc(Cl)c1)Nc1cnccc1C(=O)O ZINC000217736565 DG For-Sale Anodyne AKR1C2 22 42 O=C(/C=C\c1cccc(Cl)c1)Nc1cnccc1C(=O)O ZINC000217736565 DG For-Sale Anodyne TUBA4A 0 43 CCOc1c(OC)cc(N)c(Cl)c1C(=O)O ZINC000217736586 BE For-Sale Unstable HTR4 69 39 O=C(NCc1ccc(Cl)cc1)N1CC(N2C(=O)[C@@H]3CC=CC[C@H]3C2=O)C1 ZINC000217736587 FE In-Stock Unstable SLC6A1 29 43 Cc1nnsc1C(=O)Nc1cccc(/C=C\C(=O)O)c1 ZINC000217736592 CE For-Sale Unstable KCNK3 91 38 Cc1nnsc1C(=O)Nc1cccc(/C=C\C(=O)O)c1 ZINC000217736592 CE For-Sale Unstable KCNK9 51 38 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](C2CCCCC2)CC(=O)O4)cc1O ZINC000217736637 IJ In-Stock Unstable AKR1B1 0 48 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](C2CCCCC2)CC(=O)O4)cc1O ZINC000217736637 IJ In-Stock Unstable CYP1B1 57 35 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](C2CCCCC2)CC(=O)O4)cc1O ZINC000217736637 IJ In-Stock Unstable CYP1A1 42 48 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1cccc(Cl)c1 ZINC000217736646 JJ In-Stock Unstable THRA 17 42 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1cccc(Cl)c1 ZINC000217736646 JJ In-Stock Unstable PTGER1 23 40 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1cccc(Cl)c1 ZINC000217736646 JJ In-Stock Unstable THRB 15 42 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1cccc(Cl)c1 ZINC000217736646 JJ In-Stock Unstable UL80 26 44 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1cccc(Cl)c1 ZINC000217736646 JJ In-Stock Unstable F2R 0 45 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1cccc(Cl)c1 ZINC000217736646 JJ In-Stock Unstable GUAB 0 41 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1cccc(Cl)c1 ZINC000217736646 JJ In-Stock Unstable PTPN22 19 40 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1cccc(Cl)c1 ZINC000217736646 JJ In-Stock Unstable HIF1A 15 43 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1cccc(Cl)c1 ZINC000217736646 JJ In-Stock Unstable TAAR1 16 42 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1cccc(Cl)c1 ZINC000217736646 JJ In-Stock Unstable AKR1C3 27 48 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1cccc(Cl)c1 ZINC000217736646 JJ In-Stock Unstable IMDH_CRYPV 17 44 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1cccc(Cl)c1 ZINC000217736646 JJ In-Stock Unstable KCNK3 54 43 Cc1cccc(NC(=O)N2CC(N3C(=O)[C@H]4CC=CC[C@H]4C3=O)C2)c1 ZINC000217736688 EE In-Stock Unstable CCKAR 25 41 Cc1cccc(NC(=O)N2CC(N3C(=O)[C@H]4CC=CC[C@H]4C3=O)C2)c1 ZINC000217736688 EE In-Stock Unstable CCKBR 26 41 Cc1cccc(NC(=O)N2CC(N3C(=O)[C@H]4CC=CC[C@H]4C3=O)C2)c1 ZINC000217736688 EE In-Stock Unstable KCNK3 42 37 Cc1cccc(NC(=O)N2CC(N3C(=O)[C@H]4CC=CC[C@H]4C3=O)C2)c1 ZINC000217736688 EE In-Stock Unstable KCNK9 41 37 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](C2CCCCC2)CC(=O)O4)cc1O ZINC000217736728 IJ In-Stock Unstable AKR1B1 0 48 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](C2CCCCC2)CC(=O)O4)cc1O ZINC000217736728 IJ In-Stock Unstable CYP1B1 57 35 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](C2CCCCC2)CC(=O)O4)cc1O ZINC000217736728 IJ In-Stock Unstable CYP1A1 42 48 COc1ccccc1/C=C/NC(=O)NCCc1c[nH]c2ccccc12 ZINC000217736733 EH For-Sale Unstable EDNRB 22 43 COc1ccccc1/C=C/NC(=O)NCCc1c[nH]c2ccccc12 ZINC000217736733 EH For-Sale Unstable TACR1 40 48 COc1ccccc1/C=C/NC(=O)NCCc1c[nH]c2ccccc12 ZINC000217736733 EH For-Sale Unstable MC4R 36 48 COc1ccccc1/C=C/NC(=O)NCCc1c[nH]c2ccccc12 ZINC000217736733 EH For-Sale Unstable NQO2 19 46 COc1ccccc1/C=C/NC(=O)NCCc1c[nH]c2ccccc12 ZINC000217736733 EH For-Sale Unstable TRPV1 0 46 COc1ccccc1/C=C/NC(=O)NCCc1c[nH]c2ccccc12 ZINC000217736733 EH For-Sale Unstable CCKAR 79 47 COc1ccccc1/C=C/NC(=O)NCCc1c[nH]c2ccccc12 ZINC000217736733 EH For-Sale Unstable BRS3 28 44 COc1ccccc1/C=C/NC(=O)NCCc1c[nH]c2ccccc12 ZINC000217736733 EH For-Sale Unstable NMBR 39 49 COc1ccccc1/C=C/NC(=O)NCCc1c[nH]c2ccccc12 ZINC000217736733 EH For-Sale Unstable MTNR1A 34 48 COc1ccccc1/C=C/NC(=O)NCCc1c[nH]c2ccccc12 ZINC000217736733 EH For-Sale Unstable MTNR1B 25 47 COc1ccccc1/C=C/NC(=O)NCCc1c[nH]c2ccccc12 ZINC000217736733 EH For-Sale Unstable MMP14 58 36 COc1ccccc1/C=C/NC(=O)NCCc1c[nH]c2ccccc12 ZINC000217736733 EH For-Sale Unstable MMP11 41 32 COc1ccccc1/C=C/NC(=O)NCCc1c[nH]c2ccccc12 ZINC000217736733 EH For-Sale Unstable CCKBR 57 39 COc1ccccc1/C=C/NC(=O)NCCc1c[nH]c2ccccc12 ZINC000217736733 EH For-Sale Unstable GHSR 52 35 COc1ccccc1/C=C/NC(=O)NCCc1c[nH]c2ccccc12 ZINC000217736733 EH For-Sale Unstable ALOX15 22 40 COc1ccccc1/C=C/NC(=O)NCCc1c[nH]c2ccccc12 ZINC000217736733 EH For-Sale Unstable MMP9 19 52 COc1ccccc1/C=C/NC(=O)NCCc1c[nH]c2ccccc12 ZINC000217736733 EH For-Sale Unstable SLC15A2 0 40 Cc1cccc(NC(=O)N2CC(N3C(=O)[C@H]4CC=CC[C@@H]4C3=O)C2)c1 ZINC000217736767 EE In-Stock Unstable CCKAR 25 41 Cc1cccc(NC(=O)N2CC(N3C(=O)[C@H]4CC=CC[C@@H]4C3=O)C2)c1 ZINC000217736767 EE In-Stock Unstable CCKBR 26 41 Cc1cccc(NC(=O)N2CC(N3C(=O)[C@H]4CC=CC[C@@H]4C3=O)C2)c1 ZINC000217736767 EE In-Stock Unstable KCNK3 42 37 Cc1cccc(NC(=O)N2CC(N3C(=O)[C@H]4CC=CC[C@@H]4C3=O)C2)c1 ZINC000217736767 EE In-Stock Unstable KCNK9 41 37 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1ccc(Cl)cc1 ZINC000217736773 JJ In-Stock Unstable LTA4H 16 40 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1ccc(Cl)cc1 ZINC000217736773 JJ In-Stock Unstable PTGER1 18 42 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1ccc(Cl)cc1 ZINC000217736773 JJ In-Stock Unstable CETP 0 42 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1ccc(Cl)cc1 ZINC000217736773 JJ In-Stock Unstable GUAB 0 43 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1ccc(Cl)cc1 ZINC000217736773 JJ In-Stock Unstable MCHR1 17 43 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1ccc(Cl)cc1 ZINC000217736773 JJ In-Stock Unstable SENP1 0 40 COc1cc2c(cc1OC)CN(Cc1cc(=O)c(OCC(=O)Nc3ccc(C(C)C)cc3)co1)CC2 ZINC000217736839 JI In-Stock Unstable ABCB1B 58 40 COc1cc2c(cc1OC)CN(Cc1cc(=O)c(OCC(=O)Nc3ccc(C(C)C)cc3)co1)CC2 ZINC000217736839 JI In-Stock Unstable ABCB1 24 43 COc1cc2c(cc1OC)CN(Cc1cc(=O)c(OCC(=O)Nc3ccc(C(C)C)cc3)co1)CC2 ZINC000217736839 JI In-Stock Unstable ABCG2 35 40 Cc1cccc(NC(=O)N2CC(N3C(=O)[C@@H]4CC=CC[C@H]4C3=O)C2)c1 ZINC000217736852 EE In-Stock Unstable CCKAR 25 41 Cc1cccc(NC(=O)N2CC(N3C(=O)[C@@H]4CC=CC[C@H]4C3=O)C2)c1 ZINC000217736852 EE In-Stock Unstable CCKBR 26 41 Cc1cccc(NC(=O)N2CC(N3C(=O)[C@@H]4CC=CC[C@H]4C3=O)C2)c1 ZINC000217736852 EE In-Stock Unstable KCNK3 42 37 Cc1cccc(NC(=O)N2CC(N3C(=O)[C@@H]4CC=CC[C@H]4C3=O)C2)c1 ZINC000217736852 EE In-Stock Unstable KCNK9 41 37 CCCCCC(=O)Nc1ccc(/C=C\C(=O)O)cc1F ZINC000217736853 CG For-Sale Unstable SOAT1 20 40 CCCCCC(=O)Nc1ccc(/C=C\C(=O)O)cc1F ZINC000217736853 CG For-Sale Unstable MSR1 0 42 CCCCCC(=O)Nc1ccc(/C=C\C(=O)O)cc1F ZINC000217736853 CG For-Sale Unstable AKR1C3 28 40 CCCCCC(=O)Nc1ccc(/C=C\C(=O)O)cc1F ZINC000217736853 CG For-Sale Unstable ACAT 0 44 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1ccc(Br)cc1 ZINC000217736877 KJ In-Stock Unstable UL80 21 42 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1ccc(Br)cc1 ZINC000217736877 KJ In-Stock Unstable PRS 49 31 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1ccc(Br)cc1 ZINC000217736877 KJ In-Stock Unstable TPMT 0 40 CCCOc1cccnc1C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217736887 FH On-Demand Unstable HTR2A 19 43 CCCOc1cccnc1C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217736887 FH On-Demand Unstable SLC18A3 41 46 CCCOc1cccnc1C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217736887 FH On-Demand Unstable MLNR 17 41 CCCOc1cccnc1C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217736887 FH On-Demand Unstable WNT3A 56 36 CCCOc1cccnc1C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217736887 FH On-Demand Unstable L3MBTL3 40 31 Cc1cc(NC(=O)c2cc(Cl)c[nH]2)ccc1/C=C\C(=O)O ZINC000217736926 DG For-Sale Unstable KCNK3 45 35 COc1ccc(C(=O)COc2ccc3occ(-c4ccc(OC)c(OC)c4)c3c2)cc1OC ZINC000217736949 IK In-Stock Unstable ALDH2 87 39 Cc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1Cl ZINC000217736988 JJ In-Stock Unstable MCHR1 19 42 Cc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1Cl ZINC000217736988 JJ In-Stock Unstable MCHR2 41 41 Cc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1Cl ZINC000217736988 JJ In-Stock Unstable IMDH_CRYPV 33 40 Cc1nc(/C=C\C(=O)Nc2cnccc2C(=O)O)cs1 ZINC000217736999 CE For-Sale Unstable UL26 57 35 Cc1nc(/C=C\C(=O)Nc2cnccc2C(=O)O)cs1 ZINC000217736999 CE For-Sale Unstable SCAF_EBVB9 53 32 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1cc(Cl)cc(Cl)c1 ZINC000217737112 JK In-Stock Unstable TPMT 0 40 N[C@@H](Cc1c(Cl)nn2c1OCCC2)C(=O)O ZINC000217737145 BC For-Sale Unstable GRIA3 57 33 N[C@@H](Cc1c(Cl)nn2c1OCCC2)C(=O)O ZINC000217737145 BC For-Sale Unstable GRIA1 40 33 N[C@@H](Cc1c(Cl)nn2c1OCCC2)C(=O)O ZINC000217737145 BC For-Sale Unstable GRIA2 47 33 N[C@@H](Cc1c(Cl)nn2c1OCCC2)C(=O)O ZINC000217737145 BC For-Sale Unstable GRIA4 56 33 Cc1cc(/C=C\C(=O)O)ccc1NC(=O)Cn1cncn1 ZINC000217737189 CD For-Sale Unstable HIS3 40 31 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)cc1C(F)(F)F ZINC000217737195 FK For-Sale Unstable RBP4 22 42 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)cc1C(F)(F)F ZINC000217737195 FK For-Sale Unstable CYSP_PLAFA 41 33 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1cccc(C(F)(F)F)c1 ZINC000217737213 JJ In-Stock Unstable UL80 33 45 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1cccc(C(F)(F)F)c1 ZINC000217737213 JJ In-Stock Unstable KDR 18 40 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1cccc(C(F)(F)F)c1 ZINC000217737213 JJ In-Stock Unstable HDAC6 15 52 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1cccc(C(F)(F)F)c1 ZINC000217737213 JJ In-Stock Unstable SLC1A2 40 39 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1cccc(C(F)(F)F)c1 ZINC000217737213 JJ In-Stock Unstable HIF1A 15 41 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1cccc(C(F)(F)F)c1 ZINC000217737213 JJ In-Stock Unstable AKR1C3 20 49 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1cccc(C(F)(F)F)c1 ZINC000217737213 JJ In-Stock Unstable TRPM4 0 43 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1cccc(C(F)(F)F)c1 ZINC000217737213 JJ In-Stock Unstable KCNK3 39 46 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1cccc(C(F)(F)F)c1 ZINC000217737213 JJ In-Stock Unstable PDS 40 39 N[C@H](Cc1c(Cl)nn2c1OCCC2)C(=O)O ZINC000217737230 BC For-Sale Unstable GRIA3 57 33 N[C@H](Cc1c(Cl)nn2c1OCCC2)C(=O)O ZINC000217737230 BC For-Sale Unstable GRIA1 40 33 N[C@H](Cc1c(Cl)nn2c1OCCC2)C(=O)O ZINC000217737230 BC For-Sale Unstable GRIA2 47 33 N[C@H](Cc1c(Cl)nn2c1OCCC2)C(=O)O ZINC000217737230 BC For-Sale Unstable GRIA4 56 33 CC/C=C(\C)C(=O)Nc1cc(C(=O)O)ccn1 ZINC000217737326 BE On-Demand Unstable KDM4C 0 44 CC/C=C(\C)C(=O)Nc1cc(C(=O)O)ccn1 ZINC000217737326 BE On-Demand Unstable KDM3A 0 44 CC/C=C(\C)C(=O)Nc1cc(C(=O)O)ccn1 ZINC000217737326 BE On-Demand Unstable KDM5C 0 44 CC/C=C(\C)C(=O)Nc1cc(C(=O)O)ccn1 ZINC000217737326 BE On-Demand Unstable FTO 0 40 COc1ccccc1NC(=O)COc1c(Br)cc(C(=O)O)cc1Br ZINC000217737334 JH In-Stock Unstable LTB4R 16 46 COc1ccccc1NC(=O)COc1c(Br)cc(C(=O)O)cc1Br ZINC000217737334 JH In-Stock Unstable TPMT 0 44 COc1cc(NC(=O)N/C=C/c2ccccc2OC)c(OC)cc1Cl ZINC000217737396 FI For-Sale Unstable CYSP_PLAFA 42 36 COc1cccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)c1 ZINC000217737442 JH In-Stock Unstable DRD4 42 32 COc1cccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)c1 ZINC000217737442 JH In-Stock Unstable PDGFRB 20 42 COc1cccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)c1 ZINC000217737442 JH In-Stock Unstable LTA4H 15 40 COc1cccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)c1 ZINC000217737442 JH In-Stock Unstable MTNR1A 40 48 COc1cccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)c1 ZINC000217737442 JH In-Stock Unstable MTNR1B 40 52 COc1cccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)c1 ZINC000217737442 JH In-Stock Unstable TPMT 0 43 COc1cccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)c1 ZINC000217737442 JH In-Stock Unstable MCHR1 21 40 COc1cccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)c1 ZINC000217737442 JH In-Stock Unstable HIF1A 16 43 COc1cccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)c1 ZINC000217737442 JH In-Stock Unstable TAAR1 41 53 COc1cccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)c1 ZINC000217737442 JH In-Stock Unstable AKR1C3 43 44 COc1cccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)c1 ZINC000217737442 JH In-Stock Unstable AKR1C2 48 38 COc1cccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)c1 ZINC000217737442 JH In-Stock Unstable KCNK3 68 46 COc1cccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)c1 ZINC000217737442 JH In-Stock Unstable KCNK9 54 36 Cc1cc(/C=C\C(=O)O)ccc1NC(=O)CC(C)(C)C ZINC000217737448 CG For-Sale Unstable MMP1 0 41 Cc1cc(/C=C\C(=O)O)ccc1NC(=O)Cc1cccs1 ZINC000217737534 DG For-Sale Unstable CA5B 47 47 Cc1cc(/C=C\C(=O)O)ccc1NC(=O)Cc1cccs1 ZINC000217737534 DG For-Sale Unstable CA5A 49 47 O=C(Nc1ccccc1C(F)(F)F)N1CC(N2C(=O)[C@H]3CC=CC[C@H]3C2=O)C1 ZINC000217737541 GF In-Stock Unstable RBP4 92 48 O=C(Nc1ccccc1C(F)(F)F)N1CC(N2C(=O)[C@H]3CC=CC[C@H]3C2=O)C1 ZINC000217737541 GF In-Stock Unstable SMO 25 52 COc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217737544 JH In-Stock Unstable THRA 32 40 COc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217737544 JH In-Stock Unstable THRB 31 40 COc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217737544 JH In-Stock Unstable ADORA2B 42 38 COc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217737544 JH In-Stock Unstable CETP 0 45 COc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217737544 JH In-Stock Unstable GUAB 0 43 COc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217737544 JH In-Stock Unstable HDAC8 29 42 COc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217737544 JH In-Stock Unstable MTNR1A 41 43 COc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217737544 JH In-Stock Unstable MTNR1B 33 46 COc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217737544 JH In-Stock Unstable ACR 49 40 COc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217737544 JH In-Stock Unstable CA12 16 43 COc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217737544 JH In-Stock Unstable TPMT 0 46 COc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217737544 JH In-Stock Unstable CA9 24 43 COc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217737544 JH In-Stock Unstable MCHR1 24 47 COc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217737544 JH In-Stock Unstable AKR1C3 33 44 COc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217737544 JH In-Stock Unstable AKR1C2 51 40 COc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217737544 JH In-Stock Unstable ENPP1 47 32 COc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217737544 JH In-Stock Unstable GPR35 40 38 CC[C@@H](C(=O)N(CC(=O)Nc1ccc(F)cc1)C(C)C)c1ccccc1 ZINC000217737585 FI On-Demand Unstable KCNQ2 41 41 CC[C@@H](C(=O)N(CC(=O)Nc1ccc(F)cc1)C(C)C)c1ccccc1 ZINC000217737585 FI On-Demand Unstable NPY5R 32 42 COc1cc2c(cc1OC)CN(Cc1cc(=O)c(O)c(CN3CCOCC3)o1)CC2 ZINC000217737591 HD In-Stock Unstable ABCB1B 62 36 COc1cc2c(cc1OC)CN(Cc1cc(=O)c(O)c(CN3CCOCC3)o1)CC2 ZINC000217737591 HD In-Stock Unstable ABCB1 22 47 O=C(Nc1ccccc1C(F)(F)F)N1CC(N2C(=O)[C@H]3CC=CC[C@@H]3C2=O)C1 ZINC000217737615 GF In-Stock Unstable RBP4 92 48 O=C(Nc1ccccc1C(F)(F)F)N1CC(N2C(=O)[C@H]3CC=CC[C@@H]3C2=O)C1 ZINC000217737615 GF In-Stock Unstable SMO 25 52 COc1ccccc1/C=C/NC(=O)N1CCN(c2cccc(C)c2C)CC1 ZINC000217737631 FH For-Sale Unstable ABCB1 23 41 CC[C@H](C(=O)N(CC(=O)Nc1ccc(F)cc1)C(C)C)c1ccccc1 ZINC000217737673 FI On-Demand Unstable KCNQ2 41 41 CC[C@H](C(=O)N(CC(=O)Nc1ccc(F)cc1)C(C)C)c1ccccc1 ZINC000217737673 FI On-Demand Unstable NPY5R 32 42 O=C(Nc1ccccc1C(F)(F)F)N1CC(N2C(=O)[C@@H]3CC=CC[C@H]3C2=O)C1 ZINC000217737696 GF In-Stock Unstable RBP4 76 45 O=C(Nc1ccccc1C(F)(F)F)N1CC(N2C(=O)[C@@H]3CC=CC[C@H]3C2=O)C1 ZINC000217737696 GF In-Stock Unstable SMO 25 52 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccccc2)CC1 ZINC000217737734 EG For-Sale Unstable HTR1A 33 49 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccccc2)CC1 ZINC000217737734 EG For-Sale Unstable DRD2 27 42 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccccc2)CC1 ZINC000217737734 EG For-Sale Unstable DRD3 34 42 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccccc2)CC1 ZINC000217737734 EG For-Sale Unstable TACR1 0 40 CCOc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217737778 JI In-Stock Unstable THRA 31 42 CCOc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217737778 JI In-Stock Unstable THRB 31 42 CCOc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217737778 JI In-Stock Unstable ADORA2B 44 38 CCOc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217737778 JI In-Stock Unstable PLA2G4B 47 35 CCOc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217737778 JI In-Stock Unstable P4HTM 0 51 CCOc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217737778 JI In-Stock Unstable MCHR1 18 40 CCOc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217737778 JI In-Stock Unstable HIF1A 23 40 CCC[C@@H](O)CNC[C@@H](C)c1ccccc1 ZINC000217737820 BF For-Sale Unstable AOC3 15 49 C[C@H](NC(=O)C1CCC1)c1cccc(/C=C\C(=O)O)c1 ZINC000217737856 CF For-Sale Unstable KCNQ2 47 34 C[C@H](NC(=O)C1CCC1)c1cccc(/C=C\C(=O)O)c1 ZINC000217737856 CF For-Sale Unstable BIRC8 41 31 COC(=O)[C@@H](O)CNC(=O)c1cccnc1Cl ZINC000217737863 CB On-Demand Unstable G2YM83_BOTF4 84 41 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1ccc(Oc2ccccc2)cc1 ZINC000217737876 KK In-Stock Unstable SRD5A2 28 42 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1ccc(Oc2ccccc2)cc1 ZINC000217737876 KK In-Stock Unstable LTA4H 66 48 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1ccc(Oc2ccccc2)cc1 ZINC000217737876 KK In-Stock Unstable CA1 19 40 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1ccc(Oc2ccccc2)cc1 ZINC000217737876 KK In-Stock Unstable CETP 31 41 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1ccc(Oc2ccccc2)cc1 ZINC000217737876 KK In-Stock Unstable SLC1A2 21 40 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1ccc(Oc2ccccc2)cc1 ZINC000217737876 KK In-Stock Unstable MCHR1 24 40 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1ccc(Oc2ccccc2)cc1 ZINC000217737876 KK In-Stock Unstable Q8MMZ8_EIMTE 50 39 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1ccc(Oc2ccccc2)cc1 ZINC000217737876 KK In-Stock Unstable HIF1A 19 40 O=C(COc1c(Br)cc(C(=O)O)cc1Br)Nc1ccc(Oc2ccccc2)cc1 ZINC000217737876 KK In-Stock Unstable PFKFB3 56 40 CCC[C@H](O)CNC[C@@H](C)c1ccccc1 ZINC000217737905 BF For-Sale Unstable AOC3 15 49 COC(=O)c1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1 ZINC000217737907 JI In-Stock Unstable AKR1B1 0 42 COC(=O)c1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1 ZINC000217737907 JI In-Stock Unstable CYP1A1 28 42 COC(=O)c1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1 ZINC000217737907 JI In-Stock Unstable CYP1A2 22 42 COC(=O)[C@H](O)CNC(=O)c1cccnc1Cl ZINC000217737928 CB For-Sale Unstable G2YM83_BOTF4 84 41 C[C@@H](NC(=O)C1CCC1)c1cccc(/C=C\C(=O)O)c1 ZINC000217737938 CF For-Sale Unstable KCNQ2 47 34 C[C@@H](NC(=O)C1CCC1)c1cccc(/C=C\C(=O)O)c1 ZINC000217737938 CF For-Sale Unstable BIRC8 41 31 COc1ccccc1/C=C/NC(=O)Nc1c(C)cccc1C ZINC000217737945 CI For-Sale Unstable ACAT 0 40 O=C(NC[C@@H]1CCCN1c1nccs1)C1c2ccccc2Oc2ccccc21 ZINC000217737959 GI For-Sale Unstable TK 49 43 C[C@@H]1CCC[C@@H](CNS(=O)(=O)c2cccnc2Cl)C1 ZINC000217737960 DF On-Demand Unstable NPY2R 55 42 C[C@H](N[C@H]1CCCc2cccnc21)[C@@H]1CCCO1 ZINC000217737970 BF On-Demand Unstable CXCR4 46 35 COC(=O)c1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1 ZINC000217737976 JI In-Stock Unstable AKR1B1 0 42 COC(=O)c1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1 ZINC000217737976 JI In-Stock Unstable CYP1A1 28 42 COC(=O)c1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1 ZINC000217737976 JI In-Stock Unstable CYP1A2 22 42 CCC[C@@H](O)CNC[C@H](C)c1ccccc1 ZINC000217737982 BF For-Sale Unstable AOC3 15 49 COc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)c(OC)c1 ZINC000217738008 JH In-Stock Unstable TPMT 0 42 COc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)c(OC)c1 ZINC000217738008 JH In-Stock Unstable AKR1C2 51 37 COc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)c(OC)c1 ZINC000217738008 JH In-Stock Unstable ACAT 0 46 COc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)c(OC)c1 ZINC000217738008 JH In-Stock Unstable GPR35 43 38 COc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)c(OC)c1 ZINC000217738008 JH In-Stock Unstable FAS 19 40 O=C(NC[C@H]1CCCN1c1nccs1)C1c2ccccc2Oc2ccccc21 ZINC000217738013 GI For-Sale Unstable TK 49 43 C[C@H](NC(=O)C1CCCC1)c1cccc(/C=C\C(=O)O)c1 ZINC000217738019 CG For-Sale Unstable KCNQ2 47 34 C[C@H](NC(=O)C1CCCC1)c1cccc(/C=C\C(=O)O)c1 ZINC000217738019 CG For-Sale Unstable BIRC8 42 33 C[C@H]1CCC[C@@H](CNS(=O)(=O)c2cccnc2Cl)C1 ZINC000217738021 DF On-Demand Unstable NPY2R 55 42 COc1ccccc1/C=C/NC(=O)Nc1cc([N+](=O)[O-])ccc1OC ZINC000217738045 EG For-Sale Unstable KCNMA1 23 56 CCC[C@H](O)CNC[C@H](C)c1ccccc1 ZINC000217738058 BF For-Sale Unstable AOC3 15 49 C[C@@H]1CCC[C@H](CNS(=O)(=O)c2cccnc2Cl)C1 ZINC000217738106 DF On-Demand Unstable NPY2R 55 42 C[C@@H](NC(=O)C1CCCC1)c1cccc(/C=C\C(=O)O)c1 ZINC000217738107 CG For-Sale Unstable KCNQ2 47 34 C[C@@H](NC(=O)C1CCCC1)c1cccc(/C=C\C(=O)O)c1 ZINC000217738107 CG For-Sale Unstable BIRC8 42 33 COc1ccc(C)cc1NC(=O)COc1c(Br)cc(C(=O)O)cc1Br ZINC000217738111 JI In-Stock Unstable TPMT 0 42 COc1ccc(Br)c(C(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217738134 GG For-Sale Unstable DRD2 31 41 C[C@H]1CCC[C@H](CNS(=O)(=O)c2cccnc2Cl)C1 ZINC000217738179 DF On-Demand Unstable NPY2R 55 42 Cc1ccc(/C=C\C(=O)O)cc1NC(=O)C1CCCCC1 ZINC000217738195 CH For-Sale Unstable STK17B 40 37 CCCC#C/C=C\C[C@H](NC(=O)OC(C)(C)C)C(=O)O ZINC000217738203 CF For-Sale Unstable PAPA1_CARPA 36 47 CCCC#C/C=C\C[C@H](NC(=O)OC(C)(C)C)C(=O)O ZINC000217738203 CF For-Sale Unstable CTSK 21 47 CCCC#C/C=C\C[C@H](NC(=O)OC(C)(C)C)C(=O)O ZINC000217738203 CF For-Sale Unstable FPR1 43 36 CC(C)(C)OC(=O)N/C=C/C=C/C(=O)O ZINC000217738215 BD For-Sale Unstable CTSK 18 42 COc1ccc(Br)c(C(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217738217 GG For-Sale Unstable DRD2 31 41 COc1ccc(Br)c(C(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217738217 GG For-Sale Unstable DRD3 15 45 COc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1Cl ZINC000217738233 JJ In-Stock Unstable HTR2A 24 42 COc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1Cl ZINC000217738233 JJ In-Stock Unstable CYSP_TRYCR 0 43 COc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1Cl ZINC000217738233 JJ In-Stock Unstable COLA 52 38 COc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1Cl ZINC000217738233 JJ In-Stock Unstable CPT1A 50 38 COc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1Cl ZINC000217738233 JJ In-Stock Unstable CPT2 44 34 COc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1Cl ZINC000217738233 JJ In-Stock Unstable GRM4 18 47 COc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1Cl ZINC000217738233 JJ In-Stock Unstable PDE6A 42 34 COc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1Cl ZINC000217738233 JJ In-Stock Unstable TPMT 0 42 COc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1Cl ZINC000217738233 JJ In-Stock Unstable MCHR1 19 42 COc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1Cl ZINC000217738233 JJ In-Stock Unstable MCHR2 39 42 COc1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1Cl ZINC000217738233 JJ In-Stock Unstable ENPP1 72 36 CNS(=O)(=O)c1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1 ZINC000217738276 HE On-Demand Unstable HRH2 15 45 CNS(=O)(=O)c1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1 ZINC000217738276 HE On-Demand Unstable SLC18A3 40 51 CNS(=O)(=O)c1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1 ZINC000217738276 HE On-Demand Unstable SLC9A1 18 51 CNS(=O)(=O)c1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1 ZINC000217738276 HE On-Demand Unstable EPHX2 15 45 CNS(=O)(=O)c1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1 ZINC000217738276 HE On-Demand Unstable SFRP1 68 39 CNS(=O)(=O)c1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1 ZINC000217738276 HE On-Demand Unstable WNT3A 50 36 CNS(=O)(=O)c1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1 ZINC000217738276 HE On-Demand Unstable L3MBTL3 89 44 COCCNC(=O)COc1ccc2c(c1)O/C(=C/c1cn(C)c3ccccc13)C2=O ZINC000217738279 HF In-Stock Unstable MTOR 0 47 CCCC#C/C=C\C[C@@H](NC(=O)OC(C)(C)C)C(=O)O ZINC000217738286 CF For-Sale Unstable PAPA1_CARPA 36 47 CCCC#C/C=C\C[C@@H](NC(=O)OC(C)(C)C)C(=O)O ZINC000217738286 CF For-Sale Unstable CTSK 21 47 CCCC#C/C=C\C[C@@H](NC(=O)OC(C)(C)C)C(=O)O ZINC000217738286 CF For-Sale Unstable FPR1 43 36 Cc1onc(-c2ccccc2Cl)c1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217738312 HI For-Sale Unstable GPBAR1 29 42 COC(=O)c1ccccc1NC(=O)COc1c(Br)cc(C(=O)O)cc1Br ZINC000217738348 JH In-Stock Unstable TPMT 0 40 COC(=O)c1ccccc1NC(=O)COc1c(Br)cc(C(=O)O)cc1Br ZINC000217738348 JH In-Stock Unstable FABH 0 41 COC(=O)c1ccccc1NC(=O)COc1c(Br)cc(C(=O)O)cc1Br ZINC000217738348 JH In-Stock Unstable FAS 62 50 Cc1onc(-c2ccccc2Cl)c1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217738389 HI For-Sale Unstable GPBAR1 29 42 CC[C@@H](C)NC(=O)CN1CCO[C@@H](CN)C1 ZINC000217738399 BB On-Demand Unstable NOD1 50 32 COC(=O)c1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217738458 JH In-Stock Unstable ACR 63 39 COC(=O)c1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217738458 JH In-Stock Unstable TPMT 0 46 COC(=O)c1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217738458 JH In-Stock Unstable KDM3A 0 42 COC(=O)c1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217738458 JH In-Stock Unstable KDM5C 0 42 CC[C@H](C)NC(=O)CN1CCO[C@@H](CN)C1 ZINC000217738465 BB On-Demand Unstable NOD1 50 32 COc1ccccc1/C=C/NC(=O)NCCC(C)C ZINC000217738473 CG For-Sale Unstable DNPEP 0 40 COc1nc(Cl)nc(OC)c1C(=O)O ZINC000217738527 BC For-Sale Unstable ALS 76 37 Cc1ccc(C(=O)Nc2cccc(/C=C\C(=O)O)n2)cn1 ZINC000217738539 CE For-Sale Unstable GRM5 21 53 CCOC(=O)c1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217738556 KI In-Stock Unstable ADORA2B 20 42 CCOC(=O)c1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217738556 KI In-Stock Unstable ACR 64 35 CCOC(=O)c1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217738556 KI In-Stock Unstable NOD2 17 40 COc1ccccc1/C=C/NC(=O)NC[C@@H]1COc2ccccc2O1 ZINC000217738593 EF For-Sale Unstable ADRA1B 0 42 O=C(O)/C=C\c1cccc(NC(=O)Cc2ccccc2)n1 ZINC000217738631 CE For-Sale Unstable PTGER2 30 43 O=C(O)/C=C\c1cccc(NC(=O)Cc2ccccc2)n1 ZINC000217738631 CE For-Sale Unstable PTGER4 15 43 O=C(O)/C=C\c1cccc(NC(=O)Cc2ccccc2)n1 ZINC000217738631 CE For-Sale Unstable PTGER3 16 43 O=[N+]([O-])c1ccc(O)c(NS(=O)(=O)c2ccc(Br)cc2)c1 ZINC000217738643 FF On-Demand Bother NADE 0 41 O=[N+]([O-])c1ccc(O)c(NS(=O)(=O)c2ccc(Br)cc2)c1 ZINC000217738643 FF On-Demand Bother SNCA 24 42 O=[N+]([O-])c1ccc(O)c(NS(=O)(=O)c2ccc(Br)cc2)c1 ZINC000217738643 FF On-Demand Bother UQCRB 0 40 COc1ccccc1C(=O)N1C[C@H]2CNC[C@@H](C2)C1 ZINC000217738656 CD For-Sale Unstable CHRNA7 27 51 COc1ccccc1C(=O)N1C[C@H]2CNC[C@@H](C2)C1 ZINC000217738656 CD For-Sale Unstable MBTPS1 41 34 Cc1cc(S(=O)(=O)N2CC(N3C(=O)[C@H]4CC=CC[C@H]4C3=O)C2)ccc1F ZINC000217738660 GD In-Stock Unstable LEF 47 33 COc1ccccc1/C=C/NC(=O)NC[C@H]1COc2ccccc2O1 ZINC000217738664 EF For-Sale Unstable ADRA1B 0 42 NS(=O)(=O)c1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217738670 KF In-Stock Unstable CA2 155 51 NS(=O)(=O)c1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217738670 KF In-Stock Unstable CA6 20 44 NS(=O)(=O)c1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217738670 KF In-Stock Unstable CA1 139 51 NS(=O)(=O)c1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217738670 KF In-Stock Unstable CA7 72 50 NS(=O)(=O)c1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217738670 KF In-Stock Unstable CA13 24 43 NS(=O)(=O)c1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217738670 KF In-Stock Unstable CA5B 69 50 NS(=O)(=O)c1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217738670 KF In-Stock Unstable CA4 132 51 NS(=O)(=O)c1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217738670 KF In-Stock Unstable CA5A 75 50 NS(=O)(=O)c1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217738670 KF In-Stock Unstable CA14 52 50 NS(=O)(=O)c1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217738670 KF In-Stock Unstable CA12 90 51 NS(=O)(=O)c1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217738670 KF In-Stock Unstable CA9 97 51 NS(=O)(=O)c1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217738670 KF In-Stock Unstable CYNT 42 43 NS(=O)(=O)c1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217738670 KF In-Stock Unstable NCE103 53 44 NS(=O)(=O)c1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217738670 KF In-Stock Unstable MTCA1 56 47 NS(=O)(=O)c1ccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)cc1 ZINC000217738670 KF In-Stock Unstable P96878_MYCTU 71 47 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccc(S(=O)(=O)N2CCOCC2)cc1 ZINC000217738697 ID For-Sale Unstable TGM2 44 42 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccc(S(=O)(=O)N2CCOCC2)cc1 ZINC000217738697 ID For-Sale Unstable NAMPT 47 42 Cc1cc(S(=O)(=O)N2CC(N3C(=O)[C@H]4CC=CC[C@@H]4C3=O)C2)ccc1F ZINC000217738746 GD In-Stock Unstable LEF 47 33 COc1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)c(C)c1 ZINC000217738758 FH On-Demand Unstable CHRM2 45 40 COc1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)c(C)c1 ZINC000217738758 FH On-Demand Unstable HTR2A 15 44 COc1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)c(C)c1 ZINC000217738758 FH On-Demand Unstable OXTR 23 41 COc1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)c(C)c1 ZINC000217738758 FH On-Demand Unstable HSD11B1 18 72 COc1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)c(C)c1 ZINC000217738758 FH On-Demand Unstable CCR5 30 40 COc1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)c(C)c1 ZINC000217738758 FH On-Demand Unstable SLC18A3 43 59 COc1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)c(C)c1 ZINC000217738758 FH On-Demand Unstable WNT3A 52 33 COc1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)c(C)c1 ZINC000217738758 FH On-Demand Unstable L3MBTL3 60 40 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccccc2F)CC1 ZINC000217738768 FG For-Sale Unstable HTR1A 66 54 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccccc2F)CC1 ZINC000217738768 FG For-Sale Unstable DRD2 51 46 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccccc2F)CC1 ZINC000217738768 FG For-Sale Unstable DRD1 27 41 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccccc2F)CC1 ZINC000217738768 FG For-Sale Unstable DRD4 29 41 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccccc2F)CC1 ZINC000217738768 FG For-Sale Unstable ADRA1D 43 36 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccccc2F)CC1 ZINC000217738768 FG For-Sale Unstable HTR1B 15 54 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccccc2F)CC1 ZINC000217738768 FG For-Sale Unstable HTR2A 27 40 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccccc2F)CC1 ZINC000217738768 FG For-Sale Unstable ADRA1A 40 36 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccccc2F)CC1 ZINC000217738768 FG For-Sale Unstable DRD3 62 46 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccccc2F)CC1 ZINC000217738768 FG For-Sale Unstable HTR7 50 43 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccccc2F)CC1 ZINC000217738768 FG For-Sale Unstable SSTR1 15 43 CC(=O)c1cccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)c1 ZINC000217738785 JI In-Stock Unstable F2R 0 40 CC(=O)c1cccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)c1 ZINC000217738785 JI In-Stock Unstable GUAB 0 40 CC(=O)c1cccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)c1 ZINC000217738785 JI In-Stock Unstable HIF1A 17 47 CC(=O)c1cccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)c1 ZINC000217738785 JI In-Stock Unstable AKR1C3 45 51 CC(=O)c1cccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)c1 ZINC000217738785 JI In-Stock Unstable KCNK3 87 35 CC(=O)c1cccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)c1 ZINC000217738785 JI In-Stock Unstable KCNK9 52 34 CC(=O)c1cccc(NC(=O)COc2c(Br)cc(C(=O)O)cc2Br)c1 ZINC000217738785 JI In-Stock Unstable PARP10 0 43 O=C(/C=C\c1cccc(Br)c1)Nc1cc(C(=O)O)ccn1 ZINC000217738787 EG For-Sale Anodyne EGFR 26 40 O=C(/C=C\c1cccc(Br)c1)Nc1cc(C(=O)O)ccn1 ZINC000217738787 EG For-Sale Anodyne HDAC8 52 45 O=C(/C=C\c1cccc(Br)c1)Nc1cc(C(=O)O)ccn1 ZINC000217738787 EG For-Sale Anodyne MMP2 0 43 O=C(/C=C\c1cccc(Br)c1)Nc1cc(C(=O)O)ccn1 ZINC000217738787 EG For-Sale Anodyne HDAC6 35 45 O=C(/C=C\c1cccc(Br)c1)Nc1cc(C(=O)O)ccn1 ZINC000217738787 EG For-Sale Anodyne MMP9 0 43 O=C(/C=C\c1cccc(Br)c1)Nc1cc(C(=O)O)ccn1 ZINC000217738787 EG For-Sale Anodyne HPSE 21 42 O=C(/C=C\c1cccc(Br)c1)Nc1cc(C(=O)O)ccn1 ZINC000217738787 EG For-Sale Anodyne MMP1 23 41 O=C(/C=C\c1cccc(Br)c1)Nc1cc(C(=O)O)ccn1 ZINC000217738787 EG For-Sale Anodyne AKR1C3 17 40 Cc1ccccc1C(=O)Nc1ncc(/C=C\C(=O)O)s1 ZINC000217738788 CF For-Sale Unstable KCNK3 20 40 O=C(NC[C@H]1CCCN1c1nccs1)c1ccc(S(=O)(=O)N2CCOCC2)cc1 ZINC000217738797 ID For-Sale Unstable TGM2 44 42 O=C(NC[C@H]1CCCN1c1nccs1)c1ccc(S(=O)(=O)N2CCOCC2)cc1 ZINC000217738797 ID For-Sale Unstable NAMPT 47 42 Cc1cc(S(=O)(=O)N2CC(N3C(=O)[C@@H]4CC=CC[C@H]4C3=O)C2)ccc1F ZINC000217738836 GD In-Stock Unstable LEF 47 33 O=C(O)/C=C\c1cnc(NC(=O)CCc2ccccc2)s1 ZINC000217738877 DF For-Sale Unstable FAAH 46 36 O=C(O)/C=C\c1cnc(NC(=O)CCc2ccccc2)s1 ZINC000217738877 DF For-Sale Unstable CES1 43 36 O=C(O)/C=C\c1cnc(NC(=O)CCc2ccccc2)s1 ZINC000217738877 DF For-Sale Unstable CDK5 40 46 CCCNCC(=O)N1CC[C@@H](C)[C@@H]2CCCC[C@H]21 ZINC000217738906 CE For-Sale Unstable DPP4 15 50 COc1cccc(C(=O)N2C[C@H]3CNC[C@@H](C3)C2)c1 ZINC000217738937 CD For-Sale Unstable DRD4 49 37 COc1cccc(C(=O)N2C[C@H]3CNC[C@@H](C3)C2)c1 ZINC000217738937 CD For-Sale Unstable CHRNA7 28 51 COc1cccc(C(=O)N2C[C@H]3CNC[C@@H](C3)C2)c1 ZINC000217738937 CD For-Sale Unstable MTNR1B 29 42 COc1cccc(C(=O)N2C[C@H]3CNC[C@@H](C3)C2)c1 ZINC000217738937 CD For-Sale Unstable SCN5A 29 43 COc1cccc(C(=O)N2C[C@H]3CNC[C@@H](C3)C2)c1 ZINC000217738937 CD For-Sale Unstable TUBB2B 27 40 CCCC(=O)OCc1ccc(O)cc1 ZINC000217738958 AE For-Sale Unstable CA14 16 44 CCCC(=O)OCc1ccc(O)cc1 ZINC000217738958 AE For-Sale Unstable GRIA1 43 38 COc1ccc(CCN2C(=O)N[C@@H](CC(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)C2=O)cc1OC ZINC000217738959 JD In-Stock Unstable CHRNA4 26 45 CCCNCC(=O)N1CC[C@H](C)[C@@H]2CCCC[C@H]21 ZINC000217738982 CE For-Sale Unstable DPP4 15 50 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(OC)c(O)c2)CC(=O)O4)cc1O ZINC000217739065 JI In-Stock Unstable AKR1B1 25 52 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(OC)c(O)c2)CC(=O)O4)cc1O ZINC000217739065 JI In-Stock Unstable CYP1B1 61 38 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(OC)c(O)c2)CC(=O)O4)cc1O ZINC000217739065 JI In-Stock Unstable CYP1A1 47 52 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(OC)c(O)c2)CC(=O)O4)cc1O ZINC000217739065 JI In-Stock Unstable CYP1A2 37 42 CCCNCC(=O)N1CC[C@@H](C)[C@H]2CCCC[C@H]21 ZINC000217739073 CE For-Sale Unstable DPP4 15 50 c1cnc2c(c1)CCC[C@@H]2N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217739109 CF On-Demand Unstable CXCR4 49 35 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccc(OC(F)(F)F)cc1 ZINC000217739116 FG For-Sale Unstable GIPR 42 35 CCCCNC(=O)CC(=N)N ZINC000217739133 AC In-Stock Unstable NOD1 44 37 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(OC)c(O)c2)CC(=O)O4)cc1O ZINC000217739150 JI In-Stock Unstable AKR1B1 25 52 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(OC)c(O)c2)CC(=O)O4)cc1O ZINC000217739150 JI In-Stock Unstable CYP1B1 61 38 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(OC)c(O)c2)CC(=O)O4)cc1O ZINC000217739150 JI In-Stock Unstable CYP1A1 47 52 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(OC)c(O)c2)CC(=O)O4)cc1O ZINC000217739150 JI In-Stock Unstable CYP1A2 37 42 CC1(C)C(=O)NC(=O)CN1C(=O)/C=C\c1ccc(Br)cc1 ZINC000217739151 FD For-Sale Unstable GPR183 0 41 COc1ccccc1-n1cc(CNC(=O)c2cc(N)[nH]n2)cn1 ZINC000217739158 DD In-Stock Unstable HTR1A 19 40 COc1ccccc1-n1cc(CNC(=O)c2cc(N)[nH]n2)cn1 ZINC000217739158 DD In-Stock Unstable DRD2 27 40 CCCNCC(=O)N1CC[C@H](C)[C@H]2CCCC[C@H]21 ZINC000217739160 CE For-Sale Unstable DPP4 15 50 C[C@@H]1CCCC[C@@H]1C(=O)Nc1ccccc1 ZINC000217739175 BG On-Demand Unstable TAT_HV112 0 43 C[C@@H]1CCCC[C@@H]1C(=O)Nc1ccccc1 ZINC000217739175 BG On-Demand Unstable DGAT1 17 46 C[C@@H]1CCCC[C@@H]1C(=O)Nc1ccccc1 ZINC000217739175 BG On-Demand Unstable P95276_MYCTO 0 42 C[C@@H]1CCCC[C@@H]1C(=O)Nc1ccccc1 ZINC000217739175 BG On-Demand Unstable KCNK3 19 44 O=C(COc1ccccc1)N1C[C@H]2CNC[C@@H](C2)C1 ZINC000217739194 CD For-Sale Unstable CHRNA7 17 51 O=C(COc1ccccc1)N1C[C@H]2CNC[C@@H](C2)C1 ZINC000217739194 CD For-Sale Unstable COLA 135 40 O=C(COc1ccccc1)N1C[C@H]2CNC[C@@H](C2)C1 ZINC000217739194 CD For-Sale Unstable CPT1A 112 39 O=C(COc1ccccc1)N1C[C@H]2CNC[C@@H](C2)C1 ZINC000217739194 CD For-Sale Unstable CPT2 48 38 O=C(NC[C@H]1CCCN1c1nccs1)c1ccc(OC(F)(F)F)cc1 ZINC000217739212 FG For-Sale Unstable GIPR 42 35 COc1ccccc1/C=C/NC(=O)Nc1ccc(Br)c(C)c1 ZINC000217739227 FJ For-Sale Unstable IMPDH2 0 42 CC(C)CNC(=O)CC(=N)N ZINC000217739246 AC In-Stock Unstable F3 41 31 C[C@H]1CCCC[C@@H]1C(=O)Nc1ccccc1 ZINC000217739265 BG On-Demand Unstable TAT_HV112 0 43 C[C@H]1CCCC[C@@H]1C(=O)Nc1ccccc1 ZINC000217739265 BG On-Demand Unstable DGAT1 17 46 C[C@H]1CCCC[C@@H]1C(=O)Nc1ccccc1 ZINC000217739265 BG On-Demand Unstable P95276_MYCTO 0 42 C[C@H]1CCCC[C@@H]1C(=O)Nc1ccccc1 ZINC000217739265 BG On-Demand Unstable KCNK3 19 44 Cc1ccc(S(=O)(=O)Nc2ccc(F)cc2)cc1C(=O)N1CCC[C@@H]1c1cccn1C ZINC000217739286 II On-Demand Unstable WNT3 42 30 c1cnc2c(c1)CCC[C@@H]2N[C@H]1CCN2CCCC[C@@H]12 ZINC000217739296 CF On-Demand Unstable CXCR4 49 35 Cn1nc(-c2ccc(F)cc2)cc1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217739312 GG For-Sale Unstable HCRTR1 27 40 Cn1nc(-c2ccc(F)cc2)cc1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217739312 GG For-Sale Unstable HCRTR2 22 40 COc1cccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)c1C ZINC000217739316 FH On-Demand Unstable HTR2A 20 44 COc1cccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)c1C ZINC000217739316 FH On-Demand Unstable HSD11B1 19 69 COc1cccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)c1C ZINC000217739316 FH On-Demand Unstable CCR5 19 40 COc1cccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)c1C ZINC000217739316 FH On-Demand Unstable SLC18A3 43 51 COc1cccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)c1C ZINC000217739316 FH On-Demand Unstable WNT3A 50 31 COc1cccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)c1C ZINC000217739316 FH On-Demand Unstable L3MBTL3 58 38 C[C@@H]1CCCC[C@H]1C(=O)Nc1ccccc1 ZINC000217739346 BG On-Demand Unstable TAT_HV112 0 43 C[C@@H]1CCCC[C@H]1C(=O)Nc1ccccc1 ZINC000217739346 BG On-Demand Unstable DGAT1 17 46 C[C@@H]1CCCC[C@H]1C(=O)Nc1ccccc1 ZINC000217739346 BG On-Demand Unstable P95276_MYCTO 0 42 C[C@@H]1CCCC[C@H]1C(=O)Nc1ccccc1 ZINC000217739346 BG On-Demand Unstable KCNK3 19 44 Cc1ccc(S(=O)(=O)Nc2ccc(F)cc2)cc1C(=O)N1CCC[C@H]1c1cccn1C ZINC000217739365 II On-Demand Unstable WNT3 42 30 O=C(O)/C=C\c1ccc(NC(=O)c2ccccc2)c(F)c1 ZINC000217739375 CG For-Sale Anodyne MMP2 0 47 O=C(O)/C=C\c1ccc(NC(=O)c2ccccc2)c(F)c1 ZINC000217739375 CG For-Sale Anodyne HDAC1 22 45 O=C(O)/C=C\c1ccc(NC(=O)c2ccccc2)c(F)c1 ZINC000217739375 CG For-Sale Anodyne HDAC2 15 42 O=C(O)/C=C\c1ccc(NC(=O)c2ccccc2)c(F)c1 ZINC000217739375 CG For-Sale Anodyne MMP9 0 47 O=C(O)/C=C\c1ccc(NC(=O)c2ccccc2)c(F)c1 ZINC000217739375 CG For-Sale Anodyne MMP1 22 47 O=C(O)/C=C\c1ccc(NC(=O)c2ccccc2)c(F)c1 ZINC000217739375 CG For-Sale Anodyne KCNK3 70 41 Cn1nc(-c2ccc(F)cc2)cc1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217739395 GG For-Sale Unstable HCRTR1 27 40 Cn1nc(-c2ccc(F)cc2)cc1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217739395 GG For-Sale Unstable HCRTR2 22 40 Cc1cccc(/C=C\C(=O)Nc2cnccc2C(=O)O)c1 ZINC000217739414 CF For-Sale Unstable TRPV1 0 56 Cc1cccc(/C=C\C(=O)Nc2cnccc2C(=O)O)c1 ZINC000217739414 CF For-Sale Unstable HDAC8 46 39 Cc1cccc(/C=C\C(=O)Nc2cnccc2C(=O)O)c1 ZINC000217739414 CF For-Sale Unstable MMP2 15 47 Cc1cccc(/C=C\C(=O)Nc2cnccc2C(=O)O)c1 ZINC000217739414 CF For-Sale Unstable HDAC1 0 41 Cc1cccc(/C=C\C(=O)Nc2cnccc2C(=O)O)c1 ZINC000217739414 CF For-Sale Unstable MMP9 0 51 Cc1cccc(/C=C\C(=O)Nc2cnccc2C(=O)O)c1 ZINC000217739414 CF For-Sale Unstable MMP1 25 51 Cc1cccc(/C=C\C(=O)Nc2cnccc2C(=O)O)c1 ZINC000217739414 CF For-Sale Unstable AKR1C3 20 43 Cc1cccc(/C=C\C(=O)Nc2cnccc2C(=O)O)c1 ZINC000217739414 CF For-Sale Unstable AKR1C2 26 43 Cc1nc(N2CCOCC2)cc(Cl)c1C(=O)O ZINC000217739418 CD For-Sale Unstable PIK3CA 24 40 Cc1nc(N2CCOCC2)cc(Cl)c1C(=O)O ZINC000217739418 CD For-Sale Unstable PIK3CD 36 41 Cc1nc(N2CCOCC2)cc(Cl)c1C(=O)O ZINC000217739418 CD For-Sale Unstable PIK3CG 15 40 Cc1nc(N2CCOCC2)cc(Cl)c1C(=O)O ZINC000217739418 CD For-Sale Unstable PIK3CB 64 41 C[C@H]1CCCC[C@H]1C(=O)Nc1ccccc1 ZINC000217739421 BG On-Demand Unstable TAT_HV112 0 43 C[C@H]1CCCC[C@H]1C(=O)Nc1ccccc1 ZINC000217739421 BG On-Demand Unstable DGAT1 17 46 C[C@H]1CCCC[C@H]1C(=O)Nc1ccccc1 ZINC000217739421 BG On-Demand Unstable P95276_MYCTO 0 42 C[C@H]1CCCC[C@H]1C(=O)Nc1ccccc1 ZINC000217739421 BG On-Demand Unstable KCNK3 19 44 Cc1ccc(C(=O)Nc2ccc(/C=C\C(=O)O)c(C)c2)o1 ZINC000217739460 CG For-Sale Unstable KCNK3 49 35 Cc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)N1CCC[C@@H]1c1cccn1C ZINC000217739474 IH On-Demand Unstable SFRP1 56 32 Cc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)N1CCC[C@@H]1c1cccn1C ZINC000217739474 IH On-Demand Unstable WNT3 56 31 CN(C[C@@H]1COCCO1)C(=O)c1cc(C(C)(C)C)c(O)c(C(C)(C)C)c1 ZINC000217739531 FG In-Stock Unstable F2R 29 40 CC(C)(C)C[C@@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217739561 CE For-Sale Unstable CTSC 23 40 CC(C)(C)C[C@@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217739561 CE For-Sale Unstable MAN1B1 58 32 Cc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)N1CCC[C@H]1c1cccn1C ZINC000217739566 IH On-Demand Unstable SFRP1 56 32 Cc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)N1CCC[C@H]1c1cccn1C ZINC000217739566 IH On-Demand Unstable WNT3 56 31 C[C@@H]1CN(C[C@@H](O)c2ccccc2)CCO1 ZINC000217739591 BD On-Demand Unstable OPRK1 0 47 C[C@@H]1CN(C[C@@H](O)c2ccccc2)CCO1 ZINC000217739591 BD On-Demand Unstable IGF1R 0 43 C[C@@H]1CN(C[C@@H](O)c2ccccc2)CCO1 ZINC000217739591 BD On-Demand Unstable SLC18A3 26 43 CN(C[C@H]1COCCO1)C(=O)c1cc(C(C)(C)C)c(O)c(C(C)(C)C)c1 ZINC000217739619 FG In-Stock Unstable F2R 29 40 CC(C)(C)C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217739641 CE For-Sale Unstable CTSC 23 40 CC(C)(C)C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217739641 CE For-Sale Unstable MAN1B1 58 32 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)NCCc3c[nH]cn3)[C@H]21 ZINC000217739668 JD In-Stock Unstable HRH3 27 41 C[C@H]1CN(C[C@@H](O)c2ccccc2)CCO1 ZINC000217739676 BD On-Demand Unstable OPRK1 0 47 C[C@H]1CN(C[C@@H](O)c2ccccc2)CCO1 ZINC000217739676 BD On-Demand Unstable IGF1R 0 43 C[C@H]1CN(C[C@@H](O)c2ccccc2)CCO1 ZINC000217739676 BD On-Demand Unstable SLC18A3 26 43 O=C(/C=C\c1cccc(Cl)c1)Nc1cc(C(=O)O)ccn1 ZINC000217739681 DG For-Sale Anodyne HDAC8 44 43 O=C(/C=C\c1cccc(Cl)c1)Nc1cc(C(=O)O)ccn1 ZINC000217739681 DG For-Sale Anodyne MMP2 0 54 O=C(/C=C\c1cccc(Cl)c1)Nc1cc(C(=O)O)ccn1 ZINC000217739681 DG For-Sale Anodyne HDAC6 26 43 O=C(/C=C\c1cccc(Cl)c1)Nc1cc(C(=O)O)ccn1 ZINC000217739681 DG For-Sale Anodyne MMP9 0 51 O=C(/C=C\c1cccc(Cl)c1)Nc1cc(C(=O)O)ccn1 ZINC000217739681 DG For-Sale Anodyne MMP1 24 54 O=C(/C=C\c1cccc(Cl)c1)Nc1cc(C(=O)O)ccn1 ZINC000217739681 DG For-Sale Anodyne AKR1C3 22 44 O=C(/C=C\c1cccc(Cl)c1)Nc1cc(C(=O)O)ccn1 ZINC000217739681 DG For-Sale Anodyne TUBA4A 0 42 COC(=O)[C@@H](O)CNC(=O)COc1ccc(Cl)cc1Cl ZINC000217739702 DD On-Demand Unstable S1PR4 25 43 [N-]=[N+]=NCCCCCCCC(=O)O ZINC000217739716 AF For-Sale Unstable FABP4 15 44 [N-]=[N+]=NCCCCCCCC(=O)O ZINC000217739716 AF For-Sale Unstable FABP5 15 44 CC(C)(C)C[C@@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217739727 CE For-Sale Unstable CTSC 23 40 CC(C)(C)C[C@@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217739727 CE For-Sale Unstable MAN1B1 58 32 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)NCCc3c[nH]cn3)[C@@H]21 ZINC000217739751 JD In-Stock Unstable HRH3 27 41 C[C@@H]1CN(C[C@@H](O)COc2ccc(C#N)cc2)CCO1 ZINC000217739758 CD On-Demand Unstable ACOX1 49 29 COC(=O)[C@H](O)CNC(=O)COc1ccc(Cl)cc1Cl ZINC000217739794 DD On-Demand Unstable S1PR4 25 43 CC(C)(C)C[C@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217739802 CE For-Sale Unstable CTSC 23 40 CC(C)(C)C[C@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217739802 CE For-Sale Unstable MAN1B1 58 32 COc1cc(N2CCOCC2)cnc1C#N ZINC000217739843 BC For-Sale Unstable CHRNA4 19 41 COc1cc(N2CCOCC2)cnc1C#N ZINC000217739843 BC For-Sale Unstable TNIK 35 44 C[C@H]1CN(C[C@@H](O)COc2ccc(C#N)cc2)CCO1 ZINC000217739844 CD On-Demand Unstable ACOX1 49 29 CC(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N1CCc2n[nH]cc2C1 ZINC000217739858 DB In-Stock Unstable TRHR 59 41 CC(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N1CCc2n[nH]cc2C1 ZINC000217739858 DB In-Stock Unstable TRHR2 0 41 CC(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N1CCc2n[nH]cc2C1 ZINC000217739858 DB In-Stock Unstable GRPR 52 32 Cc1cc(/C=C\C(=O)O)ccc1NC(=O)c1ccc(Cl)o1 ZINC000217739864 DH For-Sale Unstable S1PR4 41 42 N=C(N)CC(=O)NC1CCCCCC1 ZINC000217739870 AD In-Stock Unstable EPHX2 21 43 CS(=O)(=O)c1ccc(C2(C#N)CCC2)c(F)c1 ZINC000217739905 CE For-Sale Unstable PTGS2 28 40 COc1ccccc1/C=C/NC(=O)NCCN1C(=O)CSC1=O ZINC000217739907 ED For-Sale Unstable DRD3 21 43 N#Cc1ncc(N2CCOCC2)cc1O ZINC000217739942 BC For-Sale Unstable AKR1C3 20 42 NC(=O)[C@@H]1CCN(S(=O)(=O)c2cnc(Cl)c(Cl)c2)C1 ZINC000217739975 DC For-Sale Unstable GCKR 41 32 COc1ccccc1/C=C/NC(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000217740008 FH For-Sale Unstable DRD2 0 52 COc1ccccc1/C=C/NC(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000217740008 FH For-Sale Unstable DRD3 43 55 COc1ccccc1/C=C/NC(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000217740008 FH For-Sale Unstable ADIPOR1 0 47 COc1ccccc1/C=C/NC(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000217740008 FH For-Sale Unstable ADIPOR2 0 47 CCCS(=O)(=O)Nc1ccc([N+](=O)[O-])cc1O ZINC000217740031 CD For-Sale Unstable TBXA2R 30 40 CCCS(=O)(=O)Nc1ccc([N+](=O)[O-])cc1O ZINC000217740031 CD For-Sale Unstable KCNMA1 19 40 CCCS(=O)(=O)Nc1ccc([N+](=O)[O-])cc1O ZINC000217740031 CD For-Sale Unstable ENR 0 40 COc1ccc(S(=O)(=O)N2CC(N3C(=O)[C@H]4CC=CC[C@H]4C3=O)C2)cc1Cl ZINC000217740035 HD In-Stock Unstable CYSP_TRYCR 17 40 NC(=O)[C@H]1CCN(S(=O)(=O)c2cnc(Cl)c(Cl)c2)C1 ZINC000217740059 DC For-Sale Unstable GCKR 41 32 COc1ccc(S(=O)(=O)N2CC(N3C(=O)[C@H]4CC=CC[C@@H]4C3=O)C2)cc1Cl ZINC000217740118 HD In-Stock Unstable CYSP_TRYCR 17 40 COc1ccc(S(=O)(=O)N2CC(N3C(=O)[C@@H]4CC=CC[C@H]4C3=O)C2)cc1Cl ZINC000217740191 HD In-Stock Unstable CYSP_TRYCR 17 40 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cc3ccccc3[nH]c2=O)CC(=O)O4)cc1O ZINC000217740199 JI In-Stock Unstable CYP1B1 48 35 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cc3ccccc3[nH]c2=O)CC(=O)O4)cc1O ZINC000217740199 JI In-Stock Unstable CYP1A1 35 43 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cc3cc(F)ccc3[nH]2)CC1 ZINC000217740221 FI On-Demand Unstable HTR2A 16 48 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cc3cc(F)ccc3[nH]2)CC1 ZINC000217740221 FI On-Demand Unstable GRIN2B 37 59 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cc3cc(F)ccc3[nH]2)CC1 ZINC000217740221 FI On-Demand Unstable HRH4 38 65 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cc3cc(F)ccc3[nH]2)CC1 ZINC000217740221 FI On-Demand Unstable PYGL 29 41 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cc3cc(F)ccc3[nH]2)CC1 ZINC000217740221 FI On-Demand Unstable SYK 22 42 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cc3cc(F)ccc3[nH]2)CC1 ZINC000217740221 FI On-Demand Unstable SLC18A3 38 46 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cc3cc(F)ccc3[nH]2)CC1 ZINC000217740221 FI On-Demand Unstable PLD2 45 39 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cc3cc(F)ccc3[nH]2)CC1 ZINC000217740221 FI On-Demand Unstable AKR1C3 36 51 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cc3cc(F)ccc3[nH]2)CC1 ZINC000217740221 FI On-Demand Unstable WNT3A 51 38 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cc3cc(F)ccc3[nH]2)CC1 ZINC000217740221 FI On-Demand Unstable L3MBTL3 73 38 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cc3ccccc3[nH]c2=O)CC(=O)O4)cc1O ZINC000217740285 JI In-Stock Unstable CYP1B1 48 35 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cc3ccccc3[nH]c2=O)CC(=O)O4)cc1O ZINC000217740285 JI In-Stock Unstable CYP1A1 35 43 c1cc2c(cc1CN1C[C@H]3CNC[C@@H](C3)C1)OCO2 ZINC000217740310 CD For-Sale Unstable NOS2 58 33 c1cc2c(cc1CN1C[C@H]3CNC[C@@H](C3)C1)OCO2 ZINC000217740310 CD For-Sale Unstable MCHR1 18 41 COC(=O)[C@@H](O)CNC(=O)/C=C/c1ccc2c(c1)CCO2 ZINC000217740322 CC On-Demand Unstable GPR183 0 45 COc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217740359 GF For-Sale Unstable HTR1A 40 42 COc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217740359 GF For-Sale Unstable DRD2 45 44 COc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217740359 GF For-Sale Unstable DRD4 43 47 COc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217740359 GF For-Sale Unstable ADRA1D 15 50 COc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217740359 GF For-Sale Unstable ADRA1A 15 50 COc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217740359 GF For-Sale Unstable DRD3 46 44 COc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217740359 GF For-Sale Unstable EDNRB 39 41 COc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217740359 GF For-Sale Unstable EDNRA 41 43 COc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217740359 GF For-Sale Unstable BMP1 57 43 COc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217740359 GF For-Sale Unstable SIGMAR1 18 50 COc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217740359 GF For-Sale Unstable SSTR5 44 35 COc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217740359 GF For-Sale Unstable NOS2 42 32 COc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217740359 GF For-Sale Unstable SSTR3 72 31 COc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217740359 GF For-Sale Unstable FAAH 18 43 COc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217740359 GF For-Sale Unstable MCHR1 35 57 COc1ccccc1/C=C/NC(=O)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217740359 GF For-Sale Unstable CCR8 29 40 Cc1cc(C(=O)N2CCC(Oc3ccccc3F)CC2)cc(=O)[nH]1 ZINC000217740374 EF In-Stock Unstable GRIN2B 28 42 Cc1ccc(CNC(=O)CC(=N)N)cc1 ZINC000217740441 BC In-Stock Unstable TPSAB1 22 49 CCOC(=O)N1CCN(C(=O)N/C=C/c2ccccc2OC)CC1 ZINC000217740476 EE For-Sale Unstable P2RY12 50 36 CCOC(=O)N1CCN(C(=O)N/C=C/c2ccccc2OC)CC1 ZINC000217740476 EE For-Sale Unstable MTNR1B 15 41 O=C(c1ccccc1NS(=O)(=O)c1ccc(F)cc1)N1CCn2c1nc1ccccc12 ZINC000217740480 IH On-Demand Unstable PRTN3 56 36 O=C(c1ccccc1NS(=O)(=O)c1ccc(F)cc1)N1CCn2c1nc1ccccc12 ZINC000217740480 IH On-Demand Unstable PIK3C3 45 31 FC(F)(F)[C@@H]1CCCC[C@@H]1N[C@@H]1CCCc2cccnc21 ZINC000217740481 CI On-Demand Unstable CXCR4 52 37 COC(=O)[C@@H](O)CNC(=O)[C@H]1CCC(=O)N1 ZINC000217740532 BA For-Sale Unstable TRHR 51 36 N=C(N)CC(=O)NCc1ccccc1Cl ZINC000217740538 BD In-Stock Unstable P2RX7 67 50 N=C(N)CC(=O)NCc1ccccc1Cl ZINC000217740538 BD In-Stock Unstable SCN10A 22 42 FC(F)(F)[C@@H]1CCCC[C@H]1N[C@@H]1CCCc2cccnc21 ZINC000217740566 CI For-Sale Unstable CXCR4 52 37 CCC[C@H](O)CN[C@@H]1CCC[C@@H](NC(=O)OC(C)(C)C)C1 ZINC000217740572 DF On-Demand Unstable CTSK 0 40 CCC[C@H](O)CN[C@@H]1CCC[C@@H](NC(=O)OC(C)(C)C)C1 ZINC000217740572 DF On-Demand Unstable PGA5 42 39 COC(=O)[C@H](O)CNC(=O)[C@H]1CCC(=O)N1 ZINC000217740623 BA For-Sale Unstable TRHR 51 36 N=C(N)CC(=O)NCc1ccc(Cl)cc1 ZINC000217740637 BD In-Stock Unstable P2RX7 15 50 N=C(N)CC(=O)NCc1ccc(Cl)cc1 ZINC000217740637 BD In-Stock Unstable TPSAB1 22 49 N=C(N)CC(=O)NCc1ccc(Cl)cc1 ZINC000217740637 BD In-Stock Unstable AMP1_PLAFQ 17 45 N=C(N)CC(=O)NCc1ccc(Cl)cc1 ZINC000217740637 BD In-Stock Unstable NCE103 28 42 C[C@H](NC(=O)[C@@H]1CCCO1)c1cccc(/C=C\C(=O)O)c1 ZINC000217740667 CE For-Sale Unstable KCNQ2 45 34 Cc1ccc2[nH]c(CNC(=O)CC[C@@H]3NC(=O)c4ccccc4NC3=O)nc2c1 ZINC000217740715 GE In-Stock Unstable FABK 0 41 CCC[C@H](O)CN[C@H]1CCC[C@@H](NC(=O)OC(C)(C)C)C1 ZINC000217740728 DF On-Demand Unstable CTSK 0 40 CCC[C@H](O)CN[C@H]1CCC[C@@H](NC(=O)OC(C)(C)C)C1 ZINC000217740728 DF On-Demand Unstable PGA5 42 39 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccc(-c2ccc(F)cc2)cc1 ZINC000217740736 GI For-Sale Unstable HCRTR1 24 45 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccc(-c2ccc(F)cc2)cc1 ZINC000217740736 GI For-Sale Unstable IKBKB 15 41 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccc(-c2ccc(F)cc2)cc1 ZINC000217740736 GI For-Sale Unstable HCRTR2 17 45 N=C(N)CC(=O)NCc1ccc(Cl)cc1Cl ZINC000217740749 CD In-Stock Unstable P2RX7 82 53 N=C(N)CC(=O)NCc1ccc(Cl)cc1Cl ZINC000217740749 CD In-Stock Unstable EPHX2 16 46 N=C(N)CC(=O)NCc1ccc(Cl)cc1Cl ZINC000217740749 CD In-Stock Unstable ALPL 41 35 C[C@@H](NC(=O)[C@@H]1CCCO1)c1cccc(/C=C\C(=O)O)c1 ZINC000217740761 CE For-Sale Unstable KCNQ2 45 34 COc1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)c(OC)c1OC ZINC000217740783 HH On-Demand Unstable HTR2A 19 44 COc1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)c(OC)c1OC ZINC000217740783 HH On-Demand Unstable HRH1 21 40 COc1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)c(OC)c1OC ZINC000217740783 HH On-Demand Unstable SLC18A3 45 52 COc1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)c(OC)c1OC ZINC000217740783 HH On-Demand Unstable WNT3A 40 33 COc1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)c(OC)c1OC ZINC000217740783 HH On-Demand Unstable L3MBTL3 81 39 COc1ccccc1/C=C/NC(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217740784 EJ For-Sale Unstable P2RY1 29 44 COc1ccccc1/C=C/NC(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217740784 EJ For-Sale Unstable RAF1 23 42 COc1ccccc1/C=C/NC(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217740784 EJ For-Sale Unstable EPHX2 28 49 COc1ccccc1/C=C/NC(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217740784 EJ For-Sale Unstable KCNK3 46 36 O=C(c1cn(-c2ccccc2)nc1-c1ccccc1)N1CCn2c1nc1ccccc12 ZINC000217740807 HJ On-Demand Unstable CDK2 15 42 CC(C)[C@@H](NS(=O)(=O)c1cccnc1Cl)C(N)=O ZINC000217740825 CC On-Demand Unstable ADAMTS4 50 34 O=C(NC[C@H]1CCCN1c1nccs1)c1ccc(-c2ccc(F)cc2)cc1 ZINC000217740829 GI For-Sale Unstable HCRTR1 24 45 O=C(NC[C@H]1CCCN1c1nccs1)c1ccc(-c2ccc(F)cc2)cc1 ZINC000217740829 GI For-Sale Unstable IKBKB 15 41 O=C(NC[C@H]1CCCN1c1nccs1)c1ccc(-c2ccc(F)cc2)cc1 ZINC000217740829 GI For-Sale Unstable HCRTR2 17 45 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccccc2OC(C)C)CC(=O)O4)cc1O ZINC000217740830 JK In-Stock Unstable AKR1B1 0 44 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccccc2OC(C)C)CC(=O)O4)cc1O ZINC000217740830 JK In-Stock Unstable CYP1B1 56 36 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccccc2OC(C)C)CC(=O)O4)cc1O ZINC000217740830 JK In-Stock Unstable CYP1A1 39 44 COc1ccc(CNC(=O)CC(=N)N)cc1 ZINC000217740845 BC In-Stock Unstable ANPEP 17 47 COc1ccc(CNC(=O)CC(=N)N)cc1 ZINC000217740845 BC In-Stock Unstable BMP1 45 36 COc1ccc(CNC(=O)CC(=N)N)cc1 ZINC000217740845 BC In-Stock Unstable TRPV1 24 44 COc1ccc(CNC(=O)CC(=N)N)cc1 ZINC000217740845 BC In-Stock Unstable MMP13 28 40 COc1ccc(CNC(=O)CC(=N)N)cc1 ZINC000217740845 BC In-Stock Unstable MTNR1A 63 41 COc1ccc(CNC(=O)CC(=N)N)cc1 ZINC000217740845 BC In-Stock Unstable MTNR1B 52 37 COc1ccc(CNC(=O)CC(=N)N)cc1 ZINC000217740845 BC In-Stock Unstable MMP12 18 40 COc1ccc(CNC(=O)CC(=N)N)cc1 ZINC000217740845 BC In-Stock Unstable ACR 25 41 COc1ccc(CNC(=O)CC(=N)N)cc1 ZINC000217740845 BC In-Stock Unstable CA12 15 60 COc1ccc(CNC(=O)CC(=N)N)cc1 ZINC000217740845 BC In-Stock Unstable TPSAB1 22 45 COc1ccc(CNC(=O)CC(=N)N)cc1 ZINC000217740845 BC In-Stock Unstable CA9 26 60 COc1ccc(CNC(=O)CC(=N)N)cc1 ZINC000217740845 BC In-Stock Unstable PPO2 17 42 COc1ccc(CNC(=O)CC(=N)N)cc1 ZINC000217740845 BC In-Stock Unstable PROKR1 65 41 COC(=O)c1ccc(CN[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217740862 CD For-Sale Unstable SSTR3 17 42 COc1ccccc1/C=C/NC(=O)Nc1ccc(F)cc1F ZINC000217740894 DH For-Sale Unstable P2RY1 16 45 COc1ccccc1/C=C/NC(=O)Nc1ccc(F)cc1F ZINC000217740894 DH For-Sale Unstable PYGL 15 42 COc1ccccc1/C=C/NC(=O)Nc1ccc(F)cc1F ZINC000217740894 DH For-Sale Unstable SOAT1 15 48 COc1ccccc1/C=C/NC(=O)Nc1ccc(F)cc1F ZINC000217740894 DH For-Sale Unstable PDGFRA 15 42 COc1ccccc1/C=C/NC(=O)Nc1ccc(F)cc1F ZINC000217740894 DH For-Sale Unstable TLR4 17 40 CC(C)[C@H](NS(=O)(=O)c1cccnc1Cl)C(N)=O ZINC000217740906 CC On-Demand Unstable ADAMTS4 50 34 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccccc2OC(C)C)CC(=O)O4)cc1O ZINC000217740920 JK In-Stock Unstable AKR1B1 0 44 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccccc2OC(C)C)CC(=O)O4)cc1O ZINC000217740920 JK In-Stock Unstable CYP1B1 56 36 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccccc2OC(C)C)CC(=O)O4)cc1O ZINC000217740920 JK In-Stock Unstable CYP1A1 39 44 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccc(-c2cccc(Cl)c2)cc1 ZINC000217740934 GJ For-Sale Unstable ADAM17 16 43 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccc(-c2cccc(Cl)c2)cc1 ZINC000217740934 GJ For-Sale Unstable GRM5 15 43 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccc(-c2cccc(Cl)c2)cc1 ZINC000217740934 GJ For-Sale Unstable CACNA1I 45 36 Cc1nnc(CN(C)C(=O)c2ccc(-c3cccc(F)c3)cc2)o1 ZINC000217740945 EG In-Stock Unstable HSD17B2 16 47 Cc1nnc(CN(C)C(=O)c2ccc(-c3cccc(F)c3)cc2)o1 ZINC000217740945 EG In-Stock Unstable LIMK2 24 40 COC(=O)c1ccc(CN[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217740947 CD For-Sale Unstable SSTR3 17 42 C[C@@H](NC(=O)CC(=N)N)c1ccccc1 ZINC000217740952 BD In-Stock Unstable KCNA5 23 42 C[C@@H](NC(=O)CC(=N)N)c1ccccc1 ZINC000217740952 BD In-Stock Unstable ACACA 42 41 C[C@@H](NC(=O)CC(=N)N)c1ccccc1 ZINC000217740952 BD In-Stock Unstable CTSK 32 40 C[C@@H](NC(=O)CC(=N)N)c1ccccc1 ZINC000217740952 BD In-Stock Unstable C3AR1 58 37 C[C@@H](NC(=O)CC(=N)N)c1ccccc1 ZINC000217740952 BD In-Stock Unstable F7 32 47 C[C@@H](NC(=O)CC(=N)N)c1ccccc1 ZINC000217740952 BD In-Stock Unstable AOC3 19 40 O=C(NC[C@H]1CCCN1c1nccs1)c1ccc(-c2cccc(Cl)c2)cc1 ZINC000217741016 GJ For-Sale Unstable ADAM17 16 43 O=C(NC[C@H]1CCCN1c1nccs1)c1ccc(-c2cccc(Cl)c2)cc1 ZINC000217741016 GJ For-Sale Unstable GRM5 15 43 O=C(NC[C@H]1CCCN1c1nccs1)c1ccc(-c2cccc(Cl)c2)cc1 ZINC000217741016 GJ For-Sale Unstable CACNA1I 45 36 COc1ccccc1/C=C/NC(=O)Nc1cc(F)ccc1F ZINC000217741020 DH For-Sale Unstable PDGFRA 18 42 COc1ccccc1/C=C/NC(=O)Nc1cc(F)ccc1F ZINC000217741020 DH For-Sale Unstable TLR4 16 40 C[C@H](NC(=O)CC(=N)N)c1ccccc1 ZINC000217741063 BD In-Stock Unstable KCNA5 23 42 C[C@H](NC(=O)CC(=N)N)c1ccccc1 ZINC000217741063 BD In-Stock Unstable ACACA 42 41 C[C@H](NC(=O)CC(=N)N)c1ccccc1 ZINC000217741063 BD In-Stock Unstable CTSK 32 40 C[C@H](NC(=O)CC(=N)N)c1ccccc1 ZINC000217741063 BD In-Stock Unstable C3AR1 58 37 C[C@H](NC(=O)CC(=N)N)c1ccccc1 ZINC000217741063 BD In-Stock Unstable F7 32 47 C[C@H](NC(=O)CC(=N)N)c1ccccc1 ZINC000217741063 BD In-Stock Unstable AOC3 19 40 FC(F)(F)[C@@H]1CCC[C@@H](N[C@@H]2CCCc3cccnc32)C1 ZINC000217741071 CI On-Demand Unstable CXCR4 58 36 COc1cccc(-c2ccc(C(=O)NC[C@@H]3CCCN3c3nccs3)cc2)c1 ZINC000217741124 GI For-Sale Unstable DRD4 43 34 COc1cccc(-c2ccc(C(=O)NC[C@@H]3CCCN3c3nccs3)cc2)c1 ZINC000217741124 GI For-Sale Unstable ACKR3 51 32 COc1ccccc1/C=C/NC(=O)N1CCCC[C@@H]1CCO ZINC000217741136 DF For-Sale Unstable ACKR3 67 35 FC(F)(F)[C@@H]1CCC[C@H](N[C@@H]2CCCc3cccnc32)C1 ZINC000217741160 CI On-Demand Unstable CXCR4 58 36 FCc1cc2cn[nH]c2cn1 ZINC000217741168 AD For-Sale Unstable JAK2 15 42 N=C(N)CC(=O)NCCc1ccccc1 ZINC000217741180 BC In-Stock Unstable CA2 19 55 N=C(N)CC(=O)NCCc1ccccc1 ZINC000217741180 BC In-Stock Unstable SCNN1A 23 42 N=C(N)CC(=O)NCCc1ccccc1 ZINC000217741180 BC In-Stock Unstable CA1 19 55 N=C(N)CC(=O)NCCc1ccccc1 ZINC000217741180 BC In-Stock Unstable CA7 19 55 N=C(N)CC(=O)NCCc1ccccc1 ZINC000217741180 BC In-Stock Unstable CPA1 24 43 N=C(N)CC(=O)NCCc1ccccc1 ZINC000217741180 BC In-Stock Unstable NPFFR2 58 37 N=C(N)CC(=O)NCCc1ccccc1 ZINC000217741180 BC In-Stock Unstable CA5B 41 55 N=C(N)CC(=O)NCCc1ccccc1 ZINC000217741180 BC In-Stock Unstable CA5A 41 55 N=C(N)CC(=O)NCCc1ccccc1 ZINC000217741180 BC In-Stock Unstable SCN5A 0 48 N=C(N)CC(=O)NCCc1ccccc1 ZINC000217741180 BC In-Stock Unstable CA9 15 45 N=C(N)CC(=O)NCCc1ccccc1 ZINC000217741180 BC In-Stock Unstable AMP1_PLAFQ 44 50 N=C(N)CC(=O)NCCc1ccccc1 ZINC000217741180 BC In-Stock Unstable NCE103 34 50 N=C(N)CC(=O)NCCc1ccccc1 ZINC000217741180 BC In-Stock Unstable POLG_WNV 52 34 N=C(N)CC(=O)NCCc1ccccc1 ZINC000217741180 BC In-Stock Unstable CRTM 35 40 N=C(N)CC(=O)NCCc1ccccc1 ZINC000217741180 BC In-Stock Unstable P96878_MYCTU 21 50 N=C(N)CC(=O)NCCc1ccccc1 ZINC000217741180 BC In-Stock Unstable NPFFR1 61 37 CN(CCS(C)(=O)=O)c1ccc(CBr)cc1[N+](=O)[O-] ZINC000217741188 FD For-Sale Unstable MDAA 0 47 COc1ccccc1/C=C/NC(=O)N1CCCC[C@H]1CCO ZINC000217741216 DF For-Sale Unstable ACKR3 67 35 COc1cccc(-c2ccc(C(=O)NC[C@H]3CCCN3c3nccs3)cc2)c1 ZINC000217741219 GI For-Sale Unstable DRD4 43 34 COc1cccc(-c2ccc(C(=O)NC[C@H]3CCCN3c3nccs3)cc2)c1 ZINC000217741219 GI For-Sale Unstable ACKR3 51 32 COC(=O)[C@H](N[C@@H]1CCN(C)C1)c1ccccc1 ZINC000217741223 BD For-Sale Unstable SLC6A1 39 43 COC(=O)[C@H](N[C@@H]1CCN(C)C1)c1ccccc1 ZINC000217741223 BD For-Sale Unstable SLC6A3 38 51 COc1ccc(CCNC(=O)CC(=N)N)cc1 ZINC000217741301 BC In-Stock Unstable CA2 19 50 COc1ccc(CCNC(=O)CC(=N)N)cc1 ZINC000217741301 BC In-Stock Unstable SCNN1A 38 41 COc1ccc(CCNC(=O)CC(=N)N)cc1 ZINC000217741301 BC In-Stock Unstable BMP1 48 40 COc1ccc(CCNC(=O)CC(=N)N)cc1 ZINC000217741301 BC In-Stock Unstable CA1 19 51 COc1ccc(CCNC(=O)CC(=N)N)cc1 ZINC000217741301 BC In-Stock Unstable CTSL 0 41 COc1ccc(CCNC(=O)CC(=N)N)cc1 ZINC000217741301 BC In-Stock Unstable MTNR1A 78 45 COc1ccc(CCNC(=O)CC(=N)N)cc1 ZINC000217741301 BC In-Stock Unstable MTNR1B 68 44 COc1ccc(CCNC(=O)CC(=N)N)cc1 ZINC000217741301 BC In-Stock Unstable MMP12 16 45 COc1ccc(CCNC(=O)CC(=N)N)cc1 ZINC000217741301 BC In-Stock Unstable ACR 19 40 COc1ccc(CCNC(=O)CC(=N)N)cc1 ZINC000217741301 BC In-Stock Unstable CA12 17 61 COc1ccc(CCNC(=O)CC(=N)N)cc1 ZINC000217741301 BC In-Stock Unstable PTGDR 24 44 COc1ccc(CCNC(=O)CC(=N)N)cc1 ZINC000217741301 BC In-Stock Unstable CA9 29 61 COc1ccc(CCNC(=O)CC(=N)N)cc1 ZINC000217741301 BC In-Stock Unstable MMP1 22 50 COc1ccc(CCNC(=O)CC(=N)N)cc1 ZINC000217741301 BC In-Stock Unstable AOC3 15 41 COc1ccc(CCNC(=O)CC(=N)N)cc1 ZINC000217741301 BC In-Stock Unstable PPO2 33 45 COc1ccc(CCNC(=O)CC(=N)N)cc1 ZINC000217741301 BC In-Stock Unstable NCE103 26 43 COc1ccc(CCNC(=O)CC(=N)N)cc1 ZINC000217741301 BC In-Stock Unstable PROKR1 63 39 COc1ccc(CCNC(=O)CC(=N)N)cc1 ZINC000217741301 BC In-Stock Unstable P96878_MYCTU 15 43 COC(=O)[C@H](N[C@H]1CCN(C)C1)c1ccccc1 ZINC000217741304 BD For-Sale Unstable SLC6A1 39 43 COC(=O)[C@H](N[C@H]1CCN(C)C1)c1ccccc1 ZINC000217741304 BD For-Sale Unstable SLC6A3 38 51 O[C@@H]1CCC[C@@H](N[C@@H]2CCCc3cccnc32)C1 ZINC000217741352 BE On-Demand Unstable CXCR4 54 35 O=C(O)/C=C\c1cnc(NC(=O)CC2CCCCC2)s1 ZINC000217741398 CG For-Sale Unstable CDK5 54 46 CN1CC[C@@H](N[C@@H](C(=O)O)c2ccccc2)C1 ZINC000217741414 BD For-Sale Unstable SLC6A1 33 40 CN1CC[C@@H](N[C@@H](C(=O)O)c2ccccc2)C1 ZINC000217741414 BD For-Sale Unstable SLC6A3 27 45 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccccn2)CC1 ZINC000217741419 EF For-Sale Unstable EBP 26 44 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccccn2)CC1 ZINC000217741419 EF For-Sale Unstable SSTR1 22 41 COc1ccccc1/C=C/NC(=O)N1CCN(c2ccccn2)CC1 ZINC000217741419 EF For-Sale Unstable SLC6A7 0 43 COc1ccc(CCNC(=O)CC(=N)N)cc1OC ZINC000217741424 CC In-Stock Unstable TRPV1 39 50 COc1ccc(CCNC(=O)CC(=N)N)cc1OC ZINC000217741424 CC In-Stock Unstable MTNR1A 43 36 COc1ccc(CCNC(=O)CC(=N)N)cc1OC ZINC000217741424 CC In-Stock Unstable MTNR1B 42 42 COc1ccc(CCNC(=O)CC(=N)N)cc1OC ZINC000217741424 CC In-Stock Unstable IAP 0 45 COc1ccc(CCNC(=O)CC(=N)N)cc1OC ZINC000217741424 CC In-Stock Unstable MT-ND1 26 41 COc1ccc(CCNC(=O)CC(=N)N)cc1OC ZINC000217741424 CC In-Stock Unstable CA9 20 43 COc1ccc(CCNC(=O)CC(=N)N)cc1OC ZINC000217741424 CC In-Stock Unstable NCE103 25 62 COc1ccc(CCNC(=O)CC(=N)N)cc1OC ZINC000217741424 CC In-Stock Unstable ABCG2 15 49 COc1ccc(CCNC(=O)CC(=N)N)cc1OC ZINC000217741424 CC In-Stock Unstable ENPP1 54 31 COc1ccc(CCNC(=O)CC(=N)N)cc1OC ZINC000217741424 CC In-Stock Unstable P96878_MYCTU 17 62 COc1ccc(CCNC(=O)CC(=N)N)cc1OC ZINC000217741424 CC In-Stock Unstable SCMU_MYCTU 0 43 COc1ccc(CCNC(=O)CC(=N)N)cc1OC ZINC000217741424 CC In-Stock Unstable CAN2 0 62 O=C(c1cccc(=O)[nH]1)N1CCCN(C2CCCCC2)CC1 ZINC000217741435 DD In-Stock Unstable HRH3 25 49 O=C(c1cccc(=O)[nH]1)N1CCCN(C2CCCCC2)CC1 ZINC000217741435 DD In-Stock Unstable L3MBTL3 90 46 O[C@@H]1CCC[C@H](N[C@@H]2CCCc3cccnc32)C1 ZINC000217741446 BE On-Demand Unstable CXCR4 54 35 COc1ccc(CCNC(=O)CN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@H]23)cc1 ZINC000217741470 IG In-Stock Unstable SCN9A 0 46 COc1ccc(CCNC(=O)CN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@H]23)cc1 ZINC000217741470 IG In-Stock Unstable MTNR1A 44 37 COc1ccc(CCNC(=O)CN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@H]23)cc1 ZINC000217741470 IG In-Stock Unstable CA9 15 42 CN1CC[C@H](N[C@@H](C(=O)O)c2ccccc2)C1 ZINC000217741498 BD For-Sale Unstable SLC6A1 33 40 CN1CC[C@H](N[C@@H](C(=O)O)c2ccccc2)C1 ZINC000217741498 BD For-Sale Unstable SLC6A3 27 45 CC(C)(C)c1cc(C(=O)NC[C@@H]2CCCN2c2nccs2)cc(C(C)(C)C)c1 ZINC000217741552 GK For-Sale Unstable CACNA1I 66 39 COc1ccc(CCNC(=O)CN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@@H]23)cc1 ZINC000217741556 IG In-Stock Unstable SCN9A 0 46 COc1ccc(CCNC(=O)CN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@@H]23)cc1 ZINC000217741556 IG In-Stock Unstable MTNR1A 44 37 COc1ccc(CCNC(=O)CN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@@H]23)cc1 ZINC000217741556 IG In-Stock Unstable CA9 15 42 c1cnc2c(c1)CCC[C@@H]2N[C@@H]1CCN2CCC[C@@H]12 ZINC000217741568 CE For-Sale Unstable CXCR4 52 36 CS(=O)(=O)CN1C(=O)c2ccccc2C1=O ZINC000217741606 BC In-Stock Unstable ALDH1A1 54 38 CS(=O)(=O)CN1C(=O)c2ccccc2C1=O ZINC000217741606 BC In-Stock Unstable FBPC 0 43 CC(C)(C)c1cc(C(=O)NC[C@H]2CCCN2c2nccs2)cc(C(C)(C)C)c1 ZINC000217741627 GK For-Sale Unstable CACNA1I 66 39 O=C(O)/C=C\c1cnc(NC(=O)c2cccc(F)c2)s1 ZINC000217741651 CF For-Sale Anodyne SCD1 30 41 O=C(O)/C=C\c1cnc(NC(=O)c2cccc(F)c2)s1 ZINC000217741651 CF For-Sale Anodyne SCD 0 41 O=C(O)/C=C\c1cnc(NC(=O)c2cccc(F)c2)s1 ZINC000217741651 CF For-Sale Anodyne KCNK3 49 46 O=C(O)/C=C\c1cnc(NC(=O)c2cccc(F)c2)s1 ZINC000217741651 CF For-Sale Anodyne KCNK9 32 43 Cc1cccc(C#Cc2ccc(-c3ccnn3C)cc2)n1 ZINC000217741693 CG For-Sale Unstable GRM5 25 55 c1cnc2c(c1)CCC[C@@H]2N[C@H]1CCN2CCC[C@@H]12 ZINC000217741718 CE For-Sale Unstable CXCR4 52 36 O=C(O)/C=C\c1cnc(NC(=O)Cc2ccccc2F)s1 ZINC000217741741 DF For-Sale Unstable CDK5 51 47 O=C(/C=C\c1ccc(F)cc1)Nc1cnccc1C(=O)O ZINC000217741775 CF For-Sale Anodyne MMP2 0 50 O=C(/C=C\c1ccc(F)cc1)Nc1cnccc1C(=O)O ZINC000217741775 CF For-Sale Anodyne HDAC1 0 47 O=C(/C=C\c1ccc(F)cc1)Nc1cnccc1C(=O)O ZINC000217741775 CF For-Sale Anodyne MMP9 0 50 O=C(/C=C\c1ccc(F)cc1)Nc1cnccc1C(=O)O ZINC000217741775 CF For-Sale Anodyne HPSE 40 36 O=C(/C=C\c1ccc(F)cc1)Nc1cnccc1C(=O)O ZINC000217741775 CF For-Sale Anodyne MMP1 23 50 Cc1cccc(C#Cc2ccc(-c3ccn(C)n3)cc2)n1 ZINC000217741798 CG For-Sale Unstable GRM5 26 56 O=C(O)/C=C\c1cnc(NC(=O)Cc2ccc(F)cc2)s1 ZINC000217741833 DF For-Sale Unstable CDK5 45 49 C[C@@H]1CN(C)CCN1S(=O)(=O)c1cnc(Cl)c(Cl)c1 ZINC000217741843 DD For-Sale Unstable HSD11B1 16 43 N=C(N)CC(=O)NCc1cccnc1 ZINC000217741848 AC In-Stock Unstable NAMPT 68 49 COC(=O)CNC(=O)N/C=C/c1ccccc1OC ZINC000217741876 CD For-Sale Unstable CYP1B1 19 40 COC(=O)CNC(=O)N/C=C/c1ccccc1OC ZINC000217741876 CD For-Sale Unstable TLR4 19 45 C[C@H]1CN(C)CCN1S(=O)(=O)c1cnc(Cl)c(Cl)c1 ZINC000217741921 DD For-Sale Unstable HSD11B1 16 43 O=C(CNS(=O)(=O)c1cccc(Cl)c1)NC[C@@H]1CCCN1c1nccs1 ZINC000217741937 HD For-Sale Unstable ADAMTS5 27 45 Cc1ccccc1NC(=O)CC(=N)N ZINC000217741959 AD In-Stock Unstable DDX3X 0 45 COC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217741993 EG For-Sale Unstable PPIA 20 48 COC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217741993 EG For-Sale Unstable IMPDH2 0 42 COC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217741993 EG For-Sale Unstable AKR1C3 19 40 COC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217741993 EG For-Sale Unstable KCNK3 104 45 COC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217741993 EG For-Sale Unstable KCNK9 78 44 Cc1cccc(C#Cc2ccc(-c3nn(C)cc3Br)cc2)n1 ZINC000217742014 FH For-Sale Unstable GRM5 21 51 O=C(CNS(=O)(=O)c1cccc(Cl)c1)NC[C@H]1CCCN1c1nccs1 ZINC000217742017 HD For-Sale Unstable ADAMTS5 27 45 C[C@@H]1CN(C)CCN1S(=O)(=O)c1cccnc1Cl ZINC000217742027 CD For-Sale Unstable HSD11B1 17 42 COC(=O)[C@@H](O)CNC(=O)COc1cccc(Cl)c1 ZINC000217742065 CC On-Demand Unstable PDS 80 43 Cc1cccc(NC(=O)CC(=N)N)c1 ZINC000217742069 AD In-Stock Unstable CCKAR 24 46 Cc1cccc(NC(=O)CC(=N)N)c1 ZINC000217742069 AD In-Stock Unstable F2R 0 49 Cc1cccc(NC(=O)CC(=N)N)c1 ZINC000217742069 AD In-Stock Unstable F12 0 44 Cc1cccc(NC(=O)CC(=N)N)c1 ZINC000217742069 AD In-Stock Unstable SLC1A2 42 32 Cc1cccc(NC(=O)CC(=N)N)c1 ZINC000217742069 AD In-Stock Unstable NAMPT 0 43 Cc1cccc(NC(=O)CC(=N)N)c1 ZINC000217742069 AD In-Stock Unstable PARP14 48 39 Cc1cccc(NC(=O)CC(=N)N)c1 ZINC000217742069 AD In-Stock Unstable PARP15 53 39 Cc1cccc(NC(=O)CC(=N)N)c1 ZINC000217742069 AD In-Stock Unstable PSBA 0 54 Cc1cccc(NC(=O)CC(=N)N)c1 ZINC000217742069 AD In-Stock Unstable KCNK3 92 50 Cc1cccc(NC(=O)CC(=N)N)c1 ZINC000217742069 AD In-Stock Unstable KCNK9 92 50 Cc1cccc(NC(=O)CC(=N)N)c1 ZINC000217742069 AD In-Stock Unstable PARP10 0 48 CCOC(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217742101 FG For-Sale Unstable ACR 20 40 C[C@H]1CN(C)CCN1S(=O)(=O)c1cccnc1Cl ZINC000217742108 CD For-Sale Unstable HSD11B1 17 42 CN[C@H]1Cc2ccc(Br)cc2C1 ZINC000217742113 BE For-Sale Unstable PNMT 21 50 COC(=O)[C@H](O)CNC(=O)COc1cccc(Cl)c1 ZINC000217742144 CC On-Demand Unstable PDS 80 43 CCC[C@@H](O)CNCCC(C)C ZINC000217742158 AD For-Sale Unstable Q8WS26_TRYCR 34 47 CCC[C@@H](O)CNCCC(C)C ZINC000217742158 AD For-Sale Unstable FPPS 0 47 CC1(C)[C@H]2CC[C@@]1(CS(=O)(=O)N1CC(N3C(=O)[C@H]4CC=CC[C@H]4C3=O)C1)C(=O)C2 ZINC000217742181 HD In-Stock Unstable CA5B 25 42 CC1(C)[C@H]2CC[C@@]1(CS(=O)(=O)N1CC(N3C(=O)[C@H]4CC=CC[C@H]4C3=O)C1)C(=O)C2 ZINC000217742181 HD In-Stock Unstable CA5A 27 42 CC1(C)[C@H]2CC[C@@]1(CS(=O)(=O)N1CC(N3C(=O)[C@H]4CC=CC[C@H]4C3=O)C1)C(=O)C2 ZINC000217742181 HD In-Stock Unstable CXCR3 16 51 Cc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217742189 AD In-Stock Unstable LTA4H 0 49 Cc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217742189 AD In-Stock Unstable ACR 55 50 Cc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217742189 AD In-Stock Unstable PPO2 24 41 Cc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217742189 AD In-Stock Unstable PSBA 0 48 COC(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2OC)cc1 ZINC000217742219 EF For-Sale Unstable ACR 20 40 CCOC(=O)c1ccc(S(N)(=O)=O)s1 ZINC000217742235 BC On-Demand Unstable CA2 30 48 CCOC(=O)c1ccc(S(N)(=O)=O)s1 ZINC000217742235 BC On-Demand Unstable CA14 0 44 CCC[C@H](O)CNCCC(C)C ZINC000217742250 AD For-Sale Unstable Q8WS26_TRYCR 34 47 CCC[C@H](O)CNCCC(C)C ZINC000217742250 AD For-Sale Unstable FPPS 0 47 COC(=O)Nc1ccc(S(=O)(=O)N2CC(N3C(=O)[C@H]4CC=CC[C@H]4C3=O)C2)cc1 ZINC000217742278 HD In-Stock Unstable TGM2 47 35 COC(=O)Nc1ccc(S(=O)(=O)N2CC(N3C(=O)[C@H]4CC=CC[C@H]4C3=O)C2)cc1 ZINC000217742278 HD In-Stock Unstable F13A1 76 39 O=S(=O)(NCCN1CCSCC1)c1cccnc1Cl ZINC000217742346 DD On-Demand Unstable HTR7 28 45 COC(=O)Nc1ccc(S(=O)(=O)N2CC(N3C(=O)[C@H]4CC=CC[C@@H]4C3=O)C2)cc1 ZINC000217742373 HD In-Stock Unstable TGM2 47 35 COC(=O)Nc1ccc(S(=O)(=O)N2CC(N3C(=O)[C@H]4CC=CC[C@@H]4C3=O)C2)cc1 ZINC000217742373 HD In-Stock Unstable F13A1 76 39 COC(=O)[C@@H](O)CNC(=O)[C@@H](C)Oc1ccccc1C#N ZINC000217742418 CB On-Demand Unstable ADRB1 47 37 COC(=O)Nc1ccc(S(=O)(=O)N2CC(N3C(=O)[C@@H]4CC=CC[C@H]4C3=O)C2)cc1 ZINC000217742459 HD In-Stock Unstable TGM2 47 35 COC(=O)Nc1ccc(S(=O)(=O)N2CC(N3C(=O)[C@@H]4CC=CC[C@H]4C3=O)C2)cc1 ZINC000217742459 HD In-Stock Unstable F13A1 76 39 COC(=O)[C@H](O)CNC(=O)[C@@H](C)Oc1ccccc1C#N ZINC000217742506 CB On-Demand Unstable ADRB1 47 37 COC(=O)[C@@H](O)CNC(=O)[C@H](C)Oc1ccccc1C#N ZINC000217742587 CB On-Demand Unstable ADRB1 47 37 CC(C)(C)[C@@H]1CC[C@@H](N)[C@@H](Cc2cc(F)ccc2F)C1 ZINC000217742590 CI For-Sale Unstable DPP4 19 41 Cc1n[nH]c([C@H]2CCCN2C(=O)c2cc(C)oc2C)n1 ZINC000217742620 CE In-Stock Unstable COLA 51 42 Cc1n[nH]c([C@H]2CCCN2C(=O)c2cc(C)oc2C)n1 ZINC000217742620 CE In-Stock Unstable CPT1A 45 42 CC1(C)C[C@@H]1CNS(=O)(=O)c1cccnc1Cl ZINC000217742623 CE On-Demand Unstable G2YM83_BOTF4 51 35 Cc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)N1CCn2c1nc1ccccc12 ZINC000217742635 IG On-Demand Unstable GNRHR 30 40 Cc1cccc(C)c1NC(=O)CC(=N)N ZINC000217742650 BD In-Stock Unstable S1PR4 33 40 COc1ccccc1/C=C/NC(=O)NCc1cccc(C)c1 ZINC000217742667 CG For-Sale Unstable PTGER2 28 40 COc1ccccc1/C=C/NC(=O)NCc1cccc(C)c1 ZINC000217742667 CG For-Sale Unstable PTGER4 0 40 COc1ccccc1/C=C/NC(=O)NCc1cccc(C)c1 ZINC000217742667 CG For-Sale Unstable ROCK2 27 43 COc1ccccc1/C=C/NC(=O)NCc1cccc(C)c1 ZINC000217742667 CG For-Sale Unstable KCNK3 42 40 COc1ccccc1/C=C/NC(=O)NCc1cccc(C)c1 ZINC000217742667 CG For-Sale Unstable KCNK9 45 40 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](C(C)C)CC(=O)O4)cc1O ZINC000217742672 GH In-Stock Unstable AKR1B1 23 50 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](C(C)C)CC(=O)O4)cc1O ZINC000217742672 GH In-Stock Unstable CYP1B1 59 37 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](C(C)C)CC(=O)O4)cc1O ZINC000217742672 GH In-Stock Unstable CYP1A1 45 50 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](C(C)C)CC(=O)O4)cc1O ZINC000217742672 GH In-Stock Unstable CYP1A2 36 41 CC(C)(C)[C@H]1CC[C@@H](N)[C@@H](Cc2cc(F)ccc2F)C1 ZINC000217742681 CI For-Sale Unstable DPP4 19 41 COC(=O)[C@H](O)CNC(=O)[C@H](C)Oc1ccccc1C#N ZINC000217742682 CB On-Demand Unstable ADRB1 47 37 O=C(O)/C=C\c1ccc(NC(=O)c2ccccn2)c(F)c1 ZINC000217742684 CF For-Sale Anodyne GRM4 71 55 O=C(O)/C=C\c1ccc(NC(=O)c2ccccn2)c(F)c1 ZINC000217742684 CF For-Sale Anodyne MMP2 0 43 O=C(O)/C=C\c1ccc(NC(=O)c2ccccn2)c(F)c1 ZINC000217742684 CF For-Sale Anodyne MMP9 0 43 O=C(O)/C=C\c1ccc(NC(=O)c2ccccn2)c(F)c1 ZINC000217742684 CF For-Sale Anodyne MMP1 0 43 Cc1cc(Cl)c(F)c([C@H](CN)CC(=O)O)c1 ZINC000217742688 BE For-Sale Unstable HMGCR 32 43 Cc1n[nH]c([C@@H]2CCCN2C(=O)c2cc(C)oc2C)n1 ZINC000217742707 CE In-Stock Unstable COLA 51 42 Cc1n[nH]c([C@@H]2CCCN2C(=O)c2cc(C)oc2C)n1 ZINC000217742707 CE In-Stock Unstable CPT1A 45 42 CC1(C)C[C@H]1CNS(=O)(=O)c1cccnc1Cl ZINC000217742721 CE On-Demand Unstable G2YM83_BOTF4 51 35 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](C(C)C)CC(=O)O4)cc1O ZINC000217742736 GH In-Stock Unstable AKR1B1 23 50 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](C(C)C)CC(=O)O4)cc1O ZINC000217742736 GH In-Stock Unstable CYP1B1 59 37 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](C(C)C)CC(=O)O4)cc1O ZINC000217742736 GH In-Stock Unstable CYP1A1 45 50 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](C(C)C)CC(=O)O4)cc1O ZINC000217742736 GH In-Stock Unstable CYP1A2 36 41 CCc1cccc(C)c1NC(=O)CC(=N)N ZINC000217742763 BD In-Stock Unstable S1PR4 25 44 CC(C)(C)[C@@H]1CC[C@H](N)[C@@H](Cc2cc(F)ccc2F)C1 ZINC000217742764 CI For-Sale Unstable DPP4 19 41 Cc1cc(Cl)c(F)c([C@@H](CN)CC(=O)O)c1 ZINC000217742770 BE For-Sale Unstable HMGCR 32 43 Cc1cc(NC(=O)c2ccnn2C)ccc1/C=C\C(=O)O ZINC000217742771 CE For-Sale Unstable FLT1 15 41 Cc1cc(NC(=O)c2ccnn2C)ccc1/C=C\C(=O)O ZINC000217742771 CE For-Sale Unstable KCNK3 49 36 COc1cccc(CNC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217742782 DG For-Sale Unstable DRD4 41 32 COc1cccc(CNC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217742782 DG For-Sale Unstable CYP1B1 42 46 COc1cccc(CNC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217742782 DG For-Sale Unstable ROCK1 39 44 COc1cccc(CNC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217742782 DG For-Sale Unstable MTNR1A 52 47 COc1cccc(CNC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217742782 DG For-Sale Unstable MTNR1B 55 47 COc1cccc(CNC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217742782 DG For-Sale Unstable ROCK2 52 48 COc1cccc(CNC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217742782 DG For-Sale Unstable ABCB1 16 42 COc1cccc(CNC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217742782 DG For-Sale Unstable PDS 52 41 COC(=O)[C@@H](O)CNC(=O)CCOc1cccc(Cl)c1 ZINC000217742787 DC On-Demand Unstable MTNR1A 25 41 COC(=O)[C@@H](O)CNC(=O)CCOc1cccc(Cl)c1 ZINC000217742787 DC On-Demand Unstable MTNR1B 22 41 COC(=O)[C@@H](O)CNC(=O)CCOc1cccc(Cl)c1 ZINC000217742787 DC On-Demand Unstable PDS 60 42 CC(C)(C)[C@H]1CC[C@H](N)[C@@H](Cc2cc(F)ccc2F)C1 ZINC000217742837 CI For-Sale Unstable DPP4 19 41 Cc1ccc(NC(=O)CC(=N)N)cc1C ZINC000217742855 BD In-Stock Unstable SLC1A3 40 38 Cc1ccc(NC(=O)CC(=N)N)cc1C ZINC000217742855 BD In-Stock Unstable SLC1A2 51 39 Cc1ccc(NC(=O)CC(=N)N)cc1C ZINC000217742855 BD In-Stock Unstable ENPP1 58 36 Cc1cc(NC(=O)c2cnn(C)c2)ccc1/C=C\C(=O)O ZINC000217742861 CE For-Sale Unstable PRNP 48 32 Cc1cc(NC(=O)c2cnn(C)c2)ccc1/C=C\C(=O)O ZINC000217742861 CE For-Sale Unstable KCNK3 86 37 Cc1cc(NC(=O)c2cnn(C)c2)ccc1/C=C\C(=O)O ZINC000217742861 CE For-Sale Unstable KCNK9 41 37 C[C@H](F)c1ccc(C[C@H](N)C(=O)O)c(Cl)c1 ZINC000217742874 BE For-Sale Unstable CACNA2D1 37 43 C[C@H](F)c1ccc(C[C@H](N)C(=O)O)c(Cl)c1 ZINC000217742874 BE For-Sale Unstable TPH1 41 37 COc1ccccc1/C=C/NC(=O)NCc1cccc(F)c1 ZINC000217742893 DG For-Sale Unstable GRIN2B 23 42 COc1ccccc1/C=C/NC(=O)NCc1cccc(F)c1 ZINC000217742893 DG For-Sale Unstable ROCK2 22 41 COc1ccccc1/C=C/NC(=O)NCc1cccc(F)c1 ZINC000217742893 DG For-Sale Unstable ACKR3 44 31 COc1ccc(C(=O)NC[C@@]23C[C@@H]4C[C@@](C)(C[C@@](C)(C4)C2)C3)cc1 ZINC000217742909 EI In-Stock Unstable P2RX7 22 52 O[C@@H]1CCCC[C@@H]1N[C@@H]1CCCc2cccnc21 ZINC000217742925 BE On-Demand Unstable CXCR4 60 34 CCCCCC(=O)Nc1ccc(/C=C\C(=O)O)c(C)c1 ZINC000217742935 CH For-Sale Unstable HDAC10 19 44 CCCCCC(=O)Nc1ccc(/C=C\C(=O)O)c(C)c1 ZINC000217742935 CH For-Sale Unstable HDAC3 27 52 CCCCCC(=O)Nc1ccc(/C=C\C(=O)O)c(C)c1 ZINC000217742935 CH For-Sale Unstable ENPP2 32 45 C[C@@H](F)c1ccc(C[C@H](N)C(=O)O)c(Cl)c1 ZINC000217742951 BE For-Sale Unstable CACNA2D1 37 43 C[C@@H](F)c1ccc(C[C@H](N)C(=O)O)c(Cl)c1 ZINC000217742951 BE For-Sale Unstable TPH1 41 37 O[C@@H]1CCCC[C@H]1N[C@@H]1CCCc2cccnc21 ZINC000217743004 BE On-Demand Unstable CXCR4 60 34 COc1ccccc1/C=C/NC(=O)NCc1cccc(Cl)c1 ZINC000217743005 DH For-Sale Unstable ROCK2 21 41 COc1ccccc1/C=C/NC(=O)NCc1cccc(Cl)c1 ZINC000217743005 DH For-Sale Unstable PDS 55 38 C[C@H](F)c1ccc(C[C@@H](N)C(=O)O)c(Cl)c1 ZINC000217743034 BE For-Sale Unstable CACNA2D1 37 43 C[C@H](F)c1ccc(C[C@@H](N)C(=O)O)c(Cl)c1 ZINC000217743034 BE For-Sale Unstable TPH1 41 37 COC[C@@H]1CCCN(S(=O)(=O)c2cccnc2Cl)C1 ZINC000217743072 DD On-Demand Unstable CASP3 44 32 COC[C@@H]1CCCN(S(=O)(=O)c2cccnc2Cl)C1 ZINC000217743072 DD On-Demand Unstable CASP7 48 33 CCc1ccccc1NC(=O)CC(=N)N ZINC000217743080 BD In-Stock Unstable KCNQ2 62 38 CCS(=O)(=O)CNC=O ZINC000217743096 AB In-Stock Unstable ADH1A 0 45 CCS(=O)(=O)CNC=O ZINC000217743096 AB In-Stock Unstable ADH7 0 40 CCS(=O)(=O)CNC=O ZINC000217743096 AB In-Stock Unstable ADH1B 0 45 C[C@@H](F)c1ccc(C[C@@H](N)C(=O)O)c(Cl)c1 ZINC000217743112 BE For-Sale Unstable CACNA2D1 37 43 C[C@@H](F)c1ccc(C[C@@H](N)C(=O)O)c(Cl)c1 ZINC000217743112 BE For-Sale Unstable TPH1 41 37 COC(=O)[C@@H](O)CNC(=O)/C=C/c1cccnc1 ZINC000217743144 CB On-Demand Unstable MMP2 17 41 COC(=O)[C@@H](O)CNC(=O)/C=C/c1cccnc1 ZINC000217743144 CB On-Demand Unstable MMP9 15 41 COC[C@H]1CCCN(S(=O)(=O)c2cccnc2Cl)C1 ZINC000217743155 DD On-Demand Unstable CASP3 44 32 COC[C@H]1CCCN(S(=O)(=O)c2cccnc2Cl)C1 ZINC000217743155 DD On-Demand Unstable CASP7 48 33 CCc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217743192 BD In-Stock Unstable CA2 17 44 CCc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217743192 BD In-Stock Unstable CA4 17 40 CCc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217743192 BD In-Stock Unstable ACR 54 38 CCc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217743192 BD In-Stock Unstable ENPP2 23 40 CCc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217743192 BD In-Stock Unstable PPO2 27 58 CCc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217743192 BD In-Stock Unstable RORC 17 43 CCc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217743192 BD In-Stock Unstable NAMPT 0 42 COC(=O)[C@H](O)CNC(=O)/C=C/c1cccnc1 ZINC000217743203 CB For-Sale Unstable MMP2 17 41 COC(=O)[C@H](O)CNC(=O)/C=C/c1cccnc1 ZINC000217743203 CB For-Sale Unstable MMP9 15 41 N#C[C@@H]1CCC[C@@H]1N[C@@H]1CCCc2cccnc21 ZINC000217743235 BF For-Sale Unstable CXCR4 42 32 CC(C)c1ccc(NC(=O)CC(=N)N)cc1 ZINC000217743324 BE In-Stock Unstable LTA4H 27 40 CC(C)c1ccc(NC(=O)CC(=N)N)cc1 ZINC000217743324 BE In-Stock Unstable SCN2A 17 59 CC(C)c1ccc(NC(=O)CC(=N)N)cc1 ZINC000217743324 BE In-Stock Unstable F3 45 33 CC(C)c1ccc(NC(=O)CC(=N)N)cc1 ZINC000217743324 BE In-Stock Unstable F7 30 42 CC(C)c1ccc(NC(=O)CC(=N)N)cc1 ZINC000217743324 BE In-Stock Unstable ACR 43 53 CC(C)c1ccc(NC(=O)CC(=N)N)cc1 ZINC000217743324 BE In-Stock Unstable ACAT 0 46 CC(C)c1ccc(NC(=O)CC(=N)N)cc1 ZINC000217743324 BE In-Stock Unstable PSBA 0 53 N#C[C@@H]1CCC[C@H]1N[C@@H]1CCCc2cccnc21 ZINC000217743330 BF For-Sale Unstable CXCR4 42 32 COc1ccccc1/C=C/NC(=O)NCCc1ccccc1C ZINC000217743331 DH For-Sale Unstable MTNR1A 37 43 COc1ccccc1/C=C/NC(=O)NCCc1ccccc1C ZINC000217743331 DH For-Sale Unstable MTNR1B 25 43 O=C(CCNS(=O)(=O)c1cccc(Cl)c1)NC[C@@H]1CCCN1c1nccs1 ZINC000217743352 IE For-Sale Unstable ADAMTS5 21 46 COC(=O)c1ccccc1N(C)C(=O)c1ccc(Oc2ccccc2)cc1 ZINC000217743380 FJ On-Demand Unstable SRD5A2 18 42 COC(=O)c1ccccc1N(C)C(=O)c1ccc(Oc2ccccc2)cc1 ZINC000217743380 FJ On-Demand Unstable LTA4H 36 40 COC(=O)c1ccccc1N(C)C(=O)c1ccc(Oc2ccccc2)cc1 ZINC000217743380 FJ On-Demand Unstable MT-ND1 22 41 O=C(/C=C\c1ccccc1)Nc1cnccc1C(=O)O ZINC000217743391 CE For-Sale Anodyne HDAC8 44 41 O=C(/C=C\c1ccccc1)Nc1cnccc1C(=O)O ZINC000217743391 CE For-Sale Anodyne MMP2 24 56 O=C(/C=C\c1ccccc1)Nc1cnccc1C(=O)O ZINC000217743391 CE For-Sale Anodyne HDAC6 33 49 O=C(/C=C\c1ccccc1)Nc1cnccc1C(=O)O ZINC000217743391 CE For-Sale Anodyne MMP9 16 56 O=C(CCNS(=O)(=O)c1cccc(Cl)c1)NC[C@H]1CCCN1c1nccs1 ZINC000217743434 IE For-Sale Unstable ADAMTS5 21 46 N=C(N)CC(=O)Nc1cccc2ccccc12 ZINC000217743437 BE In-Stock Unstable KCNJ11 85 35 N=C(N)CC(=O)Nc1cccc2ccccc12 ZINC000217743437 BE In-Stock Unstable TRPV1 30 41 N=C(N)CC(=O)Nc1cccc2ccccc12 ZINC000217743437 BE In-Stock Unstable HDAH 18 42 COc1ccccc1/C=C/NC(=O)NCCc1ccccc1OC ZINC000217743438 EG For-Sale Unstable MTNR1A 54 45 COc1ccccc1/C=C/NC(=O)NCCc1ccccc1OC ZINC000217743438 EG For-Sale Unstable MTNR1B 39 45 COCCNC(=O)[C@@]12CC[C@@H]3C[C@@H](C[C@@H](C3)C1)C2 ZINC000217743452 CE In-Stock Unstable ITPR1 15 52 O=C(N[C@@H]1CCN2CCCC[C@@H]12)c1ccc(CCl)cc1 ZINC000217743502 CF For-Sale Unstable SIGMAR1 15 53 O=C(N[C@@H]1CCN2CCCC[C@@H]12)c1ccc(CCl)cc1 ZINC000217743502 CF For-Sale Unstable SSTR3 31 44 O=C(N[C@@H]1CCN2CCCC[C@@H]12)c1ccc(CCl)cc1 ZINC000217743502 CF For-Sale Unstable L3MBTL3 68 39 N=C(N)CC(=O)Nc1ccccc1F ZINC000217743538 AD In-Stock Unstable CA5B 20 41 N=C(N)CC(=O)Nc1ccccc1F ZINC000217743538 AD In-Stock Unstable CA5A 23 41 COc1ccccc1/C=C/NC(=O)NCCc1ccccc1F ZINC000217743569 DG For-Sale Unstable NQO2 26 40 COc1ccccc1/C=C/NC(=O)NCCc1ccccc1F ZINC000217743569 DG For-Sale Unstable MTNR1A 48 42 COc1ccccc1/C=C/NC(=O)NCCc1ccccc1F ZINC000217743569 DG For-Sale Unstable MTNR1B 32 42 O=C(N[C@H]1CCN2CCCC[C@@H]12)c1ccc(CCl)cc1 ZINC000217743585 CF For-Sale Unstable SIGMAR1 15 53 O=C(N[C@H]1CCN2CCCC[C@@H]12)c1ccc(CCl)cc1 ZINC000217743585 CF For-Sale Unstable SSTR3 31 44 O=C(N[C@H]1CCN2CCCC[C@@H]12)c1ccc(CCl)cc1 ZINC000217743585 CF For-Sale Unstable L3MBTL3 68 39 N=C(N)CC(=O)Nc1cccc(F)c1 ZINC000217743630 AD In-Stock Unstable F2R 0 45 N=C(N)CC(=O)Nc1cccc(F)c1 ZINC000217743630 AD In-Stock Unstable FUCA1 0 49 N=C(N)CC(=O)Nc1cccc(F)c1 ZINC000217743630 AD In-Stock Unstable PARP14 42 36 N=C(N)CC(=O)Nc1cccc(F)c1 ZINC000217743630 AD In-Stock Unstable PARP15 47 34 N=C(N)CC(=O)Nc1cccc(F)c1 ZINC000217743630 AD In-Stock Unstable PSBA 0 53 N=C(N)CC(=O)Nc1cccc(F)c1 ZINC000217743630 AD In-Stock Unstable KCNK3 73 46 N=C(N)CC(=O)Nc1cccc(F)c1 ZINC000217743630 AD In-Stock Unstable KCNK9 67 43 N=C(N)CC(=O)Nc1cccc(F)c1 ZINC000217743630 AD In-Stock Unstable PARP10 0 45 O=C(CC[C@@H]1NC(=O)N(Cc2ccc3c(c2)OCO3)C1=O)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217743639 JD In-Stock Unstable SSTR3 101 34 O=C(CC[C@@H]1NC(=O)N(Cc2ccc3c(c2)OCO3)C1=O)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217743639 JD In-Stock Unstable MCHR1 22 40 CCC[C@@H](O)CNCCCN ZINC000217743647 AC For-Sale Unstable SPPS 41 36 CN1CCN(C)[C@@H](CN[C@@H]2CCCc3cccnc32)C1 ZINC000217743651 CD On-Demand Unstable CXCR4 57 41 COc1ccccc1/C=C/NC(=O)NCCc1ccccc1Cl ZINC000217743679 EH For-Sale Unstable MTNR1A 36 42 COc1ccccc1/C=C/NC(=O)NCCc1ccccc1Cl ZINC000217743679 EH For-Sale Unstable MTNR1B 27 42 COC(=O)c1ccccc1N(C)C(=O)c1cc(Br)ccc1Cl ZINC000217743692 GI On-Demand Unstable ECR 41 39 O=C(N[C@@H]1CCN2CCCC[C@@H]12)c1cccc(CCl)c1 ZINC000217743708 CF For-Sale Unstable DRD4 16 41 O=C(N[C@@H]1CCN2CCCC[C@@H]12)c1cccc(CCl)c1 ZINC000217743708 CF For-Sale Unstable SIGMAR1 21 49 O=C(N[C@@H]1CCN2CCCC[C@@H]12)c1cccc(CCl)c1 ZINC000217743708 CF For-Sale Unstable CHRNA7 21 40 O=C(N[C@@H]1CCN2CCCC[C@@H]12)c1cccc(CCl)c1 ZINC000217743708 CF For-Sale Unstable BDKRB1 15 41 O=C(N[C@@H]1CCN2CCCC[C@@H]12)c1cccc(CCl)c1 ZINC000217743708 CF For-Sale Unstable SSTR3 29 40 CCC[C@H](O)CNCCCN ZINC000217743729 AC For-Sale Unstable SPPS 41 36 N=C(N)CC(=O)Nc1ccc(F)cc1 ZINC000217743742 AD In-Stock Unstable FUCA1 23 44 N=C(N)CC(=O)Nc1ccc(F)cc1 ZINC000217743742 AD In-Stock Unstable ACR 45 35 N=C(N)CC(=O)Nc1ccc(F)cc1 ZINC000217743742 AD In-Stock Unstable PPO2 23 42 N=C(N)CC(=O)Nc1ccc(F)cc1 ZINC000217743742 AD In-Stock Unstable MTCA1 29 46 N=C(N)CC(=O)Nc1ccc(F)cc1 ZINC000217743742 AD In-Stock Unstable PSBA 0 47 Cc1cc(C)nc(NCC(=O)N2CCc3c([nH]c4ccccc34)C2)n1 ZINC000217743747 EF In-Stock Unstable DRD5 19 40 Cc1cc(C)nc(NCC(=O)N2CCc3c([nH]c4ccccc34)C2)n1 ZINC000217743747 EF In-Stock Unstable SSTR4 57 36 O=C(N[C@H]1CCN2CCCC[C@@H]12)c1cccc(CCl)c1 ZINC000217743791 CF For-Sale Unstable DRD4 16 41 O=C(N[C@H]1CCN2CCCC[C@@H]12)c1cccc(CCl)c1 ZINC000217743791 CF For-Sale Unstable SIGMAR1 21 49 O=C(N[C@H]1CCN2CCCC[C@@H]12)c1cccc(CCl)c1 ZINC000217743791 CF For-Sale Unstable CHRNA7 21 40 O=C(N[C@H]1CCN2CCCC[C@@H]12)c1cccc(CCl)c1 ZINC000217743791 CF For-Sale Unstable BDKRB1 15 41 O=C(N[C@H]1CCN2CCCC[C@@H]12)c1cccc(CCl)c1 ZINC000217743791 CF For-Sale Unstable SSTR3 29 40 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(Oc3ccccc3)cc2)CC1 ZINC000217743798 HK On-Demand Unstable HTR2A 20 53 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(Oc3ccccc3)cc2)CC1 ZINC000217743798 HK On-Demand Unstable SRD5A2 15 40 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(Oc3ccccc3)cc2)CC1 ZINC000217743798 HK On-Demand Unstable INHA 16 46 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(Oc3ccccc3)cc2)CC1 ZINC000217743798 HK On-Demand Unstable GRIN2B 18 45 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(Oc3ccccc3)cc2)CC1 ZINC000217743798 HK On-Demand Unstable LTA4H 30 42 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(Oc3ccccc3)cc2)CC1 ZINC000217743798 HK On-Demand Unstable HRH3 24 47 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(Oc3ccccc3)cc2)CC1 ZINC000217743798 HK On-Demand Unstable SLC18A3 73 65 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(Oc3ccccc3)cc2)CC1 ZINC000217743798 HK On-Demand Unstable MMP2 21 46 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(Oc3ccccc3)cc2)CC1 ZINC000217743798 HK On-Demand Unstable MMP9 21 46 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(Oc3ccccc3)cc2)CC1 ZINC000217743798 HK On-Demand Unstable EPHX2 16 43 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(Oc3ccccc3)cc2)CC1 ZINC000217743798 HK On-Demand Unstable PLAU 20 52 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(Oc3ccccc3)cc2)CC1 ZINC000217743798 HK On-Demand Unstable ST14 17 42 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(Oc3ccccc3)cc2)CC1 ZINC000217743798 HK On-Demand Unstable CCR8 22 40 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(Oc3ccccc3)cc2)CC1 ZINC000217743798 HK On-Demand Unstable WNT3A 55 36 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(Oc3ccccc3)cc2)CC1 ZINC000217743798 HK On-Demand Unstable L3MBTL3 95 47 COc1ccccc1/C=C/NC(=O)NCCc1ccccc1Br ZINC000217743807 GH For-Sale Unstable MTNR1A 33 42 COc1ccccc1/C=C/NC(=O)NCCc1ccccc1Br ZINC000217743807 GH For-Sale Unstable MTNR1B 25 42 N=C(N)CC(=O)Nc1ccccc1Cl ZINC000217743860 BD In-Stock Unstable CXCL8 56 45 N=C(N)CC(=O)Nc1ccccc1Cl ZINC000217743860 BD In-Stock Unstable KCNQ2 38 45 N=C(N)CC(=O)Nc1ccccc1Cl ZINC000217743860 BD In-Stock Unstable CA5B 20 41 N=C(N)CC(=O)Nc1ccccc1Cl ZINC000217743860 BD In-Stock Unstable CA5A 23 41 N=C(N)CC(=O)Nc1ccccc1Cl ZINC000217743860 BD In-Stock Unstable EPHB3 55 41 O=C(N[C@@H]1CCN2CCCC[C@@H]12)[C@H](Cl)c1ccccc1 ZINC000217743883 CF For-Sale Unstable VACHT_TETCF 0 42 O=C(N[C@@H]1CCN2CCCC[C@@H]12)[C@H](Cl)c1ccccc1 ZINC000217743883 CF For-Sale Unstable SIGMAR1 0 44 O=C(N[C@@H]1CCN2CCCC[C@@H]12)[C@H](Cl)c1ccccc1 ZINC000217743883 CF For-Sale Unstable SLC18A3 72 38 COC(=O)c1ccccc1N(C)C(=O)c1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217743907 HJ On-Demand Unstable TACR1 43 48 COc1ccccc1/C=C/NC(=O)NCCc1cccc(C)c1 ZINC000217743910 DH For-Sale Unstable MTNR1A 31 41 COc1ccccc1/C=C/NC(=O)NCCc1cccc(C)c1 ZINC000217743910 DH For-Sale Unstable AKR1B10 30 41 COc1ccccc1/C=C/NC(=O)NCCc1cccc(C)c1 ZINC000217743910 DH For-Sale Unstable KCNK9 40 38 CS(=O)(=O)c1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)s1 ZINC000217743912 GG On-Demand Unstable SLC18A3 35 48 CS(=O)(=O)c1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)s1 ZINC000217743912 GG On-Demand Unstable WNT3A 46 33 CS(=O)(=O)c1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)s1 ZINC000217743912 GG On-Demand Unstable L3MBTL3 70 42 CC(C)C[C@@H](O)C(=O)NCc1cc2ccccc2[nH]1 ZINC000217743946 CE In-Stock Unstable CCKAR 23 44 CC(C)(F)c1ccc([C@H](N)C(=O)O)c(Cl)c1 ZINC000217743953 BF For-Sale Unstable CACNA2D1 30 44 O=C(N[C@@H]1CCN2CCCC[C@@H]12)[C@@H](Cl)c1ccccc1 ZINC000217743963 CF For-Sale Unstable VACHT_TETCF 0 42 O=C(N[C@@H]1CCN2CCCC[C@@H]12)[C@@H](Cl)c1ccccc1 ZINC000217743963 CF For-Sale Unstable SIGMAR1 0 44 O=C(N[C@@H]1CCN2CCCC[C@@H]12)[C@@H](Cl)c1ccccc1 ZINC000217743963 CF For-Sale Unstable SLC18A3 72 38 COC(=O)C[C@H](c1cc2ccccc2[nH]c1=O)c1c(O)c2ccccc2oc1=O ZINC000217743977 GG In-Stock Unstable NQO1 53 50 C[C@H]1C[C@H](C)CC[C@@H]1N[C@@H]1CCCc2cccnc21 ZINC000217743980 CH On-Demand Unstable CXCR4 48 33 N=C(N)CC(=O)Nc1cccc(Cl)c1 ZINC000217743983 BD In-Stock Unstable ABAT 20 41 N=C(N)CC(=O)Nc1cccc(Cl)c1 ZINC000217743983 BD In-Stock Unstable PPIA 25 44 N=C(N)CC(=O)Nc1cccc(Cl)c1 ZINC000217743983 BD In-Stock Unstable F2R 0 45 N=C(N)CC(=O)Nc1cccc(Cl)c1 ZINC000217743983 BD In-Stock Unstable F13A1 24 52 N=C(N)CC(=O)Nc1cccc(Cl)c1 ZINC000217743983 BD In-Stock Unstable NAMPT 0 51 N=C(N)CC(=O)Nc1cccc(Cl)c1 ZINC000217743983 BD In-Stock Unstable KCNK3 59 46 N=C(N)CC(=O)Nc1cccc(Cl)c1 ZINC000217743983 BD In-Stock Unstable KCNK9 53 43 CC(C)(F)c1ccc([C@@H](N)C(=O)O)c(Cl)c1 ZINC000217744021 BF For-Sale Unstable CACNA2D1 30 44 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable PLG 16 42 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable ACE 66 48 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable TYR 40 48 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable PPARG 19 42 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable OPRD1 45 37 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable PPARA 23 41 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable CELA1 30 40 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable GRIN2B 24 44 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable ELANE 29 43 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable MME 140 51 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable LTA4H 20 47 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable ANPEP 79 41 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable TACR1 21 42 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable CTRA_BOVIN 44 34 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable HRAS 57 39 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable FCER2 61 33 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable GRB2 21 41 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable CASP3 18 53 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable BMP1 67 39 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable KLK3 83 40 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable CTSB 89 67 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable PAPA1_CARPA 95 50 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable CYSP_TRYCR 76 51 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable CCKAR 28 41 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable CTSK 53 53 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable CTSL 75 56 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable CPA1 51 44 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable CACNA1B 51 36 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable TIMP3 48 43 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable ITGA4 43 38 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable NAALAD2 31 42 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable CDC25B 27 40 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable CAPNS1 85 54 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable MMP2 16 47 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable MMP8 42 35 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable MMP14 42 35 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable ECE1 51 50 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable HLA-DRB1 51 36 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable CELA2A 51 34 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable REN 19 42 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable MMP11 66 38 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable CTSS 38 53 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable CAPN1 119 52 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable MMP9 25 43 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable CASP1 25 44 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable CTRC 39 43 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable CAPN2 154 67 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable ACE2 100 48 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable PLAU 19 44 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable CASP6 23 41 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable CASP9 30 41 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable TPSAB1 49 39 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable MMP1 20 44 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable FPR1 86 52 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable NPR 83 46 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable AMP1_PLAFQ 19 44 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable FFAR1 22 41 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable PSMB5 41 43 O=C(N[C@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)O)OCc1ccccc1 ZINC000217744024 GH For-Sale Unstable BLA1_STEMA 76 39 COc1cccc(CCNC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217744025 EG For-Sale Unstable DRD4 42 33 COc1cccc(CCNC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217744025 EG For-Sale Unstable HRH2 24 42 COc1cccc(CCNC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217744025 EG For-Sale Unstable CYP1B1 39 44 COc1cccc(CCNC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217744025 EG For-Sale Unstable MTNR1A 96 52 COc1cccc(CCNC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217744025 EG For-Sale Unstable MTNR1B 89 52 COc1cccc(CCNC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217744025 EG For-Sale Unstable ABCB1 16 43 COc1cccc(CCNC(=O)N/C=C/c2ccccc2OC)c1 ZINC000217744025 EG For-Sale Unstable CRTM 54 39 CC(C)C[C@H](O)C(=O)NCc1cc2ccccc2[nH]1 ZINC000217744029 CE In-Stock Unstable CCKAR 23 44 Clc1cc(CBr)ccc1N1CCN2CCCC[C@@H]2C1 ZINC000217744032 EH For-Sale Unstable L3MBTL3 44 35 O=C(N[C@H]1CCN2CCCC[C@@H]12)[C@H](Cl)c1ccccc1 ZINC000217744047 CF For-Sale Unstable VACHT_TETCF 0 42 O=C(N[C@H]1CCN2CCCC[C@@H]12)[C@H](Cl)c1ccccc1 ZINC000217744047 CF For-Sale Unstable SIGMAR1 0 44 O=C(N[C@H]1CCN2CCCC[C@@H]12)[C@H](Cl)c1ccccc1 ZINC000217744047 CF For-Sale Unstable SLC18A3 72 38 COC(=O)C[C@@H](c1cc2ccccc2[nH]c1=O)c1c(O)c2ccccc2oc1=O ZINC000217744069 GG In-Stock Unstable NQO1 53 50 N=C(N)CC(=O)Nc1ccc(Cl)cc1 ZINC000217744102 BD In-Stock Unstable ACR 48 50 N=C(N)CC(=O)Nc1ccc(Cl)cc1 ZINC000217744102 BD In-Stock Unstable SLC1A2 43 39 N=C(N)CC(=O)Nc1ccc(Cl)cc1 ZINC000217744102 BD In-Stock Unstable MTCA1 23 46 N=C(N)CC(=O)Nc1ccc(Cl)cc1 ZINC000217744102 BD In-Stock Unstable P96878_MYCTU 17 46 N=C(N)CC(=O)Nc1ccc(Cl)cc1 ZINC000217744102 BD In-Stock Unstable IMDH_CRYPV 27 40 Cc1cccc(S(=O)(=O)NCCC(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217744118 HD For-Sale Unstable FBP1 15 40 Cc1cccc(S(=O)(=O)NCCC(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217744118 HD For-Sale Unstable ADAMTS5 28 40 CC(C)(F)c1c(Cl)cccc1[C@H](N)C(=O)O ZINC000217744123 BF For-Sale Unstable CACNA2D1 25 48 O=C(N[C@H]1CCN2CCCC[C@@H]12)[C@@H](Cl)c1ccccc1 ZINC000217744130 CF For-Sale Unstable VACHT_TETCF 0 42 O=C(N[C@H]1CCN2CCCC[C@@H]12)[C@@H](Cl)c1ccccc1 ZINC000217744130 CF For-Sale Unstable SIGMAR1 0 44 O=C(N[C@H]1CCN2CCCC[C@@H]12)[C@@H](Cl)c1ccccc1 ZINC000217744130 CF For-Sale Unstable SLC18A3 72 38 COc1ccccc1/C=C/NC(=O)NCCc1cccc(F)c1 ZINC000217744133 DG For-Sale Unstable MTNR1A 27 40 COc1ccccc1/C=C/NC(=O)NCCc1cccc(F)c1 ZINC000217744133 DG For-Sale Unstable ACKR3 45 32 O=C(O)/C=C\c1ccc(NC(=O)c2ccc(Cl)cn2)cc1 ZINC000217744176 DG On-Demand Anodyne P4HTM 0 41 O=C(O)/C=C\c1ccc(NC(=O)c2ccc(Cl)cn2)cc1 ZINC000217744176 DG On-Demand Anodyne BACE1 0 42 O=C(O)/C=C\c1ccc(NC(=O)c2ccc(Cl)cn2)cc1 ZINC000217744176 DG On-Demand Anodyne MMP1 0 50 O=C(O)/C=C\c1ccc(NC(=O)c2ccc(Cl)cn2)cc1 ZINC000217744176 DG On-Demand Anodyne SMO 15 46 N=C(N)CC(=O)Nc1ccccc1Br ZINC000217744207 CD In-Stock Unstable CA5B 25 42 N=C(N)CC(=O)Nc1ccccc1Br ZINC000217744207 CD In-Stock Unstable CA5A 29 42 N=C(N)CC(=O)Nc1ccccc1Br ZINC000217744207 CD In-Stock Unstable CA9 20 44 Cc1cccc(S(=O)(=O)NCCC(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217744213 HD For-Sale Unstable FBP1 15 40 Cc1cccc(S(=O)(=O)NCCC(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217744213 HD For-Sale Unstable ADAMTS5 28 40 CC1(C)[C@H]2CC[C@](C)(C2)[C@H]1N[C@@H]1CCCc2cccnc21 ZINC000217744221 CI For-Sale Unstable CXCR4 44 32 CC(C)(F)c1c(Cl)cccc1[C@@H](N)C(=O)O ZINC000217744223 BF For-Sale Unstable CACNA2D1 25 48 COc1ccccc1/C=C/NC(=O)NCCc1cccc(Cl)c1 ZINC000217744235 EH For-Sale Unstable MTNR1A 25 40 COc1ccccc1/C=C/NC(=O)NCCc1cccc(Cl)c1 ZINC000217744235 EH For-Sale Unstable LMGT2 0 42 COC(=O)[C@@H](O)CNC(=O)/C=C/c1ccc2c(c1)OCO2 ZINC000217744298 CC On-Demand Unstable DYRK2 65 36 BrCc1ccccc1N1CCN2CCCC[C@@H]2C1 ZINC000217744299 DG For-Sale Unstable L3MBTL3 43 35 N=C(N)CC(=O)Nc1cccc(Br)c1 ZINC000217744317 CD In-Stock Unstable EGFR 49 49 N=C(N)CC(=O)Nc1cccc(Br)c1 ZINC000217744317 CD In-Stock Unstable NADD 0 44 N=C(N)CC(=O)Nc1cccc(Br)c1 ZINC000217744317 CD In-Stock Unstable KCNK3 56 33 N=C(N)CC(=O)Nc1cccc(Br)c1 ZINC000217744317 CD In-Stock Unstable KCNK9 51 33 N=C(N)CC(=O)Nc1cccc(Br)c1 ZINC000217744317 CD In-Stock Unstable MVFR 0 49 N=C(N)CC(=O)Nc1cccc(Br)c1 ZINC000217744317 CD In-Stock Unstable PARP10 0 49 C[C@H](F)c1c(Cl)cccc1C[C@H](N)C(=O)O ZINC000217744328 BE For-Sale Unstable CACNA2D1 50 45 C[C@H](F)c1c(Cl)cccc1C[C@H](N)C(=O)O ZINC000217744328 BE For-Sale Unstable CXCL8 41 32 COc1ccccc1/C=C/NC(=O)NCCc1cccc(Br)c1 ZINC000217744334 GH For-Sale Unstable MTNR1A 26 40 CCCCCCCNC[C@@H](O)CCC ZINC000217744343 BF For-Sale Unstable S1PR3 18 41 CCCCCCCNC[C@@H](O)CCC ZINC000217744343 BF For-Sale Unstable S1PR2 44 41 CCCCCCCNC[C@@H](O)CCC ZINC000217744343 BF For-Sale Unstable Q8WS26_TRYCR 45 52 CCCCCCCNC[C@@H](O)CCC ZINC000217744343 BF For-Sale Unstable CQSS 45 38 C[C@@H](CCc1ccccc1)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217744346 CF For-Sale Unstable ACE 47 40 C[C@@H](CCc1ccccc1)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217744346 CF For-Sale Unstable SLC18A2 41 37 C[C@@H](CCc1ccccc1)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217744346 CF For-Sale Unstable SIGMAR1 20 44 C[C@@H](CCc1ccccc1)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217744346 CF For-Sale Unstable SLC18A3 36 40 CC(C)(C)[C@@H]1CC[C@@H](N)[C@@H](CCCc2ccccc2)C1 ZINC000217744392 CJ For-Sale Unstable SLC18A2 43 44 C[C@@H](F)c1c(Cl)cccc1C[C@H](N)C(=O)O ZINC000217744419 BE For-Sale Unstable CACNA2D1 50 45 C[C@@H](F)c1c(Cl)cccc1C[C@H](N)C(=O)O ZINC000217744419 BE For-Sale Unstable CXCL8 41 32 BrCc1ccc(N2CCN3CCCC[C@@H]3C2)nc1 ZINC000217744421 DF For-Sale Unstable L3MBTL3 41 34 N=C(N)CC(=O)Nc1ccc(Br)cc1 ZINC000217744426 CD In-Stock Unstable ACR 48 50 N=C(N)CC(=O)Nc1ccc(Br)cc1 ZINC000217744426 CD In-Stock Unstable IDO1 15 42 N=C(N)CC(=O)Nc1ccc(Br)cc1 ZINC000217744426 CD In-Stock Unstable MTCA1 23 46 CCCCCCCNC[C@H](O)CCC ZINC000217744429 BF For-Sale Unstable S1PR3 18 41 CCCCCCCNC[C@H](O)CCC ZINC000217744429 BF For-Sale Unstable S1PR2 44 41 CCCCCCCNC[C@H](O)CCC ZINC000217744429 BF For-Sale Unstable Q8WS26_TRYCR 45 52 CCCCCCCNC[C@H](O)CCC ZINC000217744429 BF For-Sale Unstable CQSS 45 38 C[C@H](CCc1ccccc1)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217744433 CF For-Sale Unstable ACE 47 40 C[C@H](CCc1ccccc1)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217744433 CF For-Sale Unstable SLC18A2 41 37 C[C@H](CCc1ccccc1)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217744433 CF For-Sale Unstable SIGMAR1 20 44 C[C@H](CCc1ccccc1)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217744433 CF For-Sale Unstable SLC18A3 36 40 CC(C)(C)[C@H]1CC[C@@H](N)[C@@H](CCCc2ccccc2)C1 ZINC000217744464 CJ For-Sale Unstable SLC18A2 43 44 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(OCc3ccccc3)cc2)CC1 ZINC000217744474 HK On-Demand Unstable HRH2 18 41 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(OCc3ccccc3)cc2)CC1 ZINC000217744474 HK On-Demand Unstable MAOB 22 50 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(OCc3ccccc3)cc2)CC1 ZINC000217744474 HK On-Demand Unstable HTR2A 24 57 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(OCc3ccccc3)cc2)CC1 ZINC000217744474 HK On-Demand Unstable AVPR1A 24 40 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(OCc3ccccc3)cc2)CC1 ZINC000217744474 HK On-Demand Unstable GRIN2B 59 44 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(OCc3ccccc3)cc2)CC1 ZINC000217744474 HK On-Demand Unstable LTA4H 37 42 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(OCc3ccccc3)cc2)CC1 ZINC000217744474 HK On-Demand Unstable HRH3 30 53 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(OCc3ccccc3)cc2)CC1 ZINC000217744474 HK On-Demand Unstable SIGMAR1 24 49 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(OCc3ccccc3)cc2)CC1 ZINC000217744474 HK On-Demand Unstable ADAM17 27 43 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(OCc3ccccc3)cc2)CC1 ZINC000217744474 HK On-Demand Unstable SLC18A3 61 56 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(OCc3ccccc3)cc2)CC1 ZINC000217744474 HK On-Demand Unstable GRM5 16 52 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(OCc3ccccc3)cc2)CC1 ZINC000217744474 HK On-Demand Unstable SLC6A5 37 43 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(OCc3ccccc3)cc2)CC1 ZINC000217744474 HK On-Demand Unstable EPHX2 16 42 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(OCc3ccccc3)cc2)CC1 ZINC000217744474 HK On-Demand Unstable FFAR1 22 41 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(OCc3ccccc3)cc2)CC1 ZINC000217744474 HK On-Demand Unstable WNT3A 50 39 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(OCc3ccccc3)cc2)CC1 ZINC000217744474 HK On-Demand Unstable L3MBTL3 85 40 C[C@H](F)c1c(Cl)cccc1C[C@@H](N)C(=O)O ZINC000217744503 BE For-Sale Unstable CACNA2D1 50 45 C[C@H](F)c1c(Cl)cccc1C[C@@H](N)C(=O)O ZINC000217744503 BE For-Sale Unstable CXCL8 41 32 C[C@@H](CCc1ccccc1)N[C@H]1CCN2CCC[C@@H]12 ZINC000217744510 CF For-Sale Unstable ACE 47 40 C[C@@H](CCc1ccccc1)N[C@H]1CCN2CCC[C@@H]12 ZINC000217744510 CF For-Sale Unstable SLC18A2 41 37 C[C@@H](CCc1ccccc1)N[C@H]1CCN2CCC[C@@H]12 ZINC000217744510 CF For-Sale Unstable SIGMAR1 20 44 C[C@@H](CCc1ccccc1)N[C@H]1CCN2CCC[C@@H]12 ZINC000217744510 CF For-Sale Unstable SLC18A3 36 40 O=S1(=O)CCCN(S(=O)(=O)c2ccc(F)cc2)CC1 ZINC000217744515 DC On-Demand Unstable PKM 35 47 N=C(N)CC(=O)Nc1ccc(I)cc1 ZINC000217744541 DD In-Stock Unstable ACR 45 35 N=C(N)CC(=O)Nc1ccc(I)cc1 ZINC000217744541 DD In-Stock Unstable MTCA1 23 46 N=C(N)CC(=O)Nc1ccc(I)cc1 ZINC000217744541 DD In-Stock Unstable Q25615_ONCVO 58 44 CC(C)(C)[C@@H]1CC[C@H](N)[C@@H](CCCc2ccccc2)C1 ZINC000217744543 CJ For-Sale Unstable SLC18A2 43 44 C[C@@H](F)c1c(Cl)cccc1C[C@@H](N)C(=O)O ZINC000217744571 BE For-Sale Unstable CACNA2D1 50 45 C[C@@H](F)c1c(Cl)cccc1C[C@@H](N)C(=O)O ZINC000217744571 BE For-Sale Unstable CXCL8 41 32 C[C@H](CCc1ccccc1)N[C@H]1CCN2CCC[C@@H]12 ZINC000217744587 CF For-Sale Unstable ACE 47 40 C[C@H](CCc1ccccc1)N[C@H]1CCN2CCC[C@@H]12 ZINC000217744587 CF For-Sale Unstable SLC18A2 41 37 C[C@H](CCc1ccccc1)N[C@H]1CCN2CCC[C@@H]12 ZINC000217744587 CF For-Sale Unstable SIGMAR1 20 44 C[C@H](CCc1ccccc1)N[C@H]1CCN2CCC[C@@H]12 ZINC000217744587 CF For-Sale Unstable SLC18A3 36 40 COc1ccc(CCC(=O)N2CC(N3C(=O)CSC3=O)C2)cc1OCc1ccccc1 ZINC000217744619 IG In-Stock Unstable MTNR1B 17 45 CC(C)(C)[C@H]1CC[C@H](N)[C@@H](CCCc2ccccc2)C1 ZINC000217744636 CJ For-Sale Unstable SLC18A2 43 44 Cc1c(Cl)cccc1NC(=O)CC(=N)N ZINC000217744644 BD In-Stock Unstable CXCL8 43 34 O=C(O)/C=C\c1cccc(NC(=O)CCC2CCCC2)n1 ZINC000217744660 CG For-Sale Unstable LDLR 0 40 C[C@H](F)c1c(Cl)cccc1[C@H](N)CC(=O)O ZINC000217744682 BF For-Sale Unstable CXCL8 42 35 COC(=O)[C@@H](O)CNC(=O)/C=C/c1ccc(C(N)=O)cc1 ZINC000217744683 CB On-Demand Unstable HDAC8 0 44 O[C@@H]1CCCC[C@@H]1CN[C@@H]1CCCc2cccnc21 ZINC000217744692 CF On-Demand Unstable CXCR4 63 35 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccnn2C(C)C)CC(=O)O4)cc1O ZINC000217744715 JI In-Stock Unstable AKR1B1 0 44 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccnn2C(C)C)CC(=O)O4)cc1O ZINC000217744715 JI In-Stock Unstable CYP1B1 42 46 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccnn2C(C)C)CC(=O)O4)cc1O ZINC000217744715 JI In-Stock Unstable CYP1A1 33 46 O=C(CCNS(=O)(=O)c1cccc(F)c1)NC[C@@H]1CCCN1c1nccs1 ZINC000217744723 HD For-Sale Unstable ADAMTS5 29 40 Cc1cc(C(=O)Nc2cccc(/C=C\C(=O)O)n2)c(C)o1 ZINC000217744734 CF For-Sale Unstable GRM5 15 40 Cc1cc(C(=O)Nc2cccc(/C=C\C(=O)O)n2)c(C)o1 ZINC000217744734 CF For-Sale Unstable SORT1 26 42 Cc1cc(Cl)ccc1NC(=O)CC(=N)N ZINC000217744753 BD In-Stock Unstable SLC1A1 28 40 Cc1cc(Cl)ccc1NC(=O)CC(=N)N ZINC000217744753 BD In-Stock Unstable SLC1A3 28 40 Cc1cc(Cl)ccc1NC(=O)CC(=N)N ZINC000217744753 BD In-Stock Unstable SLC1A2 26 40 O[C@@H]1CCCC[C@H]1CN[C@@H]1CCCc2cccnc21 ZINC000217744770 CF On-Demand Unstable CXCR4 63 35 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccnn2C(C)C)CC(=O)O4)cc1O ZINC000217744783 JI In-Stock Unstable AKR1B1 0 44 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccnn2C(C)C)CC(=O)O4)cc1O ZINC000217744783 JI In-Stock Unstable CYP1B1 42 46 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccnn2C(C)C)CC(=O)O4)cc1O ZINC000217744783 JI In-Stock Unstable CYP1A1 33 46 C[C@@H](F)c1c(Cl)cccc1[C@H](N)CC(=O)O ZINC000217744785 BF For-Sale Unstable CXCL8 42 35 O=C(CCNS(=O)(=O)c1cccc(F)c1)NC[C@H]1CCCN1c1nccs1 ZINC000217744795 HD For-Sale Unstable ADAMTS5 29 40 COc1ccccc1/C=C/NC(=O)Nc1ccc(C)nc1 ZINC000217744808 CG For-Sale Unstable PDGFRA 40 34 COc1ccccc1/C=C/NC(=O)Nc1ccc(C)nc1 ZINC000217744808 CG For-Sale Unstable IMPDH2 0 44 Cc1ccc(Cl)cc1NC(=O)CC(=N)N ZINC000217744853 BD In-Stock Unstable KCNMA1 24 40 C[C@H](F)c1c(Cl)cccc1[C@@H](N)CC(=O)O ZINC000217744858 BF For-Sale Unstable CXCL8 42 35 Cc1cc(N2CCN3CCCC[C@@H]3C2)ccc1CBr ZINC000217744862 DH For-Sale Unstable HRH3 0 41 COc1ccccc1/C=C/NC(=O)Nc1ccc(C)cn1 ZINC000217744914 CG For-Sale Unstable GCK 21 42 COc1ccccc1/C=C/NC(=O)Nc1ccc(C)cn1 ZINC000217744914 CG For-Sale Unstable LUCI_LUCLA 41 48 C[C@@H](F)c1c(Cl)cccc1[C@@H](N)CC(=O)O ZINC000217744954 BF For-Sale Unstable CXCL8 42 35 Cc1ccc(NC(=O)CC(=N)N)cc1Cl ZINC000217744958 BD In-Stock Unstable PPIA 19 45 Cc1ccc(NC(=O)CC(=N)N)cc1Cl ZINC000217744958 BD In-Stock Unstable SLC1A1 44 41 Cc1ccc(NC(=O)CC(=N)N)cc1Cl ZINC000217744958 BD In-Stock Unstable SLC1A3 45 41 Cc1ccc(NC(=O)CC(=N)N)cc1Cl ZINC000217744958 BD In-Stock Unstable SLC1A2 50 41 BrCc1ccc(Br)cc1N1CCN2CCCC[C@@H]2C1 ZINC000217744985 GI For-Sale Unstable L3MBTL3 48 33 O=C(O)/C=C\c1cnc(NC(=O)c2cccn2C2CC2)s1 ZINC000217745009 DF For-Sale Unstable CDK5 47 35 C[C@H](F)c1c(Cl)cccc1[C@@H](CN)C(=O)O ZINC000217745049 BE For-Sale Unstable CXCL8 30 42 O[C@@H]1CCC[C@@H]1CN[C@@H]1CCCc2cccnc21 ZINC000217745082 BE For-Sale Unstable CXCR4 64 36 N=C(N)CC(=O)Nc1cccc(Cl)c1Cl ZINC000217745090 BE In-Stock Unstable CXCL8 42 36 N=C(N)CC(=O)Nc1cccc(Cl)c1Cl ZINC000217745090 BE In-Stock Unstable KCNQ2 32 40 N=C(N)CC(=O)Nc1cccc(Cl)c1Cl ZINC000217745090 BE In-Stock Unstable S100B 0 59 COc1cc2c(cc1OC)CC(=O)N(CC(=O)N[C@@H](C)CO)C=C2 ZINC000217745095 EC In-Stock Unstable HCN2 0 45 COCCn1c(C(=O)N2CC(N3C(=O)CSC3=O)C2)cc2c(=O)n3ccccc3nc21 ZINC000217745105 IC In-Stock Unstable POLR1A 68 34 BrCc1ccc(N2CCN3CCCC[C@@H]3C2)cc1 ZINC000217745107 DG For-Sale Unstable L3MBTL3 71 49 COCCCCN[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217745135 BG For-Sale Unstable TRPM8 15 42 C[C@@H](F)c1c(Cl)cccc1[C@@H](CN)C(=O)O ZINC000217745137 BE For-Sale Unstable CXCL8 30 42 O[C@@H]1CCC[C@H]1CN[C@@H]1CCCc2cccnc21 ZINC000217745156 BE On-Demand Unstable CXCR4 63 35 N=C(N)CC(=O)Nc1ccc(Cl)cc1Cl ZINC000217745193 BE In-Stock Unstable CA2 16 47 N=C(N)CC(=O)Nc1ccc(Cl)cc1Cl ZINC000217745193 BE In-Stock Unstable CA1 21 47 N=C(N)CC(=O)Nc1ccc(Cl)cc1Cl ZINC000217745193 BE In-Stock Unstable CA5B 21 43 N=C(N)CC(=O)Nc1ccc(Cl)cc1Cl ZINC000217745193 BE In-Stock Unstable CA4 21 47 N=C(N)CC(=O)Nc1ccc(Cl)cc1Cl ZINC000217745193 BE In-Stock Unstable CA5A 24 43 N=C(N)CC(=O)Nc1ccc(Cl)cc1Cl ZINC000217745193 BE In-Stock Unstable ALPL 40 37 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2csnn2)CC1 ZINC000217745195 DE On-Demand Unstable SLC18A3 34 50 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2csnn2)CC1 ZINC000217745195 DE On-Demand Unstable WNT3A 47 36 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2csnn2)CC1 ZINC000217745195 DE On-Demand Unstable L3MBTL3 60 36 C[C@H](F)c1c(Cl)cccc1[C@H](CN)C(=O)O ZINC000217745213 BE For-Sale Unstable CXCL8 30 42 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)cn1 ZINC000217745225 DH For-Sale Unstable F10 54 36 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)cn1 ZINC000217745225 DH For-Sale Unstable LUCI_LUCLA 41 41 COc1ccccc1/C=C/NC(=O)Nc1ccc(Cl)cn1 ZINC000217745225 DH For-Sale Unstable CYSP_PLAFA 43 36 COCCCCN[C@H]1C[C@H](C)CC[C@@H]1C(C)C ZINC000217745226 BG On-Demand Unstable TRPM8 15 42 OC[C@@H]1CCC[C@@H]1CN[C@@H]1CCCc2cccnc21 ZINC000217745271 CE For-Sale Unstable CXCR4 62 36 C[C@@H](F)c1c(Cl)cccc1[C@H](CN)C(=O)O ZINC000217745292 BE For-Sale Unstable CXCL8 30 42 CCOc1cccc(CN[C@@H]2CCN3CCC[C@@H]23)c1O ZINC000217745296 CE For-Sale Unstable HCN1 45 34 CCOc1cccc(CN[C@@H]2CCN3CCC[C@@H]23)c1O ZINC000217745296 CE For-Sale Unstable HCN4 42 34 N=C(N)CC(=O)Nc1cc(Cl)ccc1Cl ZINC000217745309 BE In-Stock Unstable KCNMA1 19 41 COc1ccccc1/C=C/NC(=O)Nc1cc(Cl)ccn1 ZINC000217745337 DH For-Sale Unstable CYSP_PLAFA 48 33 OC[C@@H]1CCC[C@H]1CN[C@@H]1CCCc2cccnc21 ZINC000217745361 CE For-Sale Unstable CXCR4 62 36 CCOc1cccc(CN[C@H]2CCN3CCC[C@@H]23)c1O ZINC000217745387 CE For-Sale Unstable HCN1 45 34 CCOc1cccc(CN[C@H]2CCN3CCC[C@@H]23)c1O ZINC000217745387 CE For-Sale Unstable HCN4 42 34 CCCCn1cnc(C#N)c1 ZINC000217745408 AD In-Stock Unstable CPB1 21 43 N=C(N)CC(=O)Nc1c(Cl)cccc1Cl ZINC000217745441 BE In-Stock Unstable CXCL8 51 32 N=C(N)CC(=O)Nc1c(Cl)cccc1Cl ZINC000217745441 BE In-Stock Unstable ACAT 0 40 O=C(O)/C=C\c1cccc(NC(=O)C2CCOCC2)c1 ZINC000217745460 CE For-Sale Unstable TYK2 42 36 O=C(O)/C=C\c1cccc(NC(=O)C2CCOCC2)c1 ZINC000217745460 CE For-Sale Unstable KCNK3 15 44 CC(C)(C)c1ccc(S(=O)(=O)NCCC(=O)NC[C@@H]2CCCN2c2nccs2)cc1 ZINC000217745473 JF For-Sale Unstable ADAMTS5 24 42 OC[C@@H]1CCCC[C@@H]1CN[C@@H]1CCCc2cccnc21 ZINC000217745478 CF For-Sale Unstable CXCR4 62 36 COc1ccc(S(=O)(=O)N2CCCS(=O)(=O)CC2)cc1Br ZINC000217745487 GD On-Demand Unstable PKM 18 40 COc1ccccc1/C=C/NC(=O)NCCCc1ccccc1 ZINC000217745541 DH For-Sale Unstable DRD2 18 44 COc1ccccc1/C=C/NC(=O)NCCCc1ccccc1 ZINC000217745541 DH For-Sale Unstable DRD3 29 44 COc1ccccc1/C=C/NC(=O)NCCCc1ccccc1 ZINC000217745541 DH For-Sale Unstable KCNA3 30 42 COc1ccccc1/C=C/NC(=O)NCCCc1ccccc1 ZINC000217745541 DH For-Sale Unstable SCN2A 16 41 COc1ccccc1/C=C/NC(=O)NCCCc1ccccc1 ZINC000217745541 DH For-Sale Unstable MTNR1A 34 44 COc1ccccc1/C=C/NC(=O)NCCCc1ccccc1 ZINC000217745541 DH For-Sale Unstable MTNR1B 37 46 COc1ccccc1/C=C/NC(=O)NCCCc1ccccc1 ZINC000217745541 DH For-Sale Unstable AMP1_PLAFQ 24 42 COc1ccccc1/C=C/NC(=O)NCCCc1ccccc1 ZINC000217745541 DH For-Sale Unstable CRTM 42 37 COc1ccccc1/C=C/NC(=O)NCCCc1ccccc1 ZINC000217745541 DH For-Sale Unstable AKR1B10 37 45 O=C(O)/C=C\c1cccc(NC(=O)c2ccc(Cl)o2)c1 ZINC000217745549 CG For-Sale Anodyne SCN10A 19 48 O=C(O)/C=C\c1cccc(NC(=O)c2ccc(Cl)o2)c1 ZINC000217745549 CG For-Sale Anodyne KCNK3 80 38 N=C(N)CC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217745553 BE In-Stock Unstable MAOB 18 40 N=C(N)CC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217745553 BE In-Stock Unstable CPN1 0 43 N=C(N)CC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217745553 BE In-Stock Unstable NPFFR2 18 43 N=C(N)CC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217745553 BE In-Stock Unstable SLC1A1 41 43 N=C(N)CC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217745553 BE In-Stock Unstable SLC1A3 42 43 N=C(N)CC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217745553 BE In-Stock Unstable SLC1A2 45 35 N=C(N)CC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217745553 BE In-Stock Unstable AGPAT2 46 36 N=C(N)CC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217745553 BE In-Stock Unstable MURB 0 40 N=C(N)CC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217745553 BE In-Stock Unstable SHH 56 40 N=C(N)CC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217745553 BE In-Stock Unstable PFK 0 45 N=C(N)CC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217745553 BE In-Stock Unstable ENPP1 41 32 N=C(N)CC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217745553 BE In-Stock Unstable IMDH_CRYPV 39 44 N=C(N)CC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217745553 BE In-Stock Unstable BLM 0 43 N=C(N)CC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217745553 BE In-Stock Unstable P95276_MYCTO 0 53 N=C(N)CC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217745553 BE In-Stock Unstable WRN 0 43 N=C(N)CC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217745553 BE In-Stock Unstable PPX1 0 51 CC(C)(C)c1ccc(S(=O)(=O)NCCC(=O)NC[C@H]2CCCN2c2nccs2)cc1 ZINC000217745565 JF For-Sale Unstable ADAMTS5 24 42 OC[C@@H]1CCCC[C@H]1CN[C@@H]1CCCc2cccnc21 ZINC000217745568 CF For-Sale Unstable CXCR4 62 36 Cc1ccccc1NS(=O)(=O)c1ccc(C)c(C(=O)N2CCN(CCN3CCCC3)CC2)c1 ZINC000217745602 JF On-Demand Unstable TRY2_BOVIN 45 34 Cc1ccccc1NS(=O)(=O)c1ccc(C)c(C(=O)N2CCN(CCN3CCCC3)CC2)c1 ZINC000217745602 JF On-Demand Unstable PRTN3 47 33 Cc1ccccc1NS(=O)(=O)c1ccc(C)c(C(=O)N2CCN(CCN3CCCC3)CC2)c1 ZINC000217745602 JF On-Demand Unstable CCR8 55 36 Cc1ccccc1NS(=O)(=O)c1ccc(C)c(C(=O)N2CCN(CCN3CCCC3)CC2)c1 ZINC000217745602 JF On-Demand Unstable MCL1 15 40 N#Cc1cn(-c2cccc(C(F)(F)F)c2)cn1 ZINC000217745617 BF In-Stock Mild CTSK 0 46 O=S1(=O)CCCN(S(=O)(=O)c2ccc(Cl)nc2)CC1 ZINC000217745618 DC On-Demand Unstable GCK 55 31 Cc1ccoc1C(=O)Nc1cccc(/C=C\C(=O)O)c1 ZINC000217745629 CF For-Sale Unstable HDAC8 18 40 Cc1ccoc1C(=O)Nc1cccc(/C=C\C(=O)O)c1 ZINC000217745629 CF For-Sale Unstable KCNK3 104 39 Cc1ccoc1C(=O)Nc1cccc(/C=C\C(=O)O)c1 ZINC000217745629 CF For-Sale Unstable KCNK9 61 39 COC(=O)C[C@@H](NC(=O)c1ccc(Cl)cn1)C(=O)O ZINC000217745634 CC On-Demand Unstable BLA1_STEMA 18 40 COc1ccc(OC)c2c1cc(C(=O)NC[C@@H]1CCCN3CCCC[C@H]13)n2C ZINC000217745641 GG In-Stock Unstable DRD3 0 40 COc1ccc(OC)c2c1cc(C(=O)NC[C@@H]1CCCN3CCCC[C@H]13)n2C ZINC000217745641 GG In-Stock Unstable ACKR3 63 32 COc1ccccc1/C=C/NC(=O)NCCCCc1ccccc1 ZINC000217745660 DH For-Sale Unstable DRD2 20 45 COc1ccccc1/C=C/NC(=O)NCCCCc1ccccc1 ZINC000217745660 DH For-Sale Unstable DRD3 33 45 COc1ccccc1/C=C/NC(=O)NCCCCc1ccccc1 ZINC000217745660 DH For-Sale Unstable SCN2A 17 45 COc1ccccc1/C=C/NC(=O)NCCCCc1ccccc1 ZINC000217745660 DH For-Sale Unstable MTNR1A 31 44 COc1ccccc1/C=C/NC(=O)NCCCCc1ccccc1 ZINC000217745660 DH For-Sale Unstable MTNR1B 34 43 COc1ccccc1/C=C/NC(=O)NCCCCc1ccccc1 ZINC000217745660 DH For-Sale Unstable FAAH 29 41 COc1ccccc1/C=C/NC(=O)NCCCCc1ccccc1 ZINC000217745660 DH For-Sale Unstable AMP1_PLAFQ 23 43 COc1ccccc1/C=C/NC(=O)NCCCCc1ccccc1 ZINC000217745660 DH For-Sale Unstable AKR1B10 36 44 O=C(O)/C=C\c1ccc(NC(=O)c2ccncc2)c(F)c1 ZINC000217745716 CF For-Sale Anodyne KCNK3 23 43 Cc1nc2cccc(CS(=O)(=O)Cl)c2o1 ZINC000217745733 BE For-Sale Unstable MTNR1A 15 50 Cc1nc2cccc(CS(=O)(=O)Cl)c2o1 ZINC000217745733 BE For-Sale Unstable MTNR1B 23 47 CN1CCN(Cc2ccc(O)cc2)[C@@H](c2ccccc2)C1 ZINC000217745745 CF On-Demand Unstable FABI 41 33 O=C(Cc1ccc(Br)cc1)N1CC(N2C(=O)CSC2=O)C1 ZINC000217745752 FD In-Stock Unstable GPR183 0 40 O=C(NCc1cccc(CNC(=O)c2cc(Cl)ccn2)c1)c1cc(Cl)ccn1 ZINC000217745776 HH On-Demand Unstable MMP13 23 55 O=C(NCc1cccc(CNC(=O)c2cc(Cl)ccn2)c1)c1cc(Cl)ccn1 ZINC000217745776 HH On-Demand Unstable ROCK1 18 43 O=C(NCc1cccc(CNC(=O)c2cc(Cl)ccn2)c1)c1cc(Cl)ccn1 ZINC000217745776 HH On-Demand Unstable GRM4 25 44 O=C(NCc1cccc(CNC(=O)c2cc(Cl)ccn2)c1)c1cc(Cl)ccn1 ZINC000217745776 HH On-Demand Unstable MAPK1 0 42 O=C(NCc1cccc(CNC(=O)c2cc(Cl)ccn2)c1)c1cc(Cl)ccn1 ZINC000217745776 HH On-Demand Unstable ROCK2 27 43 O=C(NCc1cccc(CNC(=O)c2cc(Cl)ccn2)c1)c1cc(Cl)ccn1 ZINC000217745776 HH On-Demand Unstable SCN10A 33 40 O=C(NCc1cccc(CNC(=O)c2cc(Cl)ccn2)c1)c1cc(Cl)ccn1 ZINC000217745776 HH On-Demand Unstable ISPE 0 43 O=C(NCc1cccc(CNC(=O)c2cc(Cl)ccn2)c1)c1cc(Cl)ccn1 ZINC000217745776 HH On-Demand Unstable PDS 54 38 N=C(N)CC(=O)Nc1cc(Cl)c(Cl)cc1Cl ZINC000217745783 CF In-Stock Unstable CA4 15 41 O=C(Cl)C(C(=O)Cl)c1cccc(C(F)(F)F)c1 ZINC000217745808 CG For-Sale Anodyne CES2 24 55 O=C(Cl)C(C(=O)Cl)c1cccc(C(F)(F)F)c1 ZINC000217745808 CG For-Sale Anodyne PDS 42 33 O=C(O)/C=C\c1ccc(NC(=O)c2cccnc2)c(F)c1 ZINC000217745811 CF For-Sale Anodyne TBXAS1 31 45 O=C(O)/C=C\c1ccc(NC(=O)c2cccnc2)c(F)c1 ZINC000217745811 CF For-Sale Anodyne HDAC1 0 50 COc1ccc(NC(=O)[C@@]23CC[C@@H]4C[C@@H](C[C@@H](C4)C2)C3)cc1 ZINC000217745848 CI In-Stock Unstable EPHX2 39 45 CO[C@@H]1[C@H]2CC[C@@H]1CN(C(=O)c1ccc3[nH]nnc3c1)C2 ZINC000217745854 CD In-Stock Unstable CHEK2 52 36 CO[C@@H]1[C@H]2CC[C@@H]1CN(C(=O)c1ccc3[nH]nnc3c1)C2 ZINC000217745854 CD In-Stock Unstable L3MBTL3 16 40 O=C(NCc1cccc(CNC(=O)c2ccc(F)c(F)c2)c1)c1ccc(F)c(F)c1 ZINC000217745866 HI On-Demand Unstable CHRM3 16 45 O=C(NCc1cccc(CNC(=O)c2ccc(F)c(F)c2)c1)c1ccc(F)c(F)c1 ZINC000217745866 HI On-Demand Unstable GRIN2B 26 45 O=C(NCc1cccc(CNC(=O)c2ccc(F)c(F)c2)c1)c1ccc(F)c(F)c1 ZINC000217745866 HI On-Demand Unstable MMP13 18 48 O=C(NCc1cccc(CNC(=O)c2ccc(F)c(F)c2)c1)c1ccc(F)c(F)c1 ZINC000217745866 HI On-Demand Unstable ROCK2 25 43 O=C(NCc1cccc(CNC(=O)c2ccc(F)c(F)c2)c1)c1ccc(F)c(F)c1 ZINC000217745866 HI On-Demand Unstable E1 0 40 O=C(NCc1cccc(CNC(=O)c2ccc(F)c(F)c2)c1)c1ccc(F)c(F)c1 ZINC000217745866 HI On-Demand Unstable TAAR1 15 46 O=C(NCc1cccc(CNC(=O)c2ccc(F)c(F)c2)c1)c1ccc(F)c(F)c1 ZINC000217745866 HI On-Demand Unstable PDS 41 34 O=C(NCc1cccc(CNC(=O)c2ccc(F)c(F)c2)c1)c1ccc(F)c(F)c1 ZINC000217745866 HI On-Demand Unstable Q76353_9HIV1 0 40 COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)ccc1O ZINC000217745878 II In-Stock Unstable AKR1B1 26 51 COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)ccc1O ZINC000217745878 II In-Stock Unstable CYP1B1 73 41 COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)ccc1O ZINC000217745878 II In-Stock Unstable CYP1A1 55 48 COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)ccc1O ZINC000217745878 II In-Stock Unstable CYP1A2 44 51 COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)ccc1O ZINC000217745878 II In-Stock Unstable ABCG2 0 40 COc1ccccc1/C=C/NC(=O)NCCC#N ZINC000217745884 BD For-Sale Unstable CYP1B1 19 40 N=C(N)CC(=O)Nc1ccc(F)cc1F ZINC000217745890 BD In-Stock Unstable CA1 19 49 N=C(N)CC(=O)Nc1ccc(F)cc1F ZINC000217745890 BD In-Stock Unstable CA5B 17 43 N=C(N)CC(=O)Nc1ccc(F)cc1F ZINC000217745890 BD In-Stock Unstable CA4 22 47 N=C(N)CC(=O)Nc1ccc(F)cc1F ZINC000217745890 BD In-Stock Unstable CA5A 20 43 COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)ccc1O ZINC000217745958 II In-Stock Unstable AKR1B1 26 51 COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)ccc1O ZINC000217745958 II In-Stock Unstable CYP1B1 73 41 COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)ccc1O ZINC000217745958 II In-Stock Unstable CYP1A1 55 48 COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)ccc1O ZINC000217745958 II In-Stock Unstable CYP1A2 44 51 COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)ccc1O ZINC000217745958 II In-Stock Unstable ABCG2 0 40 Cc1ccc(CC(=O)NCc2cccc(CNC(=O)Cc3ccc(C)cc3)c2)cc1 ZINC000217745968 HI On-Demand Unstable ANPEP 23 42 Cc1ccc(CC(=O)NCc2cccc(CNC(=O)Cc3ccc(C)cc3)c2)cc1 ZINC000217745968 HI On-Demand Unstable NQO2 30 40 Cc1ccc(CC(=O)NCc2cccc(CNC(=O)Cc3ccc(C)cc3)c2)cc1 ZINC000217745968 HI On-Demand Unstable TRPV1 20 41 Cc1ccc(CC(=O)NCc2cccc(CNC(=O)Cc3ccc(C)cc3)c2)cc1 ZINC000217745968 HI On-Demand Unstable P2RX7 41 48 Cc1ccc(CC(=O)NCc2cccc(CNC(=O)Cc3ccc(C)cc3)c2)cc1 ZINC000217745968 HI On-Demand Unstable CA5B 34 49 Cc1ccc(CC(=O)NCc2cccc(CNC(=O)Cc3ccc(C)cc3)c2)cc1 ZINC000217745968 HI On-Demand Unstable CA5A 39 49 Cc1ccc(CC(=O)NCc2cccc(CNC(=O)Cc3ccc(C)cc3)c2)cc1 ZINC000217745968 HI On-Demand Unstable ROCK2 32 40 Cc1ccc(CC(=O)NCc2cccc(CNC(=O)Cc3ccc(C)cc3)c2)cc1 ZINC000217745968 HI On-Demand Unstable FURIN 46 32 Cc1ccc(CC(=O)NCc2cccc(CNC(=O)Cc3ccc(C)cc3)c2)cc1 ZINC000217745968 HI On-Demand Unstable FBP1 15 43 Cc1ccc(CC(=O)NCc2cccc(CNC(=O)Cc3ccc(C)cc3)c2)cc1 ZINC000217745968 HI On-Demand Unstable TPSAB1 20 44 Cc1ccc(CC(=O)NCc2cccc(CNC(=O)Cc3ccc(C)cc3)c2)cc1 ZINC000217745968 HI On-Demand Unstable E1 0 47 Cc1ccc(CC(=O)NCc2cccc(CNC(=O)Cc3ccc(C)cc3)c2)cc1 ZINC000217745968 HI On-Demand Unstable NCE103 28 48 Cc1ccc(CC(=O)NCc2cccc(CNC(=O)Cc3ccc(C)cc3)c2)cc1 ZINC000217745968 HI On-Demand Unstable P96878_MYCTU 20 48 Cc1ccc(CC(=O)NCc2cccc(CNC(=O)Cc3ccc(C)cc3)c2)cc1 ZINC000217745968 HI On-Demand Unstable CAN2 0 48 Cc1ccc(CC(=O)NCc2cccc(CNC(=O)Cc3ccc(C)cc3)c2)cc1 ZINC000217745968 HI On-Demand Unstable PDS 47 36 COc1ccccc1/C=C/NC(=O)N1CCN(S(C)(=O)=O)CC1 ZINC000217745991 EC For-Sale Unstable TLR4 20 45 COc1ccc2c(ccn2CCNC(=O)C2(n3cnnn3)CCCCC2)c1 ZINC000217746060 FE In-Stock Unstable GRB2 29 42 COc1ccccc1/C=C/NC(=O)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217746093 HE For-Sale Unstable TGM2 67 40 COc1ccccc1/C=C/NC(=O)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217746093 HE For-Sale Unstable F13A1 87 40 COc1ccccc1/C=C/NC(=O)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217746093 HE For-Sale Unstable TLR4 19 42 COc1ccccc1/C=C/NC(=O)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217746093 HE For-Sale Unstable AKR1C3 47 45 N=C(N)CC(=O)Nc1ccc(Br)cc1F ZINC000217746100 CD In-Stock Unstable CA5B 18 41 N=C(N)CC(=O)Nc1ccc(Br)cc1F ZINC000217746100 CD In-Stock Unstable CA4 17 44 N=C(N)CC(=O)Nc1ccc(Br)cc1F ZINC000217746100 CD In-Stock Unstable CA5A 20 41 N=C(N)CC(=O)Nc1ccc(Br)cc1F ZINC000217746100 CD In-Stock Unstable MAP2K1 15 42 Cc1ccc(NC(=O)c2cccc(OC(F)(F)F)c2)cc1 ZINC000217746130 CI On-Demand Unstable PRSS1 15 41 Cc1ccc(NC(=O)c2cccc(OC(F)(F)F)c2)cc1 ZINC000217746130 CI On-Demand Unstable DHODH 27 44 Cc1ccc(NC(=O)c2cccc(OC(F)(F)F)c2)cc1 ZINC000217746130 CI On-Demand Unstable MAPK14 17 43 Cc1ccc(NC(=O)c2cccc(OC(F)(F)F)c2)cc1 ZINC000217746130 CI On-Demand Unstable TRPV1 22 56 Cc1ccc(NC(=O)c2cccc(OC(F)(F)F)c2)cc1 ZINC000217746130 CI On-Demand Unstable ECR 20 40 Cc1ccc(NC(=O)c2cccc(OC(F)(F)F)c2)cc1 ZINC000217746130 CI On-Demand Unstable P2RY1 52 33 Cc1ccc(NC(=O)c2cccc(OC(F)(F)F)c2)cc1 ZINC000217746130 CI On-Demand Unstable PRNP 56 39 Cc1ccc(NC(=O)c2cccc(OC(F)(F)F)c2)cc1 ZINC000217746130 CI On-Demand Unstable RAF1 35 44 Cc1ccc(NC(=O)c2cccc(OC(F)(F)F)c2)cc1 ZINC000217746130 CI On-Demand Unstable KDR 22 49 Cc1ccc(NC(=O)c2cccc(OC(F)(F)F)c2)cc1 ZINC000217746130 CI On-Demand Unstable CCR2 17 44 Cc1ccc(NC(=O)c2cccc(OC(F)(F)F)c2)cc1 ZINC000217746130 CI On-Demand Unstable P4HTM 0 40 Cc1ccc(NC(=O)c2cccc(OC(F)(F)F)c2)cc1 ZINC000217746130 CI On-Demand Unstable EPHX2 50 46 Cc1ccc(NC(=O)c2cccc(OC(F)(F)F)c2)cc1 ZINC000217746130 CI On-Demand Unstable SCN10A 48 50 Cc1ccc(NC(=O)c2cccc(OC(F)(F)F)c2)cc1 ZINC000217746130 CI On-Demand Unstable CSF1R 24 41 Cc1ccc(NC(=O)c2cccc(OC(F)(F)F)c2)cc1 ZINC000217746130 CI On-Demand Unstable TEK 34 49 Cc1ccc(NC(=O)c2cccc(OC(F)(F)F)c2)cc1 ZINC000217746130 CI On-Demand Unstable FABH 0 43 Cc1ccc(NC(=O)c2cccc(OC(F)(F)F)c2)cc1 ZINC000217746130 CI On-Demand Unstable MCHR1 18 41 Cc1ccc(NC(=O)c2cccc(OC(F)(F)F)c2)cc1 ZINC000217746130 CI On-Demand Unstable Q8MMZ8_EIMTE 43 44 Cc1ccc(NC(=O)c2cccc(OC(F)(F)F)c2)cc1 ZINC000217746130 CI On-Demand Unstable BTK 31 43 Cc1ccc(NC(=O)c2cccc(OC(F)(F)F)c2)cc1 ZINC000217746130 CI On-Demand Unstable BRAF 22 47 Cc1ccc(NC(=O)c2cccc(OC(F)(F)F)c2)cc1 ZINC000217746130 CI On-Demand Unstable TAAR1 47 49 Cc1ccc(NC(=O)c2cccc(OC(F)(F)F)c2)cc1 ZINC000217746130 CI On-Demand Unstable AKR1C3 26 43 Cc1ccc(NC(=O)c2cccc(OC(F)(F)F)c2)cc1 ZINC000217746130 CI On-Demand Unstable SHH 65 47 Cc1ccc(NC(=O)c2cccc(OC(F)(F)F)c2)cc1 ZINC000217746130 CI On-Demand Unstable NOD1 16 41 Cc1ccc(NC(=O)c2cccc(OC(F)(F)F)c2)cc1 ZINC000217746130 CI On-Demand Unstable NOD2 32 41 Cc1ccc(NC(=O)c2cccc(OC(F)(F)F)c2)cc1 ZINC000217746130 CI On-Demand Unstable SENP1 0 46 Cc1ccc(NC(=O)c2cccc(OC(F)(F)F)c2)cc1 ZINC000217746130 CI On-Demand Unstable KCNK3 105 54 Cc1ccc(NC(=O)c2cccc(OC(F)(F)F)c2)cc1 ZINC000217746130 CI On-Demand Unstable KCNK9 98 54 Cc1ccc(NC(=O)c2cccc(OC(F)(F)F)c2)cc1 ZINC000217746130 CI On-Demand Unstable BRPF1 0 45 C[C@]12C[C@@H]3C[C@](C)(C1)C[C@@](CNC(=O)COc1ccccc1)(C3)C2 ZINC000217746136 EI In-Stock Unstable P2RX7 0 40 C[C@]12C[C@@H]3C[C@](C)(C1)C[C@@](CNC(=O)COc1ccccc1)(C3)C2 ZINC000217746136 EI In-Stock Unstable LUXN 0 40 N#Cc1cccc(S(=O)(=O)N2CCCS(=O)(=O)CC2)c1 ZINC000217746162 DC On-Demand Unstable PKM 23 41 N#Cc1cccc(S(=O)(=O)N2CCCS(=O)(=O)CC2)c1 ZINC000217746162 DC On-Demand Unstable AKR1C3 41 42 O=C1N[C@@H](CCC(=O)N2CCN(Cc3nc4ccccc4c(=O)[nH]3)CC2)C(=O)Nc2ccccc21 ZINC000217746185 JD In-Stock Unstable PARP1 22 51 N=C(N)CC(=O)Nc1ccc(F)c(Cl)c1 ZINC000217746221 BD In-Stock Unstable MAOB 16 42 N=C(N)CC(=O)Nc1ccc(F)c(Cl)c1 ZINC000217746221 BD In-Stock Unstable SLC1A1 49 46 N=C(N)CC(=O)Nc1ccc(F)c(Cl)c1 ZINC000217746221 BD In-Stock Unstable SLC1A3 50 45 N=C(N)CC(=O)Nc1ccc(F)c(Cl)c1 ZINC000217746221 BD In-Stock Unstable SLC1A2 55 46 N=C(N)CC(=O)Nc1ccc(F)c(Cl)c1 ZINC000217746221 BD In-Stock Unstable AGPAT2 41 36 N=C(N)CC(=O)Nc1ccc(F)c(Cl)c1 ZINC000217746221 BD In-Stock Unstable ERBB4 42 38 N=C(N)CC(=O)Nc1ccc(F)c(Cl)c1 ZINC000217746221 BD In-Stock Unstable ENV 42 32 N=C(N)CC(=O)Nc1ccc(F)c(Cl)c1 ZINC000217746221 BD In-Stock Unstable MCHR1 15 41 Cc1ccc(/C=C\C(=O)N2CC(=O)NC(=O)C2)cc1Cl ZINC000217746256 CD For-Sale Unstable ITGAL 23 48 O=C(CCc1cccc(OCc2ccccc2)c1)NC[C@@H]1CCCN1c1nccs1 ZINC000217746271 HI For-Sale Unstable GRIN2B 17 41 O=C(CCc1cccc(OCc2ccccc2)c1)NC[C@@H]1CCCN1c1nccs1 ZINC000217746271 HI For-Sale Unstable FFAR1 16 40 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1cccc(OC(F)F)c1 ZINC000217746276 CK For-Sale Unstable TRPM8 18 50 O=S1(=O)CCCN(S(=O)(=O)c2cccc(Br)c2)CC1 ZINC000217746285 FD On-Demand Unstable AKR1C3 48 39 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](CC(C)C)C(=O)NCCN(C)C)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217746313 KG In-Stock Unstable TUBA1A 18 66 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](CC(C)C)C(=O)NCCN(C)C)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217746313 KG In-Stock Unstable TPPP 0 63 N=C(N)CC(=O)Nc1ccccc1C(F)(F)F ZINC000217746322 BD In-Stock Unstable KCNJ11 59 34 N=C(N)CC(=O)Nc1ccccc1C(F)(F)F ZINC000217746322 BD In-Stock Unstable TRPV1 17 48 N=C(N)CC(=O)Nc1ccccc1C(F)(F)F ZINC000217746322 BD In-Stock Unstable RBP4 41 36 O=C(CCc1cccc(OCc2ccccc2)c1)NC[C@H]1CCCN1c1nccs1 ZINC000217746353 HI For-Sale Unstable GRIN2B 17 41 O=C(CCc1cccc(OCc2ccccc2)c1)NC[C@H]1CCCN1c1nccs1 ZINC000217746353 HI For-Sale Unstable FFAR1 16 40 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1cccc(OC(F)F)c1 ZINC000217746363 CK For-Sale Unstable TRPM8 18 50 NC(=O)c1ncn2c(C(=O)NC34CC5CC(CC(C5)C3)C4)cc(-c3ccco3)nc12 ZINC000217746371 HF On-Demand Unstable CNR2 20 45 CC[C@@H](C)C(=O)N[C@@H](C)c1cccc(/C=C\C(=O)O)c1 ZINC000217746415 CG For-Sale Unstable ACE2 46 35 N=C(N)CC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217746417 BD In-Stock Unstable LCK 28 40 N=C(N)CC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217746417 BD In-Stock Unstable F2R 0 43 N=C(N)CC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217746417 BD In-Stock Unstable KDR 17 47 N=C(N)CC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217746417 BD In-Stock Unstable HDAC3 16 40 N=C(N)CC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217746417 BD In-Stock Unstable HDAC6 15 60 N=C(N)CC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217746417 BD In-Stock Unstable SLC1A1 31 47 N=C(N)CC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217746417 BD In-Stock Unstable SLC1A3 30 47 N=C(N)CC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217746417 BD In-Stock Unstable ACR 21 48 N=C(N)CC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217746417 BD In-Stock Unstable SLC1A2 38 47 N=C(N)CC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217746417 BD In-Stock Unstable EPHA3 24 43 N=C(N)CC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217746417 BD In-Stock Unstable BTK 23 43 N=C(N)CC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217746417 BD In-Stock Unstable EPHB4 29 43 N=C(N)CC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217746417 BD In-Stock Unstable RIPK1 41 41 N=C(N)CC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217746417 BD In-Stock Unstable KCNK3 48 35 N=C(N)CC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217746417 BD In-Stock Unstable KCNK9 49 36 N=C(N)CC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217746417 BD In-Stock Unstable PDS 39 41 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1cccc(OC(F)F)c1 ZINC000217746447 CK For-Sale Unstable TRPM8 18 50 Nc1nnc(SCC(=O)NC2CCN(Cc3ccncc3)CC2)s1 ZINC000217746464 FD In-Stock Unstable SIGMAR1 24 47 Nc1nnc(SCC(=O)NC2CCN(Cc3ccncc3)CC2)s1 ZINC000217746464 FD In-Stock Unstable SSTR5 42 35 O=C(CCc1ccc(OCc2ccccc2)cc1)NC[C@@H]1CCCN1c1nccs1 ZINC000217746470 HI For-Sale Unstable GRIN2B 20 42 O=C(CCc1ccc(OCc2ccccc2)cc1)NC[C@@H]1CCCN1c1nccs1 ZINC000217746470 HI For-Sale Unstable PREP 43 40 O=C(CCc1ccc(OCc2ccccc2)cc1)NC[C@@H]1CCCN1c1nccs1 ZINC000217746470 HI For-Sale Unstable FFAR1 25 43 NC(=O)c1ncn2c(C(=O)Nc3nc(-c4ccccc4)cs3)cc(-c3ccco3)nc12 ZINC000217746485 IG On-Demand Unstable ADORA1 0 45 NC(=O)c1ncn2c(C(=O)Nc3nc(-c4ccccc4)cs3)cc(-c3ccco3)nc12 ZINC000217746485 IG On-Demand Unstable TRPA1 19 40 CC[C@H](C)C(=O)N[C@@H](C)c1cccc(/C=C\C(=O)O)c1 ZINC000217746503 CG For-Sale Unstable ACE2 46 35 N=C(N)CC(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217746512 BD In-Stock Unstable DHODH 33 43 N=C(N)CC(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217746512 BD In-Stock Unstable TRPV1 17 50 N=C(N)CC(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217746512 BD In-Stock Unstable ATF1 17 43 N=C(N)CC(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217746512 BD In-Stock Unstable NFKB1 16 43 N=C(N)CC(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217746512 BD In-Stock Unstable SLC1A1 32 42 N=C(N)CC(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217746512 BD In-Stock Unstable SLC1A3 27 42 N=C(N)CC(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217746512 BD In-Stock Unstable ACR 48 53 N=C(N)CC(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217746512 BD In-Stock Unstable SLC1A2 54 43 N=C(N)CC(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217746512 BD In-Stock Unstable MCHR1 23 42 N=C(N)CC(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217746512 BD In-Stock Unstable KIF11 22 60 N=C(N)CC(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217746512 BD In-Stock Unstable MTCA1 15 50 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1cccc(OC(F)F)c1 ZINC000217746520 CK For-Sale Unstable TRPM8 18 50 O=C(CCc1ccc(OCc2ccccc2)cc1)NC[C@H]1CCCN1c1nccs1 ZINC000217746535 HI For-Sale Unstable GRIN2B 20 42 O=C(CCc1ccc(OCc2ccccc2)cc1)NC[C@H]1CCCN1c1nccs1 ZINC000217746535 HI For-Sale Unstable PREP 43 40 O=C(CCc1ccc(OCc2ccccc2)cc1)NC[C@H]1CCCN1c1nccs1 ZINC000217746535 HI For-Sale Unstable FFAR1 25 43 C/C(=N\O)c1ccc(NC(=O)c2ccc(Cl)cn2)cc1 ZINC000217746575 CG For-Sale Unstable BACE2 36 42 C/C(=N\O)c1ccc(NC(=O)c2ccc(Cl)cn2)cc1 ZINC000217746575 CG For-Sale Unstable GRM4 41 35 C/C(=N\O)c1ccc(NC(=O)c2ccc(Cl)cn2)cc1 ZINC000217746575 CG For-Sale Unstable P4HTM 0 47 C/C(=N\O)c1ccc(NC(=O)c2ccc(Cl)cn2)cc1 ZINC000217746575 CG For-Sale Unstable BACE1 16 42 O=C1CN(C(=O)/C=C\c2ccc(F)c(Cl)c2)CC(=O)N1 ZINC000217746576 CC For-Sale Unstable CCR2 56 41 O=C1CN(C(=O)/C=C\c2ccc(F)c(Cl)c2)CC(=O)N1 ZINC000217746576 CC For-Sale Unstable GPR183 0 44 N=C(N)CC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217746595 CF In-Stock Unstable TRPV1 15 54 N=C(N)CC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217746595 CF In-Stock Unstable NPFFR2 15 50 N=C(N)CC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217746595 CF In-Stock Unstable GUAB 0 44 N=C(N)CC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217746595 CF In-Stock Unstable RAF1 26 43 N=C(N)CC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217746595 CF In-Stock Unstable FLT1 17 44 N=C(N)CC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217746595 CF In-Stock Unstable SLC1A1 37 45 N=C(N)CC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217746595 CF In-Stock Unstable SLC1A3 42 45 N=C(N)CC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217746595 CF In-Stock Unstable SLC1A2 43 34 N=C(N)CC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217746595 CF In-Stock Unstable ENV 40 31 N=C(N)CC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217746595 CF In-Stock Unstable Q8MMZ8_EIMTE 51 47 N=C(N)CC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217746595 CF In-Stock Unstable BRAF 15 43 N=C(N)CC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217746595 CF In-Stock Unstable PTPA 0 51 N=C(N)CC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217746595 CF In-Stock Unstable SHH 42 36 N=C(N)CC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217746595 CF In-Stock Unstable PFK 0 41 N=C(N)CC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217746595 CF In-Stock Unstable IMDH_CRYPV 27 51 N=C(N)CC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217746595 CF In-Stock Unstable BLM 0 48 NC(=O)c1ncn2c(C(=O)Nc3ccc(-c4nc5ccccc5[nH]4)cc3)cc(-c3ccco3)nc12 ZINC000217746603 JH On-Demand Unstable CHEK2 53 44 NC(=O)c1ncn2c(C(=O)Nc3ccc(-c4nc5ccccc5[nH]4)cc3)cc(-c3ccco3)nc12 ZINC000217746603 JH On-Demand Unstable HPSE 24 45 NC(=O)c1ncn2c(C(=O)Nc3ccc(-c4nc5ccccc5[nH]4)cc3)cc(-c3ccco3)nc12 ZINC000217746603 JH On-Demand Unstable NR2E3 71 38 COc1ccc(CCC(=O)NC[C@@H]2CCCN2c2nccs2)cc1OCc1ccccc1 ZINC000217746646 JI For-Sale Unstable SSTR5 40 35 COc1ccccc1/C=C/NC(=O)NCCNC(=O)OC(C)(C)C ZINC000217746668 EE For-Sale Unstable DRD3 18 41 COc1ccccc1/C=C/NC(=O)NCCNC(=O)OC(C)(C)C ZINC000217746668 EE For-Sale Unstable MTNR1B 15 41 C/C(=N\O)c1cccc(NC(=O)c2ccc(Cl)cn2)c1 ZINC000217746681 CG For-Sale Unstable PPIA 22 43 C/C(=N\O)c1cccc(NC(=O)c2ccc(Cl)cn2)c1 ZINC000217746681 CG For-Sale Unstable F10 31 40 C/C(=N\O)c1cccc(NC(=O)c2ccc(Cl)cn2)c1 ZINC000217746681 CG For-Sale Unstable BACE2 44 46 C/C(=N\O)c1cccc(NC(=O)c2ccc(Cl)cn2)c1 ZINC000217746681 CG For-Sale Unstable GUAB 0 47 C/C(=N\O)c1cccc(NC(=O)c2ccc(Cl)cn2)c1 ZINC000217746681 CG For-Sale Unstable JAK1 0 40 C/C(=N\O)c1cccc(NC(=O)c2ccc(Cl)cn2)c1 ZINC000217746681 CG For-Sale Unstable GRM4 55 45 C/C(=N\O)c1cccc(NC(=O)c2ccc(Cl)cn2)c1 ZINC000217746681 CG For-Sale Unstable GRM5 17 41 C/C(=N\O)c1cccc(NC(=O)c2ccc(Cl)cn2)c1 ZINC000217746681 CG For-Sale Unstable BACE1 29 51 C/C(=N\O)c1cccc(NC(=O)c2ccc(Cl)cn2)c1 ZINC000217746681 CG For-Sale Unstable SCN10A 32 41 C/C(=N\O)c1cccc(NC(=O)c2ccc(Cl)cn2)c1 ZINC000217746681 CG For-Sale Unstable TYK2 29 40 C/C(=N\O)c1cccc(NC(=O)c2ccc(Cl)cn2)c1 ZINC000217746681 CG For-Sale Unstable CSF1R 27 41 C/C(=N\O)c1cccc(NC(=O)c2ccc(Cl)cn2)c1 ZINC000217746681 CG For-Sale Unstable TAAR1 19 42 C/C(=N\O)c1cccc(NC(=O)c2ccc(Cl)cn2)c1 ZINC000217746681 CG For-Sale Unstable IMDH_CRYPV 43 41 C/C(=N\O)c1cccc(NC(=O)c2ccc(Cl)cn2)c1 ZINC000217746681 CG For-Sale Unstable KCNK3 123 45 C/C(=N\O)c1cccc(NC(=O)c2ccc(Cl)cn2)c1 ZINC000217746681 CG For-Sale Unstable KCNK9 83 43 N=C(N)CC(=O)Nc1cc(C(F)(F)F)ccc1Cl ZINC000217746699 CF In-Stock Unstable CSNK1D 27 40 N=C(N)CC(=O)Nc1cc(C(F)(F)F)ccc1Cl ZINC000217746699 CF In-Stock Unstable ATF1 53 33 N=C(N)CC(=O)Nc1cc(C(F)(F)F)ccc1Cl ZINC000217746699 CF In-Stock Unstable NFKB1 49 33 NC(=O)c1ncn2c(C(=O)NC(c3ccccc3)c3ccccc3)cc(-c3ccco3)nc12 ZINC000217746715 IH On-Demand Unstable ADORA1 0 40 NC(=O)c1ncn2c(C(=O)NC(c3ccccc3)c3ccccc3)cc(-c3ccco3)nc12 ZINC000217746715 IH On-Demand Unstable ADORA3 0 40 CC(C)C[C@@H]1NC(=O)[C@H]2CCN2C1=O ZINC000217746726 AC For-Sale Unstable AVPR2 0 40 CC(C)C[C@@H]1NC(=O)[C@H]2CCN2C1=O ZINC000217746726 AC For-Sale Unstable OXTR 15 41 CC(C)C[C@@H]1NC(=O)[C@H]2CCN2C1=O ZINC000217746726 AC For-Sale Unstable HDAC4 0 40 COc1ccc(CCC(=O)NC[C@H]2CCCN2c2nccs2)cc1OCc1ccccc1 ZINC000217746739 JI For-Sale Unstable SSTR5 40 35 C/C(=N\O)c1ccccc1NC(=O)c1ccc(Cl)cn1 ZINC000217746749 CG For-Sale Unstable F10 38 47 C/C(=N\O)c1ccccc1NC(=O)c1ccc(Cl)cn1 ZINC000217746749 CG For-Sale Unstable EPHB3 51 34 C/C(=N\O)c1ccccc1NC(=O)c1ccc(Cl)cn1 ZINC000217746749 CG For-Sale Unstable G2YM83_BOTF4 59 34 COc1ccccc1NC(=O)CC(=N)N ZINC000217746804 BC In-Stock Unstable ACR 27 47 COc1ccccc1NC(=O)CC(=N)N ZINC000217746804 BC In-Stock Unstable KCNK3 46 42 COc1ccccc1NC(=O)CC(=N)N ZINC000217746804 BC In-Stock Unstable KCNK9 35 42 CC(C)C[C@H]1NC(=O)[C@@H]2CCN2C1=O ZINC000217746819 AC For-Sale Unstable AVPR2 0 40 CC(C)C[C@H]1NC(=O)[C@@H]2CCN2C1=O ZINC000217746819 AC For-Sale Unstable OXTR 15 41 CC(C)C[C@H]1NC(=O)[C@@H]2CCN2C1=O ZINC000217746819 AC For-Sale Unstable HDAC4 0 40 COc1ccccc1/C=C/NC(=O)NC1CCN(C(=O)OC(C)(C)C)CC1 ZINC000217746879 GG For-Sale Unstable CCR8 20 42 COc1ccccc1/C=C/NC(=O)NC1CCN(C(=O)OC(C)(C)C)CC1 ZINC000217746879 GG For-Sale Unstable GPR119 35 41 CC(C)C[C@@H]1NC(=O)[C@@H]2CCN2C1=O ZINC000217746886 AC For-Sale Unstable AVPR2 0 40 CC(C)C[C@@H]1NC(=O)[C@@H]2CCN2C1=O ZINC000217746886 AC For-Sale Unstable OXTR 15 41 CC(C)C[C@@H]1NC(=O)[C@@H]2CCN2C1=O ZINC000217746886 AC For-Sale Unstable HDAC4 0 40 COc1cccc(CN[C@@H]2CCN3CCC[C@@H]23)c1O ZINC000217746899 CD For-Sale Unstable TACR3 25 41 CCOc1ccc(-n2cnc(C#N)c2)cc1 ZINC000217746915 BE In-Stock Unstable CACNA2D1 57 41 CCOc1ccc(-n2cnc(C#N)c2)cc1 ZINC000217746915 BE In-Stock Unstable CACNA2D2 52 33 CCOc1ccc(-n2cnc(C#N)c2)cc1 ZINC000217746915 BE In-Stock Unstable CYP2C19 17 40 COc1cccc(NC(=O)CC(=N)N)c1 ZINC000217746923 BC In-Stock Unstable PRSS1 22 51 COc1cccc(NC(=O)CC(=N)N)c1 ZINC000217746923 BC In-Stock Unstable DRD4 42 33 COc1cccc(NC(=O)CC(=N)N)c1 ZINC000217746923 BC In-Stock Unstable F10 17 45 COc1cccc(NC(=O)CC(=N)N)c1 ZINC000217746923 BC In-Stock Unstable PDGFRB 18 44 COc1cccc(NC(=O)CC(=N)N)c1 ZINC000217746923 BC In-Stock Unstable PTGER3 15 43 COc1cccc(NC(=O)CC(=N)N)c1 ZINC000217746923 BC In-Stock Unstable MTNR1A 55 58 COc1cccc(NC(=O)CC(=N)N)c1 ZINC000217746923 BC In-Stock Unstable MTNR1B 51 58 COc1cccc(NC(=O)CC(=N)N)c1 ZINC000217746923 BC In-Stock Unstable FLT4 21 41 COc1cccc(NC(=O)CC(=N)N)c1 ZINC000217746923 BC In-Stock Unstable PLAU 28 60 COc1cccc(NC(=O)CC(=N)N)c1 ZINC000217746923 BC In-Stock Unstable ACR 46 41 COc1cccc(NC(=O)CC(=N)N)c1 ZINC000217746923 BC In-Stock Unstable FPR2 21 40 COc1cccc(NC(=O)CC(=N)N)c1 ZINC000217746923 BC In-Stock Unstable TAAR1 36 50 COc1cccc(NC(=O)CC(=N)N)c1 ZINC000217746923 BC In-Stock Unstable AKR1C3 23 46 COc1cccc(NC(=O)CC(=N)N)c1 ZINC000217746923 BC In-Stock Unstable AKR1C2 50 37 COc1cccc(NC(=O)CC(=N)N)c1 ZINC000217746923 BC In-Stock Unstable ENPP1 57 34 COc1cccc(NC(=O)CC(=N)N)c1 ZINC000217746923 BC In-Stock Unstable LIMK2 15 40 COc1cccc(NC(=O)CC(=N)N)c1 ZINC000217746923 BC In-Stock Unstable NAMPT 0 41 COc1cccc(NC(=O)CC(=N)N)c1 ZINC000217746923 BC In-Stock Unstable KCNK3 69 47 COc1cccc(NC(=O)CC(=N)N)c1 ZINC000217746923 BC In-Stock Unstable KCNK9 76 47 CN1CCN(c2cc(C(F)(F)F)cc(Cl)n2)CC1 ZINC000217746948 CF In-Stock Unstable HRH4 55 45 CN1CCN(c2cc(C(F)(F)F)cc(Cl)n2)CC1 ZINC000217746948 CF In-Stock Unstable MET 18 44 NC(=O)c1ncn2c(C(=O)Nc3nc(-c4ccc(Cl)cc4)cs3)cc(-c3ccco3)nc12 ZINC000217746963 JI On-Demand Unstable ADORA1 0 45 NC(=O)c1ncn2c(C(=O)Nc3nc(-c4ccc(Cl)cc4)cs3)cc(-c3ccco3)nc12 ZINC000217746963 JI On-Demand Unstable MPL 37 41 NC(=O)c1ncn2c(C(=O)Nc3nc(-c4ccc(Cl)cc4)cs3)cc(-c3ccco3)nc12 ZINC000217746963 JI On-Demand Unstable TRPA1 17 42 COc1cccc(CN[C@H]2CCN3CCC[C@@H]23)c1O ZINC000217746978 CD For-Sale Unstable TACR3 25 41 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)c(OC)c1OC ZINC000217746988 JI In-Stock Unstable AKR1B1 22 48 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)c(OC)c1OC ZINC000217746988 JI In-Stock Unstable CYP1B1 73 40 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)c(OC)c1OC ZINC000217746988 JI In-Stock Unstable CYP1A1 56 41 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)c(OC)c1OC ZINC000217746988 JI In-Stock Unstable CYP1A2 47 50 COc1ccc(NC(=O)N/C=C/c2ccccc2F)cc1OC ZINC000217746991 DH For-Sale Unstable HTR2A 15 40 COc1ccc(NC(=O)N/C=C/c2ccccc2F)cc1OC ZINC000217746991 DH For-Sale Unstable GRM4 15 43 COc1ccc(NC(=O)N/C=C/c2ccccc2F)cc1OC ZINC000217746991 DH For-Sale Unstable PDGFRA 42 39 COc1ccc(NC(=O)N/C=C/c2ccccc2F)cc1OC ZINC000217746991 DH For-Sale Unstable TLR4 16 40 COc1ccc(NC(=O)N/C=C/c2ccccc2F)cc1OC ZINC000217746991 DH For-Sale Unstable ENPP1 70 34 COc1ccccc1CCN1[C@H]2CC[C@H]1CC(N)C2 ZINC000217747016 CE For-Sale Unstable SLC18A2 26 45 COc1ccccc1CCN1[C@H]2CC[C@H]1CC(N)C2 ZINC000217747016 CE For-Sale Unstable MBTPS1 40 35 COc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217747034 BC In-Stock Unstable CA2 22 50 COc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217747034 BC In-Stock Unstable PRSS1 21 57 COc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217747034 BC In-Stock Unstable LTA4H 37 43 COc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217747034 BC In-Stock Unstable CA1 50 38 COc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217747034 BC In-Stock Unstable MTNR1A 40 47 COc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217747034 BC In-Stock Unstable MTNR1B 36 49 COc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217747034 BC In-Stock Unstable NPY5R 15 40 COc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217747034 BC In-Stock Unstable PLAU 27 44 COc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217747034 BC In-Stock Unstable F7 20 45 COc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217747034 BC In-Stock Unstable ACR 67 43 COc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217747034 BC In-Stock Unstable CA12 27 50 COc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217747034 BC In-Stock Unstable CA9 28 50 COc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217747034 BC In-Stock Unstable AKR1C3 18 40 COc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217747034 BC In-Stock Unstable PROKR1 51 32 COc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217747034 BC In-Stock Unstable AKR1C2 41 40 COc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217747034 BC In-Stock Unstable ENPP1 60 34 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)c(OC)c1OC ZINC000217747071 JI In-Stock Unstable AKR1B1 22 48 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)c(OC)c1OC ZINC000217747071 JI In-Stock Unstable CYP1B1 73 40 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)c(OC)c1OC ZINC000217747071 JI In-Stock Unstable CYP1A1 56 41 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)c(OC)c1OC ZINC000217747071 JI In-Stock Unstable CYP1A2 47 50 Cc1nc(-c2cccs2)ccc1C(=O)Nc1ccc(N2CCOCC2)cc1N1CCOCC1 ZINC000217747077 JI On-Demand Unstable CSF1R 18 44 O=C(c1ccc(S(=O)(=O)N2CCCC2)cc1)N1CC(N2C(=O)CSC2=O)C1 ZINC000217747088 HC In-Stock Unstable TGM2 44 39 O=C(c1ccc(S(=O)(=O)N2CCCC2)cc1)N1CC(N2C(=O)CSC2=O)C1 ZINC000217747088 HC In-Stock Unstable L3MBTL1 0 52 O=C(c1ccc(S(=O)(=O)N2CCCC2)cc1)N1CC(N2C(=O)CSC2=O)C1 ZINC000217747088 HC In-Stock Unstable L3MBTL3 60 52 O=C(c1ccc(S(=O)(=O)N2CCCC2)cc1)N1CC(N2C(=O)CSC2=O)C1 ZINC000217747088 HC In-Stock Unstable MBTD1 0 52 O=C(N/C=C/c1ccccc1F)NCCCN1CCCC1=O ZINC000217747104 DE For-Sale Unstable TYRO3 26 45 CCOc1ccccc1NC(=O)CC(=N)N ZINC000217747143 BD In-Stock Unstable HCN1 40 31 CCOc1ccccc1NC(=O)CC(=N)N ZINC000217747143 BD In-Stock Unstable KCNK3 34 43 CCOc1ccccc1NC(=O)CC(=N)N ZINC000217747143 BD In-Stock Unstable KCNK9 30 43 O=C(O)c1ccnc(NS(=O)(=O)/C=C\c2ccccc2)c1 ZINC000217747195 DE On-Demand Anodyne FTO 0 40 O=S1(=O)CCCN(S(=O)(=O)c2ccccc2F)CC1 ZINC000217747199 DC On-Demand Unstable PKM 20 46 O=C(C[C@@H]1NC(=O)N(Cc2cccc(F)c2)C1=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217747202 ID In-Stock Unstable CHRNA4 29 50 CCOc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217747248 BD In-Stock Unstable CA2 18 43 CCOc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217747248 BD In-Stock Unstable PRSS1 15 47 CCOc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217747248 BD In-Stock Unstable LTA4H 37 42 CCOc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217747248 BD In-Stock Unstable CA1 35 40 CCOc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217747248 BD In-Stock Unstable SCN2A 40 46 CCOc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217747248 BD In-Stock Unstable PRNP 16 51 CCOc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217747248 BD In-Stock Unstable ACR 65 41 CCOc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217747248 BD In-Stock Unstable CA12 22 43 CCOc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217747248 BD In-Stock Unstable CA9 22 43 CCOc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217747248 BD In-Stock Unstable PPO2 48 42 CCOc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217747248 BD In-Stock Unstable NCE103 19 43 Cn1cc(C(=O)Nc2cccc(/C=C\C(=O)O)n2)cn1 ZINC000217747281 CD For-Sale Unstable MAP3K5 45 35 COc1cccc(CCN2[C@H]3CC[C@H]2CC(N)C3)c1 ZINC000217747296 CE For-Sale Unstable SLC6A3 17 40 COc1cccc(CCN2[C@H]3CC[C@H]2CC(N)C3)c1 ZINC000217747296 CE For-Sale Unstable SLC18A2 37 47 COc1cccc(CCN2[C@H]3CC[C@H]2CC(N)C3)c1 ZINC000217747296 CE For-Sale Unstable KCNH2 38 48 COc1cccc(CCN2[C@H]3CC[C@H]2CC(N)C3)c1 ZINC000217747296 CE For-Sale Unstable SIGMAR1 20 57 COc1cccc(CCN2[C@H]3CC[C@H]2CC(N)C3)c1 ZINC000217747296 CE For-Sale Unstable ACHP_LYMST 19 44 COc1cccc(CCN2[C@H]3CC[C@H]2CC(N)C3)c1 ZINC000217747296 CE For-Sale Unstable Q8WSF8_APLCA 17 44 CC(=O)c1cccc(S(=O)(=O)N2CCCS(=O)(=O)CC2)c1 ZINC000217747323 EC On-Demand Unstable AKR1C3 73 46 CC(=O)c1cccc(S(=O)(=O)N2CCCS(=O)(=O)CC2)c1 ZINC000217747323 EC On-Demand Unstable AKR1C1 22 42 O=C(N/C=C/c1ccccc1F)Nc1cccc(C(=O)O)c1 ZINC000217747328 DG For-Sale Anodyne EPHX2 16 43 O=C(N/C=C/c1ccccc1F)Nc1cccc(C(=O)O)c1 ZINC000217747328 DG For-Sale Anodyne AKR1C3 32 47 O=C(N/C=C/c1ccccc1F)Nc1cccc(C(=O)O)c1 ZINC000217747328 DG For-Sale Anodyne KCNK3 78 42 O=C(N/C=C/c1ccccc1F)Nc1cccc(C(=O)O)c1 ZINC000217747328 DG For-Sale Anodyne KCNK9 40 36 COc1ccc2cc(C(=O)N3CC(N4C(=O)CSC4=O)C3)[nH]c2c1 ZINC000217747333 ED In-Stock Unstable GRIN2B 17 46 COc1ccc2cc(C(=O)N3CC(N4C(=O)CSC4=O)C3)[nH]c2c1 ZINC000217747333 ED In-Stock Unstable FPR2 28 45 NC(=O)c1ncn2c(C(=O)Nc3ncc(Cc4ccccc4Cl)s3)cc(-c3ccco3)nc12 ZINC000217747351 JI On-Demand Unstable ADORA1 0 42 NC(=O)c1ncn2c(C(=O)Nc3ncc(Cc4ccccc4Cl)s3)cc(-c3ccco3)nc12 ZINC000217747351 JI On-Demand Unstable ADORA2A 16 42 NC(=O)c1ncn2c(C(=O)Nc3ncc(Cc4ccccc4Cl)s3)cc(-c3ccco3)nc12 ZINC000217747351 JI On-Demand Unstable ADORA3 0 42 N=C(N)CC(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217747359 CF In-Stock Unstable CA2 15 59 N=C(N)CC(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217747359 CF In-Stock Unstable PRSS1 16 43 N=C(N)CC(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217747359 CF In-Stock Unstable ADRB1 21 43 N=C(N)CC(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217747359 CF In-Stock Unstable TSHR 50 35 N=C(N)CC(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217747359 CF In-Stock Unstable MAOB 24 40 N=C(N)CC(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217747359 CF In-Stock Unstable PPIA 48 40 N=C(N)CC(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217747359 CF In-Stock Unstable EPOR 0 40 N=C(N)CC(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217747359 CF In-Stock Unstable LTA4H 65 67 N=C(N)CC(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217747359 CF In-Stock Unstable HRAS 48 32 N=C(N)CC(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217747359 CF In-Stock Unstable CA1 38 59 N=C(N)CC(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217747359 CF In-Stock Unstable CA7 19 47 N=C(N)CC(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217747359 CF In-Stock Unstable SCN2A 31 56 N=C(N)CC(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217747359 CF In-Stock Unstable SLC15A1 0 43 N=C(N)CC(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217747359 CF In-Stock Unstable ADAM17 21 52 N=C(N)CC(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217747359 CF In-Stock Unstable S1PR4 23 45 N=C(N)CC(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217747359 CF In-Stock Unstable HDAC8 16 42 N=C(N)CC(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217747359 CF In-Stock Unstable CA5B 35 43 N=C(N)CC(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217747359 CF In-Stock Unstable CA5A 40 43 N=C(N)CC(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217747359 CF In-Stock Unstable S1PR1 0 45 N=C(N)CC(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217747359 CF In-Stock Unstable PLAU 37 41 N=C(N)CC(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217747359 CF In-Stock Unstable F7 17 41 N=C(N)CC(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217747359 CF In-Stock Unstable ACR 55 43 N=C(N)CC(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217747359 CF In-Stock Unstable CA12 22 59 N=C(N)CC(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217747359 CF In-Stock Unstable SLC1A2 30 42 N=C(N)CC(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217747359 CF In-Stock Unstable C5AR1 0 40 N=C(N)CC(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217747359 CF In-Stock Unstable ADAMTS4 37 40 N=C(N)CC(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217747359 CF In-Stock Unstable CA9 22 59 N=C(N)CC(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217747359 CF In-Stock Unstable TAAR1 19 43 N=C(N)CC(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217747359 CF In-Stock Unstable FFAR1 41 49 N=C(N)CC(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217747359 CF In-Stock Unstable YOPH 0 43 N=C(N)CC(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217747359 CF In-Stock Unstable PPO2 31 46 N=C(N)CC(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217747359 CF In-Stock Unstable NCE103 29 41 N=C(N)CC(=O)Nc1ccc(OCc2ccccc2)cc1 ZINC000217747359 CF In-Stock Unstable SENP1 0 41 Cc1cc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)c(C)[nH]1 ZINC000217747372 EH On-Demand Unstable HTR2A 15 46 Cc1cc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)c(C)[nH]1 ZINC000217747372 EH On-Demand Unstable SLC18A3 42 47 Cc1cc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)c(C)[nH]1 ZINC000217747372 EH On-Demand Unstable WNT3A 48 34 Cc1cc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)c(C)[nH]1 ZINC000217747372 EH On-Demand Unstable L3MBTL3 84 41 CC1CCN(Cc2ccc(C(=O)NCc3ccc4ccccc4n3)o2)CC1 ZINC000217747373 FH In-Stock Unstable MCHR1 19 45 CC1CCN(Cc2ccc(C(=O)NCc3ccc4ccccc4n3)o2)CC1 ZINC000217747373 FH In-Stock Unstable SMO 42 35 CCCCCCCC(=O)Nc1cccc(/C=C\C(=O)O)n1 ZINC000217747382 CG For-Sale Unstable SOAT1 24 47 CCCCCCCC(=O)Nc1cccc(/C=C\C(=O)O)n1 ZINC000217747382 CG For-Sale Unstable NPR 25 41 CCCCCCCC(=O)Nc1cccc(/C=C\C(=O)O)n1 ZINC000217747382 CG For-Sale Unstable ENPP2 28 40 CCCCCCCC(=O)Nc1cccc(/C=C\C(=O)O)n1 ZINC000217747382 CG For-Sale Unstable PPAF_PHAVU 0 40 CCCCCCCC(=O)Nc1cccc(/C=C\C(=O)O)n1 ZINC000217747382 CG For-Sale Unstable ACAT 0 46 CCCCCCCC(=O)Nc1cccc(/C=C\C(=O)O)n1 ZINC000217747382 CG For-Sale Unstable ACER2 0 40 O=C(C[C@H]1CCCN2CCCC[C@H]12)Nc1ccc(Cl)cc1C(=O)c1ccccc1 ZINC000217747402 HK For-Sale Unstable SLC6A1 64 35 O=C(c1cccc(Oc2ccccn2)c1)N1CC(N2C(=O)CSC2=O)C1 ZINC000217747440 FE In-Stock Unstable RHOA 0 41 CCc1nc2cccc(S(=O)(=O)Cl)c2o1 ZINC000217747464 BE For-Sale Unstable PRSS1 22 40 CCc1nc2cccc(S(=O)(=O)Cl)c2o1 ZINC000217747464 BE For-Sale Unstable MTNR1B 16 44 N=C(N)CC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217747467 CF In-Stock Unstable CA2 20 52 N=C(N)CC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217747467 CF In-Stock Unstable EPHX1 0 51 N=C(N)CC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217747467 CF In-Stock Unstable PRSS1 16 50 N=C(N)CC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217747467 CF In-Stock Unstable SRD5A2 0 41 N=C(N)CC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217747467 CF In-Stock Unstable PDGFRB 19 43 N=C(N)CC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217747467 CF In-Stock Unstable LTA4H 59 60 N=C(N)CC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217747467 CF In-Stock Unstable CA1 53 52 N=C(N)CC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217747467 CF In-Stock Unstable SCN2A 21 62 N=C(N)CC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217747467 CF In-Stock Unstable RAF1 23 41 N=C(N)CC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217747467 CF In-Stock Unstable CA5B 20 41 N=C(N)CC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217747467 CF In-Stock Unstable CA5A 23 41 N=C(N)CC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217747467 CF In-Stock Unstable MTNR1A 15 48 N=C(N)CC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217747467 CF In-Stock Unstable NPY5R 31 45 N=C(N)CC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217747467 CF In-Stock Unstable PLAU 55 40 N=C(N)CC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217747467 CF In-Stock Unstable F7 17 49 N=C(N)CC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217747467 CF In-Stock Unstable ACR 61 50 N=C(N)CC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217747467 CF In-Stock Unstable CA12 26 52 N=C(N)CC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217747467 CF In-Stock Unstable SLC1A2 28 45 N=C(N)CC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217747467 CF In-Stock Unstable SCN4A 23 41 N=C(N)CC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217747467 CF In-Stock Unstable ST14 23 43 N=C(N)CC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217747467 CF In-Stock Unstable CA9 27 52 N=C(N)CC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217747467 CF In-Stock Unstable Q8MMZ8_EIMTE 25 41 N=C(N)CC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217747467 CF In-Stock Unstable F13A1 27 53 N=C(N)CC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217747467 CF In-Stock Unstable YOPH 0 41 N=C(N)CC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217747467 CF In-Stock Unstable NCE103 31 42 N=C(N)CC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217747467 CF In-Stock Unstable P96878_MYCTU 17 52 N=C(N)CC(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000217747467 CF In-Stock Unstable PFKFB3 44 39 O=C(O)/C=C\c1cccc(NC(=O)Cc2cccs2)n1 ZINC000217747476 CE For-Sale Unstable CA5B 34 43 O=C(O)/C=C\c1cccc(NC(=O)Cc2cccs2)n1 ZINC000217747476 CE For-Sale Unstable CA5A 34 43 CCC[C@@H](O)CNCCCc1ccccc1 ZINC000217747515 BE For-Sale Unstable ADRB2 40 45 CCC[C@@H](O)CNCCCc1ccccc1 ZINC000217747515 BE For-Sale Unstable ADRB1 39 45 CCC[C@@H](O)CNCCCc1ccccc1 ZINC000217747515 BE For-Sale Unstable ADRB3 32 45 CCC[C@@H](O)CNCCCc1ccccc1 ZINC000217747515 BE For-Sale Unstable SDH1 0 43 CCC[C@@H](O)CNCCCc1ccccc1 ZINC000217747515 BE For-Sale Unstable SIGMAR1 18 50 CCC[C@@H](O)CNCCCc1ccccc1 ZINC000217747515 BE For-Sale Unstable S1PR3 16 40 CCC[C@@H](O)CNCCCc1ccccc1 ZINC000217747515 BE For-Sale Unstable ABCB1 24 47 CCC[C@@H](O)CNCCCc1ccccc1 ZINC000217747515 BE For-Sale Unstable S1PR2 38 44 CCC[C@@H](O)CNCCCc1ccccc1 ZINC000217747515 BE For-Sale Unstable AMP1_PLAFQ 23 40 CC[C@@H]1CCCC[C@@H]1NC(=O)[C@@H](Cl)c1ccccc1 ZINC000217747540 CI For-Sale Unstable XIAP 41 34 COc1ccc(-n2cnc(C#N)c2)c(OC)c1 ZINC000217747541 BD In-Stock Unstable TPPP 0 40 O=C(N/C=C/c1ccccc1F)Nc1cccc(O)c1 ZINC000217747547 CG For-Sale Anodyne KCNK3 52 37 Cc1cccc(C(=O)Nc2cccc(/C=C\C(=O)O)n2)n1 ZINC000217747561 CE For-Sale Unstable GRM5 23 68 Cc1cccc(C(=O)Nc2cccc(/C=C\C(=O)O)n2)n1 ZINC000217747561 CE For-Sale Unstable SORT1 28 50 COc1ccc(NC(=O)CC(=N)N)c(OC)c1 ZINC000217747582 BC In-Stock Unstable CYP1B1 38 57 COc1ccc(NC(=O)CC(=N)N)c(OC)c1 ZINC000217747582 BC In-Stock Unstable MTNR1A 55 37 COc1ccc(NC(=O)CC(=N)N)c(OC)c1 ZINC000217747582 BC In-Stock Unstable MTNR1B 54 38 COc1ccc(NC(=O)CC(=N)N)c(OC)c1 ZINC000217747582 BC In-Stock Unstable CA9 17 42 COc1ccc(NC(=O)CC(=N)N)c(OC)c1 ZINC000217747582 BC In-Stock Unstable AKR1C2 50 35 COc1ccc(NC(=O)CC(=N)N)c(OC)c1 ZINC000217747582 BC In-Stock Unstable ENPP1 40 31 CCC[C@H](O)CNCCCc1ccccc1 ZINC000217747601 BE For-Sale Unstable ADRB2 40 45 CCC[C@H](O)CNCCCc1ccccc1 ZINC000217747601 BE For-Sale Unstable ADRB1 39 45 CCC[C@H](O)CNCCCc1ccccc1 ZINC000217747601 BE For-Sale Unstable ADRB3 32 45 CCC[C@H](O)CNCCCc1ccccc1 ZINC000217747601 BE For-Sale Unstable SDH1 0 43 CCC[C@H](O)CNCCCc1ccccc1 ZINC000217747601 BE For-Sale Unstable SIGMAR1 18 50 CCC[C@H](O)CNCCCc1ccccc1 ZINC000217747601 BE For-Sale Unstable S1PR3 16 40 CCC[C@H](O)CNCCCc1ccccc1 ZINC000217747601 BE For-Sale Unstable ABCB1 24 47 CCC[C@H](O)CNCCCc1ccccc1 ZINC000217747601 BE For-Sale Unstable S1PR2 38 44 CCC[C@H](O)CNCCCc1ccccc1 ZINC000217747601 BE For-Sale Unstable AMP1_PLAFQ 23 40 CC[C@H]1CCCC[C@@H]1NC(=O)[C@@H](Cl)c1ccccc1 ZINC000217747628 CI For-Sale Unstable XIAP 41 34 COc1ccc(OC)c(-n2cnc(C#N)c2)c1 ZINC000217747644 BD In-Stock Unstable TPPP 0 43 O=C(CCc1ccc(Cl)cc1Cl)NC[C@@H]1CCCN1c1nccs1 ZINC000217747669 GI For-Sale Unstable MC5R 58 38 COc1ccc(OC)c(NC(=O)CC(=N)N)c1 ZINC000217747697 BC In-Stock Unstable CYP1B1 33 43 COc1ccc(OC)c(NC(=O)CC(=N)N)c1 ZINC000217747697 BC In-Stock Unstable MTNR1A 50 37 COc1ccc(OC)c(NC(=O)CC(=N)N)c1 ZINC000217747697 BC In-Stock Unstable MTNR1B 45 38 COc1ccc(OC)c(NC(=O)CC(=N)N)c1 ZINC000217747697 BC In-Stock Unstable AKR1C2 53 38 COc1ccc(OC)c(NC(=O)CC(=N)N)c1 ZINC000217747697 BC In-Stock Unstable ENPP1 55 32 CC[C@@H]1CCCC[C@H]1NC(=O)[C@@H](Cl)c1ccccc1 ZINC000217747720 CI For-Sale Unstable XIAP 41 34 O=C(CCc1ccc(Cl)cc1Cl)NC[C@H]1CCCN1c1nccs1 ZINC000217747746 GI For-Sale Unstable MC5R 58 38 CC[C@H]1CCCC[C@H]1NC(=O)[C@@H](Cl)c1ccccc1 ZINC000217747804 CI For-Sale Unstable XIAP 41 34 COc1ccc(NC(=O)CC(=N)N)cc1OC ZINC000217747812 BC In-Stock Unstable PRSS1 16 43 COc1ccc(NC(=O)CC(=N)N)cc1OC ZINC000217747812 BC In-Stock Unstable MTNR1B 15 43 COc1ccc(NC(=O)CC(=N)N)cc1OC ZINC000217747812 BC In-Stock Unstable ACR 51 43 COc1ccc(NC(=O)CC(=N)N)cc1OC ZINC000217747812 BC In-Stock Unstable QRFPR 41 34 COc1ccc(NC(=O)CC(=N)N)cc1OC ZINC000217747812 BC In-Stock Unstable ENPP1 84 47 COc1ccc(NC(=O)CC(=N)N)cc1OC ZINC000217747812 BC In-Stock Unstable DRTS_TRYCR 48 35 COc1ccc(NC(=O)CC(=N)N)cc1OC ZINC000217747812 BC In-Stock Unstable KCNK3 46 42 COc1ccc(NC(=O)CC(=N)N)cc1OC ZINC000217747812 BC In-Stock Unstable KCNK9 35 42 O=S1(=O)CCCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217747866 CC On-Demand Unstable PKM 25 43 N=C(N)CC(=O)Nc1ccc2c(c1)OCO2 ZINC000217747921 BC In-Stock Unstable PLAU 17 59 N=C(N)CC(=O)Nc1ccc2c(c1)OCO2 ZINC000217747921 BC In-Stock Unstable SLC1A2 44 33 N=C(N)CC(=O)Nc1ccc2c(c1)OCO2 ZINC000217747921 BC In-Stock Unstable DYRK2 44 33 N=C(N)CC(=O)Nc1ccc2c(c1)OCCO2 ZINC000217748031 BC In-Stock Unstable PLAU 15 49 COc1ccc2occ([C@@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(OC)c(O)c6)oc5c43)c(=O)c2c1 ZINC000217748084 KI In-Stock Unstable AKR1B1 0 43 COc1ccc2occ([C@@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(OC)c(O)c6)oc5c43)c(=O)c2c1 ZINC000217748084 KI In-Stock Unstable CYP1B1 47 33 COc1ccc2occ([C@@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(OC)c(O)c6)oc5c43)c(=O)c2c1 ZINC000217748084 KI In-Stock Unstable CYP1A1 37 44 Cc1cccc(C(=O)Nc2ncc(/C=C\C(=O)O)s2)c1 ZINC000217748085 CF For-Sale Unstable LCK 33 43 Cc1cccc(C(=O)Nc2ncc(/C=C\C(=O)O)s2)c1 ZINC000217748085 CF For-Sale Unstable MGEA5 30 40 Cc1cccc(C(=O)Nc2ncc(/C=C\C(=O)O)s2)c1 ZINC000217748085 CF For-Sale Unstable KCNK3 96 47 Cc1cccc(C(=O)Nc2ncc(/C=C\C(=O)O)s2)c1 ZINC000217748085 CF For-Sale Unstable KCNK9 57 47 CC(=O)c1ccc(S(=O)(=O)N2CCCS(=O)(=O)CC2)cc1 ZINC000217748095 EC On-Demand Unstable F13A1 38 40 CCOc1cc(CN2C[C@@H](C)[C@@H](N(C)C)C2)ccc1O ZINC000217748142 CE On-Demand Unstable SSTR5 42 34 COc1ccc(C)cc1NC(=O)CC(=N)N ZINC000217748146 BD In-Stock Unstable KCNMA1 19 47 COc1ccc(C)cc1NC(=O)CC(=N)N ZINC000217748146 BD In-Stock Unstable ENPP1 56 33 COc1ccc2occ([C@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(OC)c(O)c6)oc5c43)c(=O)c2c1 ZINC000217748160 KI In-Stock Unstable AKR1B1 0 43 COc1ccc2occ([C@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(OC)c(O)c6)oc5c43)c(=O)c2c1 ZINC000217748160 KI In-Stock Unstable CYP1B1 47 33 COc1ccc2occ([C@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(OC)c(O)c6)oc5c43)c(=O)c2c1 ZINC000217748160 KI In-Stock Unstable CYP1A1 37 44 O=C(O)/C=C\c1cnc(NC(=O)c2ccc(F)cc2Cl)s1 ZINC000217748168 EG For-Sale Anodyne PYGL 25 42 COc1cccc(NC(=O)N2CC(N3C(=O)CSC3=O)C2)c1 ZINC000217748178 DD In-Stock Unstable CCR3 15 43 COc1cccc(NC(=O)N2CC(N3C(=O)CSC3=O)C2)c1 ZINC000217748178 DD In-Stock Unstable MTNR1A 23 42 Cc1[nH]c2ccccc2c1CC(=O)NC1CCN(C(=O)N2CCOCC2)CC1 ZINC000217748180 GE In-Stock Unstable CCR8 75 44 O=C(N/C=C/c1ccccc1F)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217748213 EF For-Sale Anodyne P96878_MYCTU 46 40 CCOc1cc(CN2C[C@H](C)[C@@H](N(C)C)C2)ccc1O ZINC000217748218 CE On-Demand Unstable SSTR5 42 34 COc1ccc([C@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2oc(C)cc(=O)c2O)cc1O ZINC000217748262 JH In-Stock Unstable RORC 45 34 COc1ccc(Cl)cc1NC(=O)CC(=N)N ZINC000217748271 BD In-Stock Unstable CYSP_TRYCR 0 47 COc1ccc(Cl)cc1NC(=O)CC(=N)N ZINC000217748271 BD In-Stock Unstable COLA 51 35 COc1ccc(Cl)cc1NC(=O)CC(=N)N ZINC000217748271 BD In-Stock Unstable CPT1A 47 35 COc1ccc(Cl)cc1NC(=O)CC(=N)N ZINC000217748271 BD In-Stock Unstable KCNMA1 37 46 COc1ccc(Cl)cc1NC(=O)CC(=N)N ZINC000217748271 BD In-Stock Unstable RBP4 28 49 COc1ccc(Cl)cc1NC(=O)CC(=N)N ZINC000217748271 BD In-Stock Unstable ENPP1 56 35 N#Cc1cn(-c2cccnc2)cn1 ZINC000217748292 AD In-Stock Mild CYP2A6 18 59 O=C(NC(c1ccccc1)c1ccccc1)N1CC(N2C(=O)CSC2=O)C1 ZINC000217748295 GF In-Stock Unstable BIRC8 56 33 CN1C[C@@H]2CC[C@H](C1)N(C(=O)c1ccc3c(=O)n(C)cnc3c1)C2 ZINC000217748325 ED In-Stock Unstable HPGD 40 32 COc1ccc([C@@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2oc(C)cc(=O)c2O)cc1O ZINC000217748352 JH In-Stock Unstable RORC 45 34 CN(Cc1cccc(/C=C\C(=O)O)c1)C(=O)c1ccc[nH]1 ZINC000217748362 CE For-Sale Unstable HSD17B2 26 41 COc1ccc(NC(=O)CC(=N)N)cc1Cl ZINC000217748370 BD In-Stock Unstable CYSP_TRYCR 0 47 COc1ccc(NC(=O)CC(=N)N)cc1Cl ZINC000217748370 BD In-Stock Unstable GRM4 21 53 COc1ccc(NC(=O)CC(=N)N)cc1Cl ZINC000217748370 BD In-Stock Unstable PDE6A 43 34 COc1ccc(NC(=O)CC(=N)N)cc1Cl ZINC000217748370 BD In-Stock Unstable ACR 37 40 COc1ccc(NC(=O)CC(=N)N)cc1Cl ZINC000217748370 BD In-Stock Unstable AGPAT2 43 33 COc1ccc(NC(=O)CC(=N)N)cc1Cl ZINC000217748370 BD In-Stock Unstable CSF1R 25 41 COc1ccc(NC(=O)CC(=N)N)cc1Cl ZINC000217748370 BD In-Stock Unstable QRFPR 40 35 COc1ccc(NC(=O)CC(=N)N)cc1Cl ZINC000217748370 BD In-Stock Unstable ENPP1 71 42 COc1ccc(NC(=O)CC(=N)N)cc1Cl ZINC000217748370 BD In-Stock Unstable IMDH_CRYPV 28 40 O=C(NC12CC3CC(CC(C3)C1)C2)N1CC(N2C(=O)CSC2=O)C1 ZINC000217748381 EE In-Stock Unstable EPHX2 23 46 COCCCCNC(=O)/C=C\C(=O)O ZINC000217748383 BC For-Sale Unstable HCAR2 29 41 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1ccc(CCl)cc1 ZINC000217748390 DJ For-Sale Unstable TRPM8 23 75 Cn1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)n1 ZINC000217748407 DE On-Demand Unstable HTR2A 21 49 Cn1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)n1 ZINC000217748407 DE On-Demand Unstable SLC18A3 51 49 Cn1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)n1 ZINC000217748407 DE On-Demand Unstable WNT3A 48 36 Cn1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)n1 ZINC000217748407 DE On-Demand Unstable L3MBTL3 72 40 N#Cc1ccc(S(=O)(=O)N2CCCS(=O)(=O)CC2)cc1Cl ZINC000217748422 ED On-Demand Unstable TRPV4 42 34 CCOc1ccccc1CCC(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217748431 FG For-Sale Unstable MBTPS1 48 33 CCOc1ccccc1CCC(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217748431 FG For-Sale Unstable HCN1 44 32 CCOc1ccccc1CCC(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217748431 FG For-Sale Unstable HCN4 41 32 CSc1cccc(NC(=O)CC(=N)N)c1 ZINC000217748466 BD In-Stock Unstable F2R 0 40 CSc1cccc(NC(=O)CC(=N)N)c1 ZINC000217748466 BD In-Stock Unstable ENPP1 52 34 CSc1cccc(NC(=O)CC(=N)N)c1 ZINC000217748466 BD In-Stock Unstable KCNK3 57 33 CSc1cccc(NC(=O)CC(=N)N)c1 ZINC000217748466 BD In-Stock Unstable KCNK9 61 34 CC(=O)c1ccc(NC(=O)[C@@H](C)Sc2nnc(N3C[C@@H](C)C[C@@H](C)C3)n2Cc2ccco2)cc1 ZINC000217748469 JJ On-Demand Unstable HCRTR2 19 41 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1ccc(CCl)cc1 ZINC000217748481 DJ For-Sale Unstable TRPM8 23 75 CN(CCO)C(=O)CCc1nc2ccccc2c(=O)[nH]1 ZINC000217748483 CC In-Stock Unstable PARP1 21 55 CN(CCO)C(=O)CCc1nc2ccccc2c(=O)[nH]1 ZINC000217748483 CC In-Stock Unstable PARP3 40 55 CN(CCO)C(=O)CCc1nc2ccccc2c(=O)[nH]1 ZINC000217748483 CC In-Stock Unstable QTRT1 0 43 CN(CCO)C(=O)CCc1nc2ccccc2c(=O)[nH]1 ZINC000217748483 CC In-Stock Unstable TNKS 19 48 CCC[C@@H](O)CN[C@@H](C)c1ccc(O)cc1 ZINC000217748493 BE For-Sale Unstable NMUR2 0 43 CCOc1ccccc1CCC(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217748538 FG For-Sale Unstable MBTPS1 48 33 CCOc1ccccc1CCC(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217748538 FG For-Sale Unstable HCN1 44 32 CCOc1ccccc1CCC(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217748538 FG For-Sale Unstable HCN4 41 32 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)c1ccc(CCl)cc1 ZINC000217748558 DJ For-Sale Unstable TRPM8 23 75 O=C1CN(C(=O)/C=C\c2ccccc2)CC(=O)N1 ZINC000217748572 BC For-Sale Unstable F3 24 47 O=C1CN(C(=O)/C=C\c2ccccc2)CC(=O)N1 ZINC000217748572 BC For-Sale Unstable GPR183 0 45 COC(=O)c1ccccc1NC(=O)CC(=N)N ZINC000217748578 BC In-Stock Unstable FAS 74 60 CCC[C@H](O)CN[C@@H](C)c1ccc(O)cc1 ZINC000217748580 BE For-Sale Unstable NMUR2 0 43 Cc1oncc1C(=O)Nc1cccc(/C=C\C(=O)O)c1 ZINC000217748623 CE For-Sale Unstable BTK 20 43 Cc1oncc1C(=O)Nc1cccc(/C=C\C(=O)O)c1 ZINC000217748623 CE For-Sale Unstable KCNK3 115 40 Cc1oncc1C(=O)Nc1cccc(/C=C\C(=O)O)c1 ZINC000217748623 CE For-Sale Unstable KCNK9 81 38 CC(C)c1ccc(NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217748631 CJ For-Sale Unstable KCNQ2 40 35 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)c1ccc(CCl)cc1 ZINC000217748645 DJ For-Sale Unstable TRPM8 23 75 CCC[C@@H](O)CN[C@H](C)c1ccc(O)cc1 ZINC000217748661 BE For-Sale Unstable NMUR2 0 43 CN(C)c1ccc(/C=C\C(=O)N2CC(=O)NC(=O)C2)cc1 ZINC000217748665 CC For-Sale Unstable GPR183 0 51 COC(=O)c1ccc(NC(=O)CC(=N)N)cc1 ZINC000217748691 BC In-Stock Unstable PRSS1 26 53 COC(=O)c1ccc(NC(=O)CC(=N)N)cc1 ZINC000217748691 BC In-Stock Unstable F3 71 36 COC(=O)c1ccc(NC(=O)CC(=N)N)cc1 ZINC000217748691 BC In-Stock Unstable PLAU 19 40 COC(=O)c1ccc(NC(=O)CC(=N)N)cc1 ZINC000217748691 BC In-Stock Unstable ACR 87 53 COC(=O)c1ccc(NC(=O)CC(=N)N)cc1 ZINC000217748691 BC In-Stock Unstable PPO2 26 43 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1cccc(CCl)c1 ZINC000217748730 DJ For-Sale Unstable TRPM8 22 64 CCC[C@H](O)CN[C@H](C)c1ccc(O)cc1 ZINC000217748742 BE For-Sale Unstable NMUR2 0 43 COc1ccccc1NC(=O)N/C=C/c1ccccc1F ZINC000217748747 CH For-Sale Unstable TLR4 17 43 CCOc1ccc(-n2cnc(CO)c2)cc1 ZINC000217748773 BD In-Stock Unstable CACNA2D1 59 41 CCOc1ccc(-n2cnc(CO)c2)cc1 ZINC000217748773 BD In-Stock Unstable CACNA2D2 52 33 CCOc1ccc(-n2cnc(CO)c2)cc1 ZINC000217748773 BD In-Stock Unstable CYP2C19 18 40 CC(C)C[C@@H](CO)NC(=O)CC[C@@H]1NC(=O)N(Cc2ccc3c(c2)OCO3)C1=O ZINC000217748801 HD In-Stock Unstable NPY1R 20 40 CC(C)C[C@@H](CO)NC(=O)CC[C@@H]1NC(=O)N(Cc2ccc3c(c2)OCO3)C1=O ZINC000217748801 HD In-Stock Unstable MCHR1 22 42 CCOC(=O)c1ccc(NC(=O)CC(=N)N)cc1 ZINC000217748809 BD In-Stock Unstable PRSS1 22 50 CCOC(=O)c1ccc(NC(=O)CC(=N)N)cc1 ZINC000217748809 BD In-Stock Unstable F3 61 35 CCOC(=O)c1ccc(NC(=O)CC(=N)N)cc1 ZINC000217748809 BD In-Stock Unstable PLAU 17 43 CCOC(=O)c1ccc(NC(=O)CC(=N)N)cc1 ZINC000217748809 BD In-Stock Unstable ACR 83 50 CCOC(=O)c1ccc(NC(=O)CC(=N)N)cc1 ZINC000217748809 BD In-Stock Unstable PPO2 27 45 CCOC(=O)c1ccc(NC(=O)CC(=N)N)cc1 ZINC000217748809 BD In-Stock Unstable NOD2 17 43 CCOC(=O)c1ccc(NC(=O)CC(=N)N)cc1 ZINC000217748809 BD In-Stock Unstable SLC27A1 18 47 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1cccc(CCl)c1 ZINC000217748821 DJ For-Sale Unstable TRPM8 22 64 COc1ccc([C@@H](C)N[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217748869 CF For-Sale Unstable CHRM2 17 43 COc1ccc([C@@H](C)N[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217748869 CF For-Sale Unstable CHRM4 15 43 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)c1cccc(CCl)c1 ZINC000217748883 DJ For-Sale Unstable TRPM8 22 64 O=[N+]([O-])c1ccccc1-n1cnc(CO)c1 ZINC000217748889 BD In-Stock Unstable PQSD 0 45 Cc1cc(NC(=O)c2ccccc2)ccc1/C=C\C(=O)O ZINC000217748918 CG For-Sale Unstable PTGER2 40 38 Cc1cc(NC(=O)c2ccccc2)ccc1/C=C\C(=O)O ZINC000217748918 CG For-Sale Unstable MAPK14 20 43 Cc1cc(NC(=O)c2ccccc2)ccc1/C=C\C(=O)O ZINC000217748918 CG For-Sale Unstable TRPV1 17 40 Cc1cc(NC(=O)c2ccccc2)ccc1/C=C\C(=O)O ZINC000217748918 CG For-Sale Unstable PRNP 55 47 Cc1cc(NC(=O)c2ccccc2)ccc1/C=C\C(=O)O ZINC000217748918 CG For-Sale Unstable LDLR 0 40 Cc1cc(NC(=O)c2ccccc2)ccc1/C=C\C(=O)O ZINC000217748918 CG For-Sale Unstable GRM4 19 40 Cc1cc(NC(=O)c2ccccc2)ccc1/C=C\C(=O)O ZINC000217748918 CG For-Sale Unstable NR1H4 16 42 Cc1cc(NC(=O)c2ccccc2)ccc1/C=C\C(=O)O ZINC000217748918 CG For-Sale Unstable MCHR1 17 42 Cc1cc(NC(=O)c2ccccc2)ccc1/C=C\C(=O)O ZINC000217748918 CG For-Sale Unstable SHH 38 41 Cc1cc(NC(=O)c2ccccc2)ccc1/C=C\C(=O)O ZINC000217748918 CG For-Sale Unstable SMO 23 43 Cc1cc(NC(=O)c2ccccc2)ccc1/C=C\C(=O)O ZINC000217748918 CG For-Sale Unstable GLMU 0 40 Cc1cc(NC(=O)c2ccccc2)ccc1/C=C\C(=O)O ZINC000217748918 CG For-Sale Unstable PARP14 0 40 Cc1cc(NC(=O)c2ccccc2)ccc1/C=C\C(=O)O ZINC000217748918 CG For-Sale Unstable KCNK3 134 55 Cc1cc(NC(=O)c2ccccc2)ccc1/C=C\C(=O)O ZINC000217748918 CG For-Sale Unstable KCNK9 78 55 Cc1cc(NC(=O)c2ccccc2)ccc1/C=C\C(=O)O ZINC000217748918 CG For-Sale Unstable PARP10 0 40 CC(=O)c1cccc(NC(=O)CC(=N)N)c1 ZINC000217748928 BD In-Stock Unstable PRSS1 20 41 CC(=O)c1cccc(NC(=O)CC(=N)N)c1 ZINC000217748928 BD In-Stock Unstable CCR3 19 40 CC(=O)c1cccc(NC(=O)CC(=N)N)c1 ZINC000217748928 BD In-Stock Unstable F2R 0 41 CC(=O)c1cccc(NC(=O)CC(=N)N)c1 ZINC000217748928 BD In-Stock Unstable AMD1 18 42 CC(=O)c1cccc(NC(=O)CC(=N)N)c1 ZINC000217748928 BD In-Stock Unstable PLAU 19 40 CC(=O)c1cccc(NC(=O)CC(=N)N)c1 ZINC000217748928 BD In-Stock Unstable AKR1C3 36 53 CC(=O)c1cccc(NC(=O)CC(=N)N)c1 ZINC000217748928 BD In-Stock Unstable NAMPT 0 57 CC(=O)c1cccc(NC(=O)CC(=N)N)c1 ZINC000217748928 BD In-Stock Unstable KCNK3 91 41 CC(=O)c1cccc(NC(=O)CC(=N)N)c1 ZINC000217748928 BD In-Stock Unstable KCNK9 83 41 COc1ccc([C@H](C)N[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217748951 CF For-Sale Unstable CHRM2 17 43 COc1ccc([C@H](C)N[C@@H]2CCN3CCC[C@@H]23)cc1 ZINC000217748951 CF For-Sale Unstable CHRM4 15 43 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)c1cccc(CCl)c1 ZINC000217748958 DJ For-Sale Unstable TRPM8 22 64 C[C@H]1C[C@@H](C)CN(c2nnc(S[C@H](C)C(=O)N3CCc4ccccc43)n2Cc2ccco2)C1 ZINC000217748973 JI On-Demand Unstable HCRTR2 17 44 O=C(N/C=C/c1ccccc1F)Nc1ccc(Cl)c(Cl)c1 ZINC000217748976 EJ For-Sale Anodyne ENV 40 31 O=C(N/C=C/c1ccccc1F)Nc1ccc(Cl)c(Cl)c1 ZINC000217748976 EJ For-Sale Anodyne BLM 0 40 O=C(N/C=C/c1ccccc1F)Nc1ccc(Cl)c(Cl)c1 ZINC000217748976 EJ For-Sale Anodyne P95276_MYCTO 0 51 O=C(N/C=C/c1ccccc1F)Nc1ccc(Cl)c(Cl)c1 ZINC000217748976 EJ For-Sale Anodyne WRN 0 40 O=C(N/C=C/c1ccccc1F)Nc1ccc(Cl)c(Cl)c1 ZINC000217748976 EJ For-Sale Anodyne PPX1 0 40 Cc1ccc(C(=O)Nc2ccc(/C=C\C(=O)O)cc2C)o1 ZINC000217749010 CG For-Sale Unstable S1PR4 24 41 Cc1ccc(C(=O)Nc2ccc(/C=C\C(=O)O)cc2C)o1 ZINC000217749010 CG For-Sale Unstable CSF1R 0 51 O=C(c1ccc(Cl)cc1)C1CCN(C(=O)c2ccccc2OC(F)(F)F)CC1 ZINC000217749016 HJ On-Demand Unstable SLC6A1 17 41 O=C(c1ccc(Cl)cc1)C1CCN(C(=O)c2ccccc2OC(F)(F)F)CC1 ZINC000217749016 HJ On-Demand Unstable SLC18A3 45 44 O=C(c1ccc(Cl)cc1)C1CCN(C(=O)c2ccccc2OC(F)(F)F)CC1 ZINC000217749016 HJ On-Demand Unstable EPHX2 15 41 O=C(c1ccc(Cl)cc1)C1CCN(C(=O)c2ccccc2OC(F)(F)F)CC1 ZINC000217749016 HJ On-Demand Unstable L3MBTL3 66 40 COc1ccc([C@@H](C)N[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217749036 CF For-Sale Unstable CHRM2 17 43 COc1ccc([C@@H](C)N[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217749036 CF For-Sale Unstable CHRM4 15 43 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)[C@@H](Cl)c1ccccc1 ZINC000217749045 DJ For-Sale Unstable TRPM8 22 57 CC(=O)Nc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217749046 BC In-Stock Unstable CA2 17 48 CC(=O)Nc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217749046 BC In-Stock Unstable CA4 17 43 CC(=O)Nc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217749046 BC In-Stock Unstable ACR 55 39 CC(=O)Nc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217749046 BC In-Stock Unstable PPO2 27 47 CC(=O)Nc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217749046 BC In-Stock Unstable NAMPT 0 46 C[C@@H]1C[C@@H](C)CN(c2nnc(S[C@H](C)C(=O)N3CCc4ccccc43)n2Cc2ccco2)C1 ZINC000217749061 JI On-Demand Unstable HCRTR2 17 44 COc1ccc([C@H](C)N[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217749108 CF For-Sale Unstable CHRM2 17 43 COc1ccc([C@H](C)N[C@H]2CCN3CCC[C@@H]23)cc1 ZINC000217749108 CF For-Sale Unstable CHRM4 15 43 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)[C@@H](Cl)c1ccccc1 ZINC000217749129 DJ For-Sale Unstable TRPM8 22 57 O=C1CSC(=O)N1C1CN(S(=O)(=O)c2c(F)cccc2F)C1 ZINC000217749174 ED In-Stock Unstable PKM 21 49 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)[C@@H](Cl)c1ccccc1 ZINC000217749194 DJ For-Sale Unstable TRPM8 22 57 c1ccc2c(c1)CC[C@H]2N[C@@H]1CCN2CCC[C@@H]12 ZINC000217749222 BF For-Sale Unstable SLC18A3 50 35 Cc1cccc(C(C)C)c1NC(=O)N/C=C/c1ccccc1F ZINC000217749229 DK For-Sale Unstable SOAT1 49 39 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)[C@@H](Cl)c1ccccc1 ZINC000217749265 DJ For-Sale Unstable TRPM8 22 57 O=C1CSC(=O)N1C1CN(S(=O)(=O)c2cccc3ccccc23)C1 ZINC000217749278 FD In-Stock Unstable HTR6 17 40 c1ccc2c(c1)CC[C@H]2N[C@H]1CCN2CCC[C@@H]12 ZINC000217749303 BF For-Sale Unstable SLC18A3 50 35 CN(Cc1ccccc1)C(=O)CC(=N)N ZINC000217749311 BC In-Stock Unstable TACR1 17 43 CN(Cc1ccccc1)C(=O)CC(=N)N ZINC000217749311 BC In-Stock Unstable TSPO 20 42 CN(Cc1ccccc1)C(=O)CC(=N)N ZINC000217749311 BC In-Stock Unstable CTSB 40 45 CN(Cc1ccccc1)C(=O)CC(=N)N ZINC000217749311 BC In-Stock Unstable HSD17B2 23 43 CN(Cc1ccccc1)C(=O)CC(=N)N ZINC000217749311 BC In-Stock Unstable AOC3 16 45 CN(Cc1ccccc1)C(=O)CC(=N)N ZINC000217749311 BC In-Stock Unstable LIMK2 43 43 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)CCCl ZINC000217749393 BG For-Sale Unstable TRPM8 21 58 CC(C)(C)C(=O)NCc1cc(/C=C\C(=O)O)ccc1F ZINC000217749407 CF For-Sale Unstable AKR1C3 26 40 N=C(N)CC(=O)N(Cc1ccccc1)Cc1ccccc1 ZINC000217749411 CF In-Stock Unstable LIMK2 34 40 O=C(N/C=C/c1ccccc1F)Nc1ccc(C(=O)O)cc1 ZINC000217749423 DG For-Sale Anodyne EPHX2 15 43 COC(=O)C[C@@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(O)cc1 ZINC000217749443 FF In-Stock Unstable KCNA5 28 40 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)CCCl ZINC000217749459 BG For-Sale Unstable TRPM8 21 58 CC(=O)NCC(=O)N[C@@H](C)c1cccc(/C=C\C(=O)O)c1 ZINC000217749482 CD For-Sale Unstable F7 27 40 FC(F)c1ccc(Cl)c([C@@H]2CCCCN2)c1 ZINC000217749485 BI For-Sale Unstable SLC6A1 18 45 O=C1CSC(=O)N1C1CN(S(=O)(=O)c2ccc3c(c2)OCCO3)C1 ZINC000217749499 FC In-Stock Unstable PKM 40 54 COC(=O)C[C@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(O)cc1 ZINC000217749513 FF In-Stock Unstable KCNA5 28 40 Cc1c(Cl)cccc1NC(=O)N/C=C/c1ccccc1F ZINC000217749537 DJ For-Sale Unstable CXCL8 42 33 CC(=O)NCC(=O)N[C@H](C)c1cccc(/C=C\C(=O)O)c1 ZINC000217749559 CD For-Sale Unstable F7 27 40 FC(F)c1ccc(Cl)c([C@H]2CCCCN2)c1 ZINC000217749571 BI For-Sale Unstable SLC6A1 18 45 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)CCCl ZINC000217749574 BG For-Sale Unstable TRPM8 21 58 N=C(N)CC(=O)N1CCC(Cc2ccccc2)CC1 ZINC000217749588 CD In-Stock Unstable F2 27 56 N=C(N)CC(=O)N1CCC(Cc2ccccc2)CC1 ZINC000217749588 CD In-Stock Unstable PRSS1 28 52 N=C(N)CC(=O)N1CCC(Cc2ccccc2)CC1 ZINC000217749588 CD In-Stock Unstable CHRM2 20 42 N=C(N)CC(=O)N1CCC(Cc2ccccc2)CC1 ZINC000217749588 CD In-Stock Unstable GRIN1 0 42 N=C(N)CC(=O)N1CCC(Cc2ccccc2)CC1 ZINC000217749588 CD In-Stock Unstable GRIN2B 87 53 N=C(N)CC(=O)N1CCC(Cc2ccccc2)CC1 ZINC000217749588 CD In-Stock Unstable SIGMAR1 35 47 N=C(N)CC(=O)N1CCC(Cc2ccccc2)CC1 ZINC000217749588 CD In-Stock Unstable CCR3 63 48 N=C(N)CC(=O)N1CCC(Cc2ccccc2)CC1 ZINC000217749588 CD In-Stock Unstable C3AR1 41 37 N=C(N)CC(=O)N1CCC(Cc2ccccc2)CC1 ZINC000217749588 CD In-Stock Unstable EPHX2 19 40 N=C(N)CC(=O)N1CCC(Cc2ccccc2)CC1 ZINC000217749588 CD In-Stock Unstable ST14 63 40 N=C(N)CC(=O)N1CCC(Cc2ccccc2)CC1 ZINC000217749588 CD In-Stock Unstable GRIN2C 18 42 N=C(N)CC(=O)N1CCC(Cc2ccccc2)CC1 ZINC000217749588 CD In-Stock Unstable GRIN3A 0 42 N=C(N)CC(=O)N1CCC(Cc2ccccc2)CC1 ZINC000217749588 CD In-Stock Unstable AMP1_PLAFQ 34 57 N=C(N)CC(=O)N1CCC(Cc2ccccc2)CC1 ZINC000217749588 CD In-Stock Unstable TMPRSS11D 46 31 N=C(N)CC(=O)N1CCC(Cc2ccccc2)CC1 ZINC000217749588 CD In-Stock Unstable TMPRSS6 40 32 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)CCCl ZINC000217749624 BG For-Sale Unstable TRPM8 21 58 OCc1cn(-c2cccnc2)cn1 ZINC000217749628 AC In-Stock Unstable CYP2A6 26 59 CCOC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217749638 EH For-Sale Unstable CA1 15 43 CCOC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217749638 EH For-Sale Unstable ACR 63 36 COCC(=O)N[C@@H](C)c1cccc(/C=C\C(=O)O)c1 ZINC000217749650 CD For-Sale Unstable ACACA 22 41 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)[C@@H](C)Cl ZINC000217749693 BG For-Sale Unstable TRPM8 22 58 COc1ccc(-c2coc3ccc(OCC(N)=O)cc23)cc1 ZINC000217749734 CF In-Stock Unstable GSK3B 0 53 COCC(=O)N[C@H](C)c1cccc(/C=C\C(=O)O)c1 ZINC000217749759 CD For-Sale Unstable ACACA 22 41 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)[C@@H](C)Cl ZINC000217749781 BG For-Sale Unstable TRPM8 22 58 CC(C)c1ccccc1NC(=O)N/C=C/c1ccccc1F ZINC000217749809 CJ For-Sale Unstable ACAT 0 40 C[C@@H](N[C@@H]1CCN2CCC[C@@H]12)c1ccccc1 ZINC000217749829 BF For-Sale Unstable SLC18A3 40 36 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCCC(=O)Nc3nccs3)[C@H]21 ZINC000217749836 JH In-Stock Unstable MAP1 57 37 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)[C@@H](C)Cl ZINC000217749866 BG For-Sale Unstable TRPM8 22 58 FC(F)c1ccc(Cl)c(C2CCNCC2)c1 ZINC000217749868 BH For-Sale Unstable SLC6A2 16 53 C[C@H](NC(=O)[C@@H]1CCOC1)c1cccc(/C=C\C(=O)O)c1 ZINC000217749884 CD For-Sale Unstable KCNQ2 46 34 C[C@H](N[C@@H]1CCN2CCC[C@@H]12)c1ccccc1 ZINC000217749920 BF For-Sale Unstable SLC18A3 40 36 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCCC(=O)Nc3nccs3)[C@@H]21 ZINC000217749931 JH In-Stock Unstable MAP1 57 37 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)[C@@H](C)Cl ZINC000217749953 BG For-Sale Unstable TRPM8 22 58 C[C@@H](NC(=O)[C@@H]1CCOC1)c1cccc(/C=C\C(=O)O)c1 ZINC000217749971 CD For-Sale Unstable KCNQ2 46 34 C[C@@H](N[C@H]1CCN2CCC[C@@H]12)c1ccccc1 ZINC000217749985 BF For-Sale Unstable SLC18A3 40 36 COc1ccc(-c2n[nH]cc2C(=O)N[C@@H]2CCCc3c2[nH]c2ccc(OC)cc32)cc1 ZINC000217750004 HI In-Stock Unstable MAPKAPK2 22 44 N=C(N)CC(=O)N1CCN(Cc2ccccc2)CC1 ZINC000217750031 CC In-Stock Unstable CHRM2 18 42 N=C(N)CC(=O)N1CCN(Cc2ccccc2)CC1 ZINC000217750031 CC In-Stock Unstable DRD2 27 44 N=C(N)CC(=O)N1CCN(Cc2ccccc2)CC1 ZINC000217750031 CC In-Stock Unstable DRD4 64 43 N=C(N)CC(=O)N1CCN(Cc2ccccc2)CC1 ZINC000217750031 CC In-Stock Unstable DRD3 25 44 N=C(N)CC(=O)N1CCN(Cc2ccccc2)CC1 ZINC000217750031 CC In-Stock Unstable LTA4H 16 41 N=C(N)CC(=O)N1CCN(Cc2ccccc2)CC1 ZINC000217750031 CC In-Stock Unstable SIGMAR1 68 55 N=C(N)CC(=O)N1CCN(Cc2ccccc2)CC1 ZINC000217750031 CC In-Stock Unstable CCR3 20 40 N=C(N)CC(=O)N1CCN(Cc2ccccc2)CC1 ZINC000217750031 CC In-Stock Unstable NPFFR2 45 45 N=C(N)CC(=O)N1CCN(Cc2ccccc2)CC1 ZINC000217750031 CC In-Stock Unstable FAAH 26 50 N=C(N)CC(=O)N1CCN(Cc2ccccc2)CC1 ZINC000217750031 CC In-Stock Unstable DPP8 18 44 N=C(N)CC(=O)N1CCN(Cc2ccccc2)CC1 ZINC000217750031 CC In-Stock Unstable MGLL 0 53 N=C(N)CC(=O)N1CCN(Cc2ccccc2)CC1 ZINC000217750031 CC In-Stock Unstable ABHD6 0 45 N=C(N)CC(=O)N1CCN(Cc2ccccc2)CC1 ZINC000217750031 CC In-Stock Unstable NPFFR1 71 45 N=C(N)CC(=O)N1CCN(Cc2ccccc2)CC1 ZINC000217750031 CC In-Stock Unstable TMPRSS11D 24 40 N=C(N)CC(=O)N1CCN(Cc2ccccc2)CC1 ZINC000217750031 CC In-Stock Unstable GPR183 0 40 C=CC(=O)N[C@H]1C[C@H](C)CC[C@H]1C(C)C ZINC000217750037 BF For-Sale Unstable TRPM8 20 53 C[C@H](N[C@H]1CCN2CCC[C@@H]12)c1ccccc1 ZINC000217750083 BF For-Sale Unstable SLC18A3 40 36 COc1ccc(-c2n[nH]cc2C(=O)N[C@H]2CCCc3c2[nH]c2ccc(OC)cc32)cc1 ZINC000217750085 HI In-Stock Unstable MAPKAPK2 22 44 C=CC(=O)N[C@H]1C[C@H](C)CC[C@@H]1C(C)C ZINC000217750105 BF For-Sale Unstable TRPM8 20 53 N=C(N)CC(=O)N1CCN(c2ccccc2)CC1 ZINC000217750106 BC In-Stock Unstable HTR1A 27 44 N=C(N)CC(=O)N1CCN(c2ccccc2)CC1 ZINC000217750106 BC In-Stock Unstable HTR2A 15 44 N=C(N)CC(=O)N1CCN(c2ccccc2)CC1 ZINC000217750106 BC In-Stock Unstable ERBB2 0 45 N=C(N)CC(=O)N1CCN(c2ccccc2)CC1 ZINC000217750106 BC In-Stock Unstable MAPK1 32 49 N=C(N)CC(=O)N1CCN(c2ccccc2)CC1 ZINC000217750106 BC In-Stock Unstable ADAM10 39 44 N=C(N)CC(=O)N1CCN(c2ccccc2)CC1 ZINC000217750106 BC In-Stock Unstable AKR1C3 23 51 COc1ccc(NC(=O)N/C=C/c2ccccc2F)cc1Cl ZINC000217750126 DI For-Sale Unstable HTR2A 22 41 COc1ccc(NC(=O)N/C=C/c2ccccc2F)cc1Cl ZINC000217750126 DI For-Sale Unstable PYGL 0 42 COc1ccc(NC(=O)N/C=C/c2ccccc2F)cc1Cl ZINC000217750126 DI For-Sale Unstable GRM4 23 49 COc1ccc(NC(=O)N/C=C/c2ccccc2F)cc1Cl ZINC000217750126 DI For-Sale Unstable IMPDH2 0 46 COc1ccc(NC(=O)N/C=C/c2ccccc2F)cc1Cl ZINC000217750126 DI For-Sale Unstable CYSP_PLAFA 40 33 CCOc1ccc(/C=C\C(=O)N2CC(=O)NC(=O)C2)cc1 ZINC000217750133 CC For-Sale Unstable GPR183 0 44 C=CC(=O)N[C@H]1C[C@@H](C)CC[C@H]1C(C)C ZINC000217750187 BF For-Sale Unstable TRPM8 20 53 C[C@@H](N[C@@H]1CCN2CCC[C@@H]12)c1cccc(Br)c1 ZINC000217750188 DG For-Sale Unstable MBTD1 0 50 N=C(N)CC(=O)N1CCN(c2ccc(F)cc2)CC1 ZINC000217750222 CC In-Stock Unstable CCR1 27 45 N=C(N)CC(=O)N1CCN(c2ccc(F)cc2)CC1 ZINC000217750222 CC In-Stock Unstable AKR1C3 23 54 O=C(N/C=C/c1ccccc1F)Nc1cccc(C(F)(F)F)c1 ZINC000217750234 DJ For-Sale Anodyne KIT 16 41 O=C(N/C=C/c1ccccc1F)Nc1cccc(C(F)(F)F)c1 ZINC000217750234 DJ For-Sale Anodyne KDR 17 41 O=C(N/C=C/c1ccccc1F)Nc1cccc(C(F)(F)F)c1 ZINC000217750234 DJ For-Sale Anodyne EPHX2 15 47 O=C(N/C=C/c1ccccc1F)Nc1cccc(C(F)(F)F)c1 ZINC000217750234 DJ For-Sale Anodyne RIPK1 57 40 O=C(N/C=C/c1ccccc1F)Nc1cccc(C(F)(F)F)c1 ZINC000217750234 DJ For-Sale Anodyne TRPM4 0 42 O=C(N/C=C/c1ccccc1F)Nc1cccc(C(F)(F)F)c1 ZINC000217750234 DJ For-Sale Anodyne KCNK3 55 48 C=CC(=O)N[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217750267 BF For-Sale Unstable TRPM8 20 53 C[C@H](N[C@@H]1CCN2CCC[C@@H]12)c1cccc(Br)c1 ZINC000217750270 DG For-Sale Unstable MBTD1 0 50 COc1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1Cl ZINC000217750276 GI On-Demand Unstable HTR2A 15 44 COc1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1Cl ZINC000217750276 GI On-Demand Unstable HTR4 19 41 COc1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1Cl ZINC000217750276 GI On-Demand Unstable SLC18A3 45 53 COc1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1Cl ZINC000217750276 GI On-Demand Unstable SCN5A 20 44 COc1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1Cl ZINC000217750276 GI On-Demand Unstable L3MBTL3 78 39 Cc1cc(=O)c(O)c([C@@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccc(O)cc2)o1 ZINC000217750288 IH In-Stock Unstable FABI 51 31 Cc1cc(=O)c(O)c([C@@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccc(O)cc2)o1 ZINC000217750288 IH In-Stock Unstable DRD5 19 40 Cc1cc(=O)c(O)c([C@@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccc(O)cc2)o1 ZINC000217750288 IH In-Stock Unstable SSTR4 40 32 N=C(N)CC(=O)N1CCN(c2cccc(Cl)c2)CC1 ZINC000217750337 CD In-Stock Unstable HTR1A 30 53 N=C(N)CC(=O)N1CCN(c2cccc(Cl)c2)CC1 ZINC000217750337 CD In-Stock Unstable HTR2A 24 53 N=C(N)CC(=O)N1CCN(c2cccc(Cl)c2)CC1 ZINC000217750337 CD In-Stock Unstable DRD3 20 42 N=C(N)CC(=O)N1CCN(c2cccc(Cl)c2)CC1 ZINC000217750337 CD In-Stock Unstable HTR7 23 48 N=C(N)CC(=O)N1CCN(c2cccc(Cl)c2)CC1 ZINC000217750337 CD In-Stock Unstable MAPK1 16 49 N=C(N)CC(=O)N1CCN(c2cccc(Cl)c2)CC1 ZINC000217750337 CD In-Stock Unstable SSTR1 22 49 N=C(N)CC(=O)N1CCN(c2cccc(Cl)c2)CC1 ZINC000217750337 CD In-Stock Unstable ADAM10 16 43 CC(C)[C@H](Br)C(=O)N[C@@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217750356 DH For-Sale Unstable TRPM8 22 57 C[C@@H](N[C@H]1CCN2CCC[C@@H]12)c1cccc(Br)c1 ZINC000217750360 DG For-Sale Unstable MBTD1 0 50 Cc1cc(=O)c(O)c([C@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccc(O)cc2)o1 ZINC000217750369 IH In-Stock Unstable FABI 51 31 Cc1cc(=O)c(O)c([C@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccc(O)cc2)o1 ZINC000217750369 IH In-Stock Unstable DRD5 19 40 Cc1cc(=O)c(O)c([C@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccc(O)cc2)o1 ZINC000217750369 IH In-Stock Unstable SSTR4 40 32 O=C(O)/C=C\c1cccc(NC(=O)c2ccccc2Cl)n1 ZINC000217750403 DG For-Sale Anodyne SORT1 20 45 O=C(O)/C=C\c1cccc(NC(=O)c2ccccc2Cl)n1 ZINC000217750403 DG For-Sale Anodyne NR2E3 62 35 O=C(O)/C=C\c1cccc(NC(=O)c2ccccc2Cl)n1 ZINC000217750403 DG For-Sale Anodyne SMO 25 47 O=C(O)/C=C\c1cccc(NC(=O)c2ccccc2Cl)n1 ZINC000217750403 DG For-Sale Anodyne KCNK3 18 44 CCC[C@@H](O)CNCc1cncn1C1CC1 ZINC000217750434 BD For-Sale Unstable CAMC 0 48 COc1ccccc1N1CCN(C(=O)CC(=N)N)CC1 ZINC000217750436 CC In-Stock Unstable HTR1A 103 52 COc1ccccc1N1CCN(C(=O)CC(=N)N)CC1 ZINC000217750436 CC In-Stock Unstable ADRA2A 17 47 COc1ccccc1N1CCN(C(=O)CC(=N)N)CC1 ZINC000217750436 CC In-Stock Unstable DRD2 90 52 COc1ccccc1N1CCN(C(=O)CC(=N)N)CC1 ZINC000217750436 CC In-Stock Unstable DRD1 34 47 COc1ccccc1N1CCN(C(=O)CC(=N)N)CC1 ZINC000217750436 CC In-Stock Unstable DRD4 40 54 COc1ccccc1N1CCN(C(=O)CC(=N)N)CC1 ZINC000217750436 CC In-Stock Unstable ADRA1D 97 46 COc1ccccc1N1CCN(C(=O)CC(=N)N)CC1 ZINC000217750436 CC In-Stock Unstable HTR1D 28 45 COc1ccccc1N1CCN(C(=O)CC(=N)N)CC1 ZINC000217750436 CC In-Stock Unstable HTR1B 22 53 COc1ccccc1N1CCN(C(=O)CC(=N)N)CC1 ZINC000217750436 CC In-Stock Unstable HTR2A 45 54 COc1ccccc1N1CCN(C(=O)CC(=N)N)CC1 ZINC000217750436 CC In-Stock Unstable ADRA1A 75 46 COc1ccccc1N1CCN(C(=O)CC(=N)N)CC1 ZINC000217750436 CC In-Stock Unstable ADRA1B 65 45 COc1ccccc1N1CCN(C(=O)CC(=N)N)CC1 ZINC000217750436 CC In-Stock Unstable DRD3 76 50 COc1ccccc1N1CCN(C(=O)CC(=N)N)CC1 ZINC000217750436 CC In-Stock Unstable PDGFRB 41 39 COc1ccccc1N1CCN(C(=O)CC(=N)N)CC1 ZINC000217750436 CC In-Stock Unstable TACR1 0 50 COc1ccccc1N1CCN(C(=O)CC(=N)N)CC1 ZINC000217750436 CC In-Stock Unstable HTR7 78 50 COc1ccccc1N1CCN(C(=O)CC(=N)N)CC1 ZINC000217750436 CC In-Stock Unstable MC4R 19 44 COc1ccccc1N1CCN(C(=O)CC(=N)N)CC1 ZINC000217750436 CC In-Stock Unstable KCNQ2 47 34 COc1ccccc1N1CCN(C(=O)CC(=N)N)CC1 ZINC000217750436 CC In-Stock Unstable HTR6 0 53 COc1ccccc1N1CCN(C(=O)CC(=N)N)CC1 ZINC000217750436 CC In-Stock Unstable TACR3 28 50 COc1ccccc1N1CCN(C(=O)CC(=N)N)CC1 ZINC000217750436 CC In-Stock Unstable SSTR1 50 38 COc1ccccc1N1CCN(C(=O)CC(=N)N)CC1 ZINC000217750436 CC In-Stock Unstable ABCB1 0 41 COc1ccccc1N1CCN(C(=O)CC(=N)N)CC1 ZINC000217750436 CC In-Stock Unstable RBP4 19 45 COc1ccccc1N1CCN(C(=O)CC(=N)N)CC1 ZINC000217750436 CC In-Stock Unstable AP2S1 0 45 COc1ccccc1N1CCN(C(=O)CC(=N)N)CC1 ZINC000217750436 CC In-Stock Unstable ALPHA-1A 0 43 COc1ccccc1N1CCN(C(=O)CC(=N)N)CC1 ZINC000217750436 CC In-Stock Unstable BRPF1 0 40 C[C@H](N[C@H]1CCN2CCC[C@@H]12)c1cccc(Br)c1 ZINC000217750438 DG For-Sale Unstable MBTD1 0 50 CC(C)[C@@H](Br)C(=O)N[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217750444 DH For-Sale Unstable TRPM8 22 57 CC[C@@H](C)[C@@H](CO)NC(=O)CC[C@@H]1NC(=O)N(Cc2ccccc2)C1=O ZINC000217750467 FD In-Stock Unstable GALR1 47 34 FC(F)c1ccc([C@@H]2CCCCN2)c(Cl)c1 ZINC000217750487 BI For-Sale Unstable SLC6A1 18 45 CC(C)[C@H](Br)C(=O)N[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217750517 DH For-Sale Unstable TRPM8 22 57 CCC[C@H](O)CNCc1cncn1C1CC1 ZINC000217750519 BD For-Sale Unstable CAMC 0 48 Fc1ccc(Oc2cccc(-c3ccnc4[nH]c(C5CCNCC5)cc34)c2)cc1 ZINC000217750526 GK For-Sale Unstable CHUK 28 40 COC(=O)Nc1ccc(S(=O)(=O)N2CC(N3C(=O)CSC3=O)C2)cc1 ZINC000217750554 GC In-Stock Unstable TGM2 61 37 COC(=O)Nc1ccc(S(=O)(=O)N2CC(N3C(=O)CSC3=O)C2)cc1 ZINC000217750554 GC In-Stock Unstable F13A1 94 40 FC(F)c1ccc([C@H]2CCCCN2)c(Cl)c1 ZINC000217750566 BI For-Sale Unstable SLC6A1 18 45 COc1cc([C@@H]2CC(=O)Oc3cc4c(cc32)OCO4)ccc1O ZINC000217750574 DF In-Stock Unstable E2 0 40 COc1cc([C@@H]2CC(=O)Oc3cc4c(cc32)OCO4)ccc1O ZINC000217750574 DF In-Stock Unstable CAN2 0 42 Cc1ccc(CC(=O)Nc2ncc(/C=C\C(=O)O)s2)cc1 ZINC000217750585 DF For-Sale Unstable CDK5 41 48 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)CCCCCl ZINC000217750599 CH For-Sale Unstable TRPM8 21 64 O=C1CN(C(=O)/C=C\c2cccc(Cl)c2)CC(=O)N1 ZINC000217750607 CC For-Sale Unstable TUBA4A 0 50 O=C1CN(C(=O)/C=C\c2cccc(Cl)c2)CC(=O)N1 ZINC000217750607 CC For-Sale Unstable GPR183 0 41 COc1cc([C@H]2CC(=O)Oc3cc4c(cc32)OCO4)ccc1O ZINC000217750646 DF In-Stock Unstable E2 0 40 COc1cc([C@H]2CC(=O)Oc3cc4c(cc32)OCO4)ccc1O ZINC000217750646 DF In-Stock Unstable CAN2 0 42 CCC[C@@H](O)CNCc1cn(CCO)nn1 ZINC000217750649 BB For-Sale Unstable GBA 17 43 N=C(N)CC(=O)N1CCc2ccccc2C1 ZINC000217750654 BC In-Stock Unstable HTR7 15 40 N=C(N)CC(=O)N1CCc2ccccc2C1 ZINC000217750654 BC In-Stock Unstable HDAC6 31 40 N=C(N)CC(=O)N1CCc2ccccc2C1 ZINC000217750654 BC In-Stock Unstable DPP8 35 60 N=C(N)CC(=O)N1CCc2ccccc2C1 ZINC000217750654 BC In-Stock Unstable BCL2 0 44 N=C(N)CC(=O)N1CCc2ccccc2C1 ZINC000217750654 BC In-Stock Unstable Q6PRC7_IXORI 31 40 N=C(N)CC(=O)N1CCc2ccccc2C1 ZINC000217750654 BC In-Stock Unstable NOD2 42 36 N=C(N)CC(=O)N1CCc2ccccc2C1 ZINC000217750654 BC In-Stock Unstable TRPC6 19 40 CC(C)CCC(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217750669 CG For-Sale Unstable AKR1C3 34 49 O=C(Nc1ccc(-c2nc3ccccc3s2)cc1)c1cc2ccccc2[nH]c1=O ZINC000217750680 GK On-Demand Anodyne HPSE 21 40 O=C(Nc1ccc(-c2nc3ccccc3s2)cc1)c1cc2ccccc2[nH]c1=O ZINC000217750680 GK On-Demand Anodyne NR2E3 71 38 O=C(Nc1ccc(-c2nc3ccccc3s2)cc1)c1cc2ccccc2[nH]c1=O ZINC000217750680 GK On-Demand Anodyne SHH 19 42 O=C(Nc1ccc(-c2nc3ccccc3s2)cc1)c1cc2ccccc2[nH]c1=O ZINC000217750680 GK On-Demand Anodyne LUCI_PHOPE 15 40 O=C(Nc1ccc(-c2nc3ccccc3s2)cc1)c1cc2ccccc2[nH]c1=O ZINC000217750680 GK On-Demand Anodyne SMO 0 40 O=C(Nc1ccc(-c2nc3ccccc3s2)cc1)c1cc2ccccc2[nH]c1=O ZINC000217750680 GK On-Demand Anodyne STK33 51 34 O=C(Nc1ccc(-c2nc3ccccc3s2)cc1)c1cc2ccccc2[nH]c1=O ZINC000217750680 GK On-Demand Anodyne ETHR 15 47 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)CCCCCl ZINC000217750683 CH For-Sale Unstable TRPM8 21 64 COc1ccc(Cl)cc1NC(=O)N/C=C/c1ccccc1F ZINC000217750688 DI For-Sale Unstable RBP4 25 44 COc1ccc(Cl)cc1NC(=O)N/C=C/c1ccccc1F ZINC000217750688 DI For-Sale Unstable CYSP_PLAFA 42 35 O=C1CN(C(=O)/C=C\c2ccc(O)cc2)CC(=O)N1 ZINC000217750697 CB For-Sale Unstable F3 27 49 O=C1CN(C(=O)/C=C\c2ccc(O)cc2)CC(=O)N1 ZINC000217750697 CB For-Sale Unstable SSSIM 15 46 CCC[C@H](O)CNCc1cn(CCO)nn1 ZINC000217750731 BB For-Sale Unstable GBA 17 43 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)CCCCCl ZINC000217750757 CH For-Sale Unstable TRPM8 21 64 CCOCC(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217750758 CD For-Sale Unstable PTGER2 15 42 CCOCC(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217750758 CD For-Sale Unstable NR1H4 41 35 CCOCC(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217750758 CD For-Sale Unstable AKR1C3 32 46 N=C(N)CC(=O)NCc1ccc2c(c1)OCO2 ZINC000217750760 BC In-Stock Unstable PDE5A 30 49 N=C(N)CC(=O)NCc1ccc2c(c1)OCO2 ZINC000217750760 BC In-Stock Unstable EDNRB 29 43 N=C(N)CC(=O)NCc1ccc2c(c1)OCO2 ZINC000217750760 BC In-Stock Unstable EDNRA 25 40 N=C(N)CC(=O)NCc1ccc2c(c1)OCO2 ZINC000217750760 BC In-Stock Unstable BMP1 46 37 N=C(N)CC(=O)NCc1ccc2c(c1)OCO2 ZINC000217750760 BC In-Stock Unstable SCN9A 0 42 N=C(N)CC(=O)NCc1ccc2c(c1)OCO2 ZINC000217750760 BC In-Stock Unstable NOS2 106 41 N=C(N)CC(=O)NCc1ccc2c(c1)OCO2 ZINC000217750760 BC In-Stock Unstable MCHR1 15 40 N=C(N)CC(=O)NCc1ccc2c(c1)OCO2 ZINC000217750760 BC In-Stock Unstable LUXR 23 46 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)CCCCCl ZINC000217750829 CH For-Sale Unstable TRPM8 21 64 CCC[C@@H](C)C(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217750849 CG For-Sale Unstable AKR1C3 31 43 COC(=O)C[C@H](c1c(O)c2ccccc2oc1=O)c1cc2cccc3c2n(c1=O)CC3 ZINC000217750855 HG In-Stock Unstable NQO1 27 43 O=C(O)[C@@]1(O)COC[C@@H](O)C1 ZINC000217750890 AA For-Sale Unstable AROB 79 39 Cc1cccc(/C=C\C(=O)NCC[C@@H](C)O)c1 ZINC000217750896 BD On-Demand Unstable PYGL 23 44 Cc1cccc(/C=C\C(=O)NCC[C@@H](C)O)c1 ZINC000217750896 BD On-Demand Unstable MMP2 0 47 Cc1cccc(/C=C\C(=O)NCC[C@@H](C)O)c1 ZINC000217750896 BD On-Demand Unstable MMP9 0 47 Cc1cccc(/C=C\C(=O)NCC[C@@H](C)O)c1 ZINC000217750896 BD On-Demand Unstable MMP1 0 47 COc1ccc(NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217750912 CH For-Sale Unstable CA1 47 36 COc1ccc(NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217750912 CH For-Sale Unstable MTNR1B 18 45 COc1ccc(NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217750912 CH For-Sale Unstable CA12 21 43 COc1ccc(NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217750912 CH For-Sale Unstable PDGFRA 42 38 COc1ccc(NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217750912 CH For-Sale Unstable CA9 21 43 COc1ccc(NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217750912 CH For-Sale Unstable TLR4 16 43 CCC[C@H](C)C(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217750934 CG For-Sale Unstable AKR1C3 31 43 COC(=O)C[C@@H](c1c(O)c2ccccc2oc1=O)c1cc2cccc3c2n(c1=O)CC3 ZINC000217750939 HG In-Stock Unstable NQO1 27 43 O=C(O)[C@@]1(O)COC[C@H](O)C1 ZINC000217750967 AA For-Sale Unstable AROB 79 39 Cc1cccc(/C=C\C(=O)NCC[C@H](C)O)c1 ZINC000217750972 BD For-Sale Unstable PYGL 23 44 Cc1cccc(/C=C\C(=O)NCC[C@H](C)O)c1 ZINC000217750972 BD For-Sale Unstable HDAC8 59 39 Cc1cccc(/C=C\C(=O)NCC[C@H](C)O)c1 ZINC000217750972 BD For-Sale Unstable MMP2 0 47 Cc1cccc(/C=C\C(=O)NCC[C@H](C)O)c1 ZINC000217750972 BD For-Sale Unstable MMP9 0 47 Cc1cccc(/C=C\C(=O)NCC[C@H](C)O)c1 ZINC000217750972 BD For-Sale Unstable MMP1 0 47 O=C(O)/C=C\c1cccc(NC(=O)c2cc(Cl)c[nH]2)c1 ZINC000217751011 CG For-Sale Anodyne KCNK3 73 42 O=C(N/C=C/c1ccccc1F)Nc1ccc(Cl)cc1Cl ZINC000217751016 EJ For-Sale Anodyne PYGL 19 41 COC1CCN(C2CCN(C(=O)CC(C)(C)C)CC2)CC1 ZINC000217751027 CF In-Stock Unstable L3MBTL3 45 33 O=C(O)[C@]1(O)COC[C@@H](O)C1 ZINC000217751044 AA For-Sale Unstable AROB 79 39 COc1ccccc1CNC(=O)CC(=N)N ZINC000217751083 BC In-Stock Unstable TACR1 26 46 COc1ccccc1CNC(=O)CC(=N)N ZINC000217751083 BC In-Stock Unstable HTR7 17 43 COc1ccccc1CNC(=O)CC(=N)N ZINC000217751083 BC In-Stock Unstable P2RX7 19 48 COc1ccccc1CNC(=O)CC(=N)N ZINC000217751083 BC In-Stock Unstable ACR 24 42 Cc1cc(OC2CN(C(=O)c3cc(=O)c4ccccc4o3)C2)cc(=O)o1 ZINC000217751085 FD In-Stock Unstable TNKS 29 42 CCOC(=O)Cc1cc2cccnc2nc1C ZINC000217751096 BE In-Stock Unstable SUCNR1 44 33 O=C(N/C=C/c1ccccc1F)NCCc1ccc(O)cc1 ZINC000217751129 DG For-Sale Unstable SLC6A5 27 40 O=C(O)[C@]1(O)COC[C@H](O)C1 ZINC000217751133 AA For-Sale Unstable AROB 79 39 COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc2c1OCO2 ZINC000217751177 JI In-Stock Unstable AKR1B1 0 45 COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc2c1OCO2 ZINC000217751177 JI In-Stock Unstable CYP1B1 48 35 COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc2c1OCO2 ZINC000217751177 JI In-Stock Unstable CYP1A2 30 45 CCCCCNC(=O)CC(=N)N ZINC000217751187 AC In-Stock Unstable DNM1 0 44 CCCCCNC(=O)CC(=N)N ZINC000217751187 AC In-Stock Unstable FAAH 0 55 CCCCCNC(=O)CC(=N)N ZINC000217751187 AC In-Stock Unstable EPHX2 32 45 CCCCCNC(=O)CC(=N)N ZINC000217751187 AC In-Stock Unstable ASAH1 74 35 CCCCCNC(=O)CC(=N)N ZINC000217751187 AC In-Stock Unstable NOD1 41 38 CCCCCNC(=O)CC(=N)N ZINC000217751187 AC In-Stock Unstable CQSS 41 31 COc1cccc([C@@H](C)N[C@@H]2CCN3CCC[C@@H]23)c1 ZINC000217751222 CF For-Sale Unstable CHRNA10 28 42 CC(C)NC(=O)N/C=C/c1ccccc1F ZINC000217751225 BF For-Sale Unstable KCNQ2 52 40 COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc2c1OCO2 ZINC000217751255 JI In-Stock Unstable AKR1B1 0 45 COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc2c1OCO2 ZINC000217751255 JI In-Stock Unstable CYP1B1 48 35 COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc2c1OCO2 ZINC000217751255 JI In-Stock Unstable CYP1A2 30 45 COc1cccc([C@H](C)N[C@@H]2CCN3CCC[C@@H]23)c1 ZINC000217751295 CF For-Sale Unstable CHRNA10 28 42 CC(C)CCNC(=O)CC(=N)N ZINC000217751304 AC In-Stock Unstable DNPEP 0 46 CC(C)N(Cc1ccccc1)C(=O)N/C=C/c1ccccc1F ZINC000217751338 DI For-Sale Unstable PTGES 0 40 COc1cccc([C@@H](C)N[C@H]2CCN3CCC[C@@H]23)c1 ZINC000217751371 CF For-Sale Unstable CHRNA10 28 42 CCC[C@@H](C)NC(=O)CC(=N)N ZINC000217751422 AC In-Stock Unstable NOD1 76 40 Cc1cc(NC(=O)c2ccccn2)ccc1/C=C\C(=O)O ZINC000217751457 CF For-Sale Unstable GRM4 89 56 Cc1cc(NC(=O)c2ccccn2)ccc1/C=C\C(=O)O ZINC000217751457 CF For-Sale Unstable SHH 34 44 Cc1cc(NC(=O)c2ccccn2)ccc1/C=C\C(=O)O ZINC000217751457 CF For-Sale Unstable KCNK3 97 55 Cc1cc(NC(=O)c2ccccn2)ccc1/C=C\C(=O)O ZINC000217751457 CF For-Sale Unstable KCNK9 51 39 COc1cccc([C@H](C)N[C@H]2CCN3CCC[C@@H]23)c1 ZINC000217751460 CF For-Sale Unstable CHRNA10 28 42 CCCOCCOc1ccc(S(=O)(=O)Cl)cc1 ZINC000217751471 CE For-Sale Unstable CA7 22 56 CCC[C@H](C)NC(=O)CC(=N)N ZINC000217751515 AC In-Stock Unstable NOD1 76 40 COc1c2ccc(C(=O)NC[C@@H]3CCCN3c3nccs3)cc2nn1C ZINC000217751535 FE For-Sale Unstable ACKR3 60 32 Cc1cc(NC(=O)c2ccncc2)ccc1/C=C\C(=O)O ZINC000217751555 CF For-Sale Unstable TRPV1 15 43 Cc1cc(NC(=O)c2ccncc2)ccc1/C=C\C(=O)O ZINC000217751555 CF For-Sale Unstable PRNP 40 38 Cc1cc(NC(=O)c2ccncc2)ccc1/C=C\C(=O)O ZINC000217751555 CF For-Sale Unstable SHH 31 43 Cc1cc(NC(=O)c2ccncc2)ccc1/C=C\C(=O)O ZINC000217751555 CF For-Sale Unstable NAMPT 17 41 Cc1cc(NC(=O)c2ccncc2)ccc1/C=C\C(=O)O ZINC000217751555 CF For-Sale Unstable KCNK3 108 54 Cc1cc(NC(=O)c2ccncc2)ccc1/C=C\C(=O)O ZINC000217751555 CF For-Sale Unstable KCNK9 52 45 COc1c2ccc(C(=O)NC[C@H]3CCCN3c3nccs3)cc2nn1C ZINC000217751622 FE For-Sale Unstable ACKR3 60 32 COc1cc(-c2cc(C(=O)N3CC(Oc4cc(C)oc(=O)c4)C3)[nH]n2)cc(OC)c1OC ZINC000217751652 IE In-Stock Unstable TACR3 20 44 O=C(c1ccccc1N1CCOCC1)N1CCC[C@@H]1c1ccccn1 ZINC000217751708 EF In-Stock Unstable COLA 83 39 O=C(c1ccccc1N1CCOCC1)N1CCC[C@@H]1c1ccccn1 ZINC000217751708 EF In-Stock Unstable CPT1A 74 39 CCCCCC(=O)Nc1ccc(/C=C\C(=O)O)cc1C ZINC000217751732 CH For-Sale Unstable AKR1C3 24 41 CCCCc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217751739 BE In-Stock Unstable AGTR1 20 41 CCCCc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217751739 BE In-Stock Unstable INHA 26 40 CCCCc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217751739 BE In-Stock Unstable SCN2A 29 63 CCCCc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217751739 BE In-Stock Unstable S1PR4 33 45 CCCCc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217751739 BE In-Stock Unstable S1PR2 43 45 CCCCc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217751739 BE In-Stock Unstable S1PR1 18 45 CCCCc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217751739 BE In-Stock Unstable SPHK1 31 50 CCCCc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217751739 BE In-Stock Unstable S1PR5 35 45 CCCCc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217751739 BE In-Stock Unstable ENPP2 27 46 CCCCc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217751739 BE In-Stock Unstable PPO2 46 44 CCCCc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217751739 BE In-Stock Unstable P96878_MYCTU 15 56 CCCCc1ccc(NC(=O)CC(=N)N)cc1 ZINC000217751739 BE In-Stock Unstable ACAT 0 49 O=C(c1ccccc1N1CCOCC1)N1CCC[C@H]1c1ccccn1 ZINC000217751782 EF In-Stock Unstable COLA 83 39 O=C(c1ccccc1N1CCOCC1)N1CCC[C@H]1c1ccccn1 ZINC000217751782 EF In-Stock Unstable CPT1A 74 39 CCCCC(=O)NCc1cc(/C=C\C(=O)O)ccc1F ZINC000217751817 CF For-Sale Unstable AKR1C3 36 40 CCOC(=O)C1CCN(C(=O)N/C=C/c2ccccc2F)CC1 ZINC000217751825 DF For-Sale Unstable FDFT1 18 40 CSc1ccccc1NC(=O)CC(=N)N ZINC000217751869 BD In-Stock Unstable KCNQ2 44 34 CC[C@@H](CCO)NC(=O)CCCCCl ZINC000217751886 BD For-Sale Unstable PLA2G2C 0 43 CC[C@@H](CCO)NC(=O)CCCCCl ZINC000217751886 BD For-Sale Unstable Q6UB75_PIG 0 40 CC[C@@H](CCO)NC(=O)CCCCCl ZINC000217751886 BD For-Sale Unstable NOD1 47 36 FC(F)c1c(Cl)cccc1[C@@H]1CCCNC1 ZINC000217751889 BH For-Sale Unstable DRD2 15 51 COc1ccccc1-c1cc(C(=O)N2CC(Oc3cc(C)oc(=O)c3)C2)[nH]n1 ZINC000217751896 GE In-Stock Unstable TACR3 24 46 O=C(O)/C=C\c1ccc(F)c(CNC(=O)c2ccco2)c1 ZINC000217751913 CE For-Sale Unstable AKR1C3 27 40 CCCn1c(C(=O)NC[C@@H]2CCCN2c2nccs2)cc2c(=O)n3ccccc3nc21 ZINC000217751917 IF For-Sale Unstable POLR1A 63 33 O=C(N/C=C/c1ccccc1F)NC1CCCCC1 ZINC000217751933 CG For-Sale Unstable EPHX2 26 48 CC[C@H](CCO)NC(=O)CCCCCl ZINC000217751965 BD For-Sale Unstable PLA2G2C 0 43 CC[C@H](CCO)NC(=O)CCCCCl ZINC000217751965 BD For-Sale Unstable Q6UB75_PIG 0 40 CC[C@H](CCO)NC(=O)CCCCCl ZINC000217751965 BD For-Sale Unstable NOD1 47 36 FC(F)c1c(Cl)cccc1[C@H]1CCCNC1 ZINC000217751966 BH For-Sale Unstable DRD2 15 51 Cc1cc(OC2CN(C(=O)CNC(=O)OCc3ccccc3)C2)cc(=O)o1 ZINC000217752004 FD In-Stock Unstable PAPA1_CARPA 50 34 Cc1cc(OC2CN(C(=O)CNC(=O)OCc3ccccc3)C2)cc(=O)o1 ZINC000217752004 FD In-Stock Unstable CAPN1 40 34 Cc1cc(OC2CN(C(=O)CNC(=O)OCc3ccccc3)C2)cc(=O)o1 ZINC000217752004 FD In-Stock Unstable CAPN2 75 34 Cc1cc(OC2CN(C(=O)CNC(=O)OCc3ccccc3)C2)cc(=O)o1 ZINC000217752004 FD In-Stock Unstable NPR 57 33 Cc1cc(OC2CN(C(=O)CNC(=O)OCc3ccccc3)C2)cc(=O)o1 ZINC000217752004 FD In-Stock Unstable RHODESAIN 0 40 CCCn1c(C(=O)NC[C@H]2CCCN2c2nccs2)cc2c(=O)n3ccccc3nc21 ZINC000217752007 IF For-Sale Unstable POLR1A 63 33 COc1cc2c(cc1OC)CC(=O)N(CC(=O)NCCCN(C)C)C=C2 ZINC000217752032 FD In-Stock Unstable HCN2 0 44 FC(F)c1c(Cl)cccc1C1CCNCC1 ZINC000217752077 BH For-Sale Unstable SLC6A4 15 45 CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(-c3cccc(Cl)c3)c(Oc3ccccc3C(F)(F)F)s2)cc1 ZINC000217752085 KK Annotated Unstable CSNK1D 42 42 CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(-c3cccc(Cl)c3)c(Oc3ccccc3C(F)(F)F)s2)cc1 ZINC000217752085 KK Annotated Unstable RORC 84 64 N=C(N)CC(=O)Nc1cc(Cl)ccc1Oc1ccccc1 ZINC000217752086 DG In-Stock Unstable ENR 0 48 COCCn1c(C(=O)NC[C@@H]2CCCN2c2nccs2)cc2c(=O)n3ccccc3nc21 ZINC000217752125 JE For-Sale Unstable POLR1A 68 32 O=C(O)C1CCN(C(=O)N/C=C/c2ccccc2F)CC1 ZINC000217752145 CE For-Sale Unstable SLC6A1 71 38 COC(=O)c1ccccc1Nc1c(NC[C@@H](C)O)c(=O)c1=O ZINC000217752151 DC In-Stock Unstable CXCR2 98 37 COC(=O)c1ccccc1Nc1c(NC[C@@H](C)O)c(=O)c1=O ZINC000217752151 DC In-Stock Unstable CXCR1 71 37 COCCn1c(C(=O)NC[C@H]2CCCN2c2nccs2)cc2c(=O)n3ccccc3nc21 ZINC000217752219 JE For-Sale Unstable POLR1A 68 32 CC[C@@H]1CCN([C@@H]2C[C@@H]2c2ccccc2)CC[C@@H](C)N1 ZINC000217752225 CG For-Sale Unstable SLC18A3 45 37 O=C(N/C=C/c1ccccc1F)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217752249 HJ For-Sale Unstable NMUR2 0 46 O=C(N/C=C/c1ccccc1F)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217752249 HJ For-Sale Unstable NMUR1 0 46 O=C(NC[C@@H]1CCCN2CCCC[C@H]12)c1c[nH]nc1-c1ccc(Cl)cc1Cl ZINC000217752252 HI In-Stock Unstable ALPL 46 37 CC[C@@H](CCO)NC(=O)CCCCl ZINC000217752291 BD For-Sale Unstable PLA2G2C 0 40 Cc1cc(OC2CN(C(=O)c3csc(-c4ccccc4)n3)C2)cc(=O)o1 ZINC000217752292 FF In-Stock Unstable TRPC6 46 34 CCc1cccc(CC)c1NC(=O)CC(=N)N ZINC000217752301 BE In-Stock Unstable ACAT 0 55 CC[C@H]1CCN([C@@H]2C[C@@H]2c2ccccc2)CC[C@@H](C)N1 ZINC000217752303 CG For-Sale Unstable SLC18A3 45 37 CCCCn1c(C(=O)NC[C@@H]2CCCN2c2nccs2)cc2c(=O)n3ccccc3nc21 ZINC000217752317 JG For-Sale Unstable POLR1A 63 32 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cncc(N3CCCC3)n2)CC1 ZINC000217752318 GF On-Demand Unstable HSD11B1 15 58 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cncc(N3CCCC3)n2)CC1 ZINC000217752318 GF On-Demand Unstable SLC18A3 44 53 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cncc(N3CCCC3)n2)CC1 ZINC000217752318 GF On-Demand Unstable WNT3A 48 34 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cncc(N3CCCC3)n2)CC1 ZINC000217752318 GF On-Demand Unstable L3MBTL3 84 45 CC[C@H](CCO)NC(=O)CCCCl ZINC000217752364 BD For-Sale Unstable PLA2G2C 0 40 CCCCn1c(C(=O)NC[C@H]2CCCN2c2nccs2)cc2c(=O)n3ccccc3nc21 ZINC000217752394 JG For-Sale Unstable POLR1A 63 32 COC1CCN(C2CCN(C(=O)c3snnc3C)CC2)CC1 ZINC000217752403 DD In-Stock Unstable L3MBTL3 60 38 Cc1cccc(/C=C\C(=O)N2CC(=O)NC(=O)C2)c1 ZINC000217752411 CC For-Sale Unstable GPR183 0 44 Cc1cccc(C(C)C)c1NC(=O)CC(=N)N ZINC000217752422 BE In-Stock Unstable SOAT1 46 48 Cc1cccc(C(C)C)c1NC(=O)CC(=N)N ZINC000217752422 BE In-Stock Unstable ACAT 0 60 COc1ccc(C(=O)N2CCN(c3ncnc4c3cnn4C)CC2)c2ccccc12 ZINC000217752449 HE On-Demand Unstable PDGFRB 76 41 COc1ccc(C(=O)N2CCN(c3ncnc4c3cnn4C)CC2)c2ccccc12 ZINC000217752449 HE On-Demand Unstable PDE3B 50 34 COCCNC(=O)N/C=C/c1ccccc1F ZINC000217752455 BD For-Sale Unstable TLR4 19 44 Cc1ccc(C(=O)Nc2cc(/C=C\C(=O)O)ccc2C)s1 ZINC000217752470 DH For-Sale Unstable MAPK11 33 40 COc1ccc([C@@H](C)N2c3ccccc3C[C@@H]2C)c(O)c1 ZINC000217752475 CH For-Sale Unstable DRD4 18 42 N=C(N)CC(=O)Nc1ccccc1Oc1ccccc1 ZINC000217752529 CF In-Stock Unstable PYGM 21 48 CCCCNC(=O)N/C=C/c1ccccc1F ZINC000217752575 BF For-Sale Unstable ASAH1 58 37 N=C(N)CC(=O)Nc1ccc(Cl)cc1C(F)(F)F ZINC000217752615 CF In-Stock Unstable TMPRSS4 0 40 C[C@H]1CN[C@@H](C)CCN([C@@H]2C[C@@H]2c2ccccc2)C1 ZINC000217752631 CF For-Sale Unstable SLC18A3 24 42 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(-c3ccccc3)o2)CC1 ZINC000217752655 GJ On-Demand Unstable HTR2A 19 55 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(-c3ccccc3)o2)CC1 ZINC000217752655 GJ On-Demand Unstable GRIN2B 17 42 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(-c3ccccc3)o2)CC1 ZINC000217752655 GJ On-Demand Unstable SLC18A3 58 52 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(-c3ccccc3)o2)CC1 ZINC000217752655 GJ On-Demand Unstable WNT3A 47 36 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(-c3ccccc3)o2)CC1 ZINC000217752655 GJ On-Demand Unstable L3MBTL3 69 42 C[C@H]1CN[C@H](C)CCN([C@@H]2C[C@@H]2c2ccccc2)C1 ZINC000217752668 CF For-Sale Unstable SLC18A3 24 42 O=C(NC[C@@H]1CCCN1c1nccs1)c1cccc(Oc2ccc(F)cc2)c1 ZINC000217752692 GI For-Sale Unstable RAF1 18 42 O=C(NC[C@@H]1CCCN1c1nccs1)c1cccc(Oc2ccc(F)cc2)c1 ZINC000217752692 GI For-Sale Unstable Q8MMZ8_EIMTE 19 42 O=C(NC[C@@H]1CCCN1c1nccs1)c1cccc(Oc2ccc(F)cc2)c1 ZINC000217752692 GI For-Sale Unstable ACKR3 50 31 CC(=O)Nc1cccc(NC(=O)CC(=N)N)c1 ZINC000217752713 BC In-Stock Unstable F2R 0 46 CC(=O)Nc1cccc(NC(=O)CC(=N)N)c1 ZINC000217752713 BC In-Stock Unstable CA4 18 45 CC(=O)Nc1cccc(NC(=O)CC(=N)N)c1 ZINC000217752713 BC In-Stock Unstable CHS1 15 46 CC(=O)Nc1cccc(NC(=O)CC(=N)N)c1 ZINC000217752713 BC In-Stock Unstable NAMPT 24 53 CC(=O)Nc1cccc(NC(=O)CC(=N)N)c1 ZINC000217752713 BC In-Stock Unstable KCNK3 89 40 CC(=O)Nc1cccc(NC(=O)CC(=N)N)c1 ZINC000217752713 BC In-Stock Unstable KCNK9 85 40 O=C(NCCCNc1ccnc2ccccc12)c1ccccc1 ZINC000217752719 DG On-Demand Unstable ACHE 36 50 O=C(NCCCNc1ccnc2ccccc12)c1ccccc1 ZINC000217752719 DG On-Demand Unstable HRP1_PLAFA 93 36 O=C(NCCCNc1ccnc2ccccc12)c1ccccc1 ZINC000217752719 DG On-Demand Unstable DNMT1 36 50 O=C(NCCCNc1ccnc2ccccc12)c1ccccc1 ZINC000217752719 DG On-Demand Unstable BCHE 50 35 O=C(NCCCNc1ccnc2ccccc12)c1ccccc1 ZINC000217752719 DG On-Demand Unstable KCNN3 32 53 O=C(NCCCNc1ccnc2ccccc12)c1ccccc1 ZINC000217752719 DG On-Demand Unstable HNMT 65 47 O=C(NCCCNc1ccnc2ccccc12)c1ccccc1 ZINC000217752719 DG On-Demand Unstable METG 43 30 O=C(NCCCNc1ccnc2ccccc12)c1ccccc1 ZINC000217752719 DG On-Demand Unstable BOTA 19 46 O=C(NCCCNc1ccnc2ccccc12)c1ccccc1 ZINC000217752719 DG On-Demand Unstable KDM4E 23 42 Brc1ccc(-n2cc(-c3nc4ccccc4[nH]3)cn2)cc1 ZINC000217752761 EI On-Demand Anodyne PLAUR 36 49 O=C(NC[C@H]1CCCN1c1nccs1)c1cccc(Oc2ccc(F)cc2)c1 ZINC000217752775 GI For-Sale Unstable RAF1 18 42 O=C(NC[C@H]1CCCN1c1nccs1)c1cccc(Oc2ccc(F)cc2)c1 ZINC000217752775 GI For-Sale Unstable Q8MMZ8_EIMTE 19 42 O=C(NC[C@H]1CCCN1c1nccs1)c1cccc(Oc2ccc(F)cc2)c1 ZINC000217752775 GI For-Sale Unstable ACKR3 50 31 C[C@H]1Cc2ccccc2N1[C@H](C)c1ccc(F)cc1O ZINC000217752781 CI For-Sale Unstable DRD4 19 40 COc1ccc(/C=C\C(=O)O)cc1NC(=O)c1ccc[nH]1 ZINC000217752787 CE For-Sale Unstable TUBB1 41 36 CC[C@@H](C)NC(=O)N/C=C/c1ccccc1F ZINC000217752799 BF For-Sale Unstable KCNQ2 51 38 CCCCOC(=O)c1ccc(NC(=O)CC(=N)N)cc1 ZINC000217752802 CD In-Stock Unstable PRSS1 18 57 CCCCOC(=O)c1ccc(NC(=O)CC(=N)N)cc1 ZINC000217752802 CD In-Stock Unstable SCN2A 16 44 CCCCOC(=O)c1ccc(NC(=O)CC(=N)N)cc1 ZINC000217752802 CD In-Stock Unstable F3 45 33 CCCCOC(=O)c1ccc(NC(=O)CC(=N)N)cc1 ZINC000217752802 CD In-Stock Unstable PLA2G4B 50 35 CCCCOC(=O)c1ccc(NC(=O)CC(=N)N)cc1 ZINC000217752802 CD In-Stock Unstable ACR 79 46 CCCCOC(=O)c1ccc(NC(=O)CC(=N)N)cc1 ZINC000217752802 CD In-Stock Unstable CNGA1 0 49 CCCCOC(=O)c1ccc(NC(=O)CC(=N)N)cc1 ZINC000217752802 CD In-Stock Unstable PPO2 36 46 CCCCOC(=O)c1ccc(NC(=O)CC(=N)N)cc1 ZINC000217752802 CD In-Stock Unstable HGFAC 0 45 COC1CCN(C2CCN(C(=O)Cc3cccc(C)c3)CC2)CC1 ZINC000217752853 EF In-Stock Unstable CHRM2 52 39 COC1CCN(C2CCN(C(=O)Cc3cccc(C)c3)CC2)CC1 ZINC000217752853 EF In-Stock Unstable HRH1 18 42 COC1CCN(C2CCN(C(=O)Cc3cccc(C)c3)CC2)CC1 ZINC000217752853 EF In-Stock Unstable CCR3 39 42 COC1CCN(C2CCN(C(=O)Cc3cccc(C)c3)CC2)CC1 ZINC000217752853 EF In-Stock Unstable L3MBTL3 66 39 COc1ccc(/C=C\C(=O)O)cc1NC(=O)CCC(C)C ZINC000217752869 CG For-Sale Unstable TUBB1 42 37 COc1ccc(/C=C\C(=O)O)cc1NC(=O)CCC(C)C ZINC000217752869 CG For-Sale Unstable AKR1C3 32 44 CC[C@H](C)NC(=O)N/C=C/c1ccccc1F ZINC000217752871 BF For-Sale Unstable KCNQ2 51 38 COC(=O)c1cc(NC(=O)CC(=N)N)cc(C(=O)OC)c1 ZINC000217752877 CC In-Stock Unstable ACR 52 41 CCOC(=O)c1c(NC(=O)CCc2nc(-c3ccncc3)no2)sc2c1CCCC2 ZINC000217752918 IH On-Demand Unstable NS5B 20 50 CCOC(=O)c1c(NC(=O)CCc2nc(-c3ccncc3)no2)sc2c1CCCC2 ZINC000217752918 IH On-Demand Unstable FLT3 19 49 CCOC(=O)c1c(NC(=O)CCc2nc(-c3ccncc3)no2)sc2c1CCCC2 ZINC000217752918 IH On-Demand Unstable HCAR2 37 42 CCOC(=O)c1c(NC(=O)CCc2nc(-c3ccncc3)no2)sc2c1CCCC2 ZINC000217752918 IH On-Demand Unstable VIPR1 27 43 COC(=O)C[C@@H](C1=C(O)C(=O)c2ccccc2C1=O)c1cc(OC)c(OC)c(OC)c1 ZINC000217752946 IG In-Stock Unstable TNF 20 40 CN1CCCN(CC(=O)N2CCC[C@@H](c3cccc(C(=O)O)c3)C2)CC1 ZINC000217752964 FD In-Stock Unstable SLC6A1 55 35 CN1CCCN(CC(=O)N2CCC[C@@H](c3cccc(C(=O)O)c3)C2)CC1 ZINC000217752964 FD In-Stock Unstable NS5B 0 46 O=C(N/C=C/c1ccccc1F)N1CCCc2ccccc21 ZINC000217752968 CH For-Sale Unstable AVPR2 40 45 COc1ccc(C(=O)NC[C@@]23CC[C@@H]4C[C@@H](C[C@@H](C4)C2)C3)cc1 ZINC000217753008 DI In-Stock Unstable P2RX7 22 59 COc1ccc(C(=O)NC[C@@]23CC[C@@H]4C[C@@H](C[C@@H](C4)C2)C3)cc1 ZINC000217753008 DI In-Stock Unstable EPHX2 40 44 COc1ccc(C(=O)NC[C@@]23CC[C@@H]4C[C@@H](C[C@@H](C4)C2)C3)cc1 ZINC000217753008 DI In-Stock Unstable BOTA 16 45 COC(=O)C[C@H](C1=C(O)C(=O)c2ccccc2C1=O)c1cc(OC)c(OC)c(OC)c1 ZINC000217753021 IG In-Stock Unstable TNF 20 40 CCOC(=O)c1c(NC(=O)CN2CCCCCC2=O)sc2c1CCCC2 ZINC000217753022 GG On-Demand Unstable FLT3 16 40 COc1cc(NC(=O)CC(=N)N)c(OC)cc1Cl ZINC000217753033 CD In-Stock Unstable HTR4 41 39 CCCCCCCC(=O)Nc1ncc(/C=C\C(=O)O)s1 ZINC000217753047 CH For-Sale Unstable LASR 42 38 CCCCCCCC(=O)Nc1ncc(/C=C\C(=O)O)s1 ZINC000217753047 CH For-Sale Unstable NOD1 42 35 C[C@H](O)CCNC(=O)/C=C\c1cccc(F)c1 ZINC000217753048 BD On-Demand Unstable PYGL 24 42 C[C@H](O)CCNC(=O)/C=C\c1cccc(F)c1 ZINC000217753048 BD On-Demand Unstable HDAC8 46 35 C[C@H](O)CCNC(=O)/C=C\c1cccc(F)c1 ZINC000217753048 BD On-Demand Unstable MMP2 0 47 C[C@H](O)CCNC(=O)/C=C\c1cccc(F)c1 ZINC000217753048 BD On-Demand Unstable NR1H4 24 41 C[C@H](O)CCNC(=O)/C=C\c1cccc(F)c1 ZINC000217753048 BD On-Demand Unstable MMP9 0 47 C[C@H](O)CCNC(=O)/C=C\c1cccc(F)c1 ZINC000217753048 BD On-Demand Unstable IMPDH2 0 42 C[C@H](O)CCNC(=O)/C=C\c1cccc(F)c1 ZINC000217753048 BD On-Demand Unstable MMP1 0 47 O=C(N/C=C/c1ccccc1F)NCCc1ccccc1 ZINC000217753081 CG For-Sale Unstable CA5B 19 40 O=C(N/C=C/c1ccccc1F)NCCc1ccccc1 ZINC000217753081 CG For-Sale Unstable CA5A 18 40 O=C(NC[C@@H]1CCCN1c1nccs1)c1cccc(OCc2ccccc2)c1 ZINC000217753098 GI For-Sale Unstable DRD4 40 31 CN1CC[C@@H](NS(=O)(=O)c2cc(Br)ccc2Br)C1=O ZINC000217753108 HD On-Demand Unstable CTSC 19 54 N#C/C(=C/c1ccccc1)C(=O)NC(N)=O ZINC000217753118 BC In-Stock Unstable CA12 15 42 C[C@@H](O)CCNC(=O)/C=C\c1cccc(F)c1 ZINC000217753130 BD On-Demand Unstable PYGL 24 42 C[C@@H](O)CCNC(=O)/C=C\c1cccc(F)c1 ZINC000217753130 BD On-Demand Unstable HDAC8 46 35 C[C@@H](O)CCNC(=O)/C=C\c1cccc(F)c1 ZINC000217753130 BD On-Demand Unstable MMP2 16 46 C[C@@H](O)CCNC(=O)/C=C\c1cccc(F)c1 ZINC000217753130 BD On-Demand Unstable NR1H4 24 41 C[C@@H](O)CCNC(=O)/C=C\c1cccc(F)c1 ZINC000217753130 BD On-Demand Unstable MMP9 0 47 C[C@@H](O)CCNC(=O)/C=C\c1cccc(F)c1 ZINC000217753130 BD On-Demand Unstable IMPDH2 0 42 C[C@@H](O)CCNC(=O)/C=C\c1cccc(F)c1 ZINC000217753130 BD On-Demand Unstable MMP1 0 47 CCOC(=O)c1c(NC(=O)CCn2cnc3sccc3c2=O)sc2c1CCCC2 ZINC000217753137 IH On-Demand Unstable NS5B 20 50 CCOC(=O)c1c(NC(=O)CCn2cnc3sccc3c2=O)sc2c1CCCC2 ZINC000217753137 IH On-Demand Unstable FLT3 19 43 Cc1ccc(C(=O)Nc2ncc(/C=C\C(=O)O)s2)cc1F ZINC000217753139 DF For-Sale Unstable SCD1 26 46 Cc1ccc(C(=O)Nc2ncc(/C=C\C(=O)O)s2)cc1F ZINC000217753139 DF For-Sale Unstable SCD 17 46 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable ACE 56 37 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable MME 80 42 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable ANPEP 93 39 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable TACR1 15 42 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable FCER2 40 36 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable CASP3 20 42 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable ACACA 0 41 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable KLK3 59 34 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable CTSB 47 38 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable PAPA1_CARPA 52 34 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable CYSP_TRYCR 51 34 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable CTSG 17 41 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable CTSK 27 47 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable CTSL 41 39 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable NPFFR2 50 38 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable CTRB1 31 42 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable CAPNS1 53 33 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable MMP2 32 43 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable MMP3 69 41 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable MMP8 22 40 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable MMP14 32 41 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable HLA-DRB1 57 38 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable CELA2A 18 41 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable PCSK5 36 40 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable FURIN 49 40 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable CAPN1 70 41 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable MMP9 20 41 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable CAPN2 77 38 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable ACE2 56 36 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable LAP3 56 45 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable CTSC 21 47 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable MMP1 30 42 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable NPR 63 36 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable AMP1_PLAFQ 66 42 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable PSMB5 41 36 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable POLG_WNV 79 41 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable QRFPR 46 34 C[C@@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753143 BD In-Stock Unstable NPFFR1 57 38 N[C@@H](Cc1cnc[nH]1)C1=N/C(=C\c2ccc(O)cc2)C(=O)N1CC(=O)O ZINC000217753153 FC Annotated Unstable AKR1B1 26 40 O=C(NC[C@H]1CCCN1c1nccs1)c1cccc(OCc2ccccc2)c1 ZINC000217753186 GI For-Sale Unstable DRD4 40 31 O=C(N/C=C/c1ccccc1F)NC1CCCC1 ZINC000217753192 BG For-Sale Unstable EPHX2 22 45 CN1CC[C@H](NS(=O)(=O)c2cc(Br)ccc2Br)C1=O ZINC000217753194 HD On-Demand Unstable CTSC 19 54 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable ACE 56 37 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable MME 80 42 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable ANPEP 93 39 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable TACR1 15 42 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable FCER2 40 36 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable CASP3 20 42 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable ACACA 0 41 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable KLK3 59 34 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable CTSB 47 38 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable PAPA1_CARPA 52 34 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable CYSP_TRYCR 51 34 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable CTSG 17 41 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable CTSK 27 47 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable CTSL 41 39 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable NPFFR2 50 38 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable CTRB1 31 42 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable CAPNS1 53 33 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable MMP2 32 43 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable MMP3 69 41 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable MMP8 22 40 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable MMP14 32 41 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable HLA-DRB1 57 38 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable CELA2A 18 41 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable PCSK5 36 40 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable FURIN 49 40 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable CAPN1 70 41 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable MMP9 20 41 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable CAPN2 77 38 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable ACE2 56 36 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable LAP3 56 45 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable CTSC 21 47 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable MMP1 30 42 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable NPR 63 36 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable AMP1_PLAFQ 66 42 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable PSMB5 41 36 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable POLG_WNV 79 41 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable QRFPR 46 34 C[C@H](CCc1ccccc1)NC(=O)CC(=N)N ZINC000217753222 BD In-Stock Unstable NPFFR1 57 38 CCCCCC(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217753231 CG For-Sale Unstable AKR1C3 32 48 O=C(NC1CCN(Cc2cccnc2)CC1)[C@@H]1Cc2cc(Cl)ccc2N1 ZINC000217753264 FF In-Stock Unstable DRD4 40 41 O=C(NC1CCN(Cc2cccnc2)CC1)[C@@H]1Cc2cc(Cl)ccc2N1 ZINC000217753264 FF In-Stock Unstable ACHE 24 42 O=C(NC1CCN(Cc2cccnc2)CC1)[C@@H]1Cc2cc(Cl)ccc2N1 ZINC000217753264 FF In-Stock Unstable SIGMAR1 28 47 O=C(NC1CCN(Cc2cccnc2)CC1)[C@@H]1Cc2cc(Cl)ccc2N1 ZINC000217753264 FF In-Stock Unstable SSTR5 44 39 O=C(NC1CCN(Cc2cccnc2)CC1)[C@@H]1Cc2cc(Cl)ccc2N1 ZINC000217753264 FF In-Stock Unstable CHRNA7 36 41 O=C(NC1CCN(Cc2cccnc2)CC1)[C@@H]1Cc2cc(Cl)ccc2N1 ZINC000217753264 FF In-Stock Unstable C3AR1 46 49 O=C(NC1CCN(Cc2cccnc2)CC1)[C@@H]1Cc2cc(Cl)ccc2N1 ZINC000217753264 FF In-Stock Unstable MCHR1 41 43 O=C(O)[C@H]1CC(=O)N([C@@H]2C[C@@H]2c2ccccc2)C1 ZINC000217753275 BD For-Sale Unstable INHA 37 44 N=C(N)CC(=O)NC1CCCCCCC1 ZINC000217753310 BD In-Stock Unstable EPHX2 21 43 O=C(N/C=C/c1ccccc1F)NCc1ccccc1Cl ZINC000217753324 DH For-Sale Unstable P2RX7 44 40 C[C@H]1Cc2ccccc2N1[C@H](C)c1cc(F)ccc1O ZINC000217753339 CI For-Sale Unstable DRD4 19 40 O=C(O)[C@H]1CC(=O)N([C@H]2C[C@@H]2c2ccccc2)C1 ZINC000217753348 BD For-Sale Unstable INHA 37 44 CN(Cc1cccc(/C=C\C(=O)O)c1)C(=O)C(C)(C)C ZINC000217753350 CF For-Sale Unstable PTGER2 26 44 CN(Cc1cccc(/C=C\C(=O)O)c1)C(=O)C(C)(C)C ZINC000217753350 CF For-Sale Unstable NR1H4 40 38 CN(Cc1cccc(/C=C\C(=O)O)c1)C(=O)C(C)(C)C ZINC000217753350 CF For-Sale Unstable AKR1C3 41 41 O=C(NC1CCN(Cc2cccnc2)CC1)[C@H]1Cc2cc(Cl)ccc2N1 ZINC000217753351 FF In-Stock Unstable DRD4 40 41 O=C(NC1CCN(Cc2cccnc2)CC1)[C@H]1Cc2cc(Cl)ccc2N1 ZINC000217753351 FF In-Stock Unstable ACHE 24 42 O=C(NC1CCN(Cc2cccnc2)CC1)[C@H]1Cc2cc(Cl)ccc2N1 ZINC000217753351 FF In-Stock Unstable SIGMAR1 28 47 O=C(NC1CCN(Cc2cccnc2)CC1)[C@H]1Cc2cc(Cl)ccc2N1 ZINC000217753351 FF In-Stock Unstable SSTR5 44 39 O=C(NC1CCN(Cc2cccnc2)CC1)[C@H]1Cc2cc(Cl)ccc2N1 ZINC000217753351 FF In-Stock Unstable CHRNA7 36 41 O=C(NC1CCN(Cc2cccnc2)CC1)[C@H]1Cc2cc(Cl)ccc2N1 ZINC000217753351 FF In-Stock Unstable C3AR1 46 49 O=C(NC1CCN(Cc2cccnc2)CC1)[C@H]1Cc2cc(Cl)ccc2N1 ZINC000217753351 FF In-Stock Unstable MCHR1 41 43 CCC[C@@H](O)CNC(=O)CCCCCl ZINC000217753354 BD For-Sale Unstable CQSS 42 36 CN1CC[C@@H](NS(=O)(=O)c2ccc(Br)cc2Br)C1=O ZINC000217753364 HD On-Demand Unstable CTSC 16 43 C[C@H](O)CCNC(=O)/C=C\c1ccc(Br)s1 ZINC000217753378 DE For-Sale Unstable SCAF_EBVB9 15 42 N=C(N)CC(=O)NC(c1ccccc1)c1ccccc1 ZINC000217753409 CE In-Stock Unstable C3AR1 59 39 N=C(N)CC(=O)NC(c1ccccc1)c1ccccc1 ZINC000217753409 CE In-Stock Unstable POLG_WNV 50 30 CN1CC[C@H](NS(=O)(=O)c2ccc(Br)cc2Br)C1=O ZINC000217753435 HD On-Demand Unstable CTSC 16 43 CCC[C@H](O)CNC(=O)CCCCCl ZINC000217753446 BD For-Sale Unstable CQSS 42 36 CC[C@@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1cccc(Cl)c1 ZINC000217753456 CD For-Sale Unstable CMA1 21 40 COc1ccc(CCNC(=O)N/C=C/c2ccccc2F)cc1OC ZINC000217753457 EG For-Sale Unstable MTNR1A 15 42 COc1ccc(CCNC(=O)N/C=C/c2ccccc2F)cc1OC ZINC000217753457 EG For-Sale Unstable MTNR1B 19 44 COc1ccc(CCNC(=O)N/C=C/c2ccccc2F)cc1OC ZINC000217753457 EG For-Sale Unstable NCE103 15 45 COC1CCN(C2CCN(C(=O)Cc3ccc(F)cc3)CC2)CC1 ZINC000217753461 EE In-Stock Unstable CHRM2 51 39 COC1CCN(C2CCN(C(=O)Cc3ccc(F)cc3)CC2)CC1 ZINC000217753461 EE In-Stock Unstable HRH1 21 40 COC1CCN(C2CCN(C(=O)Cc3ccc(F)cc3)CC2)CC1 ZINC000217753461 EE In-Stock Unstable CCR3 39 58 COC1CCN(C2CCN(C(=O)Cc3ccc(F)cc3)CC2)CC1 ZINC000217753461 EE In-Stock Unstable MLNR 43 51 COC1CCN(C2CCN(C(=O)Cc3ccc(F)cc3)CC2)CC1 ZINC000217753461 EE In-Stock Unstable L3MBTL3 66 39 C[C@@H](O)CCNC(=O)/C=C\c1ccc(Br)s1 ZINC000217753468 DE On-Demand Unstable SCAF_EBVB9 15 42 O=C1CN(C(=O)/C=C\c2cccc(Br)c2)CC(=O)N1 ZINC000217753479 DC For-Sale Unstable GPR183 0 40 CC[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1cccc(Cl)c1 ZINC000217753540 CD For-Sale Unstable CMA1 21 40 CCOC(=O)[C@@H]1CCC[C@@H]1c1ccccc1 ZINC000217753556 BG On-Demand Unstable SLC6A4 19 40 CCOC(=O)[C@@H]1CCC[C@@H]1c1ccccc1 ZINC000217753556 BG On-Demand Unstable SLC6A3 31 40 CCOC(=O)[C@@H]1CCC[C@@H]1c1ccccc1 ZINC000217753556 BG On-Demand Unstable AMY2 45 32 Cc1cc(OC2CN(S(=O)(=O)c3ccccc3C#N)C2)cc(=O)o1 ZINC000217753559 ED In-Stock Unstable TRPV4 41 33 C[C@H]1Cc2ccccc2N1[C@H](C)c1cc(Cl)ccc1O ZINC000217753595 CJ For-Sale Unstable DRD4 24 45 Cc1ncsc1C(=O)Nc1cccc(/C=C\C(=O)O)c1 ZINC000217753599 CF For-Sale Unstable KCNK3 94 38 Cc1ncsc1C(=O)Nc1cccc(/C=C\C(=O)O)c1 ZINC000217753599 CF For-Sale Unstable KCNK9 56 38 CC[C@@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1cccc(Cl)c1 ZINC000217753625 CD For-Sale Unstable CMA1 21 40 COc1cccc(/C=C\C(=O)N2CC(=O)NC(=O)C2)c1 ZINC000217753634 CC For-Sale Unstable AHR 15 45 COc1cccc(/C=C\C(=O)N2CC(=O)NC(=O)C2)c1 ZINC000217753634 CC For-Sale Unstable ABCG2 15 46 COc1cccc(/C=C\C(=O)N2CC(=O)NC(=O)C2)c1 ZINC000217753634 CC For-Sale Unstable GPR183 0 46 CCCCOCCCNC(=O)N/C=C/c1ccccc1F ZINC000217753669 CG For-Sale Unstable ASAH1 41 33 Cc1nc2ccc(C(=O)NC[C@@H]3CCCN3c3nccs3)cc2s1 ZINC000217753679 FG For-Sale Unstable LCK 27 42 Cc1ccc(C(=O)Nc2cccc(/C=C\C(=O)O)c2)s1 ZINC000217753697 CG For-Sale Unstable HDAC8 17 41 Cc1ccc(C(=O)Nc2cccc(/C=C\C(=O)O)c2)s1 ZINC000217753697 CG For-Sale Unstable KCNK3 107 40 Cc1ccc(C(=O)Nc2cccc(/C=C\C(=O)O)c2)s1 ZINC000217753697 CG For-Sale Unstable KCNK9 67 40 CC[C@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1cccc(Cl)c1 ZINC000217753701 CD For-Sale Unstable CMA1 21 40 C[C@@H](NC(=O)CC(=N)N)c1ccc(Cl)cc1 ZINC000217753721 BD In-Stock Unstable ACACA 41 38 C[C@@H](NC(=O)CC(=N)N)c1ccc(Cl)cc1 ZINC000217753721 BD In-Stock Unstable PRCP 19 45 C[C@@H](NC(=O)CC(=N)N)c1ccc(Cl)cc1 ZINC000217753721 BD In-Stock Unstable F7 30 43 C[C@@H](NC(=O)CC(=N)N)c1ccc(Cl)cc1 ZINC000217753721 BD In-Stock Unstable UTS2 43 35 CCn1ncc2c(C(=O)N3CCN(c4ccc(O)cc4)CC3)cc(-c3ccccc3)nc21 ZINC000217753729 IH On-Demand Unstable P2RY12 52 35 CCn1ncc2c(C(=O)N3CCN(c4ccc(O)cc4)CC3)cc(-c3ccccc3)nc21 ZINC000217753729 IH On-Demand Unstable CCKAR 40 37 CC(C)(C)c1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1 ZINC000217753731 FJ On-Demand Unstable HTR2A 19 50 CC(C)(C)c1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1 ZINC000217753731 FJ On-Demand Unstable INHA 19 46 CC(C)(C)c1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1 ZINC000217753731 FJ On-Demand Unstable SLC18A3 47 56 CC(C)(C)c1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1 ZINC000217753731 FJ On-Demand Unstable EPHX2 17 44 CC(C)(C)c1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1 ZINC000217753731 FJ On-Demand Unstable MLYCD 20 46 CC(C)(C)c1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1 ZINC000217753731 FJ On-Demand Unstable WNT3A 48 34 CC(C)(C)c1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1 ZINC000217753731 FJ On-Demand Unstable L3MBTL3 100 45 Cc1nc2ccc(C(=O)NC[C@H]3CCCN3c3nccs3)cc2s1 ZINC000217753768 FG For-Sale Unstable LCK 27 42 O=C(N/C=C/c1ccccc1F)NCc1cccnc1 ZINC000217753774 CF For-Sale Unstable PTAFR 22 41 O=C(N/C=C/c1ccccc1F)NCc1cccnc1 ZINC000217753774 CF For-Sale Unstable NAMPT 76 51 Cc1ccsc1C(=O)Nc1cccc(/C=C\C(=O)O)c1 ZINC000217753798 CG For-Sale Unstable KCNK3 102 39 Cc1ccsc1C(=O)Nc1cccc(/C=C\C(=O)O)c1 ZINC000217753798 CG For-Sale Unstable KCNK9 59 39 CCOC(=O)c1cc(S(C)(=O)=O)cn1Cc1ccccc1 ZINC000217753800 DE In-Stock Unstable PLA2G2A 45 33 CCOC(=O)c1cc(S(C)(=O)=O)cn1Cc1ccccc1 ZINC000217753800 DE In-Stock Unstable F2RL3 21 48 CCOC(=O)c1cc(S(C)(=O)=O)cn1Cc1ccccc1 ZINC000217753800 DE In-Stock Unstable Q76353_9HIV1 0 44 C[C@H](NC(=O)CC(=N)N)c1ccc(Cl)cc1 ZINC000217753803 BD In-Stock Unstable ACACA 41 38 C[C@H](NC(=O)CC(=N)N)c1ccc(Cl)cc1 ZINC000217753803 BD In-Stock Unstable PRCP 19 45 C[C@H](NC(=O)CC(=N)N)c1ccc(Cl)cc1 ZINC000217753803 BD In-Stock Unstable F7 30 43 C[C@H](NC(=O)CC(=N)N)c1ccc(Cl)cc1 ZINC000217753803 BD In-Stock Unstable UTS2 43 35 Cc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)o1 ZINC000217753851 HI In-Stock Unstable AKR1B1 0 43 Cc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)o1 ZINC000217753851 HI In-Stock Unstable CYP1B1 29 43 Cc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)o1 ZINC000217753851 HI In-Stock Unstable CYP1A1 28 43 Cc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)o1 ZINC000217753851 HI In-Stock Unstable CYP1A2 18 40 O=C(N[C@@H]1CCCN(c2cnccn2)C1)c1ccc(N2CCCC2)cc1 ZINC000217753871 FE In-Stock Unstable PRNP 40 35 O=C(N[C@@H]1CCCN(c2cnccn2)C1)c1ccc(N2CCCC2)cc1 ZINC000217753871 FE In-Stock Unstable HPGDS 29 42 O=C(O)/C=C\c1ccc(NC(=O)c2cccs2)c(F)c1 ZINC000217753880 CG For-Sale Anodyne MMP1 0 43 C[C@@H](NC(=O)CC(=N)N)c1ccc(Br)cc1 ZINC000217753915 CD In-Stock Unstable SDH1 0 51 C[C@@H](NC(=O)CC(=N)N)c1ccc(Br)cc1 ZINC000217753915 CD In-Stock Unstable F7 30 42 Cc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)o1 ZINC000217753936 HI In-Stock Unstable AKR1B1 0 43 Cc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)o1 ZINC000217753936 HI In-Stock Unstable CYP1B1 29 43 Cc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)o1 ZINC000217753936 HI In-Stock Unstable CYP1A1 28 43 Cc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)o1 ZINC000217753936 HI In-Stock Unstable CYP1A2 18 40 O=C(N[C@H]1CCCN(c2cnccn2)C1)c1ccc(N2CCCC2)cc1 ZINC000217753968 FE In-Stock Unstable PRNP 40 35 O=C(N[C@H]1CCCN(c2cnccn2)C1)c1ccc(N2CCCC2)cc1 ZINC000217753968 FE In-Stock Unstable HPGDS 29 42 O=C(N/C=C/c1ccccc1F)N1CCC(Cc2ccccc2)CC1 ZINC000217753996 EI For-Sale Unstable GRIN2B 86 47 O=C(N/C=C/c1ccccc1F)N1CCC(Cc2ccccc2)CC1 ZINC000217753996 EI For-Sale Unstable SIGMAR1 25 41 O=C(N/C=C/c1ccccc1F)N1CCC(Cc2ccccc2)CC1 ZINC000217753996 EI For-Sale Unstable CCR3 56 46 Cc1cc(OC2CN(S(=O)(=O)C[C@@]34CC[C@@H](CC3=O)C4(C)C)C2)cc(=O)o1 ZINC000217754005 GD In-Stock Unstable CXCR3 15 47 C[C@H](NC(=O)CC(=N)N)c1ccc(Br)cc1 ZINC000217754011 CD In-Stock Unstable SDH1 0 51 C[C@H](NC(=O)CC(=N)N)c1ccc(Br)cc1 ZINC000217754011 CD In-Stock Unstable F7 30 42 O=C1CN(C(=O)/C=C\c2cc(Cl)cc(Cl)c2)CC(=O)N1 ZINC000217754017 DD For-Sale Unstable ITGAL 15 40 O=C(O)[C@@H]1[C@H]2CN(C(=O)Cc3ccc(O)c(Cl)c3)C[C@H]21 ZINC000217754110 CD In-Stock Unstable NCE103 31 49 O=C(O)[C@@H]1[C@H]2CN(C(=O)Cc3ccc(O)c(Cl)c3)C[C@H]21 ZINC000217754110 CD In-Stock Unstable P96878_MYCTU 20 45 O=C(O)[C@@H]1[C@H]2CN(C(=O)Cc3ccc(O)c(Cl)c3)C[C@H]21 ZINC000217754110 CD In-Stock Unstable CAN2 0 54 CN1CCC(N(C)C(=O)N/C=C/c2ccccc2F)CC1 ZINC000217754114 CF For-Sale Unstable NPY2R 0 41 COc1ccc([C@@H](C)NC(=O)CC(=N)N)cc1 ZINC000217754124 BD In-Stock Unstable ACACA 26 45 COc1ccc([C@@H](C)NC(=O)CC(=N)N)cc1 ZINC000217754124 BD In-Stock Unstable ACACB 35 45 COc1ccc([C@@H](C)NC(=O)CC(=N)N)cc1 ZINC000217754124 BD In-Stock Unstable F7 31 56 COc1ccc([C@@H](C)NC(=O)CC(=N)N)cc1 ZINC000217754124 BD In-Stock Unstable ACR 18 40 COc1ccc([C@@H](C)NC(=O)CC(=N)N)cc1 ZINC000217754124 BD In-Stock Unstable AOC3 17 43 COc1ccc([C@@H](C)NC(=O)CC(=N)N)cc1 ZINC000217754124 BD In-Stock Unstable DXR 24 44 Cc1cc(NC(=O)c2cccnc2)ccc1/C=C\C(=O)O ZINC000217754138 CF For-Sale Unstable ABL1 20 45 Cc1cc(NC(=O)c2cccnc2)ccc1/C=C\C(=O)O ZINC000217754138 CF For-Sale Unstable KIT 0 41 Cc1cc(NC(=O)c2cccnc2)ccc1/C=C\C(=O)O ZINC000217754138 CF For-Sale Unstable TBXAS1 40 38 Cc1cc(NC(=O)c2cccnc2)ccc1/C=C\C(=O)O ZINC000217754138 CF For-Sale Unstable MAPK9 20 40 Cc1cc(NC(=O)c2cccnc2)ccc1/C=C\C(=O)O ZINC000217754138 CF For-Sale Unstable MAPK10 18 40 Cc1cc(NC(=O)c2cccnc2)ccc1/C=C\C(=O)O ZINC000217754138 CF For-Sale Unstable CSF1R 25 51 Cc1cc(NC(=O)c2cccnc2)ccc1/C=C\C(=O)O ZINC000217754138 CF For-Sale Unstable SHH 26 47 Cc1cc(NC(=O)c2cccnc2)ccc1/C=C\C(=O)O ZINC000217754138 CF For-Sale Unstable NAMPT 21 49 Cc1cc(NC(=O)c2cccnc2)ccc1/C=C\C(=O)O ZINC000217754138 CF For-Sale Unstable KCNK3 102 44 Cc1cc(NC(=O)c2cccnc2)ccc1/C=C\C(=O)O ZINC000217754138 CF For-Sale Unstable KCNK9 50 41 CC(C)C[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@@H](CO)NC(=O)CCCCCCCCCCN)C(N)=O ZINC000217754151 KC For-Sale Unstable TACR2 47 49 CC(C)C[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@@H](CO)NC(=O)CCCCCCCCCCN)C(N)=O ZINC000217754151 KC For-Sale Unstable KLK3 136 64 CC(C)C[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@@H](CO)NC(=O)CCCCCCCCCCN)C(N)=O ZINC000217754151 KC For-Sale Unstable NMT1 73 81 CC(C)C[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@@H](CO)NC(=O)CCCCCCCCCCN)C(N)=O ZINC000217754151 KC For-Sale Unstable F2R 27 41 CC(C)C[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@@H](CO)NC(=O)CCCCCCCCCCN)C(N)=O ZINC000217754151 KC For-Sale Unstable HLA-A 63 52 CC(C)C[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@@H](CO)NC(=O)CCCCCCCCCCN)C(N)=O ZINC000217754151 KC For-Sale Unstable MMP3 15 47 CC(C)C[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@@H](CO)NC(=O)CCCCCCCCCCN)C(N)=O ZINC000217754151 KC For-Sale Unstable HLA-DRB1 86 53 CC(C)C[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@@H](CO)NC(=O)CCCCCCCCCCN)C(N)=O ZINC000217754151 KC For-Sale Unstable FURIN 69 48 CC(C)C[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@@H](CO)NC(=O)CCCCCCCCCCN)C(N)=O ZINC000217754151 KC For-Sale Unstable GHSR 15 48 CC(C)C[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@@H](CO)NC(=O)CCCCCCCCCCN)C(N)=O ZINC000217754151 KC For-Sale Unstable CAPN1 20 43 CC(C)C[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@@H](CO)NC(=O)CCCCCCCCCCN)C(N)=O ZINC000217754151 KC For-Sale Unstable PRKACA 45 36 CC(C)C[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@@H](CO)NC(=O)CCCCCCCCCCN)C(N)=O ZINC000217754151 KC For-Sale Unstable SIRT1 34 44 CC(C)C[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@@H](CO)NC(=O)CCCCCCCCCCN)C(N)=O ZINC000217754151 KC For-Sale Unstable KISS1R 55 34 CC(C)C[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@@H](CO)NC(=O)CCCCCCCCCCN)C(N)=O ZINC000217754151 KC For-Sale Unstable POLG_WNV 87 39 CC(C)C[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@@H](CO)NC(=O)CCCCCCCCCCN)C(N)=O ZINC000217754151 KC For-Sale Unstable QRFPR 50 38 CC(C)C[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@@H](CO)NC(=O)CCCCCCCCCCN)C(N)=O ZINC000217754151 KC For-Sale Unstable F2RL1 57 40 CC(C)C[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@@H](CO)NC(=O)CCCCCCCCCCN)C(N)=O ZINC000217754151 KC For-Sale Unstable NOD1 89 51 CC(C)C[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@@H](CO)NC(=O)CCCCCCCCCCN)C(N)=O ZINC000217754151 KC For-Sale Unstable HPN 77 45 COc1ccc([C@H](C)NC(=O)CC(=N)N)cc1 ZINC000217754201 BD In-Stock Unstable ACACA 26 45 COc1ccc([C@H](C)NC(=O)CC(=N)N)cc1 ZINC000217754201 BD In-Stock Unstable ACACB 35 45 COc1ccc([C@H](C)NC(=O)CC(=N)N)cc1 ZINC000217754201 BD In-Stock Unstable F7 31 56 COc1ccc([C@H](C)NC(=O)CC(=N)N)cc1 ZINC000217754201 BD In-Stock Unstable ACR 18 40 COc1ccc([C@H](C)NC(=O)CC(=N)N)cc1 ZINC000217754201 BD In-Stock Unstable AOC3 17 43 COc1ccc([C@H](C)NC(=O)CC(=N)N)cc1 ZINC000217754201 BD In-Stock Unstable DXR 24 44 COC(=O)Nc1ccc(S(=O)(=O)N2CC(Oc3cc(C)oc(=O)c3)C2)cc1 ZINC000217754221 GD In-Stock Unstable F13A1 60 36 Cc1cc(NC(=O)c2ccco2)ccc1/C=C\C(=O)O ZINC000217754222 CF For-Sale Unstable KCNK3 78 56 COc1ccc(CCNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217754233 DG For-Sale Unstable NQO2 23 40 COc1ccc(CCNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217754233 DG For-Sale Unstable MTNR1A 65 45 COc1ccc(CCNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217754233 DG For-Sale Unstable MTNR1B 57 45 COc1ccc(CCNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217754233 DG For-Sale Unstable CA9 18 45 Cc1cccc(N2CCN(CCC(=O)N(C)Cc3ncc[nH]3)CC2)c1 ZINC000217754239 ED In-Stock Unstable HTR1A 33 50 Cc1cccc(N2CCN(CCC(=O)N(C)Cc3ncc[nH]3)CC2)c1 ZINC000217754239 ED In-Stock Unstable DRD2 17 50 Cc1cccc(N2CCN(CCC(=O)N(C)Cc3ncc[nH]3)CC2)c1 ZINC000217754239 ED In-Stock Unstable HTR2A 28 50 Cc1cccc(N2CCN(CCC(=O)N(C)Cc3ncc[nH]3)CC2)c1 ZINC000217754239 ED In-Stock Unstable DRD3 19 43 Cc1cccc(N2CCN(CCC(=O)N(C)Cc3ncc[nH]3)CC2)c1 ZINC000217754239 ED In-Stock Unstable HTR7 43 38 COc1ccc([C@@H](C)NC(=O)CC(=N)N)cc1OC ZINC000217754306 CD In-Stock Unstable TNF 21 40 COc1ccc([C@@H](C)NC(=O)CC(=N)N)cc1OC ZINC000217754306 CD In-Stock Unstable TRPV1 0 52 COc1ccc([C@@H](C)NC(=O)CC(=N)N)cc1OC ZINC000217754306 CD In-Stock Unstable F7 32 42 COc1ccc([C@@H](C)NC(=O)CC(=N)N)cc1OC ZINC000217754306 CD In-Stock Unstable ENPP1 58 33 COc1ccc([C@H](C)NC(=O)CC(=N)N)cc1OC ZINC000217754383 CD In-Stock Unstable TNF 21 40 COc1ccc([C@H](C)NC(=O)CC(=N)N)cc1OC ZINC000217754383 CD In-Stock Unstable F7 32 42 COc1ccc([C@H](C)NC(=O)CC(=N)N)cc1OC ZINC000217754383 CD In-Stock Unstable ENPP1 58 33 O=C(c1ccc(F)cc1)C1CCN(C(=O)C2(c3ccccc3)CCCC2)CC1 ZINC000217754387 GJ On-Demand Unstable SLC18A3 54 51 O=C(c1ccc(F)cc1)C1CCN(C(=O)C2(c3ccccc3)CCCC2)CC1 ZINC000217754387 GJ On-Demand Unstable CACNA1G 24 41 O=C(c1ccc(F)cc1)C1CCN(C(=O)C2(c3ccccc3)CCCC2)CC1 ZINC000217754387 GJ On-Demand Unstable WNT3A 46 34 O=C(c1ccc(F)cc1)C1CCN(C(=O)C2(c3ccccc3)CCCC2)CC1 ZINC000217754387 GJ On-Demand Unstable L3MBTL3 52 34 COC(=O)C[C@@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(OCCc2ccccc2)cc1 ZINC000217754406 JJ In-Stock Unstable LTA4H 27 40 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccccc1C(=O)c1ccc(F)cc1 ZINC000217754441 HH For-Sale Unstable HCRTR1 35 44 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccccc1C(=O)c1ccc(F)cc1 ZINC000217754441 HH For-Sale Unstable PLA2G4A 79 37 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccccc1C(=O)c1ccc(F)cc1 ZINC000217754441 HH For-Sale Unstable HCRTR2 28 44 COC(=O)C[C@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(OCCc2ccccc2)cc1 ZINC000217754483 JJ In-Stock Unstable LTA4H 27 40 COc1ccccc1[C@@H](C)NC(=O)CC(=N)N ZINC000217754487 BD In-Stock Unstable ACR 23 41 COc1ccccc1[C@@H](C)NC(=O)CC(=N)N ZINC000217754487 BD In-Stock Unstable KCNK3 39 43 COc1ccccc1[C@@H](C)NC(=O)CC(=N)N ZINC000217754487 BD In-Stock Unstable KCNK9 34 43 CC[C@@H](C)N(C)CCNCc1ccc2c(c1)OCO2 ZINC000217754530 CE For-Sale Unstable NOS2 35 43 O=C(NC[C@H]1CCCN1c1nccs1)c1ccccc1C(=O)c1ccc(F)cc1 ZINC000217754534 HH For-Sale Unstable HCRTR1 35 44 O=C(NC[C@H]1CCCN1c1nccs1)c1ccccc1C(=O)c1ccc(F)cc1 ZINC000217754534 HH For-Sale Unstable PLA2G4A 79 37 O=C(NC[C@H]1CCCN1c1nccs1)c1ccccc1C(=O)c1ccc(F)cc1 ZINC000217754534 HH For-Sale Unstable HCRTR2 28 44 Cc1ccc(/C=C\C(=O)O)cc1NC(=O)Cn1cncn1 ZINC000217754542 CD For-Sale Unstable HIS3 40 31 O=C(N/C=C/c1ccccc1F)NCc1ccc(Cl)cc1 ZINC000217754545 DH For-Sale Unstable AMP1_PLAFQ 19 40 COc1ccccc1[C@H](C)NC(=O)CC(=N)N ZINC000217754574 BD In-Stock Unstable ACR 23 41 COc1ccccc1[C@H](C)NC(=O)CC(=N)N ZINC000217754574 BD In-Stock Unstable KCNK3 39 43 COc1ccccc1[C@H](C)NC(=O)CC(=N)N ZINC000217754574 BD In-Stock Unstable KCNK9 34 43 CC[C@H](C)N(C)CCNCc1ccc2c(c1)OCO2 ZINC000217754608 CE For-Sale Unstable NOS2 35 43 C[C@@H](NC(=O)N/C=C/c1ccccc1F)c1ccccc1 ZINC000217754656 CH For-Sale Unstable KCNQ2 60 47 COC1CCN(C2CCN(C(=O)c3ccc(N(C)C)cc3)CC2)CC1 ZINC000217754662 EE In-Stock Unstable CHRM2 55 38 COC1CCN(C2CCN(C(=O)c3ccc(N(C)C)cc3)CC2)CC1 ZINC000217754662 EE In-Stock Unstable HRH1 17 45 COC1CCN(C2CCN(C(=O)c3ccc(N(C)C)cc3)CC2)CC1 ZINC000217754662 EE In-Stock Unstable AVPR1A 25 51 COC1CCN(C2CCN(C(=O)c3ccc(N(C)C)cc3)CC2)CC1 ZINC000217754662 EE In-Stock Unstable HRH3 17 45 COC1CCN(C2CCN(C(=O)c3ccc(N(C)C)cc3)CC2)CC1 ZINC000217754662 EE In-Stock Unstable CCR3 46 45 COC1CCN(C2CCN(C(=O)c3ccc(N(C)C)cc3)CC2)CC1 ZINC000217754662 EE In-Stock Unstable L3MBTL3 99 57 COCCNC(=O)[C@@]12C[C@@H]3C[C@@H](C[C@@](Cl)(C3)C1)C2 ZINC000217754679 CE In-Stock Unstable EPHX2 24 42 CC(C)Oc1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2)cc1 ZINC000217754683 CD In-Stock Unstable ACACA 21 47 N=C(N)CC(=O)N[C@@H]1CCCc2ccccc21 ZINC000217754699 BD In-Stock Unstable BDKRB1 54 37 N=C(N)CC(=O)N[C@@H]1CCCc2ccccc21 ZINC000217754699 BD In-Stock Unstable KCNN3 17 40 N=C(N)CC(=O)N[C@@H]1CCCc2ccccc21 ZINC000217754699 BD In-Stock Unstable XIAP 22 41 N=C(N)CC(=O)N[C@@H]1CCCc2ccccc21 ZINC000217754699 BD In-Stock Unstable BIRC3 27 40 N=C(N)CC(=O)N[C@@H]1CCCc2ccccc21 ZINC000217754699 BD In-Stock Unstable BIRC2 42 40 C[C@H](NC(=O)N/C=C/c1ccccc1F)c1ccccc1 ZINC000217754732 CH For-Sale Unstable KCNQ2 60 47 CC(C)Oc1ccc([C@@H](C)NC(=O)[C@H]2C[C@@H](O)CN2)cc1 ZINC000217754751 CD On-Demand Unstable ACACA 0 47 CN(Cc1cc(C2CC2)[nH]n1)C(=O)CCn1ccc(=O)[nH]c1=O ZINC000217754754 DC In-Stock Unstable DUT 65 36 Cc1cc(N2CCN3CCC[C@@H]3C2)ccc1CBr ZINC000217754760 DG For-Sale Unstable HRH3 0 44 Cc1cc(N2CCN3CCC[C@@H]3C2)ccc1CBr ZINC000217754760 DG For-Sale Unstable ADCY5 40 42 N=C(N)CC(=O)N[C@H]1CCCc2ccccc21 ZINC000217754785 BD In-Stock Unstable BDKRB1 54 37 N=C(N)CC(=O)N[C@H]1CCCc2ccccc21 ZINC000217754785 BD In-Stock Unstable KCNN3 17 40 N=C(N)CC(=O)N[C@H]1CCCc2ccccc21 ZINC000217754785 BD In-Stock Unstable XIAP 22 41 N=C(N)CC(=O)N[C@H]1CCCc2ccccc21 ZINC000217754785 BD In-Stock Unstable BIRC3 27 40 N=C(N)CC(=O)N[C@H]1CCCc2ccccc21 ZINC000217754785 BD In-Stock Unstable BIRC2 42 40 Cc1ccc(/C=C\C(=O)O)cc1NC(=O)CC(C)(C)C ZINC000217754792 CG For-Sale Unstable MMP1 0 41 COCc1cc(=O)c(O)c([C@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccc(OC)c(OC)c2)o1 ZINC000217754826 KI In-Stock Unstable RORC 43 33 CC(C)Oc1ccc([C@H](C)NC(=O)[C@H]2C[C@@H](O)CN2)cc1 ZINC000217754827 CD In-Stock Unstable ACACA 21 47 O=C(N/C=C/c1ccccc1F)NC(c1ccccc1)c1ccccc1 ZINC000217754838 EJ For-Sale Anodyne KCNQ2 50 39 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cc([N+](=O)[O-])c[nH]2)CC1 ZINC000217754844 EF On-Demand Unstable SLC18A3 31 44 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cc([N+](=O)[O-])c[nH]2)CC1 ZINC000217754844 EF On-Demand Unstable L3MBTL3 50 33 Cc1ccc(/C=C\C(=O)O)cc1NC(=O)Cc1cccs1 ZINC000217754902 DG For-Sale Unstable CA5B 46 45 Cc1ccc(/C=C\C(=O)O)cc1NC(=O)Cc1cccs1 ZINC000217754902 DG For-Sale Unstable CA5A 47 45 C[C@@H](NC(=O)CC(=N)N)c1cccc(Br)c1 ZINC000217754906 CD In-Stock Unstable F7 30 61 COCc1cc(=O)c(O)c([C@@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccc(OC)c(OC)c2)o1 ZINC000217754911 KI In-Stock Unstable RORC 43 33 CC(=O)Oc1ccc(C(=O)O)cc1C(=O)O ZINC000217754913 BD For-Sale Unstable GRM2 18 40 CC(=O)Oc1ccc(C(=O)O)cc1C(=O)O ZINC000217754913 BD For-Sale Unstable AKR1C3 44 45 CC(=O)Oc1ccc(C(=O)O)cc1C(=O)O ZINC000217754913 BD For-Sale Unstable AKR1C2 44 45 CC[C@@H](C)c1ccc(S(=O)(=O)N2CCC[C@@H](O)C2)cc1 ZINC000217754917 CE On-Demand Unstable SCN2A 19 41 CC[C@@H](C)c1ccc(S(=O)(=O)N2CCC[C@@H](O)C2)cc1 ZINC000217754917 CE On-Demand Unstable AKR1C3 37 55 CCOC(=O)CN(C(=O)Cn1cnc2sc3c(c2c1=O)CCCCC3)c1ccccc1 ZINC000217754943 IG On-Demand Unstable HTR1B 18 41 COc1ccc(CNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217754956 DG For-Sale Unstable MTNR1A 19 46 COc1ccc(CNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217754956 DG For-Sale Unstable MTNR1B 16 46 COc1ccc(CNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217754956 DG For-Sale Unstable CA9 15 43 COc1ccc(CNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217754956 DG For-Sale Unstable U38 0 41 COc1ccc(CNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217754956 DG For-Sale Unstable KCNJ2 0 41 C[C@H](Oc1ccc(Cl)cc1)C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217754971 GI On-Demand Unstable CCR1 44 42 C[C@H](Oc1ccc(Cl)cc1)C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217754971 GI On-Demand Unstable SLC18A3 40 48 C[C@H](Oc1ccc(Cl)cc1)C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217754971 GI On-Demand Unstable WNT3A 52 35 C[C@H](NC(=O)CC(=N)N)c1cccc(Br)c1 ZINC000217754989 CD In-Stock Unstable F7 30 61 BrCc1ccc(N2CCN3CCC[C@@H]3C2)cc1 ZINC000217755003 CF For-Sale Unstable HRH3 0 50 BrCc1ccc(N2CCN3CCC[C@@H]3C2)cc1 ZINC000217755003 CF For-Sale Unstable ADCY5 41 42 BrCc1ccc(N2CCN3CCC[C@@H]3C2)cc1 ZINC000217755003 CF For-Sale Unstable L3MBTL3 60 46 CC[C@H](C)c1ccc(S(=O)(=O)N2CCC[C@@H](O)C2)cc1 ZINC000217755007 CE On-Demand Unstable SCN2A 19 41 CC[C@H](C)c1ccc(S(=O)(=O)N2CCC[C@@H](O)C2)cc1 ZINC000217755007 CE On-Demand Unstable AKR1C3 37 55 COc1cc(OC)c([C@@H]2CC(=O)Oc3ccc4c(c32)OC(=C(C)C)C4=O)cc1OC ZINC000217755018 HI In-Stock Unstable MT-ND4 53 35 c1ccc([C@@H]2C[C@H]2N[C@H]2CCCc3ccccc32)cc1 ZINC000217755033 CI For-Sale Unstable KCNN3 20 41 O=C(O)/C=C\c1cccc(NC(=O)c2ccccc2)n1 ZINC000217755047 CE For-Sale Anodyne GRM5 21 42 O=C(O)/C=C\c1cccc(NC(=O)c2ccccc2)n1 ZINC000217755047 CE For-Sale Anodyne LUCI_LUCLA 35 42 O=C(O)/C=C\c1cccc(NC(=O)c2ccccc2)n1 ZINC000217755047 CE For-Sale Anodyne KCNK3 78 41 COc1ccc(CNC(=O)CC(=N)N)cc1OC ZINC000217755094 CC In-Stock Unstable TRPV1 49 51 COc1ccc(CNC(=O)CC(=N)N)cc1OC ZINC000217755094 CC In-Stock Unstable PDE6A 43 33 COc1ccc(CNC(=O)CC(=N)N)cc1OC ZINC000217755094 CC In-Stock Unstable ACR 25 40 COc1ccc(CNC(=O)CC(=N)N)cc1OC ZINC000217755094 CC In-Stock Unstable MT-ND1 30 51 COc1ccc(CNC(=O)CC(=N)N)cc1OC ZINC000217755094 CC In-Stock Unstable CA9 20 41 COc1ccc(CNC(=O)CC(=N)N)cc1OC ZINC000217755094 CC In-Stock Unstable NCE103 16 45 COc1ccc(CNC(=O)CC(=N)N)cc1OC ZINC000217755094 CC In-Stock Unstable ABCG2 24 40 COc1ccc(CNC(=O)CC(=N)N)cc1OC ZINC000217755094 CC In-Stock Unstable ENPP1 56 34 COc1ccc(CNC(=O)CC(=N)N)cc1OC ZINC000217755094 CC In-Stock Unstable DRTS_TRYCR 53 39 COc1ccc(CNC(=O)CC(=N)N)cc1OC ZINC000217755094 CC In-Stock Unstable CAN2 0 45 COc1cc(OC)c([C@H]2CC(=O)Oc3ccc4c(c32)OC(=C(C)C)C4=O)cc1OC ZINC000217755099 HI In-Stock Unstable MT-ND4 53 35 c1ccc([C@@H]2C[C@@H]2N[C@H]2CCCc3ccccc32)cc1 ZINC000217755112 CI For-Sale Unstable KCNN3 20 41 CCOCC(=O)Nc1cc(/C=C\C(=O)O)ccc1OC ZINC000217755135 CD For-Sale Unstable TUBB1 47 37 CCOCC(=O)Nc1cc(/C=C\C(=O)O)ccc1OC ZINC000217755135 CD For-Sale Unstable AKR1C3 29 41 COC(=O)COc1ccc2occ(-c3ccc(OC)cc3)c2c1 ZINC000217755192 DH In-Stock Unstable ALDH2 103 49 COC(=O)COc1ccc2occ(-c3ccc(OC)cc3)c2c1 ZINC000217755192 DH In-Stock Unstable NQO2 26 45 COC(=O)COc1ccc2occ(-c3ccc(OC)cc3)c2c1 ZINC000217755192 DH In-Stock Unstable GSK3B 0 53 COC(=O)COc1ccc2occ(-c3ccc(OC)cc3)c2c1 ZINC000217755192 DH In-Stock Unstable MTNR1A 63 45 COC(=O)COc1ccc2occ(-c3ccc(OC)cc3)c2c1 ZINC000217755192 DH In-Stock Unstable MTNR1B 47 45 O=C(N/C=C/c1ccccc1F)NCc1ccc2c(c1)OCO2 ZINC000217755199 DG For-Sale Unstable PDE5A 31 41 O=C(N/C=C/c1ccccc1F)NCc1ccc2c(c1)OCO2 ZINC000217755199 DG For-Sale Unstable BMP1 42 37 O=C(N/C=C/c1ccccc1F)NCc1ccc2c(c1)OCO2 ZINC000217755199 DG For-Sale Unstable SCN9A 24 43 O=C(N/C=C/c1ccccc1F)NCc1ccc2c(c1)OCO2 ZINC000217755199 DG For-Sale Unstable NOS2 87 36 O=C(N/C=C/c1ccccc1F)NCc1ccc2c(c1)OCO2 ZINC000217755199 DG For-Sale Unstable MCHR1 18 43 N=C(N)CC(=O)NCc1ccc(F)cc1 ZINC000217755208 BC In-Stock Unstable TPSAB1 22 49 CCC[C@@H](C)C(=O)Nc1cc(/C=C\C(=O)O)ccc1OC ZINC000217755215 CG For-Sale Unstable TUBB1 41 36 CCC[C@@H](C)C(=O)Nc1cc(/C=C\C(=O)O)ccc1OC ZINC000217755215 CG For-Sale Unstable AKR1C3 29 40 COc1cccc(C(=O)NCC(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217755236 FD For-Sale Unstable DRD4 50 38 COc1cccc(C(=O)NCC(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217755236 FD For-Sale Unstable CCR2 41 43 COc1cccc(C(=O)NCC(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217755236 FD For-Sale Unstable ACKR3 51 33 CCOc1ccccc1C(=O)N1CC(Oc2cc(C)n(C)c(=O)c2)C1 ZINC000217755278 ED In-Stock Unstable HCN1 45 35 CCOc1ccccc1C(=O)N1CC(Oc2cc(C)n(C)c(=O)c2)C1 ZINC000217755278 ED In-Stock Unstable HCN4 45 35 CCC[C@H](C)C(=O)Nc1cc(/C=C\C(=O)O)ccc1OC ZINC000217755280 CG For-Sale Unstable TUBB1 41 36 CCC[C@H](C)C(=O)Nc1cc(/C=C\C(=O)O)ccc1OC ZINC000217755280 CG For-Sale Unstable AKR1C3 29 40 Cc1cccc2c(Br)c(C(=O)O)[nH]c12 ZINC000217755300 CF For-Sale Unstable ALB 16 43 Cc1cccc2c(Br)c(C(=O)O)[nH]c12 ZINC000217755300 CF For-Sale Unstable MCL1 21 43 COc1cccc(C(=O)NCC(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217755304 FD For-Sale Unstable DRD4 50 38 COc1cccc(C(=O)NCC(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217755304 FD For-Sale Unstable CCR2 41 43 COc1cccc(C(=O)NCC(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217755304 FD For-Sale Unstable ACKR3 51 33 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217755308 EE For-Sale Unstable CA2 100 56 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217755308 EE For-Sale Unstable CA1 95 56 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217755308 EE For-Sale Unstable CA7 45 48 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217755308 EE For-Sale Unstable CA5B 66 48 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217755308 EE For-Sale Unstable CA4 75 56 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217755308 EE For-Sale Unstable CA5A 71 48 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217755308 EE For-Sale Unstable CA14 32 48 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217755308 EE For-Sale Unstable CA12 80 55 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217755308 EE For-Sale Unstable CA9 83 51 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217755308 EE For-Sale Unstable IDO1 0 41 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217755308 EE For-Sale Unstable NCE103 57 46 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217755308 EE For-Sale Unstable MTCA1 64 56 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217755308 EE For-Sale Unstable P96878_MYCTU 79 56 O=c1c2c3c(sc2ncn1Cc1nc(-c2cccc(C(F)(F)F)c2)no1)CCCCC3 ZINC000217755336 IJ On-Demand Unstable RBP4 17 45 CCCCCC(=O)Nc1cc(/C=C\C(=O)O)ccc1OC ZINC000217755377 CG For-Sale Unstable TRPV1 0 42 CCCCCC(=O)Nc1cc(/C=C\C(=O)O)ccc1OC ZINC000217755377 CG For-Sale Unstable MSR1 0 40 CCCCCC(=O)Nc1cc(/C=C\C(=O)O)ccc1OC ZINC000217755377 CG For-Sale Unstable TUBB1 46 37 CCCCCC(=O)Nc1cc(/C=C\C(=O)O)ccc1OC ZINC000217755377 CG For-Sale Unstable AKR1C3 30 46 CCCCCC(=O)Nc1cc(/C=C\C(=O)O)ccc1OC ZINC000217755377 CG For-Sale Unstable ACAT 0 56 Cc1n[nH]c(C)c1CCNC(=O)c1cccc(CN2CCCCCC2)c1 ZINC000217755418 FG In-Stock Unstable DRD2 17 41 Cc1n[nH]c(C)c1CCNC(=O)c1cccc(CN2CCCCCC2)c1 ZINC000217755418 FG In-Stock Unstable DRD4 47 36 Cc1n[nH]c(C)c1CCNC(=O)c1cccc(CN2CCCCCC2)c1 ZINC000217755418 FG In-Stock Unstable HRH2 39 41 Cc1n[nH]c(C)c1CCNC(=O)c1cccc(CN2CCCCCC2)c1 ZINC000217755418 FG In-Stock Unstable CHRM3 15 44 Cc1n[nH]c(C)c1CCNC(=O)c1cccc(CN2CCCCCC2)c1 ZINC000217755418 FG In-Stock Unstable BDKRB1 28 40 Cc1n[nH]c(C)c1CCNC(=O)c1cccc(CN2CCCCCC2)c1 ZINC000217755418 FG In-Stock Unstable KDM4E 21 40 Cc1n[nH]c(C)c1CCNC(=O)c1cccc(CN2CCCCCC2)c1 ZINC000217755418 FG In-Stock Unstable HAO2 84 42 N=C(N)CC(=O)Nc1ccc(F)c(F)c1 ZINC000217755432 BD In-Stock Unstable SLC1A1 48 36 N=C(N)CC(=O)Nc1ccc(F)c(F)c1 ZINC000217755432 BD In-Stock Unstable SLC1A3 51 40 N=C(N)CC(=O)Nc1ccc(F)c(F)c1 ZINC000217755432 BD In-Stock Unstable SLC1A2 61 44 Cc1cccc2[nH]c(C(=O)O)c(Br)c12 ZINC000217755505 CF For-Sale Unstable MCL1 18 41 O=C1C[C@H](C(F)(F)F)N(C(=O)Cn2cnc3sc4c(c3c2=O)CCCCC4)c2ccccc2N1 ZINC000217755546 JI On-Demand Unstable HTR1B 18 40 C[C@H](O)CCNC(=O)/C=C\c1cc(Cl)ccc1Cl ZINC000217755563 CF For-Sale Unstable PYGL 25 45 C[C@H](O)CCNC(=O)/C=C\c1cc(Cl)ccc1Cl ZINC000217755563 CF For-Sale Unstable HDAC7 21 45 C[C@H](O)CCNC(=O)/C=C\c1cc(Cl)ccc1Cl ZINC000217755563 CF For-Sale Unstable BOTA 29 45 CC(C)C[C@@H](C(=O)O)n1cc(CNC(=O)OCC2c3ccccc3-c3ccccc32)nn1 ZINC000217755569 IH For-Sale Unstable NPR 56 32 CN1CCN(CCc2ccc(F)cc2)C[C@@H](O)C1 ZINC000217755574 CC In-Stock Unstable SLC6A4 17 43 CN1CCN(CCc2ccc(F)cc2)C[C@@H](O)C1 ZINC000217755574 CC In-Stock Unstable SLC6A3 22 40 CN1CCN(CCc2ccc(F)cc2)C[C@@H](O)C1 ZINC000217755574 CC In-Stock Unstable MC4R 0 40 CN1CCN(CCc2ccc(F)cc2)C[C@@H](O)C1 ZINC000217755574 CC In-Stock Unstable SIGMAR1 31 48 CN1CCN(CCc2ccc(F)cc2)C[C@@H](O)C1 ZINC000217755574 CC In-Stock Unstable BIRC2 30 40 Cc1cc(OC2CN(C(=O)c3ccccc3C(F)(F)F)C2)cc(=O)n1C ZINC000217755601 FF In-Stock Unstable RBP4 44 32 O=C1C[C@@H](C(F)(F)F)N(C(=O)Cn2cnc3sc4c(c3c2=O)CCCCC4)c2ccccc2N1 ZINC000217755624 JI On-Demand Unstable HTR1B 18 40 C[C@@H](O)CCNC(=O)/C=C\c1cc(Cl)ccc1Cl ZINC000217755654 CF On-Demand Unstable BOTA 29 45 N=C(N)CC(=O)Nc1ccc(F)c(C(F)(F)F)c1 ZINC000217755658 CE In-Stock Unstable SLC1A1 28 46 N=C(N)CC(=O)Nc1ccc(F)c(C(F)(F)F)c1 ZINC000217755658 CE In-Stock Unstable SLC1A3 33 46 N=C(N)CC(=O)Nc1ccc(F)c(C(F)(F)F)c1 ZINC000217755658 CE In-Stock Unstable SLC1A2 44 34 N=C(N)CC(=O)Nc1ccc(F)c(C(F)(F)F)c1 ZINC000217755658 CE In-Stock Unstable BLM 0 47 N=C(N)CC(=O)Nc1ccc(F)c(C(F)(F)F)c1 ZINC000217755658 CE In-Stock Unstable TMPRSS4 0 41 O=C(O)/C=C\c1cnc(NC(=O)c2ccccc2Cl)s1 ZINC000217755672 DG For-Sale Anodyne EPHB3 47 35 O=C(O)/C=C\c1cnc(NC(=O)c2ccccc2Cl)s1 ZINC000217755672 DG For-Sale Anodyne NR2E3 60 34 O=C(O)/C=C\c1cnc(NC(=O)c2ccccc2Cl)s1 ZINC000217755672 DG For-Sale Anodyne SMO 24 45 COc1ccccc1/C=C\C(=O)N1CC(=O)NC(=O)C1 ZINC000217755675 CC For-Sale Unstable ITGAL 35 42 CN/C(C)=C/C(=O)Nc1ccccc1 ZINC000217755688 AD For-Sale Unstable EPHX1 0 47 CN/C(C)=C/C(=O)Nc1ccccc1 ZINC000217755688 AD For-Sale Unstable MMP1 0 44 CN/C(C)=C/C(=O)Nc1ccccc1 ZINC000217755688 AD For-Sale Unstable P95276_MYCTO 0 47 CN/C(C)=C/C(=O)Nc1ccccc1 ZINC000217755688 AD For-Sale Unstable PARP14 41 35 CN/C(C)=C/C(=O)Nc1ccccc1 ZINC000217755688 AD For-Sale Unstable PARP15 0 45 CN/C(C)=C/C(=O)Nc1ccccc1 ZINC000217755688 AD For-Sale Unstable PARP10 0 40 O=C(Cc1ccc(Cl)cc1)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217755690 DG In-Stock Unstable OPRM1 0 44 O=C(Cc1ccc(Cl)cc1)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217755690 DG In-Stock Unstable OPRK1 0 44 O=C(Cc1ccc(Cl)cc1)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217755690 DG In-Stock Unstable KCNQ2 18 43 O=C(Cc1ccc(Cl)cc1)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217755690 DG In-Stock Unstable SIGMAR1 18 55 Cc1ccc(/C=C\C(=O)NCC[C@@H](C)O)s1 ZINC000217755728 BD For-Sale Unstable SCAF_EBVB9 20 41 C[C@@H](NC(=O)CC(=N)N)c1ccc(F)cc1 ZINC000217755753 BD In-Stock Unstable ACACA 41 38 C[C@@H](NC(=O)CC(=N)N)c1ccc(F)cc1 ZINC000217755753 BD In-Stock Unstable F7 30 40 O=C1CN(C(=O)/C=C\c2ccc(Cl)cc2Cl)CC(=O)N1 ZINC000217755756 DD For-Sale Unstable BOTA 25 50 N#Cc1cc(Br)ccc1CCC(=O)O ZINC000217755805 CE For-Sale Unstable FFAR1 45 43 N#Cc1cc(Br)ccc1CCC(=O)O ZINC000217755805 CE For-Sale Unstable FFAR4 39 40 Cc1ccc(/C=C\C(=O)NCC[C@H](C)O)s1 ZINC000217755814 BD For-Sale Unstable SCAF_EBVB9 20 41 C[C@H](NC(=O)CC(=N)N)c1ccc(F)cc1 ZINC000217755838 BD In-Stock Unstable ACACA 41 38 C[C@H](NC(=O)CC(=N)N)c1ccc(F)cc1 ZINC000217755838 BD In-Stock Unstable F7 30 40 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2sccc2Cl)CC1 ZINC000217755884 FI On-Demand Unstable SLC18A3 41 60 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2sccc2Cl)CC1 ZINC000217755884 FI On-Demand Unstable WNT3A 48 35 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2sccc2Cl)CC1 ZINC000217755884 FI On-Demand Unstable L3MBTL3 73 37 O=C(N/C=C/c1ccccc1F)N1CCOCC1 ZINC000217755909 CD For-Sale Unstable KCNQ2 17 40 C[C@H](C(=O)O)c1ccc(C#N)cc1Br ZINC000217755927 CF For-Sale Unstable PTGS1 19 46 C[C@H](C(=O)O)c1ccc(C#N)cc1Br ZINC000217755927 CF For-Sale Unstable PTGS2 15 46 CN[C@@H]1CC[C@H](C(C)(C)C)C[C@@H]1CCCc1ccccc1 ZINC000217755959 CK For-Sale Unstable SLC18A2 34 41 Cc1ccc2cccc(C(=O)NC[C@@H]3CCCN3c3nccs3)c2n1 ZINC000217755981 FG For-Sale Unstable HCRTR1 37 47 Cc1ccc2cccc(C(=O)NC[C@@H]3CCCN3c3nccs3)c2n1 ZINC000217755981 FG For-Sale Unstable HCRTR2 32 47 C[C@@]12CC=C3NC(=O)CC[C@@H]3[C@@H]1CCC2=O ZINC000217755986 BD Annotated Unstable CYP19A1 41 46 C[C@@H](C(=O)O)c1ccc(C#N)cc1Br ZINC000217755988 CF For-Sale Unstable PTGS1 19 46 C[C@@H](C(=O)O)c1ccc(C#N)cc1Br ZINC000217755988 CF For-Sale Unstable PTGS2 15 46 COC1CCN(C2CCN(C(=O)c3cnc4ccccc4n3)CC2)CC1 ZINC000217756015 FE In-Stock Unstable CHRM2 49 37 COC1CCN(C2CCN(C(=O)c3cnc4ccccc4n3)CC2)CC1 ZINC000217756015 FE In-Stock Unstable HRH1 17 42 COC1CCN(C2CCN(C(=O)c3cnc4ccccc4n3)CC2)CC1 ZINC000217756015 FE In-Stock Unstable HTR3A 15 58 COC1CCN(C2CCN(C(=O)c3cnc4ccccc4n3)CC2)CC1 ZINC000217756015 FE In-Stock Unstable HRH3 16 44 COC1CCN(C2CCN(C(=O)c3cnc4ccccc4n3)CC2)CC1 ZINC000217756015 FE In-Stock Unstable CCR3 42 42 COC1CCN(C2CCN(C(=O)c3cnc4ccccc4n3)CC2)CC1 ZINC000217756015 FE In-Stock Unstable L3MBTL3 87 45 CN[C@H]1CC[C@H](C(C)(C)C)C[C@@H]1CCCc1ccccc1 ZINC000217756051 CK For-Sale Unstable SLC18A2 34 41 Cc1ccc2cccc(C(=O)NC[C@H]3CCCN3c3nccs3)c2n1 ZINC000217756065 FG For-Sale Unstable HCRTR1 37 47 Cc1ccc2cccc(C(=O)NC[C@H]3CCCN3c3nccs3)c2n1 ZINC000217756065 FG For-Sale Unstable HCRTR2 32 47 N#Cc1ccc(CCC(=O)O)c(Br)c1 ZINC000217756106 CE For-Sale Unstable FFAR1 55 52 N#Cc1ccc(CCC(=O)O)c(Br)c1 ZINC000217756106 CE For-Sale Unstable FFAR4 42 43 CN[C@@H]1CC[C@@H](C(C)(C)C)C[C@@H]1CCCc1ccccc1 ZINC000217756114 CK For-Sale Unstable SLC18A2 34 41 COc1c2ccc(C(=O)N3CC(Oc4cc(C)n(C)c(=O)c4)C3)cc2nn1C ZINC000217756164 GD In-Stock Unstable HPGD 41 38 CN[C@H]1CC[C@@H](C(C)(C)C)C[C@@H]1CCCc1ccccc1 ZINC000217756195 CK For-Sale Unstable SLC18A2 34 41 O=C1CN(C(=O)/C=C\c2ccc3c(c2)CCO3)CC(=O)N1 ZINC000217756240 CC For-Sale Unstable ITGAL 17 40 O=C1CN(C(=O)/C=C\c2ccc3c(c2)CCO3)CC(=O)N1 ZINC000217756240 CC For-Sale Unstable GPR183 0 53 C[C@@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756241 CD For-Sale Unstable KCNQ2 50 38 C[C@@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756241 CD For-Sale Unstable ADAM12 24 43 Cn1c(=O)n(CCC(=O)Nc2cccc(Oc3ccccc3)c2)c2ccccc21 ZINC000217756322 GI On-Demand Unstable LTA4H 37 41 Cn1c(=O)n(CCC(=O)Nc2cccc(Oc3ccccc3)c2)c2ccccc21 ZINC000217756322 GI On-Demand Unstable ADORA2B 26 40 Cn1c(=O)n(CCC(=O)Nc2cccc(Oc3ccccc3)c2)c2ccccc21 ZINC000217756322 GI On-Demand Unstable CMA1 15 41 Cn1c(=O)n(CCC(=O)Nc2cccc(Oc3ccccc3)c2)c2ccccc21 ZINC000217756322 GI On-Demand Unstable NPY2R 0 41 Cn1c(=O)n(CCC(=O)Nc2cccc(Oc3ccccc3)c2)c2ccccc21 ZINC000217756322 GI On-Demand Unstable EPHX2 15 42 Cn1c(=O)n(CCC(=O)Nc2cccc(Oc3ccccc3)c2)c2ccccc21 ZINC000217756322 GI On-Demand Unstable CALCRL 39 43 Cn1c(=O)n(CCC(=O)Nc2cccc(Oc3ccccc3)c2)c2ccccc21 ZINC000217756322 GI On-Demand Unstable MCHR1 20 41 Cn1c(=O)n(CCC(=O)Nc2cccc(Oc3ccccc3)c2)c2ccccc21 ZINC000217756322 GI On-Demand Unstable TAAR1 40 42 Cn1c(=O)n(CCC(=O)Nc2cccc(Oc3ccccc3)c2)c2ccccc21 ZINC000217756322 GI On-Demand Unstable KCNK3 93 42 Cn1c(=O)n(CCC(=O)Nc2cccc(Oc3ccccc3)c2)c2ccccc21 ZINC000217756322 GI On-Demand Unstable KCNK9 63 36 Cn1c(=O)n(CCC(=O)Nc2cccc(Oc3ccccc3)c2)c2ccccc21 ZINC000217756322 GI On-Demand Unstable BRPF1 0 44 C[C@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756333 CD For-Sale Unstable KCNQ2 50 38 C[C@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756333 CD For-Sale Unstable ADAM12 24 43 C[C@H]1CN(C)[C@@H](C)C[C@@H]1N[C@@H]1C[C@@H]1c1ccccc1 ZINC000217756371 CF For-Sale Unstable KDM1A 25 42 Cc1cc(OC2CN(C(=O)c3cc4ccccc4[nH]3)C2)cc(=O)n1C ZINC000217756373 EE In-Stock Unstable GRIN2B 29 48 Cc1cc(OC2CN(C(=O)c3cc4ccccc4[nH]3)C2)cc(=O)n1C ZINC000217756373 EE In-Stock Unstable HRH4 36 55 Cc1cc(OC2CN(C(=O)c3cc4ccccc4[nH]3)C2)cc(=O)n1C ZINC000217756373 EE In-Stock Unstable GLRA1 33 45 Cc1cc(OC2CN(C(=O)c3cc4ccccc4[nH]3)C2)cc(=O)n1C ZINC000217756373 EE In-Stock Unstable AKR1C3 21 52 Cc1cc(NC(=O)CC(C)C)ccc1/C=C\C(=O)O ZINC000217756426 CG For-Sale Unstable SLC1A1 50 39 Cc1cc(NC(=O)CC(C)C)ccc1/C=C\C(=O)O ZINC000217756426 CG For-Sale Unstable SLC1A3 52 39 Cc1cc(NC(=O)CC(C)C)ccc1/C=C\C(=O)O ZINC000217756426 CG For-Sale Unstable SLC1A2 76 40 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](CC(C)C)C(=O)N3CCCC3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217756427 KI In-Stock Unstable TUBA1A 18 68 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](CC(C)C)C(=O)N3CCCC3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217756427 KI In-Stock Unstable TPPP 0 64 COc1nc(N)nc2cccc(Br)c12 ZINC000217756428 CD For-Sale Unstable DHFR 20 45 COc1nc(N)nc2cccc(Br)c12 ZINC000217756428 CD For-Sale Unstable DFR1 39 43 O=C(O)CCCCCNC(=O)N/C=C/c1ccccc1F ZINC000217756444 CF For-Sale Unstable HDAC2 16 40 O=C(O)CCCCCNC(=O)N/C=C/c1ccccc1F ZINC000217756444 CF For-Sale Unstable HDAC3 15 45 O=C(O)CCCCCNC(=O)N/C=C/c1ccccc1F ZINC000217756444 CF For-Sale Unstable EPHX2 0 40 O=C(O)CCCCCNC(=O)N/C=C/c1ccccc1F ZINC000217756444 CF For-Sale Unstable HDAC9 34 40 O=C(O)CCCCCNC(=O)N/C=C/c1ccccc1F ZINC000217756444 CF For-Sale Unstable HDAC7 31 40 Cc1cc(NC(=O)C2CCCCC2)ccc1/C=C\C(=O)O ZINC000217756511 CH For-Sale Unstable KCNK3 19 50 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cc3cc5c(cc3[nH]c2=O)OCO5)CC(=O)O4)cc1O ZINC000217756533 KH In-Stock Unstable CYP1A1 27 41 COc1nc(N)nc2ccc(Br)cc12 ZINC000217756536 CD For-Sale Unstable DFRA17 0 40 CC(C)[C@@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756557 CE For-Sale Unstable KCNQ2 48 37 CC(C)[C@@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756557 CE For-Sale Unstable ADAM12 18 55 Cn1c(=O)n(CCC(=O)Nc2ccccc2-c2nc3ccccc3[nH]2)c2ccccc21 ZINC000217756582 HH On-Demand Unstable SHH 20 41 Cn1c(=O)n(CCC(=O)Nc2ccccc2-c2nc3ccccc3[nH]2)c2ccccc21 ZINC000217756582 HH On-Demand Unstable STK33 58 44 Cc1cc(/C=C\C(=O)O)ccc1NC(=O)c1ccccc1 ZINC000217756583 CG For-Sale Unstable EPHX1 0 43 Cc1cc(/C=C\C(=O)O)ccc1NC(=O)c1ccccc1 ZINC000217756583 CG For-Sale Unstable HDAC8 15 41 Cc1cc(/C=C\C(=O)O)ccc1NC(=O)c1ccccc1 ZINC000217756583 CG For-Sale Unstable MMP2 0 47 Cc1cc(/C=C\C(=O)O)ccc1NC(=O)c1ccccc1 ZINC000217756583 CG For-Sale Unstable HDAC1 20 41 Cc1cc(/C=C\C(=O)O)ccc1NC(=O)c1ccccc1 ZINC000217756583 CG For-Sale Unstable HDAC2 16 42 Cc1cc(/C=C\C(=O)O)ccc1NC(=O)c1ccccc1 ZINC000217756583 CG For-Sale Unstable MMP9 0 47 Cc1cc(/C=C\C(=O)O)ccc1NC(=O)c1ccccc1 ZINC000217756583 CG For-Sale Unstable TTR 0 40 Cc1cc(/C=C\C(=O)O)ccc1NC(=O)c1ccccc1 ZINC000217756583 CG For-Sale Unstable MMP1 0 47 Cc1cc(/C=C\C(=O)O)ccc1NC(=O)c1ccccc1 ZINC000217756583 CG For-Sale Unstable KCNK3 94 43 Cc1cc(/C=C\C(=O)O)ccc1NC(=O)c1ccccc1 ZINC000217756583 CG For-Sale Unstable KCNK9 48 43 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cc3cc5c(cc3[nH]c2=O)OCO5)CC(=O)O4)cc1O ZINC000217756620 KH In-Stock Unstable CYP1A1 27 41 CC(C)[C@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756647 CE For-Sale Unstable KCNQ2 48 37 CC(C)[C@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756647 CE For-Sale Unstable ADAM12 18 55 COc1nc(N)nc2cc(Br)ccc12 ZINC000217756648 CD For-Sale Unstable DHFR 22 40 COc1nc(N)nc2cc(Br)ccc12 ZINC000217756648 CD For-Sale Unstable FOLA 48 40 Cc1cc(OC2CN(C(=O)c3c[nH]c4ccccc34)C2)cc(=O)n1C ZINC000217756685 EE In-Stock Unstable AVPR1A 21 40 COc1ccc2[nH]c3c(c2c1)CCC[C@@H]3NC(C)=O ZINC000217756723 CF In-Stock Unstable MTR1B_CHICK 0 46 COc1ccc2[nH]c3c(c2c1)CCC[C@@H]3NC(C)=O ZINC000217756723 CF In-Stock Unstable MAPKAPK2 29 54 COc1ccc2[nH]c3c(c2c1)CCC[C@@H]3NC(C)=O ZINC000217756723 CF In-Stock Unstable MTNR1A 56 42 COc1ccc2[nH]c3c(c2c1)CCC[C@@H]3NC(C)=O ZINC000217756723 CF In-Stock Unstable MTNR1B 49 42 COc1ccc2[nH]c3c(c2c1)CCC[C@@H]3NC(C)=O ZINC000217756723 CF In-Stock Unstable TUBB2B 41 35 COc1ccc2[nH]c3c(c2c1)CCC[C@@H]3NC(C)=O ZINC000217756723 CF In-Stock Unstable SIRT1 15 42 C[C@@H](N[C@H]1C[C@@H]1c1ccccc1)[C@@H]1C[C@H]2C=C[C@H]1C2 ZINC000217756732 CH For-Sale Unstable KDM1A 24 42 O=C(O)/C=C\c1ccccc1N1CC(=O)NC(=O)C1 ZINC000217756765 CC For-Sale Unstable PTGER2 36 48 O=C(O)/C=C\c1ccccc1N1CC(=O)NC(=O)C1 ZINC000217756765 CC For-Sale Unstable PTGER4 0 48 COc1ccccc1-c1cc(C(=O)N2CC(Oc3cc(C)n(C)c(=O)c3)C2)[nH]n1 ZINC000217756772 GD In-Stock Unstable TACR3 24 44 COc1ccc2[nH]c3c(c2c1)CCC[C@H]3NC(C)=O ZINC000217756787 CF In-Stock Unstable MTR1B_CHICK 0 46 COc1ccc2[nH]c3c(c2c1)CCC[C@H]3NC(C)=O ZINC000217756787 CF In-Stock Unstable MAPKAPK2 29 54 COc1ccc2[nH]c3c(c2c1)CCC[C@H]3NC(C)=O ZINC000217756787 CF In-Stock Unstable MTNR1A 56 42 COc1ccc2[nH]c3c(c2c1)CCC[C@H]3NC(C)=O ZINC000217756787 CF In-Stock Unstable MTNR1B 49 42 COc1ccc2[nH]c3c(c2c1)CCC[C@H]3NC(C)=O ZINC000217756787 CF In-Stock Unstable TUBB2B 41 35 COc1ccc2[nH]c3c(c2c1)CCC[C@H]3NC(C)=O ZINC000217756787 CF In-Stock Unstable SIRT1 15 42 C[C@H](N[C@H]1C[C@@H]1c1ccccc1)[C@@H]1C[C@H]2C=C[C@H]1C2 ZINC000217756815 CH For-Sale Unstable KDM1A 24 42 Nc1cc(Nc2ccc(Oc3ccccc3)cc2)nc(-c2ccccc2F)n1 ZINC000217756816 FK In-Stock Unstable SCN5A 28 44 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756864 CF For-Sale Unstable ACE 15 42 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756864 CF For-Sale Unstable FOLH1 23 44 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756864 CF For-Sale Unstable MME 40 46 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756864 CF For-Sale Unstable ANPEP 42 49 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756864 CF For-Sale Unstable RNPEP 24 42 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756864 CF For-Sale Unstable NAALAD2 39 42 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756864 CF For-Sale Unstable CAPNS1 51 34 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756864 CF For-Sale Unstable ECE1 17 42 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756864 CF For-Sale Unstable CAPN1 56 42 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756864 CF For-Sale Unstable CAPN2 48 34 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756864 CF For-Sale Unstable FPR1 83 44 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756864 CF For-Sale Unstable NPR 63 36 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756864 CF For-Sale Unstable AMP1_PLAFQ 17 42 C[C@@H]1C[C@@H]1C(=O)NCc1cc(/C=C\C(=O)O)ccc1F ZINC000217756866 CE For-Sale Unstable AKR1C3 27 40 COc1ccc2c(ccn2CCNC(=O)Cn2ccc3c(NC(C)=O)cccc32)c1 ZINC000217756895 HG In-Stock Unstable DRD4 40 30 COc1ccc2c(ccn2CCNC(=O)Cn2ccc3c(NC(C)=O)cccc32)c1 ZINC000217756895 HG In-Stock Unstable NQO2 24 41 COc1ccc2c(ccn2CCNC(=O)Cn2ccc3c(NC(C)=O)cccc32)c1 ZINC000217756895 HG In-Stock Unstable MTNR1A 97 42 COc1ccc2c(ccn2CCNC(=O)Cn2ccc3c(NC(C)=O)cccc32)c1 ZINC000217756895 HG In-Stock Unstable MTNR1B 86 42 C[C@H]1C[C@@H]1C(=O)NCc1cc(/C=C\C(=O)O)ccc1F ZINC000217756953 CE For-Sale Unstable AKR1C3 27 40 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756956 CF For-Sale Unstable ACE 15 42 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756956 CF For-Sale Unstable FOLH1 59 40 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756956 CF For-Sale Unstable MME 40 46 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756956 CF For-Sale Unstable ANPEP 37 49 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756956 CF For-Sale Unstable RNPEP 22 42 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756956 CF For-Sale Unstable NAALAD2 30 42 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756956 CF For-Sale Unstable CAPNS1 51 34 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756956 CF For-Sale Unstable ECE1 17 42 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756956 CF For-Sale Unstable CAPN1 56 42 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756956 CF For-Sale Unstable CAPN2 48 34 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756956 CF For-Sale Unstable FPR1 83 44 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756956 CF For-Sale Unstable NPR 63 36 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217756956 CF For-Sale Unstable AMP1_PLAFQ 17 42 Nc1cc(Nc2ccc(Oc3ccccc3)cc2)nc(-c2ccc(F)cc2)n1 ZINC000217757033 FK In-Stock Unstable SCN9A 0 53 Nc1cc(Nc2ccc(Oc3ccccc3)cc2)nc(-c2ccc(F)cc2)n1 ZINC000217757033 FK In-Stock Unstable SCN5A 30 53 Nc1cc(Nc2ccc(Oc3ccccc3)cc2)nc(-c2ccc(F)cc2)n1 ZINC000217757033 FK In-Stock Unstable SCN4A 41 38 Nc1cc(Nc2ccc(Oc3ccccc3)cc2)nc(-c2ccc(F)cc2)n1 ZINC000217757033 FK In-Stock Unstable ABCG2 0 41 CSCC[C@@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217757059 DE For-Sale Unstable FOLH1 32 44 CSCC[C@@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217757059 DE For-Sale Unstable NAALAD2 44 36 CSCC[C@@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217757059 DE For-Sale Unstable PAM 0 42 CSCC[C@@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217757059 DE For-Sale Unstable FPR1 43 41 CSCC[C@@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217757059 DE For-Sale Unstable SLC15A2 0 41 CSCC[C@@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217757059 DE For-Sale Unstable FPRL2 0 41 CC(C)c1ccc(OCC(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1 ZINC000217757073 GI On-Demand Unstable HRH2 16 41 CC(C)c1ccc(OCC(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1 ZINC000217757073 GI On-Demand Unstable HRH3 15 44 CC(C)c1ccc(OCC(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1 ZINC000217757073 GI On-Demand Unstable CPT1A 45 36 CC(C)c1ccc(OCC(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1 ZINC000217757073 GI On-Demand Unstable SLC18A3 40 47 CC(C)c1ccc(OCC(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1 ZINC000217757073 GI On-Demand Unstable MLNR 21 42 CC(C)c1ccc(OCC(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1 ZINC000217757073 GI On-Demand Unstable WNT3A 54 35 O=C(O)c1ccccc1/C=C/Cl ZINC000217757104 AF For-Sale Anodyne AKR1C2 45 42 Fc1ccc([C@@H](N[C@@H]2C[C@@H]2c2ccccc2)C2CC2)cc1 ZINC000217757127 CI For-Sale Unstable SLC6A3 20 40 Fc1ccc([C@@H](N[C@@H]2C[C@@H]2c2ccccc2)C2CC2)cc1 ZINC000217757127 CI For-Sale Unstable KDM1A 23 42 Cc1ccc(/C=C\C(=O)O)cc1NC(=O)c1ccc(Cl)o1 ZINC000217757137 DH For-Sale Unstable S1PR4 44 44 Cc1ccc(/C=C\C(=O)O)cc1NC(=O)c1ccc(Cl)o1 ZINC000217757137 DH For-Sale Unstable GPR35 54 35 CSCC[C@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217757141 DE For-Sale Unstable FOLH1 32 44 CSCC[C@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217757141 DE For-Sale Unstable NAALAD2 44 36 CSCC[C@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217757141 DE For-Sale Unstable PAM 0 42 CSCC[C@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217757141 DE For-Sale Unstable FPR1 43 41 CSCC[C@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217757141 DE For-Sale Unstable SLC15A2 0 41 CSCC[C@H](NC(=O)N/C=C/c1ccccc1F)C(=O)O ZINC000217757141 DE For-Sale Unstable FPRL2 0 41 NC(=O)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000217757185 AD On-Demand Unstable MDM2 45 33 Fc1ccc([C@@H](N[C@H]2C[C@@H]2c2ccccc2)C2CC2)cc1 ZINC000217757199 CI For-Sale Unstable SLC6A3 20 40 Fc1ccc([C@@H](N[C@H]2C[C@@H]2c2ccccc2)C2CC2)cc1 ZINC000217757199 CI For-Sale Unstable KDM1A 23 42 COc1cc([C@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc2c1OCO2 ZINC000217757203 KH In-Stock Unstable CYP1B1 45 36 COc1cc([C@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc2c1OCO2 ZINC000217757203 KH In-Stock Unstable RORC 0 40 CCOc1ccc(-c2nc(N)cc(Nc3ccc(Oc4ccccc4)cc3)n2)cc1 ZINC000217757228 GK In-Stock Unstable SCN5A 27 42 CCOc1ccc(-c2nc(N)cc(Nc3ccc(Oc4ccccc4)cc3)n2)cc1 ZINC000217757228 GK In-Stock Unstable AGPAT2 55 44 CCOc1ccc(-c2nc(N)cc(Nc3ccc(Oc4ccccc4)cc3)n2)cc1 ZINC000217757228 GK In-Stock Unstable RPS27 27 43 COc1ccc([C@@H](C)NC(=O)N/C=C/c2ccccc2F)cc1OC ZINC000217757253 EH For-Sale Unstable KCNQ2 59 45 COc1cc([C@@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc2c1OCO2 ZINC000217757283 KH In-Stock Unstable CYP1B1 45 36 COc1cc([C@@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc2c1OCO2 ZINC000217757283 KH In-Stock Unstable RORC 0 40 COc1ccc([C@H](C)NC(=O)N/C=C/c2ccccc2F)cc1OC ZINC000217757334 EH For-Sale Unstable KCNQ2 59 45 Cc1ccc(/C=C\C(=O)N2CC(=O)NC(=O)C2)cc1 ZINC000217757386 CC For-Sale Unstable GPR183 0 52 COC(=O)[C@@H](NC(=O)CC/C(C)=C/Cc1c(OC)c(C)c2c(c1OC)C(=O)OC2)C(C)C ZINC000217757392 IG In-Stock Unstable IMPDH1 0 88 COC(=O)[C@@H](NC(=O)CC/C(C)=C/Cc1c(OC)c(C)c2c(c1OC)C(=O)OC2)C(C)C ZINC000217757392 IG In-Stock Unstable IMPDH2 0 88 COc1ccc([C@@H](C)N2C[C@@H](C)C[C@@H](C)C2)c(O)c1 ZINC000217757404 CG For-Sale Unstable RORC 34 42 COc1ccc(-c2nc(N)cc(Nc3ccc(Oc4ccccc4)cc3)n2)cc1OC ZINC000217757429 HK In-Stock Unstable SCN5A 26 42 COc1ccc(-c2nc(N)cc(Nc3ccc(Oc4ccccc4)cc3)n2)cc1OC ZINC000217757429 HK In-Stock Unstable GALR2 42 38 COc1ccc(-c2nc(N)cc(Nc3ccc(Oc4ccccc4)cc3)n2)cc1OC ZINC000217757429 HK In-Stock Unstable AGPAT2 36 46 COc1ccc(-c2nc(N)cc(Nc3ccc(Oc4ccccc4)cc3)n2)cc1OC ZINC000217757429 HK In-Stock Unstable ABCG2 23 48 COc1ccc([C@@H](C)NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217757440 DH For-Sale Unstable KCNQ2 57 45 COc1ccc([C@@H](C)NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217757440 DH For-Sale Unstable ACACA 19 41 COc1ccc([C@@H](C)NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217757440 DH For-Sale Unstable ACACB 16 41 O=C(c1ccc(F)cc1)C1CCN(C(=O)COc2cccc(Cl)c2)CC1 ZINC000217757490 GH On-Demand Unstable HRH2 18 42 O=C(c1ccc(F)cc1)C1CCN(C(=O)COc2cccc(Cl)c2)CC1 ZINC000217757490 GH On-Demand Unstable HTR2A 17 47 O=C(c1ccc(F)cc1)C1CCN(C(=O)COc2cccc(Cl)c2)CC1 ZINC000217757490 GH On-Demand Unstable HRH1 15 40 O=C(c1ccc(F)cc1)C1CCN(C(=O)COc2cccc(Cl)c2)CC1 ZINC000217757490 GH On-Demand Unstable SIGMAR1 15 43 O=C(c1ccc(F)cc1)C1CCN(C(=O)COc2cccc(Cl)c2)CC1 ZINC000217757490 GH On-Demand Unstable CPT1A 104 43 O=C(c1ccc(F)cc1)C1CCN(C(=O)COc2cccc(Cl)c2)CC1 ZINC000217757490 GH On-Demand Unstable CPT2 47 43 O=C(c1ccc(F)cc1)C1CCN(C(=O)COc2cccc(Cl)c2)CC1 ZINC000217757490 GH On-Demand Unstable SLC18A3 43 43 O=C(c1ccc(F)cc1)C1CCN(C(=O)COc2cccc(Cl)c2)CC1 ZINC000217757490 GH On-Demand Unstable MLNR 24 43 O=C(c1ccc(F)cc1)C1CCN(C(=O)COc2cccc(Cl)c2)CC1 ZINC000217757490 GH On-Demand Unstable WNT3A 47 33 COc1ccc([C@H](C)NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217757508 DH For-Sale Unstable KCNQ2 57 45 COc1ccc([C@H](C)NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217757508 DH For-Sale Unstable ACACA 19 41 COc1ccc([C@H](C)NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217757508 DH For-Sale Unstable ACACB 16 41 Cc1cc(OC2CN(S(=O)(=O)c3ccc4c(c3)OCCO4)C2)cc(=O)n1C ZINC000217757530 GC In-Stock Unstable PKM 44 49 N[C@H](CN[C@@H]1C[C@@H]1c1ccccc1)c1ccccc1 ZINC000217757541 CF For-Sale Unstable KDM1A 39 41 COc1ccc(/C=C\C(=O)N2CC(=O)NC(=O)C2)cc1 ZINC000217757549 CC For-Sale Unstable PTGS2 0 47 COc1ccc(/C=C\C(=O)N2CC(=O)NC(=O)C2)cc1 ZINC000217757549 CC For-Sale Unstable GPR183 0 60 CCOc1ccc(C)cc1[C@@H](C)NC(=O)N/C=C/c1ccccc1F ZINC000217757615 EJ For-Sale Unstable KCNQ2 40 36 N[C@H](CN[C@H]1C[C@@H]1c1ccccc1)c1ccccc1 ZINC000217757629 CF For-Sale Unstable KDM1A 39 41 O=C(O)/C=C\c1cccc(NC(=O)c2ccccn2)n1 ZINC000217757641 CD For-Sale Anodyne GRM4 62 44 O=C(O)/C=C\c1cccc(NC(=O)c2ccccn2)n1 ZINC000217757641 CD For-Sale Anodyne GRM5 16 45 CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(-c3cccc(CN(C)C)c3)c(Oc3ccccc3C(F)(F)F)s2)cc1 ZINC000217757676 KK Annotated Unstable RORC 73 51 O=C(O)/C=C\c1cccc(NC(=O)c2ccncc2)n1 ZINC000217757724 CD For-Sale Anodyne KCNK3 61 48 CCOc1ccc(C)cc1[C@H](C)NC(=O)N/C=C/c1ccccc1F ZINC000217757726 EJ For-Sale Unstable KCNQ2 40 36 O=C(N[C@@H]1C[C@@H]2C[C@@H]1[C@@H]1CCC[C@@H]21)c1ccc(CCl)cc1 ZINC000217757776 DH For-Sale Unstable SSTR3 30 42 O=C(O)/C=C\c1cccc(NC(=O)c2ccc(F)cc2)n1 ZINC000217757811 CF For-Sale Anodyne HTR1F 37 40 O=C(O)/C=C\c1cccc(NC(=O)c2ccc(F)cc2)n1 ZINC000217757811 CF For-Sale Anodyne GRM5 18 42 O=C(O)/C=C\c1cccc(NC(=O)c2ccc(F)cc2)n1 ZINC000217757811 CF For-Sale Anodyne MAP3K5 41 40 O=C(O)/C=C\c1cccc(NC(=O)c2ccc(F)cc2)n1 ZINC000217757811 CF For-Sale Anodyne KCNK3 35 46 c1ccc([C@H]2C[C@H]2NC[C@@H]2NCCc3ccccc32)cc1 ZINC000217757839 CG For-Sale Unstable PRCP 63 52 O=C(N[C@H]1C[C@@H]2C[C@@H]1[C@@H]1CCC[C@@H]21)c1ccc(CCl)cc1 ZINC000217757857 DH For-Sale Unstable SSTR3 30 42 CS(=O)(=O)N(CC(=N)N)Cc1ccc(Cl)cc1 ZINC000217757878 CD In-Stock Unstable CXCR3 15 40 CS(=O)(=O)N(CC(=N)N)Cc1ccc(Cl)cc1 ZINC000217757878 CD In-Stock Unstable DAGLA 15 41 COc1ccc(Cl)cc1S(=O)(=O)N1CC(Oc2cc(C)n(C)c(=O)c2)C1 ZINC000217757891 GD In-Stock Unstable COLA 60 36 COc1ccc(Cl)cc1S(=O)(=O)N1CC(Oc2cc(C)n(C)c(=O)c2)C1 ZINC000217757891 GD In-Stock Unstable CPT1A 57 36 COc1ccc(Cl)cc1S(=O)(=O)N1CC(Oc2cc(C)n(C)c(=O)c2)C1 ZINC000217757891 GD In-Stock Unstable CPT2 44 36 COc1ccc(Cl)cc1S(=O)(=O)N1CC(Oc2cc(C)n(C)c(=O)c2)C1 ZINC000217757891 GD In-Stock Unstable CPT1B 51 36 c1ccc([C@H]2C[C@@H]2NC[C@@H]2NCCc3ccccc32)cc1 ZINC000217757916 CG For-Sale Unstable PRCP 63 52 O=C(N[C@@H]1C[C@H]2C[C@@H]1[C@@H]1CCC[C@@H]21)c1ccc(CCl)cc1 ZINC000217757934 DH For-Sale Unstable SSTR3 30 42 COc1ccc(/C=C\C(=O)O)cc1NC(=O)C(C)(C)C ZINC000217757944 CF For-Sale Unstable MMP2 0 47 COc1ccc(/C=C\C(=O)O)cc1NC(=O)C(C)(C)C ZINC000217757944 CF For-Sale Unstable TUBB1 55 41 COc1ccc(/C=C\C(=O)O)cc1NC(=O)C(C)(C)C ZINC000217757944 CF For-Sale Unstable MMP1 0 43 COc1ccc(/C=C\C(=O)O)cc1NC(=O)C(C)(C)C ZINC000217757944 CF For-Sale Unstable ABCG2 17 43 NC(=O)c1ccc(/C=C\C(=O)N2CC(=O)NC(=O)C2)cc1 ZINC000217757948 CB For-Sale Unstable GPR183 0 43 c1ccc([C@@H]2C[C@H]2NC[C@@H]2NCCc3ccccc32)cc1 ZINC000217758003 CG For-Sale Unstable PRCP 63 52 O=C1CN(C(=O)/C=C\c2ccc(Cl)cc2)CC(=O)N1 ZINC000217758023 CC For-Sale Unstable GPR183 0 43 O=C(N[C@H]1C[C@H]2C[C@@H]1[C@@H]1CCC[C@@H]21)c1ccc(CCl)cc1 ZINC000217758035 DH For-Sale Unstable SSTR3 30 42 O=C(O)/C=C\c1cnc(NC(=O)COc2ccccc2)s1 ZINC000217758038 DE For-Sale Unstable CDK5 41 41 O=C(O)/C=C\c1cnc(NC(=O)COc2ccccc2)s1 ZINC000217758038 DE For-Sale Unstable ISPD 0 42 CCc1ccc([C@@H](C)NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217758060 DI For-Sale Unstable KCNQ2 56 41 c1ccc([C@@H]2C[C@@H]2NC[C@@H]2NCCc3ccccc32)cc1 ZINC000217758078 CG For-Sale Unstable PRCP 63 52 O=C1N[C@@H](CCC(=O)N2CCc3c([nH]c4ccccc34)C2)C(=O)Nc2ccccc21 ZINC000217758093 HF In-Stock Unstable DRD5 19 41 O=C1N[C@@H](CCC(=O)N2CCc3c([nH]c4ccccc34)C2)C(=O)Nc2ccccc21 ZINC000217758093 HF In-Stock Unstable SSTR4 46 32 CCN(CC(=N)N)S(=O)(=O)c1ccc(Cl)cc1 ZINC000217758099 CD In-Stock Unstable CXCR3 17 42 CCN(CC(=N)N)S(=O)(=O)c1ccc(Cl)cc1 ZINC000217758099 CD In-Stock Unstable DAGLA 16 43 CN1CCO[C@@H](CNS(=O)(=O)N2CCC[C@@H](C(=O)O)C2)C1 ZINC000217758101 DA For-Sale Unstable SLC6A1 55 32 C[C@H](O)CCNC(=O)/C=C\c1cccc([N+](=O)[O-])c1 ZINC000217758106 CD For-Sale Unstable CACNA1D 53 35 C[C@H](O)CCNC(=O)/C=C\c1cccc([N+](=O)[O-])c1 ZINC000217758106 CD For-Sale Unstable TRPM8 0 58 CCc1ccc([C@H](C)NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217758137 DI For-Sale Unstable KCNQ2 56 41 CN1CCO[C@H](CNS(=O)(=O)N2CCC[C@@H](C(=O)O)C2)C1 ZINC000217758187 DA For-Sale Unstable SLC6A1 55 32 C[C@@H](O)CCNC(=O)/C=C\c1cccc([N+](=O)[O-])c1 ZINC000217758188 CD On-Demand Unstable CACNA1D 41 33 C[C@@H](O)CCNC(=O)/C=C\c1cccc([N+](=O)[O-])c1 ZINC000217758188 CD On-Demand Unstable TRPM8 0 58 CCCCC(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217758217 CF For-Sale Unstable PTGER2 22 40 CCCCC(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217758217 CF For-Sale Unstable AKR1C3 43 49 CN(C)S(=O)(=O)c1ccc(CCC(=N)N)cc1 ZINC000217758218 CC In-Stock Unstable CA2 26 42 CN(C)S(=O)(=O)c1ccc(CCC(=N)N)cc1 ZINC000217758218 CC In-Stock Unstable CA1 24 42 CN(C)S(=O)(=O)c1ccc(CCC(=N)N)cc1 ZINC000217758218 CC In-Stock Unstable CA7 17 41 CN(C)S(=O)(=O)c1ccc(CCC(=N)N)cc1 ZINC000217758218 CC In-Stock Unstable CA4 20 41 CN(C)S(=O)(=O)c1ccc(CCC(=N)N)cc1 ZINC000217758218 CC In-Stock Unstable AOC3 22 43 CN(C)S(=O)(=O)c1ccc(CCC(=N)N)cc1 ZINC000217758218 CC In-Stock Unstable NCE103 15 45 CN(C)S(=O)(=O)c1ccc(CCC(=N)N)cc1 ZINC000217758218 CC In-Stock Unstable CA 0 45 C[C@@H](N[C@@H]1CCN2CCC[C@@H]12)c1ccccc1O ZINC000217758222 BE For-Sale Unstable SLC18A3 55 37 C[C@@H](NC(=O)N/C=C/c1ccccc1F)c1ccc2c(c1)CCCC2 ZINC000217758242 EJ For-Sale Unstable KCNQ2 58 42 CN(Cc1cccc(/C=C\C(=O)O)c1)C(=O)c1ccco1 ZINC000217758294 CF For-Sale Unstable NR1H4 25 47 CN(Cc1cccc(/C=C\C(=O)O)c1)C(=O)c1ccco1 ZINC000217758294 CF For-Sale Unstable HSD17B2 26 42 C[C@H](N[C@@H]1CCN2CCC[C@@H]12)c1ccccc1O ZINC000217758297 BE For-Sale Unstable SLC18A3 55 37 COc1ccc(-c2ccc(S(=O)(=O)N3CC(Oc4cc(C)n(C)c(=O)c4)C3)cc2)cc1 ZINC000217758310 IF In-Stock Unstable MMP7 41 39 Cn1cccc1C(=O)N1CCC[C@@H]1c1ccccn1 ZINC000217758319 CE In-Stock Unstable COLA 65 37 Cn1cccc1C(=O)N1CCC[C@@H]1c1ccccn1 ZINC000217758319 CE In-Stock Unstable CPT1A 60 37 COc1cc(C(=O)NC[C@@H]2CCCN2c2nccs2)cc(OC)c1OC ZINC000217758325 GF For-Sale Unstable DRD2 42 46 COc1cc(C(=O)NC[C@@H]2CCCN2c2nccs2)cc(OC)c1OC ZINC000217758325 GF For-Sale Unstable CACNA1I 46 32 COc1cc(C(=O)NC[C@@H]2CCCN2c2nccs2)cc(OC)c1OC ZINC000217758325 GF For-Sale Unstable ACKR3 71 39 C[C@H](NC(=O)N/C=C/c1ccccc1F)c1ccc2c(c1)CCCC2 ZINC000217758328 EJ For-Sale Unstable KCNQ2 58 42 Cc1cc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)oc1C ZINC000217758371 EH On-Demand Unstable HSD11B1 15 64 Cc1cc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)oc1C ZINC000217758371 EH On-Demand Unstable SLC18A3 43 48 Cc1cc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)oc1C ZINC000217758371 EH On-Demand Unstable WNT3A 47 34 Cc1cc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)oc1C ZINC000217758371 EH On-Demand Unstable L3MBTL3 76 38 C[C@@H](N[C@H]1CCN2CCC[C@@H]12)c1ccccc1O ZINC000217758380 BE For-Sale Unstable SLC18A3 55 37 COc1cc(C(=O)NC[C@H]2CCCN2c2nccs2)cc(OC)c1OC ZINC000217758395 GF For-Sale Unstable DRD2 42 46 COc1cc(C(=O)NC[C@H]2CCCN2c2nccs2)cc(OC)c1OC ZINC000217758395 GF For-Sale Unstable CACNA1I 46 32 COc1cc(C(=O)NC[C@H]2CCCN2c2nccs2)cc(OC)c1OC ZINC000217758395 GF For-Sale Unstable ACKR3 71 39 N[C@H](CCN[C@@H]1C[C@@H]1c1ccccc1)c1ccccc1 ZINC000217758398 CG For-Sale Unstable KDM1A 27 46 Cn1cccc1C(=O)N1CCC[C@H]1c1ccccn1 ZINC000217758400 CE In-Stock Unstable COLA 65 37 Cn1cccc1C(=O)N1CCC[C@H]1c1ccccn1 ZINC000217758400 CE In-Stock Unstable CPT1A 60 37 C[C@]12C[C@@H]3C[C@H](C1)C[C@@](CNC(=O)c1ccc(F)cc1)(C3)C2 ZINC000217758433 DI In-Stock Unstable P2RX7 26 56 C[C@H](N[C@H]1CCN2CCC[C@@H]12)c1ccccc1O ZINC000217758468 BE For-Sale Unstable SLC18A3 55 37 CC(C)(C)c1ccc(OCC(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1 ZINC000217758472 GJ On-Demand Unstable HRH2 15 44 CC(C)(C)c1ccc(OCC(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1 ZINC000217758472 GJ On-Demand Unstable HRH3 15 44 CC(C)(C)c1ccc(OCC(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1 ZINC000217758472 GJ On-Demand Unstable CPT1A 54 36 CC(C)(C)c1ccc(OCC(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1 ZINC000217758472 GJ On-Demand Unstable SLC18A3 41 48 CC(C)(C)c1ccc(OCC(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1 ZINC000217758472 GJ On-Demand Unstable MLNR 21 42 CC(C)(C)c1ccc(OCC(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1 ZINC000217758472 GJ On-Demand Unstable WNT3A 54 34 N[C@H](CCN[C@H]1C[C@@H]1c1ccccc1)c1ccccc1 ZINC000217758488 CG For-Sale Unstable KDM1A 27 46 O=C(O)/C=C\c1cccc(NC(=O)Cc2cccs2)c1 ZINC000217758518 CG For-Sale Unstable CA5B 39 48 O=C(O)/C=C\c1cccc(NC(=O)Cc2cccs2)c1 ZINC000217758518 CG For-Sale Unstable CA5A 40 48 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable ACE 24 52 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable TYR 15 41 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable GNRHR 0 40 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable OPRM1 0 40 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable OPRD1 0 40 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable MME 33 52 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable EDNRB 54 41 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable EDNRA 38 41 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable TACR1 30 44 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable MC4R 40 38 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable BMP1 27 40 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable TACR2 22 40 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable CCKAR 84 47 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable BRS3 28 46 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable MC3R 62 37 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable MC5R 65 35 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable MMP2 28 45 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable GRPR 73 37 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable ECE1 71 52 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable LNPEP 25 40 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable MMP11 85 35 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable CCKBR 66 45 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable GHSR 70 41 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable MMP9 26 43 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable MC1R 87 38 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable MMP1 20 40 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable NPR 32 48 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable SSSIM 30 45 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable SLC15A2 0 58 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable KISS1R 70 34 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable ERAP2 43 40 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable ERAP1 0 40 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable LASB 0 43 O=C(CCn1c(=O)sc2ccccc21)N[C@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217758521 HF In-Stock Unstable NRDE 0 46 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccccc1Cl ZINC000217758522 DG For-Sale Unstable HCRTR1 33 41 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccccc1Cl ZINC000217758522 DG For-Sale Unstable HCRTR2 29 41 O=C(N/C=C/c1ccccc1F)Nc1ccc(Oc2ccccc2)cc1 ZINC000217758546 EK For-Sale Anodyne CA1 44 47 O=C(N/C=C/c1ccccc1F)Nc1ccc(Oc2ccccc2)cc1 ZINC000217758546 EK For-Sale Anodyne RAF1 28 40 O=C(N/C=C/c1ccccc1F)Nc1ccc(Oc2ccccc2)cc1 ZINC000217758546 EK For-Sale Anodyne NPY5R 21 40 O=C(N/C=C/c1ccccc1F)Nc1ccc(Oc2ccccc2)cc1 ZINC000217758546 EK For-Sale Anodyne CA12 16 47 O=C(N/C=C/c1ccccc1F)Nc1ccc(Oc2ccccc2)cc1 ZINC000217758546 EK For-Sale Anodyne CA9 17 47 O=C(N/C=C/c1ccccc1F)Nc1ccc(Oc2ccccc2)cc1 ZINC000217758546 EK For-Sale Anodyne Q8MMZ8_EIMTE 44 40 O=C(N/C=C/c1ccccc1F)Nc1ccc(Oc2ccccc2)cc1 ZINC000217758546 EK For-Sale Anodyne F13A1 21 40 O=C(CCC(=O)N1CCCCCC1)NCc1nc(-c2ccccc2)n[nH]1 ZINC000217758549 FE In-Stock Unstable COLA 44 37 O=C(NC[C@H]1CCCN1c1nccs1)c1ccccc1Cl ZINC000217758612 DG For-Sale Unstable HCRTR1 33 41 O=C(NC[C@H]1CCCN1c1nccs1)c1ccccc1Cl ZINC000217758612 DG For-Sale Unstable HCRTR2 29 41 COc1ccc(CNc2nnc(Cl)cc2C(=O)NC2CCOCC2)cc1 ZINC000217758688 GF For-Sale Unstable PDE5A 32 42 COc1ccc(CNc2nnc(Cl)cc2C(=O)NC2CCOCC2)cc1 ZINC000217758688 GF For-Sale Unstable CNR2 17 41 COc1ccc(CNc2nnc(Cl)cc2C(=O)NC2CCOCC2)cc1 ZINC000217758688 GF For-Sale Unstable PDK1 49 37 COc1ccc(CNc2nnc(Cl)cc2C(=O)NC2CCOCC2)cc1 ZINC000217758688 GF For-Sale Unstable MCHR1 22 54 COc1ccc(CNc2nnc(Cl)cc2C(=O)NC2CCOCC2)cc1 ZINC000217758688 GF For-Sale Unstable STAT6 45 38 COc1ccc(CNc2nnc(Cl)cc2C(=O)NC2CCOCC2)cc1 ZINC000217758688 GF For-Sale Unstable PROKR1 67 35 c1ccc([C@@H](N[C@@H]2C[C@@H]2c2ccccc2)C2CC2)cc1 ZINC000217758722 CI For-Sale Unstable EPHX2 15 43 c1ccc([C@@H](N[C@@H]2C[C@@H]2c2ccccc2)C2CC2)cc1 ZINC000217758722 CI For-Sale Unstable KDM1A 32 44 Cc1[nH]ncc1C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217758734 CD For-Sale Unstable ROCK1 16 41 Cc1[nH]ncc1C(=O)NCc1cccc(/C=C\C(=O)O)c1 ZINC000217758734 CD For-Sale Unstable ROCK2 20 41 COCCc1nc(CCNC(C)=O)n(Cc2ccc3c(c2)OCO3)n1 ZINC000217758740 EC In-Stock Unstable BMP1 40 34 COCCc1nc(CCNC(C)=O)n(Cc2ccc3c(c2)OCO3)n1 ZINC000217758740 EC In-Stock Unstable NOS2 98 40 COc1ccc(/C=C\C(=O)N2CC(=O)NC(=O)C2)cc1F ZINC000217758750 CC For-Sale Unstable CCR2 61 41 COc1ccc(/C=C\C(=O)N2CC(=O)NC(=O)C2)cc1F ZINC000217758750 CC For-Sale Unstable TUBB1 43 45 COc1ccc(/C=C\C(=O)N2CC(=O)NC(=O)C2)cc1F ZINC000217758750 CC For-Sale Unstable NFE2L2 0 40 COc1ccc(/C=C\C(=O)N2CC(=O)NC(=O)C2)cc1F ZINC000217758750 CC For-Sale Unstable GPR183 0 42 COc1ccc(OC)c(NC(=O)N/C=C/c2ccccc2F)c1 ZINC000217758751 DH For-Sale Unstable CYP1B1 42 40 COc1ccc(OC)c(NC(=O)N/C=C/c2ccccc2F)c1 ZINC000217758751 DH For-Sale Unstable MTNR1A 18 48 COc1ccc(OC)c(NC(=O)N/C=C/c2ccccc2F)c1 ZINC000217758751 DH For-Sale Unstable MTNR1B 19 48 COc1ccc(OC)c(NC(=O)N/C=C/c2ccccc2F)c1 ZINC000217758751 DH For-Sale Unstable AKR1C2 44 32 COc1ccc(C)cc1CN[C@@H]1CCN2CCC[C@@H]12 ZINC000217758772 CE For-Sale Unstable TACR1 35 42 Nc1nnc(Cl)cc1C(=O)NC1CCOCC1 ZINC000217758801 CC For-Sale Unstable TYRO3 15 40 c1ccc([C@@H](N[C@H]2C[C@@H]2c2ccccc2)C2CC2)cc1 ZINC000217758806 CI For-Sale Unstable EPHX2 15 43 c1ccc([C@@H](N[C@H]2C[C@@H]2c2ccccc2)C2CC2)cc1 ZINC000217758806 CI For-Sale Unstable KDM1A 32 44 Cc1cc(OC2CN(S(=O)(=O)C[C@@]34CC[C@@H](CC3=O)C4(C)C)C2)cc(=O)n1C ZINC000217758857 HD In-Stock Unstable CA5B 23 42 Cc1cc(OC2CN(S(=O)(=O)C[C@@]34CC[C@@H](CC3=O)C4(C)C)C2)cc(=O)n1C ZINC000217758857 HD In-Stock Unstable CA5A 26 42 Cc1cc(OC2CN(S(=O)(=O)C[C@@]34CC[C@@H](CC3=O)C4(C)C)C2)cc(=O)n1C ZINC000217758857 HD In-Stock Unstable CXCR3 15 47 COc1ccc(C)cc1CN[C@H]1CCN2CCC[C@@H]12 ZINC000217758863 CE For-Sale Unstable TACR1 35 42 Cc1cc(NC(=O)C2CCCC2)ccc1/C=C\C(=O)O ZINC000217758935 CG For-Sale Unstable KCNK3 19 48 Cc1[nH]ncc1C(=O)Nc1cccc(/C=C\C(=O)O)c1 ZINC000217758972 CE For-Sale Unstable BTK 24 42 Cc1[nH]ncc1C(=O)Nc1cccc(/C=C\C(=O)O)c1 ZINC000217758972 CE For-Sale Unstable KCNK3 115 40 Cc1[nH]ncc1C(=O)Nc1cccc(/C=C\C(=O)O)c1 ZINC000217758972 CE For-Sale Unstable KCNK9 83 40 CC(C)(C)OC(=O)N1C[C@@H](F)C[C@@H]1C(=O)N1CCC1 ZINC000217759035 CD On-Demand Unstable PREP 39 58 CC[C@@H](C)N(C)CCN[C@@H](C)Cc1ccccc1 ZINC000217759087 BF For-Sale Unstable LMGT2 0 40 O=C1C[C@@H](c2ccc(O)cc2)c2c(c3ccccc3oc2=O)O1 ZINC000217759098 DF In-Stock Unstable VKORC1 0 41 O=C1C[C@@H](c2ccc(O)cc2)c2c(c3ccccc3oc2=O)O1 ZINC000217759098 DF In-Stock Unstable NQO1 33 47 O=C(NCc1ccccc1)[C@@]12C[C@@H]3C[C@@H](C[C@@](Cl)(C3)C1)C2 ZINC000217759108 DH In-Stock Unstable P2RX7 0 48 O=C(NCc1ccccc1)[C@@]12C[C@@H]3C[C@@H](C[C@@](Cl)(C3)C1)C2 ZINC000217759108 DH In-Stock Unstable EPHX2 21 46 O=C(NCc1ccccc1)[C@@]12C[C@@H]3C[C@@H](C[C@@](Cl)(C3)C1)C2 ZINC000217759108 DH In-Stock Unstable CCL2 0 40 O=C(COc1ccc(-c2ccccc2)cc1)NC[C@@H]1CCCN1c1nccs1 ZINC000217759119 GH For-Sale Unstable COLA 76 37 O=C(COc1ccc(-c2ccccc2)cc1)NC[C@@H]1CCCN1c1nccs1 ZINC000217759119 GH For-Sale Unstable CPT1A 71 37 Cc1cc(NC(=O)c2cccs2)ccc1/C=C\C(=O)O ZINC000217759133 CG For-Sale Unstable NAMPT 46 34 Cc1cc(NC(=O)c2cccs2)ccc1/C=C\C(=O)O ZINC000217759133 CG For-Sale Unstable KCNK3 81 56 Cc1cc(NC(=O)c2cccs2)ccc1/C=C\C(=O)O ZINC000217759133 CG For-Sale Unstable KCNK9 44 56 NC[C@]1(N2CC[C@@H](c3ccccc3)C2)CCN(C2CC2)C1 ZINC000217759136 CE For-Sale Unstable SLC18A3 37 41 CC[C@H](C)N(C)CCN[C@@H](C)Cc1ccccc1 ZINC000217759173 BF For-Sale Unstable LMGT2 0 40 O=C1C[C@H](c2ccc(O)cc2)c2c(c3ccccc3oc2=O)O1 ZINC000217759177 DF In-Stock Unstable VKORC1 0 41 O=C1C[C@H](c2ccc(O)cc2)c2c(c3ccccc3oc2=O)O1 ZINC000217759177 DF In-Stock Unstable NQO1 33 47 O=C(N/C=C/c1ccccc1F)Nc1ccc(F)cc1 ZINC000217759202 CH For-Sale Anodyne MTCA1 17 41 O=C(COc1ccc(-c2ccccc2)cc1)NC[C@H]1CCCN1c1nccs1 ZINC000217759205 GH For-Sale Unstable COLA 76 37 O=C(COc1ccc(-c2ccccc2)cc1)NC[C@H]1CCCN1c1nccs1 ZINC000217759205 GH For-Sale Unstable CPT1A 71 37 Cc1cc(/C=C\C(=O)O)ccc1NC(=O)c1ccccn1 ZINC000217759210 CF For-Sale Unstable PYGL 0 42 Cc1cc(/C=C\C(=O)O)ccc1NC(=O)c1ccccn1 ZINC000217759210 CF For-Sale Unstable GRM4 70 48 Cc1cc(/C=C\C(=O)O)ccc1NC(=O)c1ccccn1 ZINC000217759210 CF For-Sale Unstable PYGM 23 42 Cc1cc(/C=C\C(=O)O)ccc1NC(=O)c1ccccn1 ZINC000217759210 CF For-Sale Unstable MMP1 0 43 c1ccc(C2CC(N[C@@H]3CCN4CCC[C@@H]34)C2)cc1 ZINC000217759214 CF For-Sale Unstable SLC18A3 85 48 CC[C@@H](C)[C@@H](NC(=O)[C@@H]1COc2ccccc2C1)C(=O)O ZINC000217759277 CD For-Sale Unstable ROCK2 26 44 CC[C@@H](C)[C@@H](NC(=O)[C@@H]1COc2ccccc2C1)C(=O)O ZINC000217759277 CD For-Sale Unstable GZMB 46 35 Cc1cc(/C=C\C(=O)O)ccc1NC(=O)c1ccncc1 ZINC000217759282 CF For-Sale Unstable KCNK3 42 44 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)NC[C@@H]1C[C@H]3C=C[C@@H]1C3)C(=O)OC2 ZINC000217759284 II In-Stock Unstable IMPDH1 0 59 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)NC[C@@H]1C[C@H]3C=C[C@@H]1C3)C(=O)OC2 ZINC000217759284 II In-Stock Unstable IMPDH2 0 59 c1ccc(C2CC(N[C@H]3CCN4CCC[C@@H]34)C2)cc1 ZINC000217759292 CF For-Sale Unstable SLC18A3 85 48 N#Cc1ccc(OCC(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1 ZINC000217759307 FG On-Demand Unstable HRH2 15 42 N#Cc1ccc(OCC(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1 ZINC000217759307 FG On-Demand Unstable HRH3 17 43 N#Cc1ccc(OCC(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1 ZINC000217759307 FG On-Demand Unstable CPT1A 52 50 N#Cc1ccc(OCC(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1 ZINC000217759307 FG On-Demand Unstable SLC18A3 41 46 N#Cc1ccc(OCC(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1 ZINC000217759307 FG On-Demand Unstable MLNR 25 41 N#Cc1ccc(OCC(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1 ZINC000217759307 FG On-Demand Unstable WNT3A 53 35 N#Cc1ccc(OCC(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1 ZINC000217759307 FG On-Demand Unstable MEN1 40 37 NS(=O)(=O)c1ccc(C(=O)NC[C@@H]2CCCN2c2nccs2)cc1 ZINC000217759310 FD For-Sale Unstable CA2 45 51 NS(=O)(=O)c1ccc(C(=O)NC[C@@H]2CCCN2c2nccs2)cc1 ZINC000217759310 FD For-Sale Unstable CA1 26 40 NS(=O)(=O)c1ccc(C(=O)NC[C@@H]2CCCN2c2nccs2)cc1 ZINC000217759310 FD For-Sale Unstable CA7 23 42 NS(=O)(=O)c1ccc(C(=O)NC[C@@H]2CCCN2c2nccs2)cc1 ZINC000217759310 FD For-Sale Unstable CA4 19 42 NS(=O)(=O)c1ccc(C(=O)NC[C@@H]2CCCN2c2nccs2)cc1 ZINC000217759310 FD For-Sale Unstable CA14 31 41 NS(=O)(=O)c1ccc(C(=O)NC[C@@H]2CCCN2c2nccs2)cc1 ZINC000217759310 FD For-Sale Unstable CA12 15 42 NS(=O)(=O)c1ccc(C(=O)NC[C@@H]2CCCN2c2nccs2)cc1 ZINC000217759310 FD For-Sale Unstable CA9 22 42 O=C(N/C=C/c1ccccc1F)Nc1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217759315 EI For-Sale Bother IMDH_CRYPV 29 45 O=C(N/C=C/c1ccccc1F)Nc1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217759315 EI For-Sale Bother BLM 0 46 CN(Cc1cnccn1)C(=O)C1CCN(C(=O)Cc2ccccc2)CC1 ZINC000217759331 FD In-Stock Unstable C3AR1 41 35 CC[C@H](C)[C@@H](NC(=O)[C@@H]1COc2ccccc2C1)C(=O)O ZINC000217759351 CD On-Demand Unstable ROCK2 26 44 CC[C@H](C)[C@@H](NC(=O)[C@@H]1COc2ccccc2C1)C(=O)O ZINC000217759351 CD On-Demand Unstable CDC42BPA 0 40 CC[C@H](C)[C@@H](NC(=O)[C@@H]1COc2ccccc2C1)C(=O)O ZINC000217759351 CD On-Demand Unstable ACAT 0 40 Cc1cc(/C=C\C(=O)O)ccc1NC(=O)c1cccnc1 ZINC000217759362 CF For-Sale Unstable TBXAS1 33 45 Cc1cc(/C=C\C(=O)O)ccc1NC(=O)c1cccnc1 ZINC000217759362 CF For-Sale Unstable HDAC1 0 47 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)NC[C@H]1C[C@H]3C=C[C@@H]1C3)C(=O)OC2 ZINC000217759371 II In-Stock Unstable IMPDH1 0 59 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)NC[C@H]1C[C@H]3C=C[C@@H]1C3)C(=O)OC2 ZINC000217759371 II In-Stock Unstable IMPDH2 0 59 Fc1ccc(C2CC(N[C@@H]3CCN4CCC[C@@H]34)C2)cc1 ZINC000217759392 CF For-Sale Unstable SLC18A3 40 38 NS(=O)(=O)c1ccc(C(=O)NC[C@H]2CCCN2c2nccs2)cc1 ZINC000217759400 FD For-Sale Unstable CA2 45 51 NS(=O)(=O)c1ccc(C(=O)NC[C@H]2CCCN2c2nccs2)cc1 ZINC000217759400 FD For-Sale Unstable CA1 26 40 NS(=O)(=O)c1ccc(C(=O)NC[C@H]2CCCN2c2nccs2)cc1 ZINC000217759400 FD For-Sale Unstable CA7 23 42 NS(=O)(=O)c1ccc(C(=O)NC[C@H]2CCCN2c2nccs2)cc1 ZINC000217759400 FD For-Sale Unstable CA4 19 42 NS(=O)(=O)c1ccc(C(=O)NC[C@H]2CCCN2c2nccs2)cc1 ZINC000217759400 FD For-Sale Unstable CA14 31 41 NS(=O)(=O)c1ccc(C(=O)NC[C@H]2CCCN2c2nccs2)cc1 ZINC000217759400 FD For-Sale Unstable CA12 15 42 NS(=O)(=O)c1ccc(C(=O)NC[C@H]2CCCN2c2nccs2)cc1 ZINC000217759400 FD For-Sale Unstable CA9 22 42 COc1cc([N+](=O)[O-])ccc1NC(=O)N/C=C/c1ccccc1F ZINC000217759433 EH For-Sale Unstable EPHX1 0 53 COc1cc([N+](=O)[O-])ccc1NC(=O)N/C=C/c1ccccc1F ZINC000217759433 EH For-Sale Unstable KCNMA1 24 53 COc1cc([N+](=O)[O-])ccc1NC(=O)N/C=C/c1ccccc1F ZINC000217759433 EH For-Sale Unstable WDR5 31 40 COc1cc([C@@H](C)N2C[C@@H](C)C[C@@H](C)C2)ccc1O ZINC000217759458 CG For-Sale Unstable PNLIP 0 50 COc1cc([C@@H](C)N2C[C@@H](C)C[C@@H](C)C2)ccc1O ZINC000217759458 CG For-Sale Unstable N1L 0 51 COc1cc([C@@H](C)N2C[C@@H](C)C[C@@H](C)C2)ccc1O ZINC000217759458 CG For-Sale Unstable RORC 45 42 COc1cc([C@@H](C)N2C[C@@H](C)C[C@@H](C)C2)ccc1O ZINC000217759458 CG For-Sale Unstable CAN2 0 41 COc1cc([C@@H](C)N2C[C@@H](C)C[C@@H](C)C2)ccc1O ZINC000217759458 CG For-Sale Unstable SLC22A3 0 44 Fc1ccc(C2CC(N[C@H]3CCN4CCC[C@@H]34)C2)cc1 ZINC000217759461 CF For-Sale Unstable SLC18A3 40 38 COc1ccc(CC(=O)N2CCC(N3CCC(OC)CC3)CC2)cc1OC ZINC000217759500 GE In-Stock Unstable CHRM2 58 44 COc1ccc(CC(=O)N2CCC(N3CCC(OC)CC3)CC2)cc1OC ZINC000217759500 GE In-Stock Unstable OPRK1 27 40 COc1ccc(CC(=O)N2CCC(N3CCC(OC)CC3)CC2)cc1OC ZINC000217759500 GE In-Stock Unstable CCR3 29 52 COc1ccc(CC(=O)N2CCC(N3CCC(OC)CC3)CC2)cc1OC ZINC000217759500 GE In-Stock Unstable MLNR 20 40 COc1ccc(CC(=O)N2CCC(N3CCC(OC)CC3)CC2)cc1OC ZINC000217759500 GE In-Stock Unstable EBP 18 40 COc1ccc(CC(=O)N2CCC(N3CCC(OC)CC3)CC2)cc1OC ZINC000217759500 GE In-Stock Unstable L3MBTL3 72 37 O=C(NC[C@@H]1CCCN1c1nccs1)c1cc2ccccc2[nH]1 ZINC000217759511 EG For-Sale Unstable CCKAR 23 42 O=C(NC[C@@H]1CCCN1c1nccs1)c1cc2ccccc2[nH]1 ZINC000217759511 EG For-Sale Unstable PYGL 60 39 O=C(NC[C@@H]1CCCN1c1nccs1)c1cc2ccccc2[nH]1 ZINC000217759511 EG For-Sale Unstable PLD2 30 41 O=C(NC[C@@H]1CCCN1c1nccs1)c1cc2ccccc2[nH]1 ZINC000217759511 EG For-Sale Unstable AKR1C3 22 42 CC[C@@H](Cn1ccnc1)NC(=O)c1cc(C(C)C)nc(N)n1 ZINC000217759531 DD In-Stock Unstable TBXAS1 27 40 O=C(N/C=C/c1ccccc1F)Nc1ccc([N+](=O)[O-])cc1 ZINC000217759547 DH For-Sale Bother NMBR 41 31 Clc1ccccc1C1CC(N[C@@H]2CCN3CCC[C@@H]23)C1 ZINC000217759571 CG For-Sale Unstable SLC6A1 0 52 O=C(NC[C@H]1CCCN1c1nccs1)c1cc2ccccc2[nH]1 ZINC000217759584 EG For-Sale Unstable CCKAR 23 42 O=C(NC[C@H]1CCCN1c1nccs1)c1cc2ccccc2[nH]1 ZINC000217759584 EG For-Sale Unstable PYGL 60 39 O=C(NC[C@H]1CCCN1c1nccs1)c1cc2ccccc2[nH]1 ZINC000217759584 EG For-Sale Unstable PLD2 30 41 O=C(NC[C@H]1CCCN1c1nccs1)c1cc2ccccc2[nH]1 ZINC000217759584 EG For-Sale Unstable AKR1C3 22 42 CC[C@H](Cn1ccnc1)NC(=O)c1cc(C(C)C)nc(N)n1 ZINC000217759617 DD In-Stock Unstable TBXAS1 27 40 Clc1ccccc1C1CC(N[C@H]2CCN3CCC[C@@H]23)C1 ZINC000217759645 CG For-Sale Unstable SLC6A1 0 52 O=C(N/C=C/c1ccccc1F)Nc1cccc([N+](=O)[O-])c1 ZINC000217759653 DH For-Sale Bother PPIA 15 42 O=C(N/C=C/c1ccccc1F)Nc1cccc([N+](=O)[O-])c1 ZINC000217759653 DH For-Sale Bother TRPM8 16 45 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCCCCC(=O)NCC(C)C)[C@H]21 ZINC000217759662 JI In-Stock Unstable HTR7 27 40 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCCCCC(=O)NCC(C)C)[C@@H]21 ZINC000217759728 JI In-Stock Unstable HTR7 27 40 CCOC(=O)c1c(C)n(Cc2cccnc2)c2ccc(O)cc12 ZINC000217759879 DG In-Stock Unstable PLA2G2A 69 42 CC(C)(C)OC(=O)N1Cc2ccc(S(=O)(=O)Cl)cc2C1 ZINC000217759909 DF For-Sale Unstable GPR119 43 42 CCCn1c(C)c(C(=O)OCC)c2cc(OC)ccc21 ZINC000217759981 CH In-Stock Unstable CNR1 0 58 CCCn1c(C)c(C(=O)OCC)c2cc(OC)ccc21 ZINC000217759981 CH In-Stock Unstable PTGS2 48 45 CCCn1c(C)c(C(=O)OCC)c2cc(OC)ccc21 ZINC000217759981 CH In-Stock Unstable ELANE 0 47 CCCn1c(C)c(C(=O)OCC)c2cc(OC)ccc21 ZINC000217759981 CH In-Stock Unstable CNR2 15 54 CCCn1c(C)c(C(=O)OCC)c2cc(OC)ccc21 ZINC000217759981 CH In-Stock Unstable PLA2G2A 61 47 CCCn1c(C)c(C(=O)OCC)c2cc(OC)ccc21 ZINC000217759981 CH In-Stock Unstable MTNR1A 53 40 CCCn1c(C)c(C(=O)OCC)c2cc(OC)ccc21 ZINC000217759981 CH In-Stock Unstable PTGDS 39 41 CCCn1c(C)c(C(=O)OCC)c2cc(OC)ccc21 ZINC000217759981 CH In-Stock Unstable AKR1C3 23 42 O[C@@H](CNCc1ccccc1)COc1ccccc1Br ZINC000217759984 EF On-Demand Unstable ADRB2 45 45 O[C@@H](CNCc1ccccc1)COc1ccccc1Br ZINC000217759984 EF On-Demand Unstable ADRB1 52 39 O[C@@H](CNCc1ccccc1)COc1ccccc1Br ZINC000217759984 EF On-Demand Unstable ADRB3 47 45 O[C@@H](CNCc1ccccc1)COc1ccccc1Br ZINC000217759984 EF On-Demand Unstable ABCB1 61 46 CCOC(=O)c1cc(S(=O)(=O)CC)cn1Cc1ccccc1 ZINC000217760027 DF In-Stock Unstable PLA2G2A 41 33 CCOC(=O)c1cc(S(=O)(=O)CC)cn1Cc1ccccc1 ZINC000217760027 DF In-Stock Unstable F2RL3 21 48 CCOC(=O)c1cc(S(=O)(=O)CC)cn1Cc1ccccc1 ZINC000217760027 DF In-Stock Unstable Q76353_9HIV1 0 42 COC1CCN(C2CCN(C(=O)Cc3ccc(SC(C)C)cc3)CC2)CC1 ZINC000217760059 GH In-Stock Unstable CHRM2 41 50 COC1CCN(C2CCN(C(=O)Cc3ccc(SC(C)C)cc3)CC2)CC1 ZINC000217760059 GH In-Stock Unstable CCR3 21 45 COC1CCN(C2CCN(C(=O)Cc3ccc(SC(C)C)cc3)CC2)CC1 ZINC000217760059 GH In-Stock Unstable L3MBTL3 58 36 CC(C)(C)OC(=O)N1C[C@H](O)C[C@@H]1C(=O)N1CCC1 ZINC000217760063 CC On-Demand Unstable PREP 39 60 O[C@H](CNCc1ccccc1)COc1ccccc1Br ZINC000217760072 EF On-Demand Unstable ADRB2 45 45 O[C@H](CNCc1ccccc1)COc1ccccc1Br ZINC000217760072 EF On-Demand Unstable ADRB1 52 39 O[C@H](CNCc1ccccc1)COc1ccccc1Br ZINC000217760072 EF On-Demand Unstable ADRB3 47 45 O[C@H](CNCc1ccccc1)COc1ccccc1Br ZINC000217760072 EF On-Demand Unstable ABCB1 61 46 O=C(N/C=C/c1ccccc1F)N1CCN(c2ccc(F)cc2)CC1 ZINC000217760082 EG For-Sale Unstable AKR1C3 0 45 CCOC(=O)c1c(C)n(CCOC)c2ccc(OC)cc12 ZINC000217760091 CF In-Stock Unstable CNR1 0 48 CCOC(=O)c1c(C)n(CCOC)c2ccc(OC)cc12 ZINC000217760091 CF In-Stock Unstable PTGS2 43 44 CCOC(=O)c1c(C)n(CCOC)c2ccc(OC)cc12 ZINC000217760091 CF In-Stock Unstable PLA2G2A 59 46 CCOC(=O)c1c(C)n(CCOC)c2ccc(OC)cc12 ZINC000217760091 CF In-Stock Unstable AKR1C3 19 41 O=C(c1ccc(F)cc1)C1CCN(C(=O)COc2cccc(C(F)(F)F)c2)CC1 ZINC000217760139 HI On-Demand Unstable COLA 89 43 O=C(c1ccc(F)cc1)C1CCN(C(=O)COc2cccc(C(F)(F)F)c2)CC1 ZINC000217760139 HI On-Demand Unstable CPT1A 84 43 O=C(c1ccc(F)cc1)C1CCN(C(=O)COc2cccc(C(F)(F)F)c2)CC1 ZINC000217760139 HI On-Demand Unstable CPT2 40 33 O=C(c1ccc(F)cc1)C1CCN(C(=O)COc2cccc(C(F)(F)F)c2)CC1 ZINC000217760139 HI On-Demand Unstable SLC18A3 40 41 O=C(c1ccc(F)cc1)C1CCN(C(=O)COc2cccc(C(F)(F)F)c2)CC1 ZINC000217760139 HI On-Demand Unstable MLNR 15 40 O=C(c1ccc(F)cc1)C1CCN(C(=O)COc2cccc(C(F)(F)F)c2)CC1 ZINC000217760139 HI On-Demand Unstable CHRNA10 27 43 O=C(c1ccc(F)cc1)C1CCN(C(=O)COc2cccc(C(F)(F)F)c2)CC1 ZINC000217760139 HI On-Demand Unstable CACNA1G 32 40 O=C(c1ccc(F)cc1)C1CCN(C(=O)COc2cccc(C(F)(F)F)c2)CC1 ZINC000217760139 HI On-Demand Unstable LIPG 56 40 O=C(c1ccc(F)cc1)C1CCN(C(=O)COc2cccc(C(F)(F)F)c2)CC1 ZINC000217760139 HI On-Demand Unstable WNT3A 44 31 O=C(c1ccc(F)cc1)C1CCN(C(=O)COc2cccc(C(F)(F)F)c2)CC1 ZINC000217760139 HI On-Demand Unstable PDS 44 36 O=C(O)/C=C\C(=O)NC(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000217760157 CD For-Sale Unstable SCN5A 0 41 O=C(O)/C=C\C(=O)NC(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000217760157 CD For-Sale Unstable EPHX2 24 51 O=C(O)/C=C\c1ccccc1CN1CC(=O)NC(=O)C1 ZINC000217760171 CC For-Sale Unstable PTGER2 43 48 O=C(O)/C=C\c1ccccc1CN1CC(=O)NC(=O)C1 ZINC000217760171 CC For-Sale Unstable PTGER4 0 48 O=C(O)/C=C\c1ccccc1CN1CC(=O)NC(=O)C1 ZINC000217760171 CC For-Sale Unstable PTGER3 18 48 CC(C)(C)OC(=O)N1C[C@@H](O)C[C@@H]1C(=O)N1CCC1 ZINC000217760175 CC On-Demand Unstable PREP 39 60 CCOC(=O)c1c(C)n(Cc2cccnc2)c2ccc(OC)cc12 ZINC000217760214 DH In-Stock Unstable PTGS2 36 46 CCOC(=O)c1c(C)n(Cc2cccnc2)c2ccc(OC)cc12 ZINC000217760214 DH In-Stock Unstable PPARG 19 40 CCOC(=O)c1c(C)n(Cc2cccnc2)c2ccc(OC)cc12 ZINC000217760214 DH In-Stock Unstable ALOX5AP 90 38 CCOC(=O)c1c(C)n(Cc2cccnc2)c2ccc(OC)cc12 ZINC000217760214 DH In-Stock Unstable PLA2G2A 87 54 CC(C)(C)OC(=O)N1C[C@H](O)C[C@H]1C(=O)N1CCC1 ZINC000217760254 CC On-Demand Unstable PREP 39 60 O=C(O)/C=C\C(=O)NC(=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000217760264 CD For-Sale Unstable SCN5A 0 41 O=C(O)/C=C\C(=O)NC(=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000217760264 CD For-Sale Unstable EPHX2 24 51 COc1ncccc1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217760270 DD For-Sale Unstable HCRTR1 27 40 COc1ncccc1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217760270 DD For-Sale Unstable HCRTR2 23 40 Cc1ccc(/C=C\C(=O)NCC[C@@H](C)O)cc1 ZINC000217760299 BD On-Demand Unstable PYGL 22 43 Cc1ccc(/C=C\C(=O)NCC[C@@H](C)O)cc1 ZINC000217760299 BD On-Demand Unstable HDAC8 0 43 Cc1ccc(/C=C\C(=O)NCC[C@@H](C)O)cc1 ZINC000217760299 BD On-Demand Unstable MMP2 15 48 Cc1ccc(/C=C\C(=O)NCC[C@@H](C)O)cc1 ZINC000217760299 BD On-Demand Unstable HDAC1 24 43 Cc1ccc(/C=C\C(=O)NCC[C@@H](C)O)cc1 ZINC000217760299 BD On-Demand Unstable HDAC4 0 43 CCOc1ccc(NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217760300 DI For-Sale Unstable CA1 44 40 CCOc1ccc(NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217760300 DI For-Sale Unstable FAAH 19 42 CCOc1ccc(NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217760300 DI For-Sale Unstable CA12 17 40 CCOc1ccc(NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217760300 DI For-Sale Unstable CA9 18 40 CCCn1c(C)c(C(=O)OCC)c2cc(OCC)ccc21 ZINC000217760330 CH In-Stock Unstable CNR1 0 48 CCCn1c(C)c(C(=O)OCC)c2cc(OCC)ccc21 ZINC000217760330 CH In-Stock Unstable PLA2G2A 58 48 COc1ncccc1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217760356 DD For-Sale Unstable HCRTR1 27 40 COc1ncccc1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217760356 DD For-Sale Unstable HCRTR2 23 40 O=C(NC[C@@]12CC[C@@H]3C[C@@H](C[C@@H](C3)C1)C2)Nc1ccccc1 ZINC000217760372 CI In-Stock Unstable P2RX7 34 63 O=C(NC[C@@]12CC[C@@H]3C[C@@H](C[C@@H](C3)C1)C2)Nc1ccccc1 ZINC000217760372 CI In-Stock Unstable CCR3 15 41 O=C(NC[C@@]12CC[C@@H]3C[C@@H](C[C@@H](C3)C1)C2)Nc1ccccc1 ZINC000217760372 CI In-Stock Unstable CCKBR 0 48 O=C(NC[C@@]12CC[C@@H]3C[C@@H](C[C@@H](C3)C1)C2)Nc1ccccc1 ZINC000217760372 CI In-Stock Unstable EPHX2 70 48 O=C(NC[C@@]12CC[C@@H]3C[C@@H](C[C@@H](C3)C1)C2)Nc1ccccc1 ZINC000217760372 CI In-Stock Unstable ACAT 0 49 O=C(NC[C@@]12CC[C@@H]3C[C@@H](C[C@@H](C3)C1)C2)Nc1ccccc1 ZINC000217760372 CI In-Stock Unstable P95276_MYCTO 0 44 Cc1ccc(/C=C\C(=O)NCC[C@H](C)O)cc1 ZINC000217760383 BD For-Sale Unstable PYGL 22 43 Cc1ccc(/C=C\C(=O)NCC[C@H](C)O)cc1 ZINC000217760383 BD For-Sale Unstable HDAC8 0 43 Cc1ccc(/C=C\C(=O)NCC[C@H](C)O)cc1 ZINC000217760383 BD For-Sale Unstable HDAC1 24 43 Cc1ccc(/C=C\C(=O)NCC[C@H](C)O)cc1 ZINC000217760383 BD For-Sale Unstable HDAC4 0 43 O=C(O)CC[C@@H](NC(=O)C[C@@H]1C[C@@H]2CC[C@@H]1C2)C(=O)O ZINC000217760388 CD For-Sale Unstable FOLH1 49 45 O=C(O)CC[C@@H](NC(=O)C[C@@H]1C[C@@H]2CC[C@@H]1C2)C(=O)O ZINC000217760388 CD For-Sale Unstable NAALAD2 59 45 CCOC(=O)c1c(C)n(CCOC)c2ccc(OCC)cc12 ZINC000217760434 DG In-Stock Unstable PLA2G2A 60 45 O=C(O)CC[C@H](NC(=O)C[C@@H]1C[C@@H]2CC[C@@H]1C2)C(=O)O ZINC000217760462 CD For-Sale Unstable FOLH1 49 45 O=C(O)CC[C@H](NC(=O)C[C@@H]1C[C@@H]2CC[C@@H]1C2)C(=O)O ZINC000217760462 CD For-Sale Unstable NAALAD2 59 45 O=C(O)/C=C\c1cccc(NC(=O)CCn2ccnc2)n1 ZINC000217760469 CD For-Sale Unstable TBXAS1 49 48 O=C(O)/C=C\c1cccc(NC(=O)CCn2ccnc2)n1 ZINC000217760469 CD For-Sale Unstable CYP27B1 46 35 CC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217760506 CH For-Sale Unstable PRNP 21 43 COc1ccccc1CN1CCN(C[C@@H]2[C@H]3CNC[C@H]32)CC1 ZINC000217760520 DD In-Stock Unstable HTR1A 24 40 COc1ccccc1CN1CCN(C[C@@H]2[C@H]3CNC[C@H]32)CC1 ZINC000217760520 DD In-Stock Unstable DRD2 22 43 COc1ccccc1CN1CCN(C[C@@H]2[C@H]3CNC[C@H]32)CC1 ZINC000217760520 DD In-Stock Unstable ADRA1B 18 43 COc1ccccc1CN1CCN(C[C@@H]2[C@H]3CNC[C@H]32)CC1 ZINC000217760520 DD In-Stock Unstable DRD3 21 41 COc1ccccc1CN1CCN(C[C@@H]2[C@H]3CNC[C@H]32)CC1 ZINC000217760520 DD In-Stock Unstable HTR7 19 45 COc1ccccc1CN1CCN(C[C@@H]2[C@H]3CNC[C@H]32)CC1 ZINC000217760520 DD In-Stock Unstable MBTPS1 43 33 COC1CCN(C2CCN(C(=O)C3c4ccccc4Oc4ccccc43)CC2)CC1 ZINC000217760521 HI In-Stock Unstable CHRM2 45 41 COC1CCN(C2CCN(C(=O)C3c4ccccc4Oc4ccccc43)CC2)CC1 ZINC000217760521 HI In-Stock Unstable L3MBTL3 73 38 O=C(O)CC[C@@H](NC(=O)C[C@H]1C[C@@H]2CC[C@@H]1C2)C(=O)O ZINC000217760538 CD For-Sale Unstable FOLH1 49 45 O=C(O)CC[C@@H](NC(=O)C[C@H]1C[C@@H]2CC[C@@H]1C2)C(=O)O ZINC000217760538 CD For-Sale Unstable NAALAD2 59 45 CCOC(=O)c1c(C)n(Cc2cccnc2)c2ccc(OCC)cc12 ZINC000217760547 EH In-Stock Unstable ALOX5AP 94 41 CCOC(=O)c1c(C)n(Cc2cccnc2)c2ccc(OCC)cc12 ZINC000217760547 EH In-Stock Unstable PLA2G2A 83 46 CCOC(=O)c1c(C)n(Cc2cccnc2)c2ccc(OCC)cc12 ZINC000217760547 EH In-Stock Unstable CYP3A4 17 40 O=C(O)/C=C\c1cccc(NC(=O)c2ccc(Cl)cc2)n1 ZINC000217760559 DG For-Sale Anodyne GRM5 19 40 O=C(O)/C=C\c1cccc(NC(=O)c2ccc(Cl)cc2)n1 ZINC000217760559 DG For-Sale Anodyne MAP3K5 42 42 O=C(O)/C=C\c1cccc(NC(=O)c2ccc(Cl)cc2)n1 ZINC000217760559 DG For-Sale Anodyne LUCI_LUCLA 33 43 O=C(O)/C=C\c1cccc(NC(=O)c2ccc(Cl)cc2)n1 ZINC000217760559 DG For-Sale Anodyne KCNK3 35 42 CC1(C)OB(c2ccc(C(=O)Nc3nc4c(s3)CCCC4)cc2)OC1(C)C ZINC000217760601 GH For-Sale Unstable SLC27A1 31 41 CC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2F)c1 ZINC000217760621 CH For-Sale Unstable CCR3 19 44 CC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2F)c1 ZINC000217760621 CH For-Sale Unstable AKR1C3 23 43 CC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2F)c1 ZINC000217760621 CH For-Sale Unstable KCNK3 92 39 CC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2F)c1 ZINC000217760621 CH For-Sale Unstable KCNK9 54 36 O=C(O)/C=C\c1cccc(NC(=O)c2cccnc2)n1 ZINC000217760635 CD For-Sale Anodyne TBXAS1 34 40 O=C(O)/C=C\c1cccc(NC(=O)c2cccnc2)n1 ZINC000217760635 CD For-Sale Anodyne GRM5 16 46 O=C(O)/C=C\c1cccc(NC(=O)c2cccnc2)n1 ZINC000217760635 CD For-Sale Anodyne NAMPT 18 42 CCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2C ZINC000217760672 CG In-Stock Unstable PLA2G2A 43 45 Cc1ccc(C2CC(N[C@@H]3CCN4CCC[C@@H]34)C2)cc1 ZINC000217760693 CG For-Sale Unstable SLC18A3 26 50 CCCCC(=O)Nc1cc(/C=C\C(=O)O)ccc1OC ZINC000217760719 CF For-Sale Unstable TUBB1 47 38 CCCCC(=O)Nc1cc(/C=C\C(=O)O)ccc1OC ZINC000217760719 CF For-Sale Unstable AKR1C3 41 47 CN1CCO[C@@H](CNC(=O)[C@@H](CN)Cc2ccccc2)C1 ZINC000217760726 CC For-Sale Unstable ACE 47 37 CN1CCO[C@@H](CNC(=O)[C@@H](CN)Cc2ccccc2)C1 ZINC000217760726 CC For-Sale Unstable MME 100 38 CN1CCO[C@@H](CNC(=O)[C@@H](CN)Cc2ccccc2)C1 ZINC000217760726 CC For-Sale Unstable ANPEP 96 36 CN1CCO[C@@H](CNC(=O)[C@@H](CN)Cc2ccccc2)C1 ZINC000217760726 CC For-Sale Unstable PGA5 43 31 CN1CCO[C@@H](CNC(=O)[C@@H](CN)Cc2ccccc2)C1 ZINC000217760726 CC For-Sale Unstable LAP3 58 36 O=C1CN(C(=O)/C=C\c2cccc(F)c2)CC(=O)N1 ZINC000217760736 CC For-Sale Unstable CCR2 52 40 Cc1ccc(C2CC(N[C@H]3CCN4CCC[C@@H]34)C2)cc1 ZINC000217760778 CG For-Sale Unstable SLC18A3 26 50 CCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CC ZINC000217760788 CH In-Stock Unstable PLA2G2A 63 47 CN1CCO[C@H](CNC(=O)[C@@H](CN)Cc2ccccc2)C1 ZINC000217760815 CC For-Sale Unstable ACE 47 37 CN1CCO[C@H](CNC(=O)[C@@H](CN)Cc2ccccc2)C1 ZINC000217760815 CC For-Sale Unstable MME 100 38 CN1CCO[C@H](CNC(=O)[C@@H](CN)Cc2ccccc2)C1 ZINC000217760815 CC For-Sale Unstable ANPEP 96 36 CN1CCO[C@H](CNC(=O)[C@@H](CN)Cc2ccccc2)C1 ZINC000217760815 CC For-Sale Unstable PGA5 43 31 CN1CCO[C@H](CNC(=O)[C@@H](CN)Cc2ccccc2)C1 ZINC000217760815 CC For-Sale Unstable LAP3 58 36 Cc1cc(COc2ccccc2)oc1C(=O)N1CCC[C@@H]1c1ccccn1 ZINC000217760844 FJ In-Stock Unstable CPT1A 122 46 Cc1cc(COc2ccccc2)oc1C(=O)N1CCC[C@@H]1c1ccccn1 ZINC000217760844 FJ In-Stock Unstable CPT2 44 37 O=C(CCCc1ccccc1)NC[C@@H]1CCCN1c1nccs1 ZINC000217760845 EG For-Sale Unstable GRIN2B 15 40 O=C(CCCc1ccccc1)NC[C@@H]1CCCN1c1nccs1 ZINC000217760845 EG For-Sale Unstable PREP 64 47 CCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCC ZINC000217760898 DI In-Stock Unstable PLA2G2A 61 51 O=C(N[C@@H]1C[C@@H]1c1ccccc1)[C@H]1CC=CC[C@H]1C(=O)O ZINC000217760899 CE On-Demand Unstable EPHX2 22 47 COC(=O)[C@@H](C)NC(=O)Cn1ccc2c(NC(C)=O)cccc21 ZINC000217760916 DD In-Stock Unstable NR5A1 33 40 O=C(CCCc1ccccc1)NC[C@H]1CCCN1c1nccs1 ZINC000217760924 EG For-Sale Unstable GRIN2B 15 40 O=C(CCCc1ccccc1)NC[C@H]1CCCN1c1nccs1 ZINC000217760924 EG For-Sale Unstable PREP 64 47 Cc1cc(COc2ccccc2)oc1C(=O)N1CCC[C@H]1c1ccccn1 ZINC000217760929 FJ In-Stock Unstable CPT1A 122 46 Cc1cc(COc2ccccc2)oc1C(=O)N1CCC[C@H]1c1ccccn1 ZINC000217760929 FJ In-Stock Unstable CPT2 44 37 O=C(O)[C@H]1CC=CC[C@@H]1C(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000217760985 CE For-Sale Unstable EPHX2 22 47 CCCCn1c(C)c(C(=O)OCC)c2cc(OCCC)ccc21 ZINC000217761027 DJ In-Stock Unstable CNR1 0 47 CCCCn1c(C)c(C(=O)OCC)c2cc(OCCC)ccc21 ZINC000217761027 DJ In-Stock Unstable PTGS2 0 41 CCCCn1c(C)c(C(=O)OCC)c2cc(OCCC)ccc21 ZINC000217761027 DJ In-Stock Unstable CNR2 15 45 CCCCn1c(C)c(C(=O)OCC)c2cc(OCCC)ccc21 ZINC000217761027 DJ In-Stock Unstable PLA2G2A 72 59 CCCCn1c(C)c(C(=O)OCC)c2cc(OCCC)ccc21 ZINC000217761027 DJ In-Stock Unstable PLA2G4B 67 33 COc1ccc(OCC(=O)NC[C@@H]2CCCN2c2nccs2)cc1 ZINC000217761033 EE For-Sale Unstable NOS2 17 41 CCc1cnc(NC(=O)c2ccc(B3OC(C)(C)C(C)(C)O3)cc2)s1 ZINC000217761036 FG For-Sale Unstable FDPS 16 50 O=C(O)[C@@H]1CC=CC[C@H]1C(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000217761045 CE For-Sale Unstable EPHX2 22 47 COc1ccc(OCC(=O)NC[C@H]2CCCN2c2nccs2)cc1 ZINC000217761109 EE For-Sale Unstable NOS2 17 41 CCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCOC ZINC000217761128 DH In-Stock Unstable PLA2G2A 63 48 CC(C)Oc1ccccc1[C@@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc3c21 ZINC000217761135 JK In-Stock Unstable AKR1B1 0 44 CC(C)Oc1ccccc1[C@@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc3c21 ZINC000217761135 JK In-Stock Unstable CYP1A1 28 41 CC(C)Oc1ccccc1[C@@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc3c21 ZINC000217761135 JK In-Stock Unstable CYP1A2 22 41 O=C(O)/C=C\c1cnc(NC(=O)Cc2ccccc2)s1 ZINC000217761158 CE For-Sale Unstable CSNK1D 27 48 O=C(O)/C=C\c1cnc(NC(=O)Cc2ccccc2)s1 ZINC000217761158 CE For-Sale Unstable CA5B 33 45 O=C(O)/C=C\c1cnc(NC(=O)Cc2ccccc2)s1 ZINC000217761158 CE For-Sale Unstable CA5A 38 45 O=C(O)/C=C\c1cnc(NC(=O)Cc2ccccc2)s1 ZINC000217761158 CE For-Sale Unstable CDK5 51 58 O=C(N[C@@H]1C[C@@H]1c1ccccc1)[C@H]1CCCC[C@H]1C(=O)O ZINC000217761174 CF On-Demand Unstable EPHX2 24 50 Cc1cccc(NC(=O)N/C=C/c2ccccc2F)c1 ZINC000217761177 CH For-Sale Unstable CCKAR 23 49 Cc1cccc(NC(=O)N/C=C/c2ccccc2F)c1 ZINC000217761177 CH For-Sale Unstable KDR 18 42 Cc1cccc(NC(=O)N/C=C/c2ccccc2F)c1 ZINC000217761177 CH For-Sale Unstable KCNK3 105 44 Cc1cccc(NC(=O)N/C=C/c2ccccc2F)c1 ZINC000217761177 CH For-Sale Unstable KCNK9 64 44 COC1CCN(C2CCN(C(=O)c3cc(C4CC4)on3)CC2)CC1 ZINC000217761189 EE In-Stock Unstable L3MBTL3 83 40 O=C1CN(C(=O)/C=C\c2cccc([N+](=O)[O-])c2)CC(=O)N1 ZINC000217761208 CC For-Sale Unstable CACNA1D 53 34 O=C1CN(C(=O)/C=C\c2cccc([N+](=O)[O-])c2)CC(=O)N1 ZINC000217761208 CC For-Sale Unstable TRPM8 17 50 C[C@@H](O)[C@@H](NC(=O)[C@@H]1COc2ccccc2C1)C(=O)O ZINC000217761209 CC For-Sale Unstable ROCK2 21 44 C[C@@H](O)[C@@H](NC(=O)[C@@H]1COc2ccccc2C1)C(=O)O ZINC000217761209 CC For-Sale Unstable ACAT 0 42 Cc1ccnn1Cc1ccccc1/C=C\C(=O)O ZINC000217761216 BE For-Sale Unstable PTGER2 48 47 Cc1ccnn1Cc1ccccc1/C=C\C(=O)O ZINC000217761216 BE For-Sale Unstable PTGER4 23 48 Cc1ccnn1Cc1ccccc1/C=C\C(=O)O ZINC000217761216 BE For-Sale Unstable PTGER3 19 48 Cc1ccnn1Cc1ccccc1/C=C\C(=O)O ZINC000217761216 BE For-Sale Unstable PTGDR 0 45 CCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CC(C)C ZINC000217761217 DJ In-Stock Unstable PLA2G2A 60 45 CC(C)Oc1ccccc1[C@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc3c21 ZINC000217761220 JK In-Stock Unstable AKR1B1 0 44 CC(C)Oc1ccccc1[C@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc3c21 ZINC000217761220 JK In-Stock Unstable CYP1A1 28 41 CC(C)Oc1ccccc1[C@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc3c21 ZINC000217761220 JK In-Stock Unstable CYP1A2 22 41 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable PLG 20 40 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable PRSS1 15 40 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable ACE 39 53 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable OPRM1 55 48 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable OPRD1 62 48 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable OPRK1 23 52 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable ABAT 44 36 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable MME 86 43 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable ANPEP 82 36 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable TACR1 25 57 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable MC4R 48 44 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable CMA1 28 50 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable FCER2 83 45 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable TACR2 57 58 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable RNPEP 32 42 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable PTPN2 36 44 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable KLK3 83 51 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable CTSB 50 47 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable PAPA1_CARPA 58 37 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable NMT1 37 40 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable CYSP_TRYCR 44 35 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable CCKAR 40 38 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable CTSL 36 44 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable CPA1 49 42 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable F2R 51 52 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable NPFFR2 69 45 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable C3AR1 34 41 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable TACR3 27 41 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable NAALAD2 31 43 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable MC3R 59 42 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable MC5R 48 39 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable CAPNS1 47 33 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable MMP3 24 46 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable GRIA1 66 46 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable MMP14 53 34 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable HLA-DRB1 73 60 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable HDAC1 23 52 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable HDAC2 24 40 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable MMP11 58 34 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable FURIN 57 39 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable PTPN1 20 40 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable CTSS 16 43 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable GHSR 22 51 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable CAPN1 65 42 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable MMP9 23 60 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable CAPN2 47 35 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable ACE2 64 37 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable MC1R 65 44 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable MMP1 24 47 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable FPR1 47 44 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable CTRB_BOVIN 47 35 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable BLA1_STEMA 73 44 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable KISS1R 59 34 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable POLG_WNV 93 46 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable QRFPR 72 47 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable NPFFR1 77 46 NCCCCC(=O)N[C@H](Cc1ccccc1)C(N)=O ZINC000217761236 CC On-Demand Unstable NOD1 44 43 O=C(O)[C@H]1CCCC[C@@H]1C(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000217761247 CF For-Sale Unstable EPHX2 24 50 C[C@H](O)[C@@H](NC(=O)[C@@H]1COc2ccccc2C1)C(=O)O ZINC000217761286 CC For-Sale Unstable ROCK2 21 44 C[C@H](O)[C@@H](NC(=O)[C@@H]1COc2ccccc2C1)C(=O)O ZINC000217761286 CC For-Sale Unstable ACAT 0 42 O=C1CN(C(=O)/C=C\c2ccc(Cl)c(Cl)c2)CC(=O)N1 ZINC000217761288 DD For-Sale Unstable ITGAL 22 45 O=C1CN(C(=O)/C=C\c2ccc(Cl)c(Cl)c2)CC(=O)N1 ZINC000217761288 DD For-Sale Unstable PYGL 26 45 O=C1CN(C(=O)/C=C\c2ccc(Cl)c(Cl)c2)CC(=O)N1 ZINC000217761288 DD For-Sale Unstable CCR2 22 46 O=C1CN(C(=O)/C=C\c2ccc(Cl)c(Cl)c2)CC(=O)N1 ZINC000217761288 DD For-Sale Unstable GPR183 0 55 O=C(N/C=C/c1ccccc1F)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217761299 FK For-Sale Anodyne GUAB 0 46 O=C(N/C=C/c1ccccc1F)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217761299 FK For-Sale Anodyne RAF1 32 45 O=C(N/C=C/c1ccccc1F)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217761299 FK For-Sale Anodyne ENV 40 30 O=C(N/C=C/c1ccccc1F)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217761299 FK For-Sale Anodyne Q8MMZ8_EIMTE 51 45 O=C(N/C=C/c1ccccc1F)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217761299 FK For-Sale Anodyne BRAF 15 40 O=C(N/C=C/c1ccccc1F)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217761299 FK For-Sale Anodyne PTPA 0 46 O=C(N/C=C/c1ccccc1F)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217761299 FK For-Sale Anodyne IMDH_CRYPV 33 48 O=C(N/C=C/c1ccccc1F)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217761299 FK For-Sale Anodyne BLM 0 46 COC1CCN(C2CCN(C(=O)[C@H]3CC=CCC3)CC2)CC1 ZINC000217761310 DE In-Stock Unstable L3MBTL3 56 35 CC(C)CC(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217761314 CF For-Sale Unstable PTGER2 23 41 CC(C)CC(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217761314 CF For-Sale Unstable AKR1C3 43 48 CCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217761321 FJ In-Stock Unstable ALOX5 16 45 CCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217761321 FJ In-Stock Unstable PPARG 28 41 CCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217761321 FJ In-Stock Unstable PLA2G1B 48 37 CCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217761321 FJ In-Stock Unstable ALOX5AP 97 40 CCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217761321 FJ In-Stock Unstable PLA2G2A 167 60 CCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217761321 FJ In-Stock Unstable PLA2G2E 0 42 CCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217761321 FJ In-Stock Unstable PLA2G10 40 37 CCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217761321 FJ In-Stock Unstable PLA2G2F 47 34 CCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217761321 FJ In-Stock Unstable PLA2G2D 54 34 CCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217761321 FJ In-Stock Unstable PLA2G5 48 42 CCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217761321 FJ In-Stock Unstable PTGES2 52 32 O=C(O)[C@@H]1CCCC[C@H]1C(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000217761333 CF For-Sale Unstable EPHX2 24 50 CN1C(=O)[C@@H]2CC[C@H]1CN(C(=O)CCCCc1ccccc1)C2 ZINC000217761343 DE In-Stock Unstable ACE 51 39 CN1C(=O)[C@@H]2CC[C@H]1CN(C(=O)CCCCc1ccccc1)C2 ZINC000217761343 DE In-Stock Unstable FKBP1A 39 42 CN1C(=O)[C@@H]2CC[C@H]1CN(C(=O)CCCCc1ccccc1)C2 ZINC000217761343 DE In-Stock Unstable SLC18A2 40 38 CN1C(=O)[C@@H]2CC[C@H]1CN(C(=O)CCCCc1ccccc1)C2 ZINC000217761343 DE In-Stock Unstable SSTR4 40 33 CN1C(=O)[C@@H]2CC[C@H]1CN(C(=O)CCCCc1ccccc1)C2 ZINC000217761343 DE In-Stock Unstable TRY1_BOVIN 0 43 CN1C(=O)[C@@H]2CC[C@H]1CN(C(=O)CCCCc1ccccc1)C2 ZINC000217761343 DE In-Stock Unstable PREP 55 43 CN1C(=O)[C@@H]2CC[C@H]1CN(C(=O)CCCCc1ccccc1)C2 ZINC000217761343 DE In-Stock Unstable FAAH 51 41 CN1C(=O)[C@@H]2CC[C@H]1CN(C(=O)CCCCc1ccccc1)C2 ZINC000217761343 DE In-Stock Unstable CES1 49 34 CN1C(=O)[C@@H]2CC[C@H]1CN(C(=O)CCCCc1ccccc1)C2 ZINC000217761343 DE In-Stock Unstable MGLL 0 40 CN1C(=O)[C@@H]2CC[C@H]1CN(C(=O)CCCCc1ccccc1)C2 ZINC000217761343 DE In-Stock Unstable ACHP_LYMST 16 40 CN1C(=O)[C@@H]2CC[C@H]1CN(C(=O)CCCCc1ccccc1)C2 ZINC000217761343 DE In-Stock Unstable Q8WSF8_APLCA 23 40 CN1C(=O)[C@@H]2CC[C@H]1CN(C(=O)CCCCc1ccccc1)C2 ZINC000217761343 DE In-Stock Unstable CES1D 52 31 CC(C)(C)OC(=O)N1CCC(C2CCC(=O)CC2)CC1 ZINC000217761350 CG For-Sale Unstable GPR119 45 58 C[C@H](O)[C@H](NC(=O)[C@@H]1COc2ccccc2C1)C(=O)O ZINC000217761373 CC For-Sale Unstable ROCK2 21 44 C[C@H](O)[C@H](NC(=O)[C@@H]1COc2ccccc2C1)C(=O)O ZINC000217761373 CC For-Sale Unstable ACAT 0 42 COC1CCN(C2CCN(C(=O)[C@@H]3CC=CCC3)CC2)CC1 ZINC000217761382 DE In-Stock Unstable L3MBTL3 56 35 CN(Cc1cccc(/C=C\C(=O)O)c1)C(=O)C1CCC1 ZINC000217761390 CF For-Sale Unstable NR1H4 47 48 CCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCc1ccccc1 ZINC000217761433 FK In-Stock Unstable CNR1 15 44 CCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCc1ccccc1 ZINC000217761433 FK In-Stock Unstable PPARG 28 43 CCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCc1ccccc1 ZINC000217761433 FK In-Stock Unstable PPARA 15 40 CCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCc1ccccc1 ZINC000217761433 FK In-Stock Unstable CNR2 15 43 CCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCc1ccccc1 ZINC000217761433 FK In-Stock Unstable ALOX5AP 61 31 CCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCc1ccccc1 ZINC000217761433 FK In-Stock Unstable PLA2G4A 32 42 CCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCc1ccccc1 ZINC000217761433 FK In-Stock Unstable PLA2G2A 119 51 CCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCc1ccccc1 ZINC000217761433 FK In-Stock Unstable PTGDR 22 40 CN(Cc1cccc(/C=C\C(=O)O)c1)C(=O)C1CCCC1 ZINC000217761463 CF For-Sale Unstable NR1H4 49 50 O=C(O)/C=C\C(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000217761465 BD For-Sale Unstable SCN5A 0 41 O=C(O)/C=C\C(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000217761465 BD For-Sale Unstable EPHX2 23 47 COc1ccc(CNc2nnc(Cl)cc2C(=O)O)cc1 ZINC000217761485 CE For-Sale Unstable PDE6A 42 33 COc1ccc(CNc2nnc(Cl)cc2C(=O)O)cc1 ZINC000217761485 CE For-Sale Unstable ZAP70 40 42 COc1ccc(CNc2nnc(Cl)cc2C(=O)O)cc1 ZINC000217761485 CE For-Sale Unstable PTGDR 17 41 COc1ccc(CNc2nnc(Cl)cc2C(=O)O)cc1 ZINC000217761485 CE For-Sale Unstable STAT6 53 39 COc1ccc(CNc2nnc(Cl)cc2C(=O)O)cc1 ZINC000217761485 CE For-Sale Unstable PROKR1 74 37 COc1ccc(CNc2nnc(Cl)cc2C(=O)O)cc1 ZINC000217761485 CE For-Sale Unstable AKR1C2 54 39 COc1ccc(CNc2nnc(Cl)cc2C(=O)O)cc1 ZINC000217761485 CE For-Sale Unstable DRTS_TRYCR 47 32 CCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1cccnc1 ZINC000217761536 FI In-Stock Unstable ALOX5AP 87 40 CCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1cccnc1 ZINC000217761536 FI In-Stock Unstable PLA2G2A 86 48 O=C(O)/C=C\C(=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000217761545 BD For-Sale Unstable SCN5A 0 41 O=C(O)/C=C\C(=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000217761545 BD For-Sale Unstable EPHX2 23 47 COc1ccc(NC(=O)CC[C@@H]2NC(=O)c3ccccc3NC2=O)cc1-c1nnn[nH]1 ZINC000217761665 HD In-Stock Unstable CASP2 18 41 COc1ccc(NC(=O)CC[C@@H]2NC(=O)c3ccccc3NC2=O)cc1-c1nnn[nH]1 ZINC000217761665 HD In-Stock Unstable CASP6 17 41 COc1ccc(NC(=O)CC[C@@H]2NC(=O)c3ccccc3NC2=O)cc1-c1nnn[nH]1 ZINC000217761665 HD In-Stock Unstable ENPP1 62 33 O=C(c1ccc(F)cc1)C1CCN(C(=O)COc2cc(Cl)cc(Cl)c2)CC1 ZINC000217761677 HJ On-Demand Unstable HTR2A 15 49 O=C(c1ccc(F)cc1)C1CCN(C(=O)COc2cc(Cl)cc(Cl)c2)CC1 ZINC000217761677 HJ On-Demand Unstable COLA 54 40 O=C(c1ccc(F)cc1)C1CCN(C(=O)COc2cc(Cl)cc(Cl)c2)CC1 ZINC000217761677 HJ On-Demand Unstable CPT1A 50 40 O=C(c1ccc(F)cc1)C1CCN(C(=O)COc2cc(Cl)cc(Cl)c2)CC1 ZINC000217761677 HJ On-Demand Unstable CPT2 27 40 O=C(c1ccc(F)cc1)C1CCN(C(=O)COc2cc(Cl)cc(Cl)c2)CC1 ZINC000217761677 HJ On-Demand Unstable SLC18A3 43 45 O=C(c1ccc(F)cc1)C1CCN(C(=O)COc2cc(Cl)cc(Cl)c2)CC1 ZINC000217761677 HJ On-Demand Unstable MLNR 21 43 O=C(c1ccc(F)cc1)C1CCN(C(=O)COc2cc(Cl)cc(Cl)c2)CC1 ZINC000217761677 HJ On-Demand Unstable WNT3A 53 35 Clc1ccc(C2CC(N[C@@H]3CCN4CCC[C@@H]34)C2)cc1 ZINC000217761698 CG For-Sale Unstable SLC18A3 31 50 O=C(N/C=C/c1ccccc1F)Nc1cccc(Cl)c1 ZINC000217761743 CI For-Sale Anodyne PPIA 16 40 O=C(N/C=C/c1ccccc1F)Nc1cccc(Cl)c1 ZINC000217761743 CI For-Sale Anodyne KCNK3 50 44 CCOC(=O)c1c(C)n(CC)c2ccc(OC(C)C)cc12 ZINC000217761753 CH In-Stock Unstable PLA2G2A 50 38 CO[C@@H]1CCN(C(=O)c2cccc(S(=O)(=O)N3CCCN(C)CC3)c2)C1 ZINC000217761755 GC In-Stock Unstable AKR1C3 66 42 Clc1ccc(C2CC(N[C@H]3CCN4CCC[C@@H]34)C2)cc1 ZINC000217761766 CG For-Sale Unstable SLC18A3 31 50 O=C(CCC(=O)c1ccccc1)NC[C@@H]1CCCN1c1nccs1 ZINC000217761804 EF For-Sale Unstable PREP 17 40 O=C(N/C=C/c1ccccc1F)Nc1ccc(Cl)cc1 ZINC000217761845 CI For-Sale Anodyne MTCA1 18 40 O=C(N/C=C/c1ccccc1F)Nc1ccc(Cl)cc1 ZINC000217761845 CI For-Sale Anodyne P95276_MYCTO 0 42 CCCn1c(C)c(C(=O)OCC)c2cc(OC(C)C)ccc21 ZINC000217761851 DI In-Stock Unstable PLA2G2A 45 42 CC(F)(F)c1cccc(NC(=O)Oc2ccccc2)c1 ZINC000217761865 CI For-Sale Unstable RAF1 20 43 CC(F)(F)c1cccc(NC(=O)Oc2ccccc2)c1 ZINC000217761865 CI For-Sale Unstable FAAH 25 51 CC(F)(F)c1cccc(NC(=O)Oc2ccccc2)c1 ZINC000217761865 CI For-Sale Unstable EPHX2 18 40 CC(F)(F)c1cccc(NC(=O)Oc2ccccc2)c1 ZINC000217761865 CI For-Sale Unstable Q8MMZ8_EIMTE 24 43 CC(F)(F)c1cccc(NC(=O)Oc2ccccc2)c1 ZINC000217761865 CI For-Sale Unstable AKR1C3 31 41 CC(F)(F)c1cccc(NC(=O)Oc2ccccc2)c1 ZINC000217761865 CI For-Sale Unstable AKR1C2 25 41 CC(F)(F)c1cccc(NC(=O)Oc2ccccc2)c1 ZINC000217761865 CI For-Sale Unstable KCNK3 103 45 CC(F)(F)c1cccc(NC(=O)Oc2ccccc2)c1 ZINC000217761865 CI For-Sale Unstable KCNK9 75 38 CC(F)(F)c1cccc(NC(=O)Oc2ccccc2)c1 ZINC000217761865 CI For-Sale Unstable PDS 58 47 O=C(CCC(=O)c1ccccc1)NC[C@H]1CCCN1c1nccs1 ZINC000217761890 EF For-Sale Unstable PREP 17 40 COc1cccc(C2CC(N[C@@H]3CCN4CCC[C@@H]34)C2)c1 ZINC000217761908 CF For-Sale Unstable EBP 22 40 CCCCn1c(C)c(C(=O)OCC)c2cc(OC(C)C)ccc21 ZINC000217761954 DJ In-Stock Unstable CNR1 0 45 CCCCn1c(C)c(C(=O)OCC)c2cc(OC(C)C)ccc21 ZINC000217761954 DJ In-Stock Unstable CNR2 15 45 CCCCn1c(C)c(C(=O)OCC)c2cc(OC(C)C)ccc21 ZINC000217761954 DJ In-Stock Unstable PLA2G2A 56 49 COC(=O)C[C@H](c1ccc(OC(C)C)cc1)c1c(O)c2ccccc2oc1=O ZINC000217761967 GH In-Stock Unstable NQO1 45 56 COc1cccc(C2CC(N[C@H]3CCN4CCC[C@@H]34)C2)c1 ZINC000217761993 CF For-Sale Unstable EBP 22 40 COC(=O)C[C@@H](c1ccc(OC(C)C)cc1)c1c(O)c2ccccc2oc1=O ZINC000217762056 GH In-Stock Unstable NQO1 52 56 O=C(N/C=C/c1ccccc1F)N1CCN(Cc2ccccc2)CC1 ZINC000217762057 EG For-Sale Unstable DRD2 17 43 O=C(N/C=C/c1ccccc1F)N1CCN(Cc2ccccc2)CC1 ZINC000217762057 EG For-Sale Unstable DRD4 43 40 O=C(N/C=C/c1ccccc1F)N1CCN(Cc2ccccc2)CC1 ZINC000217762057 EG For-Sale Unstable ACHE 21 40 O=C(N/C=C/c1ccccc1F)N1CCN(Cc2ccccc2)CC1 ZINC000217762057 EG For-Sale Unstable CHRM3 17 41 O=C(N/C=C/c1ccccc1F)N1CCN(Cc2ccccc2)CC1 ZINC000217762057 EG For-Sale Unstable SIGMAR1 55 45 O=C(N/C=C/c1ccccc1F)N1CCN(Cc2ccccc2)CC1 ZINC000217762057 EG For-Sale Unstable CCR3 22 45 O=C(N/C=C/c1ccccc1F)N1CCN(Cc2ccccc2)CC1 ZINC000217762057 EG For-Sale Unstable FAAH 31 50 O=C(N/C=C/c1ccccc1F)N1CCN(Cc2ccccc2)CC1 ZINC000217762057 EG For-Sale Unstable MGLL 0 43 CCOC(=O)c1c(C)n(CCOC)c2ccc(OC(C)C)cc12 ZINC000217762087 DH In-Stock Unstable PLA2G2A 47 40 O=C(O)/C=C\c1cccc(CN2CC(=O)NC(=O)C2)c1 ZINC000217762107 CC For-Sale Unstable AKR1C3 30 40 CN1CCN(C(=O)N/C=C/c2ccccc2F)CC1 ZINC000217762162 CD For-Sale Unstable HRH4 20 40 O=C(C[C@@H]1NC(=O)N(Cc2ccc3c(c2)OCO3)C1=O)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217762163 ID In-Stock Unstable NOS2 81 37 CCOC(=O)c1c(C)n(CC(C)C)c2ccc(OC(C)C)cc12 ZINC000217762199 DJ In-Stock Unstable PLA2G2A 51 37 COc1ccc2c(c1)CCC[C@@H]2NC[C@@H]1CN(C)CCO1 ZINC000217762272 CD On-Demand Unstable EBP 29 44 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OC(C)C)cc12 ZINC000217762297 FJ In-Stock Unstable PPARG 30 44 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OC(C)C)cc12 ZINC000217762297 FJ In-Stock Unstable ALOX5AP 86 34 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OC(C)C)cc12 ZINC000217762297 FJ In-Stock Unstable PLA2G2A 122 55 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OC(C)C)cc12 ZINC000217762297 FJ In-Stock Unstable PLA2G2E 0 41 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OC(C)C)cc12 ZINC000217762297 FJ In-Stock Unstable PLA2G10 63 38 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OC(C)C)cc12 ZINC000217762297 FJ In-Stock Unstable PLA2G2F 56 38 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OC(C)C)cc12 ZINC000217762297 FJ In-Stock Unstable PLA2G2D 54 34 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OC(C)C)cc12 ZINC000217762297 FJ In-Stock Unstable PLA2G5 43 38 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OC(C)C)cc12 ZINC000217762297 FJ In-Stock Unstable PTGES2 63 35 C[C@H]1CCCCN1[C@H](C)c1ccc(O)cc1 ZINC000217762322 BG For-Sale Unstable CHRM2 27 41 Cc1cc(NC(=O)c2ccsc2)ccc1/C=C\C(=O)O ZINC000217762348 CG For-Sale Unstable KCNK3 95 55 Cc1cc(NC(=O)c2ccsc2)ccc1/C=C\C(=O)O ZINC000217762348 CG For-Sale Unstable KCNK9 49 39 COc1ccc2c(c1)CCC[C@@H]2NC[C@H]1CN(C)CCO1 ZINC000217762351 CD On-Demand Unstable EBP 29 44 O=C(N/C=C/c1ccccc1F)NC1CCCCCCCCCCC1 ZINC000217762359 EK For-Sale Unstable EPHX2 26 48 CC(C)CNC(=S)NCCc1c[nH]c2ccccc12 ZINC000217762363 CF On-Demand Unstable EDNRB 29 47 CC(C)CNC(=S)NCCc1c[nH]c2ccccc12 ZINC000217762363 CF On-Demand Unstable EDNRA 47 40 CC(C)CNC(=S)NCCc1c[nH]c2ccccc12 ZINC000217762363 CF On-Demand Unstable TACR1 26 52 CC(C)CNC(=S)NCCc1c[nH]c2ccccc12 ZINC000217762363 CF On-Demand Unstable MC4R 19 46 CC(C)CNC(=S)NCCc1c[nH]c2ccccc12 ZINC000217762363 CF On-Demand Unstable CCKAR 34 46 CC(C)CNC(=S)NCCc1c[nH]c2ccccc12 ZINC000217762363 CF On-Demand Unstable MPO 42 45 CC(C)CNC(=S)NCCc1c[nH]c2ccccc12 ZINC000217762363 CF On-Demand Unstable BRS3 42 43 CC(C)CNC(=S)NCCc1c[nH]c2ccccc12 ZINC000217762363 CF On-Demand Unstable NMBR 44 48 CC(C)CNC(=S)NCCc1c[nH]c2ccccc12 ZINC000217762363 CF On-Demand Unstable MMP2 21 40 CC(C)CNC(=S)NCCc1c[nH]c2ccccc12 ZINC000217762363 CF On-Demand Unstable MMP8 30 40 CC(C)CNC(=S)NCCc1c[nH]c2ccccc12 ZINC000217762363 CF On-Demand Unstable MMP14 49 37 CC(C)CNC(=S)NCCc1c[nH]c2ccccc12 ZINC000217762363 CF On-Demand Unstable GRPR 61 34 CC(C)CNC(=S)NCCc1c[nH]c2ccccc12 ZINC000217762363 CF On-Demand Unstable CCKBR 29 41 CC(C)CNC(=S)NCCc1c[nH]c2ccccc12 ZINC000217762363 CF On-Demand Unstable GHSR 52 38 CC(C)CNC(=S)NCCc1c[nH]c2ccccc12 ZINC000217762363 CF On-Demand Unstable ALOX15 23 46 CC(C)CNC(=S)NCCc1c[nH]c2ccccc12 ZINC000217762363 CF On-Demand Unstable MMP9 18 57 CC(C)CNC(=S)NCCc1c[nH]c2ccccc12 ZINC000217762363 CF On-Demand Unstable KISS1R 53 31 O=C(N[C@@H]1C[C@@H]1c1ccccc1)[C@H]1C[C@H]1C(=O)O ZINC000217762405 BD On-Demand Unstable EPHX2 23 50 CCOC(=O)c1c(C)n(CCc2ccccc2)c2ccc(OC(C)C)cc12 ZINC000217762407 FK In-Stock Unstable CNR1 0 43 CCOC(=O)c1c(C)n(CCc2ccccc2)c2ccc(OC(C)C)cc12 ZINC000217762407 FK In-Stock Unstable PLA2G4A 20 42 CCOC(=O)c1c(C)n(CCc2ccccc2)c2ccc(OC(C)C)cc12 ZINC000217762407 FK In-Stock Unstable PLA2G2A 97 46 CCOC(=O)c1c(C)n(CCc2ccccc2)c2ccc(OC(C)C)cc12 ZINC000217762407 FK In-Stock Unstable PTGDS 40 35 O=C(N/C=C/c1ccccc1F)NCCN1CCOCC1 ZINC000217762446 CD For-Sale Unstable DRD4 43 34 O=C(N/C=C/c1ccccc1F)NCCN1CCOCC1 ZINC000217762446 CD For-Sale Unstable CASR 43 34 O=C(N/C=C/c1ccccc1F)NCCN1CCOCC1 ZINC000217762446 CD For-Sale Unstable PLD1 45 33 O=C(N/C=C/c1ccccc1F)NCCN1CCOCC1 ZINC000217762446 CD For-Sale Unstable EPHX2 24 50 O=C(N/C=C/c1ccccc1F)NCCN1CCOCC1 ZINC000217762446 CD For-Sale Unstable PLD2 75 33 O=C(N/C=C/c1ccccc1F)NCCN1CCOCC1 ZINC000217762446 CD For-Sale Unstable HPGDS 24 42 O=C(O)[C@H]1C[C@@H]1C(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000217762469 BD For-Sale Unstable EPHX2 23 50 CCOC(=O)c1c(C)n(Cc2cccnc2)c2ccc(OC(C)C)cc12 ZINC000217762505 FI In-Stock Unstable ALOX5AP 66 37 CCOC(=O)c1c(C)n(Cc2cccnc2)c2ccc(OC(C)C)cc12 ZINC000217762505 FI In-Stock Unstable PLA2G2A 70 43 C[C@H]1CCCCN1[C@H](C)Cc1ccc(O)cc1 ZINC000217762532 BG For-Sale Unstable OPRM1 23 40 C[C@H]1CCCCN1[C@H](C)Cc1ccc(O)cc1 ZINC000217762532 BG For-Sale Unstable YARS 57 33 O=C(O)[C@@H]1C[C@H]1C(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000217762548 BD On-Demand Unstable EPHX2 23 50 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccc(Oc2ccccc2)cc1 ZINC000217762603 GI For-Sale Unstable GRIN2B 19 41 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccc(Oc2ccccc2)cc1 ZINC000217762603 GI For-Sale Unstable LTA4H 38 40 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccc(Oc2ccccc2)cc1 ZINC000217762603 GI For-Sale Unstable HCRTR1 24 41 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccc(Oc2ccccc2)cc1 ZINC000217762603 GI For-Sale Unstable CPT1A 40 35 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccc(Oc2ccccc2)cc1 ZINC000217762603 GI For-Sale Unstable HCRTR2 20 41 CC[C@@H](C)C(=O)NCc1cc(/C=C\C(=O)O)ccc1F ZINC000217762619 CF For-Sale Unstable AKR1C3 36 40 O=C(NC[C@H]1CCCN1c1nccs1)c1ccc(Oc2ccccc2)cc1 ZINC000217762696 GI For-Sale Unstable GRIN2B 19 41 O=C(NC[C@H]1CCCN1c1nccs1)c1ccc(Oc2ccccc2)cc1 ZINC000217762696 GI For-Sale Unstable LTA4H 38 40 O=C(NC[C@H]1CCCN1c1nccs1)c1ccc(Oc2ccccc2)cc1 ZINC000217762696 GI For-Sale Unstable HCRTR1 24 41 O=C(NC[C@H]1CCCN1c1nccs1)c1ccc(Oc2ccccc2)cc1 ZINC000217762696 GI For-Sale Unstable CPT1A 40 35 O=C(NC[C@H]1CCCN1c1nccs1)c1ccc(Oc2ccccc2)cc1 ZINC000217762696 GI For-Sale Unstable HCRTR2 20 41 CC[C@H](C)C(=O)NCc1cc(/C=C\C(=O)O)ccc1F ZINC000217762706 CF For-Sale Unstable AKR1C3 36 40 COC(=O)c1ccc(OCc2ccccc2)c(NS(C)(=O)=O)c1 ZINC000217762712 EE On-Demand Unstable PPIA 45 37 COC(=O)c1ccc(OCc2ccccc2)c(NS(C)(=O)=O)c1 ZINC000217762712 EE On-Demand Unstable PTGER1 44 39 COC(=O)c1ccc(OCc2ccccc2)c(NS(C)(=O)=O)c1 ZINC000217762712 EE On-Demand Unstable ADAMTS4 37 42 COC(=O)c1ccc(OCc2ccccc2)c(NS(C)(=O)=O)c1 ZINC000217762712 EE On-Demand Unstable KLK_PIG 42 32 C[C@H]1CCCCN1[C@H](C)CCc1ccc(O)cc1 ZINC000217762732 BH For-Sale Unstable HRH3 24 40 O=C(N/C=C/c1ccccc1F)NCCN1CCNCC1 ZINC000217762759 CD For-Sale Unstable DRD4 41 32 O=C(N/C=C/c1ccccc1F)NCCN1CCNCC1 ZINC000217762759 CD For-Sale Unstable PLD1 63 35 O=C(N/C=C/c1ccccc1F)NCCN1CCNCC1 ZINC000217762759 CD For-Sale Unstable PLD2 98 35 O=C(N/C=C/c1ccccc1F)NCCN1CCNCC1 ZINC000217762759 CD For-Sale Unstable PFG6PD 0 43 CCC(CC)C(=O)NCc1cc(/C=C\C(=O)O)ccc1F ZINC000217762790 CF For-Sale Unstable AKR1C3 28 40 CCOc1ccc2ccccc2c1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217762801 GI For-Sale Unstable HCN1 43 32 CCOc1ccc2ccccc2c1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217762801 GI For-Sale Unstable HCN4 40 31 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccccc2COc2ccccc2)CC1 ZINC000217762810 HK On-Demand Unstable HTR2A 18 49 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccccc2COc2ccccc2)CC1 ZINC000217762810 HK On-Demand Unstable GRIN2B 46 40 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccccc2COc2ccccc2)CC1 ZINC000217762810 HK On-Demand Unstable CPT1A 45 37 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccccc2COc2ccccc2)CC1 ZINC000217762810 HK On-Demand Unstable SLC18A3 52 49 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccccc2COc2ccccc2)CC1 ZINC000217762810 HK On-Demand Unstable WNT3A 46 33 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccccc2COc2ccccc2)CC1 ZINC000217762810 HK On-Demand Unstable L3MBTL3 62 42 O=C(O)[C@@H]1CN(CCN2CCOCC2)CCN(C2CCCC2)C1 ZINC000217762836 EC In-Stock Unstable SLC6A1 75 36 Cc1ccc(CNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217762869 CH For-Sale Unstable ANPEP 16 40 CCOc1ccc2ccccc2c1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217762878 GI For-Sale Unstable HCN1 43 32 CCOc1ccc2ccccc2c1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217762878 GI For-Sale Unstable HCN4 40 31 Brc1ccccc1C1CC(N[C@@H]2CCN3CCC[C@@H]23)C1 ZINC000217762883 EH For-Sale Unstable SLC18A3 28 50 CCOc1ccc(-n2c(S[C@@H](C(N)=O)c3ccc(F)cc3)nnc2-c2cccnc2)cc1 ZINC000217762928 II On-Demand Unstable VCP 49 33 Brc1ccccc1C1CC(N[C@H]2CCN3CCC[C@@H]23)C1 ZINC000217762953 EH For-Sale Unstable SLC18A3 28 50 CC(C)CN(c1ccc(Cl)cc1CBr)C1CCCC1 ZINC000217762993 EK For-Sale Unstable NOS2 17 42 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccccc1Oc1ccccc1 ZINC000217763000 GI For-Sale Unstable HCRTR1 34 40 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccccc1Oc1ccccc1 ZINC000217763000 GI For-Sale Unstable HCRTR2 26 40 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccccc1Oc1ccccc1 ZINC000217763000 GI For-Sale Unstable HCN1 63 34 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccccc1Oc1ccccc1 ZINC000217763000 GI For-Sale Unstable HCN4 50 33 CCC[C@@H](C)Oc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCC ZINC000217763002 EK In-Stock Unstable PLA2G2A 35 40 CCOc1ccc(-n2c(S[C@H](C(N)=O)c3ccc(F)cc3)nnc2-c2cccnc2)cc1 ZINC000217763030 II On-Demand Unstable VCP 49 33 COc1cc([C@@H](C)N2CCCC[C@@H]2C)ccc1O ZINC000217763051 BG For-Sale Unstable PNLIP 0 47 COc1cc([C@@H](C)N2CCCC[C@@H]2C)ccc1O ZINC000217763051 BG For-Sale Unstable N1L 0 48 COc1cc([C@@H](C)N2CCCC[C@@H]2C)ccc1O ZINC000217763051 BG For-Sale Unstable SLC22A3 0 44 CCC[C@H](C)Oc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCC ZINC000217763083 EK In-Stock Unstable PLA2G2A 35 40 O=C(NC[C@H]1CCCN1c1nccs1)c1ccccc1Oc1ccccc1 ZINC000217763084 GI For-Sale Unstable HCRTR1 34 40 O=C(NC[C@H]1CCCN1c1nccs1)c1ccccc1Oc1ccccc1 ZINC000217763084 GI For-Sale Unstable HCRTR2 26 40 O=C(NC[C@H]1CCCN1c1nccs1)c1ccccc1Oc1ccccc1 ZINC000217763084 GI For-Sale Unstable HCN1 63 34 O=C(NC[C@H]1CCCN1c1nccs1)c1ccccc1Oc1ccccc1 ZINC000217763084 GI For-Sale Unstable HCN4 50 33 O=C(O)/C=C\c1cccc(NC(=O)Cn2cncn2)n1 ZINC000217763118 CC For-Sale Unstable HIS3 47 34 COc1ccc(CNC(=O)CN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@H]23)cc1 ZINC000217763149 IG In-Stock Unstable SCN9A 0 51 COc1ccc(CNC(=O)CN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@H]23)cc1 ZINC000217763149 IG In-Stock Unstable CA9 15 40 C[C@H]1CCCCN1[C@H](C)c1ccc2ccccc2c1O ZINC000217763167 CI For-Sale Unstable HRH3 0 40 O=C(N/C=C/c1ccccc1F)NCCCN1CCOCC1 ZINC000217763191 DD For-Sale Unstable HTR1A 22 42 O=C(N/C=C/c1ccccc1F)NCCCN1CCOCC1 ZINC000217763191 DD For-Sale Unstable DRD3 54 38 O=C(N/C=C/c1ccccc1F)NCCCN1CCOCC1 ZINC000217763191 DD For-Sale Unstable TACR2 28 42 O=C(N/C=C/c1ccccc1F)NCCCN1CCOCC1 ZINC000217763191 DD For-Sale Unstable CCR3 22 40 O=C(N/C=C/c1ccccc1F)NCCCN1CCOCC1 ZINC000217763191 DD For-Sale Unstable CHRNA7 25 43 O=C(N/C=C/c1ccccc1F)NCCCN1CCOCC1 ZINC000217763191 DD For-Sale Unstable EPHX2 26 44 CCCCn1c(C)c(C(=O)OCC)c2cc(O[C@@H](C)CCC)ccc21 ZINC000217763196 EK In-Stock Unstable PLA2G2A 48 47 O=C(O)/C=C\c1cccc(NC(=O)c2cccc(Cl)c2)n1 ZINC000217763198 DG For-Sale Anodyne GRM5 25 50 O=C(O)/C=C\c1cccc(NC(=O)c2cccc(Cl)c2)n1 ZINC000217763198 DG For-Sale Anodyne LUCI_LUCLA 34 50 O=C(O)/C=C\c1cccc(NC(=O)c2cccc(Cl)c2)n1 ZINC000217763198 DG For-Sale Anodyne KCNK3 77 49 O=C(O)/C=C\c1cccc(NC(=O)c2cccc(Cl)c2)n1 ZINC000217763198 DG For-Sale Anodyne KCNK9 37 46 O=C(CCCCc1ccccc1)NC[C@@H]1CCCN1c1nccs1 ZINC000217763217 EH For-Sale Unstable PREP 57 44 O=C(CCCCc1ccccc1)NC[C@@H]1CCCN1c1nccs1 ZINC000217763217 EH For-Sale Unstable FAAH 59 41 O=C(CCCCc1ccccc1)NC[C@@H]1CCCN1c1nccs1 ZINC000217763217 EH For-Sale Unstable CES1 60 38 O=C(CCCCc1ccccc1)NC[C@@H]1CCCN1c1nccs1 ZINC000217763217 EH For-Sale Unstable CES1D 42 29 CCc1ccc(/C=C\C(=O)N2CC(=O)NC(=O)C2)cc1 ZINC000217763230 CC For-Sale Unstable GPR183 0 43 COc1ccc(CNC(=O)CN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@@H]23)cc1 ZINC000217763235 IG In-Stock Unstable SCN9A 0 51 COc1ccc(CNC(=O)CN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@@H]23)cc1 ZINC000217763235 IG In-Stock Unstable CA9 15 40 CCCCNC(=S)NCCCCCCC(C)C ZINC000217763257 CH For-Sale Unstable NOD1 45 40 CCCCn1c(C)c(C(=O)OCC)c2cc(O[C@H](C)CCC)ccc21 ZINC000217763275 EK In-Stock Unstable PLA2G2A 48 47 COc1ccc(C(=O)C2CCN(C(=O)c3cscn3)CC2)cc1 ZINC000217763288 EF On-Demand Unstable SLC18A3 33 51 COc1ccc(C(=O)C2CCN(C(=O)c3cscn3)CC2)cc1 ZINC000217763288 EF On-Demand Unstable L3MBTL3 50 36 COc1ccc(C(=O)C2CCN(C(=O)c3cscn3)CC2)cc1 ZINC000217763288 EF On-Demand Unstable TRPC6 51 46 COc1ccc(C(=O)C2CCN(C(=O)c3cscn3)CC2)cc1 ZINC000217763288 EF On-Demand Unstable TRPC3 24 46 O=C(CCCCc1ccccc1)NC[C@H]1CCCN1c1nccs1 ZINC000217763301 EH For-Sale Unstable PREP 57 44 O=C(CCCCc1ccccc1)NC[C@H]1CCCN1c1nccs1 ZINC000217763301 EH For-Sale Unstable FAAH 59 41 O=C(CCCCc1ccccc1)NC[C@H]1CCCN1c1nccs1 ZINC000217763301 EH For-Sale Unstable CES1 60 38 O=C(CCCCc1ccccc1)NC[C@H]1CCCN1c1nccs1 ZINC000217763301 EH For-Sale Unstable CES1D 42 29 CN(N)C(=O)c1cc2ccccc2s1 ZINC000217763315 BD For-Sale Unstable LTB4R 16 45 CN(N)C(=O)c1cc2ccccc2s1 ZINC000217763315 BD For-Sale Unstable PIN1 28 40 O=C1CCC(=O)N1C1C[C@@H]2CC[C@H](C1)N2C(=O)Cc1c(F)cccc1Cl ZINC000217763323 GF In-Stock Unstable P2RX7 18 44 COc1ccc(/C=C\C(=O)O)cc1NC(=O)c1ccco1 ZINC000217763341 CF For-Sale Unstable PTGER2 0 41 COc1ccc(/C=C\C(=O)O)cc1NC(=O)c1ccco1 ZINC000217763341 CF For-Sale Unstable NR1H4 20 41 COc1ccc(/C=C\C(=O)O)cc1NC(=O)c1ccco1 ZINC000217763341 CF For-Sale Unstable AKR1C3 40 40 O=C(CC[C@@H]1NC(=O)N(Cc2ccc3c(c2)OCO3)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217763355 ID In-Stock Unstable MCHR1 22 44 C[C@H]1CCCCN1[C@H](C)c1cccc(O)c1 ZINC000217763359 BG For-Sale Unstable OPRM1 15 44 CS(=O)(=O)c1ccc(CC(=O)NCc2nnc(-c3ccccc3)o2)cc1 ZINC000217763404 FD In-Stock Unstable CA7 16 46 CS(=O)(=O)c1ccc(CC(=O)NCc2nnc(-c3ccccc3)o2)cc1 ZINC000217763404 FD In-Stock Unstable CTSF 45 33 CS(=O)(=O)c1ccc(CC(=O)NCc2nnc(-c3ccccc3)o2)cc1 ZINC000217763404 FD In-Stock Unstable CA5B 47 46 CS(=O)(=O)c1ccc(CC(=O)NCc2nnc(-c3ccccc3)o2)cc1 ZINC000217763404 FD In-Stock Unstable CA5A 49 46 CS(=O)(=O)c1ccc(CC(=O)NCc2nnc(-c3ccccc3)o2)cc1 ZINC000217763404 FD In-Stock Unstable E1 0 45 CS(=O)(=O)c1ccc(CC(=O)NCc2nnc(-c3ccccc3)o2)cc1 ZINC000217763404 FD In-Stock Unstable MT-CO2 40 38 COc1ccc(/C=C/C(=O)NC[C@@H]2CCCN2c2nccs2)cc1OC ZINC000217763406 FF For-Sale Unstable ACKR3 68 37 CN(Cc1ccccc1)C(=O)N/C=C/c1ccccc1F ZINC000217763427 CH For-Sale Unstable TSPO 17 40 CN(Cc1ccccc1)C(=O)N/C=C/c1ccccc1F ZINC000217763427 CH For-Sale Unstable LIMK2 32 42 COc1ccc(/C=C\C(=O)O)cc1NC(=O)CC(C)C ZINC000217763429 CF For-Sale Unstable TUBB1 43 39 COc1ccc(/C=C\C(=O)O)cc1NC(=O)CC(C)C ZINC000217763429 CF For-Sale Unstable AKR1C3 40 43 O=C(N[C@H]1CCC[C@@H](C(F)(F)F)C1)[C@@H](Cl)c1ccccc1 ZINC000217763440 DI For-Sale Unstable AMY2 43 30 COc1ccc(/C=C/C(=O)NC[C@H]2CCCN2c2nccs2)cc1OC ZINC000217763482 FF For-Sale Unstable ACKR3 68 37 Cc1c(F)cccc1C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217763489 EI On-Demand Unstable HTR2A 24 46 Cc1c(F)cccc1C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217763489 EI On-Demand Unstable HTR2C 15 46 Cc1c(F)cccc1C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217763489 EI On-Demand Unstable HSD11B1 21 77 Cc1c(F)cccc1C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217763489 EI On-Demand Unstable SLC18A3 50 49 Cc1c(F)cccc1C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217763489 EI On-Demand Unstable WNT3A 46 32 Cc1c(F)cccc1C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217763489 EI On-Demand Unstable L3MBTL3 83 40 Cc1ccc(C(=O)Nc2ncc(/C=C\C(=O)O)s2)cc1C ZINC000217763521 DG For-Sale Unstable SCD1 27 48 O=C(N[C@@H]1CCC[C@@H](C(F)(F)F)C1)[C@@H](Cl)c1ccccc1 ZINC000217763525 DI For-Sale Unstable AMY2 43 30 CN1CC[C@H](N2CCC[C@@H]([C@@H]3CCCN3)C2)C1 ZINC000217763640 BD For-Sale Unstable MBTD1 0 41 Cc1c(C(=O)O)[nH]c(C=O)c1F ZINC000217763641 AC For-Sale Unstable HISB 41 39 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCCCN1CCOCC1 ZINC000217763659 IC In-Stock Unstable HTR1A 19 43 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCCCN1CCOCC1 ZINC000217763659 IC In-Stock Unstable DRD2 15 45 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCCCN1CCOCC1 ZINC000217763659 IC In-Stock Unstable HTR1D 64 39 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCCCN1CCOCC1 ZINC000217763659 IC In-Stock Unstable HTR1B 61 38 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCCCN1CCOCC1 ZINC000217763659 IC In-Stock Unstable SLC6A4 0 45 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCCCN1CCOCC1 ZINC000217763659 IC In-Stock Unstable TACR1 17 44 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCCCN1CCOCC1 ZINC000217763659 IC In-Stock Unstable MC4R 42 37 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCCCN1CCOCC1 ZINC000217763659 IC In-Stock Unstable TACR2 24 42 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCCCN1CCOCC1 ZINC000217763659 IC In-Stock Unstable CCR4 29 45 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCCCN1CCOCC1 ZINC000217763659 IC In-Stock Unstable MC5R 34 41 Cc1csc(NC(=O)N/C=C/c2ccccc2F)n1 ZINC000217763677 CG For-Sale Unstable GCK 17 48 COc1cc(C)ccc1C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217763719 FH On-Demand Unstable SLC18A3 39 50 COc1cc(C)ccc1C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217763719 FH On-Demand Unstable L3MBTL3 59 39 O=C(COCC(F)(F)C(F)F)NCc1nc2cc(F)ccc2[nH]1 ZINC000217763743 EE In-Stock Unstable FABK 0 42 CSc1ccc(C[C@H](N)C(=O)O)cc1Cl ZINC000217763751 BE For-Sale Unstable OPRM1 21 42 CSc1ccc(C[C@H](N)C(=O)O)cc1Cl ZINC000217763751 BE For-Sale Unstable OPRD1 23 42 CSc1ccc(C[C@H](N)C(=O)O)cc1Cl ZINC000217763751 BE For-Sale Unstable CACNA2D1 59 49 CSc1ccc(C[C@H](N)C(=O)O)cc1Cl ZINC000217763751 BE For-Sale Unstable TPH1 76 33 CSc1ccc(C[C@H](N)C(=O)O)cc1Cl ZINC000217763751 BE For-Sale Unstable YARS 42 35 CSc1ccc(C[C@H](N)C(=O)O)cc1Cl ZINC000217763751 BE For-Sale Unstable KIF11 31 43 O=C(CC[C@@H]1NC(=O)N(Cc2ccc3c(c2)OCO3)C1=O)N[C@H](CO)c1ccccc1 ZINC000217763757 ID In-Stock Unstable MCHR1 23 46 CCC[C@@H](C)Oc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217763763 GK In-Stock Unstable PTGS2 0 44 CCC[C@@H](C)Oc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217763763 GK In-Stock Unstable PPARG 30 44 CCC[C@@H](C)Oc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217763763 GK In-Stock Unstable ALOX5AP 76 32 CCC[C@@H](C)Oc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217763763 GK In-Stock Unstable PLA2G2A 132 52 CCC[C@@H](C)Oc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217763763 GK In-Stock Unstable PLA2G2D 42 32 CCC[C@@H](C)Oc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217763763 GK In-Stock Unstable PTGES2 53 33 CN(Cc1cccc(/C=C\C(=O)O)c1)C(=O)c1cccs1 ZINC000217763786 DG For-Sale Unstable HSD17B2 38 50 CN(Cc1cccc(/C=C\C(=O)O)c1)C(=O)c1cccs1 ZINC000217763786 DG For-Sale Unstable HCAR2 0 43 CSc1ccc(C[C@@H](N)C(=O)O)cc1Cl ZINC000217763829 BE For-Sale Unstable OPRM1 21 42 CSc1ccc(C[C@@H](N)C(=O)O)cc1Cl ZINC000217763829 BE For-Sale Unstable OPRD1 23 42 CSc1ccc(C[C@@H](N)C(=O)O)cc1Cl ZINC000217763829 BE For-Sale Unstable CACNA2D1 59 49 CSc1ccc(C[C@@H](N)C(=O)O)cc1Cl ZINC000217763829 BE For-Sale Unstable TPH1 76 33 CSc1ccc(C[C@@H](N)C(=O)O)cc1Cl ZINC000217763829 BE For-Sale Unstable YARS 42 35 CSc1ccc(C[C@@H](N)C(=O)O)cc1Cl ZINC000217763829 BE For-Sale Unstable KIF11 31 43 CCC[C@H](C)Oc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217763844 GK In-Stock Unstable PTGS2 0 44 CCC[C@H](C)Oc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217763844 GK In-Stock Unstable PPARG 29 44 CCC[C@H](C)Oc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217763844 GK In-Stock Unstable ALOX5AP 76 32 CCC[C@H](C)Oc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217763844 GK In-Stock Unstable PLA2G2A 111 52 CCC[C@H](C)Oc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217763844 GK In-Stock Unstable PLA2G2D 42 32 CCC[C@H](C)Oc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217763844 GK In-Stock Unstable PTGES2 53 33 C[C@@H]1C[C@@H]1C(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217763866 CE For-Sale Unstable GRM3 16 41 C[C@@H]1C[C@@H]1C(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217763866 CE For-Sale Unstable NR1H4 40 37 C[C@@H]1C[C@@H]1C(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217763866 CE For-Sale Unstable AKR1C3 40 39 O=C1CCC(=O)N1C1C[C@@H]2CC[C@H](C1)N2C(=O)Cc1ccc(-c2ccccc2)cc1 ZINC000217763876 HH In-Stock Unstable MGLL 0 40 COc1ccc(CNC(=O)CCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@H]23)cc1OC ZINC000217763880 JH In-Stock Unstable TSHR 50 34 COc1ccc(CNC(=O)CCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@H]23)cc1OC ZINC000217763880 JH In-Stock Unstable SCN9A 0 42 COc1cccc(NC(=O)N/C=C/c2ccccc2F)c1 ZINC000217763887 CH For-Sale Unstable CCR3 15 40 COc1cccc(NC(=O)N/C=C/c2ccccc2F)c1 ZINC000217763887 CH For-Sale Unstable MTNR1A 22 45 COc1cccc(NC(=O)N/C=C/c2ccccc2F)c1 ZINC000217763887 CH For-Sale Unstable MTNR1B 28 45 COc1cccc(NC(=O)N/C=C/c2ccccc2F)c1 ZINC000217763887 CH For-Sale Unstable TAAR1 36 50 COc1cccc(NC(=O)N/C=C/c2ccccc2F)c1 ZINC000217763887 CH For-Sale Unstable TLR4 16 40 COc1cccc(NC(=O)N/C=C/c2ccccc2F)c1 ZINC000217763887 CH For-Sale Unstable KCNK3 83 47 COc1cccc(NC(=O)N/C=C/c2ccccc2F)c1 ZINC000217763887 CH For-Sale Unstable KCNK9 69 38 CCOc1ccccc1/C=C\C(=O)N1CC(=O)NC(=O)C1 ZINC000217763920 CC For-Sale Unstable PTGER2 0 40 CCOc1ccccc1/C=C\C(=O)N1CC(=O)NC(=O)C1 ZINC000217763920 CC For-Sale Unstable HCN1 51 35 CCOc1ccccc1/C=C\C(=O)N1CC(=O)NC(=O)C1 ZINC000217763920 CC For-Sale Unstable HCN4 42 33 O=C(CCC(F)(F)F)N1CCN(Cc2nnc[nH]2)CC1 ZINC000217763940 CC In-Stock Unstable ETHR 56 36 CCC[C@@H](C)Oc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCc1ccccc1 ZINC000217763946 GK In-Stock Unstable CNR1 0 42 CCC[C@@H](C)Oc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCc1ccccc1 ZINC000217763946 GK In-Stock Unstable PLA2G2A 78 43 C[C@H]1C[C@@H]1C(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217763961 CE For-Sale Unstable GRM3 16 41 C[C@H]1C[C@@H]1C(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217763961 CE For-Sale Unstable NR1H4 40 37 C[C@H]1C[C@@H]1C(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217763961 CE For-Sale Unstable AKR1C3 40 39 COc1ccc(CNC(=O)CCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@@H]23)cc1OC ZINC000217763964 JH In-Stock Unstable TSHR 50 34 COc1ccc(CNC(=O)CCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@@H]23)cc1OC ZINC000217763964 JH In-Stock Unstable SCN9A 0 42 O=C(CCC(F)(F)F)NC[C@H]1CCCN1c1nccs1 ZINC000217763969 DF For-Sale Unstable ETHR 40 39 O=C(N/C=C/c1ccccc1F)Nc1cc(Cl)ccc1O ZINC000217763990 DH For-Sale Anodyne KCNMA1 26 49 CCC[C@H](C)Oc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCc1ccccc1 ZINC000217764040 GK In-Stock Unstable CNR1 0 42 CCC[C@H](C)Oc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCc1ccccc1 ZINC000217764040 GK In-Stock Unstable PLA2G2A 75 43 O=C(CCC(F)(F)F)NC[C@@H]1CCCN1c1nccs1 ZINC000217764055 DF For-Sale Unstable ETHR 40 39 C[C@@H]1CN([C@H]2CCCc3cc(O)ccc32)C[C@@H](C)O1 ZINC000217764069 CF For-Sale Unstable DRD5 19 45 C[C@@H]1CN([C@H]2CCCc3cc(O)ccc32)C[C@@H](C)O1 ZINC000217764069 CF For-Sale Unstable HSD17B1 52 37 COc1ccc(C(OCCCC(=O)O)(c2ccccc2)c2ccccc2)cc1 ZINC000217764104 GJ For-Sale Unstable EDNRA 21 40 COc1ccc(C(OCCCC(=O)O)(c2ccccc2)c2ccccc2)cc1 ZINC000217764104 GJ For-Sale Unstable PLA2G4B 54 36 COc1ccc(C(OCCCC(=O)O)(c2ccccc2)c2ccccc2)cc1 ZINC000217764104 GJ For-Sale Unstable KIF11 15 45 COc1ccc(C(OCCCC(=O)O)(c2ccccc2)c2ccccc2)cc1 ZINC000217764104 GJ For-Sale Unstable TK2 29 41 COc1cccc(F)c1C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217764117 FH On-Demand Unstable HTR2A 23 45 COc1cccc(F)c1C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217764117 FH On-Demand Unstable HSD11B1 18 68 COc1cccc(F)c1C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217764117 FH On-Demand Unstable CCR5 34 44 COc1cccc(F)c1C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217764117 FH On-Demand Unstable SLC18A3 42 53 COc1cccc(F)c1C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217764117 FH On-Demand Unstable WNT3A 51 32 COc1cccc(F)c1C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217764117 FH On-Demand Unstable L3MBTL3 66 35 COc1cccc(F)c1C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217764117 FH On-Demand Unstable ACKR3 44 31 C[C@@H](Cc1ccccc1Cl)NC(=O)[C@@H]1C[C@@H](O)CN1 ZINC000217764141 CD For-Sale Unstable CTSC 23 42 CCC[C@@H](C)Oc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1cccnc1 ZINC000217764143 GK In-Stock Unstable PPARG 19 40 CCC[C@@H](C)Oc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1cccnc1 ZINC000217764143 GK In-Stock Unstable PLA2G2A 63 41 O=C(N/C=C/c1ccccc1F)Nc1nccs1 ZINC000217764218 CG For-Sale Anodyne MAP 0 47 O=C(N/C=C/c1ccccc1F)Nc1nccs1 ZINC000217764218 CG For-Sale Anodyne MAP1 120 47 C[C@H](Cc1ccccc1Cl)NC(=O)[C@@H]1C[C@@H](O)CN1 ZINC000217764224 CD For-Sale Unstable CTSC 23 42 COc1ccc(OC)c(CN[C@@H]2CCN3CCC[C@@H]23)c1 ZINC000217764228 CE For-Sale Unstable TACR1 37 53 CCC[C@H](C)Oc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1cccnc1 ZINC000217764247 GK In-Stock Unstable PPARG 19 40 CCC[C@H](C)Oc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1cccnc1 ZINC000217764247 GK In-Stock Unstable PLA2G2A 63 41 COc1ccc(OC)c(-c2cc(C(=O)NC[C@@H]3CCCN4CCCC[C@H]34)[nH]n2)c1 ZINC000217764286 GG In-Stock Unstable ALPL 50 35 C[C@@H](Cc1ccccc1Cl)NC(=O)[C@H]1C[C@@H](O)CN1 ZINC000217764293 CD On-Demand Unstable CTSC 23 42 COc1ccc(OC)c(CN[C@H]2CCN3CCC[C@@H]23)c1 ZINC000217764308 CE For-Sale Unstable TACR1 37 53 CSc1cccc(Cl)c1C[C@H](N)C(=O)O ZINC000217764326 BE For-Sale Unstable CACNA2D1 66 45 CSc1cccc(Cl)c1C[C@H](N)C(=O)O ZINC000217764326 BE For-Sale Unstable GRIA3 56 40 CSc1cccc(Cl)c1C[C@H](N)C(=O)O ZINC000217764326 BE For-Sale Unstable GRIA1 39 40 CSc1cccc(Cl)c1C[C@H](N)C(=O)O ZINC000217764326 BE For-Sale Unstable GRIA2 46 40 CSc1cccc(Cl)c1C[C@H](N)C(=O)O ZINC000217764326 BE For-Sale Unstable GRIA4 46 40 CSc1cccc(Cl)c1C[C@H](N)C(=O)O ZINC000217764326 BE For-Sale Unstable GRIK1 30 40 CSc1cccc(Cl)c1C[C@H](N)C(=O)O ZINC000217764326 BE For-Sale Unstable KIF11 40 42 CSc1cccc(NC(=O)N/C=C/c2ccccc2F)c1 ZINC000217764332 DI For-Sale Unstable KCNK3 53 35 C[C@H](Cc1ccccc1Cl)NC(=O)[C@H]1C[C@@H](O)CN1 ZINC000217764378 CD On-Demand Unstable CTSC 23 42 O=C(CCCn1cccn1)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217764405 ED In-Stock Unstable CHRNA4 33 59 CSc1cccc(Cl)c1C[C@@H](N)C(=O)O ZINC000217764408 BE For-Sale Unstable CACNA2D1 66 45 CSc1cccc(Cl)c1C[C@@H](N)C(=O)O ZINC000217764408 BE For-Sale Unstable GRIA3 56 40 CSc1cccc(Cl)c1C[C@@H](N)C(=O)O ZINC000217764408 BE For-Sale Unstable GRIA1 39 40 CSc1cccc(Cl)c1C[C@@H](N)C(=O)O ZINC000217764408 BE For-Sale Unstable GRIA2 46 40 CSc1cccc(Cl)c1C[C@@H](N)C(=O)O ZINC000217764408 BE For-Sale Unstable GRIA4 46 40 CSc1cccc(Cl)c1C[C@@H](N)C(=O)O ZINC000217764408 BE For-Sale Unstable GRIK1 30 40 CSc1cccc(Cl)c1C[C@@H](N)C(=O)O ZINC000217764408 BE For-Sale Unstable KIF11 40 42 COC(=O)c1ccc(NS(C)(=O)=O)cc1O ZINC000217764420 BC For-Sale Unstable CA7 15 57 O=C(N/C=C/c1ccccc1F)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217764435 IG For-Sale Unstable LPL 42 42 O=C(N/C=C/c1ccccc1F)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217764435 IG For-Sale Unstable PKM 43 41 O=C(N/C=C/c1ccccc1F)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217764435 IG For-Sale Unstable LIPG 17 42 C=CCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CC ZINC000217764472 CH In-Stock Unstable PLA2G2A 51 39 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217764540 ED For-Sale Unstable CA2 110 55 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217764540 ED For-Sale Unstable CA1 94 55 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217764540 ED For-Sale Unstable CA7 55 54 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217764540 ED For-Sale Unstable CA5B 66 54 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217764540 ED For-Sale Unstable CA4 78 55 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217764540 ED For-Sale Unstable CA5A 70 54 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217764540 ED For-Sale Unstable CA14 39 52 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217764540 ED For-Sale Unstable CA12 70 53 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217764540 ED For-Sale Unstable CA9 79 54 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217764540 ED For-Sale Unstable CYNT 24 43 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217764540 ED For-Sale Unstable MTCA1 45 52 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217764540 ED For-Sale Unstable P96878_MYCTU 58 52 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217764540 ED For-Sale Unstable NAMPT 41 38 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217764540 ED For-Sale Unstable A6YCJ1_9METZ 22 40 N[C@@H]1CCN([C@@H]2C[C@@H]2c2ccccc2)C1 ZINC000217764551 BD On-Demand Unstable SLC18A3 39 40 C=CCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCC ZINC000217764579 DI In-Stock Unstable PLA2G2A 46 44 O=C(N/C=C/c1ccccc1F)Nc1cccnc1Cl ZINC000217764661 CH For-Sale Anodyne G2YM83_BOTF4 45 32 C=CCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCOC ZINC000217764697 DG In-Stock Unstable PLA2G2A 48 42 CC[C@@H](C)N(C)CCNCc1ccc2c(c1)NC(=O)CO2 ZINC000217764742 CD On-Demand Unstable HTR1B 17 40 N[C@@H]1CCN([C@@H]2C[C@@H]2c2ccccc2)C1=O ZINC000217764745 BD For-Sale Unstable SMO 30 40 C[C@@H](N[C@@H]1CCN2CCC[C@@H]12)c1cccc(F)c1 ZINC000217764778 BF For-Sale Unstable CHRNA10 25 40 C=CCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CC(C)C ZINC000217764804 DI In-Stock Unstable PLA2G2A 44 38 N[C@@H]1CCN([C@H]2C[C@@H]2c2ccccc2)C1=O ZINC000217764821 BD For-Sale Unstable SMO 30 40 CC[C@H](C)N(C)CCNCc1ccc2c(c1)NC(=O)CO2 ZINC000217764834 CD On-Demand Unstable HTR1B 17 40 C[C@H](N[C@@H]1CCN2CCC[C@@H]12)c1cccc(F)c1 ZINC000217764856 BF For-Sale Unstable CHRNA10 25 40 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1cc(C(N)=O)ccc1F ZINC000217764863 CH For-Sale Unstable TRPM8 18 57 CSc1ccc(Cl)cc1C[C@H](N)C(=O)O ZINC000217764890 BE For-Sale Unstable CACNA2D1 65 50 CSc1ccc(Cl)cc1C[C@H](N)C(=O)O ZINC000217764890 BE For-Sale Unstable TPH1 41 31 CSc1ccc(Cl)cc1C[C@H](N)C(=O)O ZINC000217764890 BE For-Sale Unstable KIF11 31 42 C=CCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCc1ccccc1 ZINC000217764922 FJ In-Stock Unstable CNR1 0 41 C=CCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCc1ccccc1 ZINC000217764922 FJ In-Stock Unstable ALOX5AP 56 35 C=CCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCc1ccccc1 ZINC000217764922 FJ In-Stock Unstable PLA2G2A 102 45 C[C@@H](N[C@H]1CCN2CCC[C@@H]12)c1cccc(F)c1 ZINC000217764926 BF For-Sale Unstable CHRNA10 25 40 CC(C)(C)CC(=O)Nc1ccc(/C=C\C(=O)O)cc1F ZINC000217764945 CG For-Sale Unstable MMP1 0 41 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1cc(C(N)=O)ccc1F ZINC000217764950 CH For-Sale Unstable TRPM8 18 57 CSc1ccc(Cl)cc1C[C@@H](N)C(=O)O ZINC000217764970 BE For-Sale Unstable CACNA2D1 65 50 CSc1ccc(Cl)cc1C[C@@H](N)C(=O)O ZINC000217764970 BE For-Sale Unstable TPH1 41 31 CSc1ccc(Cl)cc1C[C@@H](N)C(=O)O ZINC000217764970 BE For-Sale Unstable KIF11 31 42 Nc1nc(-c2cccnc2)co1 ZINC000217765001 AD For-Sale Unstable CYP2E1 53 39 Nc1nc(-c2cccnc2)co1 ZINC000217765001 AD For-Sale Unstable CYP2A6 53 45 C[C@H](N[C@H]1CCN2CCC[C@@H]12)c1cccc(F)c1 ZINC000217765010 BF For-Sale Unstable CHRNA10 25 40 COc1ccc(C)cc1/C=C\C(=O)N1CC(=O)NC(=O)C1 ZINC000217765017 CC For-Sale Unstable GPR183 0 40 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1cc(C(N)=O)ccc1F ZINC000217765032 CH For-Sale Unstable TRPM8 18 57 Cc1cc(NC(=O)c2ccoc2C)ccc1/C=C\C(=O)O ZINC000217765034 CG For-Sale Unstable KCNK3 78 38 Cc1cc(NC(=O)c2ccoc2C)ccc1/C=C\C(=O)O ZINC000217765034 CG For-Sale Unstable KCNK9 45 36 C=CCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1cccnc1 ZINC000217765040 FI In-Stock Unstable ALOX5AP 91 40 C=CCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1cccnc1 ZINC000217765040 FI In-Stock Unstable PLA2G2A 75 42 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1cc(C(N)=O)ccc1F ZINC000217765118 CH For-Sale Unstable TRPM8 18 57 Cc1cc(NC(=O)c2occc2C)ccc1/C=C\C(=O)O ZINC000217765121 CG For-Sale Unstable KCNK3 51 35 O=C(O)Cc1ccc2nc(Cl)c(Cl)nc2c1 ZINC000217765181 CF In-Stock Unstable HPSE 48 37 O=C(O)Cc1ccc2nc(Cl)c(Cl)nc2c1 ZINC000217765181 CF In-Stock Unstable RPS6KB2 24 44 COC(=O)c1nc(NC(=O)CNc2ccc3c(cc2=O)[C@@H](NC(C)=O)CCc2cc(OC)c(OC)c(OC)c2-3)sc1C ZINC000217765183 KG In-Stock Unstable TUBA1A 17 62 COC(=O)c1nc(NC(=O)CNc2ccc3c(cc2=O)[C@@H](NC(C)=O)CCc2cc(OC)c(OC)c(OC)c2-3)sc1C ZINC000217765183 KG In-Stock Unstable TPPP 0 61 Cc1cc(NC(=O)c2ccoc2)ccc1/C=C\C(=O)O ZINC000217765196 CF For-Sale Unstable KCNK3 95 55 Cc1cc(NC(=O)c2ccoc2)ccc1/C=C\C(=O)O ZINC000217765196 CF For-Sale Unstable KCNK9 48 39 CCOC(=O)c1c(C)n(CC)c2ccc(OCC(C)C)cc12 ZINC000217765243 DI In-Stock Unstable PLA2G2A 53 39 Cc1cc(/C=C\C(=O)O)ccc1NC(=O)C1CCCCC1 ZINC000217765283 CH For-Sale Unstable STK17B 40 37 COc1ccc(CN2C(=O)N[C@@H](CC(=O)N[C@H](CO)c3ccccc3)C2=O)cc1OC ZINC000217765291 ID In-Stock Unstable ENPP1 54 31 CCCn1c(C)c(C(=O)OCC)c2cc(OCC(C)C)ccc21 ZINC000217765368 DJ In-Stock Unstable PLA2G2A 49 44 CSc1cc(Cl)cc(C[C@H](N)C(=O)O)c1 ZINC000217765474 BE For-Sale Unstable CACNA2D1 46 48 CSc1cc(Cl)cc(C[C@H](N)C(=O)O)c1 ZINC000217765474 BE For-Sale Unstable TPH1 57 33 CCCCn1c(C)c(C(=O)OCC)c2cc(OCC(C)C)ccc21 ZINC000217765477 EJ In-Stock Unstable PLA2G2A 60 52 CCn1cc(C(=O)NC[C@@H]2CCCN2c2nccs2)c(=O)c2ccc(C)nc21 ZINC000217765514 GF For-Sale Unstable CNR2 15 47 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable ACE 56 55 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable CNR1 29 65 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable MME 146 46 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable ANPEP 67 39 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable CNR2 15 54 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable CMA1 29 43 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable PTPN2 36 43 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable KLK3 32 44 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable CTSB 35 40 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable PAPA1_CARPA 44 39 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable CTSL 27 40 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable CPA1 54 44 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable TIMP3 52 36 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable LPAR1 45 52 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable SELP 30 42 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable TACR3 18 40 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable NAALAD2 31 45 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable CAPNS1 52 35 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable MMP2 18 45 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable MMP3 26 45 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable GRIA1 52 46 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable ECE1 47 41 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable HLA-DRB1 46 43 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable SOAT1 25 69 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable HDAC1 18 48 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable FAAH 43 46 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable PTPN1 27 44 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable CAPN1 54 44 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable MMP9 22 41 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable CAPN2 39 44 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable EPHX2 15 55 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable ACE2 99 46 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable MC1R 47 37 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable PIN1 42 48 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable MMP1 22 44 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable FPR1 78 48 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable CTRB_BOVIN 52 40 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable NPR 42 37 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable AMP1_PLAFQ 20 45 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable LPAR3 72 52 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable FABP3 41 51 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable BLA1_STEMA 79 46 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable FABP1 15 44 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable NOD1 104 50 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable OXER1 38 41 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217765527 IK For-Sale Unstable SLCO2A1 45 33 NC[C@@H]1CCN([C@@H]2C[C@@H]2c2ccccc2)C1 ZINC000217765533 BD On-Demand Unstable SLC18A3 41 35 CC(=O)NCC(=O)NCc1cc(/C=C\C(=O)O)ccc1F ZINC000217765545 CC For-Sale Unstable P2RX7 15 40 CCN(Cc1ccccc1)[C@@H](C(=O)NC1CC1)c1ccc(F)cc1 ZINC000217765546 EH On-Demand Unstable SIGMAR1 17 42 CCN(Cc1ccccc1)[C@@H](C(=O)NC1CC1)c1ccc(F)cc1 ZINC000217765546 EH On-Demand Unstable BACE1 15 40 CSc1cc(Cl)cc(C[C@@H](N)C(=O)O)c1 ZINC000217765556 BE For-Sale Unstable CACNA2D1 46 48 CSc1cc(Cl)cc(C[C@@H](N)C(=O)O)c1 ZINC000217765556 BE For-Sale Unstable TPH1 57 33 CCOC(=O)c1c(C)n(CCOC)c2ccc(OCC(C)C)cc12 ZINC000217765573 EH In-Stock Unstable PLA2G2A 52 42 CCn1cc(C(=O)NC[C@H]2CCCN2c2nccs2)c(=O)c2ccc(C)nc21 ZINC000217765589 GF For-Sale Unstable CNR2 15 47 CC(C)CCNC(=O)c1ccc(NC(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc1 ZINC000217765592 HG In-Stock Unstable CHRNA4 28 45 CCN(Cc1ccccc1)[C@H](C(=O)NC1CC1)c1ccc(F)cc1 ZINC000217765623 EH On-Demand Unstable SIGMAR1 17 42 CCN(Cc1ccccc1)[C@H](C(=O)NC1CC1)c1ccc(F)cc1 ZINC000217765623 EH On-Demand Unstable BACE1 15 40 COCC(=O)NCc1cc(/C=C\C(=O)O)ccc1F ZINC000217765624 CD For-Sale Unstable AKR1C3 39 40 CCOC(=O)c1c(C)n(CC(C)C)c2ccc(OCC(C)C)cc12 ZINC000217765682 EJ In-Stock Unstable PLA2G2A 55 39 N[C@@H]1CC[C@H](c2ccccc2)C[C@@H]1Cc1cccc(Br)c1 ZINC000217765695 EJ For-Sale Unstable VACHT_TETCF 0 44 Cc1ccc(C(=O)Nc2cc(/C=C\C(=O)O)ccc2C)o1 ZINC000217765704 CG For-Sale Unstable S1PR4 26 41 O=C1CN(C(=O)/C=C\c2ccc3c(c2)OCO3)CC(=O)N1 ZINC000217765727 CB For-Sale Unstable ITGAL 21 42 O=C1CN(C(=O)/C=C\c2ccc3c(c2)OCO3)CC(=O)N1 ZINC000217765727 CB For-Sale Unstable DYRK2 76 39 N[C@H]1CC[C@H](c2ccccc2)C[C@@H]1Cc1cccc(Br)c1 ZINC000217765771 EJ For-Sale Unstable VACHT_TETCF 0 44 O=C1CCC(=O)N1C1C[C@@H]2CC[C@H](C1)N2S(=O)(=O)c1ccccc1 ZINC000217765778 ED In-Stock Unstable CMA1 0 40 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCC(C)C)cc12 ZINC000217765783 FK In-Stock Unstable PTGS2 22 45 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCC(C)C)cc12 ZINC000217765783 FK In-Stock Unstable PPARG 29 42 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCC(C)C)cc12 ZINC000217765783 FK In-Stock Unstable PLA2G1B 40 37 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCC(C)C)cc12 ZINC000217765783 FK In-Stock Unstable ALOX5AP 95 42 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCC(C)C)cc12 ZINC000217765783 FK In-Stock Unstable PLA2G2A 155 53 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCC(C)C)cc12 ZINC000217765783 FK In-Stock Unstable PLA2G2E 0 41 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCC(C)C)cc12 ZINC000217765783 FK In-Stock Unstable PLA2G10 75 37 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCC(C)C)cc12 ZINC000217765783 FK In-Stock Unstable PLA2G2F 59 37 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCC(C)C)cc12 ZINC000217765783 FK In-Stock Unstable PLA2G2D 71 37 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCC(C)C)cc12 ZINC000217765783 FK In-Stock Unstable PLA2G5 48 41 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCC(C)C)cc12 ZINC000217765783 FK In-Stock Unstable PTGES2 55 35 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCC(C)C)cc12 ZINC000217765783 FK In-Stock Unstable PDS 59 39 O=C1CN(C(=O)/C=C\c2ccc([N+](=O)[O-])cc2)CC(=O)N1 ZINC000217765813 CC For-Sale Unstable SLC27A4 48 31 N[C@@H]1CC[C@@H](c2ccccc2)C[C@@H]1Cc1cccc(Br)c1 ZINC000217765844 EJ For-Sale Unstable VACHT_TETCF 0 44 CCCOc1ccc(CCC(=O)N2CCC(N3CCC(OC)CC3)CC2)cc1 ZINC000217765866 GH In-Stock Unstable CHRM2 48 45 CCCOc1ccc(CCC(=O)N2CCC(N3CCC(OC)CC3)CC2)cc1 ZINC000217765866 GH In-Stock Unstable CCR3 24 43 CCCOc1ccc(CCC(=O)N2CCC(N3CCC(OC)CC3)CC2)cc1 ZINC000217765866 GH In-Stock Unstable PLA2G4B 58 37 CCCOc1ccc(CCC(=O)N2CCC(N3CCC(OC)CC3)CC2)cc1 ZINC000217765866 GH In-Stock Unstable L3MBTL3 56 34 Fc1ccc(SCc2ccc(-n3ccnc3)cc2)cc1 ZINC000217765885 CI On-Demand Unstable CYP2C19 17 41 Fc1ccc(SCc2ccc(-n3ccnc3)cc2)cc1 ZINC000217765885 CI On-Demand Unstable CYP17A1 0 44 O=C(CC[C@@H]1NC(=O)N(Cc2cccc(Cl)c2)C1=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217765890 JE In-Stock Unstable CHRNA4 28 48 CCOC(=O)c1c(C)n(CCc2ccccc2)c2ccc(OCC(C)C)cc12 ZINC000217765897 GK In-Stock Unstable CNR1 0 41 CCOC(=O)c1c(C)n(CCc2ccccc2)c2ccc(OCC(C)C)cc12 ZINC000217765897 GK In-Stock Unstable ALOX5AP 49 36 CCOC(=O)c1c(C)n(CCc2ccccc2)c2ccc(OCC(C)C)cc12 ZINC000217765897 GK In-Stock Unstable PLA2G2A 105 45 CCOC(=O)c1c(C)n(CCc2ccccc2)c2ccc(OCC(C)C)cc12 ZINC000217765897 GK In-Stock Unstable PDS 59 38 COC(=O)c1ccccc1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217765898 EE For-Sale Unstable HCN1 56 32 COC(=O)c1ccccc1C(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217765898 EE For-Sale Unstable HCN4 48 31 O=C1CN(C(=O)/C=C\c2ccc(Br)cc2)CC(=O)N1 ZINC000217765899 DC For-Sale Unstable GPR183 0 52 N[C@H]1CC[C@@H](c2ccccc2)C[C@@H]1Cc1cccc(Br)c1 ZINC000217765905 EJ For-Sale Unstable VACHT_TETCF 0 44 CN(C(=O)OCc1ccccc1)[C@](C)(C(=O)O)c1cccc2ccccc12 ZINC000217765963 FI For-Sale Unstable SLC12A5 43 31 COC(=O)c1ccccc1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217765973 EE For-Sale Unstable HCN1 56 32 COC(=O)c1ccccc1C(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217765973 EE For-Sale Unstable HCN4 48 31 COC1CCN(C2CCN(C(=O)CCc3cccc(Cl)c3)CC2)CC1 ZINC000217765977 FG In-Stock Unstable CHRM2 42 38 COC1CCN(C2CCN(C(=O)CCc3cccc(Cl)c3)CC2)CC1 ZINC000217765977 FG In-Stock Unstable HRH1 20 42 COC1CCN(C2CCN(C(=O)CCc3cccc(Cl)c3)CC2)CC1 ZINC000217765977 FG In-Stock Unstable CCR3 47 42 COC1CCN(C2CCN(C(=O)CCc3cccc(Cl)c3)CC2)CC1 ZINC000217765977 FG In-Stock Unstable C3AR1 35 42 COC1CCN(C2CCN(C(=O)CCc3cccc(Cl)c3)CC2)CC1 ZINC000217765977 FG In-Stock Unstable L3MBTL3 63 37 N[C@@H]1CC[C@H](c2ccccc2)C[C@@H]1Cc1ccc(Br)cc1 ZINC000217765978 EJ For-Sale Unstable VACHT_TETCF 0 41 CCCCCNC(=O)N/C=C/c1ccccc1F ZINC000217765989 CG For-Sale Unstable EPHX2 25 42 CCCCCNC(=O)N/C=C/c1ccccc1F ZINC000217765989 CG For-Sale Unstable ASAH1 93 41 CCCCCNC(=O)N/C=C/c1ccccc1F ZINC000217765989 CG For-Sale Unstable ACAT 0 46 CCOC(=O)c1c(C)n(Cc2cccnc2)c2ccc(OCC(C)C)cc12 ZINC000217766007 FJ In-Stock Unstable ALOX5AP 86 39 CCOC(=O)c1c(C)n(Cc2cccnc2)c2ccc(OCC(C)C)cc12 ZINC000217766007 FJ In-Stock Unstable PLA2G2A 76 44 COc1ccc2c(c1)[C@@]1(C(=O)N2)[C@H](C(=O)c2cccs2)[C@@H](c2ccc(Cl)cc2)CN1C ZINC000217766008 JJ In-Stock Unstable SLC6A1 0 47 COc1ccc([C@@H](C)N2CCC[C@@H](C)C2)c(O)c1 ZINC000217766038 BG For-Sale Unstable RORC 47 44 N[C@H]1CC[C@H](c2ccccc2)C[C@@H]1Cc1ccc(Br)cc1 ZINC000217766066 EJ For-Sale Unstable VACHT_TETCF 0 41 O=C(NC[C@@H]1CCCN1c1nccs1)c1cccc(F)c1 ZINC000217766094 DF For-Sale Unstable DRD2 15 41 O=C(NC[C@@H]1CCCN1c1nccs1)c1cccc(F)c1 ZINC000217766094 DF For-Sale Unstable ACKR3 46 33 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CC ZINC000217766114 DI In-Stock Unstable ALOX5 15 41 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CC ZINC000217766114 DI In-Stock Unstable PTGS2 0 41 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CC ZINC000217766114 DI In-Stock Unstable PLA2G2A 71 52 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CC ZINC000217766114 DI In-Stock Unstable PLA2G4B 77 34 N[C@@H]1CC[C@@H](c2ccccc2)C[C@@H]1Cc1ccc(Br)cc1 ZINC000217766156 EJ For-Sale Unstable VACHT_TETCF 0 41 O=C(NC[C@H]1CCCN1c1nccs1)c1cccc(F)c1 ZINC000217766177 DF For-Sale Unstable DRD2 15 41 O=C(NC[C@H]1CCCN1c1nccs1)c1cccc(F)c1 ZINC000217766177 DF For-Sale Unstable ACKR3 46 33 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCC ZINC000217766201 DJ In-Stock Unstable CNR1 0 47 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCC ZINC000217766201 DJ In-Stock Unstable CNR2 15 46 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCC ZINC000217766201 DJ In-Stock Unstable PLA2G2A 68 56 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCC ZINC000217766201 DJ In-Stock Unstable PLA2G4B 76 34 CCOC(=O)[C@@H]1CCCN(C(=O)N/C=C/c2ccccc2F)C1 ZINC000217766209 DF For-Sale Unstable SLC6A1 108 37 N[C@H]1CC[C@@H](c2ccccc2)C[C@@H]1Cc1ccc(Br)cc1 ZINC000217766234 EJ For-Sale Unstable VACHT_TETCF 0 41 NNC(=O)c1ccc(CC(=O)O)cc1 ZINC000217766238 AB For-Sale Unstable CA2 15 50 NNC(=O)c1ccc(CC(=O)O)cc1 ZINC000217766238 AB For-Sale Unstable SRD5A2 0 47 NNC(=O)c1ccc(CC(=O)O)cc1 ZINC000217766238 AB For-Sale Unstable AOC2 0 47 NNC(=O)c1ccc(CC(=O)O)cc1 ZINC000217766238 AB For-Sale Unstable CAN2 0 54 NNC(=O)c1ccc(CC(=O)O)cc1 ZINC000217766238 AB For-Sale Unstable H9B8T9_CAPHI 29 50 CCOC(=O)[C@H]1CCCN(C(=O)N/C=C/c2ccccc2F)C1 ZINC000217766273 DF For-Sale Unstable SLC6A1 108 37 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCCC ZINC000217766308 EK In-Stock Unstable CNR1 15 44 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCCC ZINC000217766308 EK In-Stock Unstable CNR2 18 47 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCCC ZINC000217766308 EK In-Stock Unstable PLA2G2A 75 61 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCCC ZINC000217766308 EK In-Stock Unstable PLA2G4B 60 34 Cc1ccc(C(=O)Nc2cccc(/C=C\C(=O)O)n2)cc1 ZINC000217766383 CF For-Sale Unstable GRM5 20 41 Cc1ccc(C(=O)Nc2cccc(/C=C\C(=O)O)n2)cc1 ZINC000217766383 CF For-Sale Unstable MAP3K5 56 42 Cc1ccc(C(=O)Nc2cccc(/C=C\C(=O)O)n2)cc1 ZINC000217766383 CF For-Sale Unstable KCNK3 70 39 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCCN(C)C1CC1 ZINC000217766402 CG For-Sale Unstable TRPM8 0 40 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCOC ZINC000217766408 EH In-Stock Unstable CNR1 0 45 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCOC ZINC000217766408 EH In-Stock Unstable PTGS2 0 41 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCOC ZINC000217766408 EH In-Stock Unstable CNR2 15 45 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCOC ZINC000217766408 EH In-Stock Unstable PLA2G2A 65 53 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCOC ZINC000217766408 EH In-Stock Unstable PLA2G4B 53 32 COc1ccc(CNC(=O)c2sc3cc(Cl)ccc3c2Cl)cc1C(=O)O ZINC000217766444 HJ On-Demand Unstable PPARA 18 41 COc1ccc(CNC(=O)c2sc3cc(Cl)ccc3c2Cl)cc1C(=O)O ZINC000217766444 HJ On-Demand Unstable COLA 60 38 COc1ccc(CNC(=O)c2sc3cc(Cl)ccc3c2Cl)cc1C(=O)O ZINC000217766444 HJ On-Demand Unstable CPT1A 58 38 COc1ccc(CNC(=O)c2sc3cc(Cl)ccc3c2Cl)cc1C(=O)O ZINC000217766444 HJ On-Demand Unstable PPARD 18 41 COc1ccc(CNC(=O)c2sc3cc(Cl)ccc3c2Cl)cc1C(=O)O ZINC000217766444 HJ On-Demand Unstable UL54 61 36 COc1ccc(CNC(=O)c2sc3cc(Cl)ccc3c2Cl)cc1C(=O)O ZINC000217766444 HJ On-Demand Unstable CPT1B 55 36 COc1ccc(CNC(=O)c2sc3cc(Cl)ccc3c2Cl)cc1C(=O)O ZINC000217766444 HJ On-Demand Unstable U38 0 44 COc1ccc(/C=C\C(=O)O)cc1NC(=O)C1CCC1 ZINC000217766464 CF For-Sale Unstable NR1H4 27 40 COc1ccc(/C=C\C(=O)O)cc1NC(=O)C1CCC1 ZINC000217766464 CF For-Sale Unstable TUBB1 42 39 COc1ccc(/C=C\C(=O)O)cc1NC(=O)C1CCC1 ZINC000217766464 CF For-Sale Unstable STK17B 49 44 COc1ccc(/C=C\C(=O)O)cc1NC(=O)C1CCC1 ZINC000217766464 CF For-Sale Unstable STK17A 16 42 COc1ccc(/C=C\C(=O)O)cc1NC(=O)C1CCC1 ZINC000217766464 CF For-Sale Unstable ABCG2 15 41 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCCN(C)C1CC1 ZINC000217766492 CG For-Sale Unstable TRPM8 0 40 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CC(C)C ZINC000217766522 EJ In-Stock Unstable PLA2G2A 61 49 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CC(C)C ZINC000217766522 EJ In-Stock Unstable PLA2G4B 54 33 COc1ccc(/C=C\C(=O)O)cc1NC(=O)C1CCCC1 ZINC000217766544 CF For-Sale Unstable NR1H4 28 42 COc1ccc(/C=C\C(=O)O)cc1NC(=O)C1CCCC1 ZINC000217766544 CF For-Sale Unstable TUBB1 42 39 COc1ccc(/C=C\C(=O)O)cc1NC(=O)C1CCCC1 ZINC000217766544 CF For-Sale Unstable STK17B 51 47 COc1ccc(/C=C\C(=O)O)cc1NC(=O)C1CCCC1 ZINC000217766544 CF For-Sale Unstable STK17A 17 44 COc1ccc(/C=C\C(=O)O)cc1NC(=O)C1CCCC1 ZINC000217766544 CF For-Sale Unstable ABCG2 15 41 O=S(=O)(C[C@H]1CCCN1)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000217766547 CD For-Sale Unstable GRIA4 15 42 O=S(=O)(C[C@H]1CCCN1)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000217766547 CD For-Sale Unstable CHRNA10 29 40 COC(=O)c1ccc(OC)c(S(=O)(=O)NCCN2CCOCC2)c1 ZINC000217766549 FC On-Demand Unstable HTR1A 15 40 COC(=O)c1ccc(OC)c(S(=O)(=O)NCCN2CCOCC2)c1 ZINC000217766549 FC On-Demand Unstable CNR1 18 47 COC(=O)c1ccc(OC)c(S(=O)(=O)NCCN2CCOCC2)c1 ZINC000217766549 FC On-Demand Unstable DRD4 41 32 COC(=O)c1ccc(OC)c(S(=O)(=O)NCCN2CCOCC2)c1 ZINC000217766549 FC On-Demand Unstable HTR4 20 40 COC(=O)c1ccc(OC)c(S(=O)(=O)NCCN2CCOCC2)c1 ZINC000217766549 FC On-Demand Unstable CASR 18 42 COC(=O)c1ccc(OC)c(S(=O)(=O)NCCN2CCOCC2)c1 ZINC000217766549 FC On-Demand Unstable COLA 52 34 COC(=O)c1ccc(OC)c(S(=O)(=O)NCCN2CCOCC2)c1 ZINC000217766549 FC On-Demand Unstable CPT1A 49 34 COC(=O)c1ccc(OC)c(S(=O)(=O)NCCN2CCOCC2)c1 ZINC000217766549 FC On-Demand Unstable CPT2 40 33 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCCN(C)C1CC1 ZINC000217766583 CG For-Sale Unstable TRPM8 0 40 O=C(O)CCc1ccc2nc(Cl)c(Cl)nc2c1 ZINC000217766585 CF In-Stock Unstable TBXA2R 42 33 O=C(O)CCc1ccc2nc(Cl)c(Cl)nc2c1 ZINC000217766585 CF In-Stock Unstable FFAR1 84 47 O=C(O)CCc1ccc2nc(Cl)c(Cl)nc2c1 ZINC000217766585 CF In-Stock Unstable FFAR4 52 38 COc1ccc(-c2coc3ccc(OCC(=O)N4CCc5cc(OC)c(OC)cc5C4)cc23)cc1 ZINC000217766586 JK In-Stock Unstable ALDH2 82 38 COc1ccc(-c2coc3ccc(OCC(=O)N4CCc5cc(OC)c(OC)cc5C4)cc23)cc1 ZINC000217766586 JK In-Stock Unstable HTR1B 17 41 COc1ccc(-c2coc3ccc(OCC(=O)N4CCc5cc(OC)c(OC)cc5C4)cc23)cc1 ZINC000217766586 JK In-Stock Unstable ABCB1B 56 34 COc1ccc(-c2coc3ccc(OCC(=O)N4CCc5cc(OC)c(OC)cc5C4)cc23)cc1 ZINC000217766586 JK In-Stock Unstable ABCB1 23 58 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217766620 FK In-Stock Unstable ALOX5 26 45 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217766620 FK In-Stock Unstable CNR1 0 45 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217766620 FK In-Stock Unstable PTGS2 0 44 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217766620 FK In-Stock Unstable PPARG 32 42 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217766620 FK In-Stock Unstable PTGER2 0 43 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217766620 FK In-Stock Unstable PPARA 20 41 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217766620 FK In-Stock Unstable CNR2 18 43 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217766620 FK In-Stock Unstable PLA2G1B 50 39 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217766620 FK In-Stock Unstable ALOX5AP 97 40 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217766620 FK In-Stock Unstable PLA2G2A 172 62 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217766620 FK In-Stock Unstable PLA2G2E 0 42 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217766620 FK In-Stock Unstable PLA2G4B 79 38 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217766620 FK In-Stock Unstable PLA2G10 40 37 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217766620 FK In-Stock Unstable PLA2G2F 47 34 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217766620 FK In-Stock Unstable PLA2G2D 54 34 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217766620 FK In-Stock Unstable PTGDR 15 42 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217766620 FK In-Stock Unstable PLA2G5 48 42 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1ccccc1 ZINC000217766620 FK In-Stock Unstable PTGES2 52 32 O=S(=O)(C[C@H]1CCCN1)N[C@H]1C[C@@H]1c1ccccc1 ZINC000217766629 CD For-Sale Unstable GRIA4 15 42 O=S(=O)(C[C@H]1CCCN1)N[C@H]1C[C@@H]1c1ccccc1 ZINC000217766629 CD For-Sale Unstable CHRNA10 29 40 COc1ccc(/C=C\C(=O)O)cc1NC(=O)c1cccs1 ZINC000217766637 DG For-Sale Unstable FABP2 0 41 COc1ccc(/C=C\C(=O)O)cc1NC(=O)c1cccs1 ZINC000217766637 DG For-Sale Unstable LTB4R 0 42 COc1ccc(/C=C\C(=O)O)cc1NC(=O)c1cccs1 ZINC000217766637 DG For-Sale Unstable TUBB1 42 36 COc1ccc(/C=C\C(=O)O)cc1NC(=O)c1cccs1 ZINC000217766637 DG For-Sale Unstable KCNK9 15 40 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCCN(C)C1CC1 ZINC000217766654 CG For-Sale Unstable TRPM8 0 40 O=C(CNC(=O)c1ccccc1)NC[C@@H]1CCCN1c1nccs1 ZINC000217766683 ED For-Sale Unstable PREP 20 44 O=C(CNC(=O)c1ccccc1)NC[C@@H]1CCCN1c1nccs1 ZINC000217766683 ED For-Sale Unstable CCR2 18 42 CC[C@@H](NCCc1ccccc1OC)c1ccc(F)cc1 ZINC000217766706 CI On-Demand Unstable LEF 28 45 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2coc3ccccc3c2=O)CC(=O)O4)cc1O ZINC000217766712 JI In-Stock Unstable AKR1B1 0 44 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2coc3ccccc3c2=O)CC(=O)O4)cc1O ZINC000217766712 JI In-Stock Unstable CYP1B1 64 36 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2coc3ccccc3c2=O)CC(=O)O4)cc1O ZINC000217766712 JI In-Stock Unstable CYP1A1 49 44 COC1CCN(C2CCN(C(=O)CCc3ccccc3F)CC2)CC1 ZINC000217766721 EF In-Stock Unstable CHRM2 46 41 COC1CCN(C2CCN(C(=O)CCc3ccccc3F)CC2)CC1 ZINC000217766721 EF In-Stock Unstable CCR3 26 48 COC1CCN(C2CCN(C(=O)CCc3ccccc3F)CC2)CC1 ZINC000217766721 EF In-Stock Unstable L3MBTL3 56 37 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cccc(Oc3ccccc3)c2)CC1 ZINC000217766724 HK On-Demand Unstable HTR2A 18 50 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cccc(Oc3ccccc3)c2)CC1 ZINC000217766724 HK On-Demand Unstable INHA 20 41 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cccc(Oc3ccccc3)c2)CC1 ZINC000217766724 HK On-Demand Unstable GRIN2B 23 47 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cccc(Oc3ccccc3)c2)CC1 ZINC000217766724 HK On-Demand Unstable HRH3 24 40 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cccc(Oc3ccccc3)c2)CC1 ZINC000217766724 HK On-Demand Unstable CCR3 25 40 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cccc(Oc3ccccc3)c2)CC1 ZINC000217766724 HK On-Demand Unstable SLC18A3 66 61 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cccc(Oc3ccccc3)c2)CC1 ZINC000217766724 HK On-Demand Unstable PREP 30 43 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cccc(Oc3ccccc3)c2)CC1 ZINC000217766724 HK On-Demand Unstable SLC9A1 28 40 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cccc(Oc3ccccc3)c2)CC1 ZINC000217766724 HK On-Demand Unstable CFTR 39 48 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cccc(Oc3ccccc3)c2)CC1 ZINC000217766724 HK On-Demand Unstable EPHX2 15 41 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cccc(Oc3ccccc3)c2)CC1 ZINC000217766724 HK On-Demand Unstable CCR8 24 42 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cccc(Oc3ccccc3)c2)CC1 ZINC000217766724 HK On-Demand Unstable WNT3A 45 33 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cccc(Oc3ccccc3)c2)CC1 ZINC000217766724 HK On-Demand Unstable L3MBTL3 90 50 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCc1ccccc1 ZINC000217766736 GK In-Stock Unstable ALOX5 25 41 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCc1ccccc1 ZINC000217766736 GK In-Stock Unstable CNR1 27 49 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCc1ccccc1 ZINC000217766736 GK In-Stock Unstable PPARG 28 44 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCc1ccccc1 ZINC000217766736 GK In-Stock Unstable PTGER2 0 42 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCc1ccccc1 ZINC000217766736 GK In-Stock Unstable CNR2 21 47 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCc1ccccc1 ZINC000217766736 GK In-Stock Unstable ALOX5AP 61 31 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCc1ccccc1 ZINC000217766736 GK In-Stock Unstable PLA2G2A 107 52 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCc1ccccc1 ZINC000217766736 GK In-Stock Unstable PLA2G4B 71 36 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCc1ccccc1 ZINC000217766736 GK In-Stock Unstable PTGDR 24 44 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCc1ccccc1 ZINC000217766736 GK In-Stock Unstable PTGES 25 41 COc1ccc(Cn2ccc(C)n2)cc1/C=C\C(=O)O ZINC000217766748 CE For-Sale Unstable PTGER2 34 41 COc1ccc(Cn2ccc(C)n2)cc1/C=C\C(=O)O ZINC000217766748 CE For-Sale Unstable PTGER4 18 41 COc1ccc(Cn2ccc(C)n2)cc1/C=C\C(=O)O ZINC000217766748 CE For-Sale Unstable PTGER3 20 41 O[C@@]12C[C@H]3C[C@@H](C1)C(NCc1ccccc1)[C@H](C3)C2 ZINC000217766749 CF In-Stock Unstable HSD11B1 46 44 O=C(CNC(=O)c1ccccc1)NC[C@H]1CCCN1c1nccs1 ZINC000217766784 ED For-Sale Unstable PREP 20 44 O=C(CNC(=O)c1ccccc1)NC[C@H]1CCCN1c1nccs1 ZINC000217766784 ED For-Sale Unstable CCR2 18 42 CC[C@H](NCCc1ccccc1OC)c1ccc(F)cc1 ZINC000217766788 CI On-Demand Unstable LEF 28 45 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2coc3ccccc3c2=O)CC(=O)O4)cc1O ZINC000217766792 JI In-Stock Unstable AKR1B1 0 44 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2coc3ccccc3c2=O)CC(=O)O4)cc1O ZINC000217766792 JI In-Stock Unstable CYP1B1 64 36 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2coc3ccccc3c2=O)CC(=O)O4)cc1O ZINC000217766792 JI In-Stock Unstable CYP1A1 49 44 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1cccnc1 ZINC000217766837 FJ In-Stock Unstable ALOX5AP 87 40 CCCCOc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1cccnc1 ZINC000217766837 FJ In-Stock Unstable PLA2G2A 84 49 O=C(O)/C=C\c1cnc(NC(=O)CCC2CCCCC2)s1 ZINC000217766886 DH For-Sale Unstable CDK5 52 44 C[C@@H]1CCCN([C@H](C)CCc2ccc(O)cc2)C1 ZINC000217766897 BG For-Sale Unstable BIRC2 33 41 C[C@@H](Nc1cccc(C(N)=O)c1)C(=O)OC(C)(C)C ZINC000217766926 CD On-Demand Unstable PARP14 0 47 C[C@@H](Nc1cccc(C(N)=O)c1)C(=O)OC(C)(C)C ZINC000217766926 CD On-Demand Unstable PARP15 0 47 C[C@@H](Nc1cccc(C(N)=O)c1)C(=O)OC(C)(C)C ZINC000217766926 CD On-Demand Unstable MVFR 0 43 C[C@@H](Nc1cccc(C(N)=O)c1)C(=O)OC(C)(C)C ZINC000217766926 CD On-Demand Unstable PARP10 0 47 CCCn1c(C)c(C(=O)OCC)c2cc(OCc3ccccc3)ccc21 ZINC000217766929 FK In-Stock Unstable ALOX5 23 43 CCCn1c(C)c(C(=O)OCC)c2cc(OCc3ccccc3)ccc21 ZINC000217766929 FK In-Stock Unstable CNR1 18 46 CCCn1c(C)c(C(=O)OCC)c2cc(OCc3ccccc3)ccc21 ZINC000217766929 FK In-Stock Unstable MAOB 44 47 CCCn1c(C)c(C(=O)OCC)c2cc(OCc3ccccc3)ccc21 ZINC000217766929 FK In-Stock Unstable PPARG 23 47 CCCn1c(C)c(C(=O)OCC)c2cc(OCc3ccccc3)ccc21 ZINC000217766929 FK In-Stock Unstable CNR2 16 48 CCCn1c(C)c(C(=O)OCC)c2cc(OCc3ccccc3)ccc21 ZINC000217766929 FK In-Stock Unstable ALOX5AP 92 35 CCCn1c(C)c(C(=O)OCC)c2cc(OCc3ccccc3)ccc21 ZINC000217766929 FK In-Stock Unstable PLA2G2A 109 50 CCCn1c(C)c(C(=O)OCC)c2cc(OCc3ccccc3)ccc21 ZINC000217766929 FK In-Stock Unstable FFAR1 53 38 Cc1cc(C)cc(C(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217766941 DG For-Sale Unstable CACNA1I 53 34 c1ccc2c(c1)CC(N[C@@H]1CCN3CCC[C@@H]13)C2 ZINC000217766946 BD For-Sale Unstable VACHT_TETCF 0 43 COC(=O)[C@H](CC(C)C)NC(=O)CCn1cc(C(C)=O)c2ccccc21 ZINC000217766971 FF In-Stock Unstable CNR2 27 47 O=C(O)/C=C\c1cnc(NC(=O)c2c(F)cccc2Cl)s1 ZINC000217767004 EG For-Sale Anodyne JAK1 0 47 O=C(O)/C=C\c1cnc(NC(=O)c2c(F)cccc2Cl)s1 ZINC000217767004 EG For-Sale Anodyne TYK2 27 47 C[C@H](Nc1cccc(C(N)=O)c1)C(=O)OC(C)(C)C ZINC000217767011 CD On-Demand Unstable PARP14 0 47 C[C@H](Nc1cccc(C(N)=O)c1)C(=O)OC(C)(C)C ZINC000217767011 CD On-Demand Unstable PARP15 0 47 C[C@H](Nc1cccc(C(N)=O)c1)C(=O)OC(C)(C)C ZINC000217767011 CD On-Demand Unstable MVFR 0 43 C[C@H](Nc1cccc(C(N)=O)c1)C(=O)OC(C)(C)C ZINC000217767011 CD On-Demand Unstable PARP10 0 47 Cc1cc(C)cc(C(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217767014 DG For-Sale Unstable CACNA1I 53 34 c1ccc2c(c1)CC(N[C@H]1CCN3CCC[C@@H]13)C2 ZINC000217767016 BD For-Sale Unstable VACHT_TETCF 0 43 COC(=O)CCc1ccc2nccnc2c1 ZINC000217767028 BD In-Stock Unstable ECE2 0 44 CCOC(=O)c1c(C)n(CCOC)c2ccc(OCc3ccccc3)cc12 ZINC000217767031 FI In-Stock Unstable ALOX5 18 40 CCOC(=O)c1c(C)n(CCOC)c2ccc(OCc3ccccc3)cc12 ZINC000217767031 FI In-Stock Unstable CNR1 0 41 CCOC(=O)c1c(C)n(CCOC)c2ccc(OCc3ccccc3)cc12 ZINC000217767031 FI In-Stock Unstable MAOB 35 45 CCOC(=O)c1c(C)n(CCOC)c2ccc(OCc3ccccc3)cc12 ZINC000217767031 FI In-Stock Unstable PPARG 20 47 CCOC(=O)c1c(C)n(CCOC)c2ccc(OCc3ccccc3)cc12 ZINC000217767031 FI In-Stock Unstable ALOX5AP 91 34 CCOC(=O)c1c(C)n(CCOC)c2ccc(OCc3ccccc3)cc12 ZINC000217767031 FI In-Stock Unstable NADE 0 43 CCOC(=O)c1c(C)n(CCOC)c2ccc(OCc3ccccc3)cc12 ZINC000217767031 FI In-Stock Unstable PLA2G2A 108 50 CCOC(=O)c1c(C)n(CCOC)c2ccc(OCc3ccccc3)cc12 ZINC000217767031 FI In-Stock Unstable FFAR1 43 35 CC1(C)CC(NC(=O)N/C=C/c2ccccc2F)CC(C)(C)N1 ZINC000217767044 DG For-Sale Unstable ENV 33 42 CC1(C)CC(NC(=O)N/C=C/c2ccccc2F)CC(C)(C)N1 ZINC000217767044 DG For-Sale Unstable EZH2 49 41 CC1(C)CC(NC(=O)N/C=C/c2ccccc2F)CC(C)(C)N1 ZINC000217767044 DG For-Sale Unstable HIV1_ENV 0 42 CN(Cc1cccc(/C=C\C(=O)O)c1)C(=O)c1ccsc1 ZINC000217767083 DG For-Sale Unstable PTGER2 22 43 CN(Cc1cccc(/C=C\C(=O)O)c1)C(=O)c1ccsc1 ZINC000217767083 DG For-Sale Unstable HSD17B2 32 49 CN(Cc1cccc(/C=C\C(=O)O)c1)C(=O)c1ccsc1 ZINC000217767083 DG For-Sale Unstable AKR1C3 34 41 CN(c1ccc(Cl)cc1CBr)C1CCC(C)(C)CC1 ZINC000217767089 EK For-Sale Unstable NOS2 18 40 CN(c1ccc(Cl)cc1CBr)C1CCC(C)(C)CC1 ZINC000217767089 EK For-Sale Unstable NOS3 18 40 COc1ccc(-c2coc3ccc(OCc4ccc(C(=O)OC(C)C)o4)cc23)cc1OC ZINC000217767091 IK In-Stock Unstable ALDH2 77 35 COc1ccc(-c2coc3ccc(OCc4ccc(C(=O)OC(C)C)o4)cc23)cc1OC ZINC000217767091 IK In-Stock Unstable PRKCZ 21 40 COc1ccc(-c2coc3ccc(OCc4ccc(C(=O)OC(C)C)o4)cc23)cc1OC ZINC000217767091 IK In-Stock Unstable PRKCI 0 40 COC1CCN(C2CCN(C(=O)CCc3ccc(SC)cc3)CC2)CC1 ZINC000217767135 GG In-Stock Unstable CHRM2 17 41 COC1CCN(C2CCN(C(=O)CCc3ccc(SC)cc3)CC2)CC1 ZINC000217767135 GG In-Stock Unstable CCR3 21 41 COC1CCN(C2CCN(C(=O)CCc3ccc(SC)cc3)CC2)CC1 ZINC000217767135 GG In-Stock Unstable L3MBTL3 77 36 CCOC(=O)c1c(C)n(CC(C)C)c2ccc(OCc3ccccc3)cc12 ZINC000217767141 FK In-Stock Unstable ALOX5 19 41 CCOC(=O)c1c(C)n(CC(C)C)c2ccc(OCc3ccccc3)cc12 ZINC000217767141 FK In-Stock Unstable MAOB 32 46 CCOC(=O)c1c(C)n(CC(C)C)c2ccc(OCc3ccccc3)cc12 ZINC000217767141 FK In-Stock Unstable EDNRA 0 43 CCOC(=O)c1c(C)n(CC(C)C)c2ccc(OCc3ccccc3)cc12 ZINC000217767141 FK In-Stock Unstable ALOX5AP 92 35 CCOC(=O)c1c(C)n(CC(C)C)c2ccc(OCc3ccccc3)cc12 ZINC000217767141 FK In-Stock Unstable PLA2G2A 88 49 CCOC(=O)c1c(C)n(CC(C)C)c2ccc(OCc3ccccc3)cc12 ZINC000217767141 FK In-Stock Unstable CAPN2 67 33 CCOC(=O)c1c(C)n(CC(C)C)c2ccc(OCc3ccccc3)cc12 ZINC000217767141 FK In-Stock Unstable NPR 44 31 CCOC(=O)c1c(C)n(CC(C)C)c2ccc(OCc3ccccc3)cc12 ZINC000217767141 FK In-Stock Unstable FFAR1 56 38 O=C(O)CCc1ccc2[nH]c(S)nc2c1 ZINC000217767143 BD In-Stock Unstable FFAR1 62 38 CN(Cc1cccc(/C=C\C(=O)O)c1)C(=O)c1ccoc1 ZINC000217767172 CF For-Sale Unstable HSD17B2 25 43 CN(Cc1cccc(/C=C\C(=O)O)c1)C(=O)c1ccoc1 ZINC000217767172 CF For-Sale Unstable AKR1C3 38 40 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccccc2)CC(=O)O4)cc1O ZINC000217767200 II In-Stock Unstable AKR1B1 23 49 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccccc2)CC(=O)O4)cc1O ZINC000217767200 II In-Stock Unstable CYP1B1 75 42 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccccc2)CC(=O)O4)cc1O ZINC000217767200 II In-Stock Unstable CYP1A1 58 49 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccccc2)CC(=O)O4)cc1O ZINC000217767200 II In-Stock Unstable CYP1A2 47 42 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccccc2)CC(=O)O4)cc1O ZINC000217767200 II In-Stock Unstable ABCG2 22 42 O=S(=O)(Cl)c1ccccc1N1CCCC1 ZINC000217767238 BE For-Sale Unstable KCNQ2 67 38 COC(=O)CCc1ccc2[nH]c(S)nc2c1 ZINC000217767243 BD In-Stock Unstable P2RY12 0 46 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767244 GK In-Stock Unstable ALOX5 23 46 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767244 GK In-Stock Unstable MAOA 15 40 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767244 GK In-Stock Unstable MAOB 57 48 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767244 GK In-Stock Unstable PTGS2 0 45 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767244 GK In-Stock Unstable PPARG 32 41 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767244 GK In-Stock Unstable PTGER2 29 40 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767244 GK In-Stock Unstable EDNRA 0 40 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767244 GK In-Stock Unstable PLA2G1B 30 42 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767244 GK In-Stock Unstable ALOX5AP 108 44 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767244 GK In-Stock Unstable PLA2G2A 165 59 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767244 GK In-Stock Unstable PLA2G10 46 38 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767244 GK In-Stock Unstable PLA2G2F 49 35 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767244 GK In-Stock Unstable PLA2G2D 56 35 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767244 GK In-Stock Unstable PTGDR 0 40 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767244 GK In-Stock Unstable PLA2G5 50 44 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767244 GK In-Stock Unstable CYP2C9 38 43 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767244 GK In-Stock Unstable CYP3A4 19 41 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767244 GK In-Stock Unstable F2RL3 19 40 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767244 GK In-Stock Unstable PTGDR2 18 40 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767244 GK In-Stock Unstable PTGES2 61 33 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767244 GK In-Stock Unstable FFAR1 58 38 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767244 GK In-Stock Unstable DGAT1 0 40 CN(Cc1cccc(/C=C\C(=O)O)c1)C(=O)CC(F)(F)F ZINC000217767255 DF For-Sale Unstable PTGER2 24 42 CN(Cc1cccc(/C=C\C(=O)O)c1)C(=O)CC(F)(F)F ZINC000217767255 DF For-Sale Unstable AKR1C3 41 41 Cc1ccn(Cc2cccc(/C=C\C(=O)O)c2)n1 ZINC000217767270 BE For-Sale Unstable PTGER2 23 42 Cc1ccn(Cc2cccc(/C=C\C(=O)O)c2)n1 ZINC000217767270 BE For-Sale Unstable HDAC8 39 42 Cc1ccn(Cc2cccc(/C=C\C(=O)O)c2)n1 ZINC000217767270 BE For-Sale Unstable HDAC1 21 42 Cc1ccn(Cc2cccc(/C=C\C(=O)O)c2)n1 ZINC000217767270 BE For-Sale Unstable HDAC6 24 42 Cc1ccn(Cc2cccc(/C=C\C(=O)O)c2)n1 ZINC000217767270 BE For-Sale Unstable HDAC7 18 40 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccccc2)CC(=O)O4)cc1O ZINC000217767273 II In-Stock Unstable AKR1B1 23 49 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccccc2)CC(=O)O4)cc1O ZINC000217767273 II In-Stock Unstable CYP1B1 75 42 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccccc2)CC(=O)O4)cc1O ZINC000217767273 II In-Stock Unstable CYP1A1 58 49 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccccc2)CC(=O)O4)cc1O ZINC000217767273 II In-Stock Unstable CYP1A2 47 42 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccccc2)CC(=O)O4)cc1O ZINC000217767273 II In-Stock Unstable ABCG2 22 42 CCN(CC(=O)Nc1cccc(OC)c1)[C@@H](C)c1nc2ccccc2n1C(F)F ZINC000217767289 HI On-Demand Unstable MTNR1B 18 40 O=C(N[C@@H]1C[C@@H]1c1ccccc1)[C@@H](Cl)c1ccccc1 ZINC000217767309 CH For-Sale Unstable EPHX2 23 49 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccc(Cl)cc1Cl ZINC000217767336 FH For-Sale Unstable PREP 18 40 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccc(Cl)cc1Cl ZINC000217767336 FH For-Sale Unstable SLC6A9 48 40 Cc1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1C(F)(F)F ZINC000217767343 GJ On-Demand Unstable HTR2A 15 45 Cc1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1C(F)(F)F ZINC000217767343 GJ On-Demand Unstable HSD11B1 21 77 Cc1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1C(F)(F)F ZINC000217767343 GJ On-Demand Unstable SLC18A3 41 48 Cc1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1C(F)(F)F ZINC000217767343 GJ On-Demand Unstable SLC9A1 55 44 Cc1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1C(F)(F)F ZINC000217767343 GJ On-Demand Unstable RBP4 33 42 Cc1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1C(F)(F)F ZINC000217767343 GJ On-Demand Unstable SFRP1 70 37 Cc1ccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)cc1C(F)(F)F ZINC000217767343 GJ On-Demand Unstable L3MBTL3 86 40 COC(=O)CCc1ccc2[nH]cnc2c1 ZINC000217767345 BD In-Stock Unstable QPCT 28 44 CCOC(=O)c1c(C)n(CCc2ccccc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767354 HK In-Stock Unstable CNR1 16 43 CCOC(=O)c1c(C)n(CCc2ccccc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767354 HK In-Stock Unstable MAOB 35 46 CCOC(=O)c1c(C)n(CCc2ccccc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767354 HK In-Stock Unstable PTGER2 21 41 CCOC(=O)c1c(C)n(CCc2ccccc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767354 HK In-Stock Unstable ALOX5AP 91 35 CCOC(=O)c1c(C)n(CCc2ccccc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767354 HK In-Stock Unstable PLA2G2A 108 51 CCOC(=O)c1c(C)n(CCc2ccccc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767354 HK In-Stock Unstable PTGDR 0 41 CCOC(=O)c1c(C)n(CCc2ccccc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767354 HK In-Stock Unstable FFAR1 50 40 CCOC(=O)c1c(C)n(CCc2ccccc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767354 HK In-Stock Unstable FFAR4 43 35 CCN(CC(=O)Nc1cccc(OC)c1)[C@H](C)c1nc2ccccc2n1C(F)F ZINC000217767355 HI On-Demand Unstable MTNR1B 18 40 O=C(N[C@H]1C[C@@H]1c1ccccc1)[C@@H](Cl)c1ccccc1 ZINC000217767363 CH For-Sale Unstable EPHX2 23 49 C[C@@H]1CCCN(C(=O)N/C=C/c2ccccc2F)C1 ZINC000217767370 CG For-Sale Unstable SLC6A1 49 36 O=C(NC[C@H]1CCCN1c1nccs1)c1ccc(Cl)cc1Cl ZINC000217767419 FH For-Sale Unstable PREP 18 40 O=C(NC[C@H]1CCCN1c1nccs1)c1ccc(Cl)cc1Cl ZINC000217767419 FH For-Sale Unstable SLC6A9 48 40 COc1cc([C@@H](C)N2CCC[C@@H](C)C2)ccc1O ZINC000217767420 BG For-Sale Unstable PNLIP 0 46 COc1cc([C@@H](C)N2CCC[C@@H](C)C2)ccc1O ZINC000217767420 BG For-Sale Unstable N1L 0 47 COc1cc([C@@H](C)N2CCC[C@@H](C)C2)ccc1O ZINC000217767420 BG For-Sale Unstable SLC22A3 0 43 C[C@H]1CCCN(C(=O)N/C=C/c2ccccc2F)C1 ZINC000217767452 CG For-Sale Unstable SLC6A1 49 36 CCOC(=O)c1c(C)n(Cc2cccnc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767457 HK In-Stock Unstable MAOB 24 42 CCOC(=O)c1c(C)n(Cc2cccnc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767457 HK In-Stock Unstable PTAFR 15 40 CCOC(=O)c1c(C)n(Cc2cccnc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767457 HK In-Stock Unstable ALOX5AP 104 45 CCOC(=O)c1c(C)n(Cc2cccnc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767457 HK In-Stock Unstable PLA2G2A 100 54 CCOC(=O)c1c(C)n(Cc2cccnc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767457 HK In-Stock Unstable CYP2C9 36 42 CCOC(=O)c1c(C)n(Cc2cccnc2)c2ccc(OCc3ccccc3)cc12 ZINC000217767457 HK In-Stock Unstable CYP3A4 27 45 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccc(Cl)c(Cl)c1 ZINC000217767508 FH For-Sale Unstable CACNA1I 43 32 COC(=O)CCc1ccc2[nH]c(C)nc2c1 ZINC000217767539 BD In-Stock Unstable TYMS 42 34 COC(=O)CCc1ccc2[nH]c(C)nc2c1 ZINC000217767539 BD In-Stock Unstable GYRB 0 41 COC(=O)CCc1ccc2[nH]c(C)nc2c1 ZINC000217767539 BD In-Stock Unstable P2RY12 0 47 COC(=O)CCc1ccc2[nH]c(C)nc2c1 ZINC000217767539 BD In-Stock Unstable ALKBH3 51 34 C[C@@H](CC(F)(F)F)C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217767558 EH On-Demand Unstable HTR2A 16 49 C[C@@H](CC(F)(F)F)C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217767558 EH On-Demand Unstable SLC18A3 41 44 C[C@@H](CC(F)(F)F)C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217767558 EH On-Demand Unstable WNT3A 48 36 CCCn1c(C)c(C(=O)OCC)c2cc(OCC(=O)OCC)ccc21 ZINC000217767563 EG In-Stock Unstable PLA2G2A 53 45 CN1c2ccccc2C(=O)N2CCc3c(n(CCC(=O)N4CCCCC4)c4ccccc34)[C@H]21 ZINC000217767583 II In-Stock Unstable FABI 47 32 O=C(NC[C@H]1CCCN1c1nccs1)c1ccc(Cl)c(Cl)c1 ZINC000217767589 FH For-Sale Unstable CACNA1I 43 32 COC1CCN(C2CCN(C(=O)CCc3ccc(C(F)(F)F)cc3)CC2)CC1 ZINC000217767590 GH In-Stock Unstable CCR3 35 40 COC1CCN(C2CCN(C(=O)CCc3ccc(C(F)(F)F)cc3)CC2)CC1 ZINC000217767590 GH In-Stock Unstable SLC6A5 28 44 COC1CCN(C2CCN(C(=O)CCc3ccc(C(F)(F)F)cc3)CC2)CC1 ZINC000217767590 GH In-Stock Unstable LIPG 53 38 COC1CCN(C2CCN(C(=O)CCc3ccc(C(F)(F)F)cc3)CC2)CC1 ZINC000217767590 GH In-Stock Unstable L3MBTL3 67 36 C[C@H](CC(F)(F)F)C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217767629 EH On-Demand Unstable HTR2A 16 49 C[C@H](CC(F)(F)F)C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217767629 EH On-Demand Unstable SLC18A3 41 44 C[C@H](CC(F)(F)F)C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000217767629 EH On-Demand Unstable WNT3A 48 36 CCc1nc2cc(CCC(=O)OC)ccc2[nH]1 ZINC000217767641 BE In-Stock Unstable P2RY12 0 46 CCN(Cc1ccccc1)C(=O)N/C=C/c1ccccc1F ZINC000217767684 CI For-Sale Unstable TSPO 21 42 CCOC(=O)COc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCOC ZINC000217767704 FF In-Stock Unstable PLA2G2A 51 43 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(Br)s2)CC1 ZINC000217767742 GI On-Demand Unstable HTR2A 16 48 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(Br)s2)CC1 ZINC000217767742 GI On-Demand Unstable SLC18A3 40 54 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(Br)s2)CC1 ZINC000217767742 GI On-Demand Unstable WNT3A 46 33 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2ccc(Br)s2)CC1 ZINC000217767742 GI On-Demand Unstable L3MBTL3 79 47 O=C(O)c1sccc1S(=O)(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217767780 EF For-Sale Unstable FABP2 0 41 O=C(O)/C=C\c1ccc(NC(=O)Cc2cccs2)c(F)c1 ZINC000217767790 DG For-Sale Unstable CA7 15 60 O=C(O)/C=C\c1ccc(NC(=O)Cc2cccs2)c(F)c1 ZINC000217767790 DG For-Sale Unstable CA5B 51 60 O=C(O)/C=C\c1ccc(NC(=O)Cc2cccs2)c(F)c1 ZINC000217767790 DG For-Sale Unstable CA5A 53 60 CCOC(=O)COc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCc1ccccc1 ZINC000217767819 HI In-Stock Unstable CNR1 0 41 CCOC(=O)COc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCc1ccccc1 ZINC000217767819 HI In-Stock Unstable ALOX5AP 55 32 CCOC(=O)COc1ccc2c(c1)c(C(=O)OCC)c(C)n2CCc1ccccc1 ZINC000217767819 HI In-Stock Unstable PLA2G2A 114 46 Cc1ccn(CCOc2cccc(/C=C\C(=O)O)c2)n1 ZINC000217767845 CE For-Sale Unstable PTGER2 26 40 O=C(O)c1sccc1S(=O)(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217767862 EF For-Sale Unstable FABP2 0 41 C[C@@H](NCCCC1CCCC1)C(=O)OC(C)(C)C ZINC000217767878 CG On-Demand Unstable PFDN6 0 40 CCOc1ccc(C(=O)NC[C@@H]2CCCN2c2nccs2)cc1OCC ZINC000217767883 GG For-Sale Unstable SSTR5 48 38 CCOc1ccc(C(=O)NC[C@@H]2CCCN2c2nccs2)cc1OCC ZINC000217767883 GG For-Sale Unstable CACNA1I 50 36 CCOC(=O)COc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1cccnc1 ZINC000217767936 GH In-Stock Unstable ALOX5AP 88 39 CCOC(=O)COc1ccc2c(c1)c(C(=O)OCC)c(C)n2Cc1cccnc1 ZINC000217767936 GH In-Stock Unstable PLA2G2A 81 43 CCN(CC(=O)Nc1ccc2c(c1)OCCO2)[C@@H](C)c1nc2ccccc2n1C(F)F ZINC000217767952 II On-Demand Unstable IMDH_CRYPV 33 40 Cc1ccn(Cc2ccccc2/C=C\C(=O)O)n1 ZINC000217767953 BE For-Sale Unstable PTGER2 46 47 Cc1ccn(Cc2ccccc2/C=C\C(=O)O)n1 ZINC000217767953 BE For-Sale Unstable PTGER4 23 47 Cc1ccn(Cc2ccccc2/C=C\C(=O)O)n1 ZINC000217767953 BE For-Sale Unstable PTGER3 18 47 Cc1ccn(Cc2ccccc2/C=C\C(=O)O)n1 ZINC000217767953 BE For-Sale Unstable PTGDR 0 45 Cc1cc(NC(=O)c2cnoc2C)ccc1/C=C\C(=O)O ZINC000217767962 CF For-Sale Unstable KCNK3 58 37 C[C@H](NCCCC1CCCC1)C(=O)OC(C)(C)C ZINC000217767967 CG On-Demand Unstable PFDN6 0 40 CC(C)Cc1cc(C(=O)NC2CCN(c3ccccc3)CC2)nc(=O)[nH]1 ZINC000217767969 FE In-Stock Unstable P2RY12 49 31 CCOc1ccc(C(=O)NC[C@H]2CCCN2c2nccs2)cc1OCC ZINC000217767974 GG For-Sale Unstable SSTR5 48 38 CCOc1ccc(C(=O)NC[C@H]2CCCN2c2nccs2)cc1OCC ZINC000217767974 GG For-Sale Unstable CACNA1I 50 36 CCN(CC(=O)Nc1ccc2c(c1)OCCO2)[C@H](C)c1nc2ccccc2n1C(F)F ZINC000217768028 II On-Demand Unstable IMDH_CRYPV 33 40 COC1CCN(C2CCN(C(=O)CCc3ccc(F)c(Cl)c3)CC2)CC1 ZINC000217768034 GH In-Stock Unstable CCR3 51 38 COC1CCN(C2CCN(C(=O)CCc3ccc(F)c(Cl)c3)CC2)CC1 ZINC000217768034 GH In-Stock Unstable L3MBTL3 51 35 CC(C)c1nc2cc(NC(=O)CCN3C(=O)c4ccccc4N4C(=O)c5ccccc5[C@H]34)ccc2[nH]1 ZINC000217768077 JJ In-Stock Unstable NR2E3 59 35 Cc1cccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)n1 ZINC000217768082 EG On-Demand Unstable HTR2A 23 45 Cc1cccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)n1 ZINC000217768082 EG On-Demand Unstable HSD11B1 20 64 Cc1cccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)n1 ZINC000217768082 EG On-Demand Unstable CCR5 24 44 Cc1cccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)n1 ZINC000217768082 EG On-Demand Unstable SLC18A3 41 50 Cc1cccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)n1 ZINC000217768082 EG On-Demand Unstable WNT3A 51 36 Cc1cccc(C(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)n1 ZINC000217768082 EG On-Demand Unstable L3MBTL3 70 38 CC(C)c1nc2cc(NC(=O)CCN3C(=O)c4ccccc4N4C(=O)c5ccccc5[C@@H]34)ccc2[nH]1 ZINC000217768165 JJ In-Stock Unstable NR2E3 59 35 CCOC(=O)c1c(C)n(CC)c2ccc(OC3CCCC3)cc12 ZINC000217768181 DI In-Stock Unstable PLA2G2A 40 41 CCOC(=O)c1c(C)n(CC)c2ccc(OC3CCCC3)cc12 ZINC000217768181 DI In-Stock Unstable PFKFB3 44 34 O=C(N/C=C/c1ccccc1F)N(Cc1ccccc1)Cc1ccccc1 ZINC000217768205 FK For-Sale Unstable PTGES 26 40 COC(=O)[C@@H]1CCc2nc(N)ncc2C1 ZINC000217768229 BC In-Stock Unstable PTR1 45 32 CCCn1c(C)c(C(=O)OCC)c2cc(OC3CCCC3)ccc21 ZINC000217768290 EJ In-Stock Unstable PLA2G2A 36 41 COC(=O)[C@H]1CCc2nc(N)ncc2C1 ZINC000217768293 BC In-Stock Unstable PTR1 45 32 O=C(N/C=C/c1ccccc1F)N(CCO)Cc1ccccc1 ZINC000217768313 DG For-Sale Unstable LIMK2 18 40 CCCCn1c(C)c(C(=O)OCC)c2cc(OC3CCCC3)ccc21 ZINC000217768395 EK In-Stock Unstable CNR2 18 42 CCCCn1c(C)c(C(=O)OCC)c2cc(OC3CCCC3)ccc21 ZINC000217768395 EK In-Stock Unstable PLA2G2A 47 48 O=C1CCC(=O)N1C1C[C@@H]2CC[C@H](C1)N2S(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000217768407 HF In-Stock Unstable ELOVL6 0 42 COc1ccc(NC(=O)N/C=C/c2ccccc2F)c(OC)c1 ZINC000217768431 DH For-Sale Unstable CYP1B1 39 46 COc1ccc(NC(=O)N/C=C/c2ccccc2F)c(OC)c1 ZINC000217768431 DH For-Sale Unstable MTNR1A 19 45 COc1ccc(NC(=O)N/C=C/c2ccccc2F)c(OC)c1 ZINC000217768431 DH For-Sale Unstable MTNR1B 19 45 COc1ccc(NC(=O)N/C=C/c2ccccc2F)c(OC)c1 ZINC000217768431 DH For-Sale Unstable C5AR1 15 41 COc1ccc(NC(=O)N/C=C/c2ccccc2F)c(OC)c1 ZINC000217768431 DH For-Sale Unstable AKR1C2 40 32 COc1ccccc1-n1cc(CNC(=O)c2ccc(N)nc2)cn1 ZINC000217768435 DD In-Stock Unstable HTR1A 15 41 COc1ccccc1-n1cc(CNC(=O)c2ccc(N)nc2)cn1 ZINC000217768435 DD In-Stock Unstable DRD2 21 43 COc1ccccc1-n1cc(CNC(=O)c2ccc(N)nc2)cn1 ZINC000217768435 DD In-Stock Unstable DRD1 17 43 COc1ccccc1-n1cc(CNC(=O)c2ccc(N)nc2)cn1 ZINC000217768435 DD In-Stock Unstable DRD3 28 40 COc1ccc(C(=O)NC[C@@H]2CCCN2c2nccs2)c(OC)c1OC ZINC000217768444 GF For-Sale Unstable DRD2 46 44 COc1ccc(C(=O)NC[C@@H]2CCCN2c2nccs2)c(OC)c1OC ZINC000217768444 GF For-Sale Unstable ACKR3 64 33 COc1ccc(Cn2nccc2C)cc1/C=C\C(=O)O ZINC000217768461 CE For-Sale Unstable PTGER2 43 41 COc1ccc(Cn2nccc2C)cc1/C=C\C(=O)O ZINC000217768461 CE For-Sale Unstable PTGER4 24 41 COc1ccc(Cn2nccc2C)cc1/C=C\C(=O)O ZINC000217768461 CE For-Sale Unstable PTGER3 18 41 CCOC(=O)c1c(C)n(CCOC)c2ccc(OC3CCCC3)cc12 ZINC000217768491 EI In-Stock Unstable PLA2G2A 43 41 COc1cccc(CCN[C@@H](C)C(=O)OC(C)(C)C)c1 ZINC000217768518 CF On-Demand Unstable DRD4 40 31 COc1cccc(CCN[C@@H](C)C(=O)OC(C)(C)C)c1 ZINC000217768518 CF On-Demand Unstable MMP13 17 40 COc1cccc(CCN[C@@H](C)C(=O)OC(C)(C)C)c1 ZINC000217768518 CF On-Demand Unstable MTNR1A 63 50 COc1cccc(CCN[C@@H](C)C(=O)OC(C)(C)C)c1 ZINC000217768518 CF On-Demand Unstable MTNR1B 61 50 COc1cccc(CCN[C@@H](C)C(=O)OC(C)(C)C)c1 ZINC000217768518 CF On-Demand Unstable ABCB1 16 41 COc1ccc(C(=O)NC[C@H]2CCCN2c2nccs2)c(OC)c1OC ZINC000217768523 GF For-Sale Unstable DRD2 46 44 COc1ccc(C(=O)NC[C@H]2CCCN2c2nccs2)c(OC)c1OC ZINC000217768523 GF For-Sale Unstable ACKR3 64 33 Fc1ccccc1SCc1ccc(-n2ccnc2)cc1 ZINC000217768568 CI On-Demand Unstable CYP11B2 0 42 Fc1ccccc1SCc1ccc(-n2ccnc2)cc1 ZINC000217768568 CI On-Demand Unstable CYP2C19 18 41 CCOC(=O)c1c(C)n(CC(C)C)c2ccc(OC3CCCC3)cc12 ZINC000217768592 EK In-Stock Unstable PLA2G2A 31 40 COc1cccc(CCN[C@H](C)C(=O)OC(C)(C)C)c1 ZINC000217768604 CF On-Demand Unstable DRD4 40 31 COc1cccc(CCN[C@H](C)C(=O)OC(C)(C)C)c1 ZINC000217768604 CF On-Demand Unstable MMP13 17 40 COc1cccc(CCN[C@H](C)C(=O)OC(C)(C)C)c1 ZINC000217768604 CF On-Demand Unstable MTNR1A 63 50 COc1cccc(CCN[C@H](C)C(=O)OC(C)(C)C)c1 ZINC000217768604 CF On-Demand Unstable MTNR1B 61 50 COc1cccc(CCN[C@H](C)C(=O)OC(C)(C)C)c1 ZINC000217768604 CF On-Demand Unstable ABCB1 16 41 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)NC[C@@H]3C[C@H]4C=C[C@H]3C4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217768637 KH In-Stock Unstable TUBA1A 17 63 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)NC[C@@H]3C[C@H]4C=C[C@H]3C4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217768637 KH In-Stock Unstable TPPP 0 60 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OC3CCCC3)cc12 ZINC000217768708 GK In-Stock Unstable PRSS2 43 31 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OC3CCCC3)cc12 ZINC000217768708 GK In-Stock Unstable ALOX5AP 89 36 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OC3CCCC3)cc12 ZINC000217768708 GK In-Stock Unstable PLA2G2A 141 51 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OC3CCCC3)cc12 ZINC000217768708 GK In-Stock Unstable PLA2G2D 40 32 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OC3CCCC3)cc12 ZINC000217768708 GK In-Stock Unstable PLA2G5 36 40 CCOC(=O)c1c(C)n(Cc2ccccc2)c2ccc(OC3CCCC3)cc12 ZINC000217768708 GK In-Stock Unstable PTGES2 60 32 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)NC[C@@H]3C[C@@H]4C=C[C@H]3C4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217768713 KH In-Stock Unstable TUBA1A 17 63 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)NC[C@@H]3C[C@@H]4C=C[C@H]3C4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217768713 KH In-Stock Unstable TPPP 0 60 COc1ccc(CNc2ncnc3c(C=O)csc23)c(OC)c1 ZINC000217768765 EG For-Sale Unstable PDE6A 40 31 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)NC[C@@H]3C[C@H]4C=C[C@@H]3C4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217768811 KH In-Stock Unstable TUBA1A 17 63 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)NC[C@@H]3C[C@H]4C=C[C@@H]3C4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217768811 KH In-Stock Unstable TPPP 0 60 CCOC(=O)c1c(C)n(CCc2ccccc2)c2ccc(OC3CCCC3)cc12 ZINC000217768821 GK In-Stock Unstable KCNH2 32 43 CCOC(=O)c1c(C)n(CCc2ccccc2)c2ccc(OC3CCCC3)cc12 ZINC000217768821 GK In-Stock Unstable PLA2G2A 87 43 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)NC[C@@H]3C[C@@H]4C=C[C@@H]3C4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217768888 KH In-Stock Unstable TUBA1A 17 63 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)NC[C@@H]3C[C@@H]4C=C[C@@H]3C4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217768888 KH In-Stock Unstable TPPP 0 60 CC[C@@H](NCCc1cccc(OC)c1)c1ccc(F)cc1 ZINC000217768898 CI On-Demand Unstable MTNR1A 18 43 CC[C@@H](NCCc1cccc(OC)c1)c1ccc(F)cc1 ZINC000217768898 CI On-Demand Unstable ABCB1 0 43 CC[C@@H](NCCc1cccc(OC)c1)c1ccc(F)cc1 ZINC000217768898 CI On-Demand Unstable LEF 27 41 CCOC(=O)c1c(C)n(Cc2cccnc2)c2ccc(OC3CCCC3)cc12 ZINC000217768923 GJ In-Stock Unstable ALOX5AP 59 37 CCOC(=O)c1c(C)n(Cc2cccnc2)c2ccc(OC3CCCC3)cc12 ZINC000217768923 GJ In-Stock Unstable PLA2G2A 72 40 CCCCCC(=O)Nc1cc(/C=C\C(=O)O)ccc1C ZINC000217768946 CH For-Sale Unstable HDAC3 17 40 CCCCCC(=O)Nc1cc(/C=C\C(=O)O)ccc1C ZINC000217768946 CH For-Sale Unstable AKR1C3 24 41 CCCCCC(=O)Nc1cc(/C=C\C(=O)O)ccc1C ZINC000217768946 CH For-Sale Unstable NOD1 41 33 O=C(c1cccc(N2CCOCC2)c1)N1CCC(c2cc[nH]n2)CC1 ZINC000217768949 EE In-Stock Unstable AKR1C3 27 42 CC[C@H](NCCc1cccc(OC)c1)c1ccc(F)cc1 ZINC000217768992 CI On-Demand Unstable MTNR1A 18 43 CC[C@H](NCCc1cccc(OC)c1)c1ccc(F)cc1 ZINC000217768992 CI On-Demand Unstable ABCB1 0 43 CC[C@H](NCCc1cccc(OC)c1)c1ccc(F)cc1 ZINC000217768992 CI On-Demand Unstable LEF 27 41 CCOC(=O)[C@@H](C1CCCCC1)S(=O)(=O)CC ZINC000217769002 CD In-Stock Unstable AMY2 44 30 CCCCCCCCOc1ccc([C@@H]2CC(=O)Oc3c2c2nc4ccccc4nc2c2ccccc32)cc1 ZINC000217769012 KK In-Stock Unstable PLA2G4B 78 33 O=C(O)/C=C\c1cccc(NC(=O)CCn2cncn2)n1 ZINC000217769037 CC For-Sale Unstable HIS3 47 34 O=C(N[C@H](CCO)C(=O)O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000217769062 CC For-Sale Unstable NAALAD2 58 40 O=C(N[C@H](CCO)C(=O)O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000217769062 CC For-Sale Unstable EPHX2 21 46 O=C(N[C@H](CCO)C(=O)O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000217769062 CC For-Sale Unstable KDM1A 41 32 CCCCCCCCOc1ccc([C@H]2CC(=O)Oc3c2c2nc4ccccc4nc2c2ccccc32)cc1 ZINC000217769085 KK In-Stock Unstable PLA2G4B 78 33 CCOC(=O)[C@H](C1CCCCC1)S(=O)(=O)CC ZINC000217769094 CD In-Stock Unstable AMY2 44 30 O=C(N[C@H]1C[C@@H]1c1ccccc1)N[C@H](CCO)C(=O)O ZINC000217769147 CC For-Sale Unstable NAALAD2 58 40 O=C(N[C@H]1C[C@@H]1c1ccccc1)N[C@H](CCO)C(=O)O ZINC000217769147 CC For-Sale Unstable EPHX2 21 46 O=C(N[C@H]1C[C@@H]1c1ccccc1)N[C@H](CCO)C(=O)O ZINC000217769147 CC For-Sale Unstable KDM1A 41 32 CC[C@@H](C(=O)NC1[C@@H]2CNC[C@@H]12)c1ccccc1 ZINC000217769228 BD For-Sale Unstable KCNQ2 52 45 CC[C@@H](C(=O)NC1[C@@H]2CNC[C@@H]12)c1ccccc1 ZINC000217769228 BD For-Sale Unstable KCNQ4 0 45 Cc1c(C=O)c2cc(O)ccc2n1CCc1ccccc1 ZINC000217769240 CH In-Stock Unstable CASR 0 44 Cc1c(C=O)c2cc(O)ccc2n1CCc1ccccc1 ZINC000217769240 CH In-Stock Unstable PLA2G2A 37 41 C/C=C(\C)C(=O)O[C@@H]1[C@@H](C)[C@@]2(O)[C@@H](C=C(CO)C[C@]3(O)C(=O)C(C)=C[C@@H]23)[C@H]2C(C)(C)[C@@]21OC(=O)[C@H](C)CC ZINC000217769254 KG In-Stock Unstable PTGS1 28 68 C/C=C(\C)C(=O)O[C@@H]1[C@@H](C)[C@@]2(O)[C@@H](C=C(CO)C[C@]3(O)C(=O)C(C)=C[C@@H]23)[C@H]2C(C)(C)[C@@]21OC(=O)[C@H](C)CC ZINC000217769254 KG In-Stock Unstable PRKCD 24 71 C/C=C(\C)C(=O)O[C@@H]1[C@@H](C)[C@@]2(O)[C@@H](C=C(CO)C[C@]3(O)C(=O)C(C)=C[C@@H]23)[C@H]2C(C)(C)[C@@]21OC(=O)[C@H](C)CC ZINC000217769254 KG In-Stock Unstable PRKCE 36 69 C/C=C(\C)C(=O)O[C@@H]1[C@@H](C)[C@@]2(O)[C@@H](C=C(CO)C[C@]3(O)C(=O)C(C)=C[C@@H]23)[C@H]2C(C)(C)[C@@]21OC(=O)[C@H](C)CC ZINC000217769254 KG In-Stock Unstable PRKCG 23 69 C/C=C(\C)C(=O)O[C@@H]1[C@@H](C)[C@@]2(O)[C@@H](C=C(CO)C[C@]3(O)C(=O)C(C)=C[C@@H]23)[C@H]2C(C)(C)[C@@]21OC(=O)[C@H](C)CC ZINC000217769254 KG In-Stock Unstable PRKCH 24 69 C/C=C(\C)C(=O)O[C@@H]1[C@@H](C)[C@@]2(O)[C@@H](C=C(CO)C[C@]3(O)C(=O)C(C)=C[C@@H]23)[C@H]2C(C)(C)[C@@]21OC(=O)[C@H](C)CC ZINC000217769254 KG In-Stock Unstable PRKCA 23 69 C/C=C(\C)C(=O)O[C@@H]1[C@@H](C)[C@@]2(O)[C@@H](C=C(CO)C[C@]3(O)C(=O)C(C)=C[C@@H]23)[C@H]2C(C)(C)[C@@]21OC(=O)[C@H](C)CC ZINC000217769254 KG In-Stock Unstable TRPV4 34 66 C/C=C(\C)C(=O)O[C@@H]1[C@@H](C)[C@@]2(O)[C@@H](C=C(CO)C[C@]3(O)C(=O)C(C)=C[C@@H]23)[C@H]2C(C)(C)[C@@]21OC(=O)[C@H](C)CC ZINC000217769254 KG In-Stock Unstable VAV1 0 69 O=C(O)C[C@@H]1CCCN1C(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000217769278 CE On-Demand Unstable PREP 52 38 O=C(O)C[C@@H]1CCCN1C(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000217769278 CE On-Demand Unstable EPHX2 27 51 CC[C@H](C(=O)NC1[C@@H]2CNC[C@@H]12)c1ccccc1 ZINC000217769301 BD On-Demand Unstable KCNQ4 0 45 C/C=C(\C)C(=O)O[C@@H]1[C@@H](C)[C@@]2(O)[C@@H](C=C(CO)C[C@]3(O)C(=O)C(C)=C[C@@H]23)[C@H]2C(C)(C)[C@@]21OC(=O)[C@@H](C)CC ZINC000217769319 KG In-Stock Unstable PTGS1 28 68 C/C=C(\C)C(=O)O[C@@H]1[C@@H](C)[C@@]2(O)[C@@H](C=C(CO)C[C@]3(O)C(=O)C(C)=C[C@@H]23)[C@H]2C(C)(C)[C@@]21OC(=O)[C@@H](C)CC ZINC000217769319 KG In-Stock Unstable PRKCD 24 71 C/C=C(\C)C(=O)O[C@@H]1[C@@H](C)[C@@]2(O)[C@@H](C=C(CO)C[C@]3(O)C(=O)C(C)=C[C@@H]23)[C@H]2C(C)(C)[C@@]21OC(=O)[C@@H](C)CC ZINC000217769319 KG In-Stock Unstable PRKCE 36 69 C/C=C(\C)C(=O)O[C@@H]1[C@@H](C)[C@@]2(O)[C@@H](C=C(CO)C[C@]3(O)C(=O)C(C)=C[C@@H]23)[C@H]2C(C)(C)[C@@]21OC(=O)[C@@H](C)CC ZINC000217769319 KG In-Stock Unstable PRKCG 23 69 C/C=C(\C)C(=O)O[C@@H]1[C@@H](C)[C@@]2(O)[C@@H](C=C(CO)C[C@]3(O)C(=O)C(C)=C[C@@H]23)[C@H]2C(C)(C)[C@@]21OC(=O)[C@@H](C)CC ZINC000217769319 KG In-Stock Unstable PRKCH 24 69 C/C=C(\C)C(=O)O[C@@H]1[C@@H](C)[C@@]2(O)[C@@H](C=C(CO)C[C@]3(O)C(=O)C(C)=C[C@@H]23)[C@H]2C(C)(C)[C@@]21OC(=O)[C@@H](C)CC ZINC000217769319 KG In-Stock Unstable PRKCA 23 69 C/C=C(\C)C(=O)O[C@@H]1[C@@H](C)[C@@]2(O)[C@@H](C=C(CO)C[C@]3(O)C(=O)C(C)=C[C@@H]23)[C@H]2C(C)(C)[C@@]21OC(=O)[C@@H](C)CC ZINC000217769319 KG In-Stock Unstable TRPV4 34 66 C/C=C(\C)C(=O)O[C@@H]1[C@@H](C)[C@@]2(O)[C@@H](C=C(CO)C[C@]3(O)C(=O)C(C)=C[C@@H]23)[C@H]2C(C)(C)[C@@]21OC(=O)[C@@H](C)CC ZINC000217769319 KG In-Stock Unstable VAV1 0 69 CCCn1c(C)c(C=O)c2cc(OC)ccc21 ZINC000217769345 BG In-Stock Unstable PTGS2 37 41 CCCn1c(C)c(C=O)c2cc(OC)ccc21 ZINC000217769345 BG In-Stock Unstable PLA2G2A 37 40 O=C(O)C[C@@H]1CCCN1C(=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000217769368 CE On-Demand Unstable PREP 52 38 O=C(O)C[C@@H]1CCCN1C(=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000217769368 CE On-Demand Unstable EPHX2 27 51 CCS(=O)(=O)[C@H](C(=O)O)C1CCCCC1 ZINC000217769396 BD In-Stock Unstable AMY2 43 30 COC(=O)C[C@H](c1ccc(OC)c(O)c1)c1c(O)ccc2c(=O)c(-c3ccc(O)cc3)coc12 ZINC000217769404 JI In-Stock Unstable ALDH2 100 41 Cc1ccccc1C(=O)Nc1cccc(/C=C\C(=O)O)n1 ZINC000217769441 CF For-Sale Unstable GRM5 15 43 Cc1ccccc1C(=O)Nc1cccc(/C=C\C(=O)O)n1 ZINC000217769441 CF For-Sale Unstable SORT1 26 42 Cc1ccccc1C(=O)Nc1cccc(/C=C\C(=O)O)n1 ZINC000217769441 CF For-Sale Unstable KCNK3 40 45 Cc1ccccc1C(=O)Nc1cccc(/C=C\C(=O)O)n1 ZINC000217769441 CF For-Sale Unstable KCNK9 35 42 CCCCn1c(C)c(C=O)c2cc(OC)ccc21 ZINC000217769466 BH In-Stock Unstable PTGS2 37 40 CCCCn1c(C)c(C=O)c2cc(OC)ccc21 ZINC000217769466 BH In-Stock Unstable PLA2G2A 45 44 CCCCn1c(C)c(C=O)c2cc(OC)ccc21 ZINC000217769466 BH In-Stock Unstable GSG2 41 38 CCCCn1c(C)c(C=O)c2cc(OC)ccc21 ZINC000217769466 BH In-Stock Unstable RORB 0 50 CCS(=O)(=O)[C@@H](C(=O)O)C1CCCCC1 ZINC000217769479 BD In-Stock Unstable AMY2 43 30 COC(=O)C[C@@H](c1ccc(OC)c(O)c1)c1c(O)ccc2c(=O)c(-c3ccc(O)cc3)coc12 ZINC000217769509 JI In-Stock Unstable ALDH2 100 41 O=C(O)[C@H]1CN(C(=O)N[C@@H]2C[C@@H]2c2ccccc2)CCO1 ZINC000217769522 CD For-Sale Unstable CACNA1C 0 45 O=C(O)[C@H]1CN(C(=O)N[C@@H]2C[C@@H]2c2ccccc2)CCO1 ZINC000217769522 CD For-Sale Unstable SCN5A 25 52 O=C(O)[C@H]1CN(C(=O)N[C@@H]2C[C@@H]2c2ccccc2)CCO1 ZINC000217769522 CD For-Sale Unstable EPHX2 30 56 CCCC[C@@H](CC)C(=O)NC1[C@@H]2CNC[C@@H]12 ZINC000217769527 BD For-Sale Unstable SLC22A20 0 44 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cc(C(F)(F)F)cc(C(F)(F)F)c2)CC1 ZINC000217769571 IK On-Demand Unstable HTR2A 17 48 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cc(C(F)(F)F)cc(C(F)(F)F)c2)CC1 ZINC000217769571 IK On-Demand Unstable TACR1 67 42 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cc(C(F)(F)F)cc(C(F)(F)F)c2)CC1 ZINC000217769571 IK On-Demand Unstable CACNA1B 33 41 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cc(C(F)(F)F)cc(C(F)(F)F)c2)CC1 ZINC000217769571 IK On-Demand Unstable SLC18A3 42 51 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cc(C(F)(F)F)cc(C(F)(F)F)c2)CC1 ZINC000217769571 IK On-Demand Unstable SLC9A1 44 39 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cc(C(F)(F)F)cc(C(F)(F)F)c2)CC1 ZINC000217769571 IK On-Demand Unstable RBP4 20 45 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cc(C(F)(F)F)cc(C(F)(F)F)c2)CC1 ZINC000217769571 IK On-Demand Unstable MLYCD 18 41 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cc(C(F)(F)F)cc(C(F)(F)F)c2)CC1 ZINC000217769571 IK On-Demand Unstable SFRP1 42 41 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cc(C(F)(F)F)cc(C(F)(F)F)c2)CC1 ZINC000217769571 IK On-Demand Unstable WNT3A 45 33 O=C(c1ccc(F)cc1)C1CCN(C(=O)c2cc(C(F)(F)F)cc(C(F)(F)F)c2)CC1 ZINC000217769571 IK On-Demand Unstable L3MBTL3 89 40 Cc1ccc(NC(=O)CN(C)C)cc1Br ZINC000217769573 CE On-Demand Unstable CA4 16 40 COc1ccc2c(c1)c(C=O)c(C)n2CCc1ccccc1 ZINC000217769585 CI In-Stock Unstable PTGS2 28 44 COc1ccc2c(c1)c(C=O)c(C)n2CCc1ccccc1 ZINC000217769585 CI In-Stock Unstable PLA2G2A 66 51 COc1ccc2c(c1)c(C=O)c(C)n2CCc1ccccc1 ZINC000217769585 CI In-Stock Unstable HTR6 0 53 COc1ccc2c(c1)c(C=O)c(C)n2CCc1ccccc1 ZINC000217769585 CI In-Stock Unstable MTNR1A 33 40 O=C(O)[C@H]1CN(C(=O)N[C@H]2C[C@@H]2c2ccccc2)CCO1 ZINC000217769598 CD For-Sale Unstable CACNA1C 0 45 O=C(O)[C@H]1CN(C(=O)N[C@H]2C[C@@H]2c2ccccc2)CCO1 ZINC000217769598 CD For-Sale Unstable SCN5A 25 52 O=C(O)[C@H]1CN(C(=O)N[C@H]2C[C@@H]2c2ccccc2)CCO1 ZINC000217769598 CD For-Sale Unstable EPHX2 30 56 COc1ccc(/C=C\C(=O)O)cc1NC(=O)[C@H]1C[C@@H]1C ZINC000217769619 CE For-Sale Unstable TUBB1 43 40 COc1ccc(/C=C\C(=O)O)cc1NC(=O)[C@H]1C[C@@H]1C ZINC000217769619 CE For-Sale Unstable ABCG2 15 42 CCCC[C@H](CC)C(=O)NC1[C@@H]2CNC[C@@H]12 ZINC000217769627 BD On-Demand Unstable SLC22A20 0 44 COc1ccc2[nH]c3c(c2c1)CN(C(=O)[C@@H]1CC(=O)N(Cc2ccccc2)C1)CC3 ZINC000217769633 HG In-Stock Unstable SSTR4 49 36 COc1ccc2[nH]c3c(c2c1)CN(C(=O)[C@@H]1CC(=O)N(Cc2ccccc2)C1)CC3 ZINC000217769633 HG In-Stock Unstable MAPKAPK2 22 43 COc1ccc2[nH]c3c(c2c1)CN(C(=O)[C@@H]1CC(=O)N(Cc2ccccc2)C1)CC3 ZINC000217769633 HG In-Stock Unstable PDE11A 27 40 COc1ccc(/C=C\C(=O)O)cc1NC(=O)[C@@H]1CCCO1 ZINC000217769704 CD For-Sale Unstable ABCG2 15 40 CCOC(=O)N1CCN([C@H](C)c2ccccc2O)CC1 ZINC000217769711 CE For-Sale Unstable P2RY12 61 41 Cc1cc(NC(=O)CN(C)C)ccc1Br ZINC000217769712 CE On-Demand Unstable CA4 16 40 COc1ccc2[nH]c3c(c2c1)CN(C(=O)[C@H]1CC(=O)N(Cc2ccccc2)C1)CC3 ZINC000217769724 HG In-Stock Unstable SSTR4 49 36 COc1ccc2[nH]c3c(c2c1)CN(C(=O)[C@H]1CC(=O)N(Cc2ccccc2)C1)CC3 ZINC000217769724 HG In-Stock Unstable MAPKAPK2 22 43 COc1ccc2[nH]c3c(c2c1)CN(C(=O)[C@H]1CC(=O)N(Cc2ccccc2)C1)CC3 ZINC000217769724 HG In-Stock Unstable PDE11A 27 40 Cc1ccc(C(=O)NC[C@@H]2CCCN2c2nccs2)cc1C ZINC000217769768 DG For-Sale Unstable MAPK14 17 46 COc1ccc(/C=C\C(=O)O)cc1NC(=O)[C@H]1CCCO1 ZINC000217769782 CD For-Sale Unstable ABCG2 15 40 O=C(O)[C@H]1C[C@H](O)CN1C(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000217769810 CC For-Sale Unstable SCN5A 0 41 O=C(O)[C@H]1C[C@H](O)CN1C(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000217769810 CC For-Sale Unstable EPHX2 25 48 CCCn1c(C)c(C=O)c2cc(OCC)ccc21 ZINC000217769820 BH In-Stock Unstable PLA2G2A 21 40 CC(C)[C@@H]1CC[C@@H](N)[C@@H](CCc2ccc([N+](=O)[O-])cc2)C1 ZINC000217769832 CH For-Sale Unstable KCNJ1 23 40 CN(C)CC(=O)Nc1ccc(Br)cc1F ZINC000217769833 CE On-Demand Unstable CA1 15 48 CN(C)CC(=O)Nc1ccc(Br)cc1F ZINC000217769833 CE On-Demand Unstable CA4 21 48 Cc1ccc(C(=O)NC[C@H]2CCCN2c2nccs2)cc1C ZINC000217769854 DG For-Sale Unstable MAPK14 17 46 COc1ccc(/C=C\C(=O)O)cc1NC(=O)c1ccsc1 ZINC000217769873 DG For-Sale Unstable TUBB1 44 40 COc1ccc(/C=C\C(=O)O)cc1NC(=O)c1ccsc1 ZINC000217769873 DG For-Sale Unstable ABCG2 15 40 CC(C)[C@H]1CC[C@@H](N)[C@@H](CCc2ccc([N+](=O)[O-])cc2)C1 ZINC000217769917 CH For-Sale Unstable KCNJ1 23 40 CCCCn1c(C)c(C=O)c2cc(OCC)ccc21 ZINC000217769937 CH In-Stock Unstable PLA2G2A 34 48 O=C(O)[C@@H]1CCCCN1C(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000217769954 CE For-Sale Unstable ACE 62 42 O=C(O)[C@@H]1CCCCN1C(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000217769954 CE For-Sale Unstable FKBP1A 33 40 O=C(O)[C@@H]1CCCCN1C(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000217769954 CE For-Sale Unstable MME 20 42 O=C(O)[C@@H]1CCCCN1C(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000217769954 CE For-Sale Unstable CPT2 41 35 O=C(O)[C@@H]1CCCCN1C(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000217769954 CE For-Sale Unstable PREP 80 42 O=C(O)[C@@H]1CCCCN1C(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000217769954 CE For-Sale Unstable EPHX2 31 53 O=C(O)[C@@H]1CCCCN1C(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000217769954 CE For-Sale Unstable WNT3 40 32 O=C(O)/C=C\c1cnc(NC(=O)c2ccc(F)cc2)s1 ZINC000217769965 CF For-Sale Anodyne DGAT1 15 40 CC(C)[C@@H]1CC[C@H](N)[C@@H](CCc2ccc([N+](=O)[O-])cc2)C1 ZINC000217769999 CH For-Sale Unstable KCNJ1 23 40 O=C(O)[C@@H]1CCCCN1C(=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000217770037 CE For-Sale Unstable ACE 62 42 O=C(O)[C@@H]1CCCCN1C(=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000217770037 CE For-Sale Unstable FKBP1A 33 40 O=C(O)[C@@H]1CCCCN1C(=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000217770037 CE For-Sale Unstable MME 20 42 O=C(O)[C@@H]1CCCCN1C(=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000217770037 CE For-Sale Unstable CPT2 41 35 O=C(O)[C@@H]1CCCCN1C(=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000217770037 CE For-Sale Unstable PREP 80 42 O=C(O)[C@@H]1CCCCN1C(=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000217770037 CE For-Sale Unstable EPHX2 31 53 O=C(O)[C@@H]1CCCCN1C(=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000217770037 CE For-Sale Unstable WNT3 40 32 O=C(O)/C=C\c1cnc(NC(=O)c2ccc(Cl)cc2)s1 ZINC000217770055 DG For-Sale Anodyne LUCI_LUCLA 31 41 FC(F)c1c[nH]c2ccc(Br)cc12 ZINC000217770077 BH For-Sale Anodyne MPO 44 34 CC(C)[C@H]1CC[C@H](N)[C@@H](CCc2ccc([N+](=O)[O-])cc2)C1 ZINC000217770087 CH For-Sale Unstable KCNJ1 23 40 CCOc1ccc2c(c1)c(C=O)c(C)n2Cc1ccccc1 ZINC000217770129 CI In-Stock Unstable ALOX5AP 73 33 CCOc1ccc2c(c1)c(C=O)c(C)n2Cc1ccccc1 ZINC000217770129 CI In-Stock Unstable PLA2G2A 99 49 O=C(O)/C=C\c1cnc(NC(=O)CCCc2cccs2)s1 ZINC000217770130 DG For-Sale Unstable PTPRF 18 41 NC(=O)C[C@@H](NC(=O)N[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000217770155 CC For-Sale Unstable EPHX2 20 45 NC(=O)C[C@@H](NC(=O)N[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000217770155 CC For-Sale Unstable KDM1A 42 34 Cc1cc(OC2CCN(C(=O)c3ccc(-c4ccsc4)cc3)CC2)cc(=O)o1 ZINC000217770204 GI In-Stock Unstable OXTR 0 42 Cc1cc(OC2CCN(C(=O)c3ccc(-c4ccsc4)cc3)CC2)cc(=O)o1 ZINC000217770204 GI In-Stock Unstable PRSS2 76 32 Cc1cc(OC2CCN(C(=O)c3ccc(-c4ccsc4)cc3)CC2)cc(=O)o1 ZINC000217770204 GI In-Stock Unstable HRH3 16 41 Cc1cc(OC2CCN(C(=O)c3ccc(-c4ccsc4)cc3)CC2)cc(=O)o1 ZINC000217770204 GI In-Stock Unstable CCR3 24 43 Cc1cc(OC2CCN(C(=O)c3ccc(-c4ccsc4)cc3)CC2)cc(=O)o1 ZINC000217770204 GI In-Stock Unstable L3MBTL3 52 33 O=C(N/C=C/c1ccccc1F)Nc1ccc(Nc2ccccc2)cc1 ZINC000217770235 EK For-Sale Anodyne EPHX1 0 43 O=C(N/C=C/c1ccccc1F)Nc1ccc(Nc2ccccc2)cc1 ZINC000217770235 EK For-Sale Anodyne P95276_MYCTO 0 43 NC(=O)C[C@@H](NC(=O)N[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000217770240 CC For-Sale Unstable EPHX2 20 45 NC(=O)C[C@@H](NC(=O)N[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000217770240 CC For-Sale Unstable KDM1A 42 34 CCOc1ccc2c(c1)c(C=O)c(C)n2CCc1ccccc1 ZINC000217770255 DI In-Stock Unstable PLA2G2A 65 41 COC(=O)c1ccc(CNC(=O)[C@@H](C)N[C@@H](C)c2ccc(Cl)c(Cl)c2)cc1 ZINC000217770257 HI On-Demand Unstable TRPV1 18 46 COC(=O)c1ccc(CNC(=O)[C@@H](C)N[C@@H](C)c2ccc(Cl)c(Cl)c2)cc1 ZINC000217770257 HI On-Demand Unstable F2R 32 41 COC(=O)c1ccc(CNC(=O)[C@@H](C)N[C@@H](C)c2ccc(Cl)c(Cl)c2)cc1 ZINC000217770257 HI On-Demand Unstable F7 19 44 COC(=O)c1ccc(CNC(=O)[C@@H](C)N[C@@H](C)c2ccc(Cl)c(Cl)c2)cc1 ZINC000217770257 HI On-Demand Unstable RPA1 62 38 Cc1cc(OC2CCN(C(=O)c3cc4cc(F)ccc4s3)CC2)cc(=O)o1 ZINC000217770304 GH In-Stock Unstable PRSS2 41 37 COC(=O)c1ccc(CNC(=O)[C@H](C)N[C@@H](C)c2ccc(Cl)c(Cl)c2)cc1 ZINC000217770342 HI On-Demand Unstable TRPV1 18 46 COC(=O)c1ccc(CNC(=O)[C@H](C)N[C@@H](C)c2ccc(Cl)c(Cl)c2)cc1 ZINC000217770342 HI On-Demand Unstable F2R 32 41 COC(=O)c1ccc(CNC(=O)[C@H](C)N[C@@H](C)c2ccc(Cl)c(Cl)c2)cc1 ZINC000217770342 HI On-Demand Unstable F7 19 44 COC(=O)c1ccc(CNC(=O)[C@H](C)N[C@@H](C)c2ccc(Cl)c(Cl)c2)cc1 ZINC000217770342 HI On-Demand Unstable RPA1 62 38 Cc1ccnn1Cc1cccc(/C=C\C(=O)O)c1 ZINC000217770376 BE For-Sale Unstable PTGER2 30 42 Cc1ccnn1Cc1cccc(/C=C\C(=O)O)c1 ZINC000217770376 BE For-Sale Unstable HDAC8 38 40 Cc1ccnn1Cc1cccc(/C=C\C(=O)O)c1 ZINC000217770376 BE For-Sale Unstable HDAC1 15 40 Cc1ccnn1Cc1cccc(/C=C\C(=O)O)c1 ZINC000217770376 BE For-Sale Unstable HDAC6 22 40 COC(=O)CNC(=O)CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12 ZINC000217770391 HD In-Stock Unstable TOP1 21 41 CC[C@@H](C)C(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217770395 CF For-Sale Unstable NR1H4 37 40 CC[C@@H](C)C(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217770395 CF For-Sale Unstable AKR1C3 42 44 COC(=O)c1ccc(CNC(=O)[C@@H](C)N[C@H](C)c2ccc(Cl)c(Cl)c2)cc1 ZINC000217770423 HI On-Demand Unstable TRPV1 18 46 COC(=O)c1ccc(CNC(=O)[C@@H](C)N[C@H](C)c2ccc(Cl)c(Cl)c2)cc1 ZINC000217770423 HI On-Demand Unstable F2R 32 41 COC(=O)c1ccc(CNC(=O)[C@@H](C)N[C@H](C)c2ccc(Cl)c(Cl)c2)cc1 ZINC000217770423 HI On-Demand Unstable F7 19 44 COC(=O)c1ccc(CNC(=O)[C@@H](C)N[C@H](C)c2ccc(Cl)c(Cl)c2)cc1 ZINC000217770423 HI On-Demand Unstable RPA1 62 38 CCCOc1ccc2c(c1)c(C=O)c(C)n2CC ZINC000217770440 BH In-Stock Unstable PLA2G2A 27 40 Cc1cccc(NC(=O)N/C=C/c2ccccc2F)n1 ZINC000217770443 CG For-Sale Unstable GRM5 18 45 CC[C@H](C)C(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217770461 CF For-Sale Unstable NR1H4 37 40 CC[C@H](C)C(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217770461 CF For-Sale Unstable AKR1C3 42 44 COC(=O)CNC(=O)CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12 ZINC000217770463 HD In-Stock Unstable TOP1 21 41 CCc1nc2ccc(C(=O)N3CCC(N4CCC(OC)CC4)CC3)cc2s1 ZINC000217770485 GH In-Stock Unstable CHRM2 47 37 CCc1nc2ccc(C(=O)N3CCC(N4CCC(OC)CC4)CC3)cc2s1 ZINC000217770485 GH In-Stock Unstable HRH1 15 41 CCc1nc2ccc(C(=O)N3CCC(N4CCC(OC)CC4)CC3)cc2s1 ZINC000217770485 GH In-Stock Unstable CCR3 45 43 CCc1nc2ccc(C(=O)N3CCC(N4CCC(OC)CC4)CC3)cc2s1 ZINC000217770485 GH In-Stock Unstable GRM1 17 40 CCc1nc2ccc(C(=O)N3CCC(N4CCC(OC)CC4)CC3)cc2s1 ZINC000217770485 GH In-Stock Unstable L3MBTL3 92 46 COC(=O)c1ccc(CNC(=O)[C@H](C)N[C@H](C)c2ccc(Cl)c(Cl)c2)cc1 ZINC000217770493 HI On-Demand Unstable TRPV1 18 46 COC(=O)c1ccc(CNC(=O)[C@H](C)N[C@H](C)c2ccc(Cl)c(Cl)c2)cc1 ZINC000217770493 HI On-Demand Unstable F2R 32 41 COC(=O)c1ccc(CNC(=O)[C@H](C)N[C@H](C)c2ccc(Cl)c(Cl)c2)cc1 ZINC000217770493 HI On-Demand Unstable F7 19 44 COC(=O)c1ccc(CNC(=O)[C@H](C)N[C@H](C)c2ccc(Cl)c(Cl)c2)cc1 ZINC000217770493 HI On-Demand Unstable RPA1 62 38 COc1ccc(C(=O)O)c(Br)c1N ZINC000217770505 BD For-Sale Unstable AKR1C2 49 37 Cc1cc(OC2CCN(C(=O)c3csc(-c4ccccc4)n3)CC2)cc(=O)o1 ZINC000217770524 GH In-Stock Unstable PRSS2 63 34 Cc1cc(OC2CCN(C(=O)c3csc(-c4ccccc4)n3)CC2)cc(=O)o1 ZINC000217770524 GH In-Stock Unstable HRH3 16 42 Cc1cc(OC2CCN(C(=O)c3csc(-c4ccccc4)n3)CC2)cc(=O)o1 ZINC000217770524 GH In-Stock Unstable TRPC6 66 39 CCCOc1ccc2c(c1)c(C=O)c(C)n2CCC ZINC000217770544 CH In-Stock Unstable PLA2G2A 29 44 CCC(CC)C(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217770555 CG For-Sale Unstable PTGER2 22 40 CCC(CC)C(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217770555 CG For-Sale Unstable HSD17B2 26 40 CCC(CC)C(=O)N(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217770555 CG For-Sale Unstable AKR1C3 33 44 COc1cn(CC(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)c(C)cc1=O ZINC000217770570 FC In-Stock Unstable CHRNA4 36 48 NC[C@@H](N1CCC[C@@H]1c1cccnc1)C(F)(F)F ZINC000217770611 CE For-Sale Unstable CHRNA2 51 52 Cc1ccccc1[C@@H](C)NCC(=O)N1c2ccccc2NC(=O)C[C@@H]1C(F)(F)F ZINC000217770613 HH On-Demand Unstable CTSA 46 32 Cc1c(N)cc(C(=O)O)c(Br)c1O ZINC000217770615 BD For-Sale Unstable AKR1C2 49 40 Cc1c(N)cc(C(=O)O)c(Br)c1O ZINC000217770615 BD For-Sale Unstable AKR1C1 53 40 CN(Cc1cccc(/C=C\C(=O)O)c1)C(=O)CC(C)(C)C ZINC000217770650 CG For-Sale Unstable PTGER2 24 43 CN(Cc1cccc(/C=C\C(=O)O)c1)C(=O)CC(C)(C)C ZINC000217770650 CG For-Sale Unstable NR1H4 40 39 CN(Cc1cccc(/C=C\C(=O)O)c1)C(=O)CC(C)(C)C ZINC000217770650 CG For-Sale Unstable AKR1C3 32 42 CCCCn1c(C)c(C=O)c2cc(OCCC)ccc21 ZINC000217770670 CI In-Stock Unstable PLA2G2A 41 39 Cc1ccccc1[C@H](C)NCC(=O)N1c2ccccc2NC(=O)C[C@@H]1C(F)(F)F ZINC000217770690 HH On-Demand Unstable CTSA 46 32 CCOc1cc(C(=O)NC[C@@H]2CCCN2c2nccs2)cc(OCC)c1OCC ZINC000217770720 HH For-Sale Unstable CACNA1I 58 34 O=C(O)/C=C\c1cccc(NC(=O)c2ccccn2)c1 ZINC000217770738 CE For-Sale Anodyne HDAC8 27 45 O=C(O)/C=C\c1cccc(NC(=O)c2ccccn2)c1 ZINC000217770738 CE For-Sale Anodyne GRM4 87 60 O=C(O)/C=C\c1cccc(NC(=O)c2ccccn2)c1 ZINC000217770738 CE For-Sale Anodyne HDAC6 18 45 O=C(O)/C=C\c1cccc(NC(=O)c2ccccn2)c1 ZINC000217770738 CE For-Sale Anodyne TYK2 41 35 O=C(O)/C=C\c1cccc(NC(=O)c2ccccn2)c1 ZINC000217770738 CE For-Sale Anodyne SHH 15 42 O=C(O)/C=C\c1cccc(NC(=O)c2ccccn2)c1 ZINC000217770738 CE For-Sale Anodyne KCNK3 114 63 O=C(O)/C=C\c1cccc(NC(=O)c2ccccn2)c1 ZINC000217770738 CE For-Sale Anodyne KCNK9 73 39 O=C(N/C=C/c1ccccc1F)Nc1cccnc1 ZINC000217770746 CG For-Sale Anodyne KCNQ2 21 41 O=C(N/C=C/c1ccccc1F)Nc1cccnc1 ZINC000217770746 CG For-Sale Anodyne NAMPT 22 46 Cc1ccc(NC(=O)N2CCC(Oc3cc(C)oc(=O)c3)CC2)cc1 ZINC000217770751 EG In-Stock Unstable PRSS2 44 30 Cc1ccc(NC(=O)N2CCC(Oc3cc(C)oc(=O)c3)CC2)cc1 ZINC000217770751 EG In-Stock Unstable EPHX2 52 36 Cc1ccccc1[C@@H](C)NCC(=O)N1c2ccccc2NC(=O)C[C@H]1C(F)(F)F ZINC000217770778 HH On-Demand Unstable CTSA 46 32 CC[C@H](NCCN(C)[C@H](C)CC)c1ccc(Cl)cc1 ZINC000217770786 CI For-Sale Unstable UTS2 44 37 CCOc1cc(C(=O)NC[C@H]2CCCN2c2nccs2)cc(OCC)c1OCC ZINC000217770812 HH For-Sale Unstable CACNA1I 58 34 O=C(O)/C=C\c1cccc(NC(=O)c2ccncc2)c1 ZINC000217770814 CE For-Sale Anodyne HDAC8 18 47 O=C(O)/C=C\c1cccc(NC(=O)c2ccncc2)c1 ZINC000217770814 CE For-Sale Anodyne PRNP 17 43 O=C(O)/C=C\c1cccc(NC(=O)c2ccncc2)c1 ZINC000217770814 CE For-Sale Anodyne TAAR1 22 40 O=C(O)/C=C\c1cccc(NC(=O)c2ccncc2)c1 ZINC000217770814 CE For-Sale Anodyne KCNK3 125 64 O=C(O)/C=C\c1cccc(NC(=O)c2ccncc2)c1 ZINC000217770814 CE For-Sale Anodyne KCNK9 67 47 O=C(NC1[C@@H]2CNC[C@@H]12)[C@@H]1COc2ccccc2O1 ZINC000217770851 CC On-Demand Unstable AKT1 15 49 Cc1cc(O[C@@H]2CCN(C(=O)CCc3ccccc3)C2)cc(=O)n1C ZINC000217770863 EE In-Stock Unstable GRIN2B 22 42 Cc1cc(O[C@@H]2CCN(C(=O)CCc3ccccc3)C2)cc(=O)n1C ZINC000217770863 EE In-Stock Unstable PRSS2 55 33 Cc1ccccc1[C@H](C)NCC(=O)N1c2ccccc2NC(=O)C[C@H]1C(F)(F)F ZINC000217770872 HH On-Demand Unstable CTSA 46 32 COc1cc([C@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc(OC)c1O ZINC000217770876 KH In-Stock Unstable CYP1B1 58 41 COc1cc([C@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc(OC)c1O ZINC000217770876 KH In-Stock Unstable CYP1A1 43 41 COc1cc([C@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc(OC)c1O ZINC000217770876 KH In-Stock Unstable CYP1A2 37 41 COc1cc([C@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc(OC)c1O ZINC000217770876 KH In-Stock Unstable RORC 50 35 CC[C@H](NCCN(C)[C@@H](C)CC)c1ccc(Cl)cc1 ZINC000217770886 CI For-Sale Unstable UTS2 44 37 O=C(O)/C=C\c1ccc(NC(=O)c2ccc(Cl)o2)c(F)c1 ZINC000217770902 DG For-Sale Anodyne HPSE 50 42 O=C(O)/C=C\c1ccc(NC(=O)c2ccc(Cl)o2)c(F)c1 ZINC000217770902 DG For-Sale Anodyne GPR35 46 33 CN(Cc1nccs1)C(=O)c1cccc(OCC(=O)N2CCCCC2)c1 ZINC000217770913 FF In-Stock Unstable CPT1A 71 35 CCCOc1ccc2c(c1)c(C=O)c(C)n2Cc1ccccc1 ZINC000217770916 DJ In-Stock Unstable ALOX5AP 58 33 CCCOc1ccc2c(c1)c(C=O)c(C)n2Cc1ccccc1 ZINC000217770916 DJ In-Stock Unstable PLA2G2A 96 52 COc1ccc(N)c(Br)c1C(=O)O ZINC000217770928 BD For-Sale Unstable ALS 62 37 Cc1cc(O[C@H]2CCN(C(=O)CCc3ccccc3)C2)cc(=O)n1C ZINC000217770942 EE In-Stock Unstable GRIN2B 22 42 Cc1cc(O[C@H]2CCN(C(=O)CCc3ccccc3)C2)cc(=O)n1C ZINC000217770942 EE In-Stock Unstable PRSS2 55 33 CN(CCNS(=O)(=O)N1CCC[C@@H](C(=O)O)C1)C1CC1 ZINC000217770953 DB For-Sale Unstable SLC6A1 79 36 COc1cc([C@@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc(OC)c1O ZINC000217770960 KH In-Stock Unstable CYP1B1 58 41 COc1cc([C@@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc(OC)c1O ZINC000217770960 KH In-Stock Unstable CYP1A1 43 41 COc1cc([C@@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc(OC)c1O ZINC000217770960 KH In-Stock Unstable CYP1A2 37 41 COc1cc([C@@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc(OC)c1O ZINC000217770960 KH In-Stock Unstable RORC 50 35 COC(=O)c1ccc(CNC(=O)[C@@H](C)N[C@@H](C)c2ccccc2Br)cc1 ZINC000217770974 HH On-Demand Unstable FURIN 40 34 CCCOc1ccc2c(c1)c(C=O)c(C)n2CCc1ccccc1 ZINC000217771022 DJ In-Stock Unstable PLA2G2A 69 44 Cc1c(C(=O)O)cc(Br)c(O)c1N ZINC000217771036 BD For-Sale Unstable AKR1C2 67 48 Cc1c(C(=O)O)cc(Br)c(O)c1N ZINC000217771036 BD For-Sale Unstable AKR1C1 65 48 Cc1cc(O[C@@H]2CCN(C(=O)Cc3ccc(F)cc3)C2)cc(=O)n1C ZINC000217771062 EE In-Stock Unstable MLNR 44 52 COC(=O)c1ccc(CNC(=O)[C@H](C)N[C@@H](C)c2ccccc2Br)cc1 ZINC000217771063 HH On-Demand Unstable FURIN 40 34 CN1CCN(C(=O)C[C@H](c2cccc(O)c2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)CC1 ZINC000217771069 KH In-Stock Unstable RORC 40 35 Cc1cc(O[C@H]2CCN(C(=O)Cc3ccc(F)cc3)C2)cc(=O)n1C ZINC000217771132 EE In-Stock Unstable MLNR 44 52 COC(=O)c1ccc(CNC(=O)[C@@H](C)N[C@H](C)c2ccccc2Br)cc1 ZINC000217771134 HH On-Demand Unstable FURIN 40 34 CN1CCN(C(=O)C[C@@H](c2cccc(O)c2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)CC1 ZINC000217771139 KH In-Stock Unstable RORC 40 35 COC(=O)c1ccc(CNC(=O)[C@H](C)N[C@H](C)c2ccccc2Br)cc1 ZINC000217771228 HH On-Demand Unstable FURIN 40 34 Cc1cc(O[C@@H]2CCN(C(=O)c3ccc(F)c(F)c3)C2)cc(=O)n1C ZINC000217771250 EE In-Stock Unstable HRH3 0 45 Cc1cc(O[C@@H]2CCN(C(=O)c3ccc(F)c(F)c3)C2)cc(=O)n1C ZINC000217771250 EE In-Stock Unstable CCR3 0 40 Cc1cc(O[C@@H]2CCN(C(=O)c3ccc(F)c(F)c3)C2)cc(=O)n1C ZINC000217771250 EE In-Stock Unstable L3MBTL3 43 36 COc1ccc(CCNC(=O)CCCCCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@H]23)cc1 ZINC000217771270 JJ In-Stock Unstable HTR7 25 40 COc1ccc(CCNC(=O)CCCCCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@H]23)cc1 ZINC000217771270 JJ In-Stock Unstable SCN9A 0 45 COc1ccc(CCNC(=O)CCCCCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@H]23)cc1 ZINC000217771270 JJ In-Stock Unstable MTNR1A 50 41 COc1ccc(CCNC(=O)CCCCCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@H]23)cc1 ZINC000217771270 JJ In-Stock Unstable MTNR1B 43 35 O=C(NC[C@@H]1CCCN1c1nccs1)c1cccc2ccccc12 ZINC000217771290 EH For-Sale Unstable HCRTR1 39 44 O=C(NC[C@@H]1CCCN1c1nccs1)c1cccc2ccccc12 ZINC000217771290 EH For-Sale Unstable PREP 26 47 O=C(NC[C@@H]1CCCN1c1nccs1)c1cccc2ccccc12 ZINC000217771290 EH For-Sale Unstable HCRTR2 33 44 Cc1cc(NC(=O)[C@@H]2CCC(=O)N2)ccc1/C=C\C(=O)O ZINC000217771329 CD For-Sale Unstable HDAC10 25 40 Cc1cc(NC(=O)[C@@H]2CCC(=O)N2)ccc1/C=C\C(=O)O ZINC000217771329 CD For-Sale Unstable HDAC2 19 40 Cc1cc(NC(=O)[C@@H]2CCC(=O)N2)ccc1/C=C\C(=O)O ZINC000217771329 CD For-Sale Unstable HDAC6 18 40 Cc1cc(NC(=O)[C@@H]2CCC(=O)N2)ccc1/C=C\C(=O)O ZINC000217771329 CD For-Sale Unstable HDAC11 34 40 c1ccc(-n2cc(CN3CCN(Cc4nc5ccccc5s4)CC3)cn2)cc1 ZINC000217771350 GH On-Demand Unstable DRD4 22 62 c1ccc(-n2cc(CN3CCN(Cc4nc5ccccc5s4)CC3)cn2)cc1 ZINC000217771350 GH On-Demand Unstable LTA4H 18 41 Cc1cc(O[C@H]2CCN(C(=O)c3ccc(F)c(F)c3)C2)cc(=O)n1C ZINC000217771351 EE In-Stock Unstable HRH3 0 45 Cc1cc(O[C@H]2CCN(C(=O)c3ccc(F)c(F)c3)C2)cc(=O)n1C ZINC000217771351 EE In-Stock Unstable CCR3 0 40 Cc1cc(O[C@H]2CCN(C(=O)c3ccc(F)c(F)c3)C2)cc(=O)n1C ZINC000217771351 EE In-Stock Unstable L3MBTL3 43 36 COc1ccc(CCNC(=O)CCCCCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@@H]23)cc1 ZINC000217771359 JJ In-Stock Unstable HTR7 25 40 COc1ccc(CCNC(=O)CCCCCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@@H]23)cc1 ZINC000217771359 JJ In-Stock Unstable SCN9A 0 45 COc1ccc(CCNC(=O)CCCCCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@@H]23)cc1 ZINC000217771359 JJ In-Stock Unstable MTNR1A 50 41 COc1ccc(CCNC(=O)CCCCCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@@H]23)cc1 ZINC000217771359 JJ In-Stock Unstable MTNR1B 43 35 O=C(NC[C@H]1CCCN1c1nccs1)c1cccc2ccccc12 ZINC000217771372 EH For-Sale Unstable HCRTR1 39 44 O=C(NC[C@H]1CCCN1c1nccs1)c1cccc2ccccc12 ZINC000217771372 EH For-Sale Unstable PREP 26 47 O=C(NC[C@H]1CCCN1c1nccs1)c1cccc2ccccc12 ZINC000217771372 EH For-Sale Unstable HCRTR2 33 44 CSc1ccc(CC(=O)N2CCCO[C@@H](CN3CCCCC3)C2)cc1 ZINC000217771398 FG In-Stock Unstable OPRK1 23 43 Cc1cc(NC(=O)[C@H]2CCC(=O)N2)ccc1/C=C\C(=O)O ZINC000217771424 CD For-Sale Unstable HDAC10 25 40 Cc1cc(NC(=O)[C@H]2CCC(=O)N2)ccc1/C=C\C(=O)O ZINC000217771424 CD For-Sale Unstable HDAC2 19 40 Cc1cc(NC(=O)[C@H]2CCC(=O)N2)ccc1/C=C\C(=O)O ZINC000217771424 CD For-Sale Unstable HDAC6 18 40 Cc1cc(NC(=O)[C@H]2CCC(=O)N2)ccc1/C=C\C(=O)O ZINC000217771424 CD For-Sale Unstable HDAC11 34 40 Cc1cc(O[C@@H]2CCN(C(=O)c3nc4ccccc4s3)C2)cc(=O)n1C ZINC000217771451 FF In-Stock Unstable TRY1_BOVIN 44 35 Cc1oc(NC(=O)CN2CCN(Cc3nc4ccccc4s3)CC2)c(C#N)c1C ZINC000217771455 HG On-Demand Unstable ACOX1 53 36 Cc1oc(NC(=O)CN2CCN(Cc3nc4ccccc4s3)CC2)c(C#N)c1C ZINC000217771455 HG On-Demand Unstable SLC27A1 24 42 O=C(COc1cccnc1)NC[C@@H]1CCCN1c1nccs1 ZINC000217771478 DD For-Sale Unstable CHRNA7 51 36 CSc1ccc(CC(=O)N2CCCO[C@H](CN3CCCCC3)C2)cc1 ZINC000217771482 FG In-Stock Unstable OPRK1 23 43 CCN(C)C(=O)CNC(=O)c1cc(Cl)c2ccccc2n1 ZINC000217771505 DE On-Demand Unstable TSPO 42 41 CCN(C)C(=O)CNC(=O)c1cc(Cl)c2ccccc2n1 ZINC000217771505 DE On-Demand Unstable PYGL 30 41 Cc1cc(O[C@H]2CCN(C(=O)c3nc4ccccc4s3)C2)cc(=O)n1C ZINC000217771519 FF In-Stock Unstable TRY1_BOVIN 44 35 C[C@H](O)CCNC(=O)/C=C\c1ccccc1Cl ZINC000217771544 CE On-Demand Unstable KCNQ2 52 47 C[C@H](O)CCNC(=O)/C=C\c1ccccc1Cl ZINC000217771544 CE On-Demand Unstable UL26 18 41 C[C@H](O)CCNC(=O)/C=C\c1ccccc1Cl ZINC000217771544 CE On-Demand Unstable SCAF_EBVB9 15 41 O=C(COc1cccnc1)NC[C@H]1CCCN1c1nccs1 ZINC000217771551 DD For-Sale Unstable CHRNA7 51 36 COC(=O)c1ccc(CNC(=O)[C@@H](C)N[C@@H](C)c2cccc3ccccc23)cc1 ZINC000217771567 GH On-Demand Unstable FURIN 47 35 COC(=O)c1ccc(CNC(=O)[C@@H](C)N[C@@H](C)c2cccc3ccccc23)cc1 ZINC000217771567 GH On-Demand Unstable PROC 46 35 Cc1cccc(CN(C)c2cccc(Cl)c2CBr)n1 ZINC000217771601 EJ For-Sale Unstable DFR1 15 40 CC(=O)Nc1cccc(NC(=O)N/C=C/c2ccccc2F)c1 ZINC000217771605 DH For-Sale Unstable KCNK3 110 40 CC(=O)Nc1cccc(NC(=O)N/C=C/c2ccccc2F)c1 ZINC000217771605 DH For-Sale Unstable KCNK9 78 37 C[C@@H](O)CCNC(=O)/C=C\c1ccccc1Cl ZINC000217771629 CE On-Demand Unstable KCNQ2 52 47 C[C@@H](O)CCNC(=O)/C=C\c1ccccc1Cl ZINC000217771629 CE On-Demand Unstable U53 0 41 COC(=O)c1ccc(CNC(=O)[C@H](C)N[C@@H](C)c2cccc3ccccc23)cc1 ZINC000217771650 GH On-Demand Unstable FURIN 47 35 COC(=O)c1ccc(CNC(=O)[C@H](C)N[C@@H](C)c2cccc3ccccc23)cc1 ZINC000217771650 GH On-Demand Unstable PROC 46 35 CCOC(=O)CCNC(=O)CCNC(=O)c1ccccc1Cl ZINC000217771655 ED In-Stock Unstable ECR 43 36 O=C(Cc1cccc2ccccc12)NC[C@@H]1CCCN1c1nccs1 ZINC000217771674 FH For-Sale Unstable PREP 20 47 O=C(Cc1cccc2ccccc12)NC[C@@H]1CCCN1c1nccs1 ZINC000217771674 FH For-Sale Unstable MAPK10 17 41 Cc1n[nH]c(C)c1CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000217771687 DG In-Stock Unstable ACHE 33 46 Cc1n[nH]c(C)c1CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000217771687 DG In-Stock Unstable TACR1 0 40 Cc1n[nH]c(C)c1CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000217771687 DG In-Stock Unstable MC4R 47 41 Cc1n[nH]c(C)c1CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000217771687 DG In-Stock Unstable CTSL 0 41 Cc1n[nH]c(C)c1CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000217771687 DG In-Stock Unstable MPO 41 42 Cc1n[nH]c(C)c1CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000217771687 DG In-Stock Unstable BRS3 23 41 Cc1n[nH]c(C)c1CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000217771687 DG In-Stock Unstable MC5R 48 41 Cc1n[nH]c(C)c1CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000217771687 DG In-Stock Unstable AANAT 55 32 N[C@H](CC(=O)N[C@@H]1C[C@@H]1c1ccccc1)c1ccccc1 ZINC000217771689 CF On-Demand Unstable KDM1A 44 35 N[C@H](CC(=O)N[C@@H]1C[C@@H]1c1ccccc1)c1ccccc1 ZINC000217771689 CF On-Demand Unstable GPR88 0 48 CCCCn1c(C)c(C=O)c2cc(O[C@@H](C)CCC)ccc21 ZINC000217771712 DK In-Stock Unstable PLA2G2A 22 42 COC(=O)c1ccc(CNC(=O)[C@@H](C)N[C@H](C)c2cccc3ccccc23)cc1 ZINC000217771737 GH On-Demand Unstable FURIN 47 35 COC(=O)c1ccc(CNC(=O)[C@@H](C)N[C@H](C)c2cccc3ccccc23)cc1 ZINC000217771737 GH On-Demand Unstable PROC 46 35 O=C(Cc1cccc2ccccc12)NC[C@H]1CCCN1c1nccs1 ZINC000217771740 FH For-Sale Unstable PREP 20 47 O=C(Cc1cccc2ccccc12)NC[C@H]1CCCN1c1nccs1 ZINC000217771740 FH For-Sale Unstable MAPK10 17 41 N[C@H](CC(=O)N[C@H]1C[C@@H]1c1ccccc1)c1ccccc1 ZINC000217771761 CF On-Demand Unstable KDM1A 44 35 N[C@H](CC(=O)N[C@H]1C[C@@H]1c1ccccc1)c1ccccc1 ZINC000217771761 CF On-Demand Unstable GPR88 0 48 Cc1ccc(C(=O)Nc2ccc(/C=C\C(=O)O)c(C)c2)s1 ZINC000217771768 DH For-Sale Unstable KCNK3 49 35 CC[C@H](C)c1ccc(NC(=O)[C@H](N)[C@H](C)CC)cc1 ZINC000217771779 CH For-Sale Unstable SCN2A 29 61 CCCCn1c(C)c(C=O)c2cc(O[C@H](C)CCC)ccc21 ZINC000217771801 DK In-Stock Unstable PLA2G2A 22 42 COC(=O)c1ccc(CNC(=O)[C@H](C)N[C@H](C)c2cccc3ccccc23)cc1 ZINC000217771837 GH On-Demand Unstable FURIN 47 35 COC(=O)c1ccc(CNC(=O)[C@H](C)N[C@H](C)c2cccc3ccccc23)cc1 ZINC000217771837 GH On-Demand Unstable PROC 46 35 COC(=O)[C@@H](NC(=O)c1cccc([N+](=O)[O-])c1)[C@H](C)O ZINC000217771861 CC On-Demand Unstable CACNA1C 55 39 COC(=O)[C@@H](NC(=O)c1cccc([N+](=O)[O-])c1)[C@H](C)O ZINC000217771861 CC On-Demand Unstable CACNA1D 89 39 COC(=O)[C@@H](NC(=O)c1cccc([N+](=O)[O-])c1)[C@H](C)O ZINC000217771861 CC On-Demand Unstable UREA_CANEN 22 47 NC(=O)C[C@H](N)C(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000217771876 BB On-Demand Unstable EPHX2 21 42 O=C(O)Cc1ccc2[nH]c(Br)nc2c1 ZINC000217771901 CD In-Stock Unstable GYRB 41 32 O=C(O)Cc1ccc2[nH]c(Br)nc2c1 ZINC000217771901 CD In-Stock Unstable F7 18 44 COc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)Nc1cccc3[nH]ccc13)C(=O)OC2 ZINC000217771939 IJ In-Stock Unstable IMPDH1 0 74 COc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)Nc1cccc3[nH]ccc13)C(=O)OC2 ZINC000217771939 IJ In-Stock Unstable IMPDH2 0 74 CC[C@@H](C)c1ccc(NC(=O)[C@@H]2C[C@@H](O)CN2)cc1 ZINC000217771955 CD For-Sale Unstable SCN2A 19 48 COC(=O)[C@H](NC(=O)c1cccc([N+](=O)[O-])c1)[C@H](C)O ZINC000217771958 CC On-Demand Unstable CACNA1C 55 39 COC(=O)[C@H](NC(=O)c1cccc([N+](=O)[O-])c1)[C@H](C)O ZINC000217771958 CC On-Demand Unstable CACNA1D 89 39 COC(=O)[C@H](NC(=O)c1cccc([N+](=O)[O-])c1)[C@H](C)O ZINC000217771958 CC On-Demand Unstable UREA_CANEN 22 47 NC(=O)C[C@H](N)C(=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000217771964 BB On-Demand Unstable EPHX2 21 42 Cc1cc(O[C@@H]2CCN(C(=O)CCc3ccc(OCc4ccccc4)cc3)C2)cc(=O)n1C ZINC000217772020 IH In-Stock Unstable KCNH2 20 41 Cc1cc(O[C@@H]2CCN(C(=O)CCc3ccc(OCc4ccccc4)cc3)C2)cc(=O)n1C ZINC000217772020 IH In-Stock Unstable MCHR1 16 40 Cc1cc(O[C@@H]2CCN(C(=O)CCc3ccc(OCc4ccccc4)cc3)C2)cc(=O)n1C ZINC000217772020 IH In-Stock Unstable FFAR1 51 43 Cc1cc(O[C@@H]2CCN(C(=O)CCc3ccc(OCc4ccccc4)cc3)C2)cc(=O)n1C ZINC000217772020 IH In-Stock Unstable FFAR4 47 40 CC[C@H](C)c1ccc(NC(=O)[C@@H]2C[C@@H](O)CN2)cc1 ZINC000217772037 CD For-Sale Unstable SCN2A 19 48 COC(=O)[C@H](NC(=O)c1cccc([N+](=O)[O-])c1)[C@@H](C)O ZINC000217772051 CC On-Demand Unstable CACNA1C 55 39 COC(=O)[C@H](NC(=O)c1cccc([N+](=O)[O-])c1)[C@@H](C)O ZINC000217772051 CC On-Demand Unstable CACNA1D 89 39 COC(=O)[C@H](NC(=O)c1cccc([N+](=O)[O-])c1)[C@@H](C)O ZINC000217772051 CC On-Demand Unstable UREA_CANEN 22 47 COc1ccc(C(=O)NC[C@@H]2CCCN2c2nccs2)c(OC)c1 ZINC000217772053 EF For-Sale Unstable DRD2 34 42 COc1ccc(C(=O)NC[C@@H]2CCCN2c2nccs2)c(OC)c1 ZINC000217772053 EF For-Sale Unstable DRD3 15 42 COc1ccc(C(=O)NC[C@@H]2CCCN2c2nccs2)c(OC)c1 ZINC000217772053 EF For-Sale Unstable ACKR3 62 32 Cc1cc(O[C@H]2CCN(C(=O)CCc3ccc(OCc4ccccc4)cc3)C2)cc(=O)n1C ZINC000217772087 IH In-Stock Unstable KCNH2 20 41 Cc1cc(O[C@H]2CCN(C(=O)CCc3ccc(OCc4ccccc4)cc3)C2)cc(=O)n1C ZINC000217772087 IH In-Stock Unstable MCHR1 16 40 Cc1cc(O[C@H]2CCN(C(=O)CCc3ccc(OCc4ccccc4)cc3)C2)cc(=O)n1C ZINC000217772087 IH In-Stock Unstable FFAR1 51 43 Cc1cc(O[C@H]2CCN(C(=O)CCc3ccc(OCc4ccccc4)cc3)C2)cc(=O)n1C ZINC000217772087 IH In-Stock Unstable FFAR4 47 40 CC[C@@H](C)c1ccc(NC(=O)[C@H]2C[C@@H](O)CN2)cc1 ZINC000217772092 CD For-Sale Unstable SCN2A 19 48 CCC[C@@H](C)Oc1ccc2c(c1)c(C=O)c(C)n2Cc1ccccc1 ZINC000217772106 EK In-Stock Unstable PPARG 23 40 CCC[C@@H](C)Oc1ccc2c(c1)c(C=O)c(C)n2Cc1ccccc1 ZINC000217772106 EK In-Stock Unstable PLA2G2A 84 46 CC[C@@H](NCCOCC1CC1)c1ccc(F)cc1 ZINC000217772109 CG On-Demand Unstable LEF 19 40 COC(=O)Cc1ccc2[nH]c(Cl)nc2c1 ZINC000217772126 BD In-Stock Unstable CHEK2 41 33 COC(=O)Cc1ccc2[nH]c(Cl)nc2c1 ZINC000217772126 BD In-Stock Unstable NR2E3 44 32 COC(=O)Cc1ccc2[nH]c(Cl)nc2c1 ZINC000217772126 BD In-Stock Unstable ALKBH3 47 33 COc1ccc(C(=O)NC[C@H]2CCCN2c2nccs2)c(OC)c1 ZINC000217772143 EF For-Sale Unstable DRD2 34 42 COc1ccc(C(=O)NC[C@H]2CCCN2c2nccs2)c(OC)c1 ZINC000217772143 EF For-Sale Unstable DRD3 15 42 COc1ccc(C(=O)NC[C@H]2CCCN2c2nccs2)c(OC)c1 ZINC000217772143 EF For-Sale Unstable ACKR3 62 32 CC[C@H](C)c1ccc(NC(=O)[C@H]2C[C@@H](O)CN2)cc1 ZINC000217772173 CD For-Sale Unstable SCN2A 19 48 CCC[C@H](C)Oc1ccc2c(c1)c(C=O)c(C)n2Cc1ccccc1 ZINC000217772188 EK In-Stock Unstable PPARG 23 40 CCC[C@H](C)Oc1ccc2c(c1)c(C=O)c(C)n2Cc1ccccc1 ZINC000217772188 EK In-Stock Unstable PLA2G2A 84 46 CC[C@H](NCCOCC1CC1)c1ccc(F)cc1 ZINC000217772193 CG On-Demand Unstable LEF 19 40 CC(C)(C)OC(=O)N1CCCc2cc(CC(=O)O)ccc21 ZINC000217772235 CG In-Stock Unstable AVPR2 26 40 CC(C)(C)OC(=O)N1CCCc2cc(CC(=O)O)ccc21 ZINC000217772235 CG In-Stock Unstable GPR119 27 41 CC(C)CCC(=O)N[C@@H](C)c1cccc(/C=C\C(=O)O)c1 ZINC000217772242 CG For-Sale Unstable AKR1C3 28 41 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccc(-c2ccccc2)cc1 ZINC000217772250 FI For-Sale Unstable HCRTR1 36 45 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccc(-c2ccccc2)cc1 ZINC000217772250 FI For-Sale Unstable PRNP 41 36 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccc(-c2ccccc2)cc1 ZINC000217772250 FI For-Sale Unstable HCRTR2 17 45 O=C(N[C@@H]1C[C@@H]1c1ccccc1)[C@@H]1C[C@@H](O)CN1 ZINC000217772268 BC In-Stock Unstable EPHX2 22 42 C[C@@H](NC[C@@H](O)COc1ccc(-c2ccccc2)cc1)c1cccs1 ZINC000217772294 FJ On-Demand Unstable ADRB2 61 56 C[C@@H](NC[C@@H](O)COc1ccc(-c2ccccc2)cc1)c1cccs1 ZINC000217772294 FJ On-Demand Unstable ADRB1 68 46 C[C@@H](NC[C@@H](O)COc1ccc(-c2ccccc2)cc1)c1cccs1 ZINC000217772294 FJ On-Demand Unstable GRIN1 21 44 C[C@@H](NC[C@@H](O)COc1ccc(-c2ccccc2)cc1)c1cccs1 ZINC000217772294 FJ On-Demand Unstable ADRB3 56 43 CCC[C@@H](C)Oc1ccc2c(c1)c(C=O)c(C)n2CCc1ccccc1 ZINC000217772304 EK In-Stock Unstable PLA2G2A 53 38 O=C(NC[C@H]1CCCN1c1nccs1)c1ccc(-c2ccccc2)cc1 ZINC000217772325 FI For-Sale Unstable HCRTR1 36 45 O=C(NC[C@H]1CCCN1c1nccs1)c1ccc(-c2ccccc2)cc1 ZINC000217772325 FI For-Sale Unstable PRNP 41 36 O=C(NC[C@H]1CCCN1c1nccs1)c1ccc(-c2ccccc2)cc1 ZINC000217772325 FI For-Sale Unstable HCRTR2 17 45 CN(CCCO)S(=O)(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217772328 DD For-Sale Unstable PPX1 0 43 COC(=O)Cc1ccc2c(c1)CCCN2C(=O)OC(C)(C)C ZINC000217772336 DG In-Stock Unstable AVPR2 29 43 COC(=O)Cc1ccc2c(c1)CCCN2C(=O)OC(C)(C)C ZINC000217772336 DG In-Stock Unstable GPR119 26 42 CC(C)CCC(=O)N[C@H](C)c1cccc(/C=C\C(=O)O)c1 ZINC000217772343 CG For-Sale Unstable AKR1C3 28 41 Cc1ccc(C)c([C@@H](C)N[C@@H]2CCN(C(=O)OC(C)(C)C)C2)c1 ZINC000217772349 DH For-Sale Unstable MC4R 15 42 Cc1ccc(C)c([C@@H](C)N[C@@H]2CCN(C(=O)OC(C)(C)C)C2)c1 ZINC000217772349 DH For-Sale Unstable EPHX2 17 49 Cc1ccc(C)c([C@@H](C)N[C@@H]2CCN(C(=O)OC(C)(C)C)C2)c1 ZINC000217772349 DH For-Sale Unstable GPR119 40 46 O=C(N[C@@H]1C[C@@H]1c1ccccc1)[C@H]1C[C@H](O)CN1 ZINC000217772350 BC In-Stock Unstable EPHX2 22 42 C[C@H](NC[C@@H](O)COc1ccc(-c2ccccc2)cc1)c1cccs1 ZINC000217772374 FJ On-Demand Unstable ADRB2 61 56 C[C@H](NC[C@@H](O)COc1ccc(-c2ccccc2)cc1)c1cccs1 ZINC000217772374 FJ On-Demand Unstable ADRB1 68 46 C[C@H](NC[C@@H](O)COc1ccc(-c2ccccc2)cc1)c1cccs1 ZINC000217772374 FJ On-Demand Unstable GRIN1 21 44 C[C@H](NC[C@@H](O)COc1ccc(-c2ccccc2)cc1)c1cccs1 ZINC000217772374 FJ On-Demand Unstable ADRB3 56 43 CCC[C@H](C)Oc1ccc2c(c1)c(C=O)c(C)n2CCc1ccccc1 ZINC000217772388 EK In-Stock Unstable PLA2G2A 53 38 Cc1ccc(C)c([C@H](C)N[C@@H]2CCN(C(=O)OC(C)(C)C)C2)c1 ZINC000217772416 DH For-Sale Unstable MC4R 15 42 Cc1ccc(C)c([C@H](C)N[C@@H]2CCN(C(=O)OC(C)(C)C)C2)c1 ZINC000217772416 DH For-Sale Unstable EPHX2 17 49 Cc1ccc(C)c([C@H](C)N[C@@H]2CCN(C(=O)OC(C)(C)C)C2)c1 ZINC000217772416 DH For-Sale Unstable GPR119 40 46 O=C(N[C@@H]1C[C@@H]1c1ccccc1)[C@H]1C[C@@H](O)CN1 ZINC000217772419 BC In-Stock Unstable EPHX2 22 42 C[C@H](O)CCNC(=O)/C=C\c1ccc(Cl)cc1Cl ZINC000217772436 CF For-Sale Unstable KCNQ2 48 36 C[C@H](O)CCNC(=O)/C=C\c1ccc(Cl)cc1Cl ZINC000217772436 CF For-Sale Unstable PYGL 23 42 C[C@H](O)CCNC(=O)/C=C\c1ccc(Cl)cc1Cl ZINC000217772436 CF For-Sale Unstable HDAC9 15 47 C[C@H](O)CCNC(=O)/C=C\c1ccc(Cl)cc1Cl ZINC000217772436 CF For-Sale Unstable HDAC7 22 47 C[C@H](O)CCNC(=O)/C=C\c1ccc(Cl)cc1Cl ZINC000217772436 CF For-Sale Unstable BOTA 35 58 C[C@@H](NC[C@H](O)COc1ccc(-c2ccccc2)cc1)c1cccs1 ZINC000217772473 FJ On-Demand Unstable ADRB2 61 56 C[C@@H](NC[C@H](O)COc1ccc(-c2ccccc2)cc1)c1cccs1 ZINC000217772473 FJ On-Demand Unstable ADRB1 68 46 C[C@@H](NC[C@H](O)COc1ccc(-c2ccccc2)cc1)c1cccs1 ZINC000217772473 FJ On-Demand Unstable GRIN1 21 44 C[C@@H](NC[C@H](O)COc1ccc(-c2ccccc2)cc1)c1cccs1 ZINC000217772473 FJ On-Demand Unstable ADRB3 56 43 COC1CCN(C2CCN(C(=O)C(c3ccccc3)c3ccccc3)CC2)CC1 ZINC000217772486 GH In-Stock Unstable CHRM2 71 41 COC1CCN(C2CCN(C(=O)C(c3ccccc3)c3ccccc3)CC2)CC1 ZINC000217772486 GH In-Stock Unstable CHRM1 24 48 COC1CCN(C2CCN(C(=O)C(c3ccccc3)c3ccccc3)CC2)CC1 ZINC000217772486 GH In-Stock Unstable HRH1 18 43 COC1CCN(C2CCN(C(=O)C(c3ccccc3)c3ccccc3)CC2)CC1 ZINC000217772486 GH In-Stock Unstable SLC6A3 17 40 COC1CCN(C2CCN(C(=O)C(c3ccccc3)c3ccccc3)CC2)CC1 ZINC000217772486 GH In-Stock Unstable CHRM4 34 41 COC1CCN(C2CCN(C(=O)C(c3ccccc3)c3ccccc3)CC2)CC1 ZINC000217772486 GH In-Stock Unstable CHRM5 21 41 COC1CCN(C2CCN(C(=O)C(c3ccccc3)c3ccccc3)CC2)CC1 ZINC000217772486 GH In-Stock Unstable AGTR2 82 38 COC1CCN(C2CCN(C(=O)C(c3ccccc3)c3ccccc3)CC2)CC1 ZINC000217772486 GH In-Stock Unstable CCR3 36 43 COC1CCN(C2CCN(C(=O)C(c3ccccc3)c3ccccc3)CC2)CC1 ZINC000217772486 GH In-Stock Unstable L3MBTL3 84 45 Cc1ccc(C)c([C@@H](C)N[C@H]2CCN(C(=O)OC(C)(C)C)C2)c1 ZINC000217772501 DH For-Sale Unstable MC4R 15 42 Cc1ccc(C)c([C@@H](C)N[C@H]2CCN(C(=O)OC(C)(C)C)C2)c1 ZINC000217772501 DH For-Sale Unstable EPHX2 17 49 Cc1ccc(C)c([C@@H](C)N[C@H]2CCN(C(=O)OC(C)(C)C)C2)c1 ZINC000217772501 DH For-Sale Unstable GPR119 40 46 C[C@@H](O)CCNC(=O)/C=C\c1ccc(Cl)cc1Cl ZINC000217772531 CF For-Sale Unstable KCNQ2 48 36 C[C@@H](O)CCNC(=O)/C=C\c1ccc(Cl)cc1Cl ZINC000217772531 CF For-Sale Unstable PYGL 23 42 C[C@@H](O)CCNC(=O)/C=C\c1ccc(Cl)cc1Cl ZINC000217772531 CF For-Sale Unstable HDAC9 15 47 C[C@@H](O)CCNC(=O)/C=C\c1ccc(Cl)cc1Cl ZINC000217772531 CF For-Sale Unstable HDAC7 22 47 C[C@@H](O)CCNC(=O)/C=C\c1ccc(Cl)cc1Cl ZINC000217772531 CF For-Sale Unstable BOTA 35 58 C[C@H](NC[C@H](O)COc1ccc(-c2ccccc2)cc1)c1cccs1 ZINC000217772564 FJ On-Demand Unstable ADRB2 61 56 C[C@H](NC[C@H](O)COc1ccc(-c2ccccc2)cc1)c1cccs1 ZINC000217772564 FJ On-Demand Unstable ADRB1 68 46 C[C@H](NC[C@H](O)COc1ccc(-c2ccccc2)cc1)c1cccs1 ZINC000217772564 FJ On-Demand Unstable GRIN1 21 44 C[C@H](NC[C@H](O)COc1ccc(-c2ccccc2)cc1)c1cccs1 ZINC000217772564 FJ On-Demand Unstable ADRB3 56 43 Cc1ccc(C)c([C@H](C)N[C@H]2CCN(C(=O)OC(C)(C)C)C2)c1 ZINC000217772576 DH For-Sale Unstable MC4R 15 42 Cc1ccc(C)c([C@H](C)N[C@H]2CCN(C(=O)OC(C)(C)C)C2)c1 ZINC000217772576 DH For-Sale Unstable EPHX2 17 49 Cc1ccc(C)c([C@H](C)N[C@H]2CCN(C(=O)OC(C)(C)C)C2)c1 ZINC000217772576 DH For-Sale Unstable GPR119 40 46 C[C@H](O)CCNC(=O)/C=C\c1cccc(Br)c1 ZINC000217772620 CE For-Sale Unstable HDAC8 58 38 CC[C@@H](N[C@@H]1CCN(C(=O)OC(C)(C)C)C1)c1ccc(F)cc1 ZINC000217772692 DH On-Demand Unstable GPR119 50 49 CC[C@@H](N[C@@H]1CCN(C(=O)OC(C)(C)C)C1)c1ccc(F)cc1 ZINC000217772692 DH On-Demand Unstable SFRP1 66 41 CC[C@@H](N[C@@H]1CCN(C(=O)OC(C)(C)C)C1)c1ccc(F)cc1 ZINC000217772692 DH On-Demand Unstable WNT3 50 35 C[C@@H](O)CCNC(=O)/C=C\c1cccc(Br)c1 ZINC000217772706 CE On-Demand Unstable HDAC8 58 38 CCCCn1c(C)c(C=O)c2cc(OCC(C)C)ccc21 ZINC000217772716 CJ In-Stock Unstable PLA2G2A 22 45 O=C(C[C@H]1CCCN1)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000217772757 BD For-Sale Unstable EPHX2 22 43 O=C(C[C@H]1CCCN1)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000217772757 BD For-Sale Unstable CHRNA10 29 40 CC[C@H](N[C@@H]1CCN(C(=O)OC(C)(C)C)C1)c1ccc(F)cc1 ZINC000217772769 DH On-Demand Unstable GPR119 50 49 CC[C@H](N[C@@H]1CCN(C(=O)OC(C)(C)C)C1)c1ccc(F)cc1 ZINC000217772769 DH On-Demand Unstable SFRP1 66 41 CC[C@H](N[C@@H]1CCN(C(=O)OC(C)(C)C)C1)c1ccc(F)cc1 ZINC000217772769 DH On-Demand Unstable WNT3 50 35 Nc1ncc(Br)cc1[C@H](N)C(=O)O ZINC000217772775 BC For-Sale Unstable CACNA2D1 0 41 C[C@H](O)CCNC(=O)/C=C\c1ccc(Br)cc1 ZINC000217772778 CE For-Sale Unstable HDAC9 51 37 C[C@H](O)CCNC(=O)/C=C\c1ccc(Br)cc1 ZINC000217772778 CE For-Sale Unstable HDAC7 49 37 O=C(C[C@H]1CCCN1)N[C@H]1C[C@@H]1c1ccccc1 ZINC000217772843 BD For-Sale Unstable EPHX2 22 43 O=C(C[C@H]1CCCN1)N[C@H]1C[C@@H]1c1ccccc1 ZINC000217772843 BD For-Sale Unstable CHRNA10 29 40 CC[C@@H](N[C@H]1CCN(C(=O)OC(C)(C)C)C1)c1ccc(F)cc1 ZINC000217772849 DH On-Demand Unstable GPR119 50 49 CC[C@@H](N[C@H]1CCN(C(=O)OC(C)(C)C)C1)c1ccc(F)cc1 ZINC000217772849 DH On-Demand Unstable SFRP1 66 41 CC[C@@H](N[C@H]1CCN(C(=O)OC(C)(C)C)C1)c1ccc(F)cc1 ZINC000217772849 DH On-Demand Unstable WNT3 50 35 Nc1ncc(Br)cc1[C@@H](N)C(=O)O ZINC000217772856 BC For-Sale Unstable CACNA2D1 0 41 C[C@@H](O)CCNC(=O)/C=C\c1ccc(Br)cc1 ZINC000217772873 CE On-Demand Unstable HDAC9 51 37 C[C@@H](O)CCNC(=O)/C=C\c1ccc(Br)cc1 ZINC000217772873 CE On-Demand Unstable HDAC7 49 37 O=C(N/C=C/c1ccccc1F)Nc1ccccc1N1CCOCC1 ZINC000217772906 EG For-Sale Unstable KCNQ2 91 42 O=C(N/C=C/c1ccccc1F)Nc1ccccc1N1CCOCC1 ZINC000217772906 EG For-Sale Unstable AKR1C3 0 40 CC(C)Cc1ccc([C@@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2)cc1 ZINC000217772930 CD On-Demand Unstable CTSC 30 41 CC[C@H](N[C@H]1CCN(C(=O)OC(C)(C)C)C1)c1ccc(F)cc1 ZINC000217772936 DH On-Demand Unstable GPR119 50 49 CC[C@H](N[C@H]1CCN(C(=O)OC(C)(C)C)C1)c1ccc(F)cc1 ZINC000217772936 DH On-Demand Unstable SFRP1 66 41 CC[C@H](N[C@H]1CCN(C(=O)OC(C)(C)C)C1)c1ccc(F)cc1 ZINC000217772936 DH On-Demand Unstable WNT3 50 35 CCC[C@@H](NCCN(C)[C@@H](C)CC)c1ccc(Cl)cc1 ZINC000217772949 CJ For-Sale Unstable UTS2 45 37 O=C(CC[C@H]1CCCNC1)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000217772963 CE For-Sale Unstable EPHX2 21 40 Cc1c(C=O)c2cc(OCC(C)C)ccc2n1Cc1ccccc1 ZINC000217772970 DJ In-Stock Unstable CASR 19 41 Cc1c(C=O)c2cc(OCC(C)C)ccc2n1Cc1ccccc1 ZINC000217772970 DJ In-Stock Unstable ALOX5AP 48 32 Cc1c(C=O)c2cc(OCC(C)C)ccc2n1Cc1ccccc1 ZINC000217772970 DJ In-Stock Unstable PLA2G2A 89 47 Cc1c(C=O)c2cc(OCC(C)C)ccc2n1Cc1ccccc1 ZINC000217772970 DJ In-Stock Unstable PLA2G10 42 34 Cc1c(C=O)c2cc(OCC(C)C)ccc2n1Cc1ccccc1 ZINC000217772970 DJ In-Stock Unstable PLA2G2D 40 32 CC(C)Cc1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2)cc1 ZINC000217773001 CD On-Demand Unstable CTSC 30 41 CC(C)Cc1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2)cc1 ZINC000217773001 CD On-Demand Unstable SLC22A20 0 43 CN1CCN(c2ccc(NC(=O)N/C=C/c3ccccc3F)cc2)CC1 ZINC000217773009 FG For-Sale Unstable PRNP 51 49 CN1CCN(c2ccc(NC(=O)N/C=C/c3ccccc3F)cc2)CC1 ZINC000217773009 FG For-Sale Unstable MTOR 25 43 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccc(Cn2ccnc2)cc1 ZINC000217773010 FF In-Stock Unstable TBXAS1 25 42 Cc1cc(=O)c(O)c([C@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccsc2)o1 ZINC000217773024 II In-Stock Unstable SSTR4 45 32 O=C(CC[C@H]1CCCNC1)N[C@H]1C[C@@H]1c1ccccc1 ZINC000217773030 CE For-Sale Unstable EPHX2 21 40 CCC[C@H](NCCN(C)[C@@H](C)CC)c1ccc(Cl)cc1 ZINC000217773034 CJ For-Sale Unstable UTS2 45 37 O=C(O)CCc1ccc2[nH]c(Cl)nc2c1 ZINC000217773054 BE In-Stock Unstable GYRB 0 40 O=C(O)CCc1ccc2[nH]c(Cl)nc2c1 ZINC000217773054 BE In-Stock Unstable FFAR1 66 40 O=C(O)CCc1ccc2[nH]c(Cl)nc2c1 ZINC000217773054 BE In-Stock Unstable NR2E3 42 31 CC(C)C1=C(C(=O)N2[C@H](C(=O)N3CC4(CC4)NC[C@@H]3C)CC[C@H]2C)SC2=N[C@@](C)(c3ccc(Cl)nc3)[C@@H](c3ccc(Cl)c(F)c3)N21 ZINC000217773060 KK Annotated Unstable MDM2 19 83 CC(C)Cc1ccc([C@@H](C)NC(=O)[C@H]2C[C@@H](O)CN2)cc1 ZINC000217773079 CD On-Demand Unstable CTSC 30 41 CC(C)Cc1ccc([C@@H](C)NC(=O)[C@H]2C[C@@H](O)CN2)cc1 ZINC000217773079 CD On-Demand Unstable SLC22A20 0 43 Cc1c(C=O)c2cc(OCC(C)C)ccc2n1CCc1ccccc1 ZINC000217773080 EK In-Stock Unstable PLA2G2A 58 39 O=C(NC[C@H]1CCCN1c1nccs1)c1ccc(Cn2ccnc2)cc1 ZINC000217773091 FF In-Stock Unstable TBXAS1 25 42 Cc1cc(=O)c(O)c([C@@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccsc2)o1 ZINC000217773099 II In-Stock Unstable SSTR4 45 32 O=C(N/C=C/c1ccccc1F)Nc1ccc(N2CCCCC2)cc1 ZINC000217773120 EJ For-Sale Unstable KCNQ2 42 41 O=C(N/C=C/c1ccccc1F)Nc1ccc(N2CCCCC2)cc1 ZINC000217773120 EJ For-Sale Unstable PRNP 41 37 CCc1ccc(/C=C\C(=O)NCC[C@@H](C)O)cc1 ZINC000217773121 BE On-Demand Unstable HDAC8 19 41 CCc1ccc(/C=C\C(=O)NCC[C@@H](C)O)cc1 ZINC000217773121 BE On-Demand Unstable HDAC9 44 35 CCc1ccc(/C=C\C(=O)NCC[C@@H](C)O)cc1 ZINC000217773121 BE On-Demand Unstable HDAC7 48 35 O=C(O)CCc1ccc2[nH]c(Br)nc2c1 ZINC000217773165 CE In-Stock Unstable FFAR1 65 38 CC(C)Cc1ccc([C@H](C)NC(=O)[C@H]2C[C@@H](O)CN2)cc1 ZINC000217773170 CD On-Demand Unstable CTSC 30 41 CC(C)Cc1ccc([C@H](C)NC(=O)[C@H]2C[C@@H](O)CN2)cc1 ZINC000217773170 CD On-Demand Unstable SLC22A20 0 43 CCCCOc1ccc2c(c1)c(C=O)c(C)n2C ZINC000217773173 BG In-Stock Unstable PLA2G4B 46 30 O=C(CN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCc1ccccn1 ZINC000217773200 GF In-Stock Unstable SCN9A 0 45 CCc1ccc(/C=C\C(=O)NCC[C@H](C)O)cc1 ZINC000217773202 BE For-Sale Unstable PYGL 0 42 CCc1ccc(/C=C\C(=O)NCC[C@H](C)O)cc1 ZINC000217773202 BE For-Sale Unstable HDAC8 24 41 CCc1ccc(/C=C\C(=O)NCC[C@H](C)O)cc1 ZINC000217773202 BE For-Sale Unstable HDAC9 44 35 CCc1ccc(/C=C\C(=O)NCC[C@H](C)O)cc1 ZINC000217773202 BE For-Sale Unstable HDAC7 48 35 CCCCOc1ccc2c(c1)c(C=O)c(C)n2CC ZINC000217773266 CH In-Stock Unstable PLA2G2A 40 38 COC(=O)CCc1ccc2[nH]c(Br)nc2c1 ZINC000217773274 CE In-Stock Unstable P2RY12 0 46 O=C(CN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCc1ccccn1 ZINC000217773277 GF In-Stock Unstable SCN9A 0 45 C[C@H](O)CCNC(=O)/C=C\c1ccc(Cl)s1 ZINC000217773290 CE On-Demand Unstable SCAF_EBVB9 15 42 CCCCOc1ccc2c(c1)c(C=O)c(C)n2CCC ZINC000217773360 CI In-Stock Unstable PLA2G2A 33 48 C[C@@H](O)CCNC(=O)/C=C\c1ccc(Cl)s1 ZINC000217773369 CE On-Demand Unstable SCAF_EBVB9 15 42 Cc1cccc(CN(C)c2cc(Cl)ccc2CBr)n1 ZINC000217773377 EJ For-Sale Unstable DFR1 15 41 COC(=O)CCc1ccc2[nH]c(Cl)nc2c1 ZINC000217773384 BE In-Stock Unstable P2RY12 0 46 C[C@H](O)CCNC(=O)/C=C\c1cccc(C#N)c1 ZINC000217773444 BD For-Sale Unstable PYGL 0 40 O=C(O)/C=C\c1cccc(NC(=O)c2cccc(F)c2)n1 ZINC000217773457 CF For-Sale Anodyne HTR1F 15 42 O=C(O)/C=C\c1cccc(NC(=O)c2cccc(F)c2)n1 ZINC000217773457 CF For-Sale Anodyne GRM5 20 45 O=C(O)/C=C\c1cccc(NC(=O)c2cccc(F)c2)n1 ZINC000217773457 CF For-Sale Anodyne KCNK3 77 49 O=C(O)/C=C\c1cccc(NC(=O)c2cccc(F)c2)n1 ZINC000217773457 CF For-Sale Anodyne KCNK9 37 46 CCCCOc1ccc2c(c1)c(C=O)c(C)n2CCCC ZINC000217773458 CJ In-Stock Unstable PLA2G2A 42 40 CCCCOc1ccc2c(c1)c(C=O)c(C)n2CCCC ZINC000217773458 CJ In-Stock Unstable RORB 0 40 Cc1cccc(CN(C)c2ccc(Cl)cc2CBr)n1 ZINC000217773508 EJ For-Sale Unstable DFR1 15 40 C[C@@H](O)CCNC(=O)/C=C\c1cccc(C#N)c1 ZINC000217773522 BD On-Demand Unstable PYGL 0 40 CC(C)[C@@H]1CC[C@@H](N)[C@@H](Cc2cc(F)ccc2F)C1 ZINC000217773533 CH For-Sale Unstable DPP4 21 45 O=C(N/C=C/c1ccccc1F)Nc1cccc2ccccc12 ZINC000217773536 DJ For-Sale Anodyne TRPV1 25 40 COc1ccc(/C=C\C(=O)O)cc1NC(=O)c1ccoc1 ZINC000217773542 CF For-Sale Unstable TUBB1 48 39 COc1ccc(/C=C\C(=O)O)cc1NC(=O)c1ccoc1 ZINC000217773542 CF For-Sale Unstable ABCG2 21 40 COc1ccc(/C=C\C(=O)O)cc1NC(=O)c1ccoc1 ZINC000217773542 CF For-Sale Unstable KCNK3 22 42 CC(C)(C)c1ccc(C(=O)NC[C@@H]2CCCN2c2nccs2)cc1 ZINC000217773549 EH For-Sale Unstable IKBKB 15 44 CC(C)(C)c1ccc(C(=O)NC[C@@H]2CCCN2c2nccs2)cc1 ZINC000217773549 EH For-Sale Unstable CACNA1I 42 35 C[C@H](N)C(=O)c1c(F)cccc1Br ZINC000217773552 BE For-Sale Unstable CES2 27 43 C[C@H](N)C(=O)c1c(F)cccc1Br ZINC000217773552 BE For-Sale Unstable DAC 23 41 CCCCOc1ccc2c(c1)c(C=O)c(C)n2CC(C)C ZINC000217773570 CJ In-Stock Unstable PLA2G2A 26 42 C[C@@H](NC(=O)c1occc1COc1ccccc1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773573 HF On-Demand Unstable CA2 63 44 C[C@@H](NC(=O)c1occc1COc1ccccc1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773573 HF On-Demand Unstable CA1 47 43 C[C@@H](NC(=O)c1occc1COc1ccccc1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773573 HF On-Demand Unstable CA7 42 44 C[C@@H](NC(=O)c1occc1COc1ccccc1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773573 HF On-Demand Unstable PTGER3 41 34 C[C@@H](NC(=O)c1occc1COc1ccccc1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773573 HF On-Demand Unstable ACACA 41 37 C[C@@H](NC(=O)c1occc1COc1ccccc1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773573 HF On-Demand Unstable CA5B 48 37 C[C@@H](NC(=O)c1occc1COc1ccccc1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773573 HF On-Demand Unstable CA4 49 37 C[C@@H](NC(=O)c1occc1COc1ccccc1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773573 HF On-Demand Unstable CA5A 50 37 C[C@@H](NC(=O)c1occc1COc1ccccc1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773573 HF On-Demand Unstable CA12 36 44 C[C@@H](NC(=O)c1occc1COc1ccccc1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773573 HF On-Demand Unstable ADAMTS4 44 37 C[C@@H](NC(=O)c1occc1COc1ccccc1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773573 HF On-Demand Unstable CA9 40 35 Cc1ccccc1/C=C\C(=O)NCC[C@@H](C)O ZINC000217773599 BD On-Demand Unstable U53 0 40 C[C@@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773601 DB For-Sale Unstable CA12 21 40 C[C@@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773601 DB For-Sale Unstable CA9 22 40 C[C@@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773601 DB For-Sale Unstable P96878_MYCTU 36 40 COc1ccc(/C=C\C(=O)O)cc1NC(=O)CC(F)(F)F ZINC000217773626 DF For-Sale Unstable TUBB1 54 39 CC(C)[C@H]1CC[C@@H](N)[C@@H](Cc2cc(F)ccc2F)C1 ZINC000217773631 CH For-Sale Unstable DPP4 21 45 C[C@@H](N)C(=O)c1c(F)cccc1Br ZINC000217773637 BE For-Sale Unstable CES2 27 43 C[C@@H](N)C(=O)c1c(F)cccc1Br ZINC000217773637 BE For-Sale Unstable DAC 23 41 CC(C)(C)c1ccc(C(=O)NC[C@H]2CCCN2c2nccs2)cc1 ZINC000217773638 EH For-Sale Unstable IKBKB 15 44 CC(C)(C)c1ccc(C(=O)NC[C@H]2CCCN2c2nccs2)cc1 ZINC000217773638 EH For-Sale Unstable CACNA1I 42 35 COc1cc(C(=O)NCCN2CCNC2=O)ccc1O ZINC000217773642 CC In-Stock Unstable DRD2 25 40 COc1cc(C(=O)NCCN2CCNC2=O)ccc1O ZINC000217773642 CC In-Stock Unstable DRD4 49 37 COc1cc(C(=O)NCCN2CCNC2=O)ccc1O ZINC000217773642 CC In-Stock Unstable DRD3 30 41 COc1cc(C(=O)NCCN2CCNC2=O)ccc1O ZINC000217773642 CC In-Stock Unstable PLD1 41 40 COc1cc(C(=O)NCCN2CCNC2=O)ccc1O ZINC000217773642 CC In-Stock Unstable PLD2 62 46 COC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217773651 DG For-Sale Unstable ACR 53 39 C[C@H](NC(=O)c1occc1COc1ccccc1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773667 HF On-Demand Unstable CA2 63 44 C[C@H](NC(=O)c1occc1COc1ccccc1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773667 HF On-Demand Unstable CA1 47 43 C[C@H](NC(=O)c1occc1COc1ccccc1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773667 HF On-Demand Unstable CA7 42 44 C[C@H](NC(=O)c1occc1COc1ccccc1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773667 HF On-Demand Unstable PTGER3 41 34 C[C@H](NC(=O)c1occc1COc1ccccc1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773667 HF On-Demand Unstable ACACA 41 37 C[C@H](NC(=O)c1occc1COc1ccccc1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773667 HF On-Demand Unstable CA5B 48 37 C[C@H](NC(=O)c1occc1COc1ccccc1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773667 HF On-Demand Unstable CA4 49 37 C[C@H](NC(=O)c1occc1COc1ccccc1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773667 HF On-Demand Unstable CA5A 50 37 C[C@H](NC(=O)c1occc1COc1ccccc1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773667 HF On-Demand Unstable CA12 36 44 C[C@H](NC(=O)c1occc1COc1ccccc1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773667 HF On-Demand Unstable ADAMTS4 44 37 C[C@H](NC(=O)c1occc1COc1ccccc1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773667 HF On-Demand Unstable CA9 40 35 C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773681 DB For-Sale Unstable CA12 21 40 C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773681 DB For-Sale Unstable CA9 22 40 C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773681 DB For-Sale Unstable P96878_MYCTU 36 40 Cc1ccccc1/C=C\C(=O)NCC[C@H](C)O ZINC000217773696 BD For-Sale Unstable U53 0 40 CCCCOc1ccc2c(c1)c(C=O)c(C)n2Cc1ccccc1 ZINC000217773698 DJ In-Stock Unstable ALOX5AP 66 36 CCCCOc1ccc2c(c1)c(C=O)c(C)n2Cc1ccccc1 ZINC000217773698 DJ In-Stock Unstable PLA2G2A 112 54 CCCCOc1ccc2c(c1)c(C=O)c(C)n2Cc1ccccc1 ZINC000217773698 DJ In-Stock Unstable PLA2G4B 41 37 CC[C@@H](C)C(=O)Nc1cc(/C=C\C(=O)O)ccc1OC ZINC000217773710 CF For-Sale Unstable TUBB1 47 38 CC[C@@H](C)C(=O)Nc1cc(/C=C\C(=O)O)ccc1OC ZINC000217773710 CF For-Sale Unstable AKR1C3 40 42 CC(C)[C@@H]1CC[C@H](N)[C@@H](Cc2cc(F)ccc2F)C1 ZINC000217773714 CH For-Sale Unstable DPP4 21 45 Cc1cc(=O)c2cc(CCC(=O)O)ccc2[nH]1 ZINC000217773720 BD In-Stock Unstable FFAR1 70 43 C[C@@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773758 DB For-Sale Unstable CA12 21 40 C[C@@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773758 DB For-Sale Unstable CA9 22 40 C[C@@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773758 DB For-Sale Unstable P96878_MYCTU 36 40 COc1ccc(/C=C\C(=O)NCC[C@H](C)O)cc1F ZINC000217773795 CD For-Sale Unstable TOP2A 15 41 COc1ccc(/C=C\C(=O)NCC[C@H](C)O)cc1F ZINC000217773795 CD For-Sale Unstable DRD3 15 44 COc1ccc(/C=C\C(=O)NCC[C@H](C)O)cc1F ZINC000217773795 CD For-Sale Unstable PYGL 23 42 COc1ccc(/C=C\C(=O)NCC[C@H](C)O)cc1F ZINC000217773795 CD For-Sale Unstable HPSE 19 43 COc1ccc(/C=C\C(=O)NCC[C@H](C)O)cc1F ZINC000217773795 CD For-Sale Unstable TUBB1 48 47 CC[C@H](C)C(=O)Nc1cc(/C=C\C(=O)O)ccc1OC ZINC000217773800 CF For-Sale Unstable TUBB1 47 38 CC[C@H](C)C(=O)Nc1cc(/C=C\C(=O)O)ccc1OC ZINC000217773800 CF For-Sale Unstable AKR1C3 40 42 CC(C)[C@H]1CC[C@H](N)[C@@H](Cc2cc(F)ccc2F)C1 ZINC000217773801 CH For-Sale Unstable DPP4 21 45 CCCCOc1ccc2c(c1)c(C=O)c(C)n2CCc1ccccc1 ZINC000217773814 EK In-Stock Unstable PLA2G2A 74 46 C[C@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773849 DB For-Sale Unstable CA12 21 40 C[C@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773849 DB For-Sale Unstable CA9 22 40 C[C@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1ccc(S(N)(=O)=O)cc1 ZINC000217773849 DB For-Sale Unstable P96878_MYCTU 36 40 O=C(N/C=C/c1ccccc1F)Nc1ccc2ccccc2c1 ZINC000217773859 DJ For-Sale Anodyne UL80 47 38 O=C(N/C=C/c1ccccc1F)Nc1ccc2ccccc2c1 ZINC000217773859 DJ For-Sale Anodyne IMDH_CRYPV 26 40 COc1ccc(/C=C\C(=O)NCC[C@@H](C)O)cc1F ZINC000217773876 CD For-Sale Unstable TOP2A 15 41 COc1ccc(/C=C\C(=O)NCC[C@@H](C)O)cc1F ZINC000217773876 CD For-Sale Unstable DRD3 15 44 COc1ccc(/C=C\C(=O)NCC[C@@H](C)O)cc1F ZINC000217773876 CD For-Sale Unstable PYGL 23 42 COc1ccc(/C=C\C(=O)NCC[C@@H](C)O)cc1F ZINC000217773876 CD For-Sale Unstable HPSE 19 43 COc1ccc(/C=C\C(=O)NCC[C@@H](C)O)cc1F ZINC000217773876 CD For-Sale Unstable TUBB1 48 47 COc1ccccc1C(=O)Nc1ncc(/C=C\C(=O)O)s1 ZINC000217773883 DF For-Sale Unstable KCNA3 41 37 COc1ccccc1C(=O)Nc1ncc(/C=C\C(=O)O)s1 ZINC000217773883 DF For-Sale Unstable MAP1 24 41 COc1ccccc1C(=O)Nc1ncc(/C=C\C(=O)O)s1 ZINC000217773883 DF For-Sale Unstable KCNK3 57 45 COc1ccccc1C(=O)Nc1ncc(/C=C\C(=O)O)s1 ZINC000217773883 DF For-Sale Unstable KCNK9 53 45 Cc1cc(O[C@@H]2CCN(S(=O)(=O)c3ccccc3)C2)cc(=O)n1C ZINC000217773914 ED In-Stock Unstable AKR1C3 0 41 CCn1c(C)c(C=O)c2cc(OCc3ccccc3)ccc21 ZINC000217773919 CI In-Stock Unstable MAOB 50 44 CCn1c(C)c(C=O)c2cc(OCc3ccccc3)ccc21 ZINC000217773919 CI In-Stock Unstable PLA2G2A 66 46 Cc1cccc(C(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217773939 DF For-Sale Unstable KCNK3 44 35 COC1CCN(C2CCN(C(=O)c3ccc4cc[nH]c4c3)CC2)CC1 ZINC000217773940 EF In-Stock Unstable CHRM2 58 41 COC1CCN(C2CCN(C(=O)c3ccc4cc[nH]c4c3)CC2)CC1 ZINC000217773940 EF In-Stock Unstable HRH1 17 43 COC1CCN(C2CCN(C(=O)c3ccc4cc[nH]c4c3)CC2)CC1 ZINC000217773940 EF In-Stock Unstable INHA 19 47 COC1CCN(C2CCN(C(=O)c3ccc4cc[nH]c4c3)CC2)CC1 ZINC000217773940 EF In-Stock Unstable HRH3 20 52 COC1CCN(C2CCN(C(=O)c3ccc4cc[nH]c4c3)CC2)CC1 ZINC000217773940 EF In-Stock Unstable CCR3 47 46 COC1CCN(C2CCN(C(=O)c3ccc4cc[nH]c4c3)CC2)CC1 ZINC000217773940 EF In-Stock Unstable GHSR 16 54 COC1CCN(C2CCN(C(=O)c3ccc4cc[nH]c4c3)CC2)CC1 ZINC000217773940 EF In-Stock Unstable L3MBTL3 96 56 Cc1cc(O[C@H]2CCN(S(=O)(=O)c3ccccc3)C2)cc(=O)n1C ZINC000217773985 ED In-Stock Unstable AKR1C3 0 41 O=C(O)/C=C\c1cnc(NC(=O)c2cccc(Cl)c2)s1 ZINC000217773995 DG For-Sale Anodyne LUCI_LUCLA 25 47 O=C(O)/C=C\c1cnc(NC(=O)c2cccc(Cl)c2)s1 ZINC000217773995 DG For-Sale Anodyne SCD1 33 41 O=C(O)/C=C\c1cnc(NC(=O)c2cccc(Cl)c2)s1 ZINC000217773995 DG For-Sale Anodyne SCD 28 41 O=C(O)/C=C\c1cnc(NC(=O)c2cccc(Cl)c2)s1 ZINC000217773995 DG For-Sale Anodyne KCNK3 49 46 O=C(O)/C=C\c1cnc(NC(=O)c2cccc(Cl)c2)s1 ZINC000217773995 DG For-Sale Anodyne KCNK9 28 43 CCCn1c(C)c(C=O)c2cc(OCc3ccccc3)ccc21 ZINC000217774022 DJ In-Stock Unstable MAOB 45 42 CCCn1c(C)c(C=O)c2cc(OCc3ccccc3)ccc21 ZINC000217774022 DJ In-Stock Unstable PLA2G2A 61 45 Cc1cccc(C(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217774027 DF For-Sale Unstable KCNK3 44 35 COCc1cc(=O)c(O)c([C@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccc(OC)c(O)c2)o1 ZINC000217774061 KH In-Stock Unstable RORC 49 34 O=C(O)/C=C\c1cnc(NC(=O)Cc2cccc(F)c2)s1 ZINC000217774077 DF For-Sale Unstable CDK5 49 48 O=C(O)/C=C\c1cnc(NC(=O)Cc2cccc(F)c2)s1 ZINC000217774077 DF For-Sale Unstable HCAR2 0 42 C=C[C@@H](CI)NC(=O)OC(C)(C)C ZINC000217774114 CF For-Sale Unstable PAPA1_CARPA 43 36 C=C[C@@H](CI)NC(=O)OC(C)(C)C ZINC000217774114 CF For-Sale Unstable CTSK 28 56 C[C@H](O)CCNC(=O)/C=C\c1ccc(C#N)cc1 ZINC000217774122 BD For-Sale Unstable PYGL 0 40 CCCCn1c(C)c(C=O)c2cc(OCc3ccccc3)ccc21 ZINC000217774135 DK In-Stock Unstable MAOB 37 41 CCCCn1c(C)c(C=O)c2cc(OCc3ccccc3)ccc21 ZINC000217774135 DK In-Stock Unstable PLA2G2A 70 46 CCCCn1c(C)c(C=O)c2cc(OCc3ccccc3)ccc21 ZINC000217774135 DK In-Stock Unstable RORB 0 42 O=C(O)[C@@H]1[C@H]2CN(C(=O)C3(c4ccc(Cl)cc4)CCC3)C[C@H]21 ZINC000217774143 DF In-Stock Unstable HSD11B1 15 49 COCc1cc(=O)c(O)c([C@@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccc(OC)c(O)c2)o1 ZINC000217774151 KH In-Stock Unstable RORC 49 34 O=C(O)/C=C\c1cnc(NC(=O)Cc2ccccc2Cl)s1 ZINC000217774167 DG For-Sale Unstable CSNK1D 20 44 O=C(O)/C=C\c1cnc(NC(=O)Cc2ccccc2Cl)s1 ZINC000217774167 DG For-Sale Unstable CDK5 41 45 C[C@@H](O)CCNC(=O)/C=C\c1ccc(C#N)cc1 ZINC000217774201 BD On-Demand Unstable PYGL 0 40 COCCN(CCOC)C(=O)N/C=C/c1ccccc1F ZINC000217774220 CE For-Sale Unstable TLR4 16 43 Cc1c(C=O)c2cc(OCc3ccccc3)ccc2n1CC(C)C ZINC000217774245 DJ In-Stock Unstable MAOB 44 42 Cc1c(C=O)c2cc(OCc3ccccc3)ccc2n1CC(C)C ZINC000217774245 DJ In-Stock Unstable PLA2G2A 59 45 Cc1c(C=O)c2cc(OCc3ccccc3)ccc2n1CC(C)C ZINC000217774245 DJ In-Stock Unstable FFAR1 42 35 Cc1ccccc1CC(=O)Nc1ncc(/C=C\C(=O)O)s1 ZINC000217774249 DF For-Sale Unstable CDK5 48 46 COC1CCN(C2CCN(C(=O)Cc3ccc(Br)cc3)CC2)CC1 ZINC000217774262 GG In-Stock Unstable CHRM2 52 46 COC1CCN(C2CCN(C(=O)Cc3ccc(Br)cc3)CC2)CC1 ZINC000217774262 GG In-Stock Unstable CCR3 28 61 COC1CCN(C2CCN(C(=O)Cc3ccc(Br)cc3)CC2)CC1 ZINC000217774262 GG In-Stock Unstable L3MBTL3 78 39 CCOC(=O)[C@@H]1CCOC(=O)CC1 ZINC000217774335 AC In-Stock Unstable PPM1B 0 40 CCOC(=O)[C@@H]1CCOC(=O)CC1 ZINC000217774335 AC In-Stock Unstable PPP1CC 0 40 COc1ccc(COc2cccc(/C(C)=N\O)c2)cc1Br ZINC000217774349 FI For-Sale Unstable ACR 27 41 Cc1c(C=O)c2cc(OCc3ccccc3)ccc2n1Cc1ccccc1 ZINC000217774361 FK In-Stock Unstable MAOA 17 42 Cc1c(C=O)c2cc(OCc3ccccc3)ccc2n1Cc1ccccc1 ZINC000217774361 FK In-Stock Unstable MAOB 55 44 Cc1c(C=O)c2cc(OCc3ccccc3)ccc2n1Cc1ccccc1 ZINC000217774361 FK In-Stock Unstable ALOX5AP 92 37 Cc1c(C=O)c2cc(OCc3ccccc3)ccc2n1Cc1ccccc1 ZINC000217774361 FK In-Stock Unstable PLA2G2A 97 53 Cc1c(C=O)c2cc(OCc3ccccc3)ccc2n1Cc1ccccc1 ZINC000217774361 FK In-Stock Unstable ADAM17 16 40 Cc1c(CC(=O)NC[C@@H]2CCCN3CCCC[C@H]23)c(=O)oc2cc(O)ccc12 ZINC000217774384 GF In-Stock Unstable HSD17B3 24 46 COC1CCN(C2CCN(C(=O)Cc3cn(C)c4ccccc34)CC2)CC1 ZINC000217774385 FF In-Stock Unstable CHRM2 42 38 COC1CCN(C2CCN(C(=O)Cc3cn(C)c4ccccc34)CC2)CC1 ZINC000217774385 FF In-Stock Unstable CCR3 21 47 COC1CCN(C2CCN(C(=O)Cc3cn(C)c4ccccc34)CC2)CC1 ZINC000217774385 FF In-Stock Unstable L3MBTL3 53 36 COc1cc(NC(=O)/C=C/c2cccc(CO)c2)cc(OC)c1OC ZINC000217774392 EF On-Demand Unstable HDAC8 42 41 COc1cc(NC(=O)/C=C/c2cccc(CO)c2)cc(OC)c1OC ZINC000217774392 EF On-Demand Unstable MMP2 25 51 COc1cc(NC(=O)/C=C/c2cccc(CO)c2)cc(OC)c1OC ZINC000217774392 EF On-Demand Unstable HDAC6 28 41 COc1cc(NC(=O)/C=C/c2cccc(CO)c2)cc(OC)c1OC ZINC000217774392 EF On-Demand Unstable MMP9 21 48 COc1cc(NC(=O)/C=C/c2cccc(CO)c2)cc(OC)c1OC ZINC000217774392 EF On-Demand Unstable TUBB1 54 41 COc1cc(NC(=O)/C=C/c2cccc(CO)c2)cc(OC)c1OC ZINC000217774392 EF On-Demand Unstable MMP1 24 48 COc1cc(NC(=O)/C=C/c2cccc(CO)c2)cc(OC)c1OC ZINC000217774392 EF On-Demand Unstable METAP2 18 54 Cc1cc(Br)ccc1[C@@H]1CCCNC1 ZINC000217774395 CG For-Sale Unstable IKBKB 0 41 O=C(O)/C=C\c1ccc(OCc2ccc(F)c(Br)c2)cc1 ZINC000217774428 FI For-Sale Unstable PTGER3 16 41 O=C(O)/C=C\c1ccc(OCc2ccc(F)c(Br)c2)cc1 ZINC000217774428 FI For-Sale Unstable GYS1 46 31 O=C(O)/C=C\c1ccc(OCc2ccc(F)c(Br)c2)cc1 ZINC000217774428 FI For-Sale Unstable FFAR1 48 39 O=C(O)/C=C\c1ccc(OCc2ccc(F)c(Br)c2)cc1 ZINC000217774428 FI For-Sale Unstable AKR1C3 33 42 O=C(O)/C=C\c1ccc(OCc2ccc(F)c(Br)c2)cc1 ZINC000217774428 FI For-Sale Unstable FFAR4 35 41 CCOC(=O)[C@H]1CCOC(=O)CC1 ZINC000217774441 AC In-Stock Unstable PPM1B 0 40 CCOC(=O)[C@H]1CCOC(=O)CC1 ZINC000217774441 AC In-Stock Unstable PPP1CC 0 40 NCC[C@@H](N1CCC[C@@H]1c1cccnc1)C(F)(F)F ZINC000217774462 CE For-Sale Unstable CHRNA2 49 50 Cc1c(C=O)c2cc(OCc3ccccc3)ccc2n1CCc1ccccc1 ZINC000217774466 FK In-Stock Unstable MAOB 47 42 Cc1c(C=O)c2cc(OCc3ccccc3)ccc2n1CCc1ccccc1 ZINC000217774466 FK In-Stock Unstable PLA2G2A 66 47 Cc1c(C=O)c2cc(OCc3ccccc3)ccc2n1CCc1ccccc1 ZINC000217774466 FK In-Stock Unstable FFAR1 36 41 Cc1cc(Br)ccc1[C@H]1CCCNC1 ZINC000217774479 CG For-Sale Unstable IKBKB 0 41 O=C(O)/C=C\c1ccccc1OCc1ccc(F)c(Br)c1 ZINC000217774508 FI For-Sale Unstable PTGER2 22 51 O=C(O)/C=C\c1ccccc1OCc1ccc(F)c(Br)c1 ZINC000217774508 FI For-Sale Unstable PTGER1 55 40 O=C(O)/C=C\c1ccccc1OCc1ccc(F)c(Br)c1 ZINC000217774508 FI For-Sale Unstable PTGER4 42 50 O=C(O)/C=C\c1ccccc1OCc1ccc(F)c(Br)c1 ZINC000217774508 FI For-Sale Unstable PTGER3 34 51 O=C(O)/C=C\c1ccccc1OCc1ccc(F)c(Br)c1 ZINC000217774508 FI For-Sale Unstable PTGDR 0 45 O=C(O)/C=C\c1ccccc1OCc1ccc(F)c(Br)c1 ZINC000217774508 FI For-Sale Unstable AKR1C3 31 44 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@H]1O ZINC000217774575 KD For-Sale Unstable POLA1 43 39 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@H]1O ZINC000217774575 KD For-Sale Unstable ADORA1 98 57 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@H]1O ZINC000217774575 KD For-Sale Unstable SLC29A1 67 39 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@H]1O ZINC000217774575 KD For-Sale Unstable ADORA2A 41 45 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@H]1O ZINC000217774575 KD For-Sale Unstable DNMT1 24 42 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@H]1O ZINC000217774575 KD For-Sale Unstable P2RY6 130 44 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@H]1O ZINC000217774575 KD For-Sale Unstable ADK 51 44 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@H]1O ZINC000217774575 KD For-Sale Unstable POLB 48 39 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@H]1O ZINC000217774575 KD For-Sale Unstable P2RX3 17 69 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@H]1O ZINC000217774575 KD For-Sale Unstable AHCY 68 48 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@H]1O ZINC000217774575 KD For-Sale Unstable P2RX4 79 81 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@H]1O ZINC000217774575 KD For-Sale Unstable P2RX1 102 81 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@H]1O ZINC000217774575 KD For-Sale Unstable P2RY4 132 69 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@H]1O ZINC000217774575 KD For-Sale Unstable P2RY1 66 69 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@H]1O ZINC000217774575 KD For-Sale Unstable GAPDH 41 44 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@H]1O ZINC000217774575 KD For-Sale Unstable ITPR1 69 47 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@H]1O ZINC000217774575 KD For-Sale Unstable P2RY2 173 69 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@H]1O ZINC000217774575 KD For-Sale Unstable ADORA3 89 44 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@H]1O ZINC000217774575 KD For-Sale Unstable OXGR1 130 45 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@H]1O ZINC000217774575 KD For-Sale Unstable AANAT 81 46 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@H]1O ZINC000217774575 KD For-Sale Unstable P2RY14 62 39 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@H]1O ZINC000217774575 KD For-Sale Unstable RNASE1 70 54 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@H]1O ZINC000217774575 KD For-Sale Unstable DNMT3B 68 42 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@H]1O ZINC000217774575 KD For-Sale Unstable PANC 39 42 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@H]1O ZINC000217774575 KD For-Sale Unstable GPR17 77 57 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@H]1O ZINC000217774575 KD For-Sale Unstable HSPA5 57 34 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@H]1O ZINC000217774575 KD For-Sale Unstable DOT1L 92 42 COC1CCN(C2CCN(C(=O)c3cncc(Br)c3)CC2)CC1 ZINC000217774588 GF In-Stock Unstable CHRM2 41 36 COC1CCN(C2CCN(C(=O)c3cncc(Br)c3)CC2)CC1 ZINC000217774588 GF In-Stock Unstable CCR3 42 42 COC1CCN(C2CCN(C(=O)c3cncc(Br)c3)CC2)CC1 ZINC000217774588 GF In-Stock Unstable L3MBTL3 93 44 O=C(O)/C=C\c1cccc(OCc2ccc(F)c(Br)c2)c1 ZINC000217774603 FI For-Sale Unstable MAOB 28 42 O=C(O)/C=C\c1cccc(OCc2ccc(F)c(Br)c2)c1 ZINC000217774603 FI For-Sale Unstable PTGER2 15 41 O=C(O)/C=C\c1cccc(OCc2ccc(F)c(Br)c2)c1 ZINC000217774603 FI For-Sale Unstable PTGER4 17 46 O=C(O)/C=C\c1cccc(OCc2ccc(F)c(Br)c2)c1 ZINC000217774603 FI For-Sale Unstable FFAR1 44 39 O=C(O)/C=C\c1cccc(OCc2ccc(F)c(Br)c2)c1 ZINC000217774603 FI For-Sale Unstable AKR1C3 33 44 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@@H]1O ZINC000217774656 KD For-Sale Unstable POLA1 43 39 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@@H]1O ZINC000217774656 KD For-Sale Unstable ADORA1 98 57 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@@H]1O ZINC000217774656 KD For-Sale Unstable SLC29A1 67 39 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@@H]1O ZINC000217774656 KD For-Sale Unstable ADORA2A 41 45 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@@H]1O ZINC000217774656 KD For-Sale Unstable DNMT1 24 42 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@@H]1O ZINC000217774656 KD For-Sale Unstable P2RY6 130 44 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@@H]1O ZINC000217774656 KD For-Sale Unstable ADK 51 44 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@@H]1O ZINC000217774656 KD For-Sale Unstable POLB 48 39 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@@H]1O ZINC000217774656 KD For-Sale Unstable P2RX3 17 69 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@@H]1O ZINC000217774656 KD For-Sale Unstable AHCY 68 48 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@@H]1O ZINC000217774656 KD For-Sale Unstable P2RX4 79 81 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@@H]1O ZINC000217774656 KD For-Sale Unstable P2RX1 102 81 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@@H]1O ZINC000217774656 KD For-Sale Unstable P2RY4 132 69 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@@H]1O ZINC000217774656 KD For-Sale Unstable P2RY1 66 69 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@@H]1O ZINC000217774656 KD For-Sale Unstable GAPDH 41 44 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@@H]1O ZINC000217774656 KD For-Sale Unstable ITPR1 69 47 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@@H]1O ZINC000217774656 KD For-Sale Unstable P2RY2 173 69 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@@H]1O ZINC000217774656 KD For-Sale Unstable ADORA3 89 44 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@@H]1O ZINC000217774656 KD For-Sale Unstable OXGR1 130 45 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@@H]1O ZINC000217774656 KD For-Sale Unstable AANAT 81 46 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@@H]1O ZINC000217774656 KD For-Sale Unstable P2RY14 62 39 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@@H]1O ZINC000217774656 KD For-Sale Unstable RNASE1 70 54 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@@H]1O ZINC000217774656 KD For-Sale Unstable DNMT3B 68 42 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@@H]1O ZINC000217774656 KD For-Sale Unstable PANC 39 42 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@@H]1O ZINC000217774656 KD For-Sale Unstable GPR17 77 57 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@@H]1O ZINC000217774656 KD For-Sale Unstable HSPA5 57 34 Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)OP(=O)(O)O)[C@H](OC(=O)c2ccc(C(=O)c3ccccc3)cc2)[C@@H]1O ZINC000217774656 KD For-Sale Unstable DOT1L 92 42 O=C(O)Cc1cc(Br)c2c(c1)CCCN2 ZINC000217774670 CE In-Stock Unstable THRA 25 45 COc1ccc(CC[C@](C)(CN)N2CCCC[C@@H]2C)cc1 ZINC000217774749 CG For-Sale Unstable FKBP12.6 0 41 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217774754 HE For-Sale Unstable TGM2 50 38 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217774754 HE For-Sale Unstable NAMPT 44 44 COc1ccc(Br)cc1COc1ccc(/C(C)=N\O)cc1 ZINC000217774760 FI For-Sale Unstable TSHR 55 32 CCCCn1c(C)c(C=O)c2cc(OC(C)C)ccc21 ZINC000217774761 CI In-Stock Unstable PLA2G2A 31 44 COC(=O)Cc1ccc2c(c1)CCCN2C(=O)OCC1c2ccccc2-c2ccccc21 ZINC000217774774 IK In-Stock Unstable AVPR2 47 40 CC1(C)C[C@H]2C[C@@](C)(CN2C(=O)N/C=C/c2ccccc2F)C1 ZINC000217774788 DI For-Sale Unstable AVPR2 16 44 CC1(C)C[C@H]2C[C@@](C)(CN2C(=O)N/C=C/c2ccccc2F)C1 ZINC000217774788 DI For-Sale Unstable AVPR1A 38 44 C[C@H](O)CCNC(=O)/C=C\c1ccc(N(C)C)cc1 ZINC000217774800 CD For-Sale Unstable PYGL 0 41 C[C@H](O)CCNC(=O)/C=C\c1ccc(N(C)C)cc1 ZINC000217774800 CD For-Sale Unstable HDAC8 15 40 C[C@H](O)CCNC(=O)/C=C\c1ccc(N(C)C)cc1 ZINC000217774800 CD For-Sale Unstable HDAC1 0 40 C[C@H](O)CCNC(=O)/C=C\c1ccc(N(C)C)cc1 ZINC000217774800 CD For-Sale Unstable HDAC4 23 40 C[C@H](O)CCNC(=O)/C=C\c1ccc(N(C)C)cc1 ZINC000217774800 CD For-Sale Unstable HDAC5 26 40 O=C(NC[C@H]1CCCN1c1nccs1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217774801 HE For-Sale Unstable TGM2 50 38 O=C(NC[C@H]1CCCN1c1nccs1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217774801 HE For-Sale Unstable NAMPT 44 44 COc1cc2c(cc1OC)CN(Cc1cc(=O)c(O)c(CN3CCCCC3)o1)CC2 ZINC000217774817 HF In-Stock Unstable ABCB1B 61 35 COc1cc2c(cc1OC)CN(Cc1cc(=O)c(O)c(CN3CCCCC3)o1)CC2 ZINC000217774817 HF In-Stock Unstable ABCB1 23 47 COc1ccc(COc2ccc(/C(C)=N\O)cc2)cc1Br ZINC000217774830 FI For-Sale Unstable ACR 32 40 COc1ccc(COc2ccc(/C(C)=N\O)cc2)cc1Br ZINC000217774830 FI For-Sale Unstable KLK_PIG 33 41 C[C@@H](O)CCNC(=O)/C=C\c1ccc(N(C)C)cc1 ZINC000217774893 CD For-Sale Unstable PYGL 0 41 C[C@@H](O)CCNC(=O)/C=C\c1ccc(N(C)C)cc1 ZINC000217774893 CD For-Sale Unstable HDAC8 15 40 C[C@@H](O)CCNC(=O)/C=C\c1ccc(N(C)C)cc1 ZINC000217774893 CD For-Sale Unstable HDAC1 0 40 C[C@@H](O)CCNC(=O)/C=C\c1ccc(N(C)C)cc1 ZINC000217774893 CD For-Sale Unstable HDAC4 23 40 C[C@@H](O)CCNC(=O)/C=C\c1ccc(N(C)C)cc1 ZINC000217774893 CD For-Sale Unstable HDAC5 26 40 COc1ccc(Br)cc1COc1ccccc1/C(C)=N\O ZINC000217774915 FI For-Sale Unstable MC4R 19 40 C[C@H](N)C(=O)c1ccc(F)c(Br)c1 ZINC000217774921 BE For-Sale Unstable CES2 20 40 Cc1c(C=O)c2cc(OC(C)C)ccc2n1Cc1ccccc1 ZINC000217774953 DJ In-Stock Unstable PPARG 28 40 Cc1c(C=O)c2cc(OC(C)C)ccc2n1Cc1ccccc1 ZINC000217774953 DJ In-Stock Unstable ALOX5AP 45 35 Cc1c(C=O)c2cc(OC(C)C)ccc2n1Cc1ccccc1 ZINC000217774953 DJ In-Stock Unstable PLA2G2A 102 50 Cc1c(C=O)c2cc(OC(C)C)ccc2n1Cc1ccccc1 ZINC000217774953 DJ In-Stock Unstable PLA2G10 41 31 Cc1c(C=O)c2cc(OC(C)C)ccc2n1Cc1ccccc1 ZINC000217774953 DJ In-Stock Unstable PLA2G2D 40 31 Cc1c(C=O)c2cc(OC(C)C)ccc2n1Cc1ccccc1 ZINC000217774953 DJ In-Stock Unstable PTGES2 60 35 COC(=O)Cc1ccc2[nH]c(=O)cc(C)c2c1 ZINC000217774976 BD In-Stock Unstable AR 19 44 COC1CCN(C2CCN(C(=O)c3ccc(-n4cccc4)cc3)CC2)CC1 ZINC000217774978 FG In-Stock Unstable CHRM2 56 40 COC1CCN(C2CCN(C(=O)c3ccc(-n4cccc4)cc3)CC2)CC1 ZINC000217774978 FG In-Stock Unstable HRH1 17 41 COC1CCN(C2CCN(C(=O)c3ccc(-n4cccc4)cc3)CC2)CC1 ZINC000217774978 FG In-Stock Unstable AVPR1A 24 40 COC1CCN(C2CCN(C(=O)c3ccc(-n4cccc4)cc3)CC2)CC1 ZINC000217774978 FG In-Stock Unstable HRH3 16 46 COC1CCN(C2CCN(C(=O)c3ccc(-n4cccc4)cc3)CC2)CC1 ZINC000217774978 FG In-Stock Unstable CCR3 45 43 COC1CCN(C2CCN(C(=O)c3ccc(-n4cccc4)cc3)CC2)CC1 ZINC000217774978 FG In-Stock Unstable L3MBTL3 124 53 CN(C)c1cccc(NC(=O)N/C=C/c2ccccc2F)c1 ZINC000217774980 CH For-Sale Unstable KCNK3 48 42 O=C1CCCc2cccc(OS(=O)(=O)C(F)(F)F)c21 ZINC000217774995 CE For-Sale Unstable HPD 15 40 C[C@@H](N)C(=O)c1ccc(F)c(Br)c1 ZINC000217775010 BE For-Sale Unstable CES2 20 40 Cc1c(C=O)c2cc(OC(C)C)ccc2n1CCc1ccccc1 ZINC000217775060 DJ In-Stock Unstable PLA2G4A 20 42 Cc1c(C=O)c2cc(OC(C)C)ccc2n1CCc1ccccc1 ZINC000217775060 DJ In-Stock Unstable PLA2G2A 64 41 CN1CCc2nc(NC(=O)N/C=C/c3ccccc3F)sc2C1 ZINC000217775090 EG For-Sale Unstable F10 26 45 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000217775098 IF For-Sale Unstable TGM2 50 39 O=C(NC[C@@H]1CCCN1c1nccs1)c1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000217775098 IF For-Sale Unstable NAMPT 44 46 COc1ccc2[nH]c(C(=O)N3CCC(c4ccnc(C)n4)CC3)cc2c1 ZINC000217775114 FG In-Stock Unstable GRIN2B 32 46 COc1ccc2[nH]c(C(=O)N3CCC(c4ccnc(C)n4)CC3)cc2c1 ZINC000217775114 FG In-Stock Unstable HRH4 29 60 COc1ccc2[nH]c(C(=O)N3CCC(c4ccnc(C)n4)CC3)cc2c1 ZINC000217775114 FG In-Stock Unstable SYK 0 43 COc1ccc2[nH]c(C(=O)N3CCC(c4ccnc(C)n4)CC3)cc2c1 ZINC000217775114 FG In-Stock Unstable TUBB2B 40 43 COc1ccc2[nH]c(C(=O)N3CCC(c4ccnc(C)n4)CC3)cc2c1 ZINC000217775114 FG In-Stock Unstable FPR2 33 53 COc1ccc2[nH]c(C(=O)N3CCC(c4ccnc(C)n4)CC3)cc2c1 ZINC000217775114 FG In-Stock Unstable AKR1C3 20 48 COc1ccc2[nH]c(C(=O)N3CCC(c4ccnc(C)n4)CC3)cc2c1 ZINC000217775114 FG In-Stock Unstable MAP3K12 29 40 O=C(Cc1ccc(F)cc1)N1C[C@H]2CNC[C@@H](C2)C1 ZINC000217775167 CD For-Sale Unstable CHRNA7 31 60 O=C(Cc1ccc(F)cc1)N1C[C@H]2CNC[C@@H](C2)C1 ZINC000217775167 CD For-Sale Unstable MLNR 30 41 CCOc1ccc2ccccc2c1C(=O)N1CCC(N2CCC(OC)CC2)CC1 ZINC000217775178 GH In-Stock Unstable CHRM2 55 44 CCOc1ccc2ccccc2c1C(=O)N1CCC(N2CCC(OC)CC2)CC1 ZINC000217775178 GH In-Stock Unstable ACACA 34 46 CCOc1ccc2ccccc2c1C(=O)N1CCC(N2CCC(OC)CC2)CC1 ZINC000217775178 GH In-Stock Unstable CCR3 27 40 CCOc1ccc2ccccc2c1C(=O)N1CCC(N2CCC(OC)CC2)CC1 ZINC000217775178 GH In-Stock Unstable ACACB 28 40 CCOc1ccc2ccccc2c1C(=O)N1CCC(N2CCC(OC)CC2)CC1 ZINC000217775178 GH In-Stock Unstable L3MBTL3 82 45 O=C(NC[C@H]1CCCN1c1nccs1)c1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000217775190 IF For-Sale Unstable TGM2 50 39 O=C(NC[C@H]1CCCN1c1nccs1)c1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000217775190 IF For-Sale Unstable NAMPT 44 46 Cc1cc(O[C@@H]2CCN(S(=O)(=O)c3ccccc3C(F)(F)F)C2)cc(=O)n1C ZINC000217775284 HF In-Stock Unstable SFRP1 52 35 Nc1c[nH]c(=O)c(-c2ccccc2)n1 ZINC000217775293 AD In-Stock Unstable PTP4A1 0 43 Nc1c[nH]c(=O)c(-c2ccccc2)n1 ZINC000217775293 AD In-Stock Unstable PTP4A2 0 43 C[C@H](O)CCNC(=O)/C=C\c1cc(Cl)cc(Cl)c1 ZINC000217775341 CF For-Sale Unstable PYGL 27 49 Cc1cc(O[C@H]2CCN(S(=O)(=O)c3ccccc3C(F)(F)F)C2)cc(=O)n1C ZINC000217775380 HF In-Stock Unstable SFRP1 52 35 C[C@@H](O)CCNC(=O)/C=C\c1cc(Cl)cc(Cl)c1 ZINC000217775424 CF On-Demand Unstable PYGL 27 49 O=C(Cc1ccccc1F)N1C[C@H]2CNC[C@@H](C2)C1 ZINC000217775442 CD For-Sale Unstable CHRNA7 20 51 COc1ccc(/C=C\C(=O)NCC[C@H](C)O)cc1 ZINC000217775506 BD On-Demand Unstable PTGS2 0 53 COc1ccc(/C=C\C(=O)NCC[C@H](C)O)cc1 ZINC000217775506 BD On-Demand Unstable PYGL 0 41 COc1ccc(/C=C\C(=O)NCC[C@H](C)O)cc1 ZINC000217775506 BD On-Demand Unstable HDAC8 22 56 COc1ccc(/C=C\C(=O)NCC[C@H](C)O)cc1 ZINC000217775506 BD On-Demand Unstable MMP2 23 51 COc1ccc(/C=C\C(=O)NCC[C@H](C)O)cc1 ZINC000217775506 BD On-Demand Unstable HDAC1 24 46 COc1ccc(/C=C\C(=O)NCC[C@H](C)O)cc1 ZINC000217775506 BD On-Demand Unstable HDAC2 0 40 COc1ccc(/C=C\C(=O)NCC[C@H](C)O)cc1 ZINC000217775506 BD On-Demand Unstable HDAC4 0 46 COc1ccc(/C=C\C(=O)NCC[C@H](C)O)cc1 ZINC000217775506 BD On-Demand Unstable GPR183 0 43 O=C(O)CCc1cc(Br)c2c(c1)CCCN2 ZINC000217775515 CF In-Stock Unstable THRA 19 47 O=C(O)CCc1cc(Br)c2c(c1)CCCN2 ZINC000217775515 CF In-Stock Unstable THRB 24 47 COCCCCNC(=O)c1ccc(/C=C\C(=O)O)cc1 ZINC000217775562 CD For-Sale Unstable HDAC6 18 43 COc1ccc(/C=C\C(=O)NCC[C@@H](C)O)cc1 ZINC000217775588 BD On-Demand Unstable PTGS2 0 53 COc1ccc(/C=C\C(=O)NCC[C@@H](C)O)cc1 ZINC000217775588 BD On-Demand Unstable PYGL 0 41 COc1ccc(/C=C\C(=O)NCC[C@@H](C)O)cc1 ZINC000217775588 BD On-Demand Unstable HDAC8 22 56 COc1ccc(/C=C\C(=O)NCC[C@@H](C)O)cc1 ZINC000217775588 BD On-Demand Unstable MMP2 23 51 COc1ccc(/C=C\C(=O)NCC[C@@H](C)O)cc1 ZINC000217775588 BD On-Demand Unstable HDAC1 24 46 COc1ccc(/C=C\C(=O)NCC[C@@H](C)O)cc1 ZINC000217775588 BD On-Demand Unstable HDAC2 0 40 COc1ccc(/C=C\C(=O)NCC[C@@H](C)O)cc1 ZINC000217775588 BD On-Demand Unstable HDAC4 0 46 COc1ccc(/C=C\C(=O)NCC[C@@H](C)O)cc1 ZINC000217775588 BD On-Demand Unstable GPR183 0 43 CCCCOC(=O)Cc1ccc(C)cc1N ZINC000217775595 BE In-Stock Unstable PLA2G4B 50 33 CCN(Cc1ccc(Cl)cc1)C(=O)C(C)C ZINC000217775620 BG On-Demand Unstable TSPO 30 42 CCN(Cc1ccc(Cl)cc1)C(=O)C(C)C ZINC000217775620 BG On-Demand Unstable FFAR2 53 44 CC(C)(C)OC(=O)N1CCCc2cc(CCC(=O)O)ccc21 ZINC000217775642 DG In-Stock Unstable FFAR1 43 34 CC(C)(C)OC(=O)N1CCCc2cc(CCC(=O)O)ccc21 ZINC000217775642 DG In-Stock Unstable GPR119 20 41 O=C(N/C=C/c1ccccc1F)Nc1cccc(Br)c1 ZINC000217775663 EI For-Sale Anodyne KCNK3 42 36 COc1cc(OC)c2cc(C(=O)NC[C@@H]3CCCN4CCCC[C@H]34)n(C)c2c1 ZINC000217775667 GG In-Stock Unstable ACKR3 41 30 COCCCCNC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217775683 CD For-Sale Unstable DRD4 44 33 COCCCCNC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217775683 CD For-Sale Unstable DRD3 28 40 COCCCCNC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217775683 CD For-Sale Unstable HDAC8 19 43 COCCCCNC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217775683 CD For-Sale Unstable HDAC9 21 40 COCCCCNC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217775683 CD For-Sale Unstable HDAC7 21 40 COCCCCNC(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217775683 CD For-Sale Unstable HDA106 0 41 O=C(Cc1cccc(F)c1)N1C[C@H]2CNC[C@@H](C2)C1 ZINC000217775715 CD For-Sale Unstable CHRNA7 18 50 COC(=O)CCc1ccc2c(c1)CCCN2C(=O)OC(C)(C)C ZINC000217775750 DG In-Stock Unstable AVPR2 23 40 COC(=O)CCc1ccc2c(c1)CCCN2C(=O)OC(C)(C)C ZINC000217775750 DG In-Stock Unstable GPR119 22 41 C[C@@H](c1ccc(Cl)cc1)N(C)C[C@@H](N)c1ccccc1 ZINC000217775813 CI For-Sale Unstable AOC3 31 41 CC(C)[C@@H]1CC[C@@H](N)[C@@H](CCCc2ccccc2)C1 ZINC000217775831 CI For-Sale Unstable SLC18A2 47 48 COC(=O)CCc1ccc2c(c1)CCCN2C(=O)OCC1c2ccccc2-c2ccccc21 ZINC000217775875 IK In-Stock Unstable AVPR2 41 38 COc1cc([C@@H](C)N2CCOC[C@@H]2C)ccc1O ZINC000217775884 CE For-Sale Unstable SHBG 17 43 C[C@H](c1ccc(Cl)cc1)N(C)C[C@@H](N)c1ccccc1 ZINC000217775894 CI For-Sale Unstable AOC3 31 41 Cc1cc(OC2CCN(C(=O)c3ccco3)CC2)cc(=O)n1C ZINC000217775905 DD In-Stock Unstable PRSS2 44 31 CC(C)[C@H]1CC[C@@H](N)[C@@H](CCCc2ccccc2)C1 ZINC000217775920 CI For-Sale Unstable SLC18A2 47 48 CC(C)[C@@H]1CC[C@H](N)[C@@H](CCCc2ccccc2)C1 ZINC000217775996 CI For-Sale Unstable SLC18A2 47 48 CC(C)(C)c1ccc(NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217776006 DJ For-Sale Unstable TRPV1 20 43 Cc1cc(OC2CCN(C(=O)c3ccccc3F)CC2)cc(=O)n1C ZINC000217776017 EF In-Stock Unstable CCR3 29 44 CC(C)[C@H]1CC[C@H](N)[C@@H](CCCc2ccccc2)C1 ZINC000217776086 CI For-Sale Unstable SLC18A2 47 48 COc1ccc(CNS(C)(=O)=O)cc1C(=O)O ZINC000217776089 CC On-Demand Unstable PPARD 16 40 COc1ccc(CNS(C)(=O)=O)cc1C(=O)O ZINC000217776089 CC On-Demand Unstable AKR1C2 44 34 COc1ccc(CNS(C)(=O)=O)cc1C(=O)O ZINC000217776089 CC On-Demand Unstable DRTS_TRYCR 48 33 C[C@H](O)CCNC(=O)/C=C\c1ccccc1F ZINC000217776094 BD On-Demand Unstable KCNQ2 57 43 COc1ccc(COC/C=C\c2ccccc2)cc1Br ZINC000217776116 EJ For-Sale Unstable CYP1B1 17 43 COc1ccc(COC/C=C\c2ccccc2)cc1Br ZINC000217776116 EJ For-Sale Unstable CYP1A1 15 43 Cc1cc(C(=O)N2CCC(Oc3cc(C)n(C)c(=O)c3)CC2)c(C)o1 ZINC000217776130 EF In-Stock Unstable PRSS2 50 31 CCN(C)C(=O)CNC(=O)c1ccc(F)c([N+](=O)[O-])c1 ZINC000217776142 CC For-Sale Unstable TAAR1 18 47 COc1ccccc1C(=O)N1[C@@H](C)C[C@@H]2CNC[C@H]21 ZINC000217776145 CD For-Sale Unstable KCNA3 41 35 COCCCCNC(=O)c1ccc(/C=C\C(=O)O)c(F)c1 ZINC000217776148 CE For-Sale Unstable HDAC9 17 41 CNC(=O)c1cccc(NC(=O)C[C@@H]2NC(=O)c3ccccc3NC2=O)c1 ZINC000217776177 FD In-Stock Unstable KCNK3 57 32 C[C@@H](O)CCNC(=O)/C=C\c1ccccc1F ZINC000217776180 BD On-Demand Unstable KCNQ2 57 43 COc1ccccc1C(=O)N1[C@@H]2CNC[C@H]2C[C@H]1C ZINC000217776223 CD For-Sale Unstable KCNA3 41 35 Cc1cc(=O)c2cc(CCC(=O)O)ccc2n1C ZINC000217776232 BD In-Stock Unstable THRA 23 40 Cc1cc(=O)c2cc(CCC(=O)O)ccc2n1C ZINC000217776232 BD In-Stock Unstable THRB 21 41 Cc1cc(=O)c2cc(CCC(=O)O)ccc2n1C ZINC000217776232 BD In-Stock Unstable PLA2G4A 40 50 Cc1cc(=O)c2cc(CCC(=O)O)ccc2n1C ZINC000217776232 BD In-Stock Unstable FFAR1 58 43 Cc1cc(OC2CCN(C(=O)Cc3cccs3)CC2)cc(=O)n1C ZINC000217776249 EE In-Stock Unstable PRSS2 53 32 Cc1cc(OC2CCN(C(=O)Cc3cccs3)CC2)cc(=O)n1C ZINC000217776249 EE In-Stock Unstable ETHR 28 44 COc1ccc(NC(=O)C[C@@H]2NC(=O)N(CCc3c[nH]c4ccccc34)C2=O)cn1 ZINC000217776281 HE In-Stock Unstable GHSR 41 36 COc1ccccc1C(=O)N1[C@@H](C)C[C@H]2CNC[C@H]21 ZINC000217776312 CD For-Sale Unstable KCNA3 41 35 COC(CNC(=O)N/C=C/c1ccccc1F)OC ZINC000217776344 CD For-Sale Unstable TLR4 16 43 Cc1cc(OC2CCN(C(=O)c3cccn(C)c3=O)CC2)cc(=O)n1C ZINC000217776354 FD In-Stock Unstable PRSS2 53 31 Cc1cc(OC2CCN(C(=O)c3cccn(C)c3=O)CC2)cc(=O)n1C ZINC000217776354 FD In-Stock Unstable CCR3 17 41 O=C(NCC1C[C@@H]2CC[C@H](C1)N2)c1cccc(F)c1 ZINC000217776378 CE For-Sale Unstable GRIN2B 18 40 O=C(NCC1C[C@@H]2CC[C@H](C1)N2)c1cccc(F)c1 ZINC000217776378 CE For-Sale Unstable CACNA1I 55 42 COc1ccccc1C(=O)N1[C@@H]2CNC[C@@H]2C[C@H]1C ZINC000217776397 CD For-Sale Unstable KCNA3 41 35 C/C=C\C=C/C(=O)NCC[C@@H](C)O ZINC000217776435 AD For-Sale Unstable CNR2 0 53 CC1(C)[C@@H]2CC[C@@]1(C)[C@H](NC(=O)[C@@H](N)CCS(C)(=O)=O)C2 ZINC000217776449 DD For-Sale Unstable AVPR2 44 52 CC1(C)[C@@H]2CC[C@@]1(C)[C@H](NC(=O)[C@@H](N)CCS(C)(=O)=O)C2 ZINC000217776449 DD For-Sale Unstable OXTR 26 52 Cc1cc(OC2CCN(C(=O)c3ccc(Cl)s3)CC2)cc(=O)n1C ZINC000217776467 FG In-Stock Unstable PRSS2 59 31 O=C(NC[C@@H]1CCCN1c1nccs1)c1cc(-c2ccc3c(c2)OCO3)n[nH]1 ZINC000217776505 GF For-Sale Unstable NOS2 44 36 C/C=C/C=C\C(=O)NCC[C@@H](C)O ZINC000217776517 AD On-Demand Unstable CNR2 0 53 CC1(C)[C@H]2CC[C@@]1(C)[C@H](NC(=O)[C@@H](N)CCS(C)(=O)=O)C2 ZINC000217776531 DD On-Demand Unstable AVPR2 44 52 CC1(C)[C@H]2CC[C@@]1(C)[C@H](NC(=O)[C@@H](N)CCS(C)(=O)=O)C2 ZINC000217776531 DD On-Demand Unstable OXTR 26 52 CC[C@H](C(=O)N1CCC(Oc2cc(C)n(C)c(=O)c2)CC1)c1ccccc1 ZINC000217776568 FG In-Stock Unstable PRSS2 50 31 O=C(NC[C@H]1CCCN1c1nccs1)c1cc(-c2ccc3c(c2)OCO3)n[nH]1 ZINC000217776594 GF For-Sale Unstable NOS2 44 36 C/C=C\C=C\C(=O)NCC[C@@H](C)O ZINC000217776598 AD For-Sale Unstable CNR2 0 53 CC1(C)[C@@H]2CC[C@]1(C)[C@H](NC(=O)[C@@H](N)CCS(C)(=O)=O)C2 ZINC000217776626 DD For-Sale Unstable AVPR2 44 52 CC1(C)[C@@H]2CC[C@]1(C)[C@H](NC(=O)[C@@H](N)CCS(C)(=O)=O)C2 ZINC000217776626 DD For-Sale Unstable OXTR 26 52 CC[C@@H](C(=O)N1CCC(Oc2cc(C)n(C)c(=O)c2)CC1)c1ccccc1 ZINC000217776631 FG In-Stock Unstable PRSS2 50 31 O=C(NCC1C[C@@H]2CC[C@H](C1)N2)c1ccc(F)cc1 ZINC000217776676 CE For-Sale Unstable GRIN2B 16 41 O=C(NCC1C[C@@H]2CC[C@H](C1)N2)c1ccc(F)cc1 ZINC000217776676 CE For-Sale Unstable SSTR3 16 40 O=C(NCC1C[C@@H]2CC[C@H](C1)N2)c1ccc(F)cc1 ZINC000217776676 CE For-Sale Unstable CACNA1I 61 34 COc1cccc(/C=C\C(=O)NCC[C@H](C)O)c1 ZINC000217776680 BD For-Sale Unstable DRD4 41 31 COc1cccc(/C=C\C(=O)NCC[C@H](C)O)c1 ZINC000217776680 BD For-Sale Unstable PYGL 22 43 COc1cccc(/C=C\C(=O)NCC[C@H](C)O)c1 ZINC000217776680 BD For-Sale Unstable MTNR1B 56 45 COc1cccc(/C=C\C(=O)NCC[C@H](C)O)c1 ZINC000217776680 BD For-Sale Unstable MMP2 0 52 COc1cccc(/C=C\C(=O)NCC[C@H](C)O)c1 ZINC000217776680 BD For-Sale Unstable NR1H4 41 36 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217776691 FD For-Sale Unstable CA2 105 59 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217776691 FD For-Sale Unstable CA6 21 41 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217776691 FD For-Sale Unstable CA1 94 59 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217776691 FD For-Sale Unstable CA7 55 56 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217776691 FD For-Sale Unstable CA13 24 42 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217776691 FD For-Sale Unstable CA5B 63 56 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217776691 FD For-Sale Unstable CA4 73 57 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217776691 FD For-Sale Unstable CA5A 65 56 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217776691 FD For-Sale Unstable CA14 40 53 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217776691 FD For-Sale Unstable CA12 70 59 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217776691 FD For-Sale Unstable CA9 78 59 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217776691 FD For-Sale Unstable CAH_METTE 18 40 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217776691 FD For-Sale Unstable CYNT 27 47 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217776691 FD For-Sale Unstable NCE103 33 54 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217776691 FD For-Sale Unstable LIG1 0 45 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217776691 FD For-Sale Unstable CA15 15 40 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217776691 FD For-Sale Unstable MTCA1 43 39 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217776691 FD For-Sale Unstable P96878_MYCTU 56 43 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217776691 FD For-Sale Unstable CA 0 40 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217776691 FD For-Sale Unstable A6YCJ1_9METZ 26 53 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217776691 FD For-Sale Unstable Q5TU56_ANOGA 0 40 CC1(C)[C@H]2CC[C@]1(C)[C@H](NC(=O)[C@@H](N)CCS(C)(=O)=O)C2 ZINC000217776719 DD For-Sale Unstable AVPR2 44 52 CC1(C)[C@H]2CC[C@]1(C)[C@H](NC(=O)[C@@H](N)CCS(C)(=O)=O)C2 ZINC000217776719 DD For-Sale Unstable OXTR 26 52 COc1ccccc1-c1cc(C(=O)NC[C@@H]2CCCN2c2nccs2)[nH]n1 ZINC000217776721 GF For-Sale Unstable ACKR3 63 32 NC(=O)CCCNS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217776723 DC For-Sale Unstable AKR1C3 34 42 COC1CCN(C2CCN(C(=O)Cc3c(F)cccc3Cl)CC2)CC1 ZINC000217776725 FG In-Stock Unstable CHRM2 55 40 COC1CCN(C2CCN(C(=O)Cc3c(F)cccc3Cl)CC2)CC1 ZINC000217776725 FG In-Stock Unstable HRH1 18 40 COC1CCN(C2CCN(C(=O)Cc3c(F)cccc3Cl)CC2)CC1 ZINC000217776725 FG In-Stock Unstable CCR3 49 40 COC1CCN(C2CCN(C(=O)Cc3c(F)cccc3Cl)CC2)CC1 ZINC000217776725 FG In-Stock Unstable L3MBTL3 74 37 Oc1ccc(SCCl)cc1 ZINC000217776739 AF For-Sale Unstable H9TVJ1_CHISP 47 34 Cc1cc(OC2CCN(C(=O)c3ccc(F)cc3Cl)CC2)cc(=O)n1C ZINC000217776740 GG In-Stock Unstable HRH1 34 42 Cc1cc(OC2CCN(C(=O)c3ccc(F)cc3Cl)CC2)cc(=O)n1C ZINC000217776740 GG In-Stock Unstable P2RX7 35 51 Cc1cc(OC2CCN(C(=O)c3ccc(F)cc3Cl)CC2)cc(=O)n1C ZINC000217776740 GG In-Stock Unstable CCR3 37 42 Cc1cc(OC2CCN(C(=O)c3ccc(F)cc3Cl)CC2)cc(=O)n1C ZINC000217776740 GG In-Stock Unstable SCD1 18 42 COc1cccc(/C=C\C(=O)NCC[C@@H](C)O)c1 ZINC000217776766 BD On-Demand Unstable DRD4 41 31 COc1cccc(/C=C\C(=O)NCC[C@@H](C)O)c1 ZINC000217776766 BD On-Demand Unstable PYGL 22 43 COc1cccc(/C=C\C(=O)NCC[C@@H](C)O)c1 ZINC000217776766 BD On-Demand Unstable MMP2 0 52 COc1ccccc1-c1cc(C(=O)NC[C@H]2CCCN2c2nccs2)[nH]n1 ZINC000217776800 GF For-Sale Unstable ACKR3 63 32 CCNC(=O)Cc1ccc(C)cc1N ZINC000217776803 AD In-Stock Unstable P2RX7 18 41 CC(=O)NCCNS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217776818 DC For-Sale Unstable HDAC8 17 47 CC(=O)NCCNS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217776818 DC For-Sale Unstable AKR1C3 26 45 O=C(N/C=C/c1ccccc1F)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217776821 GK For-Sale Mild PTPA 0 46 Cc1cc(OC2CCN(C(=O)COc3ccc(Cl)cc3)CC2)cc(=O)n1C ZINC000217776865 GF In-Stock Unstable PRSS2 61 33 Cc1cc(OC2CCN(C(=O)COc3ccc(Cl)cc3)CC2)cc(=O)n1C ZINC000217776865 GF In-Stock Unstable HRH3 24 41 Cc1cc(OC2CCN(C(=O)COc3ccc(Cl)cc3)CC2)cc(=O)n1C ZINC000217776865 GF In-Stock Unstable COLA 49 38 Cc1cc(OC2CCN(C(=O)COc3ccc(Cl)cc3)CC2)cc(=O)n1C ZINC000217776865 GF In-Stock Unstable CPT1A 45 38 Cc1cc(OC2CCN(C(=O)COc3ccc(Cl)cc3)CC2)cc(=O)n1C ZINC000217776865 GF In-Stock Unstable CPT2 40 38 Cc1cc(OC2CCN(C(=O)COc3ccc(Cl)cc3)CC2)cc(=O)n1C ZINC000217776865 GF In-Stock Unstable EPHX2 15 44 Cn1ccc(NS(=O)(=O)c2cccc(/C=C\C(=O)O)c2)n1 ZINC000217776901 DD For-Sale Unstable HDAC8 37 49 Cn1ccc(NS(=O)(=O)c2cccc(/C=C\C(=O)O)c2)n1 ZINC000217776901 DD For-Sale Unstable HDAC6 16 49 Cc1cc(OC2CCN(C(=O)c3cc(=O)c4ccccc4o3)CC2)cc(=O)n1C ZINC000217776984 GE In-Stock Unstable PRSS2 70 32 Cc1cc(OC2CCN(C(=O)c3cc(=O)c4ccccc4o3)CC2)cc(=O)n1C ZINC000217776984 GE In-Stock Unstable TNKS 30 43 O=C(O)/C=C\c1cccc(S(=O)(=O)Nc2cnccn2)c1 ZINC000217777002 DD For-Sale Anodyne RHOA 0 43 Cc1cc(OC2CCN(C(=O)c3cc4ccccc4oc3=O)CC2)cc(=O)n1C ZINC000217777117 GE In-Stock Unstable PRSS2 50 30 COc1ccc(Br)c(C(=O)N2CCC(Oc3cc(C)n(C)c(=O)c3)CC2)c1 ZINC000217777244 IG In-Stock Unstable PRSS2 45 31 O=C(N/C=C/c1ccccc1F)Nc1ccc(F)c(Cl)c1 ZINC000217777311 DI For-Sale Anodyne P95276_MYCTO 0 44 C[C@H](O)CCNC(=O)/C=C\c1ccc([N+](=O)[O-])cc1 ZINC000217777329 CD On-Demand Unstable PYGL 0 40 C[C@H](O)CCNC(=O)/C=C\c1ccc([N+](=O)[O-])cc1 ZINC000217777329 CD On-Demand Unstable HDAC8 0 50 CCN(C)C(=O)CNC(=O)[C@@H]1CCCC[C@@H]1C(=O)O ZINC000217777363 CC For-Sale Unstable ACE 0 56 Cc1cc(OC2CCN(C(=O)CCc3ccccc3Br)CC2)cc(=O)n1C ZINC000217777365 IG In-Stock Unstable PRSS2 42 30 CCC[C@H](C)NC(=O)[C@@H](C)N[C@@H]1CCN(C)C1=O ZINC000217777407 CC For-Sale Unstable BIRC2 40 30 CNC(=O)CNS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217777414 CB For-Sale Unstable HDAC8 20 47 CNC(=O)CNS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217777414 CB For-Sale Unstable AKR1C3 25 40 O=C(CNC(=O)OCc1ccccc1)NC[C@@H]1CCCN1c1nccs1 ZINC000217777416 FE For-Sale Unstable GRIN2B 20 48 O=C(CNC(=O)OCc1ccccc1)NC[C@@H]1CCCN1c1nccs1 ZINC000217777416 FE For-Sale Unstable CTRA_BOVIN 41 31 O=C(CNC(=O)OCc1ccccc1)NC[C@@H]1CCCN1c1nccs1 ZINC000217777416 FE For-Sale Unstable PREP 36 47 O=C(CNC(=O)OCc1ccccc1)NC[C@@H]1CCCN1c1nccs1 ZINC000217777416 FE For-Sale Unstable CAPN2 65 35 O=C(CNC(=O)OCc1ccccc1)NC[C@@H]1CCCN1c1nccs1 ZINC000217777416 FE For-Sale Unstable NPR 47 31 C[C@@H](O)CCNC(=O)/C=C\c1ccc([N+](=O)[O-])cc1 ZINC000217777427 CD On-Demand Unstable PYGL 0 40 C[C@@H](O)CCNC(=O)/C=C\c1ccc([N+](=O)[O-])cc1 ZINC000217777427 CD On-Demand Unstable HDAC8 0 50 Brc1ccc(-c2nnn(Cc3ccc(-n4ccnc4)cc3)n2)cc1 ZINC000217777453 GG On-Demand Unstable CYP11B2 15 47 CCN(CC)c1ccc(NC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217777460 EI For-Sale Unstable GHSR 0 40 O=S(=O)(CCCCO)Nc1ccc(Cl)c(Cl)c1 ZINC000217777493 CF For-Sale Unstable GRIN1 0 40 CC(=O)Nc1ccc(CC(=O)N2CCC(Oc3cc(C)n(C)c(=O)c3)CC2)cc1 ZINC000217777495 GE In-Stock Unstable TSHR 41 31 CC(=O)Nc1ccc(CC(=O)N2CCC(Oc3cc(C)n(C)c(=O)c3)CC2)cc1 ZINC000217777495 GE In-Stock Unstable PRSS2 67 35 CC(=O)Nc1ccc(CC(=O)N2CCC(Oc3cc(C)n(C)c(=O)c3)CC2)cc1 ZINC000217777495 GE In-Stock Unstable MLNR 29 42 CC(C)n1cc(CC(=O)O)cc1Br ZINC000217777502 BE For-Sale Unstable THRA 23 41 CC(C)n1cc(CC(=O)O)cc1Br ZINC000217777502 BE For-Sale Unstable THRB 18 41 C[C@H](O)CCNC(=O)/C=C\c1c(F)cccc1Cl ZINC000217777507 CE For-Sale Unstable KCNQ2 45 32 O=C(CNC(=O)OCc1ccccc1)NC[C@H]1CCCN1c1nccs1 ZINC000217777512 FE For-Sale Unstable GRIN2B 20 48 O=C(CNC(=O)OCc1ccccc1)NC[C@H]1CCCN1c1nccs1 ZINC000217777512 FE For-Sale Unstable CTRA_BOVIN 41 31 O=C(CNC(=O)OCc1ccccc1)NC[C@H]1CCCN1c1nccs1 ZINC000217777512 FE For-Sale Unstable PREP 36 47 O=C(CNC(=O)OCc1ccccc1)NC[C@H]1CCCN1c1nccs1 ZINC000217777512 FE For-Sale Unstable CAPN2 65 35 O=C(CNC(=O)OCc1ccccc1)NC[C@H]1CCCN1c1nccs1 ZINC000217777512 FE For-Sale Unstable NPR 47 31 C[C@@H](O)CCNC(=O)/C=C\c1c(F)cccc1Cl ZINC000217777575 CE For-Sale Unstable KCNQ2 45 32 COCCCNS(=O)(=O)c1ccc(/C=C\C(=O)O)cc1Cl ZINC000217777581 ED For-Sale Unstable PYGL 0 40 CCC[C@H](C)NC(=O)[C@H](C)N[C@@H]1CCN(C)C1=O ZINC000217777583 CC For-Sale Unstable BIRC2 40 30 COc1ccc([C@@H](C#N)N2CCN(C(=O)Cn3nnc(-c4cccc(F)c4)n3)CC2)cc1 ZINC000217777602 ID On-Demand Unstable PTAFR 44 40 COc1ccc([C@@H](C#N)N2CCN(C(=O)Cn3nnc(-c4cccc(F)c4)n3)CC2)cc1 ZINC000217777602 ID On-Demand Unstable SCARB1 29 41 O=C(N/C=C/c1ccccc1F)NCc1ccc(F)cc1 ZINC000217777614 CG For-Sale Unstable Q76353_9HIV1 0 40 CCCCCNC(=O)Cc1ccc(C)cc1N ZINC000217777621 BE In-Stock Unstable GRIA1 50 34 CCCCCNC(=O)Cc1ccc(C)cc1N ZINC000217777621 BE In-Stock Unstable PA2A1_NAJMO 0 40 CCCCCNC(=O)Cc1ccc(C)cc1N ZINC000217777621 BE In-Stock Unstable ASAH1 72 35 COc1ccc([C@H](C#N)N2CCN(C(=O)Cn3nnc(-c4cccc(F)c4)n3)CC2)cc1 ZINC000217777667 ID On-Demand Unstable PTAFR 44 40 COc1ccc([C@H](C#N)N2CCN(C(=O)Cn3nnc(-c4cccc(F)c4)n3)CC2)cc1 ZINC000217777667 ID On-Demand Unstable SCARB1 29 41 COCCCNS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217777688 CD For-Sale Unstable AKR1C3 27 43 COc1cccc(C(=O)N2[C@@H](C)C[C@@H]3CNC[C@H]32)c1 ZINC000217777707 CD For-Sale Unstable DRD4 45 34 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2F)CC1 ZINC000217777709 FG For-Sale Unstable HTR1A 91 54 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2F)CC1 ZINC000217777709 FG For-Sale Unstable DRD2 69 47 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2F)CC1 ZINC000217777709 FG For-Sale Unstable DRD1 25 40 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2F)CC1 ZINC000217777709 FG For-Sale Unstable DRD4 38 46 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2F)CC1 ZINC000217777709 FG For-Sale Unstable ADRA1D 70 39 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2F)CC1 ZINC000217777709 FG For-Sale Unstable HTR1D 26 54 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2F)CC1 ZINC000217777709 FG For-Sale Unstable HTR1B 21 54 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2F)CC1 ZINC000217777709 FG For-Sale Unstable HTR2A 35 44 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2F)CC1 ZINC000217777709 FG For-Sale Unstable ADRA1A 63 40 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2F)CC1 ZINC000217777709 FG For-Sale Unstable ADRA1B 56 39 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2F)CC1 ZINC000217777709 FG For-Sale Unstable DRD3 75 46 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2F)CC1 ZINC000217777709 FG For-Sale Unstable HTR7 59 47 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2F)CC1 ZINC000217777709 FG For-Sale Unstable TACR3 24 46 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2F)CC1 ZINC000217777709 FG For-Sale Unstable RBP4 15 45 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2F)CC1 ZINC000217777709 FG For-Sale Unstable AP2S1 0 40 Cc1cc(OC2CCN(C(=O)c3ccc4cc[nH]c4c3)CC2)cc(=O)n1C ZINC000217777723 FF In-Stock Unstable GRIN2B 20 44 Cc1cc(OC2CCN(C(=O)c3ccc4cc[nH]c4c3)CC2)cc(=O)n1C ZINC000217777723 FF In-Stock Unstable PRSS2 68 35 Cc1cc(OC2CCN(C(=O)c3ccc4cc[nH]c4c3)CC2)cc(=O)n1C ZINC000217777723 FF In-Stock Unstable HRH3 20 48 Cc1cc(OC2CCN(C(=O)c3ccc4cc[nH]c4c3)CC2)cc(=O)n1C ZINC000217777723 FF In-Stock Unstable GHSR 15 50 Cc1cc(OC2CCN(C(=O)c3ccc4cc[nH]c4c3)CC2)cc(=O)n1C ZINC000217777723 FF In-Stock Unstable L3MBTL3 51 41 COc1cccc(C(=O)N2[C@@H]3CNC[C@H]3C[C@H]2C)c1 ZINC000217777783 CD For-Sale Unstable DRD4 45 34 CCC[C@@H](N)C(=O)N[C@@H]1C[C@@H]2CC[C@@]1(C)C2(C)C ZINC000217777855 CE For-Sale Unstable AVPR2 25 40 COc1cccc(C(=O)N2[C@@H](C)C[C@H]3CNC[C@H]32)c1 ZINC000217777860 CD For-Sale Unstable DRD4 45 34 COCCCCNS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217777874 DD For-Sale Unstable AKR1C3 27 45 COc1cccc(C(=O)N2[C@@H]3CNC[C@@H]3C[C@H]2C)c1 ZINC000217777936 CD For-Sale Unstable DRD4 45 34 Cc1cc(S(=O)(=O)N(C)CCO)ccc1/C=C\C(=O)O ZINC000217777943 CC For-Sale Unstable AURKAIP1 0 40 Cc1cc2c(SCC(=O)N3CCC[C@@H]3c3ccccn3)ncnc2s1 ZINC000217777948 FH In-Stock Unstable COLA 82 38 Cc1cc2c(SCC(=O)N3CCC[C@@H]3c3ccccn3)ncnc2s1 ZINC000217777948 FH In-Stock Unstable CPT1A 79 38 CCC[C@H](N)C(=O)N[C@@H]1C[C@@H]2CC[C@@]1(C)C2(C)C ZINC000217777954 CE For-Sale Unstable AVPR2 25 40 Cc1cc(OC2CCN(S(=O)(=O)c3cccs3)CC2)cc(=O)n1C ZINC000217777969 FD In-Stock Unstable FAAH 0 41 Cc1cc2c(SCC(=O)N3CCC[C@H]3c3ccccn3)ncnc2s1 ZINC000217778017 FH In-Stock Unstable COLA 82 38 Cc1cc2c(SCC(=O)N3CCC[C@H]3c3ccccn3)ncnc2s1 ZINC000217778017 FH In-Stock Unstable CPT1A 79 38 CCC[C@@H](N)C(=O)N[C@H]1C[C@@H]2CC[C@@]1(C)C2(C)C ZINC000217778026 CE For-Sale Unstable AVPR2 25 40 C[C@H](O)CCNC(=O)/C=C\c1ccc(F)c(Cl)c1 ZINC000217778050 CE For-Sale Unstable HDAC1 18 41 C[C@H](O)CCNC(=O)/C=C\c1ccc(F)c(Cl)c1 ZINC000217778050 CE For-Sale Unstable HDAC2 16 41 C[C@H](O)CCNC(=O)/C=C\c1ccc(F)c(Cl)c1 ZINC000217778050 CE For-Sale Unstable HDAC4 23 41 C[C@H](O)CCNC(=O)/C=C\c1ccc(F)c(Cl)c1 ZINC000217778050 CE For-Sale Unstable HPSE 21 40 C[C@H](O)CCNC(=O)/C=C\c1ccc(F)c(Cl)c1 ZINC000217778050 CE For-Sale Unstable HDAC9 33 41 C[C@H](O)CCNC(=O)/C=C\c1ccc(F)c(Cl)c1 ZINC000217778050 CE For-Sale Unstable HDAC7 35 41 Cc1ccc(CC(=O)N2CCCCC2)c(N)c1 ZINC000217778067 BE In-Stock Unstable ECE2 0 40 CC(C)(C)OC(=O)N[C@H](C(F)(F)F)C1(N)CC1 ZINC000217778077 CD For-Sale Unstable CTSK 22 41 CCC[C@H](N)C(=O)N[C@H]1C[C@@H]2CC[C@@]1(C)C2(C)C ZINC000217778103 CE For-Sale Unstable AVPR2 25 40 C[C@@H](O)CCNC(=O)/C=C\c1ccc(F)c(Cl)c1 ZINC000217778147 CE On-Demand Unstable HDAC4 23 41 C[C@@H](O)CCNC(=O)/C=C\c1ccc(F)c(Cl)c1 ZINC000217778147 CE On-Demand Unstable HDAC9 33 41 C[C@@H](O)CCNC(=O)/C=C\c1ccc(F)c(Cl)c1 ZINC000217778147 CE On-Demand Unstable HDAC7 31 41 C[C@@H](O)CCNC(=O)/C=C\c1ccc(F)c(Cl)c1 ZINC000217778147 CE On-Demand Unstable HD1B 0 42 CN1CCO[C@@H](CNC(=O)[C@@H](C#N)Cc2ccccc2)C1 ZINC000217778148 CC For-Sale Unstable MME 41 36 CC(C)(C)OC(=O)N[C@@H](C(F)(F)F)C1(N)CC1 ZINC000217778158 CD For-Sale Unstable CTSK 22 41 O=C(N/C=C/c1ccccc1F)NC1CCCCCC1 ZINC000217778160 CH For-Sale Unstable EPHX2 26 48 O=C(O)/C=C\c1cccc(S(=O)(=O)NCC2CCCC2)c1 ZINC000217778205 DE For-Sale Unstable NPY2R 64 41 O=C(O)/C=C\c1cccc(S(=O)(=O)NCC2CCCC2)c1 ZINC000217778205 DE For-Sale Unstable HDAC8 19 48 O=C(O)/C=C\c1cccc(S(=O)(=O)NCC2CCCC2)c1 ZINC000217778205 DE For-Sale Unstable SFRP1 40 32 CC(C)[C@@H]1CC[C@@H](N)[C@@H](Cc2cccc(C(F)(F)F)c2)C1 ZINC000217778224 CJ For-Sale Unstable PDS 15 42 COc1ccc(CN2C(=O)N[C@@H](CCC(=O)N[C@H](CO)Cc3ccccc3)C2=O)cc1 ZINC000217778226 ID In-Stock Unstable MMP1 16 42 CN1CCO[C@H](CNC(=O)[C@@H](C#N)Cc2ccccc2)C1 ZINC000217778235 CC For-Sale Unstable MME 41 36 CN(c1ccccc1C#N)c1ccc(Cl)cc1CBr ZINC000217778286 EJ For-Sale Unstable NOS2 20 40 CN(c1ccccc1C#N)c1ccc(Cl)cc1CBr ZINC000217778286 EJ For-Sale Unstable NOS3 17 40 Cc1cc(F)ccc1S(=O)(=O)N1CCC(Oc2cc(C)n(C)c(=O)c2)CC1 ZINC000217778290 GE In-Stock Unstable EPHX2 16 48 CC(C)[C@H]1CC[C@@H](N)[C@@H](Cc2cccc(C(F)(F)F)c2)C1 ZINC000217778325 CJ For-Sale Unstable PDS 15 42 COc1ccc(-n2c(=O)ssc2=O)cc1 ZINC000217778339 BD For-Sale Unstable ERCC5 15 44 COc1ccc(-n2c(=O)ssc2=O)cc1 ZINC000217778339 BD For-Sale Unstable NPBWR1 40 35 COc1cc(CN2C[C@@H](C)OC[C@@H]2C)ccc1O ZINC000217778358 CE For-Sale Unstable SHBG 16 50 CC[C@@H](C)N(C)S(=O)(=O)c1ccc(/C=C\C(=O)O)cc1Cl ZINC000217778359 EF For-Sale Unstable NR0B2 0 44 COc1cc(NC(=O)NC[C@@H]2CCCN2c2nccs2)cc(OC)c1OC ZINC000217778378 GF For-Sale Unstable DRD2 29 40 CC(C)[C@@H]1CC[C@H](N)[C@@H](Cc2cccc(C(F)(F)F)c2)C1 ZINC000217778424 CJ For-Sale Unstable PDS 15 42 COc1cc(CN2C[C@H](C)OC[C@@H]2C)ccc1O ZINC000217778442 CE For-Sale Unstable SHBG 16 50 COc1cc(NC(=O)NC[C@H]2CCCN2c2nccs2)cc(OC)c1OC ZINC000217778444 GF For-Sale Unstable DRD2 29 40 C[C@H]1C[C@@H]2CNC[C@H]2N1C(=O)[C@H]1C[C@H]1C ZINC000217778454 BC For-Sale Unstable CHRNA7 0 56 C[C@H](O)[C@@H](NC(=O)N(C)[C@@H](C)c1ccc(Cl)cc1)C(=O)O ZINC000217778455 DD For-Sale Unstable UTS2 47 37 CC[C@H](C)N(C)S(=O)(=O)c1ccc(/C=C\C(=O)O)cc1Cl ZINC000217778456 EF For-Sale Unstable NR0B2 0 44 CC(C)[C@H]1CC[C@H](N)[C@@H](Cc2cccc(C(F)(F)F)c2)C1 ZINC000217778498 CJ For-Sale Unstable PDS 15 42 Cc1cc(OC2CCN(S(=O)(=O)c3ccccc3Cl)CC2)cc(=O)n1C ZINC000217778502 GF In-Stock Unstable HRH1 25 42 Cc1cc(OC2CCN(S(=O)(=O)c3ccccc3Cl)CC2)cc(=O)n1C ZINC000217778502 GF In-Stock Unstable CCR3 31 41 C#C[C@@H](O)[C@H](NC(=O)OC(C)(C)C)C(C)C ZINC000217778532 BD For-Sale Unstable PAPA1_CARPA 43 35 C#C[C@@H](O)[C@H](NC(=O)OC(C)(C)C)C(C)C ZINC000217778532 BD For-Sale Unstable CTSK 23 47 C#C[C@@H](O)[C@H](NC(=O)OC(C)(C)C)C(C)C ZINC000217778532 BD For-Sale Unstable PGA5 41 37 C[C@H](O)[C@H](NC(=O)N(C)[C@@H](C)c1ccc(Cl)cc1)C(=O)O ZINC000217778537 DD For-Sale Unstable UTS2 47 37 C[C@H]1C[C@@H]1C(=O)N1[C@@H](C)C[C@@H]2CNC[C@H]21 ZINC000217778547 BC For-Sale Unstable CHRNA7 0 56 COCc1cc(=O)c(O)c([C@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2cc(OC)c(O)c(OC)c2)o1 ZINC000217778550 KH In-Stock Unstable RORC 42 33 Cc1ccc(CC(=O)N2CCC(C)CC2)c(N)c1 ZINC000217778570 BE In-Stock Unstable TRPC6 40 39 COC1CCN(C2CCN(C(=O)c3cccc(Cl)c3)CC2)CC1 ZINC000217778576 EG In-Stock Unstable CHRM2 57 44 COC1CCN(C2CCN(C(=O)c3cccc(Cl)c3)CC2)CC1 ZINC000217778576 EG In-Stock Unstable HRH1 21 54 COC1CCN(C2CCN(C(=O)c3cccc(Cl)c3)CC2)CC1 ZINC000217778576 EG In-Stock Unstable INHA 17 43 COC1CCN(C2CCN(C(=O)c3cccc(Cl)c3)CC2)CC1 ZINC000217778576 EG In-Stock Unstable HRH3 32 47 COC1CCN(C2CCN(C(=O)c3cccc(Cl)c3)CC2)CC1 ZINC000217778576 EG In-Stock Unstable HSD11B1 15 52 COC1CCN(C2CCN(C(=O)c3cccc(Cl)c3)CC2)CC1 ZINC000217778576 EG In-Stock Unstable CCR3 54 58 COC1CCN(C2CCN(C(=O)c3cccc(Cl)c3)CC2)CC1 ZINC000217778576 EG In-Stock Unstable L3MBTL3 89 59 Cc1cc(OC2CCN(S(=O)(=O)c3c(F)cccc3F)CC2)cc(=O)n1C ZINC000217778611 GE In-Stock Unstable PKM 29 48 C#C[C@H](O)[C@H](NC(=O)OC(C)(C)C)C(C)C ZINC000217778612 BD For-Sale Unstable PAPA1_CARPA 43 35 C#C[C@H](O)[C@H](NC(=O)OC(C)(C)C)C(C)C ZINC000217778612 BD For-Sale Unstable CTSK 23 47 C#C[C@H](O)[C@H](NC(=O)OC(C)(C)C)C(C)C ZINC000217778612 BD For-Sale Unstable PGA5 41 37 COCc1cc(=O)c(O)c([C@@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2cc(OC)c(O)c(OC)c2)o1 ZINC000217778618 KH In-Stock Unstable RORC 42 33 C[C@H]1C[C@@H]2CNC[C@H]2N1C(=O)[C@@H]1C[C@H]1C ZINC000217778638 BC For-Sale Unstable CHRNA7 0 56 Cc1ccc(CC(=O)N2C[C@@H](C)C[C@@H](C)C2)c(N)c1 ZINC000217778687 CF In-Stock Unstable RORC 22 40 COc1ccc(OCCNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217778709 EG For-Sale Unstable MTNR1A 36 45 COc1ccc(OCCNC(=O)N/C=C/c2ccccc2F)cc1 ZINC000217778709 EG For-Sale Unstable MTNR1B 29 45 CCN(CCO)S(=O)(=O)c1ccc(/C=C\C(=O)O)cc1Cl ZINC000217778719 ED For-Sale Unstable NR0B2 0 41 Cc1cc(OC2CCN(S(=O)(=O)Cc3cccc(Cl)c3)CC2)cc(=O)n1C ZINC000217778725 HF In-Stock Unstable PRSS2 44 32 C[C@H]1C[C@H]1C(=O)N1[C@@H](C)C[C@@H]2CNC[C@H]21 ZINC000217778730 BC For-Sale Unstable CHRNA7 0 56 COc1ccc2[nH]c3c(c2c1)CCC[C@@H]3NC(=O)C(C)C ZINC000217778760 CG In-Stock Unstable MAPKAPK2 27 51 COc1ccc2[nH]c3c(c2c1)CCC[C@@H]3NC(=O)C(C)C ZINC000217778760 CG In-Stock Unstable MTNR1A 44 40 Cc1ccc(CC(=O)N2C[C@H](C)C[C@@H](C)C2)c(N)c1 ZINC000217778768 CF In-Stock Unstable RORC 22 40 COC1CCN(C2CCN(C(=O)c3cnc(C)cn3)CC2)CC1 ZINC000217778801 DD In-Stock Unstable CHRM2 40 34 COC1CCN(C2CCN(C(=O)c3cnc(C)cn3)CC2)CC1 ZINC000217778801 DD In-Stock Unstable CCR3 24 40 COC1CCN(C2CCN(C(=O)c3cnc(C)cn3)CC2)CC1 ZINC000217778801 DD In-Stock Unstable L3MBTL3 70 42 Cc1cc(OC2CCN(S(=O)(=O)c3ccc(F)c(Cl)c3)CC2)cc(=O)n1C ZINC000217778826 HF In-Stock Unstable GPR119 15 43 COc1ccc2[nH]c3c(c2c1)CCC[C@H]3NC(=O)C(C)C ZINC000217778828 CG In-Stock Unstable MAPKAPK2 27 51 COc1ccc2[nH]c3c(c2c1)CCC[C@H]3NC(=O)C(C)C ZINC000217778828 CG In-Stock Unstable MTNR1A 44 40 CCN(C)C(=O)CNC(=O)[C@@H]1CCC[C@@H]1C(=O)O ZINC000217778836 CC For-Sale Unstable ACE 0 53 Cc1ccc(CC(=O)N2C[C@@H](C)C[C@H](C)C2)c(N)c1 ZINC000217778858 CF In-Stock Unstable RORC 22 40 CC(C)C[C@@H](C)NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217778894 DE For-Sale Unstable HDAC8 16 46 CC(C)C[C@@H](C)NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217778894 DE For-Sale Unstable CAPN1 17 40 CC(C)C[C@@H](C)NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217778894 DE For-Sale Unstable LEF 17 43 CC(=O)NCCNC(=O)N/C=C/c1ccccc1F ZINC000217778920 CD For-Sale Unstable MTNR1A 25 48 CC(=O)NCCNC(=O)N/C=C/c1ccccc1F ZINC000217778920 CD For-Sale Unstable MTNR1B 22 48 CCN(C)C(=O)CNC(=O)[C@H]1CCC[C@@H]1C(=O)O ZINC000217778927 CC For-Sale Unstable ACE 0 53 Cc1cc(OC2CCN(S(=O)(=O)c3ccc4c(c3)CCCC4)CC2)cc(=O)n1C ZINC000217778932 HF In-Stock Unstable CASP7 46 32 COc1ccc([C@@H]2CC(=O)Oc3ccc4c(c32)OC(C)(C)CC4=O)c(OC)c1 ZINC000217778936 GH In-Stock Unstable MT-ND4 51 32 CC(C)C[C@H](C)NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217778973 DE For-Sale Unstable HDAC8 16 46 CC(C)C[C@H](C)NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217778973 DE For-Sale Unstable CAPN1 17 40 CC(C)C[C@H](C)NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217778973 DE For-Sale Unstable LEF 17 43 CCN(C)C(=O)CNC(=O)[C@@H]1CCC[C@H]1C(=O)O ZINC000217779012 CC For-Sale Unstable ACE 0 53 COc1ccc([C@H]2CC(=O)Oc3ccc4c(c32)OC(C)(C)CC4=O)c(OC)c1 ZINC000217779030 GH In-Stock Unstable MT-ND4 51 32 Cc1cc(OC2CCN(S(=O)(=O)c3ccc4c(c3)OCCO4)CC2)cc(=O)n1C ZINC000217779031 HD In-Stock Unstable PKM 52 54 COc1ccc(C(=O)N2CCC(N3CCC(OC)CC3)CC2)c(OC)c1OC ZINC000217779032 GE In-Stock Unstable CHRM2 61 44 COc1ccc(C(=O)N2CCC(N3CCC(OC)CC3)CC2)c(OC)c1OC ZINC000217779032 GE In-Stock Unstable HRH1 15 41 COc1ccc(C(=O)N2CCC(N3CCC(OC)CC3)CC2)c(OC)c1OC ZINC000217779032 GE In-Stock Unstable CCR3 36 41 COc1ccc(C(=O)N2CCC(N3CCC(OC)CC3)CC2)c(OC)c1OC ZINC000217779032 GE In-Stock Unstable L3MBTL3 93 51 Brc1cc2cc(OCc3ccccc3)ccc2[nH]1 ZINC000217779052 DJ For-Sale Unstable MAOA 19 56 Brc1cc2cc(OCc3ccccc3)ccc2[nH]1 ZINC000217779052 DJ For-Sale Unstable MAOB 46 56 Brc1cc2cc(OCc3ccccc3)ccc2[nH]1 ZINC000217779052 DJ For-Sale Unstable SRD5A2 16 40 Brc1cc2cc(OCc3ccccc3)ccc2[nH]1 ZINC000217779052 DJ For-Sale Unstable LTA4H 18 42 CN1CC[C@@H](CCC(=O)O)CCC1=O ZINC000217779061 AD In-Stock Unstable CYP2J2 44 32 CCCCCNC(=O)[C@@H](C)N[C@@H]1CCN(C)C1=O ZINC000217779087 CC For-Sale Unstable ASAH1 85 35 CCCCCNC(=O)[C@@H](C)N[C@@H]1CCN(C)C1=O ZINC000217779087 CC For-Sale Unstable LASR 44 33 CCN(C)C(=O)CNC(=O)[C@H]1CCC[C@H]1C(=O)O ZINC000217779089 CC For-Sale Unstable ACE 0 53 Cc1cc(S(=O)(=O)NCC(=O)N2CCc3n[nH]cc3C2)ccc1F ZINC000217779123 FC In-Stock Unstable LEF 65 39 OCCN1CCN(Cc2ccc(CN3CCN(CCO)CC3)cc2)CC1 ZINC000217779127 FB On-Demand Unstable DRD2 18 44 OCCN1CCN(Cc2ccc(CN3CCN(CCO)CC3)cc2)CC1 ZINC000217779127 FB On-Demand Unstable DRD4 33 42 OCCN1CCN(Cc2ccc(CN3CCN(CCO)CC3)cc2)CC1 ZINC000217779127 FB On-Demand Unstable HRH3 24 48 OCCN1CCN(Cc2ccc(CN3CCN(CCO)CC3)cc2)CC1 ZINC000217779127 FB On-Demand Unstable SIGMAR1 67 54 OCCN1CCN(Cc2ccc(CN3CCN(CCO)CC3)cc2)CC1 ZINC000217779127 FB On-Demand Unstable CXCR4 21 41 OCCN1CCN(Cc2ccc(CN3CCN(CCO)CC3)cc2)CC1 ZINC000217779127 FB On-Demand Unstable CACNA1G 15 44 COCCNC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217779128 FC In-Stock Unstable EDNRA 24 40 COCCNC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217779128 FC In-Stock Unstable TACR1 20 40 COCCNC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217779128 FC In-Stock Unstable MC4R 41 38 COCCNC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217779128 FC In-Stock Unstable BRS3 21 40 COCCNC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217779128 FC In-Stock Unstable NMBR 29 40 COCCNC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217779128 FC In-Stock Unstable GHSR 41 36 COCCNC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217779128 FC In-Stock Unstable MMP1 15 43 O=C(N/C=C/c1ccccc1F)NC12CC3CC(CC(C3)C1)C2 ZINC000217779139 DI For-Sale Unstable EPHX2 102 50 CN1CC[C@H](CCC(=O)O)CCC1=O ZINC000217779149 AD In-Stock Unstable CYP2J2 44 32 O=C(O)CC[C@@H](NC(=O)N[C@@H]1CCN(C2CC2)C1)C(=O)O ZINC000217779164 CB For-Sale Unstable FOLH1 56 53 O=C(O)CC[C@@H](NC(=O)N[C@@H]1CCN(C2CC2)C1)C(=O)O ZINC000217779164 CB For-Sale Unstable NAALAD2 74 53 CCOc1ccc(S(=O)(=O)N2CCC(Oc3cc(C)n(C)c(=O)c3)CC2)cc1F ZINC000217779170 HE In-Stock Unstable PDE5A 35 41 CCOc1ccc(S(=O)(=O)N2CCC(Oc3cc(C)n(C)c(=O)c3)CC2)cc1F ZINC000217779170 HE In-Stock Unstable GPR119 24 41 CCCCCNC(=O)[C@H](C)N[C@@H]1CCN(C)C1=O ZINC000217779179 CC For-Sale Unstable ASAH1 85 35 CCCCCNC(=O)[C@H](C)N[C@@H]1CCN(C)C1=O ZINC000217779179 CC For-Sale Unstable LASR 44 33 Cc1ccc(CC(=O)N2CCOCC2)c(N)c1 ZINC000217779223 BC In-Stock Unstable AKR1C3 29 44 O=C(O)CC[C@@H](NC(=O)N[C@H]1CCN(C2CC2)C1)C(=O)O ZINC000217779241 CB For-Sale Unstable FOLH1 56 53 O=C(O)CC[C@@H](NC(=O)N[C@H]1CCN(C2CC2)C1)C(=O)O ZINC000217779241 CB For-Sale Unstable NAALAD2 74 53 COc1cc2c(cc1OC)CC(=O)N(CC(=O)N[C@H](CO)Cc1ccccc1)C=C2 ZINC000217779244 HD In-Stock Unstable HCN2 0 40 CCCCCNC(=O)[C@@H](C)N[C@H]1CCN(C)C1=O ZINC000217779252 CC For-Sale Unstable ASAH1 85 35 CCCCCNC(=O)[C@@H](C)N[C@H]1CCN(C)C1=O ZINC000217779252 CC For-Sale Unstable LASR 44 33 Cc1cc(OC2CCN(S(=O)(=O)c3cccc(C(F)(F)F)c3)CC2)cc(=O)n1C ZINC000217779277 IF In-Stock Unstable CACNA1B 54 39 Cc1cc(OC2CCN(S(=O)(=O)c3cccc(C(F)(F)F)c3)CC2)cc(=O)n1C ZINC000217779277 IF In-Stock Unstable PKM 18 45 CCCCCNC(=O)[C@H](C)N[C@H]1CCN(C)C1=O ZINC000217779328 CC For-Sale Unstable ASAH1 85 35 CCCCCNC(=O)[C@H](C)N[C@H]1CCN(C)C1=O ZINC000217779328 CC For-Sale Unstable LASR 44 33 COc1ccc(SCc2ccc(-n3ccnc3)cc2)cc1 ZINC000217779346 CI On-Demand Unstable CYP19A1 0 44 COc1ccc(SCc2ccc(-n3ccnc3)cc2)cc1 ZINC000217779346 CI On-Demand Unstable CYP1A2 15 50 COc1ccc(SCc2ccc(-n3ccnc3)cc2)cc1 ZINC000217779346 CI On-Demand Unstable CYP2C19 36 50 C[C@@H]1CCN(CCOCc2ccccc2)C1 ZINC000217779464 BF On-Demand Unstable DRD2 16 43 C[C@@H]1CCN(CCOCc2ccccc2)C1 ZINC000217779464 BF On-Demand Unstable SLC6A1 45 40 C[C@@H]1CCN(CCOCc2ccccc2)C1 ZINC000217779464 BF On-Demand Unstable HRH1 15 41 C[C@@H]1CCN(CCOCc2ccccc2)C1 ZINC000217779464 BF On-Demand Unstable LTA4H 26 40 C[C@@H]1CCN(CCOCc2ccccc2)C1 ZINC000217779464 BF On-Demand Unstable UGCG 48 37 C[C@@H]1CCN(CCOCc2ccccc2)C1 ZINC000217779464 BF On-Demand Unstable HRH3 15 47 C[C@@H]1CCN(CCOCc2ccccc2)C1 ZINC000217779464 BF On-Demand Unstable SIGMAR1 58 56 C[C@@H]1CCN(CCOCc2ccccc2)C1 ZINC000217779464 BF On-Demand Unstable GBA 29 42 C[C@@H]1CCN(CCOCc2ccccc2)C1 ZINC000217779464 BF On-Demand Unstable EBP 26 40 C[C@@H]1CCN(CCOCc2ccccc2)C1 ZINC000217779464 BF On-Demand Unstable GBA2 49 42 C[C@@H]1Cc2ccccc2N1C(=O)N/C=C/c1ccccc1F ZINC000217779492 CH For-Sale Unstable DRD4 26 43 C[C@@H]1Cc2ccccc2N1C(=O)N/C=C/c1ccccc1F ZINC000217779492 CH For-Sale Unstable TPP2 45 34 CCc1ccc([C@H](C)NC(=O)[C@H](N)[C@H](C)CC)cc1 ZINC000217779533 CF On-Demand Unstable ACACA 24 41 CCc1ccc([C@H](C)NC(=O)[C@H](N)[C@H](C)CC)cc1 ZINC000217779533 CF On-Demand Unstable ACACB 28 41 CCc1ccc([C@H](C)NC(=O)[C@H](N)[C@H](C)CC)cc1 ZINC000217779533 CF On-Demand Unstable CAPN2 52 36 CCc1ccc([C@H](C)NC(=O)[C@H](N)[C@H](C)CC)cc1 ZINC000217779533 CF On-Demand Unstable ACE2 56 38 CCc1ccc([C@H](C)NC(=O)[C@H](N)[C@H](C)CC)cc1 ZINC000217779533 CF On-Demand Unstable SLC15A2 0 53 C[C@H]1CCN(CCOCc2ccccc2)C1 ZINC000217779553 BF On-Demand Unstable DRD2 16 43 C[C@H]1CCN(CCOCc2ccccc2)C1 ZINC000217779553 BF On-Demand Unstable SLC6A1 45 40 C[C@H]1CCN(CCOCc2ccccc2)C1 ZINC000217779553 BF On-Demand Unstable HRH1 15 41 C[C@H]1CCN(CCOCc2ccccc2)C1 ZINC000217779553 BF On-Demand Unstable LTA4H 26 40 C[C@H]1CCN(CCOCc2ccccc2)C1 ZINC000217779553 BF On-Demand Unstable UGCG 48 37 C[C@H]1CCN(CCOCc2ccccc2)C1 ZINC000217779553 BF On-Demand Unstable HRH3 15 47 C[C@H]1CCN(CCOCc2ccccc2)C1 ZINC000217779553 BF On-Demand Unstable SIGMAR1 58 56 C[C@H]1CCN(CCOCc2ccccc2)C1 ZINC000217779553 BF On-Demand Unstable GBA 29 42 C[C@H]1CCN(CCOCc2ccccc2)C1 ZINC000217779553 BF On-Demand Unstable EBP 26 40 C[C@H]1CCN(CCOCc2ccccc2)C1 ZINC000217779553 BF On-Demand Unstable GBA2 49 42 O=C(NC[C@@H]1CCCN1c1nccs1)Nc1ccc(F)cc1 ZINC000217779571 DG For-Sale Unstable CCR3 60 40 CCN(C1CC1)S(=O)(=O)c1ccc(/C=C\C(=O)O)cc1Cl ZINC000217779573 EF For-Sale Unstable NR0B2 0 40 C[C@H]1Cc2ccccc2N1C(=O)N/C=C/c1ccccc1F ZINC000217779574 CH For-Sale Unstable DRD4 26 43 C[C@H]1Cc2ccccc2N1C(=O)N/C=C/c1ccccc1F ZINC000217779574 CH For-Sale Unstable TPP2 45 34 Cc1ccc(CC(=O)N2CCN(C)CC2)c(N)c1 ZINC000217779577 BC In-Stock Unstable HRH4 26 43 O=C(NC[C@H]1CCCN1c1nccs1)Nc1ccc(F)cc1 ZINC000217779648 DG For-Sale Unstable CCR3 60 40 Cc1ccc(CC(=O)N2CCCCCC2)c(N)c1 ZINC000217779654 BF In-Stock Unstable ECE2 0 40 Cc1cc(OC2CCN(S(=O)(=O)CCCOc3ccccc3)CC2)cc(=O)n1C ZINC000217779719 HE In-Stock Unstable MMP13 15 44 CC(C)c1nc2cc(NC(=O)[C@@H]3CC(=O)N(CCc4ccc(O)cc4)C3)ccc2[nH]1 ZINC000217779731 HG In-Stock Unstable NR2E3 46 34 CCOC(=O)c1ccn(-c2ccc(Cl)c(F)c2)n1 ZINC000217779784 CF For-Sale Unstable Q9FYV8_MAIZE 28 40 O=C(NC[C@@H]1CCCN1c1nccs1)Nc1ccc(C(F)(F)F)cc1 ZINC000217779785 FH For-Sale Unstable EPHX2 31 43 CC(C)c1nc2cc(NC(=O)[C@H]3CC(=O)N(CCc4ccc(O)cc4)C3)ccc2[nH]1 ZINC000217779819 HG In-Stock Unstable NR2E3 46 34 CN(CC1CC1)S(=O)(=O)c1ccc(/C=C\C(=O)O)cc1Cl ZINC000217779826 EE For-Sale Unstable NR0B2 0 40 O=C(NC[C@H]1CCCN1c1nccs1)Nc1ccc(C(F)(F)F)cc1 ZINC000217779868 FH For-Sale Unstable EPHX2 31 43 NC(=O)CC[C@@H](NC(=O)N[C@@H]1CCN(C2CC2)C1)C(=O)O ZINC000217779918 CB For-Sale Unstable NAALAD2 54 40 NC(=O)CC[C@@H](NC(=O)N[C@@H]1CCN(C2CC2)C1)C(=O)O ZINC000217779918 CB For-Sale Unstable SLC5A1 15 40 O=C(N/C=C/c1ccccc1F)N1CCN(c2ncccn2)CC1 ZINC000217779920 EE For-Sale Unstable FAAH 21 40 O=C(N/C=C/c1ccccc1F)N1CCN(c2ncccn2)CC1 ZINC000217779920 EE For-Sale Unstable SLC6A7 0 46 Cc1ccc(CC(=O)NC2CCCC2)c(N)c1 ZINC000217779924 BE In-Stock Unstable FAAH 17 45 Cc1ccc(CC(=O)NC2CCCC2)c(N)c1 ZINC000217779924 BE In-Stock Unstable EPHX2 27 46 COc1ccc(CN2C(=O)N[C@@H](CC(=O)NC[C@@H]3CCCN4CCCC[C@H]34)C2=O)cc1 ZINC000217779936 ID In-Stock Unstable PROKR1 42 29 CCN(C)C(=O)CNC(=O)CCC(=O)O ZINC000217779970 BB On-Demand Unstable KDM2A 48 39 COc1cccc(NC(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217779977 EF For-Sale Unstable HRH2 19 44 COc1cccc(NC(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217779977 EF For-Sale Unstable CCR3 48 45 COc1cccc(NC(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217779977 EF For-Sale Unstable CHRNA7 17 44 COc1cccc(NC(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217779977 EF For-Sale Unstable EPHX2 29 44 COc1cc(CCN)c(O)cc1Br ZINC000217779979 BD For-Sale Unstable HTR2A 17 72 COc1cc(CCN)c(O)cc1Br ZINC000217779979 BD For-Sale Unstable HTR2C 17 72 NC(=O)CC[C@@H](NC(=O)N[C@H]1CCN(C2CC2)C1)C(=O)O ZINC000217780003 CB For-Sale Unstable NAALAD2 54 40 NC(=O)CC[C@@H](NC(=O)N[C@H]1CCN(C2CC2)C1)C(=O)O ZINC000217780003 CB For-Sale Unstable SLC5A1 15 40 Cc1ccc(CC(=O)NC2CCCCC2)c(N)c1 ZINC000217780018 BF In-Stock Unstable CNR2 19 42 Cc1ccc(CC(=O)NC2CCCCC2)c(N)c1 ZINC000217780018 BF In-Stock Unstable FAAH 22 47 Cc1ccc(CC(=O)NC2CCCCC2)c(N)c1 ZINC000217780018 BF In-Stock Unstable EPHX2 36 48 COC(=O)Nc1ccc(S(=O)(=O)N2CCC(Oc3cc(C)n(C)c(=O)c3)CC2)cc1 ZINC000217780045 IE In-Stock Unstable TGM1 23 41 COC(=O)Nc1ccc(S(=O)(=O)N2CCC(Oc3cc(C)n(C)c(=O)c3)CC2)cc1 ZINC000217780045 IE In-Stock Unstable EPHX2 27 42 COC(=O)Nc1ccc(S(=O)(=O)N2CCC(Oc3cc(C)n(C)c(=O)c3)CC2)cc1 ZINC000217780045 IE In-Stock Unstable TGM2 77 42 COC(=O)Nc1ccc(S(=O)(=O)N2CCC(Oc3cc(C)n(C)c(=O)c3)CC2)cc1 ZINC000217780045 IE In-Stock Unstable F13A1 105 42 NCC1CCC(N)(C(=O)O)CC1 ZINC000217780046 AB In-Stock Unstable GRM1 0 48 COC(=O)C[C@H](c1cc(Br)cc2c1OCOC2)c1c(O)c2ccccc2oc1=O ZINC000217780047 JH In-Stock Unstable NQO1 32 42 CCN(C)C(=O)CNC(=O)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217780072 CD On-Demand Unstable TAAR1 19 47 CNC(=O)CN(C)S(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217780085 DC For-Sale Unstable HDAC8 18 41 COc1cccc(NC(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217780090 EF For-Sale Unstable HRH2 19 44 COc1cccc(NC(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217780090 EF For-Sale Unstable CCR3 48 45 COc1cccc(NC(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217780090 EF For-Sale Unstable CHRNA7 17 44 COc1cccc(NC(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217780090 EF For-Sale Unstable EPHX2 29 44 COC(=O)c1ccc(CNC(=O)[C@@H](C)N[C@@H](C)c2ccc(OC)c(Br)c2)cc1 ZINC000217780100 IH On-Demand Unstable TRPV1 24 44 COc1cc([C@H](C)N)c(O)cc1Br ZINC000217780103 BE For-Sale Unstable P2RX2 15 40 COC(=O)C[C@@H](c1cc(Br)cc2c1OCOC2)c1c(O)c2ccccc2oc1=O ZINC000217780132 JH In-Stock Unstable NQO1 32 42 CN1CC[C@@H](NC[C@@](C)(O)c2ccccc2)C1=O ZINC000217780143 BC For-Sale Unstable AMY2 43 30 CN1CC[C@@H](NC[C@@](C)(O)c2ccccc2)C1=O ZINC000217780143 BC For-Sale Unstable CYP2J2 49 37 CCOC(=O)N1CCC(NC(=O)N/C=C/c2ccccc2F)CC1 ZINC000217780151 EF For-Sale Unstable CCR8 32 41 CCN(C1CC1)S(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217780174 CD For-Sale Unstable CACNA1B 23 42 COc1cc([C@@H](C)N)c(O)cc1Br ZINC000217780176 BE For-Sale Unstable P2RX2 15 40 COC(=O)c1ccc(CNC(=O)[C@H](C)N[C@@H](C)c2ccc(OC)c(Br)c2)cc1 ZINC000217780199 IH On-Demand Unstable TRPV1 24 44 CC(C)(C)c1ccc(NC(=O)NC[C@@H]2CCCN2c2nccs2)cc1 ZINC000217780205 FI For-Sale Unstable EPHX2 23 44 CC(C)(C)c1ccc(NC(=O)NC[C@@H]2CCCN2c2nccs2)cc1 ZINC000217780205 FI For-Sale Unstable DOT1L 53 35 O=C(N[C@@H]1CCN(C2CC2)C1)N[C@H](CCO)C(=O)O ZINC000217780219 CB For-Sale Unstable NAALAD2 47 38 CN1CC[C@H](NC[C@@](C)(O)c2ccccc2)C1=O ZINC000217780234 BC For-Sale Unstable AMY2 43 30 CN1CC[C@H](NC[C@@](C)(O)c2ccccc2)C1=O ZINC000217780234 BC For-Sale Unstable CYP2J2 49 37 O=C(N/C=C/c1ccccc1F)N1CCN(c2cccc(Cl)c2)CC1 ZINC000217780264 FH For-Sale Unstable HTR1A 16 42 CS(=O)(=O)CCN1CCN(c2ncnc3[nH]ccc23)C[C@@H](O)C1 ZINC000217780282 EB In-Stock Unstable AKT2 46 43 CS(=O)(=O)CCN1CCN(c2ncnc3[nH]ccc23)C[C@@H](O)C1 ZINC000217780282 EB In-Stock Unstable AKT3 37 43 CS(=O)(=O)CCN1CCN(c2ncnc3[nH]ccc23)C[C@@H](O)C1 ZINC000217780282 EB In-Stock Unstable ROCK2 43 43 CS(=O)(=O)CCN1CCN(c2ncnc3[nH]ccc23)C[C@@H](O)C1 ZINC000217780282 EB In-Stock Unstable AKT1 24 43 C[C@@H](/C=N/NC(=N)N)c1ccccc1 ZINC000217780285 AD For-Sale Unstable NPFFR2 17 44 C[C@@H](/C=N/NC(=N)N)c1ccccc1 ZINC000217780285 AD For-Sale Unstable NPFFR1 16 40 COC(=O)c1ccc(CNC(=O)[C@@H](C)N[C@H](C)c2ccc(OC)c(Br)c2)cc1 ZINC000217780287 IH On-Demand Unstable TRPV1 24 44 CC(C)(C)c1ccc(NC(=O)NC[C@H]2CCCN2c2nccs2)cc1 ZINC000217780306 FI For-Sale Unstable EPHX2 23 44 CC(C)(C)c1ccc(NC(=O)NC[C@H]2CCCN2c2nccs2)cc1 ZINC000217780306 FI For-Sale Unstable DOT1L 53 35 O=C(N[C@H]1CCN(C2CC2)C1)N[C@H](CCO)C(=O)O ZINC000217780307 CB For-Sale Unstable NAALAD2 47 38 CN1CC[C@@H](NC[C@](C)(O)c2ccccc2)C1=O ZINC000217780322 BC For-Sale Unstable AMY2 43 30 CN1CC[C@@H](NC[C@](C)(O)c2ccccc2)C1=O ZINC000217780322 BC For-Sale Unstable CYP2J2 49 37 Cc1ccc(CC(=O)NCc2ccco2)c(N)c1 ZINC000217780326 BE In-Stock Unstable P2RX7 16 41 Nc1c(Cl)cc(Cl)cc1C(=O)NCC1CC1 ZINC000217780348 CF For-Sale Unstable HTR4 46 48 Nc1c(Cl)cc(Cl)cc1C(=O)NCC1CC1 ZINC000217780348 CF For-Sale Unstable CACNA1I 74 46 C[C@H](/C=N/NC(=N)N)c1ccccc1 ZINC000217780368 AD For-Sale Unstable NPFFR2 17 44 C[C@H](/C=N/NC(=N)N)c1ccccc1 ZINC000217780368 AD For-Sale Unstable NPFFR1 16 40 COC(=O)c1ccc(CNC(=O)[C@H](C)N[C@H](C)c2ccc(OC)c(Br)c2)cc1 ZINC000217780372 IH On-Demand Unstable TRPV1 24 44 Cc1ccc2nc(-c3ccc(NC(=O)N/C=C/c4ccccc4F)cc3)sc2c1 ZINC000217780384 HK For-Sale Unstable APP 25 51 CN1CC[C@H](NC[C@](C)(O)c2ccccc2)C1=O ZINC000217780408 BC For-Sale Unstable AMY2 43 30 CN1CC[C@H](NC[C@](C)(O)c2ccccc2)C1=O ZINC000217780408 BC For-Sale Unstable CYP2J2 49 37 O=C(NCCc1ccccc1)NC[C@@H]1CCCN1c1nccs1 ZINC000217780411 EF For-Sale Unstable PREP 47 40 O=C(NCCc1ccccc1)NC[C@@H]1CCCN1c1nccs1 ZINC000217780411 EF For-Sale Unstable GPBAR1 19 40 O=C(NCCc1ccccc1)NC[C@H]1CCCN1c1nccs1 ZINC000217780493 EF For-Sale Unstable PREP 47 40 O=C(NCCc1ccccc1)NC[C@H]1CCCN1c1nccs1 ZINC000217780493 EF For-Sale Unstable GPBAR1 19 40 O=C(N/C=C/c1ccccc1F)Nc1ccc2c(c1)OCO2 ZINC000217780511 DG For-Sale Unstable CCR2 0 42 COc1ccc2[nH]c(C(=O)NC[C@@H]3CCCN4CCCC[C@H]34)c(C)c2c1 ZINC000217780534 FG In-Stock Unstable MAPKAPK2 22 45 COc1ccc2[nH]c(C(=O)NC[C@@H]3CCCN4CCCC[C@H]34)c(C)c2c1 ZINC000217780534 FG In-Stock Unstable MTNR1A 40 42 COc1ccc2[nH]c(C(=O)NC[C@@H]3CCCN4CCCC[C@H]34)c(C)c2c1 ZINC000217780534 FG In-Stock Unstable MTNR1B 39 42 O=C1Nc2cc(I)ccc2/C1=C(\O)c1ccccc1 ZINC000217780550 FH For-Sale Anodyne FGFR1 29 41 O=C1Nc2cc(I)ccc2/C1=C(\O)c1ccccc1 ZINC000217780550 FH For-Sale Anodyne FLT1 32 41 O=C1Nc2cc(I)ccc2/C1=C(\O)c1ccccc1 ZINC000217780550 FH For-Sale Anodyne PDGFRA 50 38 O=C1Nc2cc(I)ccc2/C1=C(\O)c1ccccc1 ZINC000217780550 FH For-Sale Anodyne TGFBR1 36 40 Cc1ccc(CC(=O)Nc2nccs2)c(N)c1 ZINC000217780562 BE In-Stock Unstable MAP 0 46 Cc1ccc(CC(=O)Nc2nccs2)c(N)c1 ZINC000217780562 BE In-Stock Unstable MAP1 127 45 Cc1ccc(CC(=O)Nc2nccs2)c(N)c1 ZINC000217780562 BE In-Stock Unstable MAPK8 22 42 Cc1ccc(CC(=O)Nc2nccs2)c(N)c1 ZINC000217780562 BE In-Stock Unstable GLS 0 40 C[C@@H](CO)S(=O)(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217780648 CE For-Sale Unstable GRIN1 44 39 Cc1ccc(CC(=O)NCC2CC2)c(N)c1 ZINC000217780664 BD In-Stock Unstable CACNA1I 44 38 O=C(c1ccncc1)N1CC[C@H](N2C(=O)CSC2=O)C1 ZINC000217780671 CC In-Stock Unstable L3MBTL1 0 45 O=C(c1ccncc1)N1CC[C@H](N2C(=O)CSC2=O)C1 ZINC000217780671 CC In-Stock Unstable L3MBTL3 68 45 C[C@H](CO)S(=O)(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217780722 CE For-Sale Unstable GRIN1 44 39 COC1CCN(C2CCN(C(=O)c3cccc4ccccc34)CC2)CC1 ZINC000217780732 FH In-Stock Unstable CHRM2 71 62 COC1CCN(C2CCN(C(=O)c3cccc4ccccc34)CC2)CC1 ZINC000217780732 FH In-Stock Unstable HRH1 18 48 COC1CCN(C2CCN(C(=O)c3cccc4ccccc34)CC2)CC1 ZINC000217780732 FH In-Stock Unstable ACACA 31 42 COC1CCN(C2CCN(C(=O)c3cccc4ccccc34)CC2)CC1 ZINC000217780732 FH In-Stock Unstable CCR3 35 44 COC1CCN(C2CCN(C(=O)c3cccc4ccccc34)CC2)CC1 ZINC000217780732 FH In-Stock Unstable L3MBTL3 79 54 O=C(N/C=C/c1ccccc1F)Nc1cccc(F)c1 ZINC000217780750 CH For-Sale Anodyne KCNK3 60 46 O=C(N/C=C/c1ccccc1F)Nc1cccc(F)c1 ZINC000217780750 CH For-Sale Anodyne KCNK9 27 40 C[C@H]1CO[C@H](C)CN1Cc1cccc(O)c1 ZINC000217780761 BE On-Demand Unstable OPRD1 20 41 C[C@H]1CO[C@H](C)CN1Cc1cccc(O)c1 ZINC000217780761 BE On-Demand Unstable OPRK1 20 41 Brc1ncc(CN2CCNCC2)o1 ZINC000217780768 BC For-Sale Unstable CXCR4 21 41 O=C(c1ccncc1)N1CC[C@@H](N2C(=O)CSC2=O)C1 ZINC000217780780 CC In-Stock Unstable L3MBTL1 0 45 O=C(c1ccncc1)N1CC[C@@H](N2C(=O)CSC2=O)C1 ZINC000217780780 CC In-Stock Unstable L3MBTL3 68 45 CN(C)Cc1ccc(N/C(=C2\C(=O)Nc3cc(I)ccc32)c2ccccc2)cc1 ZINC000217780846 JK For-Sale Unstable FGFR1 18 75 CN(C)Cc1ccc(N/C(=C2\C(=O)Nc3cc(I)ccc32)c2ccccc2)cc1 ZINC000217780846 JK For-Sale Unstable FLT1 19 75 CN(C)Cc1ccc(N/C(=C2\C(=O)Nc3cc(I)ccc32)c2ccccc2)cc1 ZINC000217780846 JK For-Sale Unstable PRKAA1 25 47 CN(C)Cc1ccc(N/C(=C2\C(=O)Nc3cc(I)ccc32)c2ccccc2)cc1 ZINC000217780846 JK For-Sale Unstable FLT4 36 75 CN(C)Cc1ccc(N/C(=C2\C(=O)Nc3cc(I)ccc32)c2ccccc2)cc1 ZINC000217780846 JK For-Sale Unstable PDGFRA 84 75 CN(C)Cc1ccc(N/C(=C2\C(=O)Nc3cc(I)ccc32)c2ccccc2)cc1 ZINC000217780846 JK For-Sale Unstable TGFBR1 61 72 CN(C)Cc1ccc(N/C(=C2\C(=O)Nc3cc(I)ccc32)c2ccccc2)cc1 ZINC000217780846 JK For-Sale Unstable CAMK1G 15 47 CN(C)Cc1ccc(N/C(=C2\C(=O)Nc3cc(I)ccc32)c2ccccc2)cc1 ZINC000217780846 JK For-Sale Unstable SRPK3 15 47 CN(C)Cc1ccc(N/C(=C2\C(=O)Nc3cc(I)ccc32)c2ccccc2)cc1 ZINC000217780846 JK For-Sale Unstable RIOK3 15 47 CN(C)Cc1ccc(N/C(=C2\C(=O)Nc3cc(I)ccc32)c2ccccc2)cc1 ZINC000217780846 JK For-Sale Unstable MAP3K7 15 47 CN(C)Cc1ccc(N/C(=C2\C(=O)Nc3cc(I)ccc32)c2ccccc2)cc1 ZINC000217780846 JK For-Sale Unstable PIP5K1A 15 47 CN(C)Cc1ccc(N/C(=C2\C(=O)Nc3cc(I)ccc32)c2ccccc2)cc1 ZINC000217780846 JK For-Sale Unstable RIOK1 15 47 CN(C)Cc1ccc(N/C(=C2\C(=O)Nc3cc(I)ccc32)c2ccccc2)cc1 ZINC000217780846 JK For-Sale Unstable LTK 17 47 CN(C)Cc1ccc(N/C(=C2\C(=O)Nc3cc(I)ccc32)c2ccccc2)cc1 ZINC000217780846 JK For-Sale Unstable PIP4K2B 15 47 CN(C)Cc1ccc(N/C(=C2\C(=O)Nc3cc(I)ccc32)c2ccccc2)cc1 ZINC000217780846 JK For-Sale Unstable GRK4 15 47 C[C@H]1CN(Cc2cccc(O)c2)[C@@H](C)CO1 ZINC000217780847 BE On-Demand Unstable OPRD1 20 41 C[C@H]1CN(Cc2cccc(O)c2)[C@@H](C)CO1 ZINC000217780847 BE On-Demand Unstable OPRK1 20 41 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc3c(c2)OCO3)CC(=O)O4)cc1O ZINC000217780849 JI In-Stock Unstable AKR1B1 0 46 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc3c(c2)OCO3)CC(=O)O4)cc1O ZINC000217780849 JI In-Stock Unstable CYP1B1 48 34 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc3c(c2)OCO3)CC(=O)O4)cc1O ZINC000217780849 JI In-Stock Unstable CYP1A1 37 46 Brc1nc(CN2CCNCC2)co1 ZINC000217780883 BC For-Sale Unstable CXCR4 20 40 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc3c(c2)OCO3)CC(=O)O4)cc1O ZINC000217780938 JI In-Stock Unstable AKR1B1 0 46 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc3c(c2)OCO3)CC(=O)O4)cc1O ZINC000217780938 JI In-Stock Unstable CYP1B1 48 34 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc3c(c2)OCO3)CC(=O)O4)cc1O ZINC000217780938 JI In-Stock Unstable CYP1A1 37 46 CCCCOc1ccc(NC(=O)NC[C@@H]2CCCN2c2nccs2)cc1 ZINC000217780993 FI For-Sale Unstable ADRB1 16 40 CCCCOc1ccc(NC(=O)NC[C@@H]2CCCN2c2nccs2)cc1 ZINC000217780993 FI For-Sale Unstable EPHX2 32 42 CC(=O)NCc1ccc([N+]#N)cc1 ZINC000217781029 AD For-Sale Unstable TPSAB1 19 43 Cc1c(CC(=O)N[C@H](CO)c2ccccc2)c(=O)oc2cc(O)ccc12 ZINC000217781066 FE In-Stock Unstable HSD17B3 49 57 Cc1c(CC(=O)N[C@H](CO)c2ccccc2)c(=O)oc2cc(O)ccc12 ZINC000217781066 FE In-Stock Unstable NQO1 64 35 Cc1c(CC(=O)N[C@H](CO)c2ccccc2)c(=O)oc2cc(O)ccc12 ZINC000217781066 FE In-Stock Unstable GPR55 40 30 Cc1c(CC(=O)N[C@H](CO)c2ccccc2)c(=O)oc2cc(O)ccc12 ZINC000217781066 FE In-Stock Unstable Q81JI8_BACAN 0 41 CCCCOc1ccc(NC(=O)NC[C@H]2CCCN2c2nccs2)cc1 ZINC000217781086 FI For-Sale Unstable ADRB1 16 40 CCCCOc1ccc(NC(=O)NC[C@H]2CCCN2c2nccs2)cc1 ZINC000217781086 FI For-Sale Unstable EPHX2 32 42 O=C(COc1ccccc1)N1CC[C@H](N2C(=O)CSC2=O)C1 ZINC000217781096 DD In-Stock Unstable CPT1A 112 38 O=C(COc1ccccc1)N1CC[C@H](N2C(=O)CSC2=O)C1 ZINC000217781096 DD In-Stock Unstable CPT2 47 38 O=C(Cn1c(=O)oc2ccccc21)NCCc1noc(C2CCC2)n1 ZINC000217781139 ED In-Stock Unstable SMO 47 37 O=C(COc1ccccc1)N1CC[C@@H](N2C(=O)CSC2=O)C1 ZINC000217781173 DD In-Stock Unstable CPT1A 112 38 O=C(COc1ccccc1)N1CC[C@@H](N2C(=O)CSC2=O)C1 ZINC000217781173 DD In-Stock Unstable CPT2 47 38 C[C@@H](c1ccc(Cl)cc1)N(C)C[C@@H](O)c1cccc(N)c1 ZINC000217781181 DH For-Sale Unstable AOC3 35 50 O=C(NC[C@@H]1CCCN1c1nccs1)Nc1cccc(Cl)c1 ZINC000217781194 EH For-Sale Unstable ADAM17 19 41 O=C(NC[C@@H]1CCCN1c1nccs1)Nc1cccc(Cl)c1 ZINC000217781194 EH For-Sale Unstable GRM5 16 50 O=C(NC[C@@H]1CCCN1c1nccs1)Nc1cccc(Cl)c1 ZINC000217781194 EH For-Sale Unstable EPHX2 21 53 O=C(N/C=C/c1ccccc1F)NCCc1c[nH]c2ccccc12 ZINC000217781205 DH For-Sale Unstable CCKAR 32 42 O=C(N/C=C/c1ccccc1F)NCCc1c[nH]c2ccccc12 ZINC000217781205 DH For-Sale Unstable BCHE 15 40 O=C(N/C=C/c1ccccc1F)NCCc1c[nH]c2ccccc12 ZINC000217781205 DH For-Sale Unstable MPO 81 37 O=C(N/C=C/c1ccccc1F)NCCc1c[nH]c2ccccc12 ZINC000217781205 DH For-Sale Unstable BRS3 26 42 O=C(N/C=C/c1ccccc1F)NCCc1c[nH]c2ccccc12 ZINC000217781205 DH For-Sale Unstable NMBR 26 44 Cc1ccc(CC(=O)NCC(C)C)c(N)c1 ZINC000217781240 BD In-Stock Unstable F3 53 32 Cc1ccc(CC(=O)NCC(C)C)c(N)c1 ZINC000217781240 BD In-Stock Unstable CCR2 21 41 C[C@@H](N[C@@H]1CCN(C)C1=O)C(=O)NC1CCCCC1 ZINC000217781242 CC For-Sale Unstable EPHX2 21 44 C[C@@H](N[C@@H]1CCN(C)C1=O)C(=O)NC1CCCCC1 ZINC000217781242 CC For-Sale Unstable BIRC2 73 37 COc1cccc(C(=O)N2CC[C@H](N3C(=O)CSC3=O)C2)c1 ZINC000217781262 DD In-Stock Unstable DRD4 44 34 COc1cccc(C(=O)N2CC[C@H](N3C(=O)CSC3=O)C2)c1 ZINC000217781262 DD In-Stock Unstable AVPR1A 22 42 COc1cccc(C(=O)N2CC[C@H](N3C(=O)CSC3=O)C2)c1 ZINC000217781262 DD In-Stock Unstable SLC18A3 20 40 COc1cccc(C(=O)N2CC[C@H](N3C(=O)CSC3=O)C2)c1 ZINC000217781262 DD In-Stock Unstable L3MBTL3 41 35 CCCN(C)S(=O)(=O)c1ccc(/C=C\C(=O)O)cc1Cl ZINC000217781263 DE For-Sale Unstable NR0B2 0 42 O=C1CC[C@H](C(=O)NCCCCCCO)N1 ZINC000217781269 BB For-Sale Unstable MME 30 49 C[C@H](c1ccc(Cl)cc1)N(C)C[C@@H](O)c1cccc(N)c1 ZINC000217781270 DH For-Sale Unstable AOC3 35 50 O=C(NC[C@H]1CCCN1c1nccs1)Nc1cccc(Cl)c1 ZINC000217781283 EH For-Sale Unstable ADAM17 19 41 O=C(NC[C@H]1CCCN1c1nccs1)Nc1cccc(Cl)c1 ZINC000217781283 EH For-Sale Unstable GRM5 16 50 O=C(NC[C@H]1CCCN1c1nccs1)Nc1cccc(Cl)c1 ZINC000217781283 EH For-Sale Unstable EPHX2 21 53 CC(C)C[C@H](NC(=O)COc1cc(O)c2c(c1)OC(C)(C)CC2=O)c1nc2ccccc2[nH]1 ZINC000217781291 JI In-Stock Unstable MMP7 20 44 NC(=O)C1CCN(C(=O)N/C=C/c2ccccc2F)CC1 ZINC000217781318 CD For-Sale Unstable CCR2 0 40 C[C@H](N[C@@H]1CCN(C)C1=O)C(=O)NC1CCCCC1 ZINC000217781327 CC For-Sale Unstable EPHX2 21 44 C[C@H](N[C@@H]1CCN(C)C1=O)C(=O)NC1CCCCC1 ZINC000217781327 CC For-Sale Unstable BIRC2 73 37 C[C@@H](c1ccc(Cl)cc1)N(C)C[C@@H](O)c1ccccc1N ZINC000217781353 DH For-Sale Unstable AOC3 26 47 COc1cccc(C(=O)N2CC[C@@H](N3C(=O)CSC3=O)C2)c1 ZINC000217781361 DD In-Stock Unstable DRD4 44 34 COc1cccc(C(=O)N2CC[C@@H](N3C(=O)CSC3=O)C2)c1 ZINC000217781361 DD In-Stock Unstable AVPR1A 22 42 COc1cccc(C(=O)N2CC[C@@H](N3C(=O)CSC3=O)C2)c1 ZINC000217781361 DD In-Stock Unstable SLC18A3 20 40 COc1cccc(C(=O)N2CC[C@@H](N3C(=O)CSC3=O)C2)c1 ZINC000217781361 DD In-Stock Unstable L3MBTL3 41 35 CCOC[C@@H](C)NC(=O)N[C@@H](C(=O)O)[C@@H](C)CC ZINC000217781376 CD For-Sale Unstable ENPEP 52 37 O=C(NCc1ccc(Cl)cc1)NC[C@@H]1CCCN1c1nccs1 ZINC000217781395 FG For-Sale Unstable NOS2 18 42 C[C@@H](N[C@H]1CCN(C)C1=O)C(=O)NC1CCCCC1 ZINC000217781413 CC For-Sale Unstable EPHX2 21 44 C[C@@H](N[C@H]1CCN(C)C1=O)C(=O)NC1CCCCC1 ZINC000217781413 CC For-Sale Unstable BIRC2 73 37 C[C@H](c1ccc(Cl)cc1)N(C)C[C@@H](O)c1ccccc1N ZINC000217781451 DH For-Sale Unstable AOC3 26 47 O=C(c1ccc(Cl)cc1)N1CC[C@H](N2C(=O)CSC2=O)C1 ZINC000217781478 DE In-Stock Unstable L3MBTL1 0 47 O=C(c1ccc(Cl)cc1)N1CC[C@H](N2C(=O)CSC2=O)C1 ZINC000217781478 DE In-Stock Unstable L3MBTL3 73 47 O=C(c1ccc(Cl)cc1)N1CC[C@H](N2C(=O)CSC2=O)C1 ZINC000217781478 DE In-Stock Unstable MBTD1 0 41 O=C(NCc1ccc(Cl)cc1)NC[C@H]1CCCN1c1nccs1 ZINC000217781481 FG For-Sale Unstable NOS2 18 42 C[C@H](N[C@H]1CCN(C)C1=O)C(=O)NC1CCCCC1 ZINC000217781496 CC For-Sale Unstable EPHX2 21 44 C[C@H](N[C@H]1CCN(C)C1=O)C(=O)NC1CCCCC1 ZINC000217781496 CC For-Sale Unstable BIRC2 73 37 COc1cc(C(=O)N[C@@H]2COCC[C@H]2OC)c2ccccc2n1 ZINC000217781511 DD In-Stock Unstable ADAM17 23 40 C[C@@H](c1ccc(Cl)cc1)N(C)C[C@@H](O)c1ccc(N)cc1 ZINC000217781535 DH For-Sale Unstable AOC3 23 59 O=C(c1ccc(Cl)cc1)N1CC[C@@H](N2C(=O)CSC2=O)C1 ZINC000217781555 DE In-Stock Unstable L3MBTL1 0 47 O=C(c1ccc(Cl)cc1)N1CC[C@@H](N2C(=O)CSC2=O)C1 ZINC000217781555 DE In-Stock Unstable L3MBTL3 73 47 O=C(c1ccc(Cl)cc1)N1CC[C@@H](N2C(=O)CSC2=O)C1 ZINC000217781555 DE In-Stock Unstable MBTD1 0 41 CC(C)c1ccc(CNC(=O)OC(C)(C)C)cn1 ZINC000217781579 CG In-Stock Unstable PAPA1_CARPA 40 36 O=C(NC[C@@H]1CCCN1c1nccs1)NC(c1ccccc1)c1ccccc1 ZINC000217781586 GI For-Sale Unstable BIRC8 43 31 C[C@@H]1CCN(S(=O)(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217781604 CD For-Sale Unstable AKR1C3 61 38 C[C@H](c1ccc(Cl)cc1)N(C)C[C@@H](O)c1ccc(N)cc1 ZINC000217781621 DH For-Sale Unstable AOC3 23 59 O=C(NC[C@H]1CCCN1c1nccs1)NC(c1ccccc1)c1ccccc1 ZINC000217781674 GI For-Sale Unstable BIRC8 43 31 O=C(c1ccc(F)c(F)c1)N1CC[C@H](N2C(=O)CSC2=O)C1 ZINC000217781675 ED In-Stock Unstable L3MBTL1 0 42 O=C(c1ccc(F)c(F)c1)N1CC[C@H](N2C(=O)CSC2=O)C1 ZINC000217781675 ED In-Stock Unstable L3MBTL3 65 42 C[C@H]1CCN(S(=O)(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217781686 CD For-Sale Unstable AKR1C3 61 38 COC1CCN(C2CCN(C(=O)c3ccc(-c4ccccc4)cc3)CC2)CC1 ZINC000217781732 GI In-Stock Unstable CHRM2 64 45 COC1CCN(C2CCN(C(=O)c3ccc(-c4ccccc4)cc3)CC2)CC1 ZINC000217781732 GI In-Stock Unstable OXTR 18 41 COC1CCN(C2CCN(C(=O)c3ccc(-c4ccccc4)cc3)CC2)CC1 ZINC000217781732 GI In-Stock Unstable HRH1 21 45 COC1CCN(C2CCN(C(=O)c3ccc(-c4ccccc4)cc3)CC2)CC1 ZINC000217781732 GI In-Stock Unstable AVPR1A 32 43 COC1CCN(C2CCN(C(=O)c3ccc(-c4ccccc4)cc3)CC2)CC1 ZINC000217781732 GI In-Stock Unstable INHA 16 41 COC1CCN(C2CCN(C(=O)c3ccc(-c4ccccc4)cc3)CC2)CC1 ZINC000217781732 GI In-Stock Unstable HTR2B 16 48 COC1CCN(C2CCN(C(=O)c3ccc(-c4ccccc4)cc3)CC2)CC1 ZINC000217781732 GI In-Stock Unstable HRH3 37 41 COC1CCN(C2CCN(C(=O)c3ccc(-c4ccccc4)cc3)CC2)CC1 ZINC000217781732 GI In-Stock Unstable HSD11B1 18 51 COC1CCN(C2CCN(C(=O)c3ccc(-c4ccccc4)cc3)CC2)CC1 ZINC000217781732 GI In-Stock Unstable CCR3 49 47 COC1CCN(C2CCN(C(=O)c3ccc(-c4ccccc4)cc3)CC2)CC1 ZINC000217781732 GI In-Stock Unstable ACACB 20 40 COC1CCN(C2CCN(C(=O)c3ccc(-c4ccccc4)cc3)CC2)CC1 ZINC000217781732 GI In-Stock Unstable SLC18A3 24 43 COC1CCN(C2CCN(C(=O)c3ccc(-c4ccccc4)cc3)CC2)CC1 ZINC000217781732 GI In-Stock Unstable L3MBTL3 123 56 O=C(c1ccc(F)c(F)c1)N1CC[C@@H](N2C(=O)CSC2=O)C1 ZINC000217781768 ED In-Stock Unstable L3MBTL1 0 42 O=C(c1ccc(F)c(F)c1)N1CC[C@@H](N2C(=O)CSC2=O)C1 ZINC000217781768 ED In-Stock Unstable L3MBTL3 65 42 Cc1cc(S(=O)(=O)N2CC[C@H](C)C2)ccc1/C=C\C(=O)O ZINC000217781780 DE For-Sale Unstable AKR1C3 43 38 CCCCOC(=O)Cc1cc(C)ccc1N ZINC000217781802 BE In-Stock Unstable PLA2G4B 50 33 COC1CCN(C2CCN(C(=O)c3ccc4ccccc4c3)CC2)CC1 ZINC000217781850 FH In-Stock Unstable CHRM2 67 44 COC1CCN(C2CCN(C(=O)c3ccc4ccccc4c3)CC2)CC1 ZINC000217781850 FH In-Stock Unstable OXTR 31 40 COC1CCN(C2CCN(C(=O)c3ccc4ccccc4c3)CC2)CC1 ZINC000217781850 FH In-Stock Unstable HRH1 19 47 COC1CCN(C2CCN(C(=O)c3ccc4ccccc4c3)CC2)CC1 ZINC000217781850 FH In-Stock Unstable AVPR1A 26 45 COC1CCN(C2CCN(C(=O)c3ccc4ccccc4c3)CC2)CC1 ZINC000217781850 FH In-Stock Unstable PRSS2 44 31 COC1CCN(C2CCN(C(=O)c3ccc4ccccc4c3)CC2)CC1 ZINC000217781850 FH In-Stock Unstable HRH3 44 45 COC1CCN(C2CCN(C(=O)c3ccc4ccccc4c3)CC2)CC1 ZINC000217781850 FH In-Stock Unstable HSD11B1 15 45 COC1CCN(C2CCN(C(=O)c3ccc4ccccc4c3)CC2)CC1 ZINC000217781850 FH In-Stock Unstable CCR3 51 51 COC1CCN(C2CCN(C(=O)c3ccc4ccccc4c3)CC2)CC1 ZINC000217781850 FH In-Stock Unstable SLC18A3 19 42 COC1CCN(C2CCN(C(=O)c3ccc4ccccc4c3)CC2)CC1 ZINC000217781850 FH In-Stock Unstable AKR1C3 24 42 COC1CCN(C2CCN(C(=O)c3ccc4ccccc4c3)CC2)CC1 ZINC000217781850 FH In-Stock Unstable L3MBTL3 101 64 CCCc1ccc(C(=O)N2CC[C@H](N3C(=O)CSC3=O)C2)cc1 ZINC000217781871 EF In-Stock Unstable AVPR1A 24 54 CCCc1ccc(C(=O)N2CC[C@H](N3C(=O)CSC3=O)C2)cc1 ZINC000217781871 EF In-Stock Unstable L3MBTL1 0 43 CCCc1ccc(C(=O)N2CC[C@H](N3C(=O)CSC3=O)C2)cc1 ZINC000217781871 EF In-Stock Unstable L3MBTL3 67 43 O=C(O)[C@@H]1[C@H]2CN(C(=O)c3c(O)ccc4ccccc34)C[C@H]21 ZINC000217781922 CD In-Stock Unstable CYP73A1 0 53 CCCc1ccc(C(=O)N2CC[C@@H](N3C(=O)CSC3=O)C2)cc1 ZINC000217781952 EF In-Stock Unstable AVPR1A 24 54 CCCc1ccc(C(=O)N2CC[C@@H](N3C(=O)CSC3=O)C2)cc1 ZINC000217781952 EF In-Stock Unstable L3MBTL1 0 43 CCCc1ccc(C(=O)N2CC[C@@H](N3C(=O)CSC3=O)C2)cc1 ZINC000217781952 EF In-Stock Unstable L3MBTL3 67 43 O=C(NC[C@H]1CCCN1c1nccs1)NC12CC3CC(CC(C3)C1)C2 ZINC000217781987 FG For-Sale Unstable EPHX2 102 50 COc1ccc(CN2C(=O)N[C@@H](CC(=O)NCc3ccncc3)C2=O)cc1 ZINC000217782027 FD In-Stock Unstable PROKR1 59 36 O=C(O)/C=C\c1cccc(S(=O)(=O)NC2CCOCC2)c1 ZINC000217782043 DD For-Sale Unstable SFRP1 121 39 O=C(O)/C=C\c1cccc(S(=O)(=O)NC2CCOCC2)c1 ZINC000217782043 DD For-Sale Unstable WNT3 79 39 O=C(c1ccc(F)cc1Cl)N1CC[C@H](N2C(=O)CSC2=O)C1 ZINC000217782052 EE In-Stock Unstable P2RX7 27 48 O=C(NC[C@@H]1CCCN1c1nccs1)NC12CC3CC(CC(C3)C1)C2 ZINC000217782088 FG For-Sale Unstable EPHX2 102 50 Cc1cccc(N2CCN(C(=O)N/C=C/c3ccccc3F)CC2)c1C ZINC000217782111 FH For-Sale Unstable HTR2A 15 43 Cc1cccc(N2CCN(C(=O)N/C=C/c3ccccc3F)CC2)c1C ZINC000217782111 FH For-Sale Unstable HTR2C 19 43 O=C(c1ccc(F)cc1Cl)N1CC[C@@H](N2C(=O)CSC2=O)C1 ZINC000217782138 EE In-Stock Unstable P2RX7 27 48 COc1cc2c(cc1OC)CN(C(=O)c1cnc3cc(Cl)ccc3c1O)CC2 ZINC000217782140 GH In-Stock Unstable ABCB1B 59 35 COc1cc2c(cc1OC)CN(C(=O)c1cnc3cc(Cl)ccc3c1O)CC2 ZINC000217782140 GH In-Stock Unstable ABCB1 17 43 COc1cc2c(cc1OC)CN(C(=O)c1cnc3cc(Cl)ccc3c1O)CC2 ZINC000217782140 GH In-Stock Unstable CSF1R 39 40 CC(C)(C)OC(=O)NCc1ccc(-c2ccccc2)nc1 ZINC000217782206 CH In-Stock Unstable CYP11B1 16 44 CC(C)(C)OC(=O)NCc1ccc(-c2ccccc2)nc1 ZINC000217782206 CH In-Stock Unstable PPARA 19 42 CC(C)(C)OC(=O)NCc1ccc(-c2ccccc2)nc1 ZINC000217782206 CH In-Stock Unstable ACACA 0 41 CC(C)(C)OC(=O)NCc1ccc(-c2ccccc2)nc1 ZINC000217782206 CH In-Stock Unstable PAPA1_CARPA 59 44 CC(C)(C)OC(=O)NCc1ccc(-c2ccccc2)nc1 ZINC000217782206 CH In-Stock Unstable CCKAR 34 40 CC(C)(C)OC(=O)NCc1ccc(-c2ccccc2)nc1 ZINC000217782206 CH In-Stock Unstable CTSK 21 43 CC(C)(C)OC(=O)NCc1ccc(-c2ccccc2)nc1 ZINC000217782206 CH In-Stock Unstable CTSL 20 47 CC(C)(C)OC(=O)NCc1ccc(-c2ccccc2)nc1 ZINC000217782206 CH In-Stock Unstable ACACB 27 47 CC(C)(C)OC(=O)NCc1ccc(-c2ccccc2)nc1 ZINC000217782206 CH In-Stock Unstable CYP11B2 0 44 CC(C)(C)OC(=O)NCc1ccc(-c2ccccc2)nc1 ZINC000217782206 CH In-Stock Unstable TPH1 66 45 CC(C)(C)OC(=O)NCc1ccc(-c2ccccc2)nc1 ZINC000217782206 CH In-Stock Unstable TACR3 41 44 CC(C)(C)OC(=O)NCc1ccc(-c2ccccc2)nc1 ZINC000217782206 CH In-Stock Unstable HDAC1 23 43 CC(C)(C)OC(=O)NCc1ccc(-c2ccccc2)nc1 ZINC000217782206 CH In-Stock Unstable REN 51 40 CC(C)(C)OC(=O)NCc1ccc(-c2ccccc2)nc1 ZINC000217782206 CH In-Stock Unstable CCKBR 22 40 CC(C)(C)OC(=O)NCc1ccc(-c2ccccc2)nc1 ZINC000217782206 CH In-Stock Unstable CTSS 17 47 CC(C)(C)OC(=O)NCc1ccc(-c2ccccc2)nc1 ZINC000217782206 CH In-Stock Unstable FPR1 49 39 CC(C)(C)OC(=O)NCc1ccc(-c2ccccc2)nc1 ZINC000217782206 CH In-Stock Unstable PDS 69 40 CC(C)(C)OC(=O)NCc1ccc(-c2ccccc2)nc1 ZINC000217782206 CH In-Stock Unstable CES1D 54 35 O=C(N/C=C/c1ccccc1F)N1CCN(c2ccccc2)CC1 ZINC000217782217 EG For-Sale Unstable AKR1C3 0 43 COc1ccc(CCC(=O)N2CC[C@H](N3C(=O)CSC3=O)C2)cc1 ZINC000217782251 ED In-Stock Unstable KCNA5 16 43 COc1cc(N2CCN(C(=O)OC(C)(C)C)CC2)ccc1Nc1nc(Br)cc2cn[nH]c(=O)c12 ZINC000217782292 KH For-Sale Unstable IGF1R 42 41 COc1cc(N2CCN(C(=O)OC(C)(C)C)CC2)ccc1Nc1nc(Br)cc2cn[nH]c(=O)c12 ZINC000217782292 KH For-Sale Unstable TTK 37 40 COc1cc(N2CCN(C(=O)OC(C)(C)C)CC2)ccc1Nc1nc(Br)cc2cn[nH]c(=O)c12 ZINC000217782292 KH For-Sale Unstable MAPK7 46 37 CC(C)(C)OC(=O)NC[C@@H]1CC[C@H](c2ccccc2)NC1 ZINC000217782323 CG In-Stock Unstable PAPA1_CARPA 40 37 CC(C)(C)OC(=O)NC[C@@H]1CC[C@H](c2ccccc2)NC1 ZINC000217782323 CG In-Stock Unstable ACACB 29 48 CC(C)(C)OC(=O)NC[C@@H]1CC[C@H](c2ccccc2)NC1 ZINC000217782323 CG In-Stock Unstable VCP 55 34 COc1ccc(CCC(=O)N2CC[C@@H](N3C(=O)CSC3=O)C2)cc1 ZINC000217782337 ED In-Stock Unstable KCNA5 16 43 O=C(/C=C\c1cccc(Br)c1)NCC1(O)CCCCCC1 ZINC000217782357 FH For-Sale Unstable HDAC8 50 39 CC(C)(C)OC(=O)NC[C@H]1CC[C@H](c2ccccc2)NC1 ZINC000217782393 CG In-Stock Unstable PAPA1_CARPA 40 37 CC(C)(C)OC(=O)NC[C@H]1CC[C@H](c2ccccc2)NC1 ZINC000217782393 CG In-Stock Unstable ACACB 29 48 CC(C)(C)OC(=O)NC[C@H]1CC[C@H](c2ccccc2)NC1 ZINC000217782393 CG In-Stock Unstable VCP 55 34 CCOc1ccccc1NC(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217782422 EG For-Sale Unstable HCN1 45 33 CCOc1ccccc1NC(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217782422 EG For-Sale Unstable HCN4 42 33 COc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)NCCc1c[nH]c3ccccc13)C(=O)OC2 ZINC000217782475 JI In-Stock Unstable IMPDH1 0 75 COc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)NCCc1c[nH]c3ccccc13)C(=O)OC2 ZINC000217782475 JI In-Stock Unstable BCHE 16 42 COc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)NCCc1c[nH]c3ccccc13)C(=O)OC2 ZINC000217782475 JI In-Stock Unstable IMPDH2 0 75 CC(C)(C)OC(=O)NC[C@@H]1CC[C@@H](c2ccccc2)NC1 ZINC000217782488 CG In-Stock Unstable PAPA1_CARPA 40 37 CC(C)(C)OC(=O)NC[C@@H]1CC[C@@H](c2ccccc2)NC1 ZINC000217782488 CG In-Stock Unstable ACACB 29 48 CC(C)(C)OC(=O)NC[C@@H]1CC[C@@H](c2ccccc2)NC1 ZINC000217782488 CG In-Stock Unstable VCP 55 34 CCOc1ccccc1NC(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217782496 EG For-Sale Unstable HCN1 45 33 CCOc1ccccc1NC(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217782496 EG For-Sale Unstable HCN4 42 33 CC(=O)SC[C@@H](C)NC(=O)OC(C)(C)C ZINC000217782506 BE For-Sale Unstable CTSK 27 47 COc1ccc([N+](=O)[O-])cc1NC(=O)N/C=C/c1ccccc1F ZINC000217782567 EH For-Sale Unstable KCNMA1 23 53 COc1ccc([N+](=O)[O-])cc1NC(=O)N/C=C/c1ccccc1F ZINC000217782567 EH For-Sale Unstable WDR5 32 42 CC(C)(C)OC(=O)NC[C@H]1CC[C@@H](c2ccccc2)NC1 ZINC000217782569 CG In-Stock Unstable PAPA1_CARPA 40 37 CC(C)(C)OC(=O)NC[C@H]1CC[C@@H](c2ccccc2)NC1 ZINC000217782569 CG In-Stock Unstable ACACB 29 48 CC(C)(C)OC(=O)NC[C@H]1CC[C@@H](c2ccccc2)NC1 ZINC000217782569 CG In-Stock Unstable VCP 55 34 COc1cc2c(c(OC)c1OC)-c1ccc(NCCCC(=O)Nc3ccccn3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217782587 KI In-Stock Unstable TUBA1A 18 64 COc1cc2c(c(OC)c1OC)-c1ccc(NCCCC(=O)Nc3ccccn3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217782587 KI In-Stock Unstable TPPP 0 61 CC(C)(C)CNS(=O)(=O)c1ccc(/C=C\C(=O)O)cc1Cl ZINC000217782589 EF For-Sale Unstable NR0B2 0 43 COCc1cc(=O)c(O)c([C@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccc(OC)cc2OC)o1 ZINC000217782704 KI In-Stock Unstable DRD5 17 40 COCc1cc(=O)c(O)c([C@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccc(OC)cc2OC)o1 ZINC000217782704 KI In-Stock Unstable RORC 44 40 COCc1cc(=O)c(O)c([C@@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccc(OC)cc2OC)o1 ZINC000217782770 KI In-Stock Unstable DRD5 17 40 COCc1cc(=O)c(O)c([C@@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccc(OC)cc2OC)o1 ZINC000217782770 KI In-Stock Unstable RORC 44 40 N#C[C@]12CCC[C@H]1CN(Cc1ccccc1)C2 ZINC000217782816 BF For-Sale Unstable SIGMAR1 49 45 COc1ccc(NC(=O)NC[C@@H]2CCCN2c2nccs2)cc1 ZINC000217782821 EF For-Sale Unstable EPHX2 22 41 COc1ccc(NC(=O)NC[C@H]2CCCN2c2nccs2)cc1 ZINC000217782882 EF For-Sale Unstable EPHX2 22 41 N#C[C@]12CCC[C@@H]1CN(Cc1ccccc1)C2 ZINC000217782893 BF For-Sale Unstable SIGMAR1 49 45 CCN(C)C(=O)CNC(=O)[C@H]1CCCC[C@@H]1C(=O)O ZINC000217782944 CC For-Sale Unstable ACE 0 56 CN(C1CCCC1)S(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217782955 DE For-Sale Unstable HDAC8 17 42 Cc1cccc(NC(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217782958 DG For-Sale Unstable KIT 22 40 Cc1cccc(NC(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217782958 DG For-Sale Unstable CCKAR 31 41 Cc1cccc(NC(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217782958 DG For-Sale Unstable KDR 24 41 Cc1cccc(NC(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217782958 DG For-Sale Unstable CCKBR 44 39 Cc1cccc(NC(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217782958 DG For-Sale Unstable EPHX2 19 42 Cc1cccc(NC(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217782958 DG For-Sale Unstable TEK 23 40 CCN(C)C(=O)CNC(=O)[C@@H]1CCCC[C@H]1C(=O)O ZINC000217783021 CC For-Sale Unstable ACE 0 56 Cc1nc(-c2cccc(F)c2)sc1C(=O)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217783035 GI In-Stock Unstable PPARA 0 48 Cc1nc(-c2cccc(F)c2)sc1C(=O)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217783035 GI In-Stock Unstable SCD1 41 41 Cc1nc(-c2cccc(F)c2)sc1C(=O)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217783035 GI In-Stock Unstable SCD 34 41 Cc1cccc(NC(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217783039 DG For-Sale Unstable KIT 22 40 Cc1cccc(NC(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217783039 DG For-Sale Unstable CCKAR 31 41 Cc1cccc(NC(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217783039 DG For-Sale Unstable KDR 24 41 Cc1cccc(NC(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217783039 DG For-Sale Unstable CCKBR 44 39 Cc1cccc(NC(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217783039 DG For-Sale Unstable EPHX2 19 42 Cc1cccc(NC(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217783039 DG For-Sale Unstable TEK 23 40 O=C(O)[C@@]1(Cc2ccccc2)CCCS1(=O)=O ZINC000217783077 CD For-Sale Unstable SLC12A5 50 35 CCN(C)C(=O)CNC(=O)[C@H]1CCCC[C@H]1C(=O)O ZINC000217783112 CC For-Sale Unstable ACE 0 56 CC(C)C[C@H](NC(=O)CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)c1nc2ccccc2[nH]1 ZINC000217783146 IG In-Stock Unstable MMP7 20 47 CC(C)C[C@H](NC(=O)CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)c1nc2ccccc2[nH]1 ZINC000217783146 IG In-Stock Unstable AGAL_COFAR 0 45 CC(C)C[C@H](NC(=O)CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)c1nc2ccccc2[nH]1 ZINC000217783146 IG In-Stock Unstable HLCS 0 43 CC(C)C[C@H](NC(=O)CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)c1nc2ccccc2[nH]1 ZINC000217783146 IG In-Stock Unstable BIRA 0 41 Fc1ccc(SCCN2CCN(Cc3cn4ccccc4n3)CC2)cc1 ZINC000217783159 FG On-Demand Unstable DRD4 18 54 Fc1ccc(SCCN2CCN(Cc3cn4ccccc4n3)CC2)cc1 ZINC000217783159 FG On-Demand Unstable SLC6A4 21 42 Fc1ccc(SCCN2CCN(Cc3cn4ccccc4n3)CC2)cc1 ZINC000217783159 FG On-Demand Unstable SLC6A3 34 47 O=C(O)[C@]1(Cc2ccccc2)CCCS1(=O)=O ZINC000217783161 CD For-Sale Unstable SLC12A5 50 35 CC(C)(C)CNS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217783212 CE For-Sale Unstable HDAC8 26 49 CC(C)(C)CNS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217783212 CE For-Sale Unstable AKR1C3 32 44 CC(C)(C)CNS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217783212 CE For-Sale Unstable SFRP1 63 34 COc1ccc(-c2coc3ccc(OCC(N)=O)cc23)cc1OC ZINC000217783256 EF In-Stock Unstable ALDH2 75 42 COc1ccc([C@@H](C)CCN)cc1O ZINC000217783258 AD In-Stock Unstable TUBB1 41 40 COc1ccc([C@H](C)CCN)cc1O ZINC000217783332 AD In-Stock Unstable TUBB1 41 40 COc1ccccc1NC(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217783337 EF For-Sale Unstable ACKR3 61 31 COC(=O)C[C@H](c1ccc(OCCc2ccc(OC)cc2)cc1)c1c(O)cc(C)n(CC(=O)O)c1=O ZINC000217783354 JG In-Stock Unstable FFAR1 17 40 COc1ccccc1NC(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217783412 EF For-Sale Unstable ACKR3 61 31 CC(C)(C)Oc1ccc(C[C@@H](Br)C(=O)O)cc1 ZINC000217783419 DG For-Sale Unstable PPARG 26 40 CC(C)(C)Oc1ccc(C[C@@H](Br)C(=O)O)cc1 ZINC000217783419 DG For-Sale Unstable PPARA 33 40 CC(C)(C)Oc1ccc(C[C@@H](Br)C(=O)O)cc1 ZINC000217783419 DG For-Sale Unstable CPA1 44 36 CC(C)(C)Oc1ccc(C[C@@H](Br)C(=O)O)cc1 ZINC000217783419 DG For-Sale Unstable ACE2 45 34 COc1cc([C@@H](C)CCN)ccc1O ZINC000217783431 AD In-Stock Unstable FOLH1 35 43 COc1cc([C@@H](C)CCN)ccc1O ZINC000217783431 AD In-Stock Unstable TRPV1 0 45 COC(=O)C[C@@H](c1ccc(OCCc2ccc(OC)cc2)cc1)c1c(O)cc(C)n(CC(=O)O)c1=O ZINC000217783446 JG In-Stock Unstable FFAR1 17 40 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable F2 41 52 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable PLG 22 49 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable PRSS1 27 49 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable ACE 38 41 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable LHCGR 46 38 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable OPRM1 73 68 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable OPRD1 71 68 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable OPRK1 15 56 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable MME 95 42 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable ANPEP 76 39 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable NPR1 55 48 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable TACR1 26 57 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable HLA-DRB3 19 51 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable MC4R 82 64 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable FCER2 103 44 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable TACR2 20 45 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable RNPEP 34 42 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable NPY1R 19 57 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable KLK3 95 38 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable CTSB 62 53 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable PAPA1_CARPA 78 47 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable TRY1_BOVIN 57 42 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable CYSP_TRYCR 59 37 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable CCKAR 64 39 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable NTSR1 36 48 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable CTSK 16 47 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable CTSL 44 54 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable F2R 74 70 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable NPFFR2 111 57 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable C3AR1 41 45 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable HLA-A 55 39 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable TACR3 27 45 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable MC3R 109 58 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable MC5R 105 60 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable CAPNS1 65 36 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable MMP2 23 49 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable MMP3 48 50 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable HLA-DRB1 115 62 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable REN 49 42 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable REN1 57 42 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable LNPEP 18 42 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable MMP11 47 35 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable F11 32 41 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable PCSK5 46 39 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable PLAT 21 41 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable FURIN 105 49 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable CCKBR 43 51 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable GHSR 15 43 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable CAPN1 84 50 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable MMP9 26 45 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable CAPN2 103 41 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable ACE2 68 38 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable MC1R 163 64 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable F7 35 47 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable LAP3 39 42 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable C5AR1 21 44 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable ST14 60 39 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable MMP1 40 46 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable FPR1 80 44 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable NPR 48 33 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable AMP1_PLAFQ 24 45 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable GAG-PRO 42 35 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable XIAP 19 47 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable BLA1_STEMA 85 47 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable KISS1R 82 38 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable POLG_WNV 71 34 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable QRFPR 74 53 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable F2RL1 48 32 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable NPFFR1 104 51 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable WDR5 42 34 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable Q9NAW4_PLAFA 16 48 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable TMPRSS6 70 39 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable HPN 63 39 C[C@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783491 HA For-Sale Unstable H9B8T9_CAPHI 47 48 COc1cc([C@H](C)CCN)ccc1O ZINC000217783514 AD In-Stock Unstable PNLIP 0 57 COc1cc([C@H](C)CCN)ccc1O ZINC000217783514 AD In-Stock Unstable FOLH1 35 43 COc1cc([C@H](C)CCN)ccc1O ZINC000217783514 AD In-Stock Unstable TRPV1 0 45 COc1cc([C@H](C)CCN)ccc1O ZINC000217783514 AD In-Stock Unstable N1L 0 59 COc1cc([C@H](C)CCN)ccc1O ZINC000217783514 AD In-Stock Unstable CAN2 0 49 COc1cc([C@H](C)CCN)ccc1O ZINC000217783514 AD In-Stock Unstable SLC22A3 0 52 O=C(NCc1cccs1)NC[C@@H]1CCCN1c1nccs1 ZINC000217783522 DF For-Sale Unstable ADAM17 19 43 CCOCCNS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217783548 CD For-Sale Unstable FBP1 0 43 CCOCCNS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217783548 CD For-Sale Unstable AKR1C3 27 43 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable F2 41 52 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable PLG 22 49 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable PRSS1 27 49 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable ACE 38 41 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable LHCGR 46 38 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable OPRM1 73 68 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable OPRD1 71 68 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable OPRK1 15 56 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable OPRL1 0 56 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable F10 0 50 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable MME 95 42 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable ANPEP 76 39 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable NPR1 55 48 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable TACR1 26 57 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable CCNA2 0 47 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable AGTR2 0 42 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable BDKRB2 0 40 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable HLA-DRB3 19 51 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable MC4R 82 64 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable FCER2 103 44 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable NPY4R 0 43 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable TACR2 57 45 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable RNPEP 34 42 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable NPR3 0 48 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable PFDN6 0 62 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable NPY1R 19 57 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable KLK3 95 38 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable CTSB 62 53 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable PAPA1_CARPA 78 47 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable TRY1_BOVIN 57 42 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable CYSP_TRYCR 59 37 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable CCKAR 64 39 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable NPY2R 0 63 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable NTSR1 36 48 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable CTSK 16 47 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable CTSL 44 54 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable F2R 74 70 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable NPFFR2 111 57 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable C3AR1 41 45 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable HLA-A 55 39 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable TACR3 27 45 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable MC3R 109 58 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable MC5R 105 60 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable CAPNS1 65 36 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable MMP2 23 49 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable MMP3 48 50 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable MMP8 40 35 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable MMP14 58 38 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable HLA-DRB1 115 62 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable REN 49 42 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable REN1 57 42 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable LNPEP 18 42 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable MMP11 47 35 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable F11 32 41 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable PAM 0 44 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable PCSK5 46 39 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable PLAT 21 41 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable FURIN 105 49 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable CCKBR 43 51 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable GHSR 15 43 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable CAPN1 84 50 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable MMP9 26 45 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable CAPN2 103 41 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable ACE2 68 38 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable MC1R 163 64 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable F7 35 47 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable LAP3 39 42 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable PROTEASE 0 41 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable C5AR1 37 44 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable PSENEN 0 42 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable ST14 60 39 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable GNPAT 0 47 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable MMP1 40 46 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable FPR1 80 44 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable POL 0 45 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable NPR 48 33 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable AMP1_PLAFQ 24 45 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable GSP 0 46 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable AGRC 0 40 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable GAG-PRO 42 35 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable XIAP 19 47 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable Q95WR6_LEIDO 0 48 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable POLG_DEN26 0 53 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable SLC15A2 0 50 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable BLA1_STEMA 85 47 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable KISS1R 82 38 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable POLG_WNV 71 34 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable QRFPR 74 53 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable F2RL1 48 32 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable NPFFR1 104 51 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable LASB 0 44 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable WDR5 42 34 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable Q9NAW4_PLAFA 16 48 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable CD36 0 41 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable CBX7 0 48 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable TMPRSS6 70 39 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable HPN 63 39 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable VM1B1_BOTAS 0 45 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable CBX8 0 42 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable CBX4 0 48 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable H9B8T9_CAPHI 47 48 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable HGFAC 0 48 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable A0A0H4FQ60_PLAVI 0 40 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable Q8I6Z5_PLAF7 0 40 C[C@@H](O)[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O ZINC000217783570 HA Annotated Unstable Q91H74_9FLAV 0 42 O=C(NCc1cccs1)NC[C@H]1CCCN1c1nccs1 ZINC000217783607 DF For-Sale Unstable ADAM17 19 43 CCN(CC)c1ccc(-c2nc3ccccc3s2)c(OC)c1 ZINC000217783688 DJ In-Stock Unstable TEK 20 48 CCN(CC)c1ccc(-c2nc3ccccc3s2)c(OC)c1 ZINC000217783688 DJ In-Stock Unstable LUCI_PHOPY 19 49 CCN(CC)c1ccc(-c2nc3ccccc3s2)c(OC)c1 ZINC000217783688 DJ In-Stock Unstable LUCI_PHOPE 35 49 COc1ccc(NC(=O)NC[C@@H]2CCCN2c2nccs2)c(OC)c1 ZINC000217783698 FF For-Sale Unstable PDGFRB 15 40 COc1ccc(NC(=O)NC[C@@H]2CCCN2c2nccs2)c(OC)c1 ZINC000217783698 FF For-Sale Unstable PDGFRA 26 40 COc1ccc(NC(=O)NC[C@@H]2CCCN2c2nccs2)c(OC)c1 ZINC000217783698 FF For-Sale Unstable ACKR3 60 31 COc1ccc(NC(=O)NC[C@H]2CCCN2c2nccs2)c(OC)c1 ZINC000217783778 FF For-Sale Unstable PDGFRB 15 40 COc1ccc(NC(=O)NC[C@H]2CCCN2c2nccs2)c(OC)c1 ZINC000217783778 FF For-Sale Unstable PDGFRA 26 40 COc1ccc(NC(=O)NC[C@H]2CCCN2c2nccs2)c(OC)c1 ZINC000217783778 FF For-Sale Unstable ACKR3 60 31 Cc1ccc(C(=O)NCCc2noc(C(F)(F)F)n2)s1 ZINC000217783839 DE In-Stock Unstable HDAC4 15 41 Cc1cccc(Cc2cnc(NC(=O)CN(C)C3CCCC3)s2)c1 ZINC000217783876 EH On-Demand Unstable CDK5 57 44 Cc1cccc(Cc2cnc(NC(=O)CN(C)C3CCCC3)s2)c1 ZINC000217783876 EH On-Demand Unstable SCD 34 45 Cc1cccc(Cc2cnc(NC(=O)CN(C)C3CCCC3)s2)c1 ZINC000217783876 EH On-Demand Unstable MGEA5 33 46 COc1ccc(CNC(=O)NC[C@@H]2CCCN2c2nccs2)cc1OC ZINC000217783896 GF For-Sale Unstable PDE5A 15 40 COc1ccc(CNC(=O)NC[C@@H]2CCCN2c2nccs2)cc1OC ZINC000217783896 GF For-Sale Unstable NOS2 24 46 COc1ccc(CNC(=O)NC[C@@H]2CCCN2c2nccs2)cc1OC ZINC000217783896 GF For-Sale Unstable ACKR3 40 33 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc3cccnc23)CC(=O)O4)cc1O ZINC000217783938 JJ In-Stock Unstable CYP1B1 40 34 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc3cccnc23)CC(=O)O4)cc1O ZINC000217783938 JJ In-Stock Unstable CYP1A1 34 42 COc1ccc(CNC(=O)NC[C@H]2CCCN2c2nccs2)cc1OC ZINC000217783976 GF For-Sale Unstable PDE5A 15 40 COc1ccc(CNC(=O)NC[C@H]2CCCN2c2nccs2)cc1OC ZINC000217783976 GF For-Sale Unstable NOS2 24 46 COc1ccc(CNC(=O)NC[C@H]2CCCN2c2nccs2)cc1OC ZINC000217783976 GF For-Sale Unstable ACKR3 40 33 COc1cc([C@@H](C)N(C)[C@@H](C)C(C)C)ccc1O ZINC000217783977 CG For-Sale Unstable PNLIP 0 63 COc1cc([C@@H](C)N(C)[C@@H](C)C(C)C)ccc1O ZINC000217783977 CG For-Sale Unstable FOLH1 0 40 COc1cc([C@@H](C)N(C)[C@@H](C)C(C)C)ccc1O ZINC000217783977 CG For-Sale Unstable TTR 0 50 COc1cc([C@@H](C)N(C)[C@@H](C)C(C)C)ccc1O ZINC000217783977 CG For-Sale Unstable N1L 0 61 COc1cc([C@@H](C)N(C)[C@@H](C)C(C)C)ccc1O ZINC000217783977 CG For-Sale Unstable CAN2 0 50 COc1cc([C@@H](C)N(C)[C@@H](C)C(C)C)ccc1O ZINC000217783977 CG For-Sale Unstable SLC22A3 0 54 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc3cccnc23)CC(=O)O4)cc1O ZINC000217784024 JJ In-Stock Unstable CYP1B1 40 34 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc3cccnc23)CC(=O)O4)cc1O ZINC000217784024 JJ In-Stock Unstable CYP1A1 34 42 CC[C@@H](C)[C@@H](C)NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217784059 DE For-Sale Unstable HDAC8 15 45 CC[C@@H](C)[C@@H](C)NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217784059 DE For-Sale Unstable LEF 22 40 CCCCCNC(=O)Cc1cc(C)ccc1N ZINC000217784061 BE In-Stock Unstable PA2A1_NAJMO 0 40 CCCCCNC(=O)Cc1cc(C)ccc1N ZINC000217784061 BE In-Stock Unstable ASAH1 72 35 CCCCCNC(=O)Cc1cc(C)ccc1N ZINC000217784061 BE In-Stock Unstable ACAT 0 44 COc1cccc(NC(=O)NC[C@@H]2CCCN2c2nccs2)c1OC ZINC000217784097 FF For-Sale Unstable ACKR3 45 32 CC[C@H](C)[C@@H](C)NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217784129 DE For-Sale Unstable HDAC8 15 45 CC[C@H](C)[C@@H](C)NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217784129 DE For-Sale Unstable LEF 22 40 COc1cccc(NC(=O)NC[C@H]2CCCN2c2nccs2)c1OC ZINC000217784173 FF For-Sale Unstable ACKR3 45 32 COCCNC(=O)Cc1cc(C)ccc1N ZINC000217784180 BC In-Stock Unstable CAN2 0 48 CC[C@H](NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1)C(C)C ZINC000217784212 DE For-Sale Unstable LEF 24 44 CC[C@@H](C)c1ccccc1NC(=O)N/C=C/c1ccccc1F ZINC000217784257 DK For-Sale Unstable KCNQ2 40 39 CC[C@@H](NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1)C(C)C ZINC000217784303 DE For-Sale Unstable LEF 24 44 COC(=O)C[C@H](c1cc(OC)c(OC)c(OC)c1)c1c(O)c2ccccc2oc1=O ZINC000217784322 HG In-Stock Unstable CYP2C9 17 40 COC(=O)C[C@H](c1cc(OC)c(OC)c(OC)c1)c1c(O)c2ccccc2oc1=O ZINC000217784322 HG In-Stock Unstable NQO1 70 54 CC[C@H](C)c1ccccc1NC(=O)N/C=C/c1ccccc1F ZINC000217784350 DK For-Sale Unstable KCNQ2 40 39 COC(=O)C[C@@H](c1cc(OC)c(OC)c(OC)c1)c1c(O)c2ccccc2oc1=O ZINC000217784406 HG In-Stock Unstable CYP2C9 17 40 COC(=O)C[C@@H](c1cc(OC)c(OC)c(OC)c1)c1c(O)c2ccccc2oc1=O ZINC000217784406 HG In-Stock Unstable NQO1 70 54 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable ACE 89 46 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable OPRM1 80 53 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable OPRD1 101 53 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable OPRK1 23 45 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable P2RY12 87 40 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable FOLH1 43 50 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable MME 169 50 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable LTA4H 32 49 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable ANPEP 106 43 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable EDNRB 18 40 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable EDNRA 23 45 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable TACR1 34 55 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable CTSD 27 46 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable MC4R 28 40 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable CMA1 31 45 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable CTRA_BOVIN 22 53 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable FCER2 100 39 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable CASP3 27 46 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable BMP1 69 42 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable TACR2 52 43 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable RNPEP 36 43 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable CASP8 18 40 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable KLK3 100 38 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable CTSB 102 50 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable SRC 17 45 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable PAPA1_CARPA 98 47 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable CYSP_TRYCR 82 51 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable CCKAR 59 40 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable CTSG 31 43 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable CTSK 49 46 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable CTSL 74 50 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable CPA1 47 46 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable CACNA1B 40 36 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable CCR3 26 63 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable PGA 43 41 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable F2R 26 42 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable NPFFR2 76 37 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable TIMP3 84 37 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable CTRB1 42 41 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable NAALAD2 49 50 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable MC5R 40 34 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable CAPNS1 84 47 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable MMP2 39 46 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable MMP3 61 46 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable MMP8 33 47 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable GRIA1 56 36 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable MMP14 55 35 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable HLA-DRB1 98 45 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable CELA2A 28 43 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable REN 63 41 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable LNPEP 35 43 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable MMP11 51 35 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable YARS 67 39 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable CCKBR 49 53 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable CTSS 36 46 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable GHSR 16 45 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable CTSH 31 42 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable CAPN1 131 50 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable MMP9 37 44 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable CASP1 37 40 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable CTRC 34 45 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable CAPN2 159 51 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable ACE2 94 46 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable MC1R 69 38 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable CASP6 38 40 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable CASP9 36 40 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable LAP3 62 43 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable CTSC 34 46 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable MMP7 33 43 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable MMP1 50 47 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable FPR1 83 43 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable CTRB_BOVIN 71 48 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable NPR 91 48 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable AMP1_PLAFQ 35 49 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable FFAR1 41 35 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable PSMB2 40 44 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable PSMB5 70 40 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable BLA1_STEMA 80 42 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable BIRC2 15 51 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable ERAP2 50 39 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable QRFPR 50 38 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable PSMB8 52 35 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable NPFFR1 75 38 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable METAP2 28 50 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable NOD1 43 35 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCC(=O)O ZINC000217784418 DC For-Sale Unstable TMPRSS6 46 37 Cc1ccc(N)c(CC(=O)N2CCCCC2)c1 ZINC000217784522 BE In-Stock Unstable ECE2 0 40 COc1ccc(CCC(=O)N2[C@@H](C)C[C@@H]3CNC[C@H]32)cc1 ZINC000217784548 CD For-Sale Unstable SLC18A2 15 40 O=C(N/C=C/c1ccccc1F)NC1CCN(Cc2ccccc2)CC1 ZINC000217784562 FH For-Sale Unstable DRD2 0 52 O=C(N/C=C/c1ccccc1F)NC1CCN(Cc2ccccc2)CC1 ZINC000217784562 FH For-Sale Unstable DRD3 24 58 O=C(N/C=C/c1ccccc1F)NC1CCN(Cc2ccccc2)CC1 ZINC000217784562 FH For-Sale Unstable ADIPOR1 0 47 O=C(N/C=C/c1ccccc1F)NC1CCN(Cc2ccccc2)CC1 ZINC000217784562 FH For-Sale Unstable ADIPOR2 0 47 COc1ccc(CCC(=O)N2[C@@H]3CNC[C@H]3C[C@H]2C)cc1 ZINC000217784619 CD For-Sale Unstable SLC18A2 15 40 O=C1C[C@@H](c2coc3ccccc3c2=O)c2c(c3ccccc3oc2=O)O1 ZINC000217784621 FG In-Stock Unstable VKORC1 0 40 CC(C)[C@@H](C)NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217784660 CE For-Sale Unstable HDAC8 15 49 CC(C)[C@@H](C)NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217784660 CE For-Sale Unstable MMP12 43 37 CC(C)[C@@H](C)NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217784660 CE For-Sale Unstable LEF 26 48 COc1ccc(CN2C[C@@H]3CC[C@H](C2)[C@@H]3O)c(OC)c1OC ZINC000217784673 DD In-Stock Unstable SLC9A1 58 32 COc1ccc(CCC(=O)N2[C@@H](C)C[C@H]3CNC[C@H]32)cc1 ZINC000217784700 CD For-Sale Unstable SLC18A2 15 40 O=C1C[C@H](c2coc3ccccc3c2=O)c2c(c3ccccc3oc2=O)O1 ZINC000217784713 FG In-Stock Unstable VKORC1 0 40 CC(C)[C@H](C)NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217784749 CE For-Sale Unstable HDAC8 15 49 CC(C)[C@H](C)NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217784749 CE For-Sale Unstable MMP12 43 37 CC(C)[C@H](C)NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217784749 CE For-Sale Unstable LEF 26 48 COc1ccc(CCC(=O)N2[C@@H]3CNC[C@@H]3C[C@H]2C)cc1 ZINC000217784789 CD For-Sale Unstable SLC18A2 15 40 Cc1ccc(N)c(CC(=O)N2CCC[C@@H](C)C2)c1 ZINC000217784806 BE In-Stock Unstable RORC 29 40 CCN(C)C(=O)CNC(=O)Cc1ccccc1C(=O)O ZINC000217784807 CC On-Demand Unstable ECR 22 40 O=C(O)CNC(=O)CNC(=O)CCc1cc(O)no1 ZINC000217784810 CA In-Stock Unstable GABRR2 0 40 O=C(N/C=C/c1ccccc1F)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217784901 GG For-Sale Unstable DRD4 17 47 O=C(N/C=C/c1ccccc1F)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217784901 GG For-Sale Unstable SIGMAR1 15 52 O=C(N/C=C/c1ccccc1F)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217784901 GG For-Sale Unstable NOS2 49 35 O=C(N/C=C/c1ccccc1F)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217784901 GG For-Sale Unstable FAAH 18 41 O=C(N/C=C/c1ccccc1F)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217784901 GG For-Sale Unstable MCHR1 32 50 Cc1ccc(N)c(CC(=O)N2CCC[C@H](C)C2)c1 ZINC000217784905 BE In-Stock Unstable RORC 29 40 CCN(C(C)C)S(=O)(=O)c1ccc(/C=C\C(=O)O)cc1Cl ZINC000217784918 EF For-Sale Unstable NR0B2 0 42 O=C(C[C@@H]1NC(=O)N(Cc2cccc(Cl)c2)C1=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217784931 JD In-Stock Unstable CHRNA4 28 48 CCN(C(C)C)S(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217785014 CE For-Sale Unstable AKR1C3 27 40 CCOC(=O)N1CCN(C(=O)N/C=C/c2ccccc2F)CC1 ZINC000217785015 DE For-Sale Unstable P2RY12 60 36 CC(=O)Nc1ccc(C(=O)N2CC[C@H](N3C(=O)CSC3=O)C2)cc1 ZINC000217785020 ED In-Stock Unstable AVPR1A 34 40 CC(=O)Nc1ccc(C(=O)N2CC[C@H](N3C(=O)CSC3=O)C2)cc1 ZINC000217785020 ED In-Stock Unstable L3MBTL1 0 43 CC(=O)Nc1ccc(C(=O)N2CC[C@H](N3C(=O)CSC3=O)C2)cc1 ZINC000217785020 ED In-Stock Unstable L3MBTL3 70 43 Cc1ccc(N)c(CC(=O)N2CCC(C)CC2)c1 ZINC000217785023 BE In-Stock Unstable TRPC6 40 39 C[C@@H](c1ccc(Cl)cc1)N(C)[C@H]([C@@H](C)N)C(F)(F)F ZINC000217785031 CH For-Sale Unstable UTS2 42 33 COc1cc2ncn(CC(=O)N[C@H](CO)Cc3ccccc3)c(=O)c2cc1OC ZINC000217785040 GD In-Stock Unstable CMA1 41 34 COc1cc2ncn(CC(=O)N[C@H](CO)Cc3ccccc3)c(=O)c2cc1OC ZINC000217785040 GD In-Stock Unstable CTRA_BOVIN 43 34 COc1cc2ncn(CC(=O)N[C@H](CO)Cc3ccccc3)c(=O)c2cc1OC ZINC000217785040 GD In-Stock Unstable KDR 41 37 COc1cc2ncn(CC(=O)N[C@H](CO)Cc3ccccc3)c(=O)c2cc1OC ZINC000217785040 GD In-Stock Unstable CTRC 42 33 COc1cc2ncn(CC(=O)N[C@H](CO)Cc3ccccc3)c(=O)c2cc1OC ZINC000217785040 GD In-Stock Unstable PDGFRA 48 37 COc1cc2ncn(CC(=O)N[C@H](CO)Cc3ccccc3)c(=O)c2cc1OC ZINC000217785040 GD In-Stock Unstable SCD1 0 41 COc1cc2ncn(CC(=O)N[C@H](CO)Cc3ccccc3)c(=O)c2cc1OC ZINC000217785040 GD In-Stock Unstable ENPP1 46 30 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1ccccc1 ZINC000217785050 DE For-Sale Unstable ADAMTS5 36 47 CC(=O)Nc1ccc(C(=O)N2CC[C@@H](N3C(=O)CSC3=O)C2)cc1 ZINC000217785102 ED In-Stock Unstable AVPR1A 34 40 CC(=O)Nc1ccc(C(=O)N2CC[C@@H](N3C(=O)CSC3=O)C2)cc1 ZINC000217785102 ED In-Stock Unstable L3MBTL1 0 43 CC(=O)Nc1ccc(C(=O)N2CC[C@@H](N3C(=O)CSC3=O)C2)cc1 ZINC000217785102 ED In-Stock Unstable L3MBTL3 70 43 C[C@H](N)[C@@H](N(C)[C@@H](C)c1ccc(Cl)cc1)C(F)(F)F ZINC000217785124 CH For-Sale Unstable UTS2 42 33 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1ccccc1 ZINC000217785128 DE For-Sale Unstable ADAMTS5 36 47 Cc1ccc(N)c(CC(=O)N2C[C@@H](C)C[C@@H](C)C2)c1 ZINC000217785131 CF In-Stock Unstable RORC 26 40 O=C(c1ccc2cc[nH]c2c1)N1CC[C@H](N2C(=O)CSC2=O)C1 ZINC000217785209 EE In-Stock Unstable GHSR 0 47 O=C(c1ccc2cc[nH]c2c1)N1CC[C@H](N2C(=O)CSC2=O)C1 ZINC000217785209 EE In-Stock Unstable L3MBTL1 0 41 O=C(c1ccc2cc[nH]c2c1)N1CC[C@H](N2C(=O)CSC2=O)C1 ZINC000217785209 EE In-Stock Unstable L3MBTL3 54 34 Cc1ccc(N)c(CC(=O)N2C[C@H](C)C[C@@H](C)C2)c1 ZINC000217785210 CF In-Stock Unstable RORC 26 40 C[C@H](N)[C@H](N(C)[C@@H](C)c1ccc(Cl)cc1)C(F)(F)F ZINC000217785211 CH For-Sale Unstable UTS2 42 33 CNCCc1cc(Br)c(C)cc1F ZINC000217785246 BF For-Sale Unstable TAAR1 15 47 O=C(c1ccc2cc[nH]c2c1)N1CC[C@@H](N2C(=O)CSC2=O)C1 ZINC000217785283 EE In-Stock Unstable GHSR 0 47 O=C(c1ccc2cc[nH]c2c1)N1CC[C@@H](N2C(=O)CSC2=O)C1 ZINC000217785283 EE In-Stock Unstable L3MBTL1 0 41 O=C(c1ccc2cc[nH]c2c1)N1CC[C@@H](N2C(=O)CSC2=O)C1 ZINC000217785283 EE In-Stock Unstable L3MBTL3 54 34 Cc1ccc(N)c(CC(=O)N2C[C@@H](C)C[C@H](C)C2)c1 ZINC000217785286 CF In-Stock Unstable RORC 26 40 O=C(N/C=C/c1ccccc1F)Nc1ccc(C(F)(F)F)cc1 ZINC000217785328 DJ For-Sale Anodyne EPHX2 27 41 O=C(N/C=C/c1ccccc1F)Nc1ccc(C(F)(F)F)cc1 ZINC000217785328 DJ For-Sale Anodyne PTPA 0 41 O=C(c1cccc(Br)c1)N1CC[C@H](N2C(=O)CSC2=O)C1 ZINC000217785376 FE In-Stock Unstable L3MBTL1 0 58 O=C(c1cccc(Br)c1)N1CC[C@H](N2C(=O)CSC2=O)C1 ZINC000217785376 FE In-Stock Unstable L3MBTL3 53 37 O=C(c1cccc(Br)c1)N1CC[C@H](N2C(=O)CSC2=O)C1 ZINC000217785376 FE In-Stock Unstable MBTD1 0 46 Cc1cc(S(=O)(=O)N[C@@H](C)C(C)C)ccc1/C=C\C(=O)O ZINC000217785406 DE For-Sale Unstable MMP13 21 40 Cc1cc(S(=O)(=O)N[C@@H](C)C(C)C)ccc1/C=C\C(=O)O ZINC000217785406 DE For-Sale Unstable MMP12 64 36 Cc1cc(S(=O)(=O)N[C@@H](C)C(C)C)ccc1/C=C\C(=O)O ZINC000217785406 DE For-Sale Unstable LEF 61 40 Cc1cccc(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217785420 EE For-Sale Unstable ADAMTS5 33 44 CNCCc1cc(C)cc(Br)c1F ZINC000217785425 BF For-Sale Unstable TAAR1 15 46 O=C(c1cccc(Br)c1)N1CC[C@@H](N2C(=O)CSC2=O)C1 ZINC000217785454 FE In-Stock Unstable L3MBTL1 0 58 O=C(c1cccc(Br)c1)N1CC[C@@H](N2C(=O)CSC2=O)C1 ZINC000217785454 FE In-Stock Unstable L3MBTL3 61 43 O=C(c1cccc(Br)c1)N1CC[C@@H](N2C(=O)CSC2=O)C1 ZINC000217785454 FE In-Stock Unstable MBTD1 0 46 Cc1cc(S(=O)(=O)N[C@H](C)C(C)C)ccc1/C=C\C(=O)O ZINC000217785475 DE For-Sale Unstable MMP13 21 40 Cc1cc(S(=O)(=O)N[C@H](C)C(C)C)ccc1/C=C\C(=O)O ZINC000217785475 DE For-Sale Unstable MMP12 64 36 Cc1cc(S(=O)(=O)N[C@H](C)C(C)C)ccc1/C=C\C(=O)O ZINC000217785475 DE For-Sale Unstable LEF 61 40 Cc1cccc(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217785503 EE For-Sale Unstable ADAMTS5 33 44 CNCCc1ccc(CF)c(Br)c1 ZINC000217785526 BF For-Sale Unstable TAAR1 18 46 CCN(C)C(=O)CNC(=O)CCCCC(=O)O ZINC000217785601 BC On-Demand Unstable FABP4 16 41 CCN(C)C(=O)CNC(=O)CCCCC(=O)O ZINC000217785601 BC On-Demand Unstable FABP3 34 41 CCN(C)C(=O)CNC(=O)CCCCC(=O)O ZINC000217785601 BC On-Demand Unstable FABP5 15 41 CCN(C)C(=O)CNC(=O)CCCCC(=O)O ZINC000217785601 BC On-Demand Unstable SLC22A20 0 41 CCN(C)C(=O)CNC(=O)CCCCC(=O)O ZINC000217785601 BC On-Demand Unstable PHF8 0 40 CCN(C)C(=O)CNC(=O)CCCCC(=O)O ZINC000217785601 BC On-Demand Unstable KDM7A 0 40 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1ccccc1F ZINC000217785605 EE For-Sale Unstable ADAMTS5 32 41 COc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)N1CCN(c3ccccc3)CC1)C(=O)OC2 ZINC000217785609 JH In-Stock Unstable IMPDH1 0 68 COc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)N1CCN(c3ccccc3)CC1)C(=O)OC2 ZINC000217785609 JH In-Stock Unstable IMPDH2 0 68 C[C@H](F)c1ccc(CCN)cc1Br ZINC000217785629 BF For-Sale Unstable TAAR1 19 42 C[C@@H](c1ccccc1Cl)N(C)C[C@@H](O)c1cccc(N)c1 ZINC000217785634 DH For-Sale Unstable AOC3 39 50 Cc1ccc(N)c(CC(=O)N2CCOCC2)c1 ZINC000217785646 BC In-Stock Unstable AKR1C3 29 44 O=C(N/C=C/c1ccccc1F)N1CCCC[C@H]1CCO ZINC000217785648 CF For-Sale Unstable SLC6A1 43 35 CCN1CCN(CC(=O)N[C@@H](c2ccncc2)c2ccc(C)cc2)CC1 ZINC000217785676 FE In-Stock Unstable PRNP 22 41 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1ccccc1F ZINC000217785683 EE For-Sale Unstable ADAMTS5 32 41 C[C@H](c1ccccc1Cl)N(C)C[C@@H](O)c1cccc(N)c1 ZINC000217785703 DH For-Sale Unstable AOC3 39 50 C[C@@H](F)c1ccc(CCN)cc1Br ZINC000217785714 BF For-Sale Unstable TAAR1 19 42 O=C(N/C=C/c1ccccc1F)N1CCCC[C@@H]1CCO ZINC000217785729 CF For-Sale Unstable SLC6A1 43 35 COc1ccc(-c2csc(NC(=O)CN[C@@H](c3ccccc3)C3CC3)n2)c(OC)c1 ZINC000217785752 HJ On-Demand Unstable ROCK1 16 40 CCN1CCN(CC(=O)N[C@H](c2ccncc2)c2ccc(C)cc2)CC1 ZINC000217785756 FE In-Stock Unstable PRNP 22 41 O=C(c1cccc2ccccc12)N1CC[C@H](N2C(=O)CSC2=O)C1 ZINC000217785763 EF In-Stock Unstable L3MBTL1 0 43 O=C(c1cccc2ccccc12)N1CC[C@H](N2C(=O)CSC2=O)C1 ZINC000217785763 EF In-Stock Unstable L3MBTL3 34 43 O=C(c1cccc2ccccc12)N1CC[C@H](N2C(=O)CSC2=O)C1 ZINC000217785763 EF In-Stock Unstable MBTD1 0 43 O=C(c1cccc2ccccc12)N1CC[C@H](N2C(=O)CSC2=O)C1 ZINC000217785763 EF In-Stock Unstable TP53BP1 0 40 C[C@@H](c1ccccc1Cl)N(C)C[C@@H](O)c1ccccc1N ZINC000217785795 DH For-Sale Unstable AOC3 17 59 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1ccc(F)cc1 ZINC000217785803 EE For-Sale Unstable ADAMTS5 35 50 COc1ccc(-c2csc(NC(=O)CN[C@H](c3ccccc3)C3CC3)n2)c(OC)c1 ZINC000217785825 HJ On-Demand Unstable ROCK1 16 40 O=C(c1cccc2ccccc12)N1CC[C@@H](N2C(=O)CSC2=O)C1 ZINC000217785839 EF In-Stock Unstable L3MBTL1 0 43 O=C(c1cccc2ccccc12)N1CC[C@@H](N2C(=O)CSC2=O)C1 ZINC000217785839 EF In-Stock Unstable L3MBTL3 34 43 O=C(c1cccc2ccccc12)N1CC[C@@H](N2C(=O)CSC2=O)C1 ZINC000217785839 EF In-Stock Unstable MBTD1 0 43 O=C(c1cccc2ccccc12)N1CC[C@@H](N2C(=O)CSC2=O)C1 ZINC000217785839 EF In-Stock Unstable TP53BP1 0 40 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1ccc(F)cc1 ZINC000217785883 EE For-Sale Unstable ADAMTS5 35 50 C[C@H](c1ccccc1Cl)N(C)C[C@@H](O)c1ccccc1N ZINC000217785886 DH For-Sale Unstable AOC3 17 59 COc1cc([C@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2oc(C)cc(=O)c2O)ccc1O ZINC000217785912 JH In-Stock Unstable RORC 49 34 CCCCCCCC(=O)N1[C@@H](C)C[C@@H]2CNC[C@H]21 ZINC000217785927 CF For-Sale Unstable CQSS 50 32 O=C(Cc1c[nH]c2ccccc12)N1CC[C@H](N2C(=O)CSC2=O)C1 ZINC000217785950 EE In-Stock Unstable SSTR2 40 32 O=C(Cc1c[nH]c2ccccc12)N1CC[C@H](N2C(=O)CSC2=O)C1 ZINC000217785950 EE In-Stock Unstable TACR2 29 46 O=C(Cc1c[nH]c2ccccc12)N1CC[C@H](N2C(=O)CSC2=O)C1 ZINC000217785950 EE In-Stock Unstable MC5R 29 41 O=C(Cc1c[nH]c2ccccc12)N1CC[C@H](N2C(=O)CSC2=O)C1 ZINC000217785950 EE In-Stock Unstable CCR2 45 34 O=C(N/C=C/c1ccccc1F)N1CCN(c2ccccn2)CC1 ZINC000217785965 EF For-Sale Unstable SLC6A7 0 45 C[C@@H](c1ccccc1Cl)N(C)C[C@@H](O)c1ccc(N)cc1 ZINC000217785967 DH For-Sale Unstable AOC3 28 52 COc1cc([C@@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2oc(C)cc(=O)c2O)ccc1O ZINC000217785983 JH In-Stock Unstable RORC 49 34 CCCCCCCC(=O)N1[C@@H]2CNC[C@H]2C[C@H]1C ZINC000217786003 CF For-Sale Unstable CQSS 50 32 Cc1ccc(N)c(CC(=O)N2CCN(C)CC2)c1 ZINC000217786020 BC In-Stock Unstable HRH4 27 43 O=C(Cc1c[nH]c2ccccc12)N1CC[C@@H](N2C(=O)CSC2=O)C1 ZINC000217786024 EE In-Stock Unstable SSTR2 40 32 O=C(Cc1c[nH]c2ccccc12)N1CC[C@@H](N2C(=O)CSC2=O)C1 ZINC000217786024 EE In-Stock Unstable TACR2 29 46 O=C(Cc1c[nH]c2ccccc12)N1CC[C@@H](N2C(=O)CSC2=O)C1 ZINC000217786024 EE In-Stock Unstable MC5R 29 41 O=C(Cc1c[nH]c2ccccc12)N1CC[C@@H](N2C(=O)CSC2=O)C1 ZINC000217786024 EE In-Stock Unstable CCR2 45 34 C[C@H](c1ccccc1Cl)N(C)C[C@@H](O)c1ccc(N)cc1 ZINC000217786051 DH For-Sale Unstable AOC3 28 52 COC(=O)CCNC(=O)N/C=C/c1ccccc1F ZINC000217786083 CD For-Sale Unstable TLR4 19 44 CCCCCCCC(=O)N1[C@@H](C)C[C@H]2CNC[C@H]21 ZINC000217786093 CF For-Sale Unstable CQSS 50 32 Cc1ccc(N)c(CC(=O)N2CCCCCC2)c1 ZINC000217786105 BF In-Stock Unstable ECE2 0 40 CN1CC[C@H](NS(=O)(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217786118 DC For-Sale Unstable HDAC8 28 42 CN1CC[C@H](NS(=O)(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217786118 DC For-Sale Unstable SFRP1 131 39 CN1CC[C@H](NS(=O)(=O)c2cccc(/C=C\C(=O)O)c2)C1 ZINC000217786118 DC For-Sale Unstable WNT3 87 38 CCCCCCCC(=O)N1[C@@H]2CNC[C@@H]2C[C@H]1C ZINC000217786180 CF For-Sale Unstable CQSS 50 32 CC(C)CCN(C)S(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217786211 DE For-Sale Unstable AKR1C3 27 40 O=C(O)/C=C\c1cccc(S(=O)(=O)N2CCC[C@@H]2CO)c1 ZINC000217786293 DC For-Sale Unstable CASP3 91 38 O=C(O)/C=C\c1cccc(S(=O)(=O)N2CCC[C@@H]2CO)c1 ZINC000217786293 DC For-Sale Unstable CASP7 103 39 O=C(c1ccoc1)N1CC[C@H](N2C(=O)CSC2=O)C1 ZINC000217786322 CD In-Stock Unstable L3MBTL1 0 40 O=C(c1ccoc1)N1CC[C@H](N2C(=O)CSC2=O)C1 ZINC000217786322 CD In-Stock Unstable L3MBTL3 52 40 Cc1ccc(N)c(CC(=O)NC2CCCC2)c1 ZINC000217786325 BE In-Stock Unstable FAAH 17 45 Cc1ccc(N)c(CC(=O)NC2CCCC2)c1 ZINC000217786325 BE In-Stock Unstable EPHX2 28 46 CCc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)cc1 ZINC000217786366 FF For-Sale Unstable ADAMTS5 37 47 CCC(CC)NC(=O)c1c[nH]nc1-c1ccc(Cl)cc1 ZINC000217786377 CH On-Demand Unstable UTS2 42 33 O=C(c1ccoc1)N1CC[C@@H](N2C(=O)CSC2=O)C1 ZINC000217786405 CD In-Stock Unstable L3MBTL1 0 40 O=C(c1ccoc1)N1CC[C@@H](N2C(=O)CSC2=O)C1 ZINC000217786405 CD In-Stock Unstable L3MBTL3 52 40 COC(=O)CNC(=O)N/C=C/c1ccccc1F ZINC000217786422 CD For-Sale Unstable TLR4 23 45 CN1CCC[C@@H]2CN(c3ccc(CBr)cc3)CC[C@@H]21 ZINC000217786425 DH For-Sale Unstable HRH3 0 40 Cc1ccc(N)c(CC(=O)NC2CCCCC2)c1 ZINC000217786438 BF In-Stock Unstable CNR2 18 40 Cc1ccc(N)c(CC(=O)NC2CCCCC2)c1 ZINC000217786438 BF In-Stock Unstable FAAH 23 47 Cc1ccc(N)c(CC(=O)NC2CCCCC2)c1 ZINC000217786438 BF In-Stock Unstable EPHX2 37 48 CCc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)cc1 ZINC000217786462 FF For-Sale Unstable ADAMTS5 37 47 O=C(Cc1ccc2c(c1)OCO2)N1CC[C@H](N2C(=O)CSC2=O)C1 ZINC000217786510 ED In-Stock Unstable NOS2 68 32 O=C(Cc1ccc2c(c1)OCO2)N1CC[C@H](N2C(=O)CSC2=O)C1 ZINC000217786510 ED In-Stock Unstable SSTR3 101 35 CN1CCC[C@H]2CN(c3ccc(CBr)cc3)CC[C@@H]21 ZINC000217786517 DH For-Sale Unstable HRH3 0 40 COC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2F)c1 ZINC000217786534 DG For-Sale Unstable KCNK3 101 37 COC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2F)c1 ZINC000217786534 DG For-Sale Unstable KCNK9 71 34 CCCCCC(=O)N1[C@@H](C)C[C@@H]2CNC[C@H]21 ZINC000217786576 BD For-Sale Unstable GNAI1 0 43 CCCCCC(=O)N1[C@@H](C)C[C@@H]2CNC[C@H]21 ZINC000217786576 BD For-Sale Unstable GNAI3 0 43 CCCCCC(=O)N1[C@@H](C)C[C@@H]2CNC[C@H]21 ZINC000217786576 BD For-Sale Unstable GNAO1 0 43 Cc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)cc1C ZINC000217786579 FF For-Sale Unstable ADAMTS5 35 53 O=C(Cc1ccc2c(c1)OCO2)N1CC[C@@H](N2C(=O)CSC2=O)C1 ZINC000217786583 ED In-Stock Unstable NOS2 68 32 O=C(Cc1ccc2c(c1)OCO2)N1CC[C@@H](N2C(=O)CSC2=O)C1 ZINC000217786583 ED In-Stock Unstable SSTR3 101 35 COc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)Nc1nc(-c3ccccn3)cs1)C(=O)OC2 ZINC000217786626 JJ In-Stock Unstable IMPDH1 0 65 COc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)Nc1nc(-c3ccccn3)cs1)C(=O)OC2 ZINC000217786626 JJ In-Stock Unstable IMPDH2 0 65 CCCCCC(=O)N1[C@@H]2CNC[C@H]2C[C@H]1C ZINC000217786652 BD For-Sale Unstable GNAI1 0 43 CCCCCC(=O)N1[C@@H]2CNC[C@H]2C[C@H]1C ZINC000217786652 BD For-Sale Unstable GNAI3 0 43 CCCCCC(=O)N1[C@@H]2CNC[C@H]2C[C@H]1C ZINC000217786652 BD For-Sale Unstable GNAO1 0 43 Cc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)cc1C ZINC000217786677 FF For-Sale Unstable ADAMTS5 35 53 Clc1cncc(Cl)c1CN1CCNCC1 ZINC000217786695 BD On-Demand Unstable CXCR4 23 43 C[C@@H](c1ccccc1Cl)N(C)[C@H](c1ccccc1)[C@@H](C)N ZINC000217786724 DI For-Sale Unstable AOC3 20 41 CC[C@@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000217786734 CF For-Sale Unstable ACE 24 40 CC[C@@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000217786734 CF For-Sale Unstable MME 58 40 CC[C@@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000217786734 CF For-Sale Unstable ANPEP 67 35 CC[C@@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000217786734 CF For-Sale Unstable PGA 22 44 CC[C@@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000217786734 CF For-Sale Unstable CAPN1 50 46 CC[C@@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000217786734 CF For-Sale Unstable CAPN2 85 41 CC[C@@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000217786734 CF For-Sale Unstable ACE2 62 40 CC[C@@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000217786734 CF For-Sale Unstable CASP9 44 32 CC[C@@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000217786734 CF For-Sale Unstable NPR 40 32 CC[C@@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000217786734 CF For-Sale Unstable XIAP 49 39 CCCCCC(=O)N1[C@@H](C)C[C@H]2CNC[C@H]21 ZINC000217786735 BD For-Sale Unstable GNAI1 0 43 CCCCCC(=O)N1[C@@H](C)C[C@H]2CNC[C@H]21 ZINC000217786735 BD For-Sale Unstable GNAI3 0 43 CCCCCC(=O)N1[C@@H](C)C[C@H]2CNC[C@H]21 ZINC000217786735 BD For-Sale Unstable GNAO1 0 43 CNC(=O)[C@H](C)NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217786757 DC For-Sale Unstable MMP12 43 34 CNC(=O)[C@H](C)NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217786757 DC For-Sale Unstable LEF 28 45 Cc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)c(C)c1 ZINC000217786787 FF For-Sale Unstable ADAMTS5 30 40 C[C@H](N)[C@@H](c1ccccc1)N(C)[C@@H](C)c1ccccc1Cl ZINC000217786801 DI For-Sale Unstable AOC3 20 41 CC[C@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000217786816 CF For-Sale Unstable ACE 24 40 CC[C@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000217786816 CF For-Sale Unstable MME 58 40 CC[C@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000217786816 CF For-Sale Unstable ANPEP 67 35 CC[C@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000217786816 CF For-Sale Unstable PGA 22 44 CC[C@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000217786816 CF For-Sale Unstable CAPN1 50 46 CC[C@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000217786816 CF For-Sale Unstable CAPN2 85 41 CC[C@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000217786816 CF For-Sale Unstable ACE2 62 40 CC[C@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000217786816 CF For-Sale Unstable CASP9 44 32 CC[C@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000217786816 CF For-Sale Unstable NPR 40 32 CC[C@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000217786816 CF For-Sale Unstable XIAP 49 39 CCCCCC(=O)N1[C@@H]2CNC[C@@H]2C[C@H]1C ZINC000217786823 BD For-Sale Unstable GNAI1 0 43 CCCCCC(=O)N1[C@@H]2CNC[C@@H]2C[C@H]1C ZINC000217786823 BD For-Sale Unstable GNAI3 0 43 CCCCCC(=O)N1[C@@H]2CNC[C@@H]2C[C@H]1C ZINC000217786823 BD For-Sale Unstable GNAO1 0 43 COc1ccc(CC(=O)N[C@H](c2ccccc2)c2ccc(C)cc2C)cc1C ZINC000217786853 FK In-Stock Unstable P2RX7 0 40 COc1ccc(CC(=O)N[C@H](c2ccccc2)c2ccc(C)cc2C)cc1C ZINC000217786853 FK In-Stock Unstable RORC 42 57 CNC(=O)[C@@H](C)NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217786856 DC For-Sale Unstable MMP12 43 34 CNC(=O)[C@@H](C)NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217786856 DC For-Sale Unstable LEF 28 45 Cc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)c(C)c1 ZINC000217786868 FF For-Sale Unstable ADAMTS5 30 40 C[C@H](N)[C@H](c1ccccc1)N(C)[C@@H](C)c1ccccc1Cl ZINC000217786894 DI For-Sale Unstable AOC3 20 41 COc1ccc(CC(=O)N[C@@H](c2ccccc2)c2ccc(C)cc2C)cc1C ZINC000217786934 FK In-Stock Unstable P2RX7 0 40 COc1ccc(CC(=O)N[C@@H](c2ccccc2)c2ccc(C)cc2C)cc1C ZINC000217786934 FK In-Stock Unstable RORC 42 57 COC(=O)c1cccc(COc2ccc3occ(-c4cc(OC)c(OC)c(OC)c4)c3c2)c1 ZINC000217786941 IK In-Stock Unstable ALDH2 77 33 COC(=O)c1cccc(COc2ccc3occ(-c4cc(OC)c(OC)c(OC)c4)c3c2)c1 ZINC000217786941 IK In-Stock Unstable MAOB 56 52 COC(=O)c1cccc(COc2ccc3occ(-c4cc(OC)c(OC)c(OC)c4)c3c2)c1 ZINC000217786941 IK In-Stock Unstable GYS1 43 39 COC(=O)c1cccc(COc2ccc3occ(-c4cc(OC)c(OC)c(OC)c4)c3c2)c1 ZINC000217786941 IK In-Stock Unstable TUBB1 17 40 COC(=O)c1cccc(COc2ccc3occ(-c4cc(OC)c(OC)c(OC)c4)c3c2)c1 ZINC000217786941 IK In-Stock Unstable ADAMTS4 15 42 O=C(O)/C=C\c1cccc(S(=O)(=O)N2CCC[C@H](O)C2)c1 ZINC000217786949 DC For-Sale Unstable HDAC8 31 41 O=C(O)/C=C\c1cccc(S(=O)(=O)N2CCC[C@H](O)C2)c1 ZINC000217786949 DC For-Sale Unstable HDAC1 15 41 O=C(O)/C=C\c1cccc(S(=O)(=O)N2CCC[C@H](O)C2)c1 ZINC000217786949 DC For-Sale Unstable HDAC6 15 41 O=C(O)/C=C\c1cccc(S(=O)(=O)N2CCC[C@H](O)C2)c1 ZINC000217786949 DC For-Sale Unstable AKR1C3 58 45 O=C(O)/C=C\c1cccc(S(=O)(=O)N2CCC[C@H](O)C2)c1 ZINC000217786949 DC For-Sale Unstable AKR1C1 23 44 CC(C)[C@@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217786960 CD For-Sale Unstable CTSC 23 40 Cc1ccc(N)c(CC(=O)Nc2nccs2)c1 ZINC000217786980 BE In-Stock Unstable MAP 0 47 Cc1ccc(N)c(CC(=O)Nc2nccs2)c1 ZINC000217786980 BE In-Stock Unstable MAP1 132 47 Cc1ccc(N)c(CC(=O)Nc2nccs2)c1 ZINC000217786980 BE In-Stock Unstable MAPK8 0 45 Cc1ccc(N)c(CC(=O)Nc2nccs2)c1 ZINC000217786980 BE In-Stock Unstable GCK 19 41 Cc1ccc(N)c(CC(=O)Nc2nccs2)c1 ZINC000217786980 BE In-Stock Unstable GLS 0 40 CC(C)[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217787039 CD For-Sale Unstable CTSC 23 40 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccco2)CC(=O)O4)cc1O ZINC000217787041 HH In-Stock Unstable AKR1B1 0 49 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccco2)CC(=O)O4)cc1O ZINC000217787041 HH In-Stock Unstable CYP1B1 65 36 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccco2)CC(=O)O4)cc1O ZINC000217787041 HH In-Stock Unstable CYP1A1 48 47 CN[C@@H]1CC[C@H](C(C)C)C[C@@H]1Cc1cc(F)ccc1F ZINC000217787067 CI For-Sale Unstable DPP4 17 41 Cc1ccc(N)c(CC(=O)NCC2CC2)c1 ZINC000217787097 BD In-Stock Unstable GNRHR 0 41 Cc1ccc(N)c(CC(=O)NCC2CC2)c1 ZINC000217787097 BD In-Stock Unstable CACNA1I 44 38 O=C(O)/C=C\c1cccc(S(=O)(=O)Nc2ncccn2)c1 ZINC000217787099 DD For-Sale Anodyne HDAC8 30 55 O=C(O)/C=C\c1cccc(S(=O)(=O)Nc2ncccn2)c1 ZINC000217787099 DD For-Sale Anodyne HDAC1 15 55 O=C(O)/C=C\c1cccc(S(=O)(=O)Nc2ncccn2)c1 ZINC000217787099 DD For-Sale Anodyne RHOA 0 42 CC(C)[C@@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217787103 CD For-Sale Unstable CTSC 23 40 CCCCC[C@@H](CN)N[C@@H](CC)CCO ZINC000217787105 BD For-Sale Unstable Q6UB75_PIG 0 43 Oc1ccc2c(c1)CCC[C@@H]2N1CCC[C@@H]2CCCC[C@@H]21 ZINC000217787129 CI For-Sale Unstable DRD5 16 45 Oc1ccc2c(c1)CCC[C@@H]2N1CCC[C@@H]2CCCC[C@@H]21 ZINC000217787129 CI For-Sale Unstable HSD17B1 53 37 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccco2)CC(=O)O4)cc1O ZINC000217787136 HH In-Stock Unstable AKR1B1 0 49 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccco2)CC(=O)O4)cc1O ZINC000217787136 HH In-Stock Unstable CYP1B1 65 36 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccco2)CC(=O)O4)cc1O ZINC000217787136 HH In-Stock Unstable CYP1A1 48 47 O=C1C[C@H](C(F)(F)F)N(C(=O)CS(=O)(=O)c2ccccc2)c2ccccc2N1 ZINC000217787140 HF On-Demand Unstable SFRP1 44 32 CN[C@H]1CC[C@H](C(C)C)C[C@@H]1Cc1cc(F)ccc1F ZINC000217787154 CI For-Sale Unstable DPP4 17 41 CC(C)OC(=O)CO[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217787171 CG For-Sale Unstable SERPINE1 40 40 CC(C)OC(=O)CO[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217787171 CG For-Sale Unstable TRPM8 0 41 Cc1ccc(C)c(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217787182 FF For-Sale Unstable ADAMTS5 31 42 CCCCC[C@H](CN)N[C@@H](CC)CCO ZINC000217787189 BD For-Sale Unstable Q6UB75_PIG 0 43 CC(C)[C@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217787192 CD For-Sale Unstable CTSC 23 40 O=C1C[C@@H](C(F)(F)F)N(C(=O)CS(=O)(=O)c2ccccc2)c2ccccc2N1 ZINC000217787217 HF On-Demand Unstable SFRP1 44 32 Cc1cccc(CNC(=O)N/C=C/c2ccccc2F)c1 ZINC000217787226 CH For-Sale Unstable ANPEP 17 46 CN[C@@H]1CC[C@@H](C(C)C)C[C@@H]1Cc1cc(F)ccc1F ZINC000217787257 CI For-Sale Unstable DPP4 17 41 CC(C)OC(=O)CO[C@H]1C[C@H](C)CC[C@@H]1C(C)C ZINC000217787258 CG On-Demand Unstable SERPINE1 40 40 CC(C)OC(=O)CO[C@H]1C[C@H](C)CC[C@@H]1C(C)C ZINC000217787258 CG On-Demand Unstable TRPM8 0 41 Cc1ccc(C)c(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217787268 FF For-Sale Unstable ADAMTS5 31 42 CCCCC[C@@H](CN)N[C@H](CC)CCO ZINC000217787272 BD For-Sale Unstable Q6UB75_PIG 0 43 COc1cccc(CNC(=O)N/C=C/c2ccccc2F)c1 ZINC000217787328 DG For-Sale Unstable DRD4 43 33 COc1cccc(CNC(=O)N/C=C/c2ccccc2F)c1 ZINC000217787328 DG For-Sale Unstable MMP13 27 42 COc1cccc(CNC(=O)N/C=C/c2ccccc2F)c1 ZINC000217787328 DG For-Sale Unstable ROCK1 38 43 COc1cccc(CNC(=O)N/C=C/c2ccccc2F)c1 ZINC000217787328 DG For-Sale Unstable MTNR1A 49 46 COc1cccc(CNC(=O)N/C=C/c2ccccc2F)c1 ZINC000217787328 DG For-Sale Unstable MTNR1B 48 46 COc1cccc(CNC(=O)N/C=C/c2ccccc2F)c1 ZINC000217787328 DG For-Sale Unstable ROCK2 48 48 COc1cccc(CNC(=O)N/C=C/c2ccccc2F)c1 ZINC000217787328 DG For-Sale Unstable PDS 52 40 CN[C@H]1CC[C@@H](C(C)C)C[C@@H]1Cc1cc(F)ccc1F ZINC000217787342 CI For-Sale Unstable DPP4 17 41 CCCCC[C@H](CN)N[C@H](CC)CCO ZINC000217787362 BD For-Sale Unstable Q6UB75_PIG 0 43 COc1cc(OC)c([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1OC ZINC000217787451 JI In-Stock Unstable AKR1B1 22 46 COc1cc(OC)c([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1OC ZINC000217787451 JI In-Stock Unstable CYP1B1 57 37 COc1cc(OC)c([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1OC ZINC000217787451 JI In-Stock Unstable CYP1A1 45 48 COc1cc(OC)c([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1OC ZINC000217787451 JI In-Stock Unstable CYP1A2 37 48 COc1cc(OC)c([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1OC ZINC000217787531 JI In-Stock Unstable AKR1B1 22 46 COc1cc(OC)c([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1OC ZINC000217787531 JI In-Stock Unstable CYP1B1 57 37 COc1cc(OC)c([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1OC ZINC000217787531 JI In-Stock Unstable CYP1A1 45 48 COc1cc(OC)c([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1OC ZINC000217787531 JI In-Stock Unstable CYP1A2 37 48 COc1cccc(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217787595 FE For-Sale Unstable NPY2R 50 38 COc1cccc(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217787595 FE For-Sale Unstable CHRNA10 31 40 COc1cccc(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217787595 FE For-Sale Unstable ADAMTS5 33 44 FC(F)Oc1ccc2cn[nH]c2c1 ZINC000217787633 AE For-Sale Anodyne TRPA1 25 46 COc1cccc(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217787677 FE For-Sale Unstable NPY2R 50 38 COc1cccc(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217787677 FE For-Sale Unstable CHRNA10 31 40 COc1cccc(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217787677 FE For-Sale Unstable ADAMTS5 33 44 Cc1ccc(N)c(CC(=O)NCC(C)C)c1 ZINC000217787702 BD In-Stock Unstable F3 71 34 NC(=O)CCNS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217787731 CB For-Sale Unstable AKR1C3 35 43 COc1ccccc1S(=O)(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217787790 FE For-Sale Unstable NPY2R 43 38 COc1ccccc1S(=O)(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217787790 FE For-Sale Unstable ADAMTS5 34 43 COc1ccccc1S(=O)(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217787872 FE For-Sale Unstable NPY2R 43 38 COc1ccccc1S(=O)(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217787872 FE For-Sale Unstable ADAMTS5 34 43 O=C(CCCCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCc1cccnc1 ZINC000217787945 JI In-Stock Unstable HTR7 15 49 O=C(CCCCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCc1cccnc1 ZINC000217787945 JI In-Stock Unstable SCN9A 0 44 O=C(CCCCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCc1cccnc1 ZINC000217787945 JI In-Stock Unstable NAMPT 42 36 COc1ccccc1CCNC(=O)N/C=C/c1ccccc1F ZINC000217788018 DG For-Sale Unstable MTNR1A 29 42 COc1ccccc1CCNC(=O)N/C=C/c1ccccc1F ZINC000217788018 DG For-Sale Unstable MTNR1B 21 42 O=C(CCCCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCc1cccnc1 ZINC000217788040 JI In-Stock Unstable HTR7 15 49 O=C(CCCCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCc1cccnc1 ZINC000217788040 JI In-Stock Unstable SCN9A 0 44 O=C(CCCCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCc1cccnc1 ZINC000217788040 JI In-Stock Unstable NAMPT 42 36 CN1CCC[C@@H]1CN(C)[C@@H]1CC[C@@H]1CNC(C)(C)C ZINC000217788111 CE For-Sale Unstable CHRNA10 54 35 COc1cccc(C=O)c1OCCN1CCN(c2ccccc2)CC1 ZINC000217788119 EF In-Stock Unstable HTR1A 116 48 COc1cccc(C=O)c1OCCN1CCN(c2ccccc2)CC1 ZINC000217788119 EF In-Stock Unstable DRD2 83 59 COc1cccc(C=O)c1OCCN1CCN(c2ccccc2)CC1 ZINC000217788119 EF In-Stock Unstable DRD1 37 40 COc1cccc(C=O)c1OCCN1CCN(c2ccccc2)CC1 ZINC000217788119 EF In-Stock Unstable DRD4 56 36 COc1cccc(C=O)c1OCCN1CCN(c2ccccc2)CC1 ZINC000217788119 EF In-Stock Unstable ADRA1D 54 43 COc1cccc(C=O)c1OCCN1CCN(c2ccccc2)CC1 ZINC000217788119 EF In-Stock Unstable HTR2A 70 47 COc1cccc(C=O)c1OCCN1CCN(c2ccccc2)CC1 ZINC000217788119 EF In-Stock Unstable SLC6A4 24 43 COc1cccc(C=O)c1OCCN1CCN(c2ccccc2)CC1 ZINC000217788119 EF In-Stock Unstable ADRA1A 51 41 COc1cccc(C=O)c1OCCN1CCN(c2ccccc2)CC1 ZINC000217788119 EF In-Stock Unstable HRH1 17 40 COc1cccc(C=O)c1OCCN1CCN(c2ccccc2)CC1 ZINC000217788119 EF In-Stock Unstable ADRA1B 50 43 COc1cccc(C=O)c1OCCN1CCN(c2ccccc2)CC1 ZINC000217788119 EF In-Stock Unstable DRD3 76 45 COc1cccc(C=O)c1OCCN1CCN(c2ccccc2)CC1 ZINC000217788119 EF In-Stock Unstable HTR4 15 40 COc1cccc(C=O)c1OCCN1CCN(c2ccccc2)CC1 ZINC000217788119 EF In-Stock Unstable DRD5 30 53 COc1cccc(C=O)c1OCCN1CCN(c2ccccc2)CC1 ZINC000217788119 EF In-Stock Unstable HTR7 107 44 COc1cccc(C=O)c1OCCN1CCN(c2ccccc2)CC1 ZINC000217788119 EF In-Stock Unstable SIGMAR1 20 47 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)Nc3ccc4nc(C)[nH]c4c3)[C@H]21 ZINC000217788167 JH In-Stock Unstable TSHR 66 33 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)Nc3ccc4nc(C)[nH]c4c3)[C@H]21 ZINC000217788167 JH In-Stock Unstable ENPP1 68 34 Cc1cc(F)ccc1S(=O)(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217788172 FF For-Sale Unstable ADAMTS5 30 41 Cc1cc(F)ccc1S(=O)(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217788236 FF For-Sale Unstable ADAMTS5 30 41 C[C@@H]1CCC[C@@H](C)N1CCOc1ccc(C=O)cc1 ZINC000217788246 CG In-Stock Unstable LTA4H 42 38 C[C@@H]1CCC[C@@H](C)N1CCOc1ccc(C=O)cc1 ZINC000217788246 CG In-Stock Unstable HRH3 45 42 C[C@@H]1CCC[C@@H](C)N1CCOc1ccc(C=O)cc1 ZINC000217788246 CG In-Stock Unstable PSMB2 47 39 C[C@@H]1CCC[C@@H](C)N1CCOc1ccc(C=O)cc1 ZINC000217788246 CG In-Stock Unstable PSMB1 41 39 CCCN(CC)S(=O)(=O)c1ccc(/C=C\C(=O)O)cc1Cl ZINC000217788257 EF For-Sale Unstable NR0B2 0 41 COc1ccc([C@@H](CC(=O)Nc2ccc(-c3nc4ccccc4s3)cn2)NC(C)=O)cc1 ZINC000217788260 IJ On-Demand Unstable ACOX1 41 34 COc1ccc([C@@H](CC(=O)Nc2ccc(-c3nc4ccccc4s3)cn2)NC(C)=O)cc1 ZINC000217788260 IJ On-Demand Unstable LUCI_LUCLA 30 43 COc1ccc([C@@H](CC(=O)Nc2ccc(-c3nc4ccccc4s3)cn2)NC(C)=O)cc1 ZINC000217788260 IJ On-Demand Unstable LUCI_PHOPY 15 49 COc1ccc([C@@H](CC(=O)Nc2ccc(-c3nc4ccccc4s3)cn2)NC(C)=O)cc1 ZINC000217788260 IJ On-Demand Unstable LUCI_PHOPE 31 49 COc1ccc([C@@H](CC(=O)Nc2ccc(-c3nc4ccccc4s3)cn2)NC(C)=O)cc1 ZINC000217788260 IJ On-Demand Unstable ETHR 15 50 COc1ccc([C@@H](CC(=O)Nc2ccc(-c3nc4ccccc4s3)cn2)NC(C)=O)cc1 ZINC000217788260 IJ On-Demand Unstable ISPD 0 41 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)Nc3ccc4nc(C)[nH]c4c3)[C@@H]21 ZINC000217788263 JH In-Stock Unstable TSHR 66 33 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)Nc3ccc4nc(C)[nH]c4c3)[C@@H]21 ZINC000217788263 JH In-Stock Unstable ENPP1 68 34 C[C@H]1CCC[C@@H](C)N1CCOc1ccc(C=O)cc1 ZINC000217788328 CG In-Stock Unstable LTA4H 42 38 C[C@H]1CCC[C@@H](C)N1CCOc1ccc(C=O)cc1 ZINC000217788328 CG In-Stock Unstable HRH3 45 42 C[C@H]1CCC[C@@H](C)N1CCOc1ccc(C=O)cc1 ZINC000217788328 CG In-Stock Unstable PSMB2 47 39 C[C@H]1CCC[C@@H](C)N1CCOc1ccc(C=O)cc1 ZINC000217788328 CG In-Stock Unstable PSMB1 41 39 COc1ccc([C@H](CC(=O)Nc2ccc(-c3nc4ccccc4s3)cn2)NC(C)=O)cc1 ZINC000217788341 IJ On-Demand Unstable ACOX1 41 34 COc1ccc([C@H](CC(=O)Nc2ccc(-c3nc4ccccc4s3)cn2)NC(C)=O)cc1 ZINC000217788341 IJ On-Demand Unstable LUCI_LUCLA 30 43 COc1ccc([C@H](CC(=O)Nc2ccc(-c3nc4ccccc4s3)cn2)NC(C)=O)cc1 ZINC000217788341 IJ On-Demand Unstable LUCI_PHOPY 15 49 COc1ccc([C@H](CC(=O)Nc2ccc(-c3nc4ccccc4s3)cn2)NC(C)=O)cc1 ZINC000217788341 IJ On-Demand Unstable LUCI_PHOPE 31 49 COc1ccc([C@H](CC(=O)Nc2ccc(-c3nc4ccccc4s3)cn2)NC(C)=O)cc1 ZINC000217788341 IJ On-Demand Unstable ETHR 15 50 COc1ccc([C@H](CC(=O)Nc2ccc(-c3nc4ccccc4s3)cn2)NC(C)=O)cc1 ZINC000217788341 IJ On-Demand Unstable ISPD 0 41 O=C(O)/C=C\c1cccc(S(=O)(=O)N2CCCSCC2)c1 ZINC000217788344 ED For-Sale Unstable AKR1C3 57 38 Cc1cc(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)ccc1F ZINC000217788353 FF For-Sale Unstable ADAMTS5 33 46 Cc1cc(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)ccc1F ZINC000217788353 FF For-Sale Unstable LEF 58 37 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc3c(c2)OCCO3)CC(=O)O4)cc1O ZINC000217788365 JI In-Stock Unstable AKR1B1 0 46 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc3c(c2)OCCO3)CC(=O)O4)cc1O ZINC000217788365 JI In-Stock Unstable CYP1B1 48 34 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc3c(c2)OCCO3)CC(=O)O4)cc1O ZINC000217788365 JI In-Stock Unstable CYP1A1 37 46 C[C@H](CCc1ccc(O)cc1)N1CCC[C@@H]2CCCC[C@@H]21 ZINC000217788398 CI For-Sale Unstable BIRC2 43 38 C[C@H]1CCC[C@H](C)N1CCOc1ccc(C=O)cc1 ZINC000217788427 CG In-Stock Unstable LTA4H 42 38 C[C@H]1CCC[C@H](C)N1CCOc1ccc(C=O)cc1 ZINC000217788427 CG In-Stock Unstable HRH3 45 42 C[C@H]1CCC[C@H](C)N1CCOc1ccc(C=O)cc1 ZINC000217788427 CG In-Stock Unstable PSMB2 47 39 C[C@H]1CCC[C@H](C)N1CCOc1ccc(C=O)cc1 ZINC000217788427 CG In-Stock Unstable PSMB1 41 39 NS(=O)(=O)CCNS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217788432 EB For-Sale Unstable HDAC8 25 50 NS(=O)(=O)CCNS(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217788432 EB For-Sale Unstable AKR1C3 15 43 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc3c(c2)OCCO3)CC(=O)O4)cc1O ZINC000217788449 JI In-Stock Unstable AKR1B1 0 46 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc3c(c2)OCCO3)CC(=O)O4)cc1O ZINC000217788449 JI In-Stock Unstable CYP1B1 48 34 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc3c(c2)OCCO3)CC(=O)O4)cc1O ZINC000217788449 JI In-Stock Unstable CYP1A1 37 46 Cc1cc(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)ccc1F ZINC000217788450 FF For-Sale Unstable ADAMTS5 33 46 Cc1cc(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)ccc1F ZINC000217788450 FF For-Sale Unstable LEF 58 37 Cc1cccc(CCNC(=O)N/C=C/c2ccccc2F)c1 ZINC000217788452 CH For-Sale Unstable AKR1C3 15 41 CC(=O)N[C@@H](CC(=O)Nc1ccc(-c2nc3ccccc3s2)cn1)c1ccc(Cl)cc1 ZINC000217788453 JK On-Demand Unstable LUCI_LUCLA 32 40 CC(=O)N[C@@H](CC(=O)Nc1ccc(-c2nc3ccccc3s2)cn1)c1ccc(Cl)cc1 ZINC000217788453 JK On-Demand Unstable UTS2 43 33 COc1ccccc1CC(=O)N1[C@@H](C)C[C@@H]2CNC[C@H]21 ZINC000217788454 CD For-Sale Unstable MBTPS1 54 36 C[C@@H]1COCCN1S(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217788512 DD For-Sale Unstable AKR1C3 20 40 NC(=O)NCC(=O)NCc1cc(-c2ccccc2)n[nH]1 ZINC000217788524 CC In-Stock Unstable GSK3B 0 41 NC(=O)NCC(=O)NCc1cc(-c2ccccc2)n[nH]1 ZINC000217788524 CC In-Stock Unstable GSK3A 24 41 CC(=O)N[C@H](CC(=O)Nc1ccc(-c2nc3ccccc3s2)cn1)c1ccc(Cl)cc1 ZINC000217788530 JK On-Demand Unstable LUCI_LUCLA 32 40 CC(=O)N[C@H](CC(=O)Nc1ccc(-c2nc3ccccc3s2)cn1)c1ccc(Cl)cc1 ZINC000217788530 JK On-Demand Unstable UTS2 43 33 COc1ccccc1CC(=O)N1[C@@H]2CNC[C@H]2C[C@H]1C ZINC000217788536 CD For-Sale Unstable MBTPS1 54 36 O=S(=O)(Cc1ccc(F)cc1)NC[C@@H]1CCCN1c1nccs1 ZINC000217788552 FE For-Sale Unstable ADAMTS5 29 40 C[C@@H]1CCC[C@@H](C)N1CCOc1cccc(C=O)c1 ZINC000217788560 CG In-Stock Unstable CHRNA10 57 36 COc1cccc(CCNC(=O)N/C=C/c2ccccc2F)c1 ZINC000217788566 DG For-Sale Unstable DRD4 44 34 COc1cccc(CCNC(=O)N/C=C/c2ccccc2F)c1 ZINC000217788566 DG For-Sale Unstable NQO2 23 40 COc1cccc(CCNC(=O)N/C=C/c2ccccc2F)c1 ZINC000217788566 DG For-Sale Unstable MTNR1A 86 51 COc1cccc(CCNC(=O)N/C=C/c2ccccc2F)c1 ZINC000217788566 DG For-Sale Unstable MTNR1B 80 51 COc1cccc(CCNC(=O)N/C=C/c2ccccc2F)c1 ZINC000217788566 DG For-Sale Unstable CRTM 53 38 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)NCc3ccccn3)[C@H]21 ZINC000217788568 JF In-Stock Unstable SCN9A 0 41 C[C@H]1COCCN1S(=O)(=O)c1cccc(/C=C\C(=O)O)c1 ZINC000217788609 DD For-Sale Unstable AKR1C3 20 40 COc1ccccc1CC(=O)N1[C@@H](C)C[C@H]2CNC[C@H]21 ZINC000217788614 CD For-Sale Unstable MBTPS1 54 36 O=S(=O)(Cc1ccc(F)cc1)NC[C@H]1CCCN1c1nccs1 ZINC000217788630 FE For-Sale Unstable ADAMTS5 29 40 O=C(Nc1ccc(-c2nc3ccccc3s2)cn1)c1ccc(Cl)o1 ZINC000217788644 FJ On-Demand Anodyne LUCI_LUCLA 35 42 C[C@H]1CCC[C@@H](C)N1CCOc1cccc(C=O)c1 ZINC000217788648 CG In-Stock Unstable CHRNA10 57 36 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)NCc3ccccn3)[C@@H]21 ZINC000217788669 JF In-Stock Unstable SCN9A 0 41 COc1ccccc1CC(=O)N1[C@@H]2CNC[C@@H]2C[C@H]1C ZINC000217788706 CD For-Sale Unstable MBTPS1 54 36 C[C@H]1CCC[C@H](C)N1CCOc1cccc(C=O)c1 ZINC000217788729 CG In-Stock Unstable CHRNA10 57 36 CSc1ccc(CCN)cc1Br ZINC000217788737 BF For-Sale Unstable TAAR1 28 44 CCOc1ccccc1C(=O)N1[C@@H](C)C[C@@H]2CNC[C@H]21 ZINC000217788808 CD For-Sale Unstable HCN1 56 39 CCOc1ccccc1C(=O)N1[C@@H](C)C[C@@H]2CNC[C@H]21 ZINC000217788808 CD For-Sale Unstable HCN4 47 36 CCOc1ccccc1C(=O)N1[C@@H]2CNC[C@H]2C[C@H]1C ZINC000217788889 CD For-Sale Unstable HCN1 56 39 CCOc1ccccc1C(=O)N1[C@@H]2CNC[C@H]2C[C@H]1C ZINC000217788889 CD For-Sale Unstable HCN4 47 36 O=C1CSC(=O)N1[C@H]1CCN(S(=O)(=O)c2cccc(C(F)(F)F)c2)C1 ZINC000217788896 GE In-Stock Unstable CACNA1B 55 36 CSc1ccc(Br)cc1CCN ZINC000217788938 BF In-Stock Unstable TAAR1 23 44 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1ccccc1Cl ZINC000217788941 FF For-Sale Unstable ADAMTS5 31 40 O=C1CSC(=O)N1[C@@H]1CCN(S(=O)(=O)c2cccc(C(F)(F)F)c2)C1 ZINC000217788955 GE In-Stock Unstable CACNA1B 55 36 CCOc1ccccc1C(=O)N1[C@@H](C)C[C@H]2CNC[C@H]21 ZINC000217788975 CD For-Sale Unstable HCN1 56 39 CCOc1ccccc1C(=O)N1[C@@H](C)C[C@H]2CNC[C@H]21 ZINC000217788975 CD For-Sale Unstable HCN4 47 36 CN[C@@H]1CC[C@H](C(C)C)C[C@@H]1CCCc1ccccc1 ZINC000217789006 CJ For-Sale Unstable SLC18A2 40 44 COC1CCN(C2CCN(S(=O)(=O)c3ccccc3)CC2)CC1 ZINC000217789021 ED In-Stock Unstable CHRM2 54 56 COC1CCN(C2CCN(S(=O)(=O)c3ccccc3)CC2)CC1 ZINC000217789021 ED In-Stock Unstable HRH1 17 43 COC1CCN(C2CCN(S(=O)(=O)c3ccccc3)CC2)CC1 ZINC000217789021 ED In-Stock Unstable CCR3 32 43 COC1CCN(C2CCN(S(=O)(=O)c3ccccc3)CC2)CC1 ZINC000217789021 ED In-Stock Unstable PKM 15 42 COC1CCN(C2CCN(S(=O)(=O)c3ccccc3)CC2)CC1 ZINC000217789021 ED In-Stock Unstable F13A1 49 35 COC1CCN(C2CCN(S(=O)(=O)c3ccccc3)CC2)CC1 ZINC000217789021 ED In-Stock Unstable L3MBTL3 20 46 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1ccccc1Cl ZINC000217789025 FF For-Sale Unstable ADAMTS5 31 40 CCOc1ccccc1C(=O)N1[C@@H]2CNC[C@@H]2C[C@H]1C ZINC000217789054 CD For-Sale Unstable HCN1 56 39 CCOc1ccccc1C(=O)N1[C@@H]2CNC[C@@H]2C[C@H]1C ZINC000217789054 CD For-Sale Unstable HCN4 47 36 COCCCc1cc(O)nc(-c2cccc(Cl)c2)n1 ZINC000217789070 CG In-Stock Unstable DRTS_PLAFK 18 40 COc1ccc(-c2noc(CCC(=O)Nc3ccc(-c4nc5ccccc5s4)cn3)n2)cc1 ZINC000217789076 JJ On-Demand Unstable HCAR2 37 49 COc1ccc(-c2noc(CCC(=O)Nc3ccc(-c4nc5ccccc5s4)cn3)n2)cc1 ZINC000217789076 JJ On-Demand Unstable LUCI_LUCLA 30 43 COc1ccc(-c2noc(CCC(=O)Nc3ccc(-c4nc5ccccc5s4)cn3)n2)cc1 ZINC000217789076 JJ On-Demand Unstable LUCI_PHOPY 15 47 COc1ccc(-c2noc(CCC(=O)Nc3ccc(-c4nc5ccccc5s4)cn3)n2)cc1 ZINC000217789076 JJ On-Demand Unstable LUCI_PHOPE 37 47 COc1ccc(-c2noc(CCC(=O)Nc3ccc(-c4nc5ccccc5s4)cn3)n2)cc1 ZINC000217789076 JJ On-Demand Unstable ETHR 20 48 CN[C@H]1CC[C@H](C(C)C)C[C@@H]1CCCc1ccccc1 ZINC000217789088 CJ For-Sale Unstable SLC18A2 40 44 O=C(N/C=C/c1ccccc1F)NCCc1ccc(Cl)cc1 ZINC000217789114 DH For-Sale Unstable SLC6A5 16 40 C[C@H](NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1)C(N)=O ZINC000217789140 CB For-Sale Unstable HDAC8 15 47 C[C@H](NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1)C(N)=O ZINC000217789140 CB For-Sale Unstable LEF 19 43 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1ccc(F)c(F)c1 ZINC000217789146 FE For-Sale Unstable ADAMTS5 33 42 CN[C@@H]1CC[C@@H](C(C)C)C[C@@H]1CCCc1ccccc1 ZINC000217789169 CJ For-Sale Unstable SLC18A2 40 44 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](CC(C)C)C(=O)NCCO)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217789190 KF In-Stock Unstable TUBA1A 19 70 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](CC(C)C)C(=O)NCCO)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217789190 KF In-Stock Unstable TPPP 0 66 C[C@@H](NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1)C(N)=O ZINC000217789216 CB For-Sale Unstable HDAC8 15 47 C[C@@H](NS(=O)(=O)c1cccc(/C=C\C(=O)O)c1)C(N)=O ZINC000217789216 CB For-Sale Unstable LEF 19 43 Cc1cc2ccnc(Cl)c2n1S(=O)(=O)c1ccccc1 ZINC000217789222 DG For-Sale Unstable HTR6 27 42 Cc1cc2ccnc(Cl)c2n1S(=O)(=O)c1ccccc1 ZINC000217789222 DG For-Sale Unstable ALDH3A1 42 40 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1ccc(F)c(F)c1 ZINC000217789224 FE For-Sale Unstable ADAMTS5 33 42 CN[C@H]1CC[C@@H](C(C)C)C[C@@H]1CCCc1ccccc1 ZINC000217789243 CJ For-Sale Unstable SLC18A2 40 44 O=C(Cc1ccc(O)c(Cl)c1)NC[C@@]1(O)CCNC1 ZINC000217789248 CC In-Stock Unstable NCE103 35 50 O=C(Cc1ccc(O)c(Cl)c1)NC[C@@]1(O)CCNC1 ZINC000217789248 CC In-Stock Unstable P96878_MYCTU 23 50 O=C(Cc1ccc(O)c(Cl)c1)NC[C@@]1(O)CCNC1 ZINC000217789248 CC In-Stock Unstable CAN2 0 50 COCCCc1cc(O)nc(-c2ccco2)n1 ZINC000217789282 BE In-Stock Unstable ADORA1 24 41 COCCCc1cc(O)nc(-c2ccco2)n1 ZINC000217789282 BE In-Stock Unstable ADORA2A 34 41 COCCCc1cc(O)nc(-c2ccco2)n1 ZINC000217789282 BE In-Stock Unstable ADORA3 0 41 CC(C)[C@H](N[C@@H]1CCCC[C@@H]1C)c1ccc(Cl)cc1 ZINC000217789285 CK For-Sale Unstable SLC6A1 0 44 Cc1cc(S(=O)(=O)N[C@@H](C)C(N)=O)ccc1/C=C\C(=O)O ZINC000217789301 DC For-Sale Unstable LEF 60 38 COc1cc([C@H](C)N2CCC[C@@H]3CCCC[C@@H]32)ccc1O ZINC000217789302 CI For-Sale Unstable PNLIP 0 46 COc1cc([C@H](C)N2CCC[C@@H]3CCCC[C@@H]32)ccc1O ZINC000217789302 CI For-Sale Unstable N1L 0 47 COc1cc([C@H](C)N2CCC[C@@H]3CCCC[C@@H]32)ccc1O ZINC000217789302 CI For-Sale Unstable SLC22A3 0 43 COC(=O)C[C@H](c1c(O)c2ccccc2oc1=O)c1coc2ccccc2c1=O ZINC000217789308 GG In-Stock Unstable NQO1 54 54 O=C(Cc1ccc(O)c(Cl)c1)NC[C@]1(O)CCNC1 ZINC000217789337 CC In-Stock Unstable NCE103 35 50 O=C(Cc1ccc(O)c(Cl)c1)NC[C@]1(O)CCNC1 ZINC000217789337 CC In-Stock Unstable P96878_MYCTU 23 50 O=C(Cc1ccc(O)c(Cl)c1)NC[C@]1(O)CCNC1 ZINC000217789337 CC In-Stock Unstable CAN2 0 50 O=C(Nc1nccc2[nH]ccc12)C1CC1 ZINC000217789340 BD For-Sale Unstable GSK3B 19 42 O=C(Nc1nccc2[nH]ccc12)C1CC1 ZINC000217789340 BD For-Sale Unstable GSK3A 34 42 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1cc(F)ccc1F ZINC000217789350 FE For-Sale Unstable ADAMTS5 30 41 CC(C)[C@H](N[C@H]1CCCC[C@@H]1C)c1ccc(Cl)cc1 ZINC000217789371 CK For-Sale Unstable SLC6A1 0 44 Cc1cc(S(=O)(=O)N[C@H](C)C(N)=O)ccc1/C=C\C(=O)O ZINC000217789383 DC For-Sale Unstable LEF 60 38 COC(=O)C[C@@H](c1c(O)c2ccccc2oc1=O)c1coc2ccccc2c1=O ZINC000217789387 GG In-Stock Unstable NQO1 54 54 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1cc(F)ccc1F ZINC000217789426 FE For-Sale Unstable ADAMTS5 30 41 O=C(Nc1ccc(-c2nc3ccccc3s2)cn1)C1CCN(C(=O)c2ccc(F)cc2F)CC1 ZINC000217789430 JK On-Demand Unstable NPY5R 25 44 c1ccc([C@H]2CCCC[C@H]2N[C@H]2CCN(C3CC3)C2)cc1 ZINC000217789441 CH For-Sale Unstable SLC18A3 15 44 COc1ccccc1CN1C(=O)N[C@@H](CC(=O)NC[C@@H]2CCCN3CCCC[C@H]23)C1=O ZINC000217789500 ID In-Stock Unstable MBTPS1 52 36 COC(=O)c1ccc(S(=O)(=O)N2CC[C@H](N3C(=O)CSC3=O)C2)cc1 ZINC000217789501 GC In-Stock Unstable TGM2 48 35 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1c(F)cccc1F ZINC000217789544 FE For-Sale Unstable ADAMTS5 30 40 COC(=O)c1ccc(S(=O)(=O)N2CC[C@@H](N3C(=O)CSC3=O)C2)cc1 ZINC000217789588 GC In-Stock Unstable TGM2 48 35 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1c(F)cccc1F ZINC000217789610 FE For-Sale Unstable ADAMTS5 30 40 COc1ccc(OC)c2[nH]c(C(=O)NC[C@@H]3CCCN4CCCC[C@H]34)cc12 ZINC000217789628 FG In-Stock Unstable DRD3 0 40 COc1ccc(OC)c2[nH]c(C(=O)NC[C@@H]3CCCN4CCCC[C@H]34)cc12 ZINC000217789628 FG In-Stock Unstable ACKR3 61 31 O=C(Nc1ccc(-c2nc3ccccc3s2)cn1)c1cccc(N2CCCS2(=O)=O)c1 ZINC000217789644 JI On-Demand Unstable LUCI_LUCLA 35 41 COc1cc(OC)c2ccc(=O)oc2c1OC/C=C(/C)CCC=C(C)C ZINC000217789736 FJ For-Sale Unstable MAOA 16 55 COc1cc(OC)c2ccc(=O)oc2c1OC/C=C(/C)CCC=C(C)C ZINC000217789736 FJ For-Sale Unstable CA7 27 53 COc1cc(OC)c2ccc(=O)oc2c1OC/C=C(/C)CCC=C(C)C ZINC000217789736 FJ For-Sale Unstable PDE4D 22 60 COc1cc(OC)c2ccc(=O)oc2c1OC/C=C(/C)CCC=C(C)C ZINC000217789736 FJ For-Sale Unstable TRPA1 23 40 CCOc1cc(C=O)ccc1OCCN1CCN(c2ccccc2)CC1 ZINC000217789737 FG In-Stock Unstable HTR1A 46 45 CCOc1cc(C=O)ccc1OCCN1CCN(c2ccccc2)CC1 ZINC000217789737 FG In-Stock Unstable DRD2 33 49 CCOc1cc(C=O)ccc1OCCN1CCN(c2ccccc2)CC1 ZINC000217789737 FG In-Stock Unstable DRD1 23 53 CCOc1cc(C=O)ccc1OCCN1CCN(c2ccccc2)CC1 ZINC000217789737 FG In-Stock Unstable HTR2A 33 42 CCOc1cc(C=O)ccc1OCCN1CCN(c2ccccc2)CC1 ZINC000217789737 FG In-Stock Unstable DRD3 37 45 CCOc1cc(C=O)ccc1OCCN1CCN(c2ccccc2)CC1 ZINC000217789737 FG In-Stock Unstable DRD5 21 53 CCOc1cc(C=O)ccc1OCCN1CCN(c2ccccc2)CC1 ZINC000217789737 FG In-Stock Unstable HTR7 49 42 CCOc1cc(C=O)ccc1OCCN1CCN(c2ccccc2)CC1 ZINC000217789737 FG In-Stock Unstable SIGMAR1 15 49 CCOc1cc(C=O)ccc1OCCN1CCN(c2ccccc2)CC1 ZINC000217789737 FG In-Stock Unstable ABCB1 0 41 CCOc1cc(C=O)ccc1OCCN1CCN(c2ccccc2)CC1 ZINC000217789737 FG In-Stock Unstable ASF1A 0 40 COc1cc(-c2coc3ccc(OCc4ccc(C(=O)OC(C)C)o4)cc23)cc(OC)c1OC ZINC000217789739 JK In-Stock Unstable ALDH2 69 34 CCC(=O)Nc1nccc2[nH]ccc12 ZINC000217789787 AD For-Sale Unstable GSK3B 16 42 CCC(=O)Nc1nccc2[nH]ccc12 ZINC000217789787 AD For-Sale Unstable GSK3A 19 42 CCC(=O)Nc1nccc2[nH]ccc12 ZINC000217789787 AD For-Sale Unstable HPGDS 20 47 CCO[C@@H]1C[C@@H](N[C@@H](C(=O)OC)c2ccccc2)C1(C)C ZINC000217789799 CF For-Sale Unstable TIMP3 57 33 O=C(N/C=C/c1ccccc1F)Nc1ccc(Cl)cn1 ZINC000217789818 CH For-Sale Anodyne LUCI_LUCLA 33 43 CCO[C@H]1C[C@@H](N[C@@H](C(=O)OC)c2ccccc2)C1(C)C ZINC000217789877 CF For-Sale Unstable TIMP3 57 33 CC(=O)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)cc1 ZINC000217789911 FE For-Sale Unstable ADAMTS5 34 43 O=C(N/C=C/c1ccccc1F)Nc1cc(Cl)ccn1 ZINC000217789927 CH For-Sale Anodyne TYK2 46 36 COC(=O)C[C@H](c1ccc(O)c(OC)c1)c1oc(CN2CCCCC2)cc(=O)c1O ZINC000217789950 HF In-Stock Unstable RORC 42 33 O=C(Cn1nnc(-c2ccc(F)cc2)n1)N1CCN(c2cnccn2)CC1 ZINC000217789956 FC In-Stock Unstable SCARB1 27 40 O=C(Cn1nnc(-c2ccc(F)cc2)n1)N1CCN(c2cnccn2)CC1 ZINC000217789956 FC In-Stock Unstable SLC6A7 0 49 O=C(Cc1ccccc1)NCCC(=O)Nc1ccc(-c2nc3ccccc3s2)cn1 ZINC000217789957 HI On-Demand Unstable CSNK1D 20 49 CCO[C@@H]1C[C@H](N[C@@H](C(=O)OC)c2ccccc2)C1(C)C ZINC000217789970 CF For-Sale Unstable TIMP3 57 33 CC(=O)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)cc1 ZINC000217789985 FE For-Sale Unstable ADAMTS5 34 43 C[C@@H](c1cccc(Cl)c1)N(C)C[C@@H](O)c1cccc(N)c1 ZINC000217790033 DH For-Sale Unstable ADRB1 22 41 C[C@@H](c1cccc(Cl)c1)N(C)C[C@@H](O)c1cccc(N)c1 ZINC000217790033 DH For-Sale Unstable ADRB3 33 41 C[C@@H](c1cccc(Cl)c1)N(C)C[C@@H](O)c1cccc(N)c1 ZINC000217790033 DH For-Sale Unstable AOC3 34 45 COC(=O)C[C@@H](c1ccc(O)c(OC)c1)c1oc(CN2CCCCC2)cc(=O)c1O ZINC000217790035 HF In-Stock Unstable RORC 42 33 CCO[C@H]1C[C@H](N[C@@H](C(=O)OC)c2ccccc2)C1(C)C ZINC000217790058 CF For-Sale Unstable TIMP3 57 33 CC(C)[C@H](NC1[C@@H](C)CCC[C@@H]1C)c1ccc(Cl)cc1 ZINC000217790062 CK For-Sale Unstable SLC6A1 0 42 CC(=O)c1cccc(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217790102 FE In-Stock Unstable ADAMTS5 32 44 C[C@H](c1cccc(Cl)c1)N(C)C[C@@H](O)c1cccc(N)c1 ZINC000217790105 DH For-Sale Unstable ADRB1 22 41 C[C@H](c1cccc(Cl)c1)N(C)C[C@@H](O)c1cccc(N)c1 ZINC000217790105 DH For-Sale Unstable ADRB3 33 41 C[C@H](c1cccc(Cl)c1)N(C)C[C@@H](O)c1cccc(N)c1 ZINC000217790105 DH For-Sale Unstable AOC3 34 45 COc1cccc(C=O)c1OCCCN1CCN(c2ccccc2)CC1 ZINC000217790138 FG In-Stock Unstable HTR1A 142 53 COc1cccc(C=O)c1OCCCN1CCN(c2ccccc2)CC1 ZINC000217790138 FG In-Stock Unstable ADRA2A 17 40 COc1cccc(C=O)c1OCCCN1CCN(c2ccccc2)CC1 ZINC000217790138 FG In-Stock Unstable DRD2 101 58 COc1cccc(C=O)c1OCCCN1CCN(c2ccccc2)CC1 ZINC000217790138 FG In-Stock Unstable DRD1 46 43 COc1cccc(C=O)c1OCCCN1CCN(c2ccccc2)CC1 ZINC000217790138 FG In-Stock Unstable DRD4 60 44 COc1cccc(C=O)c1OCCCN1CCN(c2ccccc2)CC1 ZINC000217790138 FG In-Stock Unstable ADRA1D 66 47 COc1cccc(C=O)c1OCCCN1CCN(c2ccccc2)CC1 ZINC000217790138 FG In-Stock Unstable HTR1B 23 40 COc1cccc(C=O)c1OCCCN1CCN(c2ccccc2)CC1 ZINC000217790138 FG In-Stock Unstable HTR2A 88 49 COc1cccc(C=O)c1OCCCN1CCN(c2ccccc2)CC1 ZINC000217790138 FG In-Stock Unstable HTR2C 34 43 COc1cccc(C=O)c1OCCCN1CCN(c2ccccc2)CC1 ZINC000217790138 FG In-Stock Unstable SLC6A4 24 40 COc1cccc(C=O)c1OCCCN1CCN(c2ccccc2)CC1 ZINC000217790138 FG In-Stock Unstable ADRA1A 60 47 COc1cccc(C=O)c1OCCCN1CCN(c2ccccc2)CC1 ZINC000217790138 FG In-Stock Unstable ADRA1B 56 47 COc1cccc(C=O)c1OCCCN1CCN(c2ccccc2)CC1 ZINC000217790138 FG In-Stock Unstable DRD3 92 53 COc1cccc(C=O)c1OCCCN1CCN(c2ccccc2)CC1 ZINC000217790138 FG In-Stock Unstable KCNH2 0 47 COc1cccc(C=O)c1OCCCN1CCN(c2ccccc2)CC1 ZINC000217790138 FG In-Stock Unstable DRD5 33 46 COc1cccc(C=O)c1OCCCN1CCN(c2ccccc2)CC1 ZINC000217790138 FG In-Stock Unstable HTR7 125 48 COc1cccc(C=O)c1OCCCN1CCN(c2ccccc2)CC1 ZINC000217790138 FG In-Stock Unstable SIGMAR1 31 58 COc1cccc(C=O)c1OCCCN1CCN(c2ccccc2)CC1 ZINC000217790138 FG In-Stock Unstable HTR6 0 41 COc1cccc(C=O)c1OCCCN1CCN(c2ccccc2)CC1 ZINC000217790138 FG In-Stock Unstable ABCB1 28 40 COc1cccc(C=O)c1OCCCN1CCN(c2ccccc2)CC1 ZINC000217790138 FG In-Stock Unstable SLC29A2 0 40 COc1cccc(C=O)c1OCCCN1CCN(c2ccccc2)CC1 ZINC000217790138 FG In-Stock Unstable ALPHA-1A 0 42 CC(C)[C@H](NC1[C@@H](C)CCC[C@H]1C)c1ccc(Cl)cc1 ZINC000217790148 CK For-Sale Unstable SLC6A1 0 42 O=C(N/C=C/c1ccccc1F)NCCCc1ccccc1 ZINC000217790149 CH For-Sale Unstable MTNR1B 27 41 O=C(N/C=C/c1ccccc1F)NCCCc1ccccc1 ZINC000217790149 CH For-Sale Unstable AMP1_PLAFQ 29 42 O=C(N/C=C/c1ccccc1F)NCCCc1ccccc1 ZINC000217790149 CH For-Sale Unstable POLG_WNV 41 30 COC(=O)[C@@H]1CC[C@@H]1c1ccccc1 ZINC000217790164 AE In-Stock Unstable SLC6A2 16 53 COC(=O)[C@@H]1CC[C@@H]1c1ccccc1 ZINC000217790164 AE In-Stock Unstable SLC6A1 165 56 COC(=O)[C@@H]1CC[C@@H]1c1ccccc1 ZINC000217790164 AE In-Stock Unstable SLC6A4 33 55 COC(=O)[C@@H]1CC[C@@H]1c1ccccc1 ZINC000217790164 AE In-Stock Unstable SLC6A3 64 55 COC(=O)[C@@H]1CC[C@@H]1c1ccccc1 ZINC000217790164 AE In-Stock Unstable EPHX2 17 42 COC(=O)[C@@H]1CC[C@@H]1c1ccccc1 ZINC000217790164 AE In-Stock Unstable GPR88 84 36 CC(=O)c1cccc(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217790172 FE In-Stock Unstable ADAMTS5 32 44 C[C@@H](c1cccc(Cl)c1)N(C)C[C@@H](O)c1ccccc1N ZINC000217790199 DH For-Sale Unstable AOC3 23 42 COC(=O)[C@H]1CC[C@@H]1c1ccccc1 ZINC000217790245 AE In-Stock Unstable SLC6A2 16 53 COC(=O)[C@H]1CC[C@@H]1c1ccccc1 ZINC000217790245 AE In-Stock Unstable SLC6A1 165 56 COC(=O)[C@H]1CC[C@@H]1c1ccccc1 ZINC000217790245 AE In-Stock Unstable SLC6A4 33 55 COC(=O)[C@H]1CC[C@@H]1c1ccccc1 ZINC000217790245 AE In-Stock Unstable SLC6A3 64 55 COC(=O)[C@H]1CC[C@@H]1c1ccccc1 ZINC000217790245 AE In-Stock Unstable EPHX2 17 42 COC(=O)[C@H]1CC[C@@H]1c1ccccc1 ZINC000217790245 AE In-Stock Unstable GPR88 84 36 O=C(N/C=C/c1ccccc1F)NCCCCc1ccccc1 ZINC000217790246 DI For-Sale Unstable LIPC 0 51 O=C(N/C=C/c1ccccc1F)NCCCCc1ccccc1 ZINC000217790246 DI For-Sale Unstable MTNR1B 23 40 O=C(N/C=C/c1ccccc1F)NCCCCc1ccccc1 ZINC000217790246 DI For-Sale Unstable FAAH 34 41 O=C(N/C=C/c1ccccc1F)NCCCCc1ccccc1 ZINC000217790246 DI For-Sale Unstable SCN5A 0 43 O=C(N/C=C/c1ccccc1F)NCCCCc1ccccc1 ZINC000217790246 DI For-Sale Unstable SLC6A5 25 40 O=C(N/C=C/c1ccccc1F)NCCCCc1ccccc1 ZINC000217790246 DI For-Sale Unstable CES1 45 38 O=C(N/C=C/c1ccccc1F)NCCCCc1ccccc1 ZINC000217790246 DI For-Sale Unstable AMP1_PLAFQ 27 47 O=C(N/C=C/c1ccccc1F)NCCCCc1ccccc1 ZINC000217790246 DI For-Sale Unstable POLG_WNV 41 30 C[C@@H]1CCC[C@@H](C)N1CCCOc1ccc(C=O)cc1 ZINC000217790252 CH In-Stock Unstable HTR3A 24 42 C[C@@H]1CCC[C@@H](C)N1CCCOc1ccc(C=O)cc1 ZINC000217790252 CH In-Stock Unstable LTA4H 27 57 C[C@@H]1CCC[C@@H](C)N1CCCOc1ccc(C=O)cc1 ZINC000217790252 CH In-Stock Unstable HRH3 66 47 C[C@H](c1cccc(Cl)c1)N(C)C[C@@H](O)c1ccccc1N ZINC000217790284 DH For-Sale Unstable AOC3 23 42 CCCc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)cc1 ZINC000217790292 FG For-Sale Unstable ADAMTS5 40 56 C[C@H]1CCC[C@@H](C)N1CCCOc1ccc(C=O)cc1 ZINC000217790314 CH In-Stock Unstable HTR3A 24 42 C[C@H]1CCC[C@@H](C)N1CCCOc1ccc(C=O)cc1 ZINC000217790314 CH In-Stock Unstable LTA4H 27 57 C[C@H]1CCC[C@@H](C)N1CCCOc1ccc(C=O)cc1 ZINC000217790314 CH In-Stock Unstable HRH3 66 47 COC(=O)[C@@H]1CC[C@H]1c1ccccc1 ZINC000217790317 AE In-Stock Unstable SLC6A2 16 53 COC(=O)[C@@H]1CC[C@H]1c1ccccc1 ZINC000217790317 AE In-Stock Unstable SLC6A1 165 56 COC(=O)[C@@H]1CC[C@H]1c1ccccc1 ZINC000217790317 AE In-Stock Unstable SLC6A4 33 55 COC(=O)[C@@H]1CC[C@H]1c1ccccc1 ZINC000217790317 AE In-Stock Unstable SLC6A3 64 55 COC(=O)[C@@H]1CC[C@H]1c1ccccc1 ZINC000217790317 AE In-Stock Unstable EPHX2 17 42 COC(=O)[C@@H]1CC[C@H]1c1ccccc1 ZINC000217790317 AE In-Stock Unstable GPR88 84 36 COC(=O)C[C@@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(OC)c(OC)c1 ZINC000217790334 GG In-Stock Unstable TNF 25 49 CCCc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)cc1 ZINC000217790370 FG For-Sale Unstable ADAMTS5 40 56 C[C@@H](c1cccc(Cl)c1)N(C)C[C@@H](O)c1ccc(N)cc1 ZINC000217790376 DH For-Sale Unstable AOC3 33 45 O=C(COc1cccc(Cl)c1)N[C@@H]1C[C@@H]2OCC[C@@H]21 ZINC000217790386 CE In-Stock Unstable TRAR 30 42 C[C@H]1CCC[C@H](C)N1CCCOc1ccc(C=O)cc1 ZINC000217790399 CH In-Stock Unstable HTR3A 24 42 C[C@H]1CCC[C@H](C)N1CCCOc1ccc(C=O)cc1 ZINC000217790399 CH In-Stock Unstable LTA4H 27 57 C[C@H]1CCC[C@H](C)N1CCCOc1ccc(C=O)cc1 ZINC000217790399 CH In-Stock Unstable HRH3 66 47 COC(=O)[C@H]1CC[C@H]1c1ccccc1 ZINC000217790407 AE In-Stock Unstable SLC6A2 16 53 COC(=O)[C@H]1CC[C@H]1c1ccccc1 ZINC000217790407 AE In-Stock Unstable SLC6A1 165 56 COC(=O)[C@H]1CC[C@H]1c1ccccc1 ZINC000217790407 AE In-Stock Unstable SLC6A4 33 55 COC(=O)[C@H]1CC[C@H]1c1ccccc1 ZINC000217790407 AE In-Stock Unstable SLC6A3 64 55 COC(=O)[C@H]1CC[C@H]1c1ccccc1 ZINC000217790407 AE In-Stock Unstable EPHX2 17 42 COC(=O)[C@H]1CC[C@H]1c1ccccc1 ZINC000217790407 AE In-Stock Unstable GPR88 84 36 COC(=O)C[C@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(OC)c(OC)c1 ZINC000217790411 GG In-Stock Unstable TNF 25 49 C[C@H](c1cccc(Cl)c1)N(C)C[C@@H](O)c1ccc(N)cc1 ZINC000217790462 DH For-Sale Unstable AOC3 33 45 COC1CCN(C2CCN(S(=O)(=O)c3ccc(F)cc3C)CC2)CC1 ZINC000217790490 FE In-Stock Unstable EPHX2 19 51 CC(C)Cn1c([C@@H]2CCCN2C(=O)CCCC[C@H]2CCSS2)nc2ccccc21 ZINC000217790519 IK In-Stock Unstable Q7YY07_CRYPV 57 32 O=C(Nc1cc2cc[nH]c2cn1)C1CC1 ZINC000217790535 BD On-Demand Unstable ADORA2B 16 43 O=C(Nc1cc2cc[nH]c2cn1)C1CC1 ZINC000217790535 BD On-Demand Unstable GSK3B 23 52 O=C(Nc1cc2cc[nH]c2cn1)C1CC1 ZINC000217790535 BD On-Demand Unstable GSK3A 28 52 O=C(Nc1cc2cc[nH]c2cn1)C1CC1 ZINC000217790535 BD On-Demand Unstable TYK2 54 40 C[C@@H]1CCC[C@@H](C)N1CCCOc1cccc(C=O)c1 ZINC000217790540 CH In-Stock Unstable HRH3 45 41 C[C@@H]1CCC[C@@H](C)N1CCCOc1cccc(C=O)c1 ZINC000217790540 CH In-Stock Unstable CHRNA10 43 35 CC(C)Cn1c([C@@H]2CCCN2C(=O)CCCC[C@@H]2CCSS2)nc2ccccc21 ZINC000217790585 IK In-Stock Unstable Q7YY07_CRYPV 57 32 COC1CCN(C2CCN(S(=O)(=O)c3ccc(F)c(C)c3)CC2)CC1 ZINC000217790604 FE In-Stock Unstable CHRM2 49 41 COC1CCN(C2CCN(S(=O)(=O)c3ccc(F)c(C)c3)CC2)CC1 ZINC000217790604 FE In-Stock Unstable CCR3 26 43 C[C@H]1CCC[C@@H](C)N1CCCOc1cccc(C=O)c1 ZINC000217790612 CH In-Stock Unstable HRH3 45 41 C[C@H]1CCC[C@@H](C)N1CCCOc1cccc(C=O)c1 ZINC000217790612 CH In-Stock Unstable CHRNA10 43 35 Cc1cc(C)c(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)cc1C ZINC000217790665 FG For-Sale Unstable ADAMTS5 30 42 CC[C@@H](C)[C@@H](N)C(=O)N[C@H](c1ccc(Cl)cc1)C(C)C ZINC000217790686 CH For-Sale Unstable PRCP 17 62 CC[C@@H](C)[C@@H](N)C(=O)N[C@H](c1ccc(Cl)cc1)C(C)C ZINC000217790686 CH For-Sale Unstable UTS2 41 32 COC(=O)C[C@H](c1ccc(OC)c(OC)c1OC)c1c(Cc2ccc3c(c2)CCC(C)(C)O3)[nH][nH]c1=O ZINC000217790690 KI In-Stock Unstable NDUFA4 0 40 C[C@H]1CCC[C@H](C)N1CCCOc1cccc(C=O)c1 ZINC000217790693 CH In-Stock Unstable HRH3 45 41 C[C@H]1CCC[C@H](C)N1CCCOc1cccc(C=O)c1 ZINC000217790693 CH In-Stock Unstable CHRNA10 43 35 O=C(N/C=C/c1ccccc1F)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217790698 GF For-Sale Unstable TGM2 73 39 O=C(N/C=C/c1ccccc1F)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217790698 GF For-Sale Unstable F13A1 88 39 Cc1cc(C)c(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)cc1C ZINC000217790743 FG For-Sale Unstable ADAMTS5 30 42 CCN(C)C(=O)CNC(=O)c1ncccc1C(=O)O ZINC000217790757 CB For-Sale Unstable EGLN1 0 41 CCN(C)C(=O)CNC(=O)c1ncccc1C(=O)O ZINC000217790757 CB For-Sale Unstable OSIGBA0132E09-OSIGBA0108L24.11 0 40 CC[C@H](C)[C@@H](N)C(=O)N[C@H](c1ccc(Cl)cc1)C(C)C ZINC000217790764 CH For-Sale Unstable PRCP 17 62 CC[C@H](C)[C@@H](N)C(=O)N[C@H](c1ccc(Cl)cc1)C(C)C ZINC000217790764 CH For-Sale Unstable UTS2 41 32 COc1ccc(N2C[C@H](C(=O)N3CCC(N4C(=O)CSC4=O)CC3)CC2=O)cc1 ZINC000217790777 HD In-Stock Unstable CHRM2 20 40 COC(=O)C[C@@H](c1ccc(OC)c(OC)c1OC)c1c(Cc2ccc3c(c2)CCC(C)(C)O3)[nH][nH]c1=O ZINC000217790782 KI In-Stock Unstable NDUFA4 0 40 Cc1ccc(S(=O)(=O)N2CCN(C(=O)N/C=C/c3ccccc3F)CC2)cc1 ZINC000217790808 HF For-Sale Unstable TGM2 73 38 Cc1ccc(S(=O)(=O)N2CCN(C(=O)N/C=C/c3ccccc3F)CC2)cc1 ZINC000217790808 HF For-Sale Unstable F13A1 87 38 CC[C@H]1CCCN1[C@H](CC)c1ccc(O)cc1 ZINC000217790831 BH For-Sale Unstable CYP17A1 0 42 COc1ccc(N2C[C@@H](C(=O)N3CCC(N4C(=O)CSC4=O)CC3)CC2=O)cc1 ZINC000217790843 HD In-Stock Unstable CHRM2 20 40 CC(C)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)cc1 ZINC000217790857 FG For-Sale Unstable ADAMTS5 34 43 CC(C)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)cc1 ZINC000217790940 FG For-Sale Unstable ADAMTS5 34 43 O=C(c1ccc2noc(-c3ccccc3)c2c1)N1CCC(N2C(=O)CSC2=O)CC1 ZINC000217791059 HH In-Stock Unstable AVPR1A 22 40 O=C(c1ccc2noc(-c3ccccc3)c2c1)N1CCC(N2C(=O)CSC2=O)CC1 ZINC000217791059 HH In-Stock Unstable L3MBTL1 0 41 O=C(c1ccc2noc(-c3ccccc3)c2c1)N1CCC(N2C(=O)CSC2=O)CC1 ZINC000217791059 HH In-Stock Unstable L3MBTL3 56 41 CCOc1ccccc1S(=O)(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217791061 FE For-Sale Unstable ADAMTS5 33 41 COc1cc([C@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc2c1OCO2 ZINC000217791087 KH In-Stock Unstable RORC 0 42 COc1cc(C=O)ccc1OCCCN1[C@@H](C)CCC[C@@H]1C ZINC000217791105 DH In-Stock Unstable EHMT2 47 32 COC1CCN(C2CCN(S(=O)(=O)c3ccc(F)c(F)c3)CC2)CC1 ZINC000217791127 FE In-Stock Unstable CHRM2 48 42 COC1CCN(C2CCN(S(=O)(=O)c3ccc(F)c(F)c3)CC2)CC1 ZINC000217791127 FE In-Stock Unstable CCR3 26 46 COC1CCN(C2CCN(S(=O)(=O)c3ccc(F)c(F)c3)CC2)CC1 ZINC000217791127 FE In-Stock Unstable APP 17 42 COC1CCN(C2CCN(S(=O)(=O)c3ccc(F)c(F)c3)CC2)CC1 ZINC000217791127 FE In-Stock Unstable PKM 41 38 CCOc1ccccc1S(=O)(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217791147 FE For-Sale Unstable ADAMTS5 33 41 COCC[C@@H](NC(=O)NC[C@@H]1CN(C)CCO1)C(=O)O ZINC000217791171 CB For-Sale Unstable NPPA 40 32 Cc1c(C(=O)N2CCC(N3C(=O)CSC3=O)CC2)cnn1-c1ccccc1 ZINC000217791172 GE In-Stock Unstable SLC9A2 0 44 C[C@@H](c1cccc(Cl)c1)N(C)[C@H](c1ccccc1)[C@@H](C)N ZINC000217791175 DI For-Sale Unstable OPRL1 0 43 C[C@@H](c1cccc(Cl)c1)N(C)[C@H](c1ccccc1)[C@@H](C)N ZINC000217791175 DI For-Sale Unstable AOC3 19 44 COc1cc([C@@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc2c1OCO2 ZINC000217791187 KH In-Stock Unstable RORC 0 42 COc1cc(C=O)ccc1OCCCN1[C@@H](C)CCC[C@H]1C ZINC000217791198 DH In-Stock Unstable EHMT2 47 32 COCC[C@@H](NC(=O)NC[C@H]1CN(C)CCO1)C(=O)O ZINC000217791252 CB For-Sale Unstable NPPA 40 32 COc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)cc1C ZINC000217791261 FE For-Sale Unstable ADAMTS5 32 47 C[C@H](N)[C@@H](c1ccccc1)N(C)[C@@H](C)c1cccc(Cl)c1 ZINC000217791266 DI For-Sale Unstable OPRL1 0 43 C[C@H](N)[C@@H](c1ccccc1)N(C)[C@@H](C)c1cccc(Cl)c1 ZINC000217791266 DI For-Sale Unstable AOC3 19 44 COc1cc(C=O)ccc1OCCCN1[C@H](C)CCC[C@H]1C ZINC000217791281 DH In-Stock Unstable EHMT2 47 32 O=C(c1ccc(-c2ccccc2)cc1)N1CCC(N2C(=O)CSC2=O)CC1 ZINC000217791282 GH In-Stock Unstable AVPR1A 33 50 O=C(c1ccc(-c2ccccc2)cc1)N1CCC(N2C(=O)CSC2=O)CC1 ZINC000217791282 GH In-Stock Unstable L3MBTL3 97 45 CCN(C)C(=O)CNC(=O)c1ccccc1C(=O)O ZINC000217791302 CC For-Sale Unstable ECR 40 37 CCN(C)C(=O)CNC(=O)c1ccccc1C(=O)O ZINC000217791302 CC For-Sale Unstable HCN1 51 32 C[C@H]1CCCN1[C@H](C)Cc1ccc(O)cc1 ZINC000217791316 BF For-Sale Unstable OPRM1 25 40 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)cc1C ZINC000217791345 FE For-Sale Unstable ADAMTS5 32 47 C[C@H](N)[C@H](c1ccccc1)N(C)[C@@H](C)c1cccc(Cl)c1 ZINC000217791348 DI For-Sale Unstable OPRL1 0 43 C[C@H](N)[C@H](c1ccccc1)N(C)[C@@H](C)c1cccc(Cl)c1 ZINC000217791348 DI For-Sale Unstable AOC3 19 44 CC(C)(C)OC(=O)NCCNC(=O)N/C=C/c1ccccc1F ZINC000217791359 DF For-Sale Unstable PAPA1_CARPA 36 41 CC(C)(C)OC(=O)NCCNC(=O)N/C=C/c1ccccc1F ZINC000217791359 DF For-Sale Unstable CTSK 18 40 COc1cc(F)ccc1-c1ccnc2[nH]c(I)cc12 ZINC000217791372 FH For-Sale Unstable GRIN2B 36 41 COc1cc(F)ccc1-c1ccnc2[nH]c(I)cc12 ZINC000217791372 FH For-Sale Unstable KIT 18 42 O=C(Cn1nnc2ccccc21)N1CCC(N2C(=O)CSC2=O)CC1 ZINC000217791387 FD In-Stock Unstable MGLL 0 42 COc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791390 FG In-Stock Unstable HTR1A 122 54 COc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791390 FG In-Stock Unstable DRD2 82 49 COc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791390 FG In-Stock Unstable DRD1 44 39 COc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791390 FG In-Stock Unstable DRD4 55 43 COc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791390 FG In-Stock Unstable ACHE 18 45 COc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791390 FG In-Stock Unstable ADRA1D 43 45 COc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791390 FG In-Stock Unstable HTR2A 79 48 COc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791390 FG In-Stock Unstable HTR2C 25 41 COc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791390 FG In-Stock Unstable SLC6A4 21 49 COc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791390 FG In-Stock Unstable ADRA1A 44 48 COc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791390 FG In-Stock Unstable HRH1 17 42 COc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791390 FG In-Stock Unstable ADRA1B 38 41 COc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791390 FG In-Stock Unstable DRD3 82 54 COc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791390 FG In-Stock Unstable DRD5 33 47 COc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791390 FG In-Stock Unstable HTR7 105 41 COc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791390 FG In-Stock Unstable SIGMAR1 39 54 COc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791390 FG In-Stock Unstable BCHE 18 41 COc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791390 FG In-Stock Unstable ABCB1 25 41 COc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791390 FG In-Stock Unstable MET 51 38 COc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791390 FG In-Stock Unstable MCHR1 0 42 COc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791390 FG In-Stock Unstable EHMT2 77 41 COc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791390 FG In-Stock Unstable SLC29A2 0 40 COc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791390 FG In-Stock Unstable ASF1A 0 44 O=S(=O)(Nc1ccc2c(c1)CCC2)c1ccc(CO)o1 ZINC000217791417 CE For-Sale Unstable MLNR 15 40 COCCN(CC(=O)O)C(=O)/C=C\c1ccc(OC)cc1 ZINC000217791423 CD On-Demand Unstable GPR183 0 41 COc1ccc(C)cc1S(=O)(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217791460 FE For-Sale Unstable ADAMTS5 30 40 CC(C)(C)OC(=O)N1CCN(C(=O)N/C=C/c2ccccc2F)CC1 ZINC000217791480 EG For-Sale Unstable F13A1 16 42 CC(C)(C)OC(=O)N1CCN(C(=O)N/C=C/c2ccccc2F)CC1 ZINC000217791480 EG For-Sale Unstable GPR119 37 44 O=C(N[C@@H]1CCCCNC1=O)[C@@H]1C[C@@H]2CCCC[C@@H]2N1 ZINC000217791523 CC For-Sale Unstable MMP1 0 40 C[C@H]1CCCN1[C@H](C)CCc1ccc(O)cc1 ZINC000217791537 BG For-Sale Unstable HRH3 32 42 C[C@H]1CCCN1[C@H](C)CCc1ccc(O)cc1 ZINC000217791537 BG For-Sale Unstable BIRC2 32 40 COC1CCN(C2CCN(S(=O)(=O)c3ccc(C(C)=O)cc3)CC2)CC1 ZINC000217791551 GE In-Stock Unstable CHRM2 61 52 COC1CCN(C2CCN(S(=O)(=O)c3ccc(C(C)=O)cc3)CC2)CC1 ZINC000217791551 GE In-Stock Unstable MMP13 18 40 COC1CCN(C2CCN(S(=O)(=O)c3ccc(C(C)=O)cc3)CC2)CC1 ZINC000217791551 GE In-Stock Unstable MMP3 16 40 COC1CCN(C2CCN(S(=O)(=O)c3ccc(C(C)=O)cc3)CC2)CC1 ZINC000217791551 GE In-Stock Unstable TGM2 59 38 COC1CCN(C2CCN(S(=O)(=O)c3ccc(C(C)=O)cc3)CC2)CC1 ZINC000217791551 GE In-Stock Unstable MMP7 20 40 COC1CCN(C2CCN(S(=O)(=O)c3ccc(C(C)=O)cc3)CC2)CC1 ZINC000217791551 GE In-Stock Unstable F13A1 56 37 COC1CCN(C2CCN(S(=O)(=O)c3ccc(C(C)=O)cc3)CC2)CC1 ZINC000217791551 GE In-Stock Unstable L3MBTL3 70 56 COC1CCN(C2CCN(S(=O)(=O)c3ccc(C(C)=O)cc3)CC2)CC1 ZINC000217791551 GE In-Stock Unstable NAMPT 18 45 COc1ccc(C)cc1S(=O)(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217791566 FE For-Sale Unstable ADAMTS5 30 40 CC(C)(C)OC(=O)N1CCC(NC(=O)N/C=C/c2ccccc2F)CC1 ZINC000217791592 FG For-Sale Unstable EPHX2 42 36 CC(C)(C)OC(=O)N1CCC(NC(=O)N/C=C/c2ccccc2F)CC1 ZINC000217791592 FG For-Sale Unstable CCR8 19 42 CC(C)(C)OC(=O)N1CCC(NC(=O)N/C=C/c2ccccc2F)CC1 ZINC000217791592 FG For-Sale Unstable GPR119 46 47 CC(C)(C)OC(=O)N1CCC(NC(=O)N/C=C/c2ccccc2F)CC1 ZINC000217791592 FG For-Sale Unstable SFRP1 30 40 COc1ccc2occ([C@H](CC(N)=O)c3oc(C)cc(=O)c3O)c(=O)c2c1 ZINC000217791607 FD In-Stock Unstable ALDH2 58 35 O=C1NCCCC[C@@H]1NC(=O)[C@@H]1C[C@@H]2CCCC[C@@H]2N1 ZINC000217791624 CC On-Demand Unstable MMP1 18 40 O=C(COc1ccc(-c2ccccc2)cc1)c1nccs1 ZINC000217791640 CI Annotated Unstable FFAR1 17 40 O=C1CN(C(=O)c2ccncc2O)CCN1Cc1ccc(F)cc1 ZINC000217791669 ED In-Stock Unstable P2RX7 31 40 C[C@H]1CCCN1[C@H](C)c1ccccc1O ZINC000217791670 BF For-Sale Unstable HRH3 26 50 COc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)c(C)c1 ZINC000217791693 FE For-Sale Unstable ADAMTS5 30 40 COc1ccc2occ([C@@H](CC(N)=O)c3oc(C)cc(=O)c3O)c(=O)c2c1 ZINC000217791704 FD In-Stock Unstable ALDH2 58 35 COc1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1OC ZINC000217791713 EI For-Sale Unstable GRM4 21 44 COc1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1OC ZINC000217791713 EI For-Sale Unstable IMPDH2 0 51 COc1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1OC ZINC000217791713 EI For-Sale Unstable ENPP1 71 35 COc1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1OC ZINC000217791713 EI For-Sale Unstable IMDH_CRYPV 36 41 COc1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1OC ZINC000217791713 EI For-Sale Unstable CYSP_PLAFA 42 36 O=C1NCCCC[C@@H]1NC(=O)[C@H]1C[C@@H]2CCCC[C@@H]2N1 ZINC000217791719 CC For-Sale Unstable MMP1 0 40 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)c(C)c1 ZINC000217791767 FE For-Sale Unstable ADAMTS5 30 40 O=C(CCn1c2c(c3ccccc31)CCCC2)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217791827 HH In-Stock Unstable FABI 52 32 O=C(CCn1c2c(c3ccccc31)CCCC2)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217791827 HH In-Stock Unstable FABP4 49 36 O=C(CCn1c2c(c3ccccc31)CCCC2)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217791827 HH In-Stock Unstable CHRNA4 39 52 N#Cc1nccnc1O[C@H]1CCCN(C(=O)CCn2cnc3ccccc3c2=O)C1 ZINC000217791830 HD In-Stock Unstable PREP 35 40 N#Cc1nccnc1O[C@H]1CCCN(C(=O)CCn2cnc3ccccc3c2=O)C1 ZINC000217791830 HD In-Stock Unstable FAP 0 40 O=C(N/C=C/c1ccccc1Cl)NCCCN1CCCC1=O ZINC000217791831 DF For-Sale Unstable TYRO3 25 44 CCOc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791840 FG In-Stock Unstable HTR1A 78 53 CCOc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791840 FG In-Stock Unstable DRD2 55 53 CCOc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791840 FG In-Stock Unstable DRD4 36 40 CCOc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791840 FG In-Stock Unstable HTR2A 56 47 CCOc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791840 FG In-Stock Unstable SLC6A4 15 41 CCOc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791840 FG In-Stock Unstable ADRA1A 25 47 CCOc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791840 FG In-Stock Unstable HRH1 18 53 CCOc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791840 FG In-Stock Unstable DRD3 59 53 CCOc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791840 FG In-Stock Unstable DRD5 33 46 CCOc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791840 FG In-Stock Unstable HTR7 82 45 CCOc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791840 FG In-Stock Unstable SIGMAR1 29 48 CCOc1cc(C=O)ccc1OCCCN1CCN(c2ccccc2)CC1 ZINC000217791840 FG In-Stock Unstable ABCB1 15 40 COc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)cc1F ZINC000217791877 FE For-Sale Unstable ADAMTS5 32 41 N#Cc1nccnc1O[C@@H]1CCCN(C(=O)CCn2cnc3ccccc3c2=O)C1 ZINC000217791900 HD In-Stock Unstable PREP 35 40 N#Cc1nccnc1O[C@@H]1CCCN(C(=O)CCn2cnc3ccccc3c2=O)C1 ZINC000217791900 HD In-Stock Unstable FAP 0 40 COc1cc([C@@H](C)N2CCC[C@@H]2C)ccc1O ZINC000217791903 BF For-Sale Unstable PNLIP 0 48 COc1cc([C@@H](C)N2CCC[C@@H]2C)ccc1O ZINC000217791903 BF For-Sale Unstable N1L 0 49 COc1cc([C@@H](C)N2CCC[C@@H]2C)ccc1O ZINC000217791903 BF For-Sale Unstable SLC22A3 0 45 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(Br)cc1 ZINC000217791921 FJ For-Sale Anodyne SMO 15 40 COc1ccc([C@@H]2CC(=O)Oc3ccc4c(c32)OC(=C(C)C)C4=O)cc1OC ZINC000217791923 GI In-Stock Unstable MT-ND4 52 32 CCN(CC)CCCCOc1c(C=O)cccc1OC ZINC000217791941 CG In-Stock Unstable ACHE 0 49 CCN(CC)CCCCOc1c(C=O)cccc1OC ZINC000217791941 CG In-Stock Unstable BCHE 0 49 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)cc1F ZINC000217791961 FE For-Sale Unstable ADAMTS5 32 41 COc1ccc([C@H]2CC(=O)Oc3ccc4c(c32)OC(=C(C)C)C4=O)cc1OC ZINC000217792012 GI In-Stock Unstable MT-ND4 52 32 O=C(N/C=C/c1ccccc1Cl)Nc1cccc(C(=O)O)c1 ZINC000217792018 DH For-Sale Anodyne PPIA 20 40 O=C(N/C=C/c1ccccc1Cl)Nc1cccc(C(=O)O)c1 ZINC000217792018 DH For-Sale Anodyne EPHX2 15 43 O=C(N/C=C/c1ccccc1Cl)Nc1cccc(C(=O)O)c1 ZINC000217792018 DH For-Sale Anodyne AKR1C3 36 47 O=C(N/C=C/c1ccccc1Cl)Nc1cccc(C(=O)O)c1 ZINC000217792018 DH For-Sale Anodyne IMDH_CRYPV 40 34 O=C(N/C=C/c1ccccc1Cl)Nc1cccc(C(=O)O)c1 ZINC000217792018 DH For-Sale Anodyne KCNK3 74 46 O=C(N[C@@H]1CCCCNC1=O)[C@@H]1C[C@@H](O)CN1 ZINC000217792028 BA For-Sale Unstable MMP1 0 40 C[C@H]1CCCN1[C@H](C)c1ccc2ccccc2c1O ZINC000217792033 CI For-Sale Unstable HRH3 35 44 Cc1c(Cl)cccc1S(=O)(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217792059 FG For-Sale Unstable ADAMTS5 31 40 COC(=O)[C@@H]1CC[C@@H]1Sc1ccccc1 ZINC000217792078 BF In-Stock Unstable SLC6A1 51 40 O=C(N[C@@H]1CCCCNC1=O)[C@H]1C[C@@H](O)CN1 ZINC000217792108 BA For-Sale Unstable MMP1 0 40 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(-c3cccc(C(=O)O)c3)o2)CC(=O)O4)cc1O ZINC000217792112 KK In-Stock Unstable CYP1B1 41 36 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(-c3cccc(C(=O)O)c3)o2)CC(=O)O4)cc1O ZINC000217792112 KK In-Stock Unstable CYP1A1 33 42 Cc1c(Cl)cccc1S(=O)(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217792148 FG For-Sale Unstable ADAMTS5 31 40 COC(=O)[C@H]1CC[C@@H]1Sc1ccccc1 ZINC000217792166 BF In-Stock Unstable SLC6A1 51 40 COc1cccc(C=O)c1OCCCCN1CCCC1 ZINC000217792169 CF In-Stock Unstable HTR1A 73 40 COc1cccc(C=O)c1OCCCCN1CCCC1 ZINC000217792169 CF In-Stock Unstable DRD2 64 44 COc1cccc(C=O)c1OCCCCN1CCCC1 ZINC000217792169 CF In-Stock Unstable DRD1 32 42 COc1cccc(C=O)c1OCCCCN1CCCC1 ZINC000217792169 CF In-Stock Unstable DRD4 31 40 COc1cccc(C=O)c1OCCCCN1CCCC1 ZINC000217792169 CF In-Stock Unstable ACHE 24 48 COc1cccc(C=O)c1OCCCCN1CCCC1 ZINC000217792169 CF In-Stock Unstable ADRA1D 39 41 COc1cccc(C=O)c1OCCCCN1CCCC1 ZINC000217792169 CF In-Stock Unstable HTR2A 44 42 COc1cccc(C=O)c1OCCCCN1CCCC1 ZINC000217792169 CF In-Stock Unstable ADRA1B 28 41 COc1cccc(C=O)c1OCCCCN1CCCC1 ZINC000217792169 CF In-Stock Unstable DRD3 58 42 COc1cccc(C=O)c1OCCCCN1CCCC1 ZINC000217792169 CF In-Stock Unstable KCNH2 0 46 COc1cccc(C=O)c1OCCCCN1CCCC1 ZINC000217792169 CF In-Stock Unstable HTR4 21 47 COc1cccc(C=O)c1OCCCCN1CCCC1 ZINC000217792169 CF In-Stock Unstable DRD5 18 42 COc1cccc(C=O)c1OCCCCN1CCCC1 ZINC000217792169 CF In-Stock Unstable HTR7 58 42 COc1cccc(C=O)c1OCCCCN1CCCC1 ZINC000217792169 CF In-Stock Unstable HRH3 58 42 COc1cccc(C=O)c1OCCCCN1CCCC1 ZINC000217792169 CF In-Stock Unstable SIGMAR1 35 50 COc1cccc(C=O)c1OCCCCN1CCCC1 ZINC000217792169 CF In-Stock Unstable CHRNA7 16 40 COc1cccc(C=O)c1OCCCCN1CCCC1 ZINC000217792169 CF In-Stock Unstable EBP 41 42 COc1cccc(C=O)c1OCCCCN1CCCC1 ZINC000217792169 CF In-Stock Unstable HNMT 62 32 COc1cccc(C=O)c1OCCCCN1CCCC1 ZINC000217792169 CF In-Stock Unstable ABCB1 22 41 COc1cccc(C=O)c1OCCCCN1CCCC1 ZINC000217792169 CF In-Stock Unstable PSMB2 44 33 COc1cccc(C=O)c1OCCCCN1CCCC1 ZINC000217792169 CF In-Stock Unstable EHMT2 53 37 COc1cccc(C=O)c1OCCCCN1CCCC1 ZINC000217792169 CF In-Stock Unstable SLC29A2 0 44 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(-c3cccc(C(=O)O)c3)o2)CC(=O)O4)cc1O ZINC000217792208 KK In-Stock Unstable CYP1B1 41 36 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(-c3cccc(C(=O)O)c3)o2)CC(=O)O4)cc1O ZINC000217792208 KK In-Stock Unstable CYP1A1 33 42 O=C(N/C=C/c1ccccc1Cl)Nc1cccc(O)c1 ZINC000217792221 CH For-Sale Anodyne KCNK3 55 41 COc1ccc(CNC(=O)c2cc(=O)nc[nH]2)cc1 ZINC000217792223 CC In-Stock Unstable ROCK2 23 48 COc1ccc(CNC(=O)c2cc(=O)nc[nH]2)cc1 ZINC000217792223 CC In-Stock Unstable CA9 15 43 COc1ccc(CNC(=O)c2cc(=O)nc[nH]2)cc1 ZINC000217792223 CC In-Stock Unstable U38 0 44 COc1ccc(CNC(=O)c2cc(=O)nc[nH]2)cc1 ZINC000217792223 CC In-Stock Unstable PROKR1 54 33 COc1ccc(CNC(=O)c2cc(=O)nc[nH]2)cc1 ZINC000217792223 CC In-Stock Unstable Q76353_9HIV1 0 45 COC(=O)[C@@H]1CC[C@H]1Sc1ccccc1 ZINC000217792242 BF In-Stock Unstable SLC6A1 51 40 Cc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)cc1Cl ZINC000217792260 FG For-Sale Unstable ADAMTS5 34 46 COc1cccc(C=O)c1OCCCCN1CCCCC1 ZINC000217792274 CG In-Stock Unstable HTR1A 69 40 COc1cccc(C=O)c1OCCCCN1CCCCC1 ZINC000217792274 CG In-Stock Unstable DRD2 61 43 COc1cccc(C=O)c1OCCCCN1CCCCC1 ZINC000217792274 CG In-Stock Unstable DRD1 30 42 COc1cccc(C=O)c1OCCCCN1CCCCC1 ZINC000217792274 CG In-Stock Unstable ACHE 27 48 COc1cccc(C=O)c1OCCCCN1CCCCC1 ZINC000217792274 CG In-Stock Unstable ADRA1D 38 40 COc1cccc(C=O)c1OCCCCN1CCCCC1 ZINC000217792274 CG In-Stock Unstable HTR2A 40 41 COc1cccc(C=O)c1OCCCCN1CCCCC1 ZINC000217792274 CG In-Stock Unstable ADRA1B 27 40 COc1cccc(C=O)c1OCCCCN1CCCCC1 ZINC000217792274 CG In-Stock Unstable DRD3 57 41 COc1cccc(C=O)c1OCCCCN1CCCCC1 ZINC000217792274 CG In-Stock Unstable KCNH2 0 48 COc1cccc(C=O)c1OCCCCN1CCCCC1 ZINC000217792274 CG In-Stock Unstable HTR4 20 49 COc1cccc(C=O)c1OCCCCN1CCCCC1 ZINC000217792274 CG In-Stock Unstable DRD5 20 42 COc1cccc(C=O)c1OCCCCN1CCCCC1 ZINC000217792274 CG In-Stock Unstable HTR7 56 41 COc1cccc(C=O)c1OCCCCN1CCCCC1 ZINC000217792274 CG In-Stock Unstable HRH3 68 43 COc1cccc(C=O)c1OCCCCN1CCCCC1 ZINC000217792274 CG In-Stock Unstable SIGMAR1 36 49 COc1cccc(C=O)c1OCCCCN1CCCCC1 ZINC000217792274 CG In-Stock Unstable NPY1R 40 33 COc1cccc(C=O)c1OCCCCN1CCCCC1 ZINC000217792274 CG In-Stock Unstable CHRNA7 18 41 COc1cccc(C=O)c1OCCCCN1CCCCC1 ZINC000217792274 CG In-Stock Unstable EBP 36 46 COc1cccc(C=O)c1OCCCCN1CCCCC1 ZINC000217792274 CG In-Stock Unstable HNMT 74 34 COc1cccc(C=O)c1OCCCCN1CCCCC1 ZINC000217792274 CG In-Stock Unstable ABCB1 21 43 COc1cccc(C=O)c1OCCCCN1CCCCC1 ZINC000217792274 CG In-Stock Unstable PSMB2 46 35 COc1cccc(C=O)c1OCCCCN1CCCCC1 ZINC000217792274 CG In-Stock Unstable PSMB1 40 35 COc1cccc(C=O)c1OCCCCN1CCCCC1 ZINC000217792274 CG In-Stock Unstable EHMT2 47 36 C[C@H]1CCCN1[C@H](C)c1cccc(O)c1 ZINC000217792305 BF For-Sale Unstable OPRM1 15 45 COC(=O)[C@H]1CC[C@H]1Sc1ccccc1 ZINC000217792306 BF In-Stock Unstable SLC6A1 51 40 Cc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)cc1Cl ZINC000217792309 FG For-Sale Unstable ADAMTS5 34 46 Cc1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217792323 CI For-Sale Unstable LPL 42 33 Cc1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217792323 CI For-Sale Unstable SMO 17 40 COC(=O)c1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)cc1 ZINC000217792325 JI In-Stock Unstable AKR1B1 0 46 COC(=O)c1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)cc1 ZINC000217792325 JI In-Stock Unstable CYP1B1 48 34 COC(=O)c1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)cc1 ZINC000217792325 JI In-Stock Unstable CYP1A1 37 46 CC(C)=C1C(=O)Cc2cccc(O)c21 ZINC000217792335 AE For-Sale Unstable Q9BEG3_BOVIN 43 38 CC1(C)CC(COc2ccccc2)C1 ZINC000217792393 AH In-Stock Unstable CHRNA10 58 46 COc1cccc(C=O)c1OCCCCN1CCOCC1 ZINC000217792397 CD In-Stock Unstable HTR1A 61 39 COc1cccc(C=O)c1OCCCCN1CCOCC1 ZINC000217792397 CD In-Stock Unstable DRD2 55 44 COc1cccc(C=O)c1OCCCCN1CCOCC1 ZINC000217792397 CD In-Stock Unstable DRD1 23 41 COc1cccc(C=O)c1OCCCCN1CCOCC1 ZINC000217792397 CD In-Stock Unstable ACHE 15 42 COc1cccc(C=O)c1OCCCCN1CCOCC1 ZINC000217792397 CD In-Stock Unstable HTR2A 35 42 COc1cccc(C=O)c1OCCCCN1CCOCC1 ZINC000217792397 CD In-Stock Unstable ADRA1A 32 43 COc1cccc(C=O)c1OCCCCN1CCOCC1 ZINC000217792397 CD In-Stock Unstable DRD3 49 42 COc1cccc(C=O)c1OCCCCN1CCOCC1 ZINC000217792397 CD In-Stock Unstable DRD5 15 41 COc1cccc(C=O)c1OCCCCN1CCOCC1 ZINC000217792397 CD In-Stock Unstable HTR7 49 41 COc1cccc(C=O)c1OCCCCN1CCOCC1 ZINC000217792397 CD In-Stock Unstable SIGMAR1 27 43 COc1cccc(C=O)c1OCCCCN1CCOCC1 ZINC000217792397 CD In-Stock Unstable ABCB1 15 45 COc1cccc(C=O)c1OCCCCN1CCOCC1 ZINC000217792397 CD In-Stock Unstable EPHX2 16 43 COc1cccc(C=O)c1OCCCCN1CCOCC1 ZINC000217792397 CD In-Stock Unstable AURKA 19 41 COc1cccc(C=O)c1OCCCCN1CCOCC1 ZINC000217792397 CD In-Stock Unstable SLC29A2 0 41 COc1cccc(C=O)c1OCCCCN1CCOCC1 ZINC000217792397 CD In-Stock Unstable AURKB-A 0 41 COC(=O)c1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)cc1 ZINC000217792426 JI In-Stock Unstable AKR1B1 0 46 COC(=O)c1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)cc1 ZINC000217792426 JI In-Stock Unstable CYP1B1 48 34 COC(=O)c1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)cc1 ZINC000217792426 JI In-Stock Unstable CYP1A1 37 46 COc1ccc(NC(=O)c2cc(=O)nc[nH]2)c(OC)c1 ZINC000217792459 CD In-Stock Unstable CYP1B1 17 55 COc1ccc(NC(=O)c2cc(=O)nc[nH]2)c(OC)c1 ZINC000217792459 CD In-Stock Unstable LUCI_LUCLA 16 41 Cc1ccc(Cl)cc1S(=O)(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217792468 FG For-Sale Unstable ADAMTS5 31 43 COc1cccc(C=O)c1OCCCCN1CCC(C)CC1 ZINC000217792490 DG In-Stock Unstable HTR1A 65 40 COc1cccc(C=O)c1OCCCCN1CCC(C)CC1 ZINC000217792490 DG In-Stock Unstable DRD2 58 41 COc1cccc(C=O)c1OCCCCN1CCC(C)CC1 ZINC000217792490 DG In-Stock Unstable HTR2A 40 39 COc1cccc(C=O)c1OCCCCN1CCC(C)CC1 ZINC000217792490 DG In-Stock Unstable DRD3 49 41 COc1cccc(C=O)c1OCCCCN1CCC(C)CC1 ZINC000217792490 DG In-Stock Unstable HTR7 56 39 COc1cccc(C=O)c1OCCCCN1CCC(C)CC1 ZINC000217792490 DG In-Stock Unstable SIGMAR1 24 41 COc1cccc(C=O)c1OCCCCN1CCC(C)CC1 ZINC000217792490 DG In-Stock Unstable EBP 47 44 COc1cccc(C=O)c1OCCCCN1CCC(C)CC1 ZINC000217792490 DG In-Stock Unstable SLC29A2 0 40 CCCCCS[C@@H](C)C(=O)OC(C)(C)C ZINC000217792503 BH On-Demand Unstable EST1_PIG 49 35 CCCCCS[C@@H](C)C(=O)OC(C)(C)C ZINC000217792503 BH On-Demand Unstable CQSS 40 32 Nc1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217792535 CH For-Sale Unstable SMO 15 40 Cc1ccc(Cl)cc1S(=O)(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217792549 FG For-Sale Unstable ADAMTS5 31 43 O=C1C[C@@H](c2ccncc2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217792565 HH In-Stock Unstable AKR1B1 0 44 O=C1C[C@@H](c2ccncc2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217792565 HH In-Stock Unstable CYP1B1 28 41 O=C1C[C@@H](c2ccncc2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217792565 HH In-Stock Unstable CYP1A1 25 41 O=C1C[C@@H](c2ccncc2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217792565 HH In-Stock Unstable CYP1A2 19 41 CC(=O)c1cccc(NC(=O)c2cc(=O)nc[nH]2)c1 ZINC000217792571 CD In-Stock Unstable AKR1C3 25 44 CC(=O)c1cccc(NC(=O)c2cc(=O)nc[nH]2)c1 ZINC000217792571 CD In-Stock Unstable KCNK3 95 43 CC(=O)c1cccc(NC(=O)c2cc(=O)nc[nH]2)c1 ZINC000217792571 CD In-Stock Unstable KCNK9 78 42 CC1(C)CC(COc2cccc(Br)c2)C1 ZINC000217792588 CI In-Stock Unstable CHRNA10 62 38 CCCCCS[C@H](C)C(=O)OC(C)(C)C ZINC000217792599 BH On-Demand Unstable EST1_PIG 49 35 CCCCCS[C@H](C)C(=O)OC(C)(C)C ZINC000217792599 BH On-Demand Unstable CQSS 40 32 COc1cccc(C=O)c1OCCCCN1CCCC[C@@H]1C ZINC000217792603 DH In-Stock Unstable HRH3 52 46 COc1cccc(C=O)c1OCCCCN1CCCC[C@@H]1C ZINC000217792603 DH In-Stock Unstable EBP 29 47 COc1cccc(C=O)c1OCCCCN1CCCC[C@@H]1C ZINC000217792603 DH In-Stock Unstable ACKR3 55 32 O=C1C[C@H](c2ccncc2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217792656 HH In-Stock Unstable AKR1B1 0 44 O=C1C[C@H](c2ccncc2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217792656 HH In-Stock Unstable CYP1B1 28 41 O=C1C[C@H](c2ccncc2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217792656 HH In-Stock Unstable CYP1A1 25 41 O=C1C[C@H](c2ccncc2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217792656 HH In-Stock Unstable CYP1A2 19 41 CCOC(=O)c1ccc(NC(=O)c2cc(=O)nc[nH]2)cc1 ZINC000217792674 CD In-Stock Unstable PRNP 40 34 CCOC(=O)c1ccc(NC(=O)c2cc(=O)nc[nH]2)cc1 ZINC000217792674 CD In-Stock Unstable ACR 57 36 CCOC(=O)c1ccc(NC(=O)c2cc(=O)nc[nH]2)cc1 ZINC000217792674 CD In-Stock Unstable NOD2 18 43 COc1ccc(S(=O)(=O)N2CCC(N3CCC(OC)CC3)CC2)cc1F ZINC000217792681 GE In-Stock Unstable CHRM2 52 42 COc1cccc(C=O)c1OCCCCN1CCCC[C@H]1C ZINC000217792686 DH In-Stock Unstable HRH3 52 46 COc1cccc(C=O)c1OCCCCN1CCCC[C@H]1C ZINC000217792686 DH In-Stock Unstable EBP 29 47 COc1cccc(C=O)c1OCCCCN1CCCC[C@H]1C ZINC000217792686 DH In-Stock Unstable ACKR3 55 32 Cc1c(F)ccc(C(=O)O)c1O ZINC000217792744 AD For-Sale Unstable GRM3 24 42 Cc1c(F)ccc(C(=O)O)c1O ZINC000217792744 AD For-Sale Unstable GRM2 23 46 Cc1c(F)ccc(C(=O)O)c1O ZINC000217792744 AD For-Sale Unstable AKR1C2 50 42 Cc1c(F)ccc(C(=O)O)c1O ZINC000217792744 AD For-Sale Unstable AKR1C1 54 42 Cc1c(F)ccc(C(=O)O)c1O ZINC000217792744 AD For-Sale Unstable HAAO 43 35 CC(=O)Nc1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217792749 EI For-Sale Unstable SMO 15 40 COC(=O)C[C@H](c1cc(OC)c(OC(C)=O)c(OC)c1)c1c(O)c2ccccc2oc1=O ZINC000217792756 IG In-Stock Unstable NQO1 59 48 O=C(Nc1nc2ccccc2s1)c1cc(=O)nc[nH]1 ZINC000217792799 CD In-Stock Anodyne CSNK1D 35 48 O=C(Nc1nc2ccccc2s1)c1cc(=O)nc[nH]1 ZINC000217792799 CD In-Stock Anodyne FABK 0 43 O=C(Nc1nc2ccccc2s1)c1cc(=O)nc[nH]1 ZINC000217792799 CD In-Stock Anodyne PORCN 0 40 COC(=O)C[C@@H](c1cc(OC)c(OC(C)=O)c(OC)c1)c1c(O)c2ccccc2oc1=O ZINC000217792809 IG In-Stock Unstable NQO1 59 48 O=S(=O)(Cc1cccc(Cl)c1)NC[C@@H]1CCCN1c1nccs1 ZINC000217792836 FF For-Sale Unstable ADAMTS5 27 42 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217792840 FG For-Sale Anodyne LPL 48 33 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217792840 FG For-Sale Anodyne CA12 27 44 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217792840 FG For-Sale Anodyne CA9 21 44 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217792840 FG For-Sale Anodyne PFK 0 42 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217792840 FG For-Sale Anodyne MTCA1 43 40 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217792840 FG For-Sale Anodyne P96878_MYCTU 54 40 O=S(=O)(Cc1cccc(Cl)c1)NC[C@H]1CCCN1c1nccs1 ZINC000217792894 FF For-Sale Unstable ADAMTS5 27 42 NS(=O)(=O)c1ccc(NC(=O)c2cc(=O)nc[nH]2)cc1 ZINC000217792921 CB In-Stock Unstable CA2 102 52 NS(=O)(=O)c1ccc(NC(=O)c2cc(=O)nc[nH]2)cc1 ZINC000217792921 CB In-Stock Unstable CA1 91 56 NS(=O)(=O)c1ccc(NC(=O)c2cc(=O)nc[nH]2)cc1 ZINC000217792921 CB In-Stock Unstable CA7 48 42 NS(=O)(=O)c1ccc(NC(=O)c2cc(=O)nc[nH]2)cc1 ZINC000217792921 CB In-Stock Unstable CA5B 47 42 NS(=O)(=O)c1ccc(NC(=O)c2cc(=O)nc[nH]2)cc1 ZINC000217792921 CB In-Stock Unstable CA4 83 56 NS(=O)(=O)c1ccc(NC(=O)c2cc(=O)nc[nH]2)cc1 ZINC000217792921 CB In-Stock Unstable CA5A 53 42 NS(=O)(=O)c1ccc(NC(=O)c2cc(=O)nc[nH]2)cc1 ZINC000217792921 CB In-Stock Unstable CA14 45 40 NS(=O)(=O)c1ccc(NC(=O)c2cc(=O)nc[nH]2)cc1 ZINC000217792921 CB In-Stock Unstable CA12 67 42 NS(=O)(=O)c1ccc(NC(=O)c2cc(=O)nc[nH]2)cc1 ZINC000217792921 CB In-Stock Unstable CA9 68 46 NS(=O)(=O)c1ccc(NC(=O)c2cc(=O)nc[nH]2)cc1 ZINC000217792921 CB In-Stock Unstable UREA_CANEN 28 42 NS(=O)(=O)c1ccc(NC(=O)c2cc(=O)nc[nH]2)cc1 ZINC000217792921 CB In-Stock Unstable CYNT 44 49 NS(=O)(=O)c1ccc(NC(=O)c2cc(=O)nc[nH]2)cc1 ZINC000217792921 CB In-Stock Unstable MTCA1 43 44 NS(=O)(=O)c1ccc(NC(=O)c2cc(=O)nc[nH]2)cc1 ZINC000217792921 CB In-Stock Unstable P96878_MYCTU 60 47 O=C(N/C=C/c1ccccc1Cl)Nc1cccc(S(=O)(=O)O)c1 ZINC000217792929 FG For-Sale Anodyne LPL 42 33 COC1CCN(C2CCN(S(=O)(=O)c3ccc(C)c(Cl)c3)CC2)CC1 ZINC000217792937 GF In-Stock Unstable CHRM2 48 42 COC1CCN(C2CCN(S(=O)(=O)c3ccc(C)c(Cl)c3)CC2)CC1 ZINC000217792937 GF In-Stock Unstable HRH1 18 42 COC1CCN(C2CCN(S(=O)(=O)c3ccc(C)c(Cl)c3)CC2)CC1 ZINC000217792937 GF In-Stock Unstable CCR3 19 40 COc1ccc([C@@H](C)N2CC[C@@H](C)C2)c(O)c1 ZINC000217792959 BF For-Sale Unstable RORC 44 38 CN(C)C(=O)[C@H](N)Cc1ccncc1 ZINC000217793023 AC For-Sale Unstable SLC15A1 59 37 COc1cccc(C=O)c1OCCCCN1CCCCCC1 ZINC000217793050 DH In-Stock Unstable HTR1A 96 42 COc1cccc(C=O)c1OCCCCN1CCCCCC1 ZINC000217793050 DH In-Stock Unstable DRD2 74 43 COc1cccc(C=O)c1OCCCCN1CCCCCC1 ZINC000217793050 DH In-Stock Unstable DRD1 30 42 COc1cccc(C=O)c1OCCCCN1CCCCCC1 ZINC000217793050 DH In-Stock Unstable DRD4 36 40 COc1cccc(C=O)c1OCCCCN1CCCCCC1 ZINC000217793050 DH In-Stock Unstable ACHE 29 48 COc1cccc(C=O)c1OCCCCN1CCCCCC1 ZINC000217793050 DH In-Stock Unstable ADRA1D 41 40 COc1cccc(C=O)c1OCCCCN1CCCCCC1 ZINC000217793050 DH In-Stock Unstable HTR2A 41 41 COc1cccc(C=O)c1OCCCCN1CCCCCC1 ZINC000217793050 DH In-Stock Unstable ADRA1A 46 42 COc1cccc(C=O)c1OCCCCN1CCCCCC1 ZINC000217793050 DH In-Stock Unstable ADRA1B 37 42 COc1cccc(C=O)c1OCCCCN1CCCCCC1 ZINC000217793050 DH In-Stock Unstable DRD3 75 43 COc1cccc(C=O)c1OCCCCN1CCCCCC1 ZINC000217793050 DH In-Stock Unstable KCNH2 0 48 COc1cccc(C=O)c1OCCCCN1CCCCCC1 ZINC000217793050 DH In-Stock Unstable HTR4 25 49 COc1cccc(C=O)c1OCCCCN1CCCCCC1 ZINC000217793050 DH In-Stock Unstable DRD5 20 42 COc1cccc(C=O)c1OCCCCN1CCCCCC1 ZINC000217793050 DH In-Stock Unstable HTR7 57 41 COc1cccc(C=O)c1OCCCCN1CCCCCC1 ZINC000217793050 DH In-Stock Unstable HRH3 73 48 COc1cccc(C=O)c1OCCCCN1CCCCCC1 ZINC000217793050 DH In-Stock Unstable SIGMAR1 44 49 COc1cccc(C=O)c1OCCCCN1CCCCCC1 ZINC000217793050 DH In-Stock Unstable NPY1R 40 33 COc1cccc(C=O)c1OCCCCN1CCCCCC1 ZINC000217793050 DH In-Stock Unstable CHRNA7 18 41 COc1cccc(C=O)c1OCCCCN1CCCCCC1 ZINC000217793050 DH In-Stock Unstable EBP 47 46 COc1cccc(C=O)c1OCCCCN1CCCCCC1 ZINC000217793050 DH In-Stock Unstable HNMT 84 36 COc1cccc(C=O)c1OCCCCN1CCCCCC1 ZINC000217793050 DH In-Stock Unstable ABCB1 21 43 COc1cccc(C=O)c1OCCCCN1CCCCCC1 ZINC000217793050 DH In-Stock Unstable PSMB2 46 35 COc1cccc(C=O)c1OCCCCN1CCCCCC1 ZINC000217793050 DH In-Stock Unstable PSMB1 40 35 COc1cccc(C=O)c1OCCCCN1CCCCCC1 ZINC000217793050 DH In-Stock Unstable EHMT2 48 36 COc1cccc(C=O)c1OCCCCN1CCCCCC1 ZINC000217793050 DH In-Stock Unstable SLC29A2 0 43 CC(=O)NS(=O)(=O)c1ccc(NC(=O)c2cc(=O)nc[nH]2)cc1 ZINC000217793056 EB In-Stock Unstable IDO1 29 41 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1cccc2ccccc12 ZINC000217793057 FG For-Sale Unstable NPY1R 52 45 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1cccc2ccccc12 ZINC000217793057 FG For-Sale Unstable NPY2R 48 45 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1cccc2ccccc12 ZINC000217793057 FG For-Sale Unstable NPY5R 21 45 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1cccc2ccccc12 ZINC000217793057 FG For-Sale Unstable ADAMTS5 32 40 COC(=O)C[C@H](c1ccc2c(c1)OCCO2)c1c(OC)ccc2c(=O)c(-c3ccc(OC)cc3)coc12 ZINC000217793083 KJ In-Stock Unstable ALDH2 82 35 COC(=O)C[C@H](c1ccc2c(c1)OCCO2)c1c(OC)ccc2c(=O)c(-c3ccc(OC)cc3)coc12 ZINC000217793083 KJ In-Stock Unstable RORC 46 38 O=C(O)[C@H]1CCCN(S(=O)(=O)Cl)C1 ZINC000217793099 BC In-Stock Unstable SLC6A1 82 35 COC1CCN(C2CCN(S(=O)(=O)Cc3ccccc3Cl)CC2)CC1 ZINC000217793127 GF In-Stock Unstable CHRM2 54 41 COC1CCN(C2CCN(S(=O)(=O)Cc3ccccc3Cl)CC2)CC1 ZINC000217793127 GF In-Stock Unstable HRH1 16 41 COC1CCN(C2CCN(S(=O)(=O)Cc3ccccc3Cl)CC2)CC1 ZINC000217793127 GF In-Stock Unstable CCR3 29 41 COC(=O)C[C@@H](c1ccc2c(c1)OCCO2)c1c(OC)ccc2c(=O)c(-c3ccc(OC)cc3)coc12 ZINC000217793143 KJ In-Stock Unstable ALDH2 82 35 COC(=O)C[C@@H](c1ccc2c(c1)OCCO2)c1c(OC)ccc2c(=O)c(-c3ccc(OC)cc3)coc12 ZINC000217793143 KJ In-Stock Unstable RORC 46 38 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1cccc2ccccc12 ZINC000217793148 FG For-Sale Unstable NPY1R 52 45 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1cccc2ccccc12 ZINC000217793148 FG For-Sale Unstable NPY2R 48 45 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1cccc2ccccc12 ZINC000217793148 FG For-Sale Unstable NPY5R 21 45 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1cccc2ccccc12 ZINC000217793148 FG For-Sale Unstable ADAMTS5 32 40 O=C(O)[C@@H]1CCCN(S(=O)(=O)Cl)C1 ZINC000217793177 BC In-Stock Unstable SLC6A1 82 35 O=C(Nc1ccc(F)c(Cl)c1)c1cc(=O)nc[nH]1 ZINC000217793185 CD In-Stock Anodyne MAOB 19 47 O=C(Nc1ccc(F)c(Cl)c1)c1cc(=O)nc[nH]1 ZINC000217793185 CD In-Stock Anodyne GRM4 41 38 O=C(Nc1ccc(F)c(Cl)c1)c1cc(=O)nc[nH]1 ZINC000217793185 CD In-Stock Anodyne ERBB4 41 36 O=C(Nc1ccc(F)c(Cl)c1)c1cc(=O)nc[nH]1 ZINC000217793185 CD In-Stock Anodyne P95276_MYCTO 0 41 COc1cccc(C=O)c1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217793187 FG In-Stock Unstable HTR1A 158 50 COc1cccc(C=O)c1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217793187 FG In-Stock Unstable ADRA2A 17 42 COc1cccc(C=O)c1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217793187 FG In-Stock Unstable DRD2 111 57 COc1cccc(C=O)c1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217793187 FG In-Stock Unstable DRD1 52 45 COc1cccc(C=O)c1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217793187 FG In-Stock Unstable DRD4 62 48 COc1cccc(C=O)c1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217793187 FG In-Stock Unstable ACHE 16 42 COc1cccc(C=O)c1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217793187 FG In-Stock Unstable ADRA1D 72 46 COc1cccc(C=O)c1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217793187 FG In-Stock Unstable HTR1B 23 42 COc1cccc(C=O)c1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217793187 FG In-Stock Unstable HTR2A 96 50 COc1cccc(C=O)c1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217793187 FG In-Stock Unstable HTR2C 40 46 COc1cccc(C=O)c1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217793187 FG In-Stock Unstable SLC6A4 29 41 COc1cccc(C=O)c1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217793187 FG In-Stock Unstable ADRA1A 67 44 COc1cccc(C=O)c1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217793187 FG In-Stock Unstable HRH1 22 42 COc1cccc(C=O)c1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217793187 FG In-Stock Unstable ADRA1B 59 46 COc1cccc(C=O)c1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217793187 FG In-Stock Unstable DRD3 102 49 COc1cccc(C=O)c1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217793187 FG In-Stock Unstable KCNH2 0 49 COc1cccc(C=O)c1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217793187 FG In-Stock Unstable DRD5 34 46 COc1cccc(C=O)c1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217793187 FG In-Stock Unstable TACR1 0 40 COc1cccc(C=O)c1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217793187 FG In-Stock Unstable HTR7 136 50 COc1cccc(C=O)c1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217793187 FG In-Stock Unstable SIGMAR1 36 48 COc1cccc(C=O)c1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217793187 FG In-Stock Unstable HTR6 0 42 COc1cccc(C=O)c1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217793187 FG In-Stock Unstable ABCB1 34 44 COc1cccc(C=O)c1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217793187 FG In-Stock Unstable CACNA1G 25 40 COc1cccc(C=O)c1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217793187 FG In-Stock Unstable SLC29A2 0 41 COc1cccc(C=O)c1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217793187 FG In-Stock Unstable AP2S1 0 41 COc1cccc(C=O)c1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217793187 FG In-Stock Unstable ALPHA-1A 0 44 Brc1cccc(OCC2=CCC2)c1 ZINC000217793195 BH In-Stock Unstable MAOB 18 42 C[C@@H]1CCN([C@H](C)c2ccc(O)cc2)C1 ZINC000217793264 BF For-Sale Unstable ERG2 17 41 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1ccc(F)c(Cl)c1 ZINC000217793272 GF For-Sale Unstable ADAMTS5 32 43 O=C(Nc1ccc(F)c(C(F)(F)F)c1)c1cc(=O)nc[nH]1 ZINC000217793276 DE In-Stock Anodyne RIPK1 35 41 O=C(Nc1ccc(F)c(C(F)(F)F)c1)c1cc(=O)nc[nH]1 ZINC000217793276 DE In-Stock Anodyne TMPRSS4 0 41 CCN(CC)CCCCOc1ccc(C=O)cc1 ZINC000217793283 BF In-Stock Unstable THRA 31 43 CCN(CC)CCCCOc1ccc(C=O)cc1 ZINC000217793283 BF In-Stock Unstable ACHE 25 62 CCN(CC)CCCCOc1ccc(C=O)cc1 ZINC000217793283 BF In-Stock Unstable LTA4H 18 50 CCN(CC)CCCCOc1ccc(C=O)cc1 ZINC000217793283 BF In-Stock Unstable ERG2 17 40 CCN(CC)CCCCOc1ccc(C=O)cc1 ZINC000217793283 BF In-Stock Unstable THRB 0 43 CCN(CC)CCCCOc1ccc(C=O)cc1 ZINC000217793283 BF In-Stock Unstable KCNQ1 0 47 CCN(CC)CCCCOc1ccc(C=O)cc1 ZINC000217793283 BF In-Stock Unstable BCHE 0 64 CCN(CC)CCCCOc1ccc(C=O)cc1 ZINC000217793283 BF In-Stock Unstable PLA2G4B 56 34 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1ccc(F)c(Cl)c1 ZINC000217793344 GF For-Sale Unstable ADAMTS5 32 43 O=C(Nc1ncccc1O)c1cc(-c2ccc(Cl)cc2)n[nH]1 ZINC000217793360 DG On-Demand Anodyne TACR3 15 41 O=C(Nc1ncccc1O)c1cc(-c2ccc(Cl)cc2)n[nH]1 ZINC000217793360 DG On-Demand Anodyne SCN10A 44 35 O=C(Nc1ncccc1O)c1cc(-c2ccc(Cl)cc2)n[nH]1 ZINC000217793360 DG On-Demand Anodyne ALPL 69 41 O=C(NCc1ccc(F)cc1)c1cc(=O)nc[nH]1 ZINC000217793392 BC In-Stock Unstable NAMPT 29 42 O=C(NCc1ccc(F)cc1)c1cc(=O)nc[nH]1 ZINC000217793392 BC In-Stock Unstable Q76353_9HIV1 0 43 COc1ccccc1NC(=O)N/C=C/c1ccccc1Cl ZINC000217793401 DI For-Sale Unstable CXCL8 41 32 CC1CCN(CCCCOc2ccc(C=O)cc2)CC1 ZINC000217793412 CG In-Stock Unstable ACHE 19 45 CC1CCN(CCCCOc2ccc(C=O)cc2)CC1 ZINC000217793412 CG In-Stock Unstable HTR2A 15 48 CC1CCN(CCCCOc2ccc(C=O)cc2)CC1 ZINC000217793412 CG In-Stock Unstable KCNH2 0 43 CC1CCN(CCCCOc2ccc(C=O)cc2)CC1 ZINC000217793412 CG In-Stock Unstable LTA4H 49 43 CC1CCN(CCCCOc2ccc(C=O)cc2)CC1 ZINC000217793412 CG In-Stock Unstable HRH3 85 48 CC1CCN(CCCCOc2ccc(C=O)cc2)CC1 ZINC000217793412 CG In-Stock Unstable SIGMAR1 24 50 CC1CCN(CCCCOc2ccc(C=O)cc2)CC1 ZINC000217793412 CG In-Stock Unstable EBP 39 63 CC1CCN(CCCCOc2ccc(C=O)cc2)CC1 ZINC000217793412 CG In-Stock Unstable PSMB2 47 38 CC1CCN(CCCCOc2ccc(C=O)cc2)CC1 ZINC000217793412 CG In-Stock Unstable PSMB1 41 38 CC1CCN(CCCCOc2ccc(C=O)cc2)CC1 ZINC000217793412 CG In-Stock Unstable MEN1 51 35 C[C@@H]1CCN([C@H](C)Cc2ccc(O)cc2)C1 ZINC000217793445 BF For-Sale Unstable OPRM1 15 40 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1ccc2c(c1)CCCC2 ZINC000217793456 GF For-Sale Unstable ADAMTS5 33 41 COC(=O)[C@@H](CC(C)C)NC(=O)[C@@H]1C[C@@H](O)CN1 ZINC000217793497 CB For-Sale Unstable NPR 15 40 CC(C)(C)OC(=O)N1CC[C@@H](N)[C@@H](C2CC2)CC1 ZINC000217793506 CE For-Sale Unstable GPR119 37 47 Cc1ccccc1NC(=O)N/C=C/c1ccccc1Cl ZINC000217793508 CI For-Sale Unstable CXCL8 40 39 Cc1ccccc1NC(=O)N/C=C/c1ccccc1Cl ZINC000217793508 CI For-Sale Unstable DDX3X 0 41 C[C@@H]1CCCN(CCCCOc2ccc(C=O)cc2)C1 ZINC000217793518 CG In-Stock Unstable ACHE 15 44 C[C@@H]1CCCN(CCCCOc2ccc(C=O)cc2)C1 ZINC000217793518 CG In-Stock Unstable SLC6A1 76 38 C[C@@H]1CCCN(CCCCOc2ccc(C=O)cc2)C1 ZINC000217793518 CG In-Stock Unstable KCNH2 0 50 C[C@@H]1CCCN(CCCCOc2ccc(C=O)cc2)C1 ZINC000217793518 CG In-Stock Unstable LTA4H 43 38 C[C@@H]1CCCN(CCCCOc2ccc(C=O)cc2)C1 ZINC000217793518 CG In-Stock Unstable HRH3 87 50 C[C@@H]1CCCN(CCCCOc2ccc(C=O)cc2)C1 ZINC000217793518 CG In-Stock Unstable SIGMAR1 15 46 C[C@@H]1CCCN(CCCCOc2ccc(C=O)cc2)C1 ZINC000217793518 CG In-Stock Unstable EBP 26 46 C[C@@H]1CCCN(CCCCOc2ccc(C=O)cc2)C1 ZINC000217793518 CG In-Stock Unstable PSMB2 47 38 C[C@@H]1CCCN(CCCCOc2ccc(C=O)cc2)C1 ZINC000217793518 CG In-Stock Unstable PSMB1 41 38 N#Cc1cccc(OCC2=CCC2)c1 ZINC000217793519 AF In-Stock Unstable CHRNA10 27 49 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1ccc2c(c1)CCCC2 ZINC000217793531 GF For-Sale Unstable ADAMTS5 33 41 CC(C)(C)OC(=O)N1CC[C@@H](C2CC2)[C@H](N)CC1 ZINC000217793584 CE For-Sale Unstable GPR119 37 47 COC(=O)[C@@H](CC(C)C)NC(=O)[C@H]1C[C@@H](O)CN1 ZINC000217793587 CB For-Sale Unstable NPR 15 40 Cc1cccc(NC(=O)c2cc(=O)nc[nH]2)c1 ZINC000217793594 BD In-Stock Unstable CCKAR 15 40 Cc1cccc(NC(=O)c2cc(=O)nc[nH]2)c1 ZINC000217793594 BD In-Stock Unstable F12 0 43 Cc1cccc(NC(=O)c2cc(=O)nc[nH]2)c1 ZINC000217793594 BD In-Stock Unstable SCN10A 28 41 Cc1cccc(NC(=O)c2cc(=O)nc[nH]2)c1 ZINC000217793594 BD In-Stock Unstable SLC11A2 24 46 Cc1cccc(NC(=O)c2cc(=O)nc[nH]2)c1 ZINC000217793594 BD In-Stock Unstable KCNK3 99 49 Cc1cccc(NC(=O)c2cc(=O)nc[nH]2)c1 ZINC000217793594 BD In-Stock Unstable KCNK9 90 49 C[C@H]1CCCN(CCCCOc2ccc(C=O)cc2)C1 ZINC000217793612 CG In-Stock Unstable ACHE 15 44 C[C@H]1CCCN(CCCCOc2ccc(C=O)cc2)C1 ZINC000217793612 CG In-Stock Unstable SLC6A1 76 38 C[C@H]1CCCN(CCCCOc2ccc(C=O)cc2)C1 ZINC000217793612 CG In-Stock Unstable KCNH2 0 50 C[C@H]1CCCN(CCCCOc2ccc(C=O)cc2)C1 ZINC000217793612 CG In-Stock Unstable LTA4H 43 38 C[C@H]1CCCN(CCCCOc2ccc(C=O)cc2)C1 ZINC000217793612 CG In-Stock Unstable HRH3 87 50 C[C@H]1CCCN(CCCCOc2ccc(C=O)cc2)C1 ZINC000217793612 CG In-Stock Unstable SIGMAR1 15 46 C[C@H]1CCCN(CCCCOc2ccc(C=O)cc2)C1 ZINC000217793612 CG In-Stock Unstable EBP 26 46 C[C@H]1CCCN(CCCCOc2ccc(C=O)cc2)C1 ZINC000217793612 CG In-Stock Unstable PSMB2 47 38 C[C@H]1CCCN(CCCCOc2ccc(C=O)cc2)C1 ZINC000217793612 CG In-Stock Unstable PSMB1 41 38 Cc1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1Cl ZINC000217793622 DK For-Sale Unstable LPL 48 33 CC(C)(C)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)cc1 ZINC000217793640 GG For-Sale Unstable ADAMTS5 29 51 COc1ccc(C(=O)N[C@@H](CC(=O)O)c2ccccc2Cl)nc1Br ZINC000217793646 HG Annotated Unstable MME 15 41 COc1ccc(C(=O)N[C@@H](CC(=O)O)c2ccccc2Cl)nc1Br ZINC000217793646 HG Annotated Unstable CTSA 89 44 CC(C)(C)OC(=O)N1CC[C@H](N)[C@@H](C2CC2)CC1 ZINC000217793658 CE For-Sale Unstable GPR119 37 47 COCCN(CC(=O)O)C(=O)/C=C\c1ccc(Cl)cc1Cl ZINC000217793660 EF For-Sale Unstable BOTA 24 44 CC(C)(C)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)cc1 ZINC000217793680 GG For-Sale Unstable ADAMTS5 37 51 COc1ccc(C(=O)N[C@H](CC(=O)O)c2ccccc2Cl)nc1Br ZINC000217793711 HG Annotated Unstable MME 15 41 COc1ccc(C(=O)N[C@H](CC(=O)O)c2ccccc2Cl)nc1Br ZINC000217793711 HG Annotated Unstable CTSA 89 44 CC(C)(C)OC(=O)N1CC[C@H](N)[C@H](C2CC2)CC1 ZINC000217793717 CE For-Sale Unstable GPR119 37 47 Cc1cccc(C(C)C)c1NC(=O)N/C=C/c1ccccc1Cl ZINC000217793732 EK For-Sale Unstable CXCL8 33 44 Cc1cccc(C(C)C)c1NC(=O)N/C=C/c1ccccc1Cl ZINC000217793732 EK For-Sale Unstable SOAT1 48 41 Cc1cccc(C(C)C)c1NC(=O)N/C=C/c1ccccc1Cl ZINC000217793732 EK For-Sale Unstable ACAT 0 45 C[C@@H]1CCC[C@@H](C)N1CCCCOc1ccc(C=O)cc1 ZINC000217793736 CH In-Stock Unstable LTA4H 29 56 C[C@@H]1CCC[C@@H](C)N1CCCCOc1ccc(C=O)cc1 ZINC000217793736 CH In-Stock Unstable HRH3 51 42 Cc1ccccc1-c1cc(C(=O)Nc2ccnn2[C@@H](C)C2CC2)c2cnn(C(C)C)c2n1 ZINC000217793748 IK On-Demand Unstable EZH2 15 43 Cn1nc(OCC2CC2)c2cc(N)ccc21 ZINC000217793752 BD In-Stock Unstable HTR4 71 36 O=C(Nc1ccc(Cl)cc1)c1cc(=O)nc[nH]1 ZINC000217793785 BD In-Stock Anodyne P95276_MYCTO 0 43 C[C@@H]1CCN([C@H](C)CCc2ccc(O)cc2)C1 ZINC000217793797 BG For-Sale Unstable ERG2 17 40 C[C@H]1CCC[C@@H](C)N1CCCCOc1ccc(C=O)cc1 ZINC000217793803 CH In-Stock Unstable LTA4H 29 56 C[C@H]1CCC[C@@H](C)N1CCCCOc1ccc(C=O)cc1 ZINC000217793803 CH In-Stock Unstable HRH3 51 42 Cc1ccccc1-c1cc(C(=O)Nc2ccnn2[C@H](C)C2CC2)c2cnn(C(C)C)c2n1 ZINC000217793818 IK On-Demand Unstable EZH2 15 43 CC(C)(C)OC(=O)N1CC[C@H](C2CCC2)[C@H](N)C1 ZINC000217793836 CE For-Sale Unstable GPR119 30 42 CC(C)(C)OC(=O)N1CC[C@@H](C2CCC2)[C@H](N)C1 ZINC000217793877 CE For-Sale Unstable GPR119 30 42 CS(=O)(=O)Nc1cccc(NC(=O)c2cc(=O)nc[nH]2)c1 ZINC000217793906 DC In-Stock Unstable KCNK3 81 38 CS(=O)(=O)Nc1cccc(NC(=O)c2cc(=O)nc[nH]2)c1 ZINC000217793906 DC In-Stock Unstable KCNK9 72 37 C[C@H]1CCC[C@H](C)N1CCCCOc1ccc(C=O)cc1 ZINC000217793908 CH In-Stock Unstable LTA4H 29 56 C[C@H]1CCC[C@H](C)N1CCCCOc1ccc(C=O)cc1 ZINC000217793908 CH In-Stock Unstable HRH3 51 42 CN(CCc1ccncc1)C(=O)[C@@H]1CCCN1C(=O)C1CCCCC1 ZINC000217793926 EF In-Stock Unstable FKBP1A 41 41 CN(CCc1ccncc1)C(=O)[C@@H]1CCCN1C(=O)C1CCCCC1 ZINC000217793926 EF In-Stock Unstable PREP 81 37 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(C(=O)O)cc1 ZINC000217793935 DH For-Sale Anodyne SMO 23 44 CC(C)(C)OC(=O)N1CC[C@H](C2CCC2)[C@@H](N)C1 ZINC000217793963 CE For-Sale Unstable GPR119 30 42 C[C@@H]1C[C@@H](C)CN(CCCCOc2ccc(C=O)cc2)C1 ZINC000217794017 CH In-Stock Unstable HRH3 55 40 C[C@@H]1C[C@@H](C)CN(CCCCOc2ccc(C=O)cc2)C1 ZINC000217794017 CH In-Stock Unstable EBP 19 43 Cc1c(Cl)cccc1NC(=O)N/C=C/c1ccccc1Cl ZINC000217794018 DK For-Sale Unstable CXCL8 44 36 Cc1ccnc(NS(=O)(=O)c2ccc(NC(=O)c3cc(=O)nc[nH]3)cc2)n1 ZINC000217794019 GC In-Stock Unstable GRM4 16 42 Cc1ccnc(NS(=O)(=O)c2ccc(NC(=O)c3cc(=O)nc[nH]3)cc2)n1 ZINC000217794019 GC In-Stock Unstable SMG1 48 31 CC(=O)Nc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)cc1 ZINC000217794023 GE For-Sale Unstable ADAMTS5 34 42 O=C(O)Cc1cc(I)ccc1O ZINC000217794039 CD For-Sale Unstable THRA 41 43 O=C(O)Cc1cc(I)ccc1O ZINC000217794039 CD For-Sale Unstable THRB 25 43 O=C(O)Cc1cc(I)ccc1O ZINC000217794039 CD For-Sale Unstable CAN2 0 45 O=C(O)Cc1cc(I)ccc1O ZINC000217794039 CD For-Sale Unstable SLCO1C1 0 43 CC(C)(C)OC(=O)N1CC[C@@H](C2CCC2)[C@@H](N)C1 ZINC000217794049 CE For-Sale Unstable GPR119 30 42 CC(=O)Nc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)cc1 ZINC000217794092 GE For-Sale Unstable ADAMTS5 34 42 C[C@H]1C[C@@H](C)CN(CCCCOc2ccc(C=O)cc2)C1 ZINC000217794098 CH In-Stock Unstable HRH3 55 40 C[C@H]1C[C@@H](C)CN(CCCCOc2ccc(C=O)cc2)C1 ZINC000217794098 CH In-Stock Unstable EBP 19 43 O=C(Nc1ccc(OCc2ccccc2)cc1)c1cc(=O)nc[nH]1 ZINC000217794117 DF In-Stock Unstable TSHR 59 37 O=C(Nc1ccc(OCc2ccccc2)cc1)c1cc(=O)nc[nH]1 ZINC000217794117 DF In-Stock Unstable PPIA 45 35 O=C(Nc1ccc(OCc2ccccc2)cc1)c1cc(=O)nc[nH]1 ZINC000217794117 DF In-Stock Unstable LTA4H 28 48 O=C(Nc1ccc(OCc2ccccc2)cc1)c1cc(=O)nc[nH]1 ZINC000217794117 DF In-Stock Unstable HRAS 46 30 O=C(Nc1ccc(OCc2ccccc2)cc1)c1cc(=O)nc[nH]1 ZINC000217794117 DF In-Stock Unstable ADAM17 25 45 O=C(Nc1ccc(OCc2ccccc2)cc1)c1cc(=O)nc[nH]1 ZINC000217794117 DF In-Stock Unstable FFAR1 38 44 O=C(Nc1ccc(OCc2ccccc2)cc1)c1cc(=O)nc[nH]1 ZINC000217794117 DF In-Stock Unstable YOPH 0 42 O=C(Nc1ccc(OCc2ccccc2)cc1)c1cc(=O)nc[nH]1 ZINC000217794117 DF In-Stock Unstable SENP1 0 40 CCOC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217794122 EI For-Sale Unstable CA1 18 43 CCOC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217794122 EI For-Sale Unstable ACR 63 36 CCOC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217794122 EI For-Sale Unstable NOD2 17 42 CCOC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217794122 EI For-Sale Unstable SENP1 0 41 CC(C)(C)OC(=O)N1CC[C@H](CN)[C@H](C2CC2)C1 ZINC000217794124 CE For-Sale Unstable GPR119 33 42 Cc1ccc(-c2cnc(CCC(=O)Nc3ccc(N4CCOCC4)cc3N3CCOCC3)o2)cc1 ZINC000217794128 JH On-Demand Unstable PRKDC 65 33 Cc1ccc(-c2cnc(CCC(=O)Nc3ccc(N4CCOCC4)cc3N3CCOCC3)o2)cc1 ZINC000217794128 JH On-Demand Unstable CSF1R 0 42 Cc1ccc(-c2cnc(CCC(=O)Nc3ccc(N4CCOCC4)cc3N3CCOCC3)o2)cc1 ZINC000217794128 JH On-Demand Unstable AKR1C3 0 40 COCCN(CC(=O)O)C(=O)/C=C\c1cccc(Cl)c1 ZINC000217794132 CD On-Demand Unstable NR1H4 22 40 COCCN(CC(=O)O)C(=O)/C=C\c1cccc(Cl)c1 ZINC000217794132 CD On-Demand Unstable TUBA4A 0 41 CC(C)(C)OC(=O)N1CC[C@@H](CN)[C@H](C2CC2)C1 ZINC000217794168 CE For-Sale Unstable GPR119 33 42 C[C@H]1C[C@H](C)CN(CCCCOc2ccc(C=O)cc2)C1 ZINC000217794188 CH In-Stock Unstable HRH3 55 40 C[C@H]1C[C@H](C)CN(CCCCOc2ccc(C=O)cc2)C1 ZINC000217794188 CH In-Stock Unstable EBP 19 43 O=C(N/C=C/c1ccccc1Cl)Nc1ccccc1Cl ZINC000217794212 DJ For-Sale Anodyne CXCL8 53 40 O=C(N/C=C/c1ccccc1Cl)Nc1ccccc1Cl ZINC000217794212 DJ For-Sale Anodyne EPHB3 51 35 CC(C)(C)OC(=O)N1CC[C@H](CN)[C@@H](C2CC2)C1 ZINC000217794247 CE For-Sale Unstable GPR119 33 42 COc1cc([C@@H](C)N2CC[C@@H](C)C2)ccc1O ZINC000217794268 BF For-Sale Unstable PNLIP 0 48 COc1cc([C@@H](C)N2CC[C@@H](C)C2)ccc1O ZINC000217794268 BF For-Sale Unstable N1L 0 49 COc1cc([C@@H](C)N2CC[C@@H](C)C2)ccc1O ZINC000217794268 BF For-Sale Unstable RORC 50 38 COc1cc([C@@H](C)N2CC[C@@H](C)C2)ccc1O ZINC000217794268 BF For-Sale Unstable SLC22A3 0 42 O=Cc1ccc(OCCCCN2CCN(c3ccccc3)CC2)cc1 ZINC000217794308 EG In-Stock Unstable HTR1A 110 70 O=Cc1ccc(OCCCCN2CCN(c3ccccc3)CC2)cc1 ZINC000217794308 EG In-Stock Unstable DRD2 74 66 O=Cc1ccc(OCCCCN2CCN(c3ccccc3)CC2)cc1 ZINC000217794308 EG In-Stock Unstable DRD1 37 50 O=Cc1ccc(OCCCCN2CCN(c3ccccc3)CC2)cc1 ZINC000217794308 EG In-Stock Unstable DRD4 45 46 O=Cc1ccc(OCCCCN2CCN(c3ccccc3)CC2)cc1 ZINC000217794308 EG In-Stock Unstable ACHE 28 44 O=Cc1ccc(OCCCCN2CCN(c3ccccc3)CC2)cc1 ZINC000217794308 EG In-Stock Unstable ADRA1D 22 40 O=Cc1ccc(OCCCCN2CCN(c3ccccc3)CC2)cc1 ZINC000217794308 EG In-Stock Unstable HTR2A 72 53 O=Cc1ccc(OCCCCN2CCN(c3ccccc3)CC2)cc1 ZINC000217794308 EG In-Stock Unstable HTR2C 28 41 O=Cc1ccc(OCCCCN2CCN(c3ccccc3)CC2)cc1 ZINC000217794308 EG In-Stock Unstable SLC6A4 20 44 O=Cc1ccc(OCCCCN2CCN(c3ccccc3)CC2)cc1 ZINC000217794308 EG In-Stock Unstable ADRA1A 33 53 O=Cc1ccc(OCCCCN2CCN(c3ccccc3)CC2)cc1 ZINC000217794308 EG In-Stock Unstable HRH1 24 70 O=Cc1ccc(OCCCCN2CCN(c3ccccc3)CC2)cc1 ZINC000217794308 EG In-Stock Unstable DRD3 76 70 O=Cc1ccc(OCCCCN2CCN(c3ccccc3)CC2)cc1 ZINC000217794308 EG In-Stock Unstable KCNH2 23 59 O=Cc1ccc(OCCCCN2CCN(c3ccccc3)CC2)cc1 ZINC000217794308 EG In-Stock Unstable DRD5 49 47 O=Cc1ccc(OCCCCN2CCN(c3ccccc3)CC2)cc1 ZINC000217794308 EG In-Stock Unstable LTA4H 72 45 O=Cc1ccc(OCCCCN2CCN(c3ccccc3)CC2)cc1 ZINC000217794308 EG In-Stock Unstable HTR7 117 54 O=Cc1ccc(OCCCCN2CCN(c3ccccc3)CC2)cc1 ZINC000217794308 EG In-Stock Unstable HRH3 70 47 O=Cc1ccc(OCCCCN2CCN(c3ccccc3)CC2)cc1 ZINC000217794308 EG In-Stock Unstable SIGMAR1 46 47 O=Cc1ccc(OCCCCN2CCN(c3ccccc3)CC2)cc1 ZINC000217794308 EG In-Stock Unstable BCHE 23 44 O=Cc1ccc(OCCCCN2CCN(c3ccccc3)CC2)cc1 ZINC000217794308 EG In-Stock Unstable HTR6 0 44 O=Cc1ccc(OCCCCN2CCN(c3ccccc3)CC2)cc1 ZINC000217794308 EG In-Stock Unstable PLA2G4B 40 35 O=Cc1ccc(OCCCCN2CCN(c3ccccc3)CC2)cc1 ZINC000217794308 EG In-Stock Unstable ABCB1 24 45 O=Cc1ccc(OCCCCN2CCN(c3ccccc3)CC2)cc1 ZINC000217794308 EG In-Stock Unstable EPHX2 17 46 O=Cc1ccc(OCCCCN2CCN(c3ccccc3)CC2)cc1 ZINC000217794308 EG In-Stock Unstable PSMB2 50 41 O=Cc1ccc(OCCCCN2CCN(c3ccccc3)CC2)cc1 ZINC000217794308 EG In-Stock Unstable PSMB5 17 41 O=Cc1ccc(OCCCCN2CCN(c3ccccc3)CC2)cc1 ZINC000217794308 EG In-Stock Unstable PSMB1 43 41 O=Cc1ccc(OCCCCN2CCN(c3ccccc3)CC2)cc1 ZINC000217794308 EG In-Stock Unstable MEN1 46 35 O=Cc1ccc(OCCCCN2CCN(c3ccccc3)CC2)cc1 ZINC000217794308 EG In-Stock Unstable AP2S1 0 41 CC(C)c1ccccc1NC(=O)N/C=C/c1ccccc1Cl ZINC000217794337 DK For-Sale Unstable CXCL8 44 39 O=C(CC[C@@H]1NC(=O)N(Cc2ccc3c(c2)OCO3)C1=O)NCCc1ccc(O)cc1 ZINC000217794364 ID In-Stock Unstable NOS2 70 36 O=C(CC[C@@H]1NC(=O)N(Cc2ccc3c(c2)OCO3)C1=O)NCCc1ccc(O)cc1 ZINC000217794364 ID In-Stock Unstable MCHR1 23 41 O=C(c1ccno1)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217794367 FF In-Stock Unstable HRH3 23 42 CC(C)(C)OC(=O)N1CC[C@@H](CN)[C@@H](C2CC2)C1 ZINC000217794386 CE For-Sale Unstable GPR119 33 42 CCN(CC)CCCCOc1cccc(C=O)c1 ZINC000217794415 BF In-Stock Unstable THRA 0 40 CCN(CC)CCCCOc1cccc(C=O)c1 ZINC000217794415 BF In-Stock Unstable ACHE 28 52 CCN(CC)CCCCOc1cccc(C=O)c1 ZINC000217794415 BF In-Stock Unstable BCHE 16 48 CCN(CC)CCCCOc1cccc(C=O)c1 ZINC000217794415 BF In-Stock Unstable SQLE 49 34 CCN(CC)CCCCOc1cccc(C=O)c1 ZINC000217794415 BF In-Stock Unstable GALR3 31 40 O=C(N/C=C/c1ccccc1Cl)Nc1cccc(Cl)c1Cl ZINC000217794421 EK For-Sale Anodyne CXCL8 42 35 COc1cc(C)c(C)cc1S(=O)(=O)NC[C@@H]1CCCN1c1nccs1 ZINC000217794431 GF For-Sale Unstable ADAMTS5 29 40 O=C(c1ccno1)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217794446 FF In-Stock Unstable HRH3 23 42 C[C@@H](c1ccccc1F)N(C)C[C@@H](O)c1cccc(N)c1 ZINC000217794481 CG For-Sale Unstable AOC3 29 40 CC(C)(C)OC(=O)N1CC[C@H](N)[C@H](C2CCC2)C1 ZINC000217794482 CE For-Sale Unstable GPR119 30 42 COc1cccc(NC(=O)CC/C(C)=C/Cc2c(O)c3c(c(C)c2OC)COC3=O)c1 ZINC000217794484 II In-Stock Unstable IMPDH1 0 70 COc1cccc(NC(=O)CC/C(C)=C/Cc2c(O)c3c(c(C)c2OC)COC3=O)c1 ZINC000217794484 II In-Stock Unstable MTNR1A 17 41 COc1cccc(NC(=O)CC/C(C)=C/Cc2c(O)c3c(c(C)c2OC)COC3=O)c1 ZINC000217794484 II In-Stock Unstable MTNR1B 18 41 COc1cccc(NC(=O)CC/C(C)=C/Cc2c(O)c3c(c(C)c2OC)COC3=O)c1 ZINC000217794484 II In-Stock Unstable IMPDH2 0 70 COc1cc(C)c(C)cc1S(=O)(=O)NC[C@H]1CCCN1c1nccs1 ZINC000217794509 GF For-Sale Unstable ADAMTS5 29 40 COCCN(CC(=O)O)C(=O)/C=C\c1ccc(Cl)c(Cl)c1 ZINC000217794519 EF For-Sale Unstable PYGL 0 45 O=Cc1cccc(OCCCCN2CCCC2)c1 ZINC000217794565 BF In-Stock Unstable HTR1A 17 41 O=Cc1cccc(OCCCCN2CCCC2)c1 ZINC000217794565 BF In-Stock Unstable DRD2 26 44 O=Cc1cccc(OCCCCN2CCCC2)c1 ZINC000217794565 BF In-Stock Unstable DRD1 15 44 O=Cc1cccc(OCCCCN2CCCC2)c1 ZINC000217794565 BF In-Stock Unstable ACHE 29 49 O=Cc1cccc(OCCCCN2CCCC2)c1 ZINC000217794565 BF In-Stock Unstable HRH2 34 42 O=Cc1cccc(OCCCCN2CCCC2)c1 ZINC000217794565 BF In-Stock Unstable HTR2A 20 44 O=Cc1cccc(OCCCCN2CCCC2)c1 ZINC000217794565 BF In-Stock Unstable SLC6A4 16 41 O=Cc1cccc(OCCCCN2CCCC2)c1 ZINC000217794565 BF In-Stock Unstable DRD3 19 44 O=Cc1cccc(OCCCCN2CCCC2)c1 ZINC000217794565 BF In-Stock Unstable KCNH2 17 40 O=Cc1cccc(OCCCCN2CCCC2)c1 ZINC000217794565 BF In-Stock Unstable DRD5 24 40 O=Cc1cccc(OCCCCN2CCCC2)c1 ZINC000217794565 BF In-Stock Unstable LTA4H 50 51 O=Cc1cccc(OCCCCN2CCCC2)c1 ZINC000217794565 BF In-Stock Unstable HRH3 81 51 O=Cc1cccc(OCCCCN2CCCC2)c1 ZINC000217794565 BF In-Stock Unstable SIGMAR1 37 46 O=Cc1cccc(OCCCCN2CCCC2)c1 ZINC000217794565 BF In-Stock Unstable BCHE 21 43 O=Cc1cccc(OCCCCN2CCCC2)c1 ZINC000217794565 BF In-Stock Unstable CHRNA7 0 45 O=Cc1cccc(OCCCCN2CCCC2)c1 ZINC000217794565 BF In-Stock Unstable HNMT 60 35 O=Cc1cccc(OCCCCN2CCCC2)c1 ZINC000217794565 BF In-Stock Unstable EPHX2 21 45 O=Cc1cccc(OCCCCN2CCCC2)c1 ZINC000217794565 BF In-Stock Unstable PSMB2 52 42 O=Cc1cccc(OCCCCN2CCCC2)c1 ZINC000217794565 BF In-Stock Unstable PSMB5 18 42 O=Cc1cccc(OCCCCN2CCCC2)c1 ZINC000217794565 BF In-Stock Unstable PSMB1 45 42 C/C=C\c1ccc(OC[C@](C)(O)C(=O)O)c(OC)c1 ZINC000217794566 CD For-Sale Unstable CYP1B1 19 42 C/C=C\c1ccc(OC[C@](C)(O)C(=O)O)c(OC)c1 ZINC000217794566 CD For-Sale Unstable APP 21 43 C/C=C\c1ccc(OC[C@](C)(O)C(=O)O)c(OC)c1 ZINC000217794566 CD For-Sale Unstable CYP1A1 21 42 C/C=C\c1ccc(OC[C@](C)(O)C(=O)O)c(OC)c1 ZINC000217794566 CD For-Sale Unstable TUBB1 57 40 CC(C)(C)OC(=O)N1CC[C@@H](N)[C@H](C2CCC2)C1 ZINC000217794573 CE For-Sale Unstable GPR119 30 42 C[C@H](c1ccccc1F)N(C)C[C@@H](O)c1cccc(N)c1 ZINC000217794578 CG For-Sale Unstable AOC3 29 40 C[C@@H]1CCN([C@H](C)c2cc(Cl)ccc2O)C1 ZINC000217794637 BG For-Sale Unstable EBP 19 41 C[C@@H](c1ccccc1F)N(C)C[C@@H](O)c1ccccc1N ZINC000217794640 CG For-Sale Unstable AOC3 15 40 C/C=C\c1ccc(OC[C@@](C)(O)C(=O)O)c(OC)c1 ZINC000217794641 CD For-Sale Unstable CYP1B1 19 42 C/C=C\c1ccc(OC[C@@](C)(O)C(=O)O)c(OC)c1 ZINC000217794641 CD For-Sale Unstable APP 21 43 C/C=C\c1ccc(OC[C@@](C)(O)C(=O)O)c(OC)c1 ZINC000217794641 CD For-Sale Unstable CYP1A1 21 42 C/C=C\c1ccc(OC[C@@](C)(O)C(=O)O)c(OC)c1 ZINC000217794641 CD For-Sale Unstable TUBB1 57 40 CC(C)(C)OC(=O)N1CC[C@H](N)[C@@H](C2CCC2)C1 ZINC000217794647 CE For-Sale Unstable GPR119 30 42 COc1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1Cl ZINC000217794652 EJ For-Sale Unstable GCGR 0 42 COc1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1Cl ZINC000217794652 EJ For-Sale Unstable GRM4 25 52 COc1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1Cl ZINC000217794652 EJ For-Sale Unstable IMPDH2 0 48 COc1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1Cl ZINC000217794652 EJ For-Sale Unstable CYSP_PLAFA 41 36 COC(=O)c1cccc(S(=O)(=O)N[C@@H](C(=O)OC(C)(C)C)c2ccccc2)c1 ZINC000217794654 HF On-Demand Unstable TRY2_BOVIN 43 33 O=C(NCl)c1cccc(C(=O)NCl)n1 ZINC000217794669 BC For-Sale Anodyne GRM4 18 41 CC1CCN(CCCCOc2cccc(C=O)c2)CC1 ZINC000217794672 CG In-Stock Unstable HTR1A 15 40 CC1CCN(CCCCOc2cccc(C=O)c2)CC1 ZINC000217794672 CG In-Stock Unstable DRD2 22 42 CC1CCN(CCCCOc2cccc(C=O)c2)CC1 ZINC000217794672 CG In-Stock Unstable ACHE 20 41 CC1CCN(CCCCOc2cccc(C=O)c2)CC1 ZINC000217794672 CG In-Stock Unstable HRH3 62 40 CC1CCN(CCCCOc2cccc(C=O)c2)CC1 ZINC000217794672 CG In-Stock Unstable SIGMAR1 26 50 CC1CCN(CCCCOc2cccc(C=O)c2)CC1 ZINC000217794672 CG In-Stock Unstable EBP 40 51 CC1CCN(CCCCOc2cccc(C=O)c2)CC1 ZINC000217794672 CG In-Stock Unstable EPHX2 20 44 CC1CCN(CCCCOc2cccc(C=O)c2)CC1 ZINC000217794672 CG In-Stock Unstable CHRNA10 42 36 CC1CCN(CCCCOc2cccc(C=O)c2)CC1 ZINC000217794672 CG In-Stock Unstable MEN1 43 32 O=C(NCc1ccccn1)[C@@H]1CC[C@@H](CNS(=O)(=O)c2ccccc2)CC1 ZINC000217794704 GE In-Stock Unstable NPY2R 86 55 O=C(NCc1ccccn1)[C@@H]1CC[C@@H](CNS(=O)(=O)c2ccccc2)CC1 ZINC000217794704 GE In-Stock Unstable NPY5R 29 55 O=C(NCc1ccccn1)[C@@H]1CC[C@@H](CNS(=O)(=O)c2ccccc2)CC1 ZINC000217794704 GE In-Stock Unstable VCP 43 36 CC(C)(C)OC(=O)N1CC[C@@H](N)[C@@H](C2CCC2)C1 ZINC000217794724 CE For-Sale Unstable GPR119 30 42 COC(=O)c1cccc(S(=O)(=O)N[C@H](C(=O)OC(C)(C)C)c2ccccc2)c1 ZINC000217794728 HF On-Demand Unstable TRY2_BOVIN 43 33 C[C@@H]1CCCCN1CCCCOc1cccc(C=O)c1 ZINC000217794735 CH In-Stock Unstable HTR3A 25 48 C[C@@H]1CCCCN1CCCCOc1cccc(C=O)c1 ZINC000217794735 CH In-Stock Unstable KCNH2 0 46 C[C@@H]1CCCCN1CCCCOc1cccc(C=O)c1 ZINC000217794735 CH In-Stock Unstable HRH3 84 45 O=C(/C=C/c1ccco1)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217794747 GH In-Stock Unstable HRH3 22 41 C[C@@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1ccc2c(c1)OCO2 ZINC000217794750 CC On-Demand Unstable KCNQ2 22 47 C[C@@H]1CCN([C@H](C)c2cccc(O)c2)C1 ZINC000217794760 BF For-Sale Unstable OPRM1 15 51 C[C@H](c1ccccc1F)N(C)C[C@@H](O)c1ccccc1N ZINC000217794761 CG For-Sale Unstable AOC3 15 40 O=C(N/C=C/c1ccccc1Cl)Nc1cccc(C(F)(F)F)c1 ZINC000217794768 EK For-Sale Anodyne KIT 15 40 O=C(N/C=C/c1ccccc1Cl)Nc1cccc(C(F)(F)F)c1 ZINC000217794768 EK For-Sale Anodyne KDR 15 40 O=C(N/C=C/c1ccccc1Cl)Nc1cccc(C(F)(F)F)c1 ZINC000217794768 EK For-Sale Anodyne EPHX2 16 46 O=C(N/C=C/c1ccccc1Cl)Nc1cccc(C(F)(F)F)c1 ZINC000217794768 EK For-Sale Anodyne TYK2 22 40 O=C(N/C=C/c1ccccc1Cl)Nc1cccc(C(F)(F)F)c1 ZINC000217794768 EK For-Sale Anodyne TEK 25 40 O=C(N/C=C/c1ccccc1Cl)Nc1cccc(C(F)(F)F)c1 ZINC000217794768 EK For-Sale Anodyne BRAF 17 40 O=C(N/C=C/c1ccccc1Cl)Nc1cccc(C(F)(F)F)c1 ZINC000217794768 EK For-Sale Anodyne RIPK1 45 39 O=C(N/C=C/c1ccccc1Cl)Nc1cccc(C(F)(F)F)c1 ZINC000217794768 EK For-Sale Anodyne IMDH_CRYPV 48 40 O=C(N/C=C/c1ccccc1Cl)Nc1cccc(C(F)(F)F)c1 ZINC000217794768 EK For-Sale Anodyne TRPM4 0 41 O=C(N/C=C/c1ccccc1Cl)Nc1cccc(C(F)(F)F)c1 ZINC000217794768 EK For-Sale Anodyne KCNK3 49 47 C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1ccc2c(c1)OCO2 ZINC000217794800 CC On-Demand Unstable KCNQ2 22 47 O=C(/C=C/c1ccco1)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217794809 GH In-Stock Unstable HRH3 22 41 CCOc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)cc1C ZINC000217794820 GF For-Sale Unstable ADAMTS5 32 46 C[C@H]1CCCCN1CCCCOc1cccc(C=O)c1 ZINC000217794822 CH In-Stock Unstable HTR3A 25 48 C[C@H]1CCCCN1CCCCOc1cccc(C=O)c1 ZINC000217794822 CH In-Stock Unstable KCNH2 0 46 C[C@H]1CCCCN1CCCCOc1cccc(C=O)c1 ZINC000217794822 CH In-Stock Unstable HRH3 84 45 C[C@@H](c1ccccc1F)N(C)C[C@@H](O)c1ccc(N)cc1 ZINC000217794849 CG For-Sale Unstable AOC3 22 43 C[C@@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1ccc2c(c1)OCO2 ZINC000217794876 CC On-Demand Unstable KCNQ2 22 47 CCOc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)cc1C ZINC000217794911 GF For-Sale Unstable ADAMTS5 32 46 C[C@H](c1ccccc1F)N(C)C[C@@H](O)c1ccc(N)cc1 ZINC000217794913 CG For-Sale Unstable AOC3 22 43 Cn1cccc(C(=O)N2CCC[C@H](Cc3nc(-c4ccccc4F)no3)C2)c1=O ZINC000217794916 GF In-Stock Unstable HRH3 25 45 C[C@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1ccc2c(c1)OCO2 ZINC000217794949 CC On-Demand Unstable KCNQ2 22 47 Cc1nc(C2CCN(C(=O)c3cc4sccc4[nH]3)CC2)no1 ZINC000217794957 DF In-Stock Unstable HRH4 31 57 Cc1nc(C2CCN(C(=O)c3cc4sccc4[nH]3)CC2)no1 ZINC000217794957 DF In-Stock Unstable AKR1C3 0 41 Cc1nc(C2CCN(C(=O)c3cc4sccc4[nH]3)CC2)no1 ZINC000217794957 DF In-Stock Unstable ETHR 49 39 CCCc1nc2ccccc2n1CC(=O)OCC ZINC000217794964 BF For-Sale Unstable AGTR1 47 44 CCCc1nc2ccccc2n1CC(=O)OCC ZINC000217794964 BF For-Sale Unstable PIN4 0 43 CCCc1nc2ccccc2n1CC(=O)OCC ZINC000217794964 BF For-Sale Unstable AGTR1B 34 43 CCCc1nc2ccccc2n1CC(=O)OCC ZINC000217794964 BF For-Sale Unstable CA13 15 48 CCCc1nc2ccccc2n1CC(=O)OCC ZINC000217794964 BF For-Sale Unstable RPS6KB1 21 40 CCCc1nc2ccccc2n1CC(=O)OCC ZINC000217794964 BF For-Sale Unstable PTGDR2 16 48 Cn1cccc(C(=O)N2CCC[C@@H](Cc3nc(-c4ccccc4F)no3)C2)c1=O ZINC000217794993 GF In-Stock Unstable HRH3 25 45 COc1ccc(S(=O)(=O)N2CCC(N3CCC(OC)CC3)CC2)cc1Cl ZINC000217795017 HF In-Stock Unstable CHRM2 56 43 COc1ccc(S(=O)(=O)N2CCC(N3CCC(OC)CC3)CC2)cc1Cl ZINC000217795017 HF In-Stock Unstable HRH1 18 44 COc1ccc(S(=O)(=O)N2CCC(N3CCC(OC)CC3)CC2)cc1Cl ZINC000217795017 HF In-Stock Unstable CCR3 18 44 COc1ccc(S(=O)(=O)N2CCC(N3CCC(OC)CC3)CC2)cc1Cl ZINC000217795017 HF In-Stock Unstable HTR6 15 42 COc1c(C)cc(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)cc1C ZINC000217795058 GF For-Sale Unstable ADAMTS5 30 41 O=C(/C=C/c1ccccc1Cl)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217795112 IK In-Stock Unstable HRH3 17 42 COc1c(C)cc(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)cc1C ZINC000217795131 GF For-Sale Unstable ADAMTS5 30 41 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(O)cc1 ZINC000217795146 CH For-Sale Anodyne SMO 15 40 O=C(/C=C/c1ccccc1Cl)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217795205 IK In-Stock Unstable HRH3 17 42 Nc1nc(CN2CCN(CCOc3cccc(Cl)c3)CC2)nc2ccccc12 ZINC000217795207 GG On-Demand Unstable HTR1A 18 44 Nc1nc(CN2CCN(CCOc3cccc(Cl)c3)CC2)nc2ccccc12 ZINC000217795207 GG On-Demand Unstable DRD2 17 40 Nc1nc(CN2CCN(CCOc3cccc(Cl)c3)CC2)nc2ccccc12 ZINC000217795207 GG On-Demand Unstable ACHE 20 42 Nc1nc(CN2CCN(CCOc3cccc(Cl)c3)CC2)nc2ccccc12 ZINC000217795207 GG On-Demand Unstable HTR1D 19 44 Nc1nc(CN2CCN(CCOc3cccc(Cl)c3)CC2)nc2ccccc12 ZINC000217795207 GG On-Demand Unstable LTA4H 42 42 Nc1nc(CN2CCN(CCOc3cccc(Cl)c3)CC2)nc2ccccc12 ZINC000217795207 GG On-Demand Unstable HTR7 16 42 Nc1nc(CN2CCN(CCOc3cccc(Cl)c3)CC2)nc2ccccc12 ZINC000217795207 GG On-Demand Unstable HRH3 17 47 Nc1nc(CN2CCN(CCOc3cccc(Cl)c3)CC2)nc2ccccc12 ZINC000217795207 GG On-Demand Unstable NORA 0 44 O=Cc1cccc(OCCCCN2CCCCCC2)c1 ZINC000217795222 CH In-Stock Unstable ESR1 46 37 O=Cc1cccc(OCCCCN2CCCCCC2)c1 ZINC000217795222 CH In-Stock Unstable HTR1A 15 40 O=Cc1cccc(OCCCCN2CCCCCC2)c1 ZINC000217795222 CH In-Stock Unstable DRD2 24 43 O=Cc1cccc(OCCCCN2CCCCCC2)c1 ZINC000217795222 CH In-Stock Unstable ACHE 30 51 O=Cc1cccc(OCCCCN2CCCCCC2)c1 ZINC000217795222 CH In-Stock Unstable HRH2 38 44 O=Cc1cccc(OCCCCN2CCCCCC2)c1 ZINC000217795222 CH In-Stock Unstable HTR2A 19 43 O=Cc1cccc(OCCCCN2CCCCCC2)c1 ZINC000217795222 CH In-Stock Unstable SLC6A4 17 43 O=Cc1cccc(OCCCCN2CCCCCC2)c1 ZINC000217795222 CH In-Stock Unstable DRD3 17 43 O=Cc1cccc(OCCCCN2CCCCCC2)c1 ZINC000217795222 CH In-Stock Unstable KCNH2 17 42 O=Cc1cccc(OCCCCN2CCCCCC2)c1 ZINC000217795222 CH In-Stock Unstable LTA4H 48 50 O=Cc1cccc(OCCCCN2CCCCCC2)c1 ZINC000217795222 CH In-Stock Unstable HRH3 85 53 O=Cc1cccc(OCCCCN2CCCCCC2)c1 ZINC000217795222 CH In-Stock Unstable SIGMAR1 37 47 O=Cc1cccc(OCCCCN2CCCCCC2)c1 ZINC000217795222 CH In-Stock Unstable NPY1R 40 33 O=Cc1cccc(OCCCCN2CCCCCC2)c1 ZINC000217795222 CH In-Stock Unstable BCHE 20 45 O=Cc1cccc(OCCCCN2CCCCCC2)c1 ZINC000217795222 CH In-Stock Unstable CHRNA7 22 40 O=Cc1cccc(OCCCCN2CCCCCC2)c1 ZINC000217795222 CH In-Stock Unstable HNMT 69 34 O=Cc1cccc(OCCCCN2CCCCCC2)c1 ZINC000217795222 CH In-Stock Unstable ABCB1 18 41 O=Cc1cccc(OCCCCN2CCCCCC2)c1 ZINC000217795222 CH In-Stock Unstable EPHX2 20 47 O=Cc1cccc(OCCCCN2CCCCCC2)c1 ZINC000217795222 CH In-Stock Unstable PSMB2 55 44 O=Cc1cccc(OCCCCN2CCCCCC2)c1 ZINC000217795222 CH In-Stock Unstable PSMB5 19 44 O=Cc1cccc(OCCCCN2CCCCCC2)c1 ZINC000217795222 CH In-Stock Unstable PSMB1 47 44 CCc1ccc(OC)c(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217795246 GF For-Sale Unstable ADAMTS5 32 40 COc1ccc(Cl)cc1NC(=O)N/C=C/c1ccccc1Cl ZINC000217795261 EJ For-Sale Unstable CPT1A 42 29 COc1ccc(Cl)cc1NC(=O)N/C=C/c1ccccc1Cl ZINC000217795261 EJ For-Sale Unstable RBP4 25 50 COc1ccc(Cl)cc1NC(=O)N/C=C/c1ccccc1Cl ZINC000217795261 EJ For-Sale Unstable CYSP_PLAFA 51 38 O=C(c1ccc(=O)[nH]n1)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217795296 GE In-Stock Unstable HRH3 23 43 CC(C)C[C@H](NC(=O)CC[C@@H]1NC(=O)c2ccccc2NC1=O)c1nc2ccccc2[nH]1 ZINC000217795302 IG In-Stock Unstable MMP7 21 49 C[C@@H]1C[C@@H](C)CN(CCCCOc2cccc(C=O)c2)C1 ZINC000217795307 CH In-Stock Unstable HRH3 21 42 CCc1ccc(OC)c(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217795342 GF For-Sale Unstable ADAMTS5 32 40 C[C@H]1C[C@@H](C)CN(CCCCOc2cccc(C=O)c2)C1 ZINC000217795345 CH In-Stock Unstable HRH3 21 42 O=C(c1ccc(=O)[nH]n1)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217795373 GE In-Stock Unstable HRH3 23 43 CC(C)C[C@H](NC(=O)CC[C@H]1NC(=O)c2ccccc2NC1=O)c1nc2ccccc2[nH]1 ZINC000217795377 IG In-Stock Unstable MMP7 21 49 C/C=C\c1ccc(OC[C@](C)(O)C(=O)OC)c(OC)c1 ZINC000217795387 CE For-Sale Unstable TUBB1 57 39 C[C@H]1C[C@H](C)CN(CCCCOc2cccc(C=O)c2)C1 ZINC000217795431 CH In-Stock Unstable HRH3 21 42 C/C=C\c1ccc(OC[C@@](C)(O)C(=O)OC)c(OC)c1 ZINC000217795457 CE For-Sale Unstable TUBB1 57 39 CC[C@@H](O)/C=C/CN(Cc1ccccc1)C(=O)OC(C)(C)C ZINC000217795458 DH For-Sale Unstable FPR1 40 34 COc1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217795469 DI For-Sale Unstable CA1 46 36 COc1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217795469 DI For-Sale Unstable MTNR1B 19 45 COc1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217795469 DI For-Sale Unstable CA12 23 43 COc1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217795469 DI For-Sale Unstable CA9 23 43 COc1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217795469 DI For-Sale Unstable Q8MMZ8_EIMTE 0 41 COc1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217795469 DI For-Sale Unstable TLR4 16 43 COc1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217795469 DI For-Sale Unstable AKR1C2 42 37 C[C@@H](NC(=O)Cn1nnc(-c2ccccc2)n1)c1cc(F)c(Cl)cc1Cl ZINC000217795478 GH On-Demand Unstable SCARB1 48 40 COc1ccc2cc([C@@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(O)cc6)oc5c43)c(=O)[nH]c2c1 ZINC000217795485 JI In-Stock Unstable AKR1B1 0 42 COc1ccc2cc([C@@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(O)cc6)oc5c43)c(=O)[nH]c2c1 ZINC000217795485 JI In-Stock Unstable CYP1B1 28 42 COc1ccc2cc([C@@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(O)cc6)oc5c43)c(=O)[nH]c2c1 ZINC000217795485 JI In-Stock Unstable CYP1A1 23 42 COc1ccc2cc([C@@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(O)cc6)oc5c43)c(=O)[nH]c2c1 ZINC000217795485 JI In-Stock Unstable CYP1A2 16 42 COc1ccc(NC(=O)N2[C@@H](C)C[C@@H]3CNC[C@H]32)cc1 ZINC000217795531 CD For-Sale Unstable ELOVL6 0 45 C[C@H](NC(=O)Cn1nnc(-c2ccccc2)n1)c1cc(F)c(Cl)cc1Cl ZINC000217795535 GH On-Demand Unstable SCARB1 48 40 COc1ccc2cc([C@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(O)cc6)oc5c43)c(=O)[nH]c2c1 ZINC000217795552 JI In-Stock Unstable AKR1B1 0 42 COc1ccc2cc([C@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(O)cc6)oc5c43)c(=O)[nH]c2c1 ZINC000217795552 JI In-Stock Unstable CYP1B1 28 42 COc1ccc2cc([C@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(O)cc6)oc5c43)c(=O)[nH]c2c1 ZINC000217795552 JI In-Stock Unstable CYP1A1 23 42 COc1ccc2cc([C@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(O)cc6)oc5c43)c(=O)[nH]c2c1 ZINC000217795552 JI In-Stock Unstable CYP1A2 16 42 O=Cc1cccc(OCCCCN2CCN(c3ccccc3)CC2)c1 ZINC000217795557 EG In-Stock Unstable HTR1A 98 64 O=Cc1cccc(OCCCCN2CCN(c3ccccc3)CC2)c1 ZINC000217795557 EG In-Stock Unstable DRD2 66 54 O=Cc1cccc(OCCCCN2CCN(c3ccccc3)CC2)c1 ZINC000217795557 EG In-Stock Unstable DRD1 31 44 O=Cc1cccc(OCCCCN2CCN(c3ccccc3)CC2)c1 ZINC000217795557 EG In-Stock Unstable DRD4 45 37 O=Cc1cccc(OCCCCN2CCN(c3ccccc3)CC2)c1 ZINC000217795557 EG In-Stock Unstable ACHE 24 41 O=Cc1cccc(OCCCCN2CCN(c3ccccc3)CC2)c1 ZINC000217795557 EG In-Stock Unstable HTR2A 70 64 O=Cc1cccc(OCCCCN2CCN(c3ccccc3)CC2)c1 ZINC000217795557 EG In-Stock Unstable HTR2C 30 42 O=Cc1cccc(OCCCCN2CCN(c3ccccc3)CC2)c1 ZINC000217795557 EG In-Stock Unstable SLC6A4 19 44 O=Cc1cccc(OCCCCN2CCN(c3ccccc3)CC2)c1 ZINC000217795557 EG In-Stock Unstable ADRA1A 28 52 O=Cc1cccc(OCCCCN2CCN(c3ccccc3)CC2)c1 ZINC000217795557 EG In-Stock Unstable HRH1 18 48 O=Cc1cccc(OCCCCN2CCN(c3ccccc3)CC2)c1 ZINC000217795557 EG In-Stock Unstable ADRA1B 15 41 O=Cc1cccc(OCCCCN2CCN(c3ccccc3)CC2)c1 ZINC000217795557 EG In-Stock Unstable DRD3 72 64 O=Cc1cccc(OCCCCN2CCN(c3ccccc3)CC2)c1 ZINC000217795557 EG In-Stock Unstable SLC6A3 18 41 O=Cc1cccc(OCCCCN2CCN(c3ccccc3)CC2)c1 ZINC000217795557 EG In-Stock Unstable KCNH2 0 53 O=Cc1cccc(OCCCCN2CCN(c3ccccc3)CC2)c1 ZINC000217795557 EG In-Stock Unstable DRD5 39 44 O=Cc1cccc(OCCCCN2CCN(c3ccccc3)CC2)c1 ZINC000217795557 EG In-Stock Unstable LTA4H 35 42 O=Cc1cccc(OCCCCN2CCN(c3ccccc3)CC2)c1 ZINC000217795557 EG In-Stock Unstable HTR7 105 43 O=Cc1cccc(OCCCCN2CCN(c3ccccc3)CC2)c1 ZINC000217795557 EG In-Stock Unstable SIGMAR1 42 46 O=Cc1cccc(OCCCCN2CCN(c3ccccc3)CC2)c1 ZINC000217795557 EG In-Stock Unstable ABCB1 25 42 O=Cc1cccc(OCCCCN2CCN(c3ccccc3)CC2)c1 ZINC000217795557 EG In-Stock Unstable EPHX2 20 48 O=Cc1cccc(OCCCCN2CCN(c3ccccc3)CC2)c1 ZINC000217795557 EG In-Stock Unstable CACNA1G 0 42 O=Cc1cccc(OCCCCN2CCN(c3ccccc3)CC2)c1 ZINC000217795557 EG In-Stock Unstable ALPHA-1A 0 40 CCN(CC)CCCCOc1ccccc1C=O ZINC000217795636 BF In-Stock Unstable ACHE 0 49 CCN(CC)CCCCOc1ccccc1C=O ZINC000217795636 BF In-Stock Unstable BCHE 0 49 CCN(CC)CCCCOc1ccccc1C=O ZINC000217795636 BF In-Stock Unstable AMY2 42 38 O=C(c1cncc(Br)c1)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217795645 II In-Stock Unstable HRH3 23 41 CS(=O)(=O)c1cc(F)cc(CCC(=O)O)c1 ZINC000217795675 BD For-Sale Unstable TBXA2R 54 43 CS(=O)(=O)c1cc(F)cc(CCC(=O)O)c1 ZINC000217795675 BD For-Sale Unstable FFAR1 51 40 COC1CCN(C2CCN(S(=O)(=O)c3ccccc3Br)CC2)CC1 ZINC000217795677 HF In-Stock Unstable CHRM2 23 41 COC1CCN(C2CCN(S(=O)(=O)c3ccccc3Br)CC2)CC1 ZINC000217795677 HF In-Stock Unstable CCR1 17 46 O=C(N/C=C/c1ccccc1Cl)NCCc1ccc(O)cc1 ZINC000217795680 DH For-Sale Unstable SLC6A5 27 40 O=C(N/C=C/c1ccccc1Cl)NCCc1ccc(O)cc1 ZINC000217795680 DH For-Sale Unstable NCE103 30 42 COc1ccc(OC)c(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)c1 ZINC000217795685 GE For-Sale Unstable ADAMTS5 31 41 O=C(c1cncc(Br)c1)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217795712 II In-Stock Unstable HRH3 23 41 O=Cc1ccccc1OCCCCN1CCCC1 ZINC000217795724 BF In-Stock Unstable HTR1A 61 38 O=Cc1ccccc1OCCCCN1CCCC1 ZINC000217795724 BF In-Stock Unstable DRD2 60 47 O=Cc1ccccc1OCCCCN1CCCC1 ZINC000217795724 BF In-Stock Unstable DRD1 33 56 O=Cc1ccccc1OCCCCN1CCCC1 ZINC000217795724 BF In-Stock Unstable ACHE 22 45 O=Cc1ccccc1OCCCCN1CCCC1 ZINC000217795724 BF In-Stock Unstable HRH2 16 40 O=Cc1ccccc1OCCCCN1CCCC1 ZINC000217795724 BF In-Stock Unstable ADRA1D 25 41 O=Cc1ccccc1OCCCCN1CCCC1 ZINC000217795724 BF In-Stock Unstable HTR2A 35 40 O=Cc1ccccc1OCCCCN1CCCC1 ZINC000217795724 BF In-Stock Unstable HTR2C 15 40 O=Cc1ccccc1OCCCCN1CCCC1 ZINC000217795724 BF In-Stock Unstable SLC6A1 82 40 O=Cc1ccccc1OCCCCN1CCCC1 ZINC000217795724 BF In-Stock Unstable DRD3 51 41 O=Cc1ccccc1OCCCCN1CCCC1 ZINC000217795724 BF In-Stock Unstable KCNH2 0 45 O=Cc1ccccc1OCCCCN1CCCC1 ZINC000217795724 BF In-Stock Unstable DRD5 39 56 O=Cc1ccccc1OCCCCN1CCCC1 ZINC000217795724 BF In-Stock Unstable LTA4H 47 45 O=Cc1ccccc1OCCCCN1CCCC1 ZINC000217795724 BF In-Stock Unstable HTR7 63 40 O=Cc1ccccc1OCCCCN1CCCC1 ZINC000217795724 BF In-Stock Unstable HRH3 68 48 O=Cc1ccccc1OCCCCN1CCCC1 ZINC000217795724 BF In-Stock Unstable SIGMAR1 46 40 O=Cc1ccccc1OCCCCN1CCCC1 ZINC000217795724 BF In-Stock Unstable NPY1R 44 37 O=Cc1ccccc1OCCCCN1CCCC1 ZINC000217795724 BF In-Stock Unstable BCHE 15 40 O=Cc1ccccc1OCCCCN1CCCC1 ZINC000217795724 BF In-Stock Unstable CHRNA7 20 40 O=Cc1ccccc1OCCCCN1CCCC1 ZINC000217795724 BF In-Stock Unstable HNMT 73 36 O=Cc1ccccc1OCCCCN1CCCC1 ZINC000217795724 BF In-Stock Unstable ABCB1 23 53 O=Cc1ccccc1OCCCCN1CCCC1 ZINC000217795724 BF In-Stock Unstable PSMB2 49 39 O=Cc1ccccc1OCCCCN1CCCC1 ZINC000217795724 BF In-Stock Unstable PSMB1 43 40 COc1ccc(OC)c(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)c1 ZINC000217795755 GE For-Sale Unstable ADAMTS5 31 41 CC(C)NC(=O)N/C=C/c1ccccc1Cl ZINC000217795768 BG For-Sale Unstable KCNQ2 22 45 CN(C)c1ccc(Cl)cc1NC(=O)CCn1c(=O)n(C)c2ccccc21 ZINC000217795778 FG On-Demand Unstable CXCR3 17 40 COc1ccc(NC(=O)N2[C@@H]3CNC[C@@H]3C[C@H]2C)cc1 ZINC000217795795 CD For-Sale Unstable ELOVL6 0 45 CCOCC(=O)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217795812 EF In-Stock Unstable HRH3 25 44 CC1CCN(CCCCOc2ccccc2C=O)CC1 ZINC000217795824 CG In-Stock Unstable HTR1A 63 39 CC1CCN(CCCCOc2ccccc2C=O)CC1 ZINC000217795824 CG In-Stock Unstable DRD2 60 42 CC1CCN(CCCCOc2ccccc2C=O)CC1 ZINC000217795824 CG In-Stock Unstable DRD1 21 41 CC1CCN(CCCCOc2ccccc2C=O)CC1 ZINC000217795824 CG In-Stock Unstable ACHE 15 44 CC1CCN(CCCCOc2ccccc2C=O)CC1 ZINC000217795824 CG In-Stock Unstable ADRA1D 26 40 CC1CCN(CCCCOc2ccccc2C=O)CC1 ZINC000217795824 CG In-Stock Unstable DRD3 42 37 CC1CCN(CCCCOc2ccccc2C=O)CC1 ZINC000217795824 CG In-Stock Unstable DRD5 25 41 CC1CCN(CCCCOc2ccccc2C=O)CC1 ZINC000217795824 CG In-Stock Unstable HTR7 68 39 CC1CCN(CCCCOc2ccccc2C=O)CC1 ZINC000217795824 CG In-Stock Unstable SIGMAR1 33 45 CC1CCN(CCCCOc2ccccc2C=O)CC1 ZINC000217795824 CG In-Stock Unstable NPY1R 42 35 CC1CCN(CCCCOc2ccccc2C=O)CC1 ZINC000217795824 CG In-Stock Unstable EBP 31 48 CC1CCN(CCCCOc2ccccc2C=O)CC1 ZINC000217795824 CG In-Stock Unstable ABCB1 15 40 CC1CCN(CCCCOc2ccccc2C=O)CC1 ZINC000217795824 CG In-Stock Unstable CYP2J2 45 32 CCN(CCNC(=O)[C@@H]1CCC[C@@H]1C(=O)O)C1CC1 ZINC000217795827 CD For-Sale Unstable ACE 0 43 CCOc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)cc1F ZINC000217795860 GF For-Sale Unstable ADAMTS5 32 41 CCCCNC(=O)N1[C@@H](C)C[C@@H]2CNC[C@H]21 ZINC000217795874 BD For-Sale Unstable ASAH1 51 31 CCOCC(=O)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217795878 EF In-Stock Unstable HRH3 25 44 Cc1ccc2ncc(N3CCN[C@H](C(C)C)C3)nc2c1 ZINC000217795902 CE For-Sale Unstable PRKCQ 15 43 Cc1cc(-c2cc(C(=O)N3CCN(c4cccc(O)c4)CC3)c3cnn(C(C)C)c3n2)c(C)o1 ZINC000217795911 JJ On-Demand Unstable CCKAR 36 40 C[C@H](F)CS(=O)(=O)c1ccc(C(=O)O)cc1 ZINC000217795916 BD For-Sale Unstable CA2 19 45 C[C@H](F)CS(=O)(=O)c1ccc(C(=O)O)cc1 ZINC000217795916 BD For-Sale Unstable SRD5A2 44 38 CCOc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)cc1F ZINC000217795923 GF For-Sale Unstable ADAMTS5 32 41 CCCCCC[C@@H](CN)N[C@@H](CC)CCO ZINC000217795925 BE For-Sale Unstable Q6UB75_PIG 0 46 CCN(CCNC(=O)[C@H]1CCC[C@@H]1C(=O)O)C1CC1 ZINC000217795928 CD For-Sale Unstable ACE 0 43 C[C@@H]1CCCCN1CCCCOc1ccccc1C=O ZINC000217795941 CH In-Stock Unstable HTR3A 18 40 C[C@@H]1CCCCN1CCCCOc1ccccc1C=O ZINC000217795941 CH In-Stock Unstable KCNH2 0 42 C[C@@H]1CCCCN1CCCCOc1ccccc1C=O ZINC000217795941 CH In-Stock Unstable HRH3 66 45 CCCCNC(=O)N1[C@@H]2CNC[C@H]2C[C@H]1C ZINC000217795969 BD For-Sale Unstable ASAH1 51 31 C[C@@H](F)CS(=O)(=O)c1ccc(C(=O)O)cc1 ZINC000217795971 BD For-Sale Unstable CA2 19 45 C[C@@H](F)CS(=O)(=O)c1ccc(C(=O)O)cc1 ZINC000217795971 BD For-Sale Unstable SRD5A2 44 38 Cc1ccc2ncc(N3CCN[C@@H](C(C)C)C3)nc2c1 ZINC000217795978 CE For-Sale Unstable PRKCQ 15 43 CCOC(=O)CCC(=O)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217795992 GG In-Stock Unstable HRH3 24 43 COC(=O)c1ccc(OCC(=O)C(C)(C)C)c(Br)n1 ZINC000217796000 EF For-Sale Unstable VDR 15 43 CCCCCC[C@H](CN)N[C@@H](CC)CCO ZINC000217796010 BE For-Sale Unstable Q6UB75_PIG 0 46 C[C@H]1CCCCN1CCCCOc1ccccc1C=O ZINC000217796020 CH In-Stock Unstable HTR3A 18 40 C[C@H]1CCCCN1CCCCOc1ccccc1C=O ZINC000217796020 CH In-Stock Unstable KCNH2 0 42 C[C@H]1CCCCN1CCCCOc1ccccc1C=O ZINC000217796020 CH In-Stock Unstable HRH3 66 45 CCCCNC(=O)N1[C@@H](C)C[C@H]2CNC[C@H]21 ZINC000217796057 BD For-Sale Unstable ASAH1 51 31 CCOC(=O)CCC(=O)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217796065 GG In-Stock Unstable HRH3 24 43 C[C@H](F)CS(=O)(=O)c1cccc(C(=O)O)c1 ZINC000217796091 BD For-Sale Unstable AKR1C3 64 43 Cc1ccccc1-c1cc(C(=O)N2CCN(c3cccc(O)c3)CC2)c2cnn(C(C)C)c2n1 ZINC000217796096 JJ On-Demand Unstable CCKAR 37 42 CCCCCC[C@@H](CN)N[C@H](CC)CCO ZINC000217796119 BE For-Sale Unstable Q6UB75_PIG 0 46 CC[C@H](CO)[C@@H](CO)NC(=O)OC(C)(C)C ZINC000217796135 BC For-Sale Unstable PAPA1_CARPA 43 39 CC[C@H](CO)[C@@H](CO)NC(=O)OC(C)(C)C ZINC000217796135 BC For-Sale Unstable CTSK 25 49 CC[C@H](CO)[C@@H](CO)NC(=O)OC(C)(C)C ZINC000217796135 BC For-Sale Unstable PGA5 42 37 CC[C@H](CO)[C@@H](CO)NC(=O)OC(C)(C)C ZINC000217796135 BC For-Sale Unstable POL 0 45 CCCCNC(=O)N1[C@@H]2CNC[C@@H]2C[C@H]1C ZINC000217796142 BD For-Sale Unstable ASAH1 51 31 C[C@@H](F)CS(=O)(=O)c1cccc(C(=O)O)c1 ZINC000217796160 BD For-Sale Unstable AKR1C3 64 43 COc1ccccc1C(=O)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217796172 GH In-Stock Unstable HRH3 25 52 CCn1ncc2c(C(=O)N3CCN(c4cccc(O)c4)CC3)cc(-c3ccccc3)nc21 ZINC000217796180 IH On-Demand Unstable P2RY12 41 39 CCn1ncc2c(C(=O)N3CCN(c4cccc(O)c4)CC3)cc(-c3ccccc3)nc21 ZINC000217796180 IH On-Demand Unstable CCKAR 40 43 COC1CCN(C2CCN(S(=O)(=O)Cc3cc(F)ccc3F)CC2)CC1 ZINC000217796188 GE In-Stock Unstable CHRM2 29 43 CCCCCC[C@H](CN)N[C@H](CC)CCO ZINC000217796190 BE For-Sale Unstable Q6UB75_PIG 0 46 CC[C@@H](CO)[C@H](CO)NC(=O)OC(C)(C)C ZINC000217796213 BC For-Sale Unstable PAPA1_CARPA 43 39 CC[C@@H](CO)[C@H](CO)NC(=O)OC(C)(C)C ZINC000217796213 BC For-Sale Unstable CTSK 25 49 CC[C@@H](CO)[C@H](CO)NC(=O)OC(C)(C)C ZINC000217796213 BC For-Sale Unstable PGA5 42 37 CC[C@@H](CO)[C@H](CO)NC(=O)OC(C)(C)C ZINC000217796213 BC For-Sale Unstable POL 0 45 COc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)cc1Cl ZINC000217796217 GF For-Sale Unstable ADAMTS5 31 41 COc1ccccc1C(=O)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217796240 GH In-Stock Unstable HRH3 25 52 NCCCOc1ccccc1OCc1ccccc1 ZINC000217796277 CF In-Stock Unstable PTGER2 24 44 NCCCOc1ccccc1OCc1ccccc1 ZINC000217796277 CF In-Stock Unstable PPIA 44 36 NCCCOc1ccccc1OCc1ccccc1 ZINC000217796277 CF In-Stock Unstable PTGER1 37 41 NCCCOc1ccccc1OCc1ccccc1 ZINC000217796277 CF In-Stock Unstable PTGER4 18 41 NCCCOc1ccccc1OCc1ccccc1 ZINC000217796277 CF In-Stock Unstable TAAR1 23 49 CN1CCC[C@@H]1CNCc1nccn1C(F)F ZINC000217796284 BD For-Sale Unstable CHRNA10 44 36 O=C(CCc1ncc(-c2ccccc2Cl)o1)N1CCN(c2cccc(O)c2)CC1 ZINC000217796285 HH On-Demand Unstable SSTR1 44 43 CC[C@H](CO)[C@H](CO)NC(=O)OC(C)(C)C ZINC000217796300 BC For-Sale Unstable PAPA1_CARPA 43 39 CC[C@H](CO)[C@H](CO)NC(=O)OC(C)(C)C ZINC000217796300 BC For-Sale Unstable CTSK 25 49 CC[C@H](CO)[C@H](CO)NC(=O)OC(C)(C)C ZINC000217796300 BC For-Sale Unstable PGA5 42 37 CC[C@H](CO)[C@H](CO)NC(=O)OC(C)(C)C ZINC000217796300 BC For-Sale Unstable POL 0 45 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)cc1Cl ZINC000217796309 GF For-Sale Unstable ADAMTS5 31 41 CCOC(=O)C1CCN(C(=O)N/C=C/c2ccccc2Cl)CC1 ZINC000217796321 EG For-Sale Unstable FDFT1 23 41 O=Cc1ccccc1OCCCCN1CCCCCC1 ZINC000217796332 CH In-Stock Unstable HTR1A 56 38 O=Cc1ccccc1OCCCCN1CCCCCC1 ZINC000217796332 CH In-Stock Unstable DRD2 56 47 O=Cc1ccccc1OCCCCN1CCCCCC1 ZINC000217796332 CH In-Stock Unstable DRD1 29 55 O=Cc1ccccc1OCCCCN1CCCCCC1 ZINC000217796332 CH In-Stock Unstable ACHE 22 46 O=Cc1ccccc1OCCCCN1CCCCCC1 ZINC000217796332 CH In-Stock Unstable ADRA1D 24 40 O=Cc1ccccc1OCCCCN1CCCCCC1 ZINC000217796332 CH In-Stock Unstable HTR2A 31 42 O=Cc1ccccc1OCCCCN1CCCCCC1 ZINC000217796332 CH In-Stock Unstable SLC6A1 72 39 O=Cc1ccccc1OCCCCN1CCCCCC1 ZINC000217796332 CH In-Stock Unstable DRD3 49 40 O=Cc1ccccc1OCCCCN1CCCCCC1 ZINC000217796332 CH In-Stock Unstable KCNH2 0 48 O=Cc1ccccc1OCCCCN1CCCCCC1 ZINC000217796332 CH In-Stock Unstable HTR4 15 47 O=Cc1ccccc1OCCCCN1CCCCCC1 ZINC000217796332 CH In-Stock Unstable DRD5 39 55 O=Cc1ccccc1OCCCCN1CCCCCC1 ZINC000217796332 CH In-Stock Unstable LTA4H 46 44 O=Cc1ccccc1OCCCCN1CCCCCC1 ZINC000217796332 CH In-Stock Unstable HTR7 57 39 O=Cc1ccccc1OCCCCN1CCCCCC1 ZINC000217796332 CH In-Stock Unstable HRH3 73 50 O=Cc1ccccc1OCCCCN1CCCCCC1 ZINC000217796332 CH In-Stock Unstable SIGMAR1 46 41 O=Cc1ccccc1OCCCCN1CCCCCC1 ZINC000217796332 CH In-Stock Unstable NPY1R 46 38 O=Cc1ccccc1OCCCCN1CCCCCC1 ZINC000217796332 CH In-Stock Unstable CHRNA7 23 42 O=Cc1ccccc1OCCCCN1CCCCCC1 ZINC000217796332 CH In-Stock Unstable HNMT 77 38 O=Cc1ccccc1OCCCCN1CCCCCC1 ZINC000217796332 CH In-Stock Unstable ABCB1 30 55 O=Cc1ccccc1OCCCCN1CCCCCC1 ZINC000217796332 CH In-Stock Unstable PSMB2 52 41 O=Cc1ccccc1OCCCCN1CCCCCC1 ZINC000217796332 CH In-Stock Unstable PSMB5 18 41 O=Cc1ccccc1OCCCCN1CCCCCC1 ZINC000217796332 CH In-Stock Unstable PSMB1 45 43 CN1CCC[C@H]1CNCc1nccn1C(F)F ZINC000217796351 BD For-Sale Unstable CHRNA10 44 36 NC(=O)[C@H]1CCCN1C(=O)CC1CC1 ZINC000217796374 AC On-Demand Unstable ACE 15 45 NC(=O)[C@H]1CCCN1C(=O)CC1CC1 ZINC000217796374 AC On-Demand Unstable TRHR 59 38 NC(=O)[C@H]1CCCN1C(=O)CC1CC1 ZINC000217796374 AC On-Demand Unstable DPP4 16 48 NC(=O)[C@H]1CCCN1C(=O)CC1CC1 ZINC000217796374 AC On-Demand Unstable PREP 48 43 NC(=O)[C@H]1CCCN1C(=O)CC1CC1 ZINC000217796374 AC On-Demand Unstable TPP2 40 53 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable ACE 29 61 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable TYR 16 44 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable GNRHR 0 43 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable OPRM1 17 44 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable OPRD1 0 45 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable MME 46 54 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable EDNRB 62 47 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable EDNRA 52 47 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable TACR1 39 47 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable MC4R 47 41 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable BMP1 29 42 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable TACR2 26 44 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable CCKAR 135 49 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable BRS3 31 50 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable NMBR 31 44 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable MC3R 66 37 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable MC5R 67 35 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable MMP2 30 47 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable MMP8 39 42 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable MMP14 27 42 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable GRPR 76 38 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable ECE1 79 54 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable LNPEP 31 43 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable SSTR3 28 41 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable MMP11 104 38 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable CCKBR 106 43 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable GHSR 78 42 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable MMP9 29 47 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable MC1R 97 41 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable ADAM9 41 42 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable MMP1 21 44 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable FPR1 19 47 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable NPR 35 52 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable SSSIM 32 48 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable SLC15A2 0 61 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable KISS1R 75 36 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable ERAP2 47 44 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable PSMB8 25 40 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable ERAP1 0 44 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable LASB 0 45 Cc1cc(=O)n(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c2ccccc12 ZINC000217796378 HF In-Stock Unstable NRDE 0 48 O=C(c1ccccc1Br)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217796384 IJ In-Stock Unstable HRH3 20 44 O=C(CCc1ncc(-c2ccc(Cl)cc2)o1)N1CCN(c2cccc(O)c2)CC1 ZINC000217796387 HH On-Demand Unstable VDR 0 41 O=C(CCc1ncc(-c2ccc(Cl)cc2)o1)N1CCN(c2cccc(O)c2)CC1 ZINC000217796387 HH On-Demand Unstable MAPK1 16 41 O=C(CCc1ncc(-c2ccc(Cl)cc2)o1)N1CCN(c2cccc(O)c2)CC1 ZINC000217796387 HH On-Demand Unstable AKR1C3 0 43 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1ccc(C(F)(F)F)cc1 ZINC000217796440 GG For-Sale Unstable ADAMTS5 29 56 O=C(N/C=C/c1ccccc1Cl)NC1CCCCC1 ZINC000217796449 CH For-Sale Unstable EPHX2 36 48 NC(=O)[C@@H]1CCCN1C(=O)CC1CC1 ZINC000217796459 AC On-Demand Unstable ACE 15 45 NC(=O)[C@@H]1CCCN1C(=O)CC1CC1 ZINC000217796459 AC On-Demand Unstable TRHR 59 38 NC(=O)[C@@H]1CCCN1C(=O)CC1CC1 ZINC000217796459 AC On-Demand Unstable DPP4 16 48 NC(=O)[C@@H]1CCCN1C(=O)CC1CC1 ZINC000217796459 AC On-Demand Unstable PREP 48 43 NC(=O)[C@@H]1CCCN1C(=O)CC1CC1 ZINC000217796459 AC On-Demand Unstable TPP2 40 53 O=C(c1ccccc1Br)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217796472 IJ In-Stock Unstable HRH3 20 44 O=C(CCc1ncc(-c2ccc(F)cc2F)o1)N1CCN(c2cccc(O)c2)CC1 ZINC000217796477 HH On-Demand Unstable SSTR1 35 41 COc1ccc(CCNC(=O)[C@@H](NC(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)C(C)C)cc1OC ZINC000217796505 JE In-Stock Unstable CHRNA4 26 44 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1ccc(C(F)(F)F)cc1 ZINC000217796518 GG For-Sale Unstable OXTR 20 40 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1ccc(C(F)(F)F)cc1 ZINC000217796518 GG For-Sale Unstable ADAMTS5 37 57 O=C(c1ccccc1C(F)(F)F)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217796575 IJ In-Stock Unstable HRH3 19 43 O=C(c1ccccc1C(F)(F)F)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217796575 IJ In-Stock Unstable RBP4 42 35 O=C(c1ccccc1C(F)(F)F)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217796575 IJ In-Stock Unstable SCD1 22 41 O=C(c1ccccc1C(F)(F)F)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217796575 IJ In-Stock Unstable SCD 23 41 O=C(CCc1ncc(-c2ccc(Cl)cc2Cl)o1)N1CCN(c2cccc(O)c2)CC1 ZINC000217796579 IJ On-Demand Unstable SSTR1 35 42 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1cccc(C(F)(F)F)c1 ZINC000217796611 GG For-Sale Unstable CACNA1B 46 34 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1cccc(C(F)(F)F)c1 ZINC000217796611 GG For-Sale Unstable ADAMTS5 34 51 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1cccc(C(F)(F)F)c1 ZINC000217796611 GG For-Sale Unstable SFRP1 53 31 COc1ccc(O)c(CS(=O)(=O)Cl)c1F ZINC000217796618 CD For-Sale Unstable TUBB1 42 36 O=C(c1ccccc1C(F)(F)F)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217796640 IJ In-Stock Unstable HRH3 19 43 O=C(c1ccccc1C(F)(F)F)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217796640 IJ In-Stock Unstable RBP4 42 35 O=C(c1ccccc1C(F)(F)F)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217796640 IJ In-Stock Unstable SCD1 22 41 O=C(c1ccccc1C(F)(F)F)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217796640 IJ In-Stock Unstable SCD 23 41 O=C(O)C1CCN(C(=O)N/C=C/c2ccccc2Cl)CC1 ZINC000217796673 DF For-Sale Unstable SLC6A1 55 38 O=C(O)C1CCN(C(=O)N/C=C/c2ccccc2Cl)CC1 ZINC000217796673 DF For-Sale Unstable ITGAL 21 40 O=C(O)C1CCN(C(=O)N/C=C/c2ccccc2Cl)CC1 ZINC000217796673 DF For-Sale Unstable EPHX2 15 47 COc1ccc(-c2noc(CCC(=O)N3CCN(c4cccc(O)c4)CC3)n2)cc1 ZINC000217796677 HF On-Demand Unstable CCKAR 37 40 COc1ccc(-c2noc(CCC(=O)N3CCN(c4cccc(O)c4)CC3)n2)cc1 ZINC000217796677 HF On-Demand Unstable PDK1 37 42 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1cccc(C(F)(F)F)c1 ZINC000217796679 GG For-Sale Unstable CACNA1B 46 34 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1cccc(C(F)(F)F)c1 ZINC000217796679 GG For-Sale Unstable ADAMTS5 34 51 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1cccc(C(F)(F)F)c1 ZINC000217796679 GG For-Sale Unstable SFRP1 53 31 O=Cc1ccccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217796693 EG In-Stock Unstable HTR1A 148 58 O=Cc1ccccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217796693 EG In-Stock Unstable DRD2 104 55 O=Cc1ccccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217796693 EG In-Stock Unstable DRD1 52 44 O=Cc1ccccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217796693 EG In-Stock Unstable DRD4 66 42 O=Cc1ccccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217796693 EG In-Stock Unstable ADRA1D 53 45 O=Cc1ccccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217796693 EG In-Stock Unstable HTR1B 20 41 O=Cc1ccccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217796693 EG In-Stock Unstable HTR2A 93 46 O=Cc1ccccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217796693 EG In-Stock Unstable HTR2C 35 41 O=Cc1ccccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217796693 EG In-Stock Unstable SLC6A4 29 42 O=Cc1ccccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217796693 EG In-Stock Unstable ADRA1A 50 45 O=Cc1ccccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217796693 EG In-Stock Unstable HRH1 22 43 O=Cc1ccccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217796693 EG In-Stock Unstable DRD3 92 58 O=Cc1ccccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217796693 EG In-Stock Unstable DRD5 38 56 O=Cc1ccccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217796693 EG In-Stock Unstable HTR7 134 49 O=Cc1ccccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217796693 EG In-Stock Unstable HRH3 18 45 O=Cc1ccccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217796693 EG In-Stock Unstable SIGMAR1 41 47 O=Cc1ccccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217796693 EG In-Stock Unstable HTR6 0 43 O=Cc1ccccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217796693 EG In-Stock Unstable ABCB1 30 53 O=Cc1ccccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217796693 EG In-Stock Unstable AP2S1 0 41 COc1ccc(O)c(F)c1CS(=O)(=O)Cl ZINC000217796694 CD For-Sale Unstable TUBB1 43 37 O=C(COc1ccc(Cl)cc1)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217796743 II In-Stock Unstable HRH3 30 48 O=C(COc1ccc(Cl)cc1)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217796743 II In-Stock Unstable COLA 121 45 O=C(COc1ccc(Cl)cc1)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217796743 II In-Stock Unstable CPT1A 109 45 O=C(COc1ccc(Cl)cc1)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217796743 II In-Stock Unstable GPR183 0 43 COc1cc(C(=O)N[C@@H](CC(=O)O)c2ccccc2C)cc(Cl)n1 ZINC000217796751 EF Annotated Unstable MME 15 49 COc1cc(C(=O)N[C@@H](CC(=O)O)c2ccccc2C)cc(Cl)n1 ZINC000217796751 EF Annotated Unstable ALS 71 36 COc1cc(C(=O)N[C@@H](CC(=O)O)c2ccccc2C)cc(Cl)n1 ZINC000217796751 EF Annotated Unstable UTS2 65 34 COc1cc(C(=O)N[C@@H](CC(=O)O)c2ccccc2C)cc(Cl)n1 ZINC000217796751 EF Annotated Unstable CTSA 114 51 O=C(Nc1nc(CC(=O)N2CCN(c3cccc(O)c3)CC2)cs1)c1ccccc1 ZINC000217796754 HF On-Demand Unstable PDE5A 16 53 O=C(Nc1nc(CC(=O)N2CCN(c3cccc(O)c3)CC2)cs1)c1ccccc1 ZINC000217796754 HF On-Demand Unstable VDR 16 40 O=C(Nc1nc(CC(=O)N2CCN(c3cccc(O)c3)CC2)cs1)c1ccccc1 ZINC000217796754 HF On-Demand Unstable COLA 19 42 O=C(Nc1nc(CC(=O)N2CCN(c3cccc(O)c3)CC2)cs1)c1ccccc1 ZINC000217796754 HF On-Demand Unstable CPT1A 29 42 O=C(Nc1nc(CC(=O)N2CCN(c3cccc(O)c3)CC2)cs1)c1ccccc1 ZINC000217796754 HF On-Demand Unstable PRNP 46 34 O=C(Nc1nc(CC(=O)N2CCN(c3cccc(O)c3)CC2)cs1)c1ccccc1 ZINC000217796754 HF On-Demand Unstable MAPK1 30 40 O=C(Nc1nc(CC(=O)N2CCN(c3cccc(O)c3)CC2)cs1)c1ccccc1 ZINC000217796754 HF On-Demand Unstable CPT1B 38 42 O=C(N/C=C/c1ccccc1Cl)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217796757 IK For-Sale Unstable NMUR2 0 46 O=C(N/C=C/c1ccccc1Cl)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217796757 IK For-Sale Unstable NMUR1 0 46 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1cc(Cl)ccc1Cl ZINC000217796815 GG For-Sale Unstable ADAMTS5 29 41 CCN(CC)CCCCOc1ccc(C=O)cc1OC ZINC000217796817 CG In-Stock Unstable THRA 22 43 CCN(CC)CCCCOc1ccc(C=O)cc1OC ZINC000217796817 CG In-Stock Unstable ACHE 0 50 CCN(CC)CCCCOc1ccc(C=O)cc1OC ZINC000217796817 CG In-Stock Unstable BCHE 0 44 O=C(COc1ccc(Cl)cc1)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217796837 II In-Stock Unstable HRH3 30 48 O=C(COc1ccc(Cl)cc1)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217796837 II In-Stock Unstable COLA 121 45 O=C(COc1ccc(Cl)cc1)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217796837 II In-Stock Unstable CPT1A 109 45 O=C(COc1ccc(Cl)cc1)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217796837 II In-Stock Unstable GPR183 0 43 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1cc(Cl)ccc1Cl ZINC000217796884 GG For-Sale Unstable ADAMTS5 29 41 COc1cc(C=O)ccc1OCCCCN1CCCC1 ZINC000217796909 CF In-Stock Unstable DRD2 37 41 COc1cc(C=O)ccc1OCCCCN1CCCC1 ZINC000217796909 CF In-Stock Unstable DRD1 19 40 COc1cc(C=O)ccc1OCCCCN1CCCC1 ZINC000217796909 CF In-Stock Unstable ACHE 28 53 COc1cc(C=O)ccc1OCCCCN1CCCC1 ZINC000217796909 CF In-Stock Unstable HTR2A 22 42 COc1cc(C=O)ccc1OCCCCN1CCCC1 ZINC000217796909 CF In-Stock Unstable HTR4 38 41 COc1cc(C=O)ccc1OCCCCN1CCCC1 ZINC000217796909 CF In-Stock Unstable DRD5 17 40 COc1cc(C=O)ccc1OCCCCN1CCCC1 ZINC000217796909 CF In-Stock Unstable HRH3 55 42 COc1cc(C=O)ccc1OCCCCN1CCCC1 ZINC000217796909 CF In-Stock Unstable SIGMAR1 33 45 COc1cc(C=O)ccc1OCCCCN1CCCC1 ZINC000217796909 CF In-Stock Unstable ABCB1 16 40 COc1cc(C=O)ccc1OCCCCN1CCCC1 ZINC000217796909 CF In-Stock Unstable MET 46 41 COc1cc(C=O)ccc1OCCCCN1CCCC1 ZINC000217796909 CF In-Stock Unstable MCHR1 0 43 COc1cc(C=O)ccc1OCCCCN1CCCC1 ZINC000217796909 CF In-Stock Unstable PSMB2 43 34 COc1cc(C=O)ccc1OCCCCN1CCCC1 ZINC000217796909 CF In-Stock Unstable EHMT1 0 44 COc1cc(C=O)ccc1OCCCCN1CCCC1 ZINC000217796909 CF In-Stock Unstable EHMT2 83 44 COc1cc(C=O)ccc1OCCCCN1CCCC1 ZINC000217796909 CF In-Stock Unstable SLC29A2 0 44 COc1cc(C=O)ccc1OCCCCN1CCCC1 ZINC000217796909 CF In-Stock Unstable ASF1A 0 49 CCN([C@H](C)COC)[C@@H]1CCCc2cc(O)ccc21 ZINC000217796922 CG For-Sale Unstable HSD17B1 68 37 COc1ccc(CC(=O)N2CCC[C@H](Cc3nc(-c4ccccc4F)no3)C2)cc1OC ZINC000217796952 IH In-Stock Unstable HRH3 26 47 COc1ccc(CC(=O)N2CCC[C@H](Cc3nc(-c4ccccc4F)no3)C2)cc1OC ZINC000217796952 IH In-Stock Unstable ACKR3 47 35 CC(C)COc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)cc1 ZINC000217796993 GG For-Sale Unstable ADAMTS5 33 42 COc1ccc(CC(=O)N2CCC[C@@H](Cc3nc(-c4ccccc4F)no3)C2)cc1OC ZINC000217797017 IH In-Stock Unstable HRH3 26 47 COc1ccc(CC(=O)N2CCC[C@@H](Cc3nc(-c4ccccc4F)no3)C2)cc1OC ZINC000217797017 IH In-Stock Unstable ACKR3 47 35 COCCN(CC(=O)O)C(=O)/C=C\c1ccc(O)cc1 ZINC000217797027 CC On-Demand Unstable F3 24 41 COCCN(CC(=O)O)C(=O)/C=C\c1ccc(O)cc1 ZINC000217797027 CC On-Demand Unstable AKR1B10 26 42 COc1cc(C=O)ccc1OCCCCN1CCC(C)CC1 ZINC000217797034 DG In-Stock Unstable DRD2 23 45 COc1cc(C=O)ccc1OCCCCN1CCC(C)CC1 ZINC000217797034 DG In-Stock Unstable ACHE 20 42 COc1cc(C=O)ccc1OCCCCN1CCC(C)CC1 ZINC000217797034 DG In-Stock Unstable HTR4 46 44 COc1cc(C=O)ccc1OCCCCN1CCC(C)CC1 ZINC000217797034 DG In-Stock Unstable SIGMAR1 22 42 COc1cc(C=O)ccc1OCCCCN1CCC(C)CC1 ZINC000217797034 DG In-Stock Unstable EBP 38 43 COc1cc(C=O)ccc1OCCCCN1CCC(C)CC1 ZINC000217797034 DG In-Stock Unstable MET 33 41 COc1cc(C=O)ccc1OCCCCN1CCC(C)CC1 ZINC000217797034 DG In-Stock Unstable EHMT2 68 35 COc1cc(C=O)ccc1OCCCCN1CCC(C)CC1 ZINC000217797034 DG In-Stock Unstable SLC29A2 0 41 COc1cc(C=O)ccc1OCCCCN1CCC(C)CC1 ZINC000217797034 DG In-Stock Unstable ASF1A 0 40 CCCCNC(=O)N/C=C/c1ccccc1Cl ZINC000217797051 CG For-Sale Unstable ACAT 0 47 CC(C)COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)cc1 ZINC000217797061 GG For-Sale Unstable ADAMTS5 33 42 COc1ccc(CN2C(=O)N[C@@H](CC(=O)NCCc3ccc(O)cc3)C2=O)cc1OC ZINC000217797135 ID In-Stock Unstable CAN2 0 48 COc1cc(C=O)ccc1OCCCCN1CCC[C@@H](C)C1 ZINC000217797155 DG In-Stock Unstable ACHE 15 41 COc1cc(C=O)ccc1OCCCCN1CCC[C@@H](C)C1 ZINC000217797155 DG In-Stock Unstable SLC6A1 48 35 COc1cc(C=O)ccc1OCCCCN1CCC[C@@H](C)C1 ZINC000217797155 DG In-Stock Unstable HTR4 20 44 COc1cc(C=O)ccc1OCCCCN1CCC[C@@H](C)C1 ZINC000217797155 DG In-Stock Unstable EBP 21 44 COc1cc(C=O)ccc1OCCCCN1CCC[C@@H](C)C1 ZINC000217797155 DG In-Stock Unstable EHMT2 72 37 COc1cc(C=O)ccc1OCCCCN1CCC[C@@H](C)C1 ZINC000217797155 DG In-Stock Unstable ACKR3 65 35 COc1cc(C=O)ccc1OCCCCN1CCC[C@@H](C)C1 ZINC000217797155 DG In-Stock Unstable ASF1A 0 40 O=C(Cc1cccs1)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217797159 GH In-Stock Unstable HRH3 19 40 O=C(Cc1cccs1)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217797159 GH In-Stock Unstable ETHR 53 49 CCCOc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)cc1C ZINC000217797185 GG For-Sale Unstable ADAMTS5 33 47 O=C(Cc1cccs1)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217797221 GH In-Stock Unstable HRH3 19 40 O=C(Cc1cccs1)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217797221 GH In-Stock Unstable ETHR 53 49 COc1cc(C=O)ccc1OCCCCN1CCC[C@H](C)C1 ZINC000217797222 DG In-Stock Unstable ACHE 15 41 COc1cc(C=O)ccc1OCCCCN1CCC[C@H](C)C1 ZINC000217797222 DG In-Stock Unstable SLC6A1 48 35 COc1cc(C=O)ccc1OCCCCN1CCC[C@H](C)C1 ZINC000217797222 DG In-Stock Unstable HTR4 20 44 COc1cc(C=O)ccc1OCCCCN1CCC[C@H](C)C1 ZINC000217797222 DG In-Stock Unstable EBP 21 44 COc1cc(C=O)ccc1OCCCCN1CCC[C@H](C)C1 ZINC000217797222 DG In-Stock Unstable EHMT2 72 37 COc1cc(C=O)ccc1OCCCCN1CCC[C@H](C)C1 ZINC000217797222 DG In-Stock Unstable ACKR3 65 35 COc1cc(C=O)ccc1OCCCCN1CCC[C@H](C)C1 ZINC000217797222 DG In-Stock Unstable ASF1A 0 40 C[C@H]1[C@H](C)CCC[C@H]1NC(=O)Nc1cccc([C@@H](C)O)c1 ZINC000217797247 CH For-Sale Unstable EPHX2 17 40 COc1ccc(-c2coc3ccc(OCC(=O)c4ccc(NC(C)=O)cc4)cc23)cc1OC ZINC000217797265 IK In-Stock Unstable ALDH2 82 36 COc1ccc(-c2coc3ccc(OCC(=O)c4ccc(NC(C)=O)cc4)cc23)cc1OC ZINC000217797265 IK In-Stock Unstable TSHR 44 34 COc1ccc(-c2coc3ccc(OCC(=O)c4ccc(NC(C)=O)cc4)cc23)cc1OC ZINC000217797265 IK In-Stock Unstable KIT 19 41 COc1ccc(-c2coc3ccc(OCC(=O)c4ccc(NC(C)=O)cc4)cc23)cc1OC ZINC000217797265 IK In-Stock Unstable PDGFRA 47 35 CCCOc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)cc1C ZINC000217797273 GG For-Sale Unstable ADAMTS5 33 47 C[C@H](O)c1cccc(NC(=O)N[C@@H]2CCC[C@@H](C)[C@@H]2C)c1 ZINC000217797318 CH For-Sale Unstable EPHX2 17 40 COc1cc(C=O)ccc1OCCCCN1CCCC[C@@H]1C ZINC000217797330 DH In-Stock Unstable HRH3 50 42 COc1cc(C=O)ccc1OCCCCN1CCCC[C@@H]1C ZINC000217797330 DH In-Stock Unstable ACKR3 55 47 O=C(c1ccco1)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217797336 FH In-Stock Unstable HRH3 26 48 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](CC(C)C)C(=O)Nc3nc[nH]n3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217797378 KG In-Stock Unstable TUBA1A 18 63 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](CC(C)C)C(=O)Nc3nc[nH]n3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217797378 KG In-Stock Unstable TPPP 0 60 C[C@@H]1[C@@H](NC(=O)Nc2cccc([C@@H](C)O)c2)CCC[C@H]1C ZINC000217797403 CH For-Sale Unstable EPHX2 17 40 COc1cc(C=O)ccc1OCCCCN1CCCC[C@H]1C ZINC000217797421 DH In-Stock Unstable HRH3 50 42 COc1cc(C=O)ccc1OCCCCN1CCCC[C@H]1C ZINC000217797421 DH In-Stock Unstable ACKR3 55 47 O=C(c1ccco1)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217797427 FH In-Stock Unstable HRH3 26 48 O=C(N/C=C/c1ccccc1Cl)N1CCCc2ccccc21 ZINC000217797428 DI For-Sale Unstable AVPR2 52 49 C[C@H](O)c1cccc(NC(=O)N[C@H]2CCC[C@@H](C)[C@@H]2C)c1 ZINC000217797483 CH For-Sale Unstable EPHX2 17 40 O=C(N/C=C/c1ccccc1Cl)NCCc1ccccc1 ZINC000217797533 DH For-Sale Unstable CA5B 15 40 O=C(N/C=C/c1ccccc1Cl)NCCc1ccccc1 ZINC000217797533 DH For-Sale Unstable CA5A 18 40 O=C(N/C=C/c1ccccc1Cl)NCCc1ccccc1 ZINC000217797533 DH For-Sale Unstable NCE103 24 45 CCOC(=O)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217797534 EG In-Stock Unstable HRH3 28 46 C[C@H]1[C@H](C)CCC[C@H]1NC(=O)Nc1ccc([C@@H](C)O)cc1 ZINC000217797548 CH For-Sale Unstable EPHX2 28 50 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1ccc(OC(F)(F)F)cc1 ZINC000217797584 HF For-Sale Unstable ADAMTS5 26 46 CCOC(=O)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217797605 EG In-Stock Unstable HRH3 28 46 O=C(CCn1ccc(=O)[nH]c1=O)NCCc1nccc(-c2ccccc2)n1 ZINC000217797623 FC In-Stock Unstable DUT 70 38 O=C(CCn1ccc(=O)[nH]c1=O)NCCc1nccc(-c2ccccc2)n1 ZINC000217797623 FC In-Stock Unstable Q8II92_PLAF7 55 41 O=C(N/C=C/c1ccccc1Cl)NC1CCCC1 ZINC000217797629 CH For-Sale Unstable EPHX2 31 45 C[C@H](O)c1ccc(NC(=O)N[C@@H]2CCC[C@@H](C)[C@@H]2C)cc1 ZINC000217797641 CH For-Sale Unstable EPHX2 28 50 C[C@@H](NCc1cccn1C)[C@@H]1CCCN(C(=O)OC(C)(C)C)C1 ZINC000217797670 DG On-Demand Unstable GPR119 26 43 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1ccc(OC(F)(F)F)cc1 ZINC000217797692 HF For-Sale Unstable ADAMTS5 26 46 O=C(N/C=C/c1ccccc1Cl)NCc1ccccc1Cl ZINC000217797707 DI For-Sale Unstable P2RX7 28 43 O=C(N/C=C/c1ccccc1Cl)NCc1ccccc1Cl ZINC000217797707 DI For-Sale Unstable SLC6A12 0 40 C[C@H](NCc1cccn1C)[C@@H]1CCCN(C(=O)OC(C)(C)C)C1 ZINC000217797712 DG On-Demand Unstable GPR119 26 43 C[C@@H]1[C@@H](NC(=O)Nc2ccc([C@@H](C)O)cc2)CCC[C@H]1C ZINC000217797716 CH For-Sale Unstable EPHX2 28 50 COC(=O)c1ccccc1C(=O)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217797736 HH In-Stock Unstable HRH3 28 48 C=C(C)COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)ccc1OC ZINC000217797738 KK In-Stock Unstable AKR1B1 0 45 C=C(C)COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)ccc1OC ZINC000217797738 KK In-Stock Unstable CYP1B1 49 36 C=C(C)COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)ccc1OC ZINC000217797738 KK In-Stock Unstable CYP1A1 37 43 C[C@@H](NCc1cccn1C)[C@H]1CCCN(C(=O)OC(C)(C)C)C1 ZINC000217797790 DG On-Demand Unstable GPR119 26 43 C[C@H](O)c1ccc(NC(=O)N[C@H]2CCC[C@@H](C)[C@@H]2C)cc1 ZINC000217797794 CH For-Sale Unstable EPHX2 28 50 COc1ccc(CCNC(=O)N/C=C/c2ccccc2Cl)cc1OC ZINC000217797798 FH For-Sale Unstable CAN2 0 53 C=C(C)COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)ccc1OC ZINC000217797829 KK In-Stock Unstable AKR1B1 0 45 C=C(C)COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)ccc1OC ZINC000217797829 KK In-Stock Unstable CYP1B1 49 36 C=C(C)COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)ccc1OC ZINC000217797829 KK In-Stock Unstable CYP1A1 37 43 COC(=O)c1ccccc1C(=O)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217797836 HH In-Stock Unstable HRH3 28 48 N[C@H]1CC[C@@H](n2cc(C(=O)N3CCC[C@H]3C(=O)N3CCCCC3)nn2)CC1 ZINC000217797841 FD In-Stock Unstable PREP 69 49 C[C@H](NCc1cccn1C)[C@H]1CCCN(C(=O)OC(C)(C)C)C1 ZINC000217797861 DG On-Demand Unstable GPR119 26 43 COc1ccc2[nH]c(=O)c([C@@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(O)cc6)oc5c43)cc2c1 ZINC000217797951 JI In-Stock Unstable AKR1B1 0 42 COc1ccc2[nH]c(=O)c([C@@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(O)cc6)oc5c43)cc2c1 ZINC000217797951 JI In-Stock Unstable CYP1B1 28 42 COc1ccc2[nH]c(=O)c([C@@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(O)cc6)oc5c43)cc2c1 ZINC000217797951 JI In-Stock Unstable CYP1A1 24 42 COc1ccc2[nH]c(=O)c([C@@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(O)cc6)oc5c43)cc2c1 ZINC000217797951 JI In-Stock Unstable CYP1A2 18 42 Cc1nnsc1C(=O)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217797967 GG In-Stock Unstable HRH3 20 41 NC(=O)[C@@H]1CCCN([C@@H]2CCC[C@@H]2O)C1 ZINC000217797968 BC For-Sale Unstable VACHT_TETCF 0 42 NC(=O)[C@@H]1CCCN([C@@H]2CCC[C@@H]2O)C1 ZINC000217797968 BC For-Sale Unstable SLC18A3 38 43 NC(=O)[C@@H]1CCCN([C@@H]2CCC[C@@H]2O)C1 ZINC000217797968 BC For-Sale Unstable L3MBTL3 51 34 C[C@H](O)c1cccc(NC(=O)N[C@@H]2CCCC[C@@H]2C)c1 ZINC000217797973 CG For-Sale Unstable EPHX2 18 44 O=S(=O)(CCCO)Nc1ccc2c(c1)CCC2 ZINC000217798003 CD For-Sale Unstable MLNR 0 41 C[C@H](O)c1cccc(NC(=O)N[C@H]2CCCC[C@@H]2C)c1 ZINC000217798048 CG For-Sale Unstable EPHX2 18 44 COc1ccc2[nH]c(=O)c([C@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(O)cc6)oc5c43)cc2c1 ZINC000217798049 JI In-Stock Unstable AKR1B1 0 42 COc1ccc2[nH]c(=O)c([C@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(O)cc6)oc5c43)cc2c1 ZINC000217798049 JI In-Stock Unstable CYP1B1 28 42 COc1ccc2[nH]c(=O)c([C@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(O)cc6)oc5c43)cc2c1 ZINC000217798049 JI In-Stock Unstable CYP1A1 24 42 COc1ccc2[nH]c(=O)c([C@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(O)cc6)oc5c43)cc2c1 ZINC000217798049 JI In-Stock Unstable CYP1A2 18 42 Cc1nnsc1C(=O)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217798051 GG In-Stock Unstable HRH3 20 41 O[C@@H]1CCC[C@@H]1N1CCCc2ccccc21 ZINC000217798058 BE In-Stock Unstable VACHT_TETCF 0 44 COc1cc(C=O)ccc1OCCCCN1CCN(C)CC1 ZINC000217798060 DD In-Stock Unstable HTR1A 41 38 COc1cc(C=O)ccc1OCCCCN1CCN(C)CC1 ZINC000217798060 DD In-Stock Unstable DRD2 43 42 COc1cc(C=O)ccc1OCCCCN1CCN(C)CC1 ZINC000217798060 DD In-Stock Unstable ACHE 21 46 COc1cc(C=O)ccc1OCCCCN1CCN(C)CC1 ZINC000217798060 DD In-Stock Unstable HTR2A 28 44 COc1cc(C=O)ccc1OCCCCN1CCN(C)CC1 ZINC000217798060 DD In-Stock Unstable DRD3 42 42 COc1cc(C=O)ccc1OCCCCN1CCN(C)CC1 ZINC000217798060 DD In-Stock Unstable SIGMAR1 22 47 COc1cc(C=O)ccc1OCCCCN1CCN(C)CC1 ZINC000217798060 DD In-Stock Unstable SLC9A1 52 33 COc1cc(C=O)ccc1OCCCCN1CCN(C)CC1 ZINC000217798060 DD In-Stock Unstable EBP 15 40 COc1cc(C=O)ccc1OCCCCN1CCN(C)CC1 ZINC000217798060 DD In-Stock Unstable ABCB1 18 46 COc1cc(C=O)ccc1OCCCCN1CCN(C)CC1 ZINC000217798060 DD In-Stock Unstable SLC29A2 0 46 COc1cc(C=O)ccc1OCCCCN1CCN(C)CC1 ZINC000217798060 DD In-Stock Unstable ASF1A 0 42 CC[C@@H](CCO)NCCCn1ccnc1 ZINC000217798079 BD For-Sale Unstable TBXAS1 31 46 CC[C@@H](CCO)NCCCn1ccnc1 ZINC000217798079 BD For-Sale Unstable CAMC 0 44 CC[C@@H](CCO)NCCCn1ccnc1 ZINC000217798079 BD For-Sale Unstable QPCT 41 39 S=C1CCCN1CCCCN1CCN(c2cccc3sccc23)CC1 ZINC000217798104 FI For-Sale Unstable HTR1A 68 45 S=C1CCCN1CCCCN1CCN(c2cccc3sccc23)CC1 ZINC000217798104 FI For-Sale Unstable DRD2 56 44 S=C1CCCN1CCCCN1CCN(c2cccc3sccc23)CC1 ZINC000217798104 FI For-Sale Unstable DRD1 17 41 S=C1CCCN1CCCCN1CCN(c2cccc3sccc23)CC1 ZINC000217798104 FI For-Sale Unstable HTR2A 27 44 S=C1CCCN1CCCCN1CCN(c2cccc3sccc23)CC1 ZINC000217798104 FI For-Sale Unstable DRD3 36 44 C[C@H](O)c1ccc(NC(=O)N[C@@H]2CCCC[C@@H]2C)cc1 ZINC000217798123 CG For-Sale Unstable EPHX2 31 56 O=C(N/C=C/c1ccccc1Cl)NCc1cccnc1 ZINC000217798142 CG For-Sale Unstable PTAFR 25 41 O=C(N/C=C/c1ccccc1Cl)NCc1cccnc1 ZINC000217798142 CG For-Sale Unstable NAMPT 88 52 O[C@@H]1CCC[C@H]1N1CCCc2ccccc21 ZINC000217798150 BE In-Stock Unstable VACHT_TETCF 0 44 CC[C@H](CCO)NCCCn1ccnc1 ZINC000217798155 BD For-Sale Unstable TBXAS1 31 46 CC[C@H](CCO)NCCCn1ccnc1 ZINC000217798155 BD For-Sale Unstable CAMC 0 44 CC[C@H](CCO)NCCCn1ccnc1 ZINC000217798155 BD For-Sale Unstable QPCT 41 39 COc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217798173 FG In-Stock Unstable HTR1A 138 50 COc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217798173 FG In-Stock Unstable DRD2 89 48 COc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217798173 FG In-Stock Unstable DRD1 48 41 COc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217798173 FG In-Stock Unstable DRD4 58 50 COc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217798173 FG In-Stock Unstable ACHE 22 44 COc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217798173 FG In-Stock Unstable ADRA1D 51 44 COc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217798173 FG In-Stock Unstable HTR2A 88 47 COc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217798173 FG In-Stock Unstable HTR2C 31 43 COc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217798173 FG In-Stock Unstable SLC6A4 24 48 COc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217798173 FG In-Stock Unstable ADRA1A 49 45 COc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217798173 FG In-Stock Unstable ADRA1B 43 43 COc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217798173 FG In-Stock Unstable DRD3 89 50 COc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217798173 FG In-Stock Unstable DRD5 33 46 COc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217798173 FG In-Stock Unstable HTR7 118 43 COc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217798173 FG In-Stock Unstable SIGMAR1 40 53 COc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217798173 FG In-Stock Unstable BCHE 25 40 COc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217798173 FG In-Stock Unstable HTR6 0 40 COc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217798173 FG In-Stock Unstable ABCB1 28 45 COc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217798173 FG In-Stock Unstable MET 50 37 COc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217798173 FG In-Stock Unstable MCHR1 0 41 COc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217798173 FG In-Stock Unstable CACNA1G 26 40 COc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217798173 FG In-Stock Unstable EHMT2 50 39 COc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217798173 FG In-Stock Unstable SLC29A2 0 42 COc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217798173 FG In-Stock Unstable ACKR3 38 40 COc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217798173 FG In-Stock Unstable ASF1A 0 45 O=C(c1nc2ccccc2s1)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217798179 HJ In-Stock Unstable HRH3 18 40 O=C(c1nc2ccccc2s1)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217798179 HJ In-Stock Unstable TRY1_BOVIN 40 36 COC(=O)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)cc1 ZINC000217798192 GD For-Sale Unstable ADAMTS5 33 42 C[C@H](O)c1ccc(NC(=O)N[C@H]2CCCC[C@@H]2C)cc1 ZINC000217798210 CG For-Sale Unstable EPHX2 31 56 C[C@@H]1CCc2ccccc2N1C(=O)C1CCN(c2nc3ccccc3o2)CC1 ZINC000217798244 GI On-Demand Unstable HCRTR1 17 48 C[C@@H]1CCc2ccccc2N1C(=O)C1CCN(c2nc3ccccc3o2)CC1 ZINC000217798244 GI On-Demand Unstable SORD 15 40 O=C(c1nc2ccccc2s1)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217798259 HJ In-Stock Unstable HRH3 18 40 O=C(c1nc2ccccc2s1)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217798259 HJ In-Stock Unstable TRY1_BOVIN 40 36 O[C@@H]1CCC[C@@H]1N1CCc2ccccc2C1 ZINC000217798270 BD In-Stock Unstable VACHT_TETCF 0 51 O[C@@H]1CCC[C@@H]1N1CCc2ccccc2C1 ZINC000217798270 BD In-Stock Unstable CHRNA6 0 41 O[C@@H]1CCC[C@@H]1N1CCc2ccccc2C1 ZINC000217798270 BD In-Stock Unstable SLC18A3 42 38 CC(C)(C)NC(=O)N/C=C/c1ccccc1Cl ZINC000217798271 CG For-Sale Unstable ECR 44 35 COC(=O)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)cc1 ZINC000217798290 GD For-Sale Unstable ADAMTS5 33 42 C[C@H]1CCc2ccccc2N1C(=O)C1CCN(c2nc3ccccc3o2)CC1 ZINC000217798358 GI On-Demand Unstable HCRTR1 17 48 C[C@H]1CCc2ccccc2N1C(=O)C1CCN(c2nc3ccccc3o2)CC1 ZINC000217798358 GI On-Demand Unstable SORD 15 40 O[C@@H]1CCC[C@H]1N1CCc2ccccc2C1 ZINC000217798360 BD In-Stock Unstable VACHT_TETCF 0 51 O[C@@H]1CCC[C@H]1N1CCc2ccccc2C1 ZINC000217798360 BD In-Stock Unstable CHRNA6 0 41 O[C@@H]1CCC[C@H]1N1CCc2ccccc2C1 ZINC000217798360 BD In-Stock Unstable SLC18A3 42 38 O=C(CSc1ccc(F)cc1)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217798362 IJ In-Stock Unstable HRH3 18 41 CCOc1cc(C=O)ccc1OCCCCN(C)C ZINC000217798363 CF In-Stock Unstable THRA 42 42 CCOc1cc(C=O)ccc1OCCCCN(C)C ZINC000217798363 CF In-Stock Unstable THRB 0 42 O=C(N/C=C/c1ccccc1Cl)N1CCC(Cc2ccccc2)CC1 ZINC000217798385 FJ For-Sale Unstable GRIN2B 82 47 O=C(N/C=C/c1ccccc1Cl)N1CCC(Cc2ccccc2)CC1 ZINC000217798385 FJ For-Sale Unstable SIGMAR1 30 43 O=C(N/C=C/c1ccccc1Cl)N1CCC(Cc2ccccc2)CC1 ZINC000217798385 FJ For-Sale Unstable CCR3 53 43 c1ccc(C(OC2CC3(CNC3)C2)c2ccccc2)cc1 ZINC000217798398 CH In-Stock Unstable CHRM1 0 43 c1ccc(C(OC2CC3(CNC3)C2)c2ccccc2)cc1 ZINC000217798398 CH In-Stock Unstable SLC6A3 15 43 C[C@H]1C[C@@H](C)CN(C(=O)Nc2cccc([C@H](C)O)c2)C1 ZINC000217798448 CG For-Sale Unstable RBP4 46 32 O=C(CSc1ccc(F)cc1)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217798449 IJ In-Stock Unstable HRH3 18 41 CCOc1cc(C=O)ccc1OCCCCN1CCCC1 ZINC000217798474 CG In-Stock Unstable ACHE 19 44 CCOc1cc(C=O)ccc1OCCCCN1CCCC1 ZINC000217798474 CG In-Stock Unstable LTA4H 20 40 CCOc1cc(C=O)ccc1OCCCCN1CCCC1 ZINC000217798474 CG In-Stock Unstable HRH3 53 41 CCOc1cc(C=O)ccc1OCCCCN1CCCC1 ZINC000217798474 CG In-Stock Unstable PSMB2 44 34 COc1ccc(CCN2C(=O)N[C@@H](CC(=O)NCCc3ccc(O)cc3)C2=O)cc1OC ZINC000217798475 ID In-Stock Unstable NCE103 15 49 COc1ccc(CCN2C(=O)N[C@@H](CC(=O)NCCc3ccc(O)cc3)C2=O)cc1OC ZINC000217798475 ID In-Stock Unstable CAN2 0 49 C[C@@H]1CCCCN1C(=O)C[C@@H](CC(=O)O)c1ccccc1 ZINC000217798476 CG In-Stock Unstable COLA 72 35 C[C@@H]1CCCCN1C(=O)C[C@@H](CC(=O)O)c1ccccc1 ZINC000217798476 CG In-Stock Unstable CPT1A 70 34 C[C@@H]1CCCCN1C(=O)C[C@@H](CC(=O)O)c1ccccc1 ZINC000217798476 CG In-Stock Unstable PREP 49 36 C[C@@H]1CCCCN1C(=O)C[C@@H](CC(=O)O)c1ccccc1 ZINC000217798476 CG In-Stock Unstable MTNR1B 29 40 CCN(CC)c1ccc(NC(=S)NCCO)cc1 ZINC000217798480 CD For-Sale Unstable QPCT 46 38 C[C@H]1CCCCN1C(=O)C[C@@H](CC(=O)O)c1ccccc1 ZINC000217798539 CG In-Stock Unstable COLA 72 35 C[C@H]1CCCCN1C(=O)C[C@@H](CC(=O)O)c1ccccc1 ZINC000217798539 CG In-Stock Unstable CPT1A 70 34 C[C@H]1CCCCN1C(=O)C[C@@H](CC(=O)O)c1ccccc1 ZINC000217798539 CG In-Stock Unstable PREP 49 36 C[C@H]1CCCCN1C(=O)C[C@@H](CC(=O)O)c1ccccc1 ZINC000217798539 CG In-Stock Unstable MTNR1B 29 40 C[C@H](O)c1cccc(NC(=O)N2C[C@H](C)C[C@@H](C)C2)c1 ZINC000217798564 CG For-Sale Unstable RBP4 46 32 COc1ccc(CCNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217798599 EH For-Sale Unstable MTNR1A 66 45 COc1ccc(CCNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217798599 EH For-Sale Unstable MTNR1B 57 45 COc1ccc(CCNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217798599 EH For-Sale Unstable CA9 18 45 COc1ccc(CCNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217798599 EH For-Sale Unstable NCE103 23 41 COc1ccc(CCNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217798599 EH For-Sale Unstable CAN2 0 41 CCOc1cc(C=O)ccc1OCCCCN1CCC(C)CC1 ZINC000217798603 DH In-Stock Unstable HRH3 15 41 CCOc1cc(C=O)ccc1OCCCCN1CCC(C)CC1 ZINC000217798603 DH In-Stock Unstable SIGMAR1 16 40 CCOc1cc(C=O)ccc1OCCCCN1CCC(C)CC1 ZINC000217798603 DH In-Stock Unstable EBP 16 43 C[C@@H]1CCCCN1C(=O)C[C@H](CC(=O)O)c1ccccc1 ZINC000217798613 CG In-Stock Unstable COLA 72 35 C[C@@H]1CCCCN1C(=O)C[C@H](CC(=O)O)c1ccccc1 ZINC000217798613 CG In-Stock Unstable CPT1A 70 34 C[C@@H]1CCCCN1C(=O)C[C@H](CC(=O)O)c1ccccc1 ZINC000217798613 CG In-Stock Unstable PREP 49 36 C[C@@H]1CCCCN1C(=O)C[C@H](CC(=O)O)c1ccccc1 ZINC000217798613 CG In-Stock Unstable MTNR1B 29 40 O[C@@H]1CCC[C@@H]1N1CCc2ccccc21 ZINC000217798623 BD For-Sale Unstable VACHT_TETCF 0 44 C[C@H]1C[C@@H](C)CN(C(=O)Nc2ccc([C@H](C)O)cc2)C1 ZINC000217798630 CG For-Sale Unstable EPHX2 27 44 C[C@H]1C[C@@H](C)CN(C(=O)Nc2ccc([C@H](C)O)cc2)C1 ZINC000217798630 CG For-Sale Unstable RBP4 41 31 O=S(=O)(Cc1ccc(C(F)(F)F)cc1)NC[C@@H]1CCCN1c1nccs1 ZINC000217798656 HG For-Sale Unstable ADAMTS5 31 45 C[C@H]1CCCCN1C(=O)C[C@H](CC(=O)O)c1ccccc1 ZINC000217798676 CG In-Stock Unstable COLA 72 35 C[C@H]1CCCCN1C(=O)C[C@H](CC(=O)O)c1ccccc1 ZINC000217798676 CG In-Stock Unstable CPT1A 70 34 C[C@H]1CCCCN1C(=O)C[C@H](CC(=O)O)c1ccccc1 ZINC000217798676 CG In-Stock Unstable PREP 49 36 C[C@H]1CCCCN1C(=O)C[C@H](CC(=O)O)c1ccccc1 ZINC000217798676 CG In-Stock Unstable MTNR1B 29 40 O=C(N/C=C/c1ccccc1Cl)NC[C@@H]1CCCO1 ZINC000217798694 CF For-Sale Unstable OXTR 25 44 CCOc1cc(C=O)ccc1OCCCCN1CCCC[C@@H]1C ZINC000217798696 DH In-Stock Unstable HRH3 44 41 CCN1Cc2ccccc2C[C@@H]1C(=O)N1CC(c2nc3ccccc3[nH]2)C1 ZINC000217798705 FF In-Stock Unstable PREP 22 41 CCN1Cc2ccccc2C[C@@H]1C(=O)N1CC(c2nc3ccccc3[nH]2)C1 ZINC000217798705 FF In-Stock Unstable ADAM9 69 37 O[C@@H]1CCC[C@H]1N1CCc2ccccc21 ZINC000217798711 BD For-Sale Unstable VACHT_TETCF 0 44 C[C@H](O)c1ccc(NC(=O)N2C[C@H](C)C[C@@H](C)C2)cc1 ZINC000217798715 CG For-Sale Unstable EPHX2 27 44 C[C@H](O)c1ccc(NC(=O)N2C[C@H](C)C[C@@H](C)C2)cc1 ZINC000217798715 CG For-Sale Unstable RBP4 41 31 O=S(=O)(Cc1ccc(C(F)(F)F)cc1)NC[C@H]1CCCN1c1nccs1 ZINC000217798732 HG For-Sale Unstable ADAMTS5 31 45 CCN(CCNC(=O)c1ccc(Cl)c([N+](=O)[O-])c1)C1CC1 ZINC000217798737 DE On-Demand Unstable TAAR1 15 43 Cc1cc(C(=O)N2CCC[C@H](Cc3nc(-c4ccccc4F)no3)C2)no1 ZINC000217798741 FG In-Stock Unstable HRH3 29 46 CCN1Cc2ccccc2C[C@H]1C(=O)N1CC(c2nc3ccccc3[nH]2)C1 ZINC000217798759 FF In-Stock Unstable PREP 22 41 CCN1Cc2ccccc2C[C@H]1C(=O)N1CC(c2nc3ccccc3[nH]2)C1 ZINC000217798759 FF In-Stock Unstable ADAM9 69 37 CCOc1cc(C=O)ccc1OCCCCN1CCCC[C@H]1C ZINC000217798769 DH In-Stock Unstable HRH3 44 41 O=C(N/C=C/c1ccccc1Cl)NC[C@H]1CCCO1 ZINC000217798778 CF For-Sale Unstable OXTR 25 44 C[C@@H]1CCCN(C(=O)C[C@@H](CC(=O)O)c2ccccc2)C1 ZINC000217798785 CF In-Stock Unstable PREP 45 37 CC1(C)CCc2cc(CC(=O)N[C@H](CO)Cc3ccccc3)ccc2O1 ZINC000217798787 FG In-Stock Unstable MME 46 43 CC1(C)CCc2cc(CC(=O)N[C@H](CO)Cc3ccccc3)ccc2O1 ZINC000217798787 FG In-Stock Unstable TIMP3 53 33 CC1(C)CCc2cc(CC(=O)N[C@H](CO)Cc3ccccc3)ccc2O1 ZINC000217798787 FG In-Stock Unstable DAGLA 25 44 CC1(C)CCc2cc(CC(=O)N[C@H](CO)Cc3ccccc3)ccc2O1 ZINC000217798787 FG In-Stock Unstable PSMB8 55 31 C[C@@H]1CCc2ccccc2N1C(=O)CCc1ncc(-c2ccc(Cl)cc2)o1 ZINC000217798800 GK On-Demand Unstable DRD4 24 40 C[C@@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1ccc(C#N)cc1 ZINC000217798801 CC For-Sale Unstable CTSC 30 48 Cc1cc(C(=O)N2CCC[C@@H](Cc3nc(-c4ccccc4F)no3)C2)no1 ZINC000217798814 FG In-Stock Unstable HRH3 29 46 O[C@@H]1CCCN([C@H]2CCC[C@H]2O)C1 ZINC000217798816 AC For-Sale Unstable VACHT_TETCF 0 41 O[C@@H]1CCCN([C@H]2CCC[C@H]2O)C1 ZINC000217798816 AC For-Sale Unstable SLC18A3 26 47 O[C@@H]1CCCN([C@H]2CCC[C@H]2O)C1 ZINC000217798816 AC For-Sale Unstable MAN2B1 0 45 O[C@@H]1CCCN([C@H]2CCC[C@H]2O)C1 ZINC000217798816 AC For-Sale Unstable MAN2C1 0 45 O[C@@H]1CCCN([C@H]2CCC[C@H]2O)C1 ZINC000217798816 AC For-Sale Unstable ALPHA-MAN-IA 0 45 C[C@@H](c1ccc(Cl)cc1)N(C)[C@H](C)C(=O)c1ccccc1 ZINC000217798820 DJ For-Sale Unstable SLC6A1 0 40 C[C@@H](c1ccc(Cl)cc1)N(C)[C@H](C)C(=O)c1ccccc1 ZINC000217798820 DJ For-Sale Unstable SLC6A9 0 41 C[C@@H](c1ccc(Cl)cc1)N(C)[C@H](C)C(=O)c1ccccc1 ZINC000217798820 DJ For-Sale Unstable UTS2 65 43 C[C@H]1CCCN(C(=O)C[C@@H](CC(=O)O)c2ccccc2)C1 ZINC000217798856 CF In-Stock Unstable PREP 45 37 C[C@@H](NC(=O)N/C=C/c1ccccc1Cl)c1ccccc1 ZINC000217798861 DI For-Sale Unstable KCNQ2 54 50 C[C@@H](NC(=O)N/C=C/c1ccccc1Cl)c1ccccc1 ZINC000217798861 DI For-Sale Unstable MENB 0 40 C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1ccc(C#N)cc1 ZINC000217798875 CC For-Sale Unstable CTSC 30 48 C[C@H]1CCc2ccccc2N1C(=O)CCc1ncc(-c2ccc(Cl)cc2)o1 ZINC000217798883 GK On-Demand Unstable DRD4 24 40 O[C@H]1CCC[C@@H]1N1CCC[C@@H](O)C1 ZINC000217798885 AC For-Sale Unstable VACHT_TETCF 0 41 O[C@H]1CCC[C@@H]1N1CCC[C@@H](O)C1 ZINC000217798885 AC For-Sale Unstable SLC18A3 26 47 O[C@H]1CCC[C@@H]1N1CCC[C@@H](O)C1 ZINC000217798885 AC For-Sale Unstable MAN2B1 0 45 O[C@H]1CCC[C@@H]1N1CCC[C@@H](O)C1 ZINC000217798885 AC For-Sale Unstable MAN2C1 0 45 O[C@H]1CCC[C@@H]1N1CCC[C@@H](O)C1 ZINC000217798885 AC For-Sale Unstable ALPHA-MAN-IA 0 45 O=C(CCSc1ccccc1)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217798891 IJ In-Stock Unstable HRH3 20 43 COc1cc2cc(C(=O)NC[C@@H]3CCCN4CCCC[C@H]34)n(C)c2cc1OC ZINC000217798913 GG In-Stock Unstable HTR4 17 51 C[C@@H]1CCCN(C(=O)C[C@H](CC(=O)O)c2ccccc2)C1 ZINC000217798932 CF In-Stock Unstable PREP 45 37 O[C@@H]1CCCN([C@@H]2CCC[C@H]2O)C1 ZINC000217798955 AC On-Demand Unstable VACHT_TETCF 0 41 O[C@@H]1CCCN([C@@H]2CCC[C@H]2O)C1 ZINC000217798955 AC On-Demand Unstable SLC18A3 26 47 O[C@@H]1CCCN([C@@H]2CCC[C@H]2O)C1 ZINC000217798955 AC On-Demand Unstable MAN2B1 0 45 O[C@@H]1CCCN([C@@H]2CCC[C@H]2O)C1 ZINC000217798955 AC On-Demand Unstable MAN2C1 0 45 O[C@@H]1CCCN([C@@H]2CCC[C@H]2O)C1 ZINC000217798955 AC On-Demand Unstable ALPHA-MAN-IA 0 45 C[C@@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1ccc(C#N)cc1 ZINC000217798958 CC For-Sale Unstable CTSC 30 48 C[C@H](NC(=O)N/C=C/c1ccccc1Cl)c1ccccc1 ZINC000217798959 DI For-Sale Unstable KCNQ2 54 50 C[C@H](NC(=O)N/C=C/c1ccccc1Cl)c1ccccc1 ZINC000217798959 DI For-Sale Unstable MENB 0 40 O=C(CCSc1ccccc1)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217798980 IJ In-Stock Unstable HRH3 20 43 C[C@@H](c1ccccc1Cl)N(C)[C@H](C)C(=O)c1ccccc1 ZINC000217798993 DJ For-Sale Unstable CXCL8 45 38 C[C@H]1CCCN(C(=O)C[C@H](CC(=O)O)c2ccccc2)C1 ZINC000217799013 CF In-Stock Unstable PREP 45 37 CCOc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)cc1 ZINC000217799014 FE For-Sale Unstable ADAMTS5 35 43 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc3nccnc23)CC(=O)O4)cc1O ZINC000217799018 JI In-Stock Unstable AKR1B1 0 42 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc3nccnc23)CC(=O)O4)cc1O ZINC000217799018 JI In-Stock Unstable CYP1B1 47 36 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc3nccnc23)CC(=O)O4)cc1O ZINC000217799018 JI In-Stock Unstable CYP1A1 34 42 C[C@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1ccc(C#N)cc1 ZINC000217799044 CC For-Sale Unstable CTSC 30 48 O[C@H]1CCC[C@H]1N1CCC[C@@H](O)C1 ZINC000217799045 AC For-Sale Unstable VACHT_TETCF 0 41 O[C@H]1CCC[C@H]1N1CCC[C@@H](O)C1 ZINC000217799045 AC For-Sale Unstable SLC18A3 26 47 O[C@H]1CCC[C@H]1N1CCC[C@@H](O)C1 ZINC000217799045 AC For-Sale Unstable MAN2B1 0 45 O[C@H]1CCC[C@H]1N1CCC[C@@H](O)C1 ZINC000217799045 AC For-Sale Unstable MAN2C1 0 45 O[C@H]1CCC[C@H]1N1CCC[C@@H](O)C1 ZINC000217799045 AC For-Sale Unstable ALPHA-MAN-IA 0 45 O=C(N/C=C/c1ccccc1Cl)NC(c1ccccc1)c1ccccc1 ZINC000217799068 FK For-Sale Anodyne KCNQ2 21 42 CN(C)c1ccc(C(=O)N2CCC[C@H](Cc3nc(-c4ccccc4F)no3)C2)cc1 ZINC000217799082 HI In-Stock Unstable HRH3 24 49 COc1ccccc1[C@@H](O)P(=O)(OC)OC ZINC000217799083 BE In-Stock Unstable KCNK3 32 40 COc1ccccc1[C@@H](O)P(=O)(OC)OC ZINC000217799083 BE In-Stock Unstable KCNK9 28 40 CCOc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)cc1 ZINC000217799084 FE For-Sale Unstable ADAMTS5 35 43 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc3nccnc23)CC(=O)O4)cc1O ZINC000217799089 JI In-Stock Unstable AKR1B1 0 42 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc3nccnc23)CC(=O)O4)cc1O ZINC000217799089 JI In-Stock Unstable CYP1B1 47 36 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc3nccnc23)CC(=O)O4)cc1O ZINC000217799089 JI In-Stock Unstable CYP1A1 34 42 COc1ccccc1[C@H](O)P(=O)(OC)OC ZINC000217799162 BE In-Stock Unstable KCNK3 32 40 COc1ccccc1[C@H](O)P(=O)(OC)OC ZINC000217799162 BE In-Stock Unstable KCNK9 28 40 CN(C)c1ccc(C(=O)N2CCC[C@@H](Cc3nc(-c4ccccc4F)no3)C2)cc1 ZINC000217799166 HI In-Stock Unstable HRH3 24 49 CCOc1cc(C=O)ccc1OCCCCN1CCCCCC1 ZINC000217799168 DH In-Stock Unstable ACHE 20 46 CCOc1cc(C=O)ccc1OCCCCN1CCCCCC1 ZINC000217799168 DH In-Stock Unstable HTR4 19 44 CCOc1cc(C=O)ccc1OCCCCN1CCCCCC1 ZINC000217799168 DH In-Stock Unstable THRB 0 40 CCOc1cc(C=O)ccc1OCCCCN1CCCCCC1 ZINC000217799168 DH In-Stock Unstable HRH3 70 43 CCOc1cc(C=O)ccc1OCCCCN1CCCCCC1 ZINC000217799168 DH In-Stock Unstable HNMT 45 30 CCOc1cc(C=O)ccc1OCCCCN1CCCCCC1 ZINC000217799168 DH In-Stock Unstable PSMB2 46 36 CCOc1cc(C=O)ccc1OCCCCN1CCCCCC1 ZINC000217799168 DH In-Stock Unstable PSMB1 40 36 OC[C@@H]1CCCN([C@@H]2CCC[C@@H]2O)C1 ZINC000217799177 AC For-Sale Unstable SLC18A3 37 46 OC[C@@H]1CCCN([C@@H]2CCC[C@@H]2O)C1 ZINC000217799177 AC For-Sale Unstable MAN2B1 0 40 OC[C@@H]1CCCN([C@@H]2CCC[C@@H]2O)C1 ZINC000217799177 AC For-Sale Unstable MAN2C1 0 40 OC[C@@H]1CCCN([C@@H]2CCC[C@@H]2O)C1 ZINC000217799177 AC For-Sale Unstable ALPHA-MAN-IA 0 40 COc1ccc(CNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217799182 DH For-Sale Unstable ANPEP 22 44 COc1ccc(CNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217799182 DH For-Sale Unstable MTNR1A 21 46 COc1ccc(CNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217799182 DH For-Sale Unstable MTNR1B 15 46 COc1ccc(CNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217799182 DH For-Sale Unstable CA9 18 43 COc1ccc(CNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217799182 DH For-Sale Unstable PROKR1 44 33 C[C@@H](c1cccc(Cl)c1)N(C)[C@H](C)C(=O)c1ccccc1 ZINC000217799193 DJ For-Sale Unstable ADRB1 24 41 C[C@@H](c1cccc(Cl)c1)N(C)[C@H](C)C(=O)c1ccccc1 ZINC000217799193 DJ For-Sale Unstable ADRB3 36 41 C[C@@H](c1cccc(Cl)c1)N(C)[C@H](C)C(=O)c1ccccc1 ZINC000217799193 DJ For-Sale Unstable SLC22A7 0 40 C[C@@H](c1cccc(Cl)c1)N(C)[C@H](C)C(=O)c1ccccc1 ZINC000217799193 DJ For-Sale Unstable PDS 21 40 CCn1ccnc1CNC1CCN(C(=O)OC(C)(C)C)CC1 ZINC000217799215 DE On-Demand Unstable GPR119 43 46 CN(C)c1ccc(NC(=S)NCCO)cc1 ZINC000217799239 BD For-Sale Unstable QPCT 41 36 N[C@@H]1C[C@@H]1NS(=O)(=O)N1CCc2ccccc2C1 ZINC000217799249 CB For-Sale Unstable AKR1C3 62 44 CC1=C(c2ccccc2)[C@@H]1C(=O)NCCc1nc2cc(Cl)ccc2[nH]1 ZINC000217799308 FH In-Stock Unstable F9 36 51 CC1=C(c2ccccc2)[C@@H]1C(=O)NCCc1nc2cc(Cl)ccc2[nH]1 ZINC000217799308 FH In-Stock Unstable CYSP_TRYCR 0 51 CC1=C(c2ccccc2)[C@@H]1C(=O)NCCc1nc2cc(Cl)ccc2[nH]1 ZINC000217799308 FH In-Stock Unstable PYGL 50 36 CC1=C(c2ccccc2)[C@@H]1C(=O)NCCc1nc2cc(Cl)ccc2[nH]1 ZINC000217799308 FH In-Stock Unstable PIN1 34 45 CC1=C(c2ccccc2)[C@@H]1C(=O)NCCc1nc2cc(Cl)ccc2[nH]1 ZINC000217799308 FH In-Stock Unstable NR2E3 61 32 O[C@@H]1CCC[C@@H]1N1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217799335 BE For-Sale Unstable VACHT_TETCF 0 46 O[C@@H]1CCC[C@@H]1N1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217799335 BE For-Sale Unstable CYP2D26 0 44 O[C@@H]1CCC[C@@H]1N1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217799335 BE For-Sale Unstable SLC18A3 52 75 Cn1cccc1CNC1CCN(C(=O)OC(C)(C)C)CC1 ZINC000217799340 CF On-Demand Unstable CCR8 21 41 Cn1cccc1CNC1CCN(C(=O)OC(C)(C)C)CC1 ZINC000217799340 CF On-Demand Unstable GPR119 44 44 N[C@@H]1C[C@H]1NS(=O)(=O)N1CCc2ccccc2C1 ZINC000217799344 CB For-Sale Unstable AKR1C3 62 44 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1ccc(F)cc1F ZINC000217799376 FE For-Sale Unstable ADAMTS5 30 41 O=C(CN1CCN(Cc2cnc(-c3ccccc3)s2)CC1)NCc1ccccc1 ZINC000217799386 HG On-Demand Unstable ACHE 15 40 O=C(CN1CCN(Cc2cnc(-c3ccccc3)s2)CC1)NCc1ccccc1 ZINC000217799386 HG On-Demand Unstable SIGMAR1 19 41 O=C(CN1CCN(Cc2cnc(-c3ccccc3)s2)CC1)NCc1ccccc1 ZINC000217799386 HG On-Demand Unstable MGEA5 36 44 CC1=C(c2ccccc2)[C@H]1C(=O)NCCc1nc2cc(Cl)ccc2[nH]1 ZINC000217799388 FH In-Stock Unstable F9 36 51 CC1=C(c2ccccc2)[C@H]1C(=O)NCCc1nc2cc(Cl)ccc2[nH]1 ZINC000217799388 FH In-Stock Unstable CYSP_TRYCR 0 51 CC1=C(c2ccccc2)[C@H]1C(=O)NCCc1nc2cc(Cl)ccc2[nH]1 ZINC000217799388 FH In-Stock Unstable PYGL 50 36 CC1=C(c2ccccc2)[C@H]1C(=O)NCCc1nc2cc(Cl)ccc2[nH]1 ZINC000217799388 FH In-Stock Unstable PIN1 34 45 CC1=C(c2ccccc2)[C@H]1C(=O)NCCc1nc2cc(Cl)ccc2[nH]1 ZINC000217799388 FH In-Stock Unstable NR2E3 61 32 O=C(N/C=C/c1ccccc1Cl)NCc1ccc2c(c1)OCO2 ZINC000217799391 EH For-Sale Unstable PDE5A 30 41 O=C(N/C=C/c1ccccc1Cl)NCc1ccc2c(c1)OCO2 ZINC000217799391 EH For-Sale Unstable KCNQ2 15 50 O=C(N/C=C/c1ccccc1Cl)NCc1ccc2c(c1)OCO2 ZINC000217799391 EH For-Sale Unstable SCN9A 24 43 O=C(N/C=C/c1ccccc1Cl)NCc1ccc2c(c1)OCO2 ZINC000217799391 EH For-Sale Unstable NOS2 84 36 O=C(N/C=C/c1ccccc1Cl)NCc1ccc2c(c1)OCO2 ZINC000217799391 EH For-Sale Unstable MCHR1 18 43 COc1ccc(/C=C2\Oc3c(ccc4c3[C@H](c3ccc(O)c(Cl)c3)CC(=O)O4)C2=O)cc1 ZINC000217799398 IK In-Stock Unstable HSD17B3 18 41 O[C@H]1CCC[C@@H]1N1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217799416 BE For-Sale Unstable VACHT_TETCF 0 46 O[C@H]1CCC[C@@H]1N1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217799416 BE For-Sale Unstable CYP2D26 0 44 O[C@H]1CCC[C@@H]1N1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217799416 BE For-Sale Unstable SLC18A3 52 75 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1ccc(F)cc1F ZINC000217799459 FE For-Sale Unstable ADAMTS5 30 41 Cn1cc(C(=O)N2CCC[C@H](Cc3nc(-c4ccccc4F)no3)C2)nn1 ZINC000217799464 FE In-Stock Unstable HRH3 27 46 COc1ccc(/C=C2\Oc3c(ccc4c3[C@@H](c3ccc(O)c(Cl)c3)CC(=O)O4)C2=O)cc1 ZINC000217799481 IK In-Stock Unstable HSD17B3 18 41 O[C@@H]1CCC[C@H]1N1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217799487 BE For-Sale Unstable VACHT_TETCF 0 46 O[C@@H]1CCC[C@H]1N1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217799487 BE For-Sale Unstable CYP2D26 0 44 O[C@@H]1CCC[C@H]1N1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217799487 BE For-Sale Unstable SLC18A3 52 75 O=C(CN1CCN(CCOc2cc(Cl)ccc2Cl)CC1)NCc1ccccc1 ZINC000217799490 HG On-Demand Unstable HTR1A 28 42 O=C(CN1CCN(CCOc2cc(Cl)ccc2Cl)CC1)NCc1ccccc1 ZINC000217799490 HG On-Demand Unstable DRD2 36 42 O=C(CN1CCN(CCOc2cc(Cl)ccc2Cl)CC1)NCc1ccccc1 ZINC000217799490 HG On-Demand Unstable DRD4 44 35 O=C(CN1CCN(CCOc2cc(Cl)ccc2Cl)CC1)NCc1ccccc1 ZINC000217799490 HG On-Demand Unstable SLC6A4 15 41 O=C(CN1CCN(CCOc2cc(Cl)ccc2Cl)CC1)NCc1ccccc1 ZINC000217799490 HG On-Demand Unstable HRH1 25 42 O=C(CN1CCN(CCOc2cc(Cl)ccc2Cl)CC1)NCc1ccccc1 ZINC000217799490 HG On-Demand Unstable PTGER1 44 37 O=C(CN1CCN(CCOc2cc(Cl)ccc2Cl)CC1)NCc1ccccc1 ZINC000217799490 HG On-Demand Unstable HRP1_PLAFA 55 35 O=C(CN1CCN(CCOc2cc(Cl)ccc2Cl)CC1)NCc1ccccc1 ZINC000217799490 HG On-Demand Unstable HTR7 44 50 O=C(CN1CCN(CCOc2cc(Cl)ccc2Cl)CC1)NCc1ccccc1 ZINC000217799490 HG On-Demand Unstable KCNA5 0 53 O=C(CN1CCN(CCOc2cc(Cl)ccc2Cl)CC1)NCc1ccccc1 ZINC000217799490 HG On-Demand Unstable SIGMAR1 32 42 O=C(CN1CCN(CCOc2cc(Cl)ccc2Cl)CC1)NCc1ccccc1 ZINC000217799490 HG On-Demand Unstable RPA1 56 37 O=C(CN1CCN(CCOc2cc(Cl)ccc2Cl)CC1)NCc1ccccc1 ZINC000217799490 HG On-Demand Unstable PDS 44 39 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217799493 FF For-Sale Unstable CA2 100 57 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217799493 FF For-Sale Unstable CA1 95 57 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217799493 FF For-Sale Unstable CA7 40 48 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217799493 FF For-Sale Unstable CA5B 51 48 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217799493 FF For-Sale Unstable CA4 70 56 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217799493 FF For-Sale Unstable CA5A 58 48 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217799493 FF For-Sale Unstable CA14 37 48 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217799493 FF For-Sale Unstable CA12 86 57 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217799493 FF For-Sale Unstable CA9 84 57 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217799493 FF For-Sale Unstable UREA_CANEN 32 40 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217799493 FF For-Sale Unstable NCE103 47 46 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217799493 FF For-Sale Unstable MTCA1 65 56 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217799493 FF For-Sale Unstable P96878_MYCTU 83 56 CN(C)CC[C@@H](CCO)c1ccccc1 ZINC000217799516 BE In-Stock Unstable ADRA1D 0 44 CN(C)CC[C@@H](CCO)c1ccccc1 ZINC000217799516 BE In-Stock Unstable HRH1 16 44 CN(C)CC[C@@H](CCO)c1ccccc1 ZINC000217799516 BE In-Stock Unstable UTS2 49 37 COc1nc(Br)nc2ccc(O)cc12 ZINC000217799544 CE For-Sale Unstable ESRRA 48 44 COc1nc(Br)nc2ccc(O)cc12 ZINC000217799544 CE For-Sale Unstable ESRRB 51 44 Cn1cc(C(=O)N2CCC[C@@H](Cc3nc(-c4ccccc4F)no3)C2)nn1 ZINC000217799545 FE In-Stock Unstable HRH3 27 46 CCOc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217799562 GH In-Stock Unstable HTR1A 97 49 CCOc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217799562 GH In-Stock Unstable DRD2 65 46 CCOc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217799562 GH In-Stock Unstable DRD1 36 46 CCOc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217799562 GH In-Stock Unstable DRD4 41 41 CCOc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217799562 GH In-Stock Unstable HTR2A 67 45 CCOc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217799562 GH In-Stock Unstable SLC6A4 17 41 CCOc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217799562 GH In-Stock Unstable ADRA1A 32 44 CCOc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217799562 GH In-Stock Unstable DRD3 71 49 CCOc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217799562 GH In-Stock Unstable DRD5 32 46 CCOc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217799562 GH In-Stock Unstable HTR7 99 52 CCOc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217799562 GH In-Stock Unstable SIGMAR1 30 48 CCOc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217799562 GH In-Stock Unstable HTR6 0 41 CCOc1cc(C=O)ccc1OCCCCN1CCN(c2ccccc2)CC1 ZINC000217799562 GH In-Stock Unstable ABCB1 23 44 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1cc(F)cc(F)c1 ZINC000217799570 FE For-Sale Unstable ADAMTS5 32 43 CCCCCC[C@@H](C)NCCN(C)[C@@H](C)CC ZINC000217799588 BH For-Sale Unstable ADH1B 0 41 CCCCCC[C@@H](C)NCCN(C)[C@@H](C)CC ZINC000217799588 BH For-Sale Unstable ADH1C 0 41 Cc1cccc(OCC(C)C)c1C ZINC000217799589 AG On-Demand Unstable ADRB2 0 43 CN(C)CC[C@H](CCO)c1ccccc1 ZINC000217799601 BE In-Stock Unstable ADRA1D 0 44 CN(C)CC[C@H](CCO)c1ccccc1 ZINC000217799601 BE In-Stock Unstable HRH1 16 44 CN(C)CC[C@H](CCO)c1ccccc1 ZINC000217799601 BE In-Stock Unstable UTS2 49 37 O=S1(=O)CC[C@H](N[C@@H]2CCCC[C@@H]2c2ccccc2)C1 ZINC000217799619 CE For-Sale Unstable GRIA4 15 43 C[C@H](O)c1cccc(NC(=O)N[C@@H]2CCC[C@@H](C)C2)c1 ZINC000217799631 CG For-Sale Unstable EPHX2 38 48 Cc1noc(C)c1CC(=O)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217799653 GH In-Stock Unstable HRH3 20 41 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1cc(F)cc(F)c1 ZINC000217799660 FE For-Sale Unstable ADAMTS5 32 43 O[C@@H]1CCC[C@@H]1N1CCC[C@@H]2CCCC[C@H]21 ZINC000217799668 BF For-Sale Unstable SLC18A3 42 53 CCCCCC[C@H](C)NCCN(C)[C@@H](C)CC ZINC000217799673 BH For-Sale Unstable ADH1B 0 41 CCCCCC[C@H](C)NCCN(C)[C@@H](C)CC ZINC000217799673 BH For-Sale Unstable ADH1C 0 41 OCC[C@@H](CCN1CCOCC1)c1ccccc1 ZINC000217799698 BD In-Stock Unstable CASR 54 42 O=S1(=O)CC[C@H](N[C@H]2CCCC[C@@H]2c2ccccc2)C1 ZINC000217799712 CE For-Sale Unstable GRIA4 15 43 C[C@H](O)c1cccc(NC(=O)N[C@H]2CCC[C@@H](C)C2)c1 ZINC000217799715 CG For-Sale Unstable EPHX2 38 48 O[C@H]1CCC[C@@H]1N1CCC[C@@H]2CCCC[C@H]21 ZINC000217799728 BF For-Sale Unstable SLC18A3 42 53 Cc1noc(C)c1CC(=O)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217799736 GH In-Stock Unstable HRH3 20 41 OCC[C@H](CCN1CCOCC1)c1ccccc1 ZINC000217799782 BD In-Stock Unstable CASR 54 42 C[C@H](O)c1ccc(NC(=O)N[C@@H]2CCC[C@@H](C)C2)cc1 ZINC000217799795 CG For-Sale Unstable EPHX2 49 43 O[C@@H]1CCC[C@H]1N1CCC[C@@H]2CCCC[C@H]21 ZINC000217799802 BF For-Sale Unstable SLC18A3 42 53 Cc1c(Br)cccc1NC(=O)c1cccc(Cl)c1F ZINC000217799811 EJ On-Demand Unstable EPHB3 45 39 Cc1c(Br)cccc1NC(=O)c1cccc(Cl)c1F ZINC000217799811 EJ On-Demand Unstable SMO 20 41 Cc1c(Br)cccc1NC(=O)c1cccc(Cl)c1F ZINC000217799811 EJ On-Demand Unstable G2YM83_BOTF4 68 35 Cc1c(Br)cccc1NC(=O)c1cccc(Cl)c1F ZINC000217799811 EJ On-Demand Unstable H9CNL0_SPOEX 0 45 CN(CC(=O)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1)S(C)(=O)=O ZINC000217799839 HD In-Stock Unstable HRH3 18 41 C[C@H](O)c1ccc(NC(=O)N[C@H]2CCC[C@@H](C)C2)cc1 ZINC000217799870 CG For-Sale Unstable EPHX2 49 43 CCC(=O)c1cc(C(=O)OC)c(O)cc1F ZINC000217799909 BD For-Sale Unstable CA7 17 50 CCC(=O)c1cc(C(=O)OC)c(O)cc1F ZINC000217799909 BD For-Sale Unstable CA14 15 50 C[C@@H](c1ccccc1F)N(C)[C@H](C)C(=O)c1ccccc1 ZINC000217799915 CI For-Sale Unstable CES2 20 40 CN(CC(=O)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1)S(C)(=O)=O ZINC000217799924 HD In-Stock Unstable HRH3 18 41 Cc1ccc(Br)c(C(=O)Nc2cccc(Br)c2C)c1 ZINC000217799933 GK On-Demand Unstable KCNK3 67 36 Cc1ccc(Br)c(C(=O)Nc2cccc(Br)c2C)c1 ZINC000217799933 GK On-Demand Unstable KCNK9 59 36 Cc1ccc(Br)c(C(=O)Nc2cccc(Br)c2C)c1 ZINC000217799933 GK On-Demand Unstable H9CNL0_SPOEX 0 42 C[C@@H](Cc1nnnn1Cc1ccccc1)C(=O)O ZINC000217799942 BC For-Sale Unstable MME 50 37 C[C@@H](Cc1nnnn1Cc1ccccc1)C(=O)O ZINC000217799942 BC For-Sale Unstable CPA1 51 33 C[C@@H](Cc1nnnn1Cc1ccccc1)C(=O)O ZINC000217799942 BC For-Sale Unstable CAPNS1 46 34 C[C@@H](Cc1nnnn1Cc1ccccc1)C(=O)O ZINC000217799942 BC For-Sale Unstable GHSR 19 41 C[C@@H](Cc1nnnn1Cc1ccccc1)C(=O)O ZINC000217799942 BC For-Sale Unstable CAPN2 51 32 C[C@@H](Cc1nnnn1Cc1ccccc1)C(=O)O ZINC000217799942 BC For-Sale Unstable ACE2 40 33 C[C@@H](Cc1nnnn1Cc1ccccc1)C(=O)O ZINC000217799942 BC For-Sale Unstable FPR1 51 40 C[C@@H](Cc1nnnn1Cc1ccccc1)C(=O)O ZINC000217799942 BC For-Sale Unstable DAGLA 35 41 Cc1cccc(CN2CCN(C(=O)CN3CCN(CC(=O)NCc4ccccc4)CC3)CC2)c1 ZINC000217799955 JD On-Demand Unstable HTR1A 18 43 Cc1cccc(CN2CCN(C(=O)CN3CCN(CC(=O)NCc4ccccc4)CC3)CC2)c1 ZINC000217799955 JD On-Demand Unstable DRD2 24 42 Cc1cccc(CN2CCN(C(=O)CN3CCN(CC(=O)NCc4ccccc4)CC3)CC2)c1 ZINC000217799955 JD On-Demand Unstable DRD4 58 48 Cc1cccc(CN2CCN(C(=O)CN3CCN(CC(=O)NCc4ccccc4)CC3)CC2)c1 ZINC000217799955 JD On-Demand Unstable ACHE 24 45 Cc1cccc(CN2CCN(C(=O)CN3CCN(CC(=O)NCc4ccccc4)CC3)CC2)c1 ZINC000217799955 JD On-Demand Unstable HRH2 28 41 Cc1cccc(CN2CCN(C(=O)CN3CCN(CC(=O)NCc4ccccc4)CC3)CC2)c1 ZINC000217799955 JD On-Demand Unstable AVPR1B 18 40 Cc1cccc(CN2CCN(C(=O)CN3CCN(CC(=O)NCc4ccccc4)CC3)CC2)c1 ZINC000217799955 JD On-Demand Unstable CHRM3 20 49 Cc1cccc(CN2CCN(C(=O)CN3CCN(CC(=O)NCc4ccccc4)CC3)CC2)c1 ZINC000217799955 JD On-Demand Unstable SIGMAR1 33 48 Cc1cccc(CN2CCN(C(=O)CN3CCN(CC(=O)NCc4ccccc4)CC3)CC2)c1 ZINC000217799955 JD On-Demand Unstable FAAH 27 47 Cc1cccc(CN2CCN(C(=O)CN3CCN(CC(=O)NCc4ccccc4)CC3)CC2)c1 ZINC000217799955 JD On-Demand Unstable NPFFR1 50 34 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1ccc2ccccc2c1 ZINC000217799973 FG For-Sale Unstable F2 17 42 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1ccc2ccccc2c1 ZINC000217799973 FG For-Sale Unstable HTR7 17 45 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1ccc2ccccc2c1 ZINC000217799973 FG For-Sale Unstable NPY1R 45 45 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1ccc2ccccc2c1 ZINC000217799973 FG For-Sale Unstable TRY2_BOVIN 42 35 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1ccc2ccccc2c1 ZINC000217799973 FG For-Sale Unstable NPY2R 23 45 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1ccc2ccccc2c1 ZINC000217799973 FG For-Sale Unstable ADAMTS5 35 53 COc1ccc(CN2C(=O)N[C@@H](CC(=O)N[C@H](CO)c3ccccc3)C2=O)cc1 ZINC000217799979 GD In-Stock Unstable SOAT1 0 46 COc1ccc(CN2C(=O)N[C@@H](CC(=O)N[C@H](CO)c3ccccc3)C2=O)cc1 ZINC000217799979 GD In-Stock Unstable GPR88 0 48 C[C@@H](Cc1cccs1)NC(=O)[C@@H]1C[C@@H](O)CN1 ZINC000217799984 CC For-Sale Unstable CTSC 44 37 COC1CCN(C2CCN(S(=O)(=O)c3ccccc3C(F)(F)F)CC2)CC1 ZINC000217799991 HF In-Stock Unstable CHRM2 27 41 COC1CCN(C2CCN(S(=O)(=O)c3ccccc3C(F)(F)F)CC2)CC1 ZINC000217799991 HF In-Stock Unstable CCR1 15 43 COC1CCN(C2CCN(S(=O)(=O)c3ccccc3C(F)(F)F)CC2)CC1 ZINC000217799991 HF In-Stock Unstable SFRP1 41 38 Cc1cc(O)ccc1NC(=O)N/C=C/c1ccccc1Cl ZINC000217800002 DI For-Sale Unstable LPL 48 35 C[C@H](Cc1nnnn1Cc1ccccc1)C(=O)O ZINC000217800022 BC For-Sale Unstable MME 50 37 C[C@H](Cc1nnnn1Cc1ccccc1)C(=O)O ZINC000217800022 BC For-Sale Unstable CPA1 51 33 C[C@H](Cc1nnnn1Cc1ccccc1)C(=O)O ZINC000217800022 BC For-Sale Unstable CAPNS1 46 34 C[C@H](Cc1nnnn1Cc1ccccc1)C(=O)O ZINC000217800022 BC For-Sale Unstable GHSR 19 41 C[C@H](Cc1nnnn1Cc1ccccc1)C(=O)O ZINC000217800022 BC For-Sale Unstable CAPN2 51 32 C[C@H](Cc1nnnn1Cc1ccccc1)C(=O)O ZINC000217800022 BC For-Sale Unstable ACE2 40 33 C[C@H](Cc1nnnn1Cc1ccccc1)C(=O)O ZINC000217800022 BC For-Sale Unstable FPR1 51 40 C[C@H](Cc1nnnn1Cc1ccccc1)C(=O)O ZINC000217800022 BC For-Sale Unstable DAGLA 35 41 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1ccc2ccccc2c1 ZINC000217800036 FG For-Sale Unstable F2 17 42 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1ccc2ccccc2c1 ZINC000217800036 FG For-Sale Unstable HTR7 17 45 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1ccc2ccccc2c1 ZINC000217800036 FG For-Sale Unstable NPY1R 45 45 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1ccc2ccccc2c1 ZINC000217800036 FG For-Sale Unstable TRY2_BOVIN 42 35 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1ccc2ccccc2c1 ZINC000217800036 FG For-Sale Unstable NPY2R 23 45 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1ccc2ccccc2c1 ZINC000217800036 FG For-Sale Unstable ADAMTS5 35 53 COc1ccc2cc(C(=O)N3CCC[C@H](Cc4nc(-c5ccccc5F)no4)C3)[nH]c2c1 ZINC000217800039 II In-Stock Unstable GRIN2B 26 45 COc1ccc2cc(C(=O)N3CCC[C@H](Cc4nc(-c5ccccc5F)no4)C3)[nH]c2c1 ZINC000217800039 II In-Stock Unstable HRH3 29 45 COc1ccc2cc(C(=O)N3CCC[C@H](Cc4nc(-c5ccccc5F)no4)C3)[nH]c2c1 ZINC000217800039 II In-Stock Unstable SYK 0 40 COc1ccc2cc(C(=O)N3CCC[C@H](Cc4nc(-c5ccccc5F)no4)C3)[nH]c2c1 ZINC000217800039 II In-Stock Unstable FPR2 28 43 COc1ccc2cc(C(=O)N3CCC[C@H](Cc4nc(-c5ccccc5F)no4)C3)[nH]c2c1 ZINC000217800039 II In-Stock Unstable AKR1C3 0 41 Cc1ccccc1-c1cc(C(=O)Nc2cccc(CO)c2)c2cnn(C(C)C)c2n1 ZINC000217800071 HJ On-Demand Unstable EZH2 15 41 Cc1ccccc1-c1cc(C(=O)Nc2cccc(CO)c2)c2cnn(C(C)C)c2n1 ZINC000217800071 HJ On-Demand Unstable KCNK3 58 37 Cc1ccccc1-c1cc(C(=O)Nc2cccc(CO)c2)c2cnn(C(C)C)c2n1 ZINC000217800071 HJ On-Demand Unstable KCNK9 57 37 COc1ccc2cc(C(=O)N3CCC[C@@H](Cc4nc(-c5ccccc5F)no4)C3)[nH]c2c1 ZINC000217800113 II In-Stock Unstable GRIN2B 26 45 COc1ccc2cc(C(=O)N3CCC[C@@H](Cc4nc(-c5ccccc5F)no4)C3)[nH]c2c1 ZINC000217800113 II In-Stock Unstable HRH3 29 45 COc1ccc2cc(C(=O)N3CCC[C@@H](Cc4nc(-c5ccccc5F)no4)C3)[nH]c2c1 ZINC000217800113 II In-Stock Unstable SYK 0 40 COc1ccc2cc(C(=O)N3CCC[C@@H](Cc4nc(-c5ccccc5F)no4)C3)[nH]c2c1 ZINC000217800113 II In-Stock Unstable FPR2 28 43 COc1ccc2cc(C(=O)N3CCC[C@@H](Cc4nc(-c5ccccc5F)no4)C3)[nH]c2c1 ZINC000217800113 II In-Stock Unstable AKR1C3 0 41 O=C(N/C=C/c1ccccc1Cl)N1CCOCC1 ZINC000217800121 CE For-Sale Unstable AKR1C3 31 47 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1ccc(Cl)cc1 ZINC000217800142 FF For-Sale Unstable ADAMTS5 34 50 COc1ccc2[nH]c(Br)nc(=O)c2c1 ZINC000217800176 CD For-Sale Unstable CYP1B1 35 41 COc1ccc2[nH]c(Br)nc(=O)c2c1 ZINC000217800176 CD For-Sale Unstable TUBB2B 59 47 COc1ccc2[nH]c(Br)nc(=O)c2c1 ZINC000217800176 CD For-Sale Unstable CYP1A2 24 41 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1ccc(Cl)cc1 ZINC000217800213 FF For-Sale Unstable ADAMTS5 34 50 O=C(c1ccc(OC(F)(F)F)cc1)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217800217 IJ In-Stock Unstable HRH3 30 44 Cc1cc(CN[C@H]2C[C@H](C)CC[C@H]2C(C)C)no1 ZINC000217800249 CH For-Sale Unstable TRPM8 15 41 Cc1ccc([C@H](CCO)CCN(C)C)cc1 ZINC000217800273 BE In-Stock Unstable UTS2 51 42 COc1ccc2c(=O)nc(Br)[nH]c2c1 ZINC000217800279 CD For-Sale Unstable CYP1B1 32 41 COc1ccc2c(=O)nc(Br)[nH]c2c1 ZINC000217800279 CD For-Sale Unstable TUBB2B 57 38 COc1ccc2c(=O)nc(Br)[nH]c2c1 ZINC000217800279 CD For-Sale Unstable CYP1A2 25 41 COc1ccc2c(=O)nc(Br)[nH]c2c1 ZINC000217800279 CD For-Sale Unstable CYP2C19 27 41 CC[C@@H](C)N(C)CCNC(=O)c1ccc(Br)c(Cl)c1 ZINC000217800292 EH On-Demand Unstable CA2 16 42 O=C(c1ccc(OC(F)(F)F)cc1)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217800307 IJ In-Stock Unstable HRH3 30 44 COc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)cc1 ZINC000217800318 FE For-Sale Unstable ADAMTS5 36 49 Cc1cc(CN[C@H]2C[C@@H](C)CC[C@H]2C(C)C)no1 ZINC000217800339 CH For-Sale Unstable TRPM8 15 41 Cc1ccc([C@@H](CCO)CCN(C)C)cc1 ZINC000217800351 BE In-Stock Unstable UTS2 51 42 CC[C@H](C)N(C)CCNC(=O)c1ccc(Br)c(Cl)c1 ZINC000217800394 EH On-Demand Unstable CA2 16 42 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)cc1 ZINC000217800395 FE For-Sale Unstable ADAMTS5 36 49 CCN(CCNC(=O)CCCCC(=O)O)C1CC1 ZINC000217800396 CD For-Sale Unstable DNM1 0 45 Cc1noc(C)c1C(=O)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217800434 GH In-Stock Unstable HRH3 23 42 C[C@H](C(=O)O)c1ccc(SCC(F)F)cc1 ZINC000217800448 BG For-Sale Unstable PTGS1 20 49 O[C@@H]1CCC[C@@H]1N1CCc2sccc2C1 ZINC000217800478 BE For-Sale Unstable VACHT_TETCF 0 40 O[C@@H]1CCC[C@@H]1N1CCc2sccc2C1 ZINC000217800478 BE For-Sale Unstable SLC18A3 36 44 O=S(=O)(Cc1ccc(Cl)cc1)NC[C@@H]1CCCN1c1nccs1 ZINC000217800512 FF For-Sale Unstable ADAMTS5 29 40 Cc1noc(C)c1C(=O)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217800522 GH In-Stock Unstable HRH3 23 42 C[C@@H](C(=O)O)c1ccc(SCC(F)F)cc1 ZINC000217800542 BG For-Sale Unstable PTGS1 20 49 O[C@@H]1CCC[C@H]1N1CCc2sccc2C1 ZINC000217800554 BE On-Demand Unstable VACHT_TETCF 0 40 O[C@@H]1CCC[C@H]1N1CCc2sccc2C1 ZINC000217800554 BE On-Demand Unstable SLC18A3 24 42 O=S(=O)(Cc1ccc(Cl)cc1)NC[C@H]1CCCN1c1nccs1 ZINC000217800596 FF For-Sale Unstable ADAMTS5 29 40 O=C(c1ccccc1SC(F)F)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217800632 IK In-Stock Unstable HRH3 21 45 O=C(O)CCCCCNC(=O)N/C=C/c1ccccc1Cl ZINC000217800638 DG For-Sale Unstable EPHX2 0 40 O=C(O)CCCCCNC(=O)N/C=C/c1ccccc1Cl ZINC000217800638 DG For-Sale Unstable HDA106 0 43 CCn1ncc2c(C(=O)N3CC=C(c4ccc(O)cc4)CC3)cc(-c3ccccc3)nc21 ZINC000217800680 HJ On-Demand Unstable MT-CO2 44 33 O=C(c1ccccc1SC(F)F)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217800707 IK In-Stock Unstable HRH3 21 45 CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(-c3cccc(C#N)c3)c(Oc3ccc(C(F)(F)F)cc3Cl)s2)cc1 ZINC000217800723 KK Annotated Unstable CSNK1D 37 41 CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(-c3cccc(C#N)c3)c(Oc3ccc(C(F)(F)F)cc3Cl)s2)cc1 ZINC000217800723 KK Annotated Unstable PTGDR2 21 41 CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(-c3cccc(C#N)c3)c(Oc3ccc(C(F)(F)F)cc3Cl)s2)cc1 ZINC000217800723 KK Annotated Unstable RORC 73 51 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1ccc(F)c(C(N)=O)c1 ZINC000217800726 CH For-Sale Unstable TRPM8 17 50 O=C(c1cc(-c2ccc(Cl)cc2)n[nH]1)N1CC=C(c2ccc(O)cc2)CC1 ZINC000217800793 GI On-Demand Unstable TACR3 26 51 O=C(c1cc(-c2ccc(Cl)cc2)n[nH]1)N1CC=C(c2ccc(O)cc2)CC1 ZINC000217800793 GI On-Demand Unstable ALPL 50 43 O=C(c1noc2c1CCCC2)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217800806 HH In-Stock Unstable HRH3 18 40 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1ccc(F)c(C(N)=O)c1 ZINC000217800811 CH For-Sale Unstable TRPM8 17 50 Nc1c(C(=O)O)[nH]c2cc(Br)ccc12 ZINC000217800816 CE For-Sale Unstable PRS 40 36 CNCC[C@@H](CCO)c1cccc(C)c1 ZINC000217800839 BE In-Stock Unstable SLC6A2 15 51 C[C@H](C(=O)O)c1cccc(SCC(F)F)c1 ZINC000217800849 BG For-Sale Unstable PTGS1 22 49 C[C@H](C(=O)O)c1cccc(SCC(F)F)c1 ZINC000217800849 BG For-Sale Unstable CXCL8 19 49 O=C(c1noc2c1CCCC2)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217800876 HH In-Stock Unstable HRH3 18 40 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1ccc(F)c(C(N)=O)c1 ZINC000217800895 CH For-Sale Unstable TRPM8 17 50 CNCC[C@H](CCO)c1cccc(C)c1 ZINC000217800914 BE In-Stock Unstable SLC6A2 15 51 C[C@@H](C(=O)O)c1cccc(SCC(F)F)c1 ZINC000217800937 BG For-Sale Unstable PTGS1 22 49 C[C@@H](C(=O)O)c1cccc(SCC(F)F)c1 ZINC000217800937 BG For-Sale Unstable CXCL8 19 49 CC[C@@H](CCO)NCCc1cccnc1 ZINC000217800941 BD For-Sale Unstable TBXAS1 42 39 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1ccc(F)c(C(N)=O)c1 ZINC000217800964 CH For-Sale Unstable TRPM8 17 50 O=C(c1ccc(C(F)(F)F)nc1)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217800991 II In-Stock Unstable HRH3 21 41 Cc1cccc([C@H](CCO)CCN(C)C)c1 ZINC000217801013 BE In-Stock Unstable UTS2 44 36 CC[C@H](CCO)NCCc1cccnc1 ZINC000217801022 BD For-Sale Unstable TBXAS1 42 39 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1Cl)C(=O)O ZINC000217801029 DG For-Sale Unstable ACE 15 42 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1Cl)C(=O)O ZINC000217801029 DG For-Sale Unstable FOLH1 25 44 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1Cl)C(=O)O ZINC000217801029 DG For-Sale Unstable MME 39 45 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1Cl)C(=O)O ZINC000217801029 DG For-Sale Unstable ANPEP 41 47 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1Cl)C(=O)O ZINC000217801029 DG For-Sale Unstable RNPEP 24 42 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1Cl)C(=O)O ZINC000217801029 DG For-Sale Unstable CAPNS1 51 34 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1Cl)C(=O)O ZINC000217801029 DG For-Sale Unstable CAPN1 58 42 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1Cl)C(=O)O ZINC000217801029 DG For-Sale Unstable CAPN2 65 34 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1Cl)C(=O)O ZINC000217801029 DG For-Sale Unstable FPR1 83 44 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1Cl)C(=O)O ZINC000217801029 DG For-Sale Unstable NPR 60 35 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1Cl)C(=O)O ZINC000217801029 DG For-Sale Unstable AMP1_PLAFQ 17 42 CC(F)(F)CCSc1cccc(C(=O)O)c1 ZINC000217801044 BH For-Sale Unstable AKR1C3 40 37 O=C(c1ccc(C(F)(F)F)nc1)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217801074 II In-Stock Unstable HRH3 21 41 Cc1cccc([C@@H](CCO)CCN(C)C)c1 ZINC000217801093 BE In-Stock Unstable UTS2 44 36 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1Cl)C(=O)O ZINC000217801111 DG For-Sale Unstable ACE 15 42 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1Cl)C(=O)O ZINC000217801111 DG For-Sale Unstable FOLH1 25 44 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1Cl)C(=O)O ZINC000217801111 DG For-Sale Unstable MME 39 45 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1Cl)C(=O)O ZINC000217801111 DG For-Sale Unstable ANPEP 41 47 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1Cl)C(=O)O ZINC000217801111 DG For-Sale Unstable RNPEP 24 42 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1Cl)C(=O)O ZINC000217801111 DG For-Sale Unstable CAPNS1 51 34 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1Cl)C(=O)O ZINC000217801111 DG For-Sale Unstable CAPN1 58 42 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1Cl)C(=O)O ZINC000217801111 DG For-Sale Unstable CAPN2 65 34 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1Cl)C(=O)O ZINC000217801111 DG For-Sale Unstable FPR1 83 44 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1Cl)C(=O)O ZINC000217801111 DG For-Sale Unstable NPR 60 35 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1Cl)C(=O)O ZINC000217801111 DG For-Sale Unstable AMP1_PLAFQ 17 42 O=C(O)Cn1cnc2cc(Br)ccc21 ZINC000217801122 CD For-Sale Unstable NR1I2 48 37 COc1cccc(CCNc2ncnc3c2CCCC3)c1 ZINC000217801149 CG On-Demand Unstable ACHE 17 42 COc1cccc(CCNc2ncnc3c2CCCC3)c1 ZINC000217801149 CG On-Demand Unstable BCHE 23 42 O=C(Cc1ccc(C(F)(F)F)cc1)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217801176 IJ In-Stock Unstable HRH3 23 45 Cc1cccc([C@@H](CCO)CCN2CCOCC2)c1 ZINC000217801184 CE In-Stock Unstable CASR 33 41 COc1ccc(CCN2C(=O)N[C@@H](CC(=O)NCc3ccccc3)C2=O)cc1OC ZINC000217801194 HD In-Stock Unstable PLG 45 31 COc1ccc(CCN2C(=O)N[C@@H](CC(=O)NCc3ccccc3)C2=O)cc1OC ZINC000217801194 HD In-Stock Unstable TSHR 49 35 COc1ccc(CCN2C(=O)N[C@@H](CC(=O)NCc3ccccc3)C2=O)cc1OC ZINC000217801194 HD In-Stock Unstable FKBP1A 21 41 COc1ccc(CCN2C(=O)N[C@@H](CC(=O)NCc3ccccc3)C2=O)cc1OC ZINC000217801194 HD In-Stock Unstable HCRTR1 24 46 COc1ccc(CCN2C(=O)N[C@@H](CC(=O)NCc3ccccc3)C2=O)cc1OC ZINC000217801194 HD In-Stock Unstable BCHE 17 41 COc1ccc(CCN2C(=O)N[C@@H](CC(=O)NCc3ccccc3)C2=O)cc1OC ZINC000217801194 HD In-Stock Unstable MTNR1B 15 43 COc1ccc(CCN2C(=O)N[C@@H](CC(=O)NCc3ccccc3)C2=O)cc1OC ZINC000217801194 HD In-Stock Unstable HCRTR2 26 43 COc1ccc(CCN2C(=O)N[C@@H](CC(=O)NCc3ccccc3)C2=O)cc1OC ZINC000217801194 HD In-Stock Unstable CACNA1G 47 35 COc1ccc(CCN2C(=O)N[C@@H](CC(=O)NCc3ccccc3)C2=O)cc1OC ZINC000217801194 HD In-Stock Unstable ABCG2 22 41 CSCC[C@@H](NC(=O)N/C=C/c1ccccc1Cl)C(=O)O ZINC000217801210 EF For-Sale Unstable FOLH1 22 42 CSCC[C@@H](NC(=O)N/C=C/c1ccccc1Cl)C(=O)O ZINC000217801210 EF For-Sale Unstable PAM 0 42 CSCC[C@@H](NC(=O)N/C=C/c1ccccc1Cl)C(=O)O ZINC000217801210 EF For-Sale Unstable FPR1 43 43 CSCC[C@@H](NC(=O)N/C=C/c1ccccc1Cl)C(=O)O ZINC000217801210 EF For-Sale Unstable SLC15A2 0 41 CSCC[C@@H](NC(=O)N/C=C/c1ccccc1Cl)C(=O)O ZINC000217801210 EF For-Sale Unstable FPRL2 0 41 CC[C@@H](C)c1ccc(O[C@@H](C)C(=O)OC)cc1 ZINC000217801250 BG For-Sale Unstable ACACA 51 38 CC[C@@H](C)c1ccc(O[C@@H](C)C(=O)OC)cc1 ZINC000217801250 BG For-Sale Unstable SCN2A 17 44 Cc1cccc([C@H](CCO)CCN2CCOCC2)c1 ZINC000217801257 CE In-Stock Unstable CASR 33 41 O=C(Cc1ccc(C(F)(F)F)cc1)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217801261 IJ In-Stock Unstable HRH3 23 45 C[C@H](C(=O)O)c1ccccc1SCC(F)F ZINC000217801264 BG For-Sale Unstable PTGS1 19 42 Cc1nc2cc(CNC(=O)CCC(F)(F)F)ccc2n1C ZINC000217801277 CF In-Stock Unstable NAMPT 41 36 CSCC[C@H](NC(=O)N/C=C/c1ccccc1Cl)C(=O)O ZINC000217801292 EF For-Sale Unstable FOLH1 22 42 CSCC[C@H](NC(=O)N/C=C/c1ccccc1Cl)C(=O)O ZINC000217801292 EF For-Sale Unstable PAM 0 42 CSCC[C@H](NC(=O)N/C=C/c1ccccc1Cl)C(=O)O ZINC000217801292 EF For-Sale Unstable FPR1 43 43 CSCC[C@H](NC(=O)N/C=C/c1ccccc1Cl)C(=O)O ZINC000217801292 EF For-Sale Unstable SLC15A2 0 41 CSCC[C@H](NC(=O)N/C=C/c1ccccc1Cl)C(=O)O ZINC000217801292 EF For-Sale Unstable FPRL2 0 41 CCOc1cc(F)cc(C#N)c1 ZINC000217801298 AE On-Demand Unstable GRM5 28 40 CC[C@H](C)c1ccc(O[C@@H](C)C(=O)OC)cc1 ZINC000217801329 BG For-Sale Unstable ACACA 51 38 CC[C@H](C)c1ccc(O[C@@H](C)C(=O)OC)cc1 ZINC000217801329 BG For-Sale Unstable SCN2A 17 44 O=C(O)Cn1c(Br)nc2ccccc21 ZINC000217801340 CD For-Sale Unstable AKR1B1 16 43 O=C(O)Cn1c(Br)nc2ccccc21 ZINC000217801340 CD For-Sale Unstable PLM2_PLAFA 15 46 O=C(O)Cn1c(Br)nc2ccccc21 ZINC000217801340 CD For-Sale Unstable PTGDR2 37 58 O=C(O)Cn1c(Br)nc2ccccc21 ZINC000217801340 CD For-Sale Unstable IMDH_CRYPV 37 44 C[C@@H](C(=O)O)c1ccccc1SCC(F)F ZINC000217801344 BG For-Sale Unstable PTGS1 19 42 C[C@@H]1CCC[C@@H](N(C)[C@H](C)Cc2ccc(O)cc2)C1 ZINC000217801350 CH For-Sale Unstable YARS 56 34 O=C(Cc1ccsc1)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217801378 GH In-Stock Unstable HRH3 20 40 COc1ccc([C@@H](C)NC(=O)N/C=C/c2ccccc2Cl)cc1OC ZINC000217801389 FI For-Sale Unstable KCNQ2 53 50 CCOc1ccccc1N1CCN(C[C@@H]2[C@H]3CNC[C@H]32)CC1 ZINC000217801408 DD In-Stock Unstable HTR1A 72 46 CCOc1ccccc1N1CCN(C[C@@H]2[C@H]3CNC[C@H]32)CC1 ZINC000217801408 DD In-Stock Unstable DRD2 66 45 CCOc1ccccc1N1CCN(C[C@@H]2[C@H]3CNC[C@H]32)CC1 ZINC000217801408 DD In-Stock Unstable DRD4 33 51 CCOc1ccccc1N1CCN(C[C@@H]2[C@H]3CNC[C@H]32)CC1 ZINC000217801408 DD In-Stock Unstable ADRA1D 58 42 CCOc1ccccc1N1CCN(C[C@@H]2[C@H]3CNC[C@H]32)CC1 ZINC000217801408 DD In-Stock Unstable HTR2A 29 44 CCOc1ccccc1N1CCN(C[C@@H]2[C@H]3CNC[C@H]32)CC1 ZINC000217801408 DD In-Stock Unstable ADRA1A 47 44 CCOc1ccccc1N1CCN(C[C@@H]2[C@H]3CNC[C@H]32)CC1 ZINC000217801408 DD In-Stock Unstable ADRA1B 36 42 CCOc1ccccc1N1CCN(C[C@@H]2[C@H]3CNC[C@H]32)CC1 ZINC000217801408 DD In-Stock Unstable DRD3 54 42 CCOc1ccccc1N1CCN(C[C@@H]2[C@H]3CNC[C@H]32)CC1 ZINC000217801408 DD In-Stock Unstable HTR7 50 43 CC[C@@H](C)c1ccc(O[C@H](C)C(=O)OC)cc1 ZINC000217801414 BG For-Sale Unstable ACACA 51 38 CC[C@@H](C)c1ccc(O[C@H](C)C(=O)OC)cc1 ZINC000217801414 BG For-Sale Unstable SCN2A 17 44 O=C(Cc1ccsc1)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217801462 GH In-Stock Unstable HRH3 20 40 COc1ccc([C@H](C)NC(=O)N/C=C/c2ccccc2Cl)cc1OC ZINC000217801470 FI For-Sale Unstable KCNQ2 53 50 O=c1[nH]c2cc(S(=O)(=O)NC[C@@H]3CCCN3c3nccs3)ccc2o1 ZINC000217801479 GD For-Sale Unstable ADAMTS5 30 40 CC[C@H](C)c1ccc(O[C@H](C)C(=O)OC)cc1 ZINC000217801486 BG For-Sale Unstable ACACA 51 38 CC[C@H](C)c1ccc(O[C@H](C)C(=O)OC)cc1 ZINC000217801486 BG For-Sale Unstable SCN2A 17 44 CC(=O)OC(C)(C)C(=O)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217801561 GF In-Stock Unstable HRH3 23 43 O=c1[nH]c2cc(S(=O)(=O)NC[C@H]3CCCN3c3nccs3)ccc2o1 ZINC000217801563 GD For-Sale Unstable ADAMTS5 30 40 O=C(Nc1cc(F)ccc1Cl)c1ccc(Br)c(Cl)c1 ZINC000217801576 FK On-Demand Anodyne PYGL 24 42 O=C(Nc1cc(F)ccc1Cl)c1ccc(Br)c(Cl)c1 ZINC000217801576 FK On-Demand Anodyne TAAR1 17 43 O=C(Nc1cc(F)ccc1Cl)c1ccc(Br)c(Cl)c1 ZINC000217801576 FK On-Demand Anodyne GPR35 24 40 COc1ccc([C@@H](C)NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217801581 EI For-Sale Unstable KCNQ2 51 47 COc1ccc([C@@H](C)NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217801581 EI For-Sale Unstable ACACA 48 41 COc1ccc([C@@H](C)NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217801581 EI For-Sale Unstable ACACB 16 41 CC(=O)OC(C)(C)C(=O)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217801657 GF In-Stock Unstable HRH3 23 43 COc1ccc([C@H](C)NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217801668 EI For-Sale Unstable KCNQ2 51 47 COc1ccc([C@H](C)NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217801668 EI For-Sale Unstable ACACA 48 41 COc1ccc([C@H](C)NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217801668 EI For-Sale Unstable ACACB 16 41 COc1ccccc1Oc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)cc1 ZINC000217801685 IH For-Sale Unstable ADAMTS5 34 44 COc1ccccc1Oc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)cc1 ZINC000217801761 IH For-Sale Unstable ADAMTS5 34 44 O=C(CCc1cccc(Cl)c1)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217801770 IJ In-Stock Unstable HRH3 22 44 CCCc1nc2ccccc2n1CCS(=O)(=O)CCC ZINC000217801827 CF For-Sale Unstable AGTR1 18 41 Cc1cc(S(=O)(=O)NCC(=O)N[C@@H](C)c2n[nH]c(=O)[nH]2)ccc1F ZINC000217801833 FB In-Stock Unstable LEF 70 42 O=C(CCc1cccc(Cl)c1)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217801847 IJ In-Stock Unstable HRH3 22 44 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1ccc(Oc2ccccc2Cl)cc1 ZINC000217801866 IJ For-Sale Unstable ADAMTS5 26 41 O=C1C[C@@H](c2ccc(C(=O)O)cc2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217801909 II In-Stock Unstable AKR1B1 0 43 O=C1C[C@@H](c2ccc(C(=O)O)cc2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217801909 II In-Stock Unstable CYP1A1 22 41 O=C1C[C@@H](c2ccc(C(=O)O)cc2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217801909 II In-Stock Unstable CYP1A2 17 40 Cc1cc(S(=O)(=O)NCC(=O)N[C@H](C)c2n[nH]c(=O)[nH]2)ccc1F ZINC000217801914 FB In-Stock Unstable LEF 70 42 COC(C)(C)C(=O)Nc1nc(CCl)cs1 ZINC000217801924 BE For-Sale Unstable PDE5A 0 40 O=C(c1ccc(F)c(F)c1F)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217801942 HI In-Stock Unstable HRH3 20 43 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1ccc(Oc2ccccc2Cl)cc1 ZINC000217801959 IJ For-Sale Unstable ADAMTS5 26 41 O=C1C[C@H](c2ccc(C(=O)O)cc2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217801976 II In-Stock Unstable AKR1B1 0 43 O=C1C[C@H](c2ccc(C(=O)O)cc2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217801976 II In-Stock Unstable CYP1A1 22 41 O=C1C[C@H](c2ccc(C(=O)O)cc2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217801976 II In-Stock Unstable CYP1A2 17 40 O=C1CC(c2ccc(OCC3CCCC3)cc2)CC(=O)O1 ZINC000217801985 CG In-Stock Unstable HPGD 22 46 O=C(c1ccc(F)c(F)c1F)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217802004 HI In-Stock Unstable HRH3 20 43 CN1CCC[C@@H]1CNc1ncnc2c1CCCC2 ZINC000217802054 BD On-Demand Unstable CHRNA10 52 38 Cc1ccccc1Oc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)cc1 ZINC000217802079 II For-Sale Unstable ADAMTS5 27 42 O=C(CCCCCNc1ncccn1)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217802080 GE In-Stock Unstable CHRNA4 30 51 COC(=O)c1cc(C)ccc1C(C)=O ZINC000217802085 AD For-Sale Unstable CA7 17 47 COC(=O)c1cc(C)ccc1C(C)=O ZINC000217802085 AD For-Sale Unstable CA14 15 47 COC(=O)c1cc(C)ccc1C(C)=O ZINC000217802085 AD For-Sale Unstable KCNK3 43 35 COC(=O)c1cc(C)ccc1C(C)=O ZINC000217802085 AD For-Sale Unstable KCNK9 43 35 O=C(Nc1ccccc1Cl)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217802130 HK In-Stock Unstable HRH3 22 46 O=C(Nc1ccccc1Cl)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217802130 HK In-Stock Unstable SMO 49 46 CN1CCC[C@H]1CNc1ncnc2c1CCCC2 ZINC000217802137 BD On-Demand Unstable CHRNA10 52 38 CCOC(=O)CCC(=O)c1ccc(O)c(OCC)c1 ZINC000217802147 CE For-Sale Unstable CA14 18 46 CCc1ccc([C@@H](C)NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217802155 EJ For-Sale Unstable KCNQ2 50 47 Cc1ccccc1Oc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)cc1 ZINC000217802157 II For-Sale Unstable ADAMTS5 27 42 COc1cc2c(c(OC)c1OC)-c1ccc(NCCCCCC(=O)NCc3nc4ccccc4[nH]3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217802177 KK In-Stock Unstable TUBA1A 16 59 O=C(Nc1ccccc1Cl)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217802204 HK In-Stock Unstable HRH3 22 46 O=C(Nc1ccccc1Cl)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217802204 HK In-Stock Unstable SMO 49 46 CCc1ccc([C@H](C)NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217802229 EJ For-Sale Unstable KCNQ2 50 47 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1c(Cl)cccc1Cl ZINC000217802264 GG For-Sale Unstable ADAMTS5 24 41 O=C1CC(c2ccc(OCC3CCCCC3)cc2)CC(=O)O1 ZINC000217802278 DH In-Stock Unstable HPGD 23 45 O=C(Nc1ccc(C(F)(F)F)cc1)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217802307 IK In-Stock Unstable HRH3 22 44 O=C(Nc1ccc(C(F)(F)F)cc1)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217802307 IK In-Stock Unstable EPHX2 43 47 O=C(Nc1ccc(C(F)(F)F)cc1)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217802307 IK In-Stock Unstable TRPM8 51 43 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1c(Cl)cccc1Cl ZINC000217802350 GG For-Sale Unstable ADAMTS5 31 41 C[C@@H](NC(=O)N/C=C/c1ccccc1Cl)c1ccc2c(c1)CCCC2 ZINC000217802354 FK For-Sale Unstable KCNQ2 52 52 O=C(Nc1ccc(C(F)(F)F)cc1)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217802380 IK In-Stock Unstable HRH3 22 44 O=C(Nc1ccc(C(F)(F)F)cc1)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217802380 IK In-Stock Unstable EPHX2 43 47 O=C(Nc1ccc(C(F)(F)F)cc1)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217802380 IK In-Stock Unstable TRPM8 51 43 C[C@@H](c1ccccc1Cl)N(C)[C@@]1(CN)CCN(C2CC2)C1 ZINC000217802395 DF For-Sale Unstable OPRM1 20 42 C[C@@H](c1ccccc1Cl)N(C)[C@@]1(CN)CCN(C2CC2)C1 ZINC000217802395 DF For-Sale Unstable OPRL1 55 42 C[C@H](NC(=O)N/C=C/c1ccccc1Cl)c1ccc2c(c1)CCCC2 ZINC000217802443 FK For-Sale Unstable KCNQ2 52 52 COc1ccc2ccccc2c1CN1C[C@@H]2CC[C@H](C1)[C@@H]2O ZINC000217802459 CG In-Stock Unstable XIAP 50 36 Cc1ccc(-c2ccc(S(=O)(=O)NC[C@@H]3CCCN3c3nccs3)cc2)cc1 ZINC000217802465 HI For-Sale Unstable ADAMTS5 36 46 C[C@H](c1ccccc1Cl)N(C)[C@@]1(CN)CCN(C2CC2)C1 ZINC000217802468 DF For-Sale Unstable OPRM1 20 42 C[C@H](c1ccccc1Cl)N(C)[C@@]1(CN)CCN(C2CC2)C1 ZINC000217802468 DF For-Sale Unstable OPRL1 55 42 Cc1ccccc1NC(=O)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217802483 GJ In-Stock Unstable HRH3 25 45 Cc1ccccc1NC(=O)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217802483 GJ In-Stock Unstable CCR3 24 40 Cc1ccccc1NC(=O)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217802483 GJ In-Stock Unstable Q8MHZ5_SHEEP 40 31 Cc1ccccc1NC(=O)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217802483 GJ In-Stock Unstable SMO 36 44 Cc1ccc(-c2ccc(S(=O)(=O)NC[C@H]3CCCN3c3nccs3)cc2)cc1 ZINC000217802549 HI For-Sale Unstable ADAMTS5 36 46 CCc1cccc(CC)c1NC(=O)N/C=C/c1ccccc1Cl ZINC000217802550 EK For-Sale Unstable CXCL8 42 37 CCc1cccc(CC)c1NC(=O)N/C=C/c1ccccc1Cl ZINC000217802550 EK For-Sale Unstable ACAT 0 41 Cc1ccccc1NC(=O)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217802559 GJ In-Stock Unstable HRH3 25 45 Cc1ccccc1NC(=O)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217802559 GJ In-Stock Unstable CCR3 24 40 Cc1ccccc1NC(=O)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217802559 GJ In-Stock Unstable Q8MHZ5_SHEEP 40 31 Cc1ccccc1NC(=O)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217802559 GJ In-Stock Unstable SMO 36 44 O=C(Cn1nnc(-c2ccccc2)n1)Nc1ccccc1Nc1ccccc1 ZINC000217802604 FH On-Demand Unstable SCARB1 31 40 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(Oc2ccccc2)cc1 ZINC000217802659 FK For-Sale Anodyne CA1 43 47 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(Oc2ccccc2)cc1 ZINC000217802659 FK For-Sale Anodyne RAF1 32 40 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(Oc2ccccc2)cc1 ZINC000217802659 FK For-Sale Anodyne NPY5R 0 43 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(Oc2ccccc2)cc1 ZINC000217802659 FK For-Sale Anodyne CA12 17 47 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(Oc2ccccc2)cc1 ZINC000217802659 FK For-Sale Anodyne CA9 18 47 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(Oc2ccccc2)cc1 ZINC000217802659 FK For-Sale Anodyne Q8MMZ8_EIMTE 47 41 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(Oc2ccccc2)cc1 ZINC000217802659 FK For-Sale Anodyne F13A1 15 40 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(Oc2ccccc2)cc1 ZINC000217802659 FK For-Sale Anodyne SMO 15 40 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1ccc(-c2ccc(Cl)cc2)cc1 ZINC000217802662 II For-Sale Unstable ADAMTS5 29 48 O=C(Cn1cnc2sc(-c3ccccc3)cc2c1=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217802673 JF In-Stock Unstable CHRNA4 26 42 O=C(NCc1ccc2c(c1)OCO2)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217802680 IH In-Stock Unstable HRH3 20 42 O=C(NCc1ccc2c(c1)OCO2)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217802680 IH In-Stock Unstable NOS2 101 41 O=C(NCc1ccc2c(c1)OCO2)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217802680 IH In-Stock Unstable SSTR3 106 35 CC(C)(C)[C@@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217802708 CD For-Sale Unstable CTSC 23 40 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1ccc(-c2ccc(Cl)cc2)cc1 ZINC000217802747 II For-Sale Unstable ADAMTS5 29 48 O=C(NCc1ccc2c(c1)OCO2)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217802751 IH In-Stock Unstable HRH3 20 42 O=C(NCc1ccc2c(c1)OCO2)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217802751 IH In-Stock Unstable NOS2 101 41 O=C(NCc1ccc2c(c1)OCO2)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217802751 IH In-Stock Unstable SSTR3 106 35 CC1(CNC(=O)Cc2ccc(O)c(Cl)c2)COC1 ZINC000217802780 CD In-Stock Unstable NCE103 38 55 CC1(CNC(=O)Cc2ccc(O)c(Cl)c2)COC1 ZINC000217802780 CD In-Stock Unstable P96878_MYCTU 24 53 CC1(CNC(=O)Cc2ccc(O)c(Cl)c2)COC1 ZINC000217802780 CD In-Stock Unstable CAN2 0 55 CC(C)(C)[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217802789 CD For-Sale Unstable CTSC 23 40 O=C(Nc1ccccc1Nc1ccccc1)C1CCN(c2nc3ccccc3o2)CC1 ZINC000217802820 HK On-Demand Unstable PTGES 37 43 O=S(=O)(NC1[C@@H]2CNC[C@@H]12)N1CCc2ccccc2C1 ZINC000217802847 CC For-Sale Unstable AKR1C3 57 43 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1ccc(-c2ccc(F)cc2)cc1 ZINC000217802865 HH For-Sale Unstable ADAMTS5 27 43 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1ccc(-c2ccc(F)cc2)cc1 ZINC000217802865 HH For-Sale Unstable PIK3C3 46 33 CC(C)(C)[C@@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217802868 CD For-Sale Unstable CTSC 23 40 COc1ccc(OC)c(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217802876 EI For-Sale Unstable CYP1B1 42 40 COc1ccc(OC)c(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217802876 EI For-Sale Unstable MTNR1A 21 48 COc1ccc(OC)c(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217802876 EI For-Sale Unstable MTNR1B 23 48 COc1ccc(OC)c(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217802876 EI For-Sale Unstable AKR1C2 46 35 COc1ccc(OC)c(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217802876 EI For-Sale Unstable CYSP_PLAFA 53 45 CS(=O)(=O)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217802878 EE In-Stock Unstable HRH3 16 40 CCCn1c(CNCCOCC2CC2)nc2ccccc21 ZINC000217802890 CF On-Demand Unstable HRH1 17 41 C[C@@H](NS(=O)(=O)c1ccc(Br)c(F)c1)C(=O)OC(C)(C)C ZINC000217802910 GF On-Demand Unstable CA2 22 40 C[C@@H](NS(=O)(=O)c1ccc(Br)c(F)c1)C(=O)OC(C)(C)C ZINC000217802910 GF On-Demand Unstable CA1 18 40 C[C@@H](NS(=O)(=O)c1ccc(Br)c(F)c1)C(=O)OC(C)(C)C ZINC000217802910 GF On-Demand Unstable MMP13 17 40 C[C@@H](NS(=O)(=O)c1ccc(Br)c(F)c1)C(=O)OC(C)(C)C ZINC000217802910 GF On-Demand Unstable CA4 20 40 C[C@@H](NS(=O)(=O)c1ccc(Br)c(F)c1)C(=O)OC(C)(C)C ZINC000217802910 GF On-Demand Unstable CA14 20 40 C[C@@H](NS(=O)(=O)c1ccc(Br)c(F)c1)C(=O)OC(C)(C)C ZINC000217802910 GF On-Demand Unstable LEF 66 41 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1ccc(-c2ccc(F)cc2)cc1 ZINC000217802942 HH For-Sale Unstable ADAMTS5 34 48 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1ccc(-c2ccc(F)cc2)cc1 ZINC000217802942 HH For-Sale Unstable PIK3C3 46 33 CC(C)(C)[C@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217802948 CD For-Sale Unstable CTSC 23 40 CS(=O)(=O)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217802967 EE In-Stock Unstable HRH3 16 40 COc1ccc(CNC(=O)CCCCCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@H]23)cc1 ZINC000217802977 JJ In-Stock Unstable HTR7 35 46 COc1ccc(CNC(=O)CCCCCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@H]23)cc1 ZINC000217802977 JJ In-Stock Unstable SCN9A 0 50 CC[C@@H](C)c1ccc(OCCCc2ccccc2)cc1 ZINC000217803046 CK For-Sale Unstable ALOX5 24 52 CC[C@@H](C)c1ccc(OCCCc2ccccc2)cc1 ZINC000217803046 CK For-Sale Unstable PPARG 17 41 CC[C@@H](C)c1ccc(OCCCc2ccccc2)cc1 ZINC000217803046 CK For-Sale Unstable LTA4H 44 44 CC[C@@H](C)c1ccc(OCCCc2ccccc2)cc1 ZINC000217803046 CK For-Sale Unstable SIGMAR1 25 50 CC[C@@H](C)c1ccc(OCCCc2ccccc2)cc1 ZINC000217803046 CK For-Sale Unstable SCN2A 30 40 CC[C@@H](C)c1ccc(OCCCc2ccccc2)cc1 ZINC000217803046 CK For-Sale Unstable PLA2G4B 57 42 CC[C@@H](C)c1ccc(OCCCc2ccccc2)cc1 ZINC000217803046 CK For-Sale Unstable TAAR1 30 55 CC[C@@H](C)c1ccc(OCCCc2ccccc2)cc1 ZINC000217803046 CK For-Sale Unstable FFAR1 20 43 COc1ccc(CNC(=O)CCCCCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@@H]23)cc1 ZINC000217803057 JJ In-Stock Unstable HTR7 35 46 COc1ccc(CNC(=O)CCCCCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@@H]23)cc1 ZINC000217803057 JJ In-Stock Unstable SCN9A 0 50 CCOC(=O)c1ccc(NCCCCN)cc1 ZINC000217803062 BE For-Sale Unstable ACR 53 40 COc1ccc(-c2ccc(S(=O)(=O)NC[C@@H]3CCCN3c3nccs3)cc2)cc1 ZINC000217803072 IH For-Sale Unstable MMP13 26 41 COc1ccc(-c2ccc(S(=O)(=O)NC[C@@H]3CCCN3c3nccs3)cc2)cc1 ZINC000217803072 IH For-Sale Unstable ADAMTS5 36 51 CC[C@H](C)c1ccc(OCCCc2ccccc2)cc1 ZINC000217803137 CK For-Sale Unstable ALOX5 24 52 CC[C@H](C)c1ccc(OCCCc2ccccc2)cc1 ZINC000217803137 CK For-Sale Unstable PPARG 17 41 CC[C@H](C)c1ccc(OCCCc2ccccc2)cc1 ZINC000217803137 CK For-Sale Unstable LTA4H 44 44 CC[C@H](C)c1ccc(OCCCc2ccccc2)cc1 ZINC000217803137 CK For-Sale Unstable SIGMAR1 25 50 CC[C@H](C)c1ccc(OCCCc2ccccc2)cc1 ZINC000217803137 CK For-Sale Unstable SCN2A 30 40 CC[C@H](C)c1ccc(OCCCc2ccccc2)cc1 ZINC000217803137 CK For-Sale Unstable PLA2G4B 57 42 CC[C@H](C)c1ccc(OCCCc2ccccc2)cc1 ZINC000217803137 CK For-Sale Unstable TAAR1 30 55 CC[C@H](C)c1ccc(OCCCc2ccccc2)cc1 ZINC000217803137 CK For-Sale Unstable FFAR1 20 43 COc1ccc(-c2ccc(S(=O)(=O)NC[C@H]3CCCN3c3nccs3)cc2)cc1 ZINC000217803154 IH For-Sale Unstable MMP13 26 41 COc1ccc(-c2ccc(S(=O)(=O)NC[C@H]3CCCN3c3nccs3)cc2)cc1 ZINC000217803154 IH For-Sale Unstable ADAMTS5 36 51 CCCCC[C@H](C#CC(F)(F)F)OC(C)=O ZINC000217803165 BG For-Sale Unstable CES2 47 33 CCCCC[C@H](C#CC(F)(F)F)OC(C)=O ZINC000217803165 BG For-Sale Unstable EST1_PIG 69 33 CCCCC[C@H](C#CC(F)(F)F)OC(C)=O ZINC000217803165 BG For-Sale Unstable CES2C 55 33 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1ccc(-c2ccc(Cl)c(Cl)c2)cc1 ZINC000217803273 JK For-Sale Unstable ADAMTS5 33 43 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(F)cc1 ZINC000217803293 CI For-Sale Anodyne SMO 16 40 O=C(O)[C@@H]1[C@H]2CN(C(=O)c3nc4ccccc4[nH]3)C[C@H]21 ZINC000217803299 CC In-Stock Unstable GRIN2B 28 47 COc1ccc([C@@H](CC(=O)Nc2ccccc2Nc2ccccc2)NC(C)=O)cc1 ZINC000217803336 HJ On-Demand Unstable AKR1C3 27 41 COc1ccc([C@@H](CC(=O)Nc2ccccc2Nc2ccccc2)NC(C)=O)cc1 ZINC000217803336 HJ On-Demand Unstable AKR1C2 71 46 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1ccc(-c2ccc(Cl)c(Cl)c2)cc1 ZINC000217803344 JK For-Sale Unstable ADAMTS5 33 43 CC(C)(F)CCS(=O)(=O)c1cccc(O)c1 ZINC000217803367 BE For-Sale Unstable HSD17B1 15 42 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217803396 FJ For-Sale Bother IMDH_CRYPV 33 48 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217803396 FJ For-Sale Bother BLM 0 49 COc1ccc([C@H](CC(=O)Nc2ccccc2Nc2ccccc2)NC(C)=O)cc1 ZINC000217803409 HJ On-Demand Unstable AKR1C3 27 41 COc1ccc([C@H](CC(=O)Nc2ccccc2Nc2ccccc2)NC(C)=O)cc1 ZINC000217803409 HJ On-Demand Unstable AKR1C2 71 46 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1ccc(-c2cccc(Cl)c2)cc1 ZINC000217803460 II For-Sale Unstable ADAMTS5 26 45 CC(=O)N[C@@H](CC(=O)Nc1ccccc1Nc1ccccc1)c1ccc(Cl)cc1 ZINC000217803506 HK On-Demand Unstable AKR1C2 30 42 CC(=O)N[C@@H](CC(=O)Nc1ccccc1Nc1ccccc1)c1ccc(Cl)cc1 ZINC000217803506 HK On-Demand Unstable UTS2 45 37 COc1cc([N+](=O)[O-])ccc1NC(=O)N/C=C/c1ccccc1Cl ZINC000217803512 EI For-Sale Unstable EPHX1 0 54 COc1cc([N+](=O)[O-])ccc1NC(=O)N/C=C/c1ccccc1Cl ZINC000217803512 EI For-Sale Unstable PYGL 16 43 COc1cc([N+](=O)[O-])ccc1NC(=O)N/C=C/c1ccccc1Cl ZINC000217803512 EI For-Sale Unstable KCNMA1 25 54 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1ccc(-c2cccc(Cl)c2)cc1 ZINC000217803533 II For-Sale Unstable ADAMTS5 26 45 C/C=C\c1ccccc1OC[C@](C)(O)C(=O)O ZINC000217803540 BD For-Sale Unstable PTGER2 0 42 CSCC[C@H](NC(=O)c1cccc2c1ccn2C)C(=O)O ZINC000217803545 DE In-Stock Unstable CCKAR 0 56 CCOC[C@@H](C)NC(=O)/C=C\C(=O)O ZINC000217803549 BC For-Sale Unstable HCAR2 31 40 CC(=O)N[C@H](CC(=O)Nc1ccccc1Nc1ccccc1)c1ccc(Cl)cc1 ZINC000217803588 HK On-Demand Unstable AKR1C2 30 42 CC(=O)N[C@H](CC(=O)Nc1ccccc1Nc1ccccc1)c1ccc(Cl)cc1 ZINC000217803588 HK On-Demand Unstable UTS2 45 37 O=C(N/C=C/c1ccccc1Cl)Nc1ccc([N+](=O)[O-])cc1 ZINC000217803601 DI For-Sale Bother NADE 0 49 O=C(N/C=C/c1ccccc1Cl)Nc1ccc([N+](=O)[O-])cc1 ZINC000217803601 DI For-Sale Bother NMBR 47 32 C/C=C\c1ccccc1OC[C@@](C)(O)C(=O)O ZINC000217803613 BD For-Sale Unstable PTGER2 0 42 CCOC[C@H](C)NC(=O)/C=C\C(=O)O ZINC000217803629 BC For-Sale Unstable HCAR2 31 40 CC(=O)c1cccc(S(=O)(=O)N2CCC[C@H](Cc3nc(-c4ccccc4F)no3)C2)c1 ZINC000217803646 IH In-Stock Unstable HRH3 18 40 CC(=O)c1cccc(S(=O)(=O)N2CCC[C@H](Cc3nc(-c4ccccc4F)no3)C2)c1 ZINC000217803646 IH In-Stock Unstable AKR1C3 44 36 Cc1cccc(OCCCc2ccccc2)c1C ZINC000217803670 BI For-Sale Unstable SIGMAR1 24 44 Cc1cccc(OCCCc2ccccc2)c1C ZINC000217803670 BI For-Sale Unstable MCL1 40 38 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1ccc(-c2cc(Cl)cc(Cl)c2)cc1 ZINC000217803676 JK For-Sale Unstable ADAMTS5 33 43 O=C(N/C=C/c1ccccc1Cl)Nc1cccc([N+](=O)[O-])c1 ZINC000217803678 DI For-Sale Bother PPIA 17 42 O=C(N/C=C/c1ccccc1Cl)Nc1cccc([N+](=O)[O-])c1 ZINC000217803678 DI For-Sale Bother DDX3X 0 52 O=C(N/C=C/c1ccccc1Cl)Nc1cccc([N+](=O)[O-])c1 ZINC000217803678 DI For-Sale Bother TRPM8 0 48 O=C(N/C=C/c1ccccc1Cl)Nc1cccc([N+](=O)[O-])c1 ZINC000217803678 DI For-Sale Bother OSIGBA0132E09-OSIGBA0108L24.11 0 42 NC1(C2(NC(=O)OCc3ccccc3)CC2)CC1 ZINC000217803684 BD For-Sale Unstable ACE 18 43 NC1(C2(NC(=O)OCc3ccccc3)CC2)CC1 ZINC000217803684 BD For-Sale Unstable MME 22 40 NC1(C2(NC(=O)OCc3ccccc3)CC2)CC1 ZINC000217803684 BD For-Sale Unstable BMP1 54 34 NC1(C2(NC(=O)OCc3ccccc3)CC2)CC1 ZINC000217803684 BD For-Sale Unstable KLK3 59 36 NC1(C2(NC(=O)OCc3ccccc3)CC2)CC1 ZINC000217803684 BD For-Sale Unstable CTSB 46 40 NC1(C2(NC(=O)OCc3ccccc3)CC2)CC1 ZINC000217803684 BD For-Sale Unstable PAPA1_CARPA 57 39 NC1(C2(NC(=O)OCc3ccccc3)CC2)CC1 ZINC000217803684 BD For-Sale Unstable CYSP_TRYCR 57 41 NC1(C2(NC(=O)OCc3ccccc3)CC2)CC1 ZINC000217803684 BD For-Sale Unstable CTSK 28 52 NC1(C2(NC(=O)OCc3ccccc3)CC2)CC1 ZINC000217803684 BD For-Sale Unstable CTSL 35 41 NC1(C2(NC(=O)OCc3ccccc3)CC2)CC1 ZINC000217803684 BD For-Sale Unstable CAPNS1 62 39 NC1(C2(NC(=O)OCc3ccccc3)CC2)CC1 ZINC000217803684 BD For-Sale Unstable ECE1 18 42 NC1(C2(NC(=O)OCc3ccccc3)CC2)CC1 ZINC000217803684 BD For-Sale Unstable CTSS 18 44 NC1(C2(NC(=O)OCc3ccccc3)CC2)CC1 ZINC000217803684 BD For-Sale Unstable CAPN1 64 40 NC1(C2(NC(=O)OCc3ccccc3)CC2)CC1 ZINC000217803684 BD For-Sale Unstable CASP1 23 40 NC1(C2(NC(=O)OCc3ccccc3)CC2)CC1 ZINC000217803684 BD For-Sale Unstable CAPN2 95 39 NC1(C2(NC(=O)OCc3ccccc3)CC2)CC1 ZINC000217803684 BD For-Sale Unstable NPR 65 37 NC1(C2(NC(=O)OCc3ccccc3)CC2)CC1 ZINC000217803684 BD For-Sale Unstable KDM1A 17 43 NC1(C2(NC(=O)OCc3ccccc3)CC2)CC1 ZINC000217803684 BD For-Sale Unstable SLC12A5 71 40 Cn1c(=O)n(CCC(=O)Nc2ccccc2Nc2ccccc2)c2ccccc21 ZINC000217803692 GI On-Demand Unstable CMA1 17 40 CC(=O)c1cccc(S(=O)(=O)N2CCC[C@@H](Cc3nc(-c4ccccc4F)no3)C2)c1 ZINC000217803728 IH In-Stock Unstable HRH3 18 40 CC(=O)c1cccc(S(=O)(=O)N2CCC[C@@H](Cc3nc(-c4ccccc4F)no3)C2)c1 ZINC000217803728 IH In-Stock Unstable AKR1C3 44 36 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1ccc(-c2cc(Cl)cc(Cl)c2)cc1 ZINC000217803737 JK For-Sale Unstable ADAMTS5 33 43 O=C(CCc1ncc(-c2ccccc2)o1)Nc1ccccc1Nc1ccccc1 ZINC000217803784 GK On-Demand Unstable FAAH 43 41 O=C(CCc1ncc(-c2ccccc2)o1)Nc1ccccc1Nc1ccccc1 ZINC000217803784 GK On-Demand Unstable CES1 27 41 O=C(CCc1ncc(-c2ccccc2)o1)Nc1ccccc1Nc1ccccc1 ZINC000217803784 GK On-Demand Unstable HCAR2 36 40 COC(=O)C[C@H](c1ccc(OC)c(OC)c1)c1c(O)cc(C)n(CCc2ccc(O)cc2)c1=O ZINC000217803788 JH In-Stock Unstable TNF 21 40 Cc1nnc(CCNC(=O)CCc2nc3ccccc3[nH]2)s1 ZINC000217803810 DE In-Stock Unstable CYSP_TRYCR 0 57 Cc1nnc(CCNC(=O)CCc2nc3ccccc3[nH]2)s1 ZINC000217803810 DE In-Stock Unstable FABK 0 41 Cc1nnc(CCNC(=O)CCc2nc3ccccc3[nH]2)s1 ZINC000217803810 DE In-Stock Unstable ISPE 0 42 COC(=O)C[C@@H](c1ccc(OC)c(OC)c1)c1c(O)cc(C)n(CCc2ccc(O)cc2)c1=O ZINC000217803853 JH In-Stock Unstable TNF 21 40 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217803869 JJ For-Sale Unstable ADAMTS5 35 49 CC[C@@H](CCO)NCCc1cccs1 ZINC000217803895 BE For-Sale Unstable ADAM17 0 43 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1ccc(-c2cccc(C(F)(F)F)c2)cc1 ZINC000217803925 JJ For-Sale Unstable ADAMTS5 35 49 COc1ccc(-c2noc(CCC(=O)Nc3ccccc3Nc3ccccc3)n2)cc1 ZINC000217803963 HK On-Demand Unstable HCAR2 43 61 COc1ccc(-c2noc(CCC(=O)Nc3ccccc3Nc3ccccc3)n2)cc1 ZINC000217803963 HK On-Demand Unstable AKR1C3 19 42 COc1ccc(-c2noc(CCC(=O)Nc3ccccc3Nc3ccccc3)n2)cc1 ZINC000217803963 HK On-Demand Unstable AKR1C2 57 42 CC[C@H](CCO)NCCc1cccs1 ZINC000217803986 BE For-Sale Unstable ADAM17 0 43 Cc1cccc(-c2ccc(S(=O)(=O)NC[C@@H]3CCCN3c3nccs3)cc2)c1 ZINC000217804032 HI For-Sale Unstable ADAMTS5 35 46 O=S(=O)(C1CC1)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217804041 FF In-Stock Unstable HRH3 18 42 CC(C)[C@H](NC(=O)CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)c1nc2ccccc2n1C ZINC000217804044 IG In-Stock Unstable AGAL_COFAR 0 44 CC(C)[C@H](NC(=O)CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)c1nc2ccccc2n1C ZINC000217804044 IG In-Stock Unstable HLCS 0 41 CC(C)[C@H](NC(=O)CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)c1nc2ccccc2n1C ZINC000217804044 IG In-Stock Unstable BIRA 0 43 O=C(N/C=C/c1ccccc1Cl)N1CCN(c2ccc(F)cc2)CC1 ZINC000217804048 FH For-Sale Unstable AKR1C3 0 43 O=C(Nc1ccccc1Nc1ccccc1)c1cccc(N2CCCS2(=O)=O)c1 ZINC000217804063 HI On-Demand Unstable CDK1 20 42 O=C(Nc1ccccc1Nc1ccccc1)c1cccc(N2CCCS2(=O)=O)c1 ZINC000217804063 HI On-Demand Unstable CDK4 22 42 O=C(Nc1ccccc1Nc1ccccc1)c1cccc(N2CCCS2(=O)=O)c1 ZINC000217804063 HI On-Demand Unstable KCNK3 85 38 O=C(Nc1ccccc1Nc1ccccc1)c1cccc(N2CCCS2(=O)=O)c1 ZINC000217804063 HI On-Demand Unstable KCNK9 41 36 Cc1cccc(-c2ccc(S(=O)(=O)NC[C@H]3CCCN3c3nccs3)cc2)c1 ZINC000217804118 HI For-Sale Unstable ADAMTS5 35 46 O=S(=O)(C1CC1)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217804136 FF In-Stock Unstable HRH3 18 42 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)Nc3ccc4[nH]cnc4c3)[C@H]21 ZINC000217804160 JG In-Stock Unstable TSHR 50 34 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)Nc3ccc4[nH]cnc4c3)[C@H]21 ZINC000217804160 JG In-Stock Unstable ENPP1 55 33 O=C(Nc1ccccc1Nc1ccccc1)c1ccc(S(=O)(=O)NC2CC2)cc1 ZINC000217804175 HI On-Demand Unstable APOB 0 40 O=C(Nc1ccccc1Nc1ccccc1)c1ccc(S(=O)(=O)NC2CC2)cc1 ZINC000217804175 HI On-Demand Unstable HDAC1 18 40 O=C(Nc1ccccc1Nc1ccccc1)c1ccc(S(=O)(=O)NC2CC2)cc1 ZINC000217804175 HI On-Demand Unstable MTTP 17 40 O=C(Nc1ccccc1Nc1ccccc1)c1ccc(S(=O)(=O)NC2CC2)cc1 ZINC000217804175 HI On-Demand Unstable PTGDR 17 40 O=C(Nc1ccccc1Nc1ccccc1)c1ccc(S(=O)(=O)NC2CC2)cc1 ZINC000217804175 HI On-Demand Unstable CCR8 91 49 O=C(Nc1ccccc1Nc1ccccc1)c1ccc(S(=O)(=O)NC2CC2)cc1 ZINC000217804175 HI On-Demand Unstable SFRP1 98 36 O=C(Nc1ccccc1Nc1ccccc1)c1ccc(S(=O)(=O)NC2CC2)cc1 ZINC000217804175 HI On-Demand Unstable WNT3 59 33 O=C(Nc1ccccc1Nc1ccccc1)c1ccc(S(=O)(=O)NC2CC2)cc1 ZINC000217804175 HI On-Demand Unstable KCNK3 44 35 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1ccc(Cl)c(C(F)(F)F)c1 ZINC000217804235 IH For-Sale Unstable ADAMTS5 32 45 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1ccc(Cl)c(C(F)(F)F)c1 ZINC000217804235 IH For-Sale Unstable SFRP1 106 33 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1ccc(Cl)c(C(F)(F)F)c1 ZINC000217804235 IH For-Sale Unstable WNT3 67 31 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)Nc3ccc4[nH]cnc4c3)[C@@H]21 ZINC000217804244 JG In-Stock Unstable TSHR 50 34 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)Nc3ccc4[nH]cnc4c3)[C@@H]21 ZINC000217804244 JG In-Stock Unstable ENPP1 55 33 C[C@H](Cc1ccc(O)cc1)N1CCO[C@@H]2CCC[C@@H]21 ZINC000217804253 CF For-Sale Unstable YARS 46 32 Nc1ccc(F)cc1C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217804262 CD For-Sale Unstable VACHT_TETCF 0 41 C[C@@H](c1cccc(Cl)c1)N(C)[C@@]1(CN)CCN(C2CC2)C1 ZINC000217804268 DF For-Sale Unstable OPRL1 15 40 CC(C)NS(=O)(=O)c1cccc(C(=O)Nc2ccccc2Nc2ccccc2)c1 ZINC000217804276 HI On-Demand Unstable MMP13 20 42 CC(C)NS(=O)(=O)c1cccc(C(=O)Nc2ccccc2Nc2ccccc2)c1 ZINC000217804276 HI On-Demand Unstable CPT1A 0 41 CC(C)NS(=O)(=O)c1cccc(C(=O)Nc2ccccc2Nc2ccccc2)c1 ZINC000217804276 HI On-Demand Unstable PPARD 30 41 CC(C)NS(=O)(=O)c1cccc(C(=O)Nc2ccccc2Nc2ccccc2)c1 ZINC000217804276 HI On-Demand Unstable AKR1C3 65 44 CC(C)NS(=O)(=O)c1cccc(C(=O)Nc2ccccc2Nc2ccccc2)c1 ZINC000217804276 HI On-Demand Unstable KCNK3 109 41 CC(C)NS(=O)(=O)c1cccc(C(=O)Nc2ccccc2Nc2ccccc2)c1 ZINC000217804276 HI On-Demand Unstable KCNK9 66 41 COc1cccc(-n2cc(CNC(=O)c3ccccc3C#N)cn2)c1 ZINC000217804279 EF In-Stock Unstable DRD4 44 34 COc1cccc(-n2cc(CNC(=O)c3ccccc3C#N)cn2)c1 ZINC000217804279 EF In-Stock Unstable ROCK1 27 44 CCOc1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217804285 DJ For-Sale Unstable CA1 45 40 CCOc1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217804285 DJ For-Sale Unstable PRNP 18 44 CCOc1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217804285 DJ For-Sale Unstable CA12 18 40 CCOc1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217804285 DJ For-Sale Unstable CA9 19 40 O[C@@H]1CCC[C@@H]1N[C@@H]1CCCc2ccccc21 ZINC000217804288 BF On-Demand Unstable KCNN3 22 43 O[C@@H]1CCC[C@@H]1N[C@@H]1CCCc2ccccc21 ZINC000217804288 BF On-Demand Unstable TSPAN17 0 42 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1ccc(Cl)c(C(F)(F)F)c1 ZINC000217804321 IH For-Sale Unstable ADAMTS5 32 45 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1ccc(Cl)c(C(F)(F)F)c1 ZINC000217804321 IH For-Sale Unstable SFRP1 106 33 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1ccc(Cl)c(C(F)(F)F)c1 ZINC000217804321 IH For-Sale Unstable WNT3 67 31 CCOC(=O)c1nnn(Cc2cccc(F)c2)c1C ZINC000217804330 CD On-Demand Unstable ELANE 0 47 C[C@H](c1cccc(Cl)c1)N(C)[C@@]1(CN)CCN(C2CC2)C1 ZINC000217804343 DF For-Sale Unstable OPRL1 15 40 Nc1ccc(F)cc1C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217804356 CD For-Sale Unstable SIGMAR1 0 42 O[C@@H]1CCC[C@H]1N[C@@H]1CCCc2ccccc21 ZINC000217804365 BF On-Demand Unstable KCNN3 22 43 O[C@@H]1CCC[C@H]1N[C@@H]1CCCc2ccccc21 ZINC000217804365 BF On-Demand Unstable TSPAN17 0 42 COc1ccc([C@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1OC ZINC000217804377 KH In-Stock Unstable PRKDC 16 41 COc1ccc([C@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1OC ZINC000217804377 KH In-Stock Unstable CYP1B1 60 39 COc1ccc([C@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1OC ZINC000217804377 KH In-Stock Unstable CYP1A1 45 39 COc1ccc([C@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1OC ZINC000217804377 KH In-Stock Unstable RORC 54 38 COc1cc(S(=O)(=O)Cl)cc(C)c1Cl ZINC000217804423 CF For-Sale Unstable FFAR4 17 44 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1ccc(Oc2ccccc2)cc1 ZINC000217804430 HH For-Sale Unstable ADAMTS5 35 44 COc1ccc([C@@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1OC ZINC000217804458 KH In-Stock Unstable PRKDC 16 41 COc1ccc([C@@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1OC ZINC000217804458 KH In-Stock Unstable CYP1B1 60 39 COc1ccc([C@@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1OC ZINC000217804458 KH In-Stock Unstable CYP1A1 45 39 COc1ccc([C@@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1OC ZINC000217804458 KH In-Stock Unstable RORC 54 38 C[C@@](O)(COC/C=C\c1ccccc1)C(=O)O ZINC000217804471 BD For-Sale Unstable CACNA1B 49 38 CC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217804491 DI For-Sale Unstable GUAB 0 41 CC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217804491 DI For-Sale Unstable IMDH_CRYPV 41 36 CC(C)NS(=O)(=O)c1ccc(C(=O)Nc2ccccc2Nc2ccccc2)cc1 ZINC000217804494 HI On-Demand Unstable CA2 23 42 CC(C)NS(=O)(=O)c1ccc(C(=O)Nc2ccccc2Nc2ccccc2)cc1 ZINC000217804494 HI On-Demand Unstable CA1 19 43 CC(C)NS(=O)(=O)c1ccc(C(=O)Nc2ccccc2Nc2ccccc2)cc1 ZINC000217804494 HI On-Demand Unstable KCNA5 0 40 CC(C)NS(=O)(=O)c1ccc(C(=O)Nc2ccccc2Nc2ccccc2)cc1 ZINC000217804494 HI On-Demand Unstable MMP13 39 43 CC(C)NS(=O)(=O)c1ccc(C(=O)Nc2ccccc2Nc2ccccc2)cc1 ZINC000217804494 HI On-Demand Unstable PRNP 40 36 CC(C)NS(=O)(=O)c1ccc(C(=O)Nc2ccccc2Nc2ccccc2)cc1 ZINC000217804494 HI On-Demand Unstable CA4 18 42 CC(C)NS(=O)(=O)c1ccc(C(=O)Nc2ccccc2Nc2ccccc2)cc1 ZINC000217804494 HI On-Demand Unstable MMP2 32 55 CC(C)NS(=O)(=O)c1ccc(C(=O)Nc2ccccc2Nc2ccccc2)cc1 ZINC000217804494 HI On-Demand Unstable HDAC1 26 43 CC(C)NS(=O)(=O)c1ccc(C(=O)Nc2ccccc2Nc2ccccc2)cc1 ZINC000217804494 HI On-Demand Unstable HDAC2 16 43 CC(C)NS(=O)(=O)c1ccc(C(=O)Nc2ccccc2Nc2ccccc2)cc1 ZINC000217804494 HI On-Demand Unstable PRTN3 51 32 CC(C)NS(=O)(=O)c1ccc(C(=O)Nc2ccccc2Nc2ccccc2)cc1 ZINC000217804494 HI On-Demand Unstable MMP9 16 46 CC(C)NS(=O)(=O)c1ccc(C(=O)Nc2ccccc2Nc2ccccc2)cc1 ZINC000217804494 HI On-Demand Unstable CA12 17 48 CC(C)NS(=O)(=O)c1ccc(C(=O)Nc2ccccc2Nc2ccccc2)cc1 ZINC000217804494 HI On-Demand Unstable ADAMTS4 55 36 CC(C)NS(=O)(=O)c1ccc(C(=O)Nc2ccccc2Nc2ccccc2)cc1 ZINC000217804494 HI On-Demand Unstable CA9 15 48 CC(C)NS(=O)(=O)c1ccc(C(=O)Nc2ccccc2Nc2ccccc2)cc1 ZINC000217804494 HI On-Demand Unstable E1 0 42 CC(C)NS(=O)(=O)c1ccc(C(=O)Nc2ccccc2Nc2ccccc2)cc1 ZINC000217804494 HI On-Demand Unstable IDO1 23 40 CC(C)NS(=O)(=O)c1ccc(C(=O)Nc2ccccc2Nc2ccccc2)cc1 ZINC000217804494 HI On-Demand Unstable CYNT 16 41 CC(C)NS(=O)(=O)c1ccc(C(=O)Nc2ccccc2Nc2ccccc2)cc1 ZINC000217804494 HI On-Demand Unstable AKR1C2 42 38 CC(C)NS(=O)(=O)c1ccc(C(=O)Nc2ccccc2Nc2ccccc2)cc1 ZINC000217804494 HI On-Demand Unstable LIMK2 43 40 CC(C)NS(=O)(=O)c1ccc(C(=O)Nc2ccccc2Nc2ccccc2)cc1 ZINC000217804494 HI On-Demand Unstable DAC 20 40 CC(C)NS(=O)(=O)c1ccc(C(=O)Nc2ccccc2Nc2ccccc2)cc1 ZINC000217804494 HI On-Demand Unstable KCNK3 66 37 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1ccc(Oc2ccccc2)cc1 ZINC000217804510 HH For-Sale Unstable ADAMTS5 35 44 COCCOCCNC(=O)/C=C\C(=O)O ZINC000217804516 BB For-Sale Unstable HCAR2 29 41 C[C@](O)(COC/C=C\c1ccccc1)C(=O)O ZINC000217804548 BD For-Sale Unstable CACNA1B 49 38 COc1cc(C)c(Cl)c(S(=O)(=O)Cl)c1 ZINC000217804554 CF For-Sale Unstable FFAR4 21 44 COc1ccc(S(=O)(=O)N2[C@@H](C)C[C@@H]3CNC[C@H]32)cc1 ZINC000217804585 CD For-Sale Unstable MMP13 47 44 COc1ccc(S(=O)(=O)N2[C@@H](C)C[C@@H]3CNC[C@H]32)cc1 ZINC000217804585 CD For-Sale Unstable MMP2 28 41 COc1ccc(S(=O)(=O)N2[C@@H](C)C[C@@H]3CNC[C@H]32)cc1 ZINC000217804585 CD For-Sale Unstable MMP3 55 44 COc1ccc(S(=O)(=O)N2[C@@H](C)C[C@@H]3CNC[C@H]32)cc1 ZINC000217804585 CD For-Sale Unstable MMP8 30 41 COc1ccc(S(=O)(=O)N2[C@@H](C)C[C@@H]3CNC[C@H]32)cc1 ZINC000217804585 CD For-Sale Unstable MMP9 39 44 COc1ccc(S(=O)(=O)N2[C@@H](C)C[C@@H]3CNC[C@H]32)cc1 ZINC000217804585 CD For-Sale Unstable MMP7 50 41 COc1ccc(S(=O)(=O)N2[C@@H](C)C[C@@H]3CNC[C@H]32)cc1 ZINC000217804585 CD For-Sale Unstable MMP1 49 44 CC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217804592 DI For-Sale Unstable CCR3 17 40 CC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217804592 DI For-Sale Unstable GUAB 0 43 CC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217804592 DI For-Sale Unstable AKR1C3 23 43 CC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217804592 DI For-Sale Unstable IMDH_CRYPV 57 40 CC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217804592 DI For-Sale Unstable KCNK3 91 43 CC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217804592 DI For-Sale Unstable KCNK9 49 36 COC(=O)[C@](C)(O)COC/C=C\c1ccccc1 ZINC000217804611 CD For-Sale Unstable CACNA1B 48 36 C[C@H](F)CN(C(=O)OC(C)(C)C)[C@@H]1CCNC1 ZINC000217804640 BD For-Sale Unstable SLC6A2 31 45 C[C@H](F)CN(C(=O)OC(C)(C)C)[C@@H]1CCNC1 ZINC000217804640 BD For-Sale Unstable MBTPS1 44 31 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1ccc(Br)cc1 ZINC000217804647 HF For-Sale Unstable ADAMTS5 26 43 COc1ccc(S(=O)(=O)N2[C@@H]3CNC[C@H]3C[C@H]2C)cc1 ZINC000217804651 CD For-Sale Unstable MMP13 47 44 COc1ccc(S(=O)(=O)N2[C@@H]3CNC[C@H]3C[C@H]2C)cc1 ZINC000217804651 CD For-Sale Unstable MMP2 28 41 COc1ccc(S(=O)(=O)N2[C@@H]3CNC[C@H]3C[C@H]2C)cc1 ZINC000217804651 CD For-Sale Unstable MMP3 55 44 COc1ccc(S(=O)(=O)N2[C@@H]3CNC[C@H]3C[C@H]2C)cc1 ZINC000217804651 CD For-Sale Unstable MMP8 30 41 COc1ccc(S(=O)(=O)N2[C@@H]3CNC[C@H]3C[C@H]2C)cc1 ZINC000217804651 CD For-Sale Unstable MMP9 39 44 COc1ccc(S(=O)(=O)N2[C@@H]3CNC[C@H]3C[C@H]2C)cc1 ZINC000217804651 CD For-Sale Unstable MMP7 50 41 COc1ccc(S(=O)(=O)N2[C@@H]3CNC[C@H]3C[C@H]2C)cc1 ZINC000217804651 CD For-Sale Unstable MMP1 49 44 Cc1cc(F)ccc1S(=O)(=O)N1CCC[C@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217804663 IH In-Stock Unstable Q8MHZ5_SHEEP 40 32 COC(=O)[C@@](C)(O)COC/C=C\c1ccccc1 ZINC000217804701 CD For-Sale Unstable CACNA1B 48 36 O=C(N[C@@H]1CCN2CCCC[C@@H]12)c1ccc2c(c1)CCN2 ZINC000217804709 CE On-Demand Unstable L3MBTL3 44 32 CC(C)OC(=O)[C@@H]1CCc2ccccc2C1 ZINC000217804711 BF On-Demand Unstable NPY1R 40 36 C[C@@H](CCc1ccc(O)cc1)N1CCO[C@@H]2CCC[C@@H]21 ZINC000217804715 CF For-Sale Unstable BIRC2 40 38 C[C@@H](F)CN(C(=O)OC(C)(C)C)[C@@H]1CCNC1 ZINC000217804726 BD For-Sale Unstable SLC6A2 31 45 C[C@@H](F)CN(C(=O)OC(C)(C)C)[C@@H]1CCNC1 ZINC000217804726 BD For-Sale Unstable MBTPS1 44 31 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1ccc(Br)cc1 ZINC000217804733 HF For-Sale Unstable ADAMTS5 26 43 Cc1cc(F)ccc1S(=O)(=O)N1CCC[C@@H](Cc2nc(-c3ccccc3F)no2)C1 ZINC000217804747 IH In-Stock Unstable Q8MHZ5_SHEEP 40 32 O=C(NN1CCCCC1)c1ccc(=O)[nH]n1 ZINC000217804760 BB On-Demand Unstable CNR1 51 32 COC(=O)C[C@H](c1ccccc1OCCc1ccc(OC)cc1)c1c(O)c2ccccc2oc1=O ZINC000217804773 JJ In-Stock Unstable NQO1 30 51 COC(=O)C[C@H](c1ccccc1OCCc1ccc(OC)cc1)c1c(O)c2ccccc2oc1=O ZINC000217804773 JJ In-Stock Unstable ABCG2 20 42 CC(C)OC(=O)[C@H]1CCc2ccccc2C1 ZINC000217804788 BF On-Demand Unstable NPY1R 40 36 O=C(N[C@H]1CCN2CCCC[C@@H]12)c1ccc2c(c1)CCN2 ZINC000217804792 CE On-Demand Unstable L3MBTL3 44 32 C[C@H](CCc1ccc(O)cc1)N1CCO[C@@H]2CCC[C@@H]21 ZINC000217804795 CF For-Sale Unstable BIRC2 40 38 C[C@H](F)CN(C(=O)OC(C)(C)C)[C@H]1CCNC1 ZINC000217804815 BD For-Sale Unstable SLC6A2 31 45 C[C@H](F)CN(C(=O)OC(C)(C)C)[C@H]1CCNC1 ZINC000217804815 BD For-Sale Unstable MBTPS1 44 31 COC(=O)C[C@@H](c1ccccc1OCCc1ccc(OC)cc1)c1c(O)c2ccccc2oc1=O ZINC000217804818 JJ In-Stock Unstable NQO1 30 51 COC(=O)C[C@@H](c1ccccc1OCCc1ccc(OC)cc1)c1c(O)c2ccccc2oc1=O ZINC000217804818 JJ In-Stock Unstable ABCG2 20 42 Cc1cccc(NC(=O)N/C=C/c2ccccc2Cl)c1C ZINC000217804822 DJ For-Sale Unstable CXCL8 45 39 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2nccs2)cc1 ZINC000217804846 HC For-Sale Unstable ADAMTS5 26 43 C[C@@H](c1cccc(Cl)c1)N(C)[C@@H](CN)Cc1ccccc1 ZINC000217804873 DH For-Sale Unstable ADRB3 19 41 C[C@@H](c1cccc(Cl)c1)N(C)[C@@H](CN)Cc1ccccc1 ZINC000217804873 DH For-Sale Unstable AOC3 18 42 C[C@@H](c1cccc(Cl)c1)N(C)[C@@H](CN)Cc1ccccc1 ZINC000217804873 DH For-Sale Unstable TAAR1 15 40 C[C@@H](F)CN(C(=O)OC(C)(C)C)[C@H]1CCNC1 ZINC000217804898 BD For-Sale Unstable SLC6A2 31 45 C[C@@H](F)CN(C(=O)OC(C)(C)C)[C@H]1CCNC1 ZINC000217804898 BD For-Sale Unstable MBTPS1 44 31 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2nccs2)cc1 ZINC000217804914 HC For-Sale Unstable ADAMTS5 26 43 C[C@H](c1cccc(Cl)c1)N(C)[C@@H](CN)Cc1ccccc1 ZINC000217804922 DH For-Sale Unstable ADRB3 19 41 C[C@H](c1cccc(Cl)c1)N(C)[C@@H](CN)Cc1ccccc1 ZINC000217804922 DH For-Sale Unstable AOC3 18 42 C[C@H](c1cccc(Cl)c1)N(C)[C@@H](CN)Cc1ccccc1 ZINC000217804922 DH For-Sale Unstable TAAR1 15 40 NCc1ccc(C(=O)N[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217804932 CD On-Demand Unstable SIGMAR1 0 50 NCc1ccc(C(=O)N[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217804932 CD On-Demand Unstable SSTR3 28 44 NCc1ccc(C(=O)N[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217804932 CD On-Demand Unstable L3MBTL3 63 36 c1ccc(Cn2cc(NC3=NCCC3)cn2)cc1 ZINC000217804943 BF In-Stock Unstable ITK 30 45 c1ccc(Cn2cc(NC3=NCCC3)cn2)cc1 ZINC000217804943 BF In-Stock Unstable PANC 48 40 C[C@@H](c1cccc(Cl)c1)N(C)[C@@]1(CN)CN2CCC1CC2 ZINC000217805014 DF For-Sale Unstable OPRL1 15 41 NCc1ccc(C(=O)N[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217805017 CD On-Demand Unstable SIGMAR1 0 50 NCc1ccc(C(=O)N[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217805017 CD On-Demand Unstable SSTR3 28 44 NCc1ccc(C(=O)N[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217805017 CD On-Demand Unstable L3MBTL3 63 36 COc1ccc(C)cc1NC(=O)N/C=C/c1ccccc1Cl ZINC000217805032 DI For-Sale Unstable KCNMA1 18 41 COc1ccc(C)cc1NC(=O)N/C=C/c1ccccc1Cl ZINC000217805032 DI For-Sale Unstable CYSP_PLAFA 40 35 O=S(=O)(Cc1cccc(C(F)(F)F)c1)NC[C@@H]1CCCN1c1nccs1 ZINC000217805035 HG In-Stock Unstable ADAMTS5 26 41 O=S(=O)(Cc1cccc(C(F)(F)F)c1)NC[C@H]1CCCN1c1nccs1 ZINC000217805095 HG In-Stock Unstable ADAMTS5 26 41 C[C@H](c1cccc(Cl)c1)N(C)[C@@]1(CN)CN2CCC1CC2 ZINC000217805107 DF For-Sale Unstable OPRL1 15 41 Cc1cccc(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217805126 CI For-Sale Unstable LPL 42 32 Cc1cccc(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217805126 CI For-Sale Unstable PTGER3 0 47 Cc1cccc(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217805126 CI For-Sale Unstable CCKAR 25 49 Cc1cccc(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217805126 CI For-Sale Unstable KDR 18 42 Cc1cccc(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217805126 CI For-Sale Unstable CCKBR 36 41 Cc1cccc(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217805126 CI For-Sale Unstable KCNK3 104 50 Cc1cccc(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217805126 CI For-Sale Unstable KCNK9 59 44 Nc1cccc(C(=O)N[C@@H]2CCN3CCCC[C@@H]23)c1 ZINC000217805166 CD On-Demand Unstable VACHT_TETCF 0 41 Nc1cccc(C(=O)N[C@@H]2CCN3CCCC[C@@H]23)c1 ZINC000217805166 CD On-Demand Unstable SIGMAR1 0 44 Cc1ccc(Cn2cc(NC3=NCCC3)cn2)cc1 ZINC000217805187 CF In-Stock Unstable PANC 40 34 CN[C@@H](C)c1ccc(NC(=O)N[C@@H]2CCCC[C@@H]2C)cc1 ZINC000217805204 CH For-Sale Unstable EPHX2 26 53 Cc1cccc(Oc2ccc(S(=O)(=O)NC[C@@H]3CCCN3c3nccs3)cc2)c1 ZINC000217805205 II For-Sale Unstable ADAMTS5 26 40 Nc1cccc(C(=O)N[C@H]2CCN3CCCC[C@@H]23)c1 ZINC000217805229 CD On-Demand Unstable VACHT_TETCF 0 41 Nc1cccc(C(=O)N[C@H]2CCN3CCCC[C@@H]23)c1 ZINC000217805229 CD On-Demand Unstable SIGMAR1 0 44 O=C(N[C@@H](CCn1cncn1)c1ccccc1)c1ccc2[nH]nnc2c1 ZINC000217805251 EE In-Stock Unstable HIS3 43 35 O=C(N[C@@H](CCn1cncn1)c1ccccc1)c1ccc2[nH]nnc2c1 ZINC000217805251 EE In-Stock Unstable CYP51 0 42 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217805257 GK For-Sale Anodyne GUAB 0 48 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217805257 GK For-Sale Anodyne RAF1 34 47 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217805257 GK For-Sale Anodyne Q8MMZ8_EIMTE 54 47 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217805257 GK For-Sale Anodyne BRAF 15 41 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217805257 GK For-Sale Anodyne PTPA 0 47 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217805257 GK For-Sale Anodyne IMDH_CRYPV 37 50 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217805257 GK For-Sale Anodyne BLM 0 47 CC(C)(C)OC(=O)N1CCC(NCCF)CC1 ZINC000217805260 BD On-Demand Unstable GPR119 41 42 CN[C@@H](C)c1ccc(NC(=O)N[C@H]2CCCC[C@@H]2C)cc1 ZINC000217805288 CH For-Sale Unstable EPHX2 26 53 Cc1cccc(Oc2ccc(S(=O)(=O)NC[C@H]3CCCN3c3nccs3)cc2)c1 ZINC000217805303 II For-Sale Unstable ADAMTS5 26 40 O=C(N[C@H](CCn1cncn1)c1ccccc1)c1ccc2[nH]nnc2c1 ZINC000217805367 EE In-Stock Unstable HIS3 43 35 O=C(N[C@H](CCn1cncn1)c1ccccc1)c1ccc2[nH]nnc2c1 ZINC000217805367 EE In-Stock Unstable CYP51 0 42 C[C@H](F)CN[C@@H]1CCN(C(=O)OC(C)(C)C)C1 ZINC000217805385 BD For-Sale Unstable GPR119 33 43 Nc1ccc(C(=O)N[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217805409 CD On-Demand Unstable VACHT_TETCF 0 40 Nc1ccc(C(=O)N[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217805409 CD On-Demand Unstable SIGMAR1 0 44 Nc1ccc(C(=O)N[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217805409 CD On-Demand Unstable L3MBTL3 70 36 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1cccc(-c2ccccc2)c1 ZINC000217805410 GH For-Sale Unstable ADAMTS5 34 46 COC(=O)C[C@H](c1ccc2ncccc2c1)c1c(O)c2ccccc2oc1=O ZINC000217805413 GH In-Stock Unstable NQO1 53 49 C[C@@H](F)CN[C@@H]1CCN(C(=O)OC(C)(C)C)C1 ZINC000217805456 BD For-Sale Unstable GPR119 33 43 COC(=O)C[C@@H](c1ccc2ncccc2c1)c1c(O)c2ccccc2oc1=O ZINC000217805487 GH In-Stock Unstable NQO1 53 49 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1cccc(-c2ccccc2)c1 ZINC000217805489 GH For-Sale Unstable ADAMTS5 34 46 Nc1ccc(C(=O)N[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217805490 CD On-Demand Unstable VACHT_TETCF 0 40 Nc1ccc(C(=O)N[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217805490 CD On-Demand Unstable SIGMAR1 0 44 Nc1ccc(C(=O)N[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217805490 CD On-Demand Unstable L3MBTL3 70 36 COC(=O)c1ccc(Cn2cc(NC3=NCCC3)cn2)o1 ZINC000217805523 CD In-Stock Unstable PANC 52 38 C[C@H](F)CN[C@H]1CCN(C(=O)OC(C)(C)C)C1 ZINC000217805533 BD For-Sale Unstable GPR119 33 43 CC(C)CCc1cc(C(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)[nH]n1 ZINC000217805601 FE In-Stock Unstable CHRNA4 30 46 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1cccc(-c2ccc(Cl)cc2)c1 ZINC000217805605 II For-Sale Unstable DCK 33 40 O=S(=O)(NC[C@@H]1CCCN1c1nccs1)c1cccc(-c2ccc(Cl)cc2)c1 ZINC000217805605 II For-Sale Unstable ADAMTS5 25 45 C[C@H](N)c1cccc(NC(=O)N[C@@H]2CCCC[C@@H]2C)c1 ZINC000217805612 CG For-Sale Unstable EPHX2 16 44 C[C@H](N)c1cccc(NC(=O)N[C@@H]2CCCC[C@@H]2C)c1 ZINC000217805612 CG For-Sale Unstable METAP2 0 40 C[C@@H](F)CN[C@H]1CCN(C(=O)OC(C)(C)C)C1 ZINC000217805613 BD For-Sale Unstable GPR119 33 43 CCN1CCN(c2ccccc2NC(=O)CCn2c(=O)n(C)c3ccccc32)CC1 ZINC000217805675 HF On-Demand Unstable HTR1A 59 43 CCN1CCN(c2ccccc2NC(=O)CCn2c(=O)n(C)c3ccccc32)CC1 ZINC000217805675 HF On-Demand Unstable ADRA1D 24 45 CCN1CCN(c2ccccc2NC(=O)CCn2c(=O)n(C)c3ccccc32)CC1 ZINC000217805675 HF On-Demand Unstable HTR7 61 39 CCN1CCN(c2ccccc2NC(=O)CCn2c(=O)n(C)c3ccccc32)CC1 ZINC000217805675 HF On-Demand Unstable KCNQ2 82 43 CCN1CCN(c2ccccc2NC(=O)CCn2c(=O)n(C)c3ccccc32)CC1 ZINC000217805675 HF On-Demand Unstable PRNP 29 42 C[C@H](N)c1cccc(NC(=O)N[C@H]2CCCC[C@@H]2C)c1 ZINC000217805694 CG For-Sale Unstable EPHX2 16 44 C[C@H](N)c1cccc(NC(=O)N[C@H]2CCCC[C@@H]2C)c1 ZINC000217805694 CG For-Sale Unstable METAP2 0 40 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1cccc(-c2ccc(Cl)cc2)c1 ZINC000217805696 II For-Sale Unstable DCK 33 40 O=S(=O)(NC[C@H]1CCCN1c1nccs1)c1cccc(-c2ccc(Cl)cc2)c1 ZINC000217805696 II For-Sale Unstable ADAMTS5 25 45 O=C(N/C=C/c1ccccc1Cl)Nc1cccc(Cl)c1 ZINC000217805724 DJ For-Sale Anodyne PPIA 18 42 O=C(N/C=C/c1ccccc1Cl)Nc1cccc(Cl)c1 ZINC000217805724 DJ For-Sale Anodyne KCNK3 57 46 O=C(N/C=C/c1ccccc1Cl)Nc1cccc(Cl)c1 ZINC000217805724 DJ For-Sale Anodyne KCNK9 27 40 COc1ccc(CCNC(=O)Cn2ccc3c(NC(C)=O)cccc32)cc1OC ZINC000217805830 GF In-Stock Unstable NR5A1 30 41 C[C@H](N)c1ccc(NC(=O)N[C@@H]2CCCC[C@@H]2C)cc1 ZINC000217805838 CG For-Sale Unstable EPHX2 29 58 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(Cl)cc1 ZINC000217805846 DJ For-Sale Anodyne SMO 16 41 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(Cl)cc1 ZINC000217805846 DJ For-Sale Anodyne P95276_MYCTO 0 46 C[C@H](N)c1ccc(NC(=O)N[C@H]2CCCC[C@@H]2C)cc1 ZINC000217805909 CG For-Sale Unstable EPHX2 29 58 CCC(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217806020 BE For-Sale Unstable MTNR1A 28 40 CCC(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217806020 BE For-Sale Unstable MTNR1B 30 40 CCCn1c(CNC[C@@H]2CC2(C)C)nc2ccccc21 ZINC000217806031 CH On-Demand Unstable HRH1 15 43 O=C(N/C=C/c1ccccc1Cl)N1CCN(Cc2ccccc2)CC1 ZINC000217806046 FH For-Sale Unstable DRD3 23 40 O=C(N/C=C/c1ccccc1Cl)N1CCN(Cc2ccccc2)CC1 ZINC000217806046 FH For-Sale Unstable FAAH 0 53 O=C(N/C=C/c1ccccc1Cl)N1CCN(Cc2ccccc2)CC1 ZINC000217806046 FH For-Sale Unstable MGLL 0 44 O=C(N/C=C/c1ccccc1Cl)N1CCN(Cc2ccccc2)CC1 ZINC000217806046 FH For-Sale Unstable ABHD6 0 41 O=C(N/C=C/c1ccccc1Cl)N1CCN(Cc2ccccc2)CC1 ZINC000217806046 FH For-Sale Unstable GPR183 0 40 CCC(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217806112 BE For-Sale Unstable MTNR1A 28 40 CCC(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217806112 BE For-Sale Unstable MTNR1B 30 40 O=C([C@H]1C[C@H]1c1ccc(Br)cc1)N1CCOCC1 ZINC000217806116 DE On-Demand Unstable PRCP 21 55 O=C([C@H]1C[C@H]1c1ccc(Br)cc1)N1CCOCC1 ZINC000217806116 DE On-Demand Unstable AKR1C3 29 49 CCCn1c(CNC[C@H]2CC2(C)C)nc2ccccc21 ZINC000217806122 CH On-Demand Unstable HRH1 15 43 CN[C@@H](C)c1ccc(NC(=O)N2C[C@@H](C)C[C@@H](C)C2)cc1 ZINC000217806129 CG For-Sale Unstable EPHX2 17 43 CC(=O)Nc1cccc2c1ccn2CC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217806135 HE In-Stock Unstable CHRNA4 28 48 Nc1ccc(CC(=O)N[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217806173 CD On-Demand Unstable OPRK1 0 41 Nc1ccc(CC(=O)N[C@@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217806173 CD On-Demand Unstable SIGMAR1 23 41 COC(=O)c1ccc(C(=O)N2CCC[C@H](Cc3nc(C4CC4)no3)C2)cc1 ZINC000217806182 FF In-Stock Unstable GRM3 15 45 CN[C@@H](C)c1ccc(NC(=O)N2C[C@H](C)C[C@@H](C)C2)cc1 ZINC000217806201 CG For-Sale Unstable EPHX2 17 43 CC1(C)[C@@H]2CC[C@]1(C)[C@@H](NC(=O)c1ccc(F)cc1)C2 ZINC000217806208 CH In-Stock Unstable SSTR3 16 40 O=C([C@@H]1C[C@H]1c1ccc(Br)cc1)N1CCOCC1 ZINC000217806209 DE On-Demand Unstable PRCP 21 55 O=C([C@@H]1C[C@H]1c1ccc(Br)cc1)N1CCOCC1 ZINC000217806209 DE On-Demand Unstable AKR1C3 29 49 CCCCC(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217806227 CF For-Sale Unstable P2RY12 59 33 COC(=O)c1ccc(C(=O)N2CCC[C@@H](Cc3nc(C4CC4)no3)C2)cc1 ZINC000217806254 FF In-Stock Unstable GRM3 15 45 Nc1ccc(CC(=O)N[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217806259 CD On-Demand Unstable OPRK1 0 41 Nc1ccc(CC(=O)N[C@H]2CCN3CCCC[C@@H]23)cc1 ZINC000217806259 CD On-Demand Unstable SIGMAR1 23 41 O=C([C@@H]1C[C@@H]1c1ccc(Br)cc1)N1CCOCC1 ZINC000217806267 DE On-Demand Unstable PRCP 21 55 O=C([C@@H]1C[C@@H]1c1ccc(Br)cc1)N1CCOCC1 ZINC000217806267 DE On-Demand Unstable AKR1C3 29 49 CCCCC(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217806297 CF For-Sale Unstable P2RY12 59 33 O=C(N/C=C/c1ccccc1Cl)NC1CCCCCCCCCCC1 ZINC000217806361 FK For-Sale Unstable EPHX2 36 48 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)Nc3ccc4c(c3)ncn4C)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217806411 KH In-Stock Unstable TUBA1A 19 61 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)Nc3ccc4c(c3)ncn4C)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217806411 KH In-Stock Unstable TPPP 0 58 O=C(N/C=C/c1ccccc1Cl)NCCN1CCOCC1 ZINC000217806463 DD For-Sale Unstable DRD4 46 38 O=C(N/C=C/c1ccccc1Cl)NCCN1CCOCC1 ZINC000217806463 DD For-Sale Unstable DRD3 22 41 O=C(N/C=C/c1ccccc1Cl)NCCN1CCOCC1 ZINC000217806463 DD For-Sale Unstable CASR 43 34 O=C(N/C=C/c1ccccc1Cl)NCCN1CCOCC1 ZINC000217806463 DD For-Sale Unstable EPHX2 22 47 O=C(N/C=C/c1ccccc1Cl)NCCN1CCOCC1 ZINC000217806463 DD For-Sale Unstable HPGDS 23 40 O=C([C@H]1C[C@H]1c1ccc(Br)cc1)N1CCCC1 ZINC000217806516 CG On-Demand Unstable SLC6A1 15 47 O=C([C@H]1C[C@H]1c1ccc(Br)cc1)N1CCCC1 ZINC000217806516 CG On-Demand Unstable PRCP 15 44 O=C([C@H]1C[C@H]1c1ccc(Br)cc1)N1CCCC1 ZINC000217806516 CG On-Demand Unstable PREP 46 50 CNC[C@H]1OC(=O)N2c3ccc(OC)cc3CC[C@H]12 ZINC000217806557 CD For-Sale Unstable SRD5A1 15 41 Cc1ccc(C(=O)N[C@@H]2CCN3CCCC[C@@H]23)cc1N ZINC000217806561 CD On-Demand Unstable SIGMAR1 0 42 Cc1ccc(C(=O)N[C@@H]2CCN3CCCC[C@@H]23)cc1N ZINC000217806561 CD On-Demand Unstable L3MBTL3 56 39 CN(C)[C@@H]1[C@H]2CC[C@@H]1CN(C(=O)CN1CCC(c3ccccc3)CC1)C2 ZINC000217806605 FF In-Stock Unstable CCR5 50 47 COc1ccc(O)c(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217806610 FG On-Demand Unstable DRD2 37 54 COc1ccc(O)c(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217806610 FG On-Demand Unstable CNR1 19 44 COc1ccc(O)c(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217806610 FG On-Demand Unstable DRD4 77 60 COc1ccc(O)c(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217806610 FG On-Demand Unstable ACHE 27 58 COc1ccc(O)c(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217806610 FG On-Demand Unstable HTR2A 15 60 COc1ccc(O)c(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217806610 FG On-Demand Unstable SLC6A1 23 48 COc1ccc(O)c(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217806610 FG On-Demand Unstable HRH1 21 43 COc1ccc(O)c(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217806610 FG On-Demand Unstable DRD3 40 53 COc1ccc(O)c(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217806610 FG On-Demand Unstable AVPR1A 20 42 COc1ccc(O)c(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217806610 FG On-Demand Unstable HTR3A 21 44 COc1ccc(O)c(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217806610 FG On-Demand Unstable AVPR1B 41 33 COc1ccc(O)c(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217806610 FG On-Demand Unstable KCNH2 25 51 COc1ccc(O)c(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217806610 FG On-Demand Unstable HTR4 59 53 COc1ccc(O)c(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217806610 FG On-Demand Unstable CHRM3 15 44 COc1ccc(O)c(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217806610 FG On-Demand Unstable LTA4H 22 41 COc1ccc(O)c(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217806610 FG On-Demand Unstable CNR2 21 44 COc1ccc(O)c(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217806610 FG On-Demand Unstable SIGMAR1 49 56 COc1ccc(O)c(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217806610 FG On-Demand Unstable SSTR5 82 43 COc1ccc(O)c(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217806610 FG On-Demand Unstable CCR1 27 44 COc1ccc(O)c(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217806610 FG On-Demand Unstable CCR3 64 48 COc1ccc(O)c(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217806610 FG On-Demand Unstable ADAM17 17 42 COc1ccc(O)c(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217806610 FG On-Demand Unstable UTS2R 22 48 COc1ccc(O)c(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217806610 FG On-Demand Unstable MTNR1B 16 41 COc1ccc(O)c(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217806610 FG On-Demand Unstable FAAH 23 40 COc1ccc(O)c(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217806610 FG On-Demand Unstable CCR2 19 45 COc1ccc(O)c(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217806610 FG On-Demand Unstable SLC6A5 36 43 COc1ccc(O)c(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217806610 FG On-Demand Unstable PDK1 64 53 COc1ccc(O)c(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217806610 FG On-Demand Unstable CXCR3 47 45 COc1ccc(O)c(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217806610 FG On-Demand Unstable MCHR1 77 74 COc1ccc(O)c(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217806610 FG On-Demand Unstable CACNA1I 51 42 COc1ccc(O)c(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217806610 FG On-Demand Unstable CCR8 21 43 O=C([C@@H]1C[C@H]1c1ccc(Br)cc1)N1CCCC1 ZINC000217806621 CG On-Demand Unstable SLC6A1 15 47 O=C([C@@H]1C[C@H]1c1ccc(Br)cc1)N1CCCC1 ZINC000217806621 CG On-Demand Unstable PRCP 15 44 O=C([C@@H]1C[C@H]1c1ccc(Br)cc1)N1CCCC1 ZINC000217806621 CG On-Demand Unstable PREP 46 50 Cc1ccc(C(=O)N[C@H]2CCN3CCCC[C@@H]23)cc1N ZINC000217806632 CD On-Demand Unstable SIGMAR1 0 42 Cc1ccc(C(=O)N[C@H]2CCN3CCCC[C@@H]23)cc1N ZINC000217806632 CD On-Demand Unstable L3MBTL3 56 39 CNC[C@@H]1OC(=O)N2c3ccc(OC)cc3CC[C@H]12 ZINC000217806640 CD For-Sale Unstable SRD5A1 15 41 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1 ZINC000217806643 CG For-Sale Unstable ACE 15 40 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1 ZINC000217806643 CG For-Sale Unstable DRD2 28 43 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1 ZINC000217806643 CG For-Sale Unstable SLC6A1 34 42 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1 ZINC000217806643 CG For-Sale Unstable GRIN2B 15 40 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1 ZINC000217806643 CG For-Sale Unstable HCRTR1 24 53 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1 ZINC000217806643 CG For-Sale Unstable PREP 34 50 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1 ZINC000217806643 CG For-Sale Unstable HCRTR2 17 53 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1 ZINC000217806643 CG For-Sale Unstable CACNA1I 55 34 C[C@H]1C[C@@H](C)CN(C(=O)Nc2ccc([C@H](C)N)cc2)C1 ZINC000217806666 CG For-Sale Unstable DPP4 16 44 C[C@H]1C[C@@H](C)CN(C(=O)Nc2ccc([C@H](C)N)cc2)C1 ZINC000217806666 CG For-Sale Unstable EPHX2 20 43 NCCN1CCN(C(=O)N/C=C/c2ccccc2Cl)CC1 ZINC000217806689 DD For-Sale Unstable DRD3 19 40 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccccc1 ZINC000217806705 CG For-Sale Unstable ACE 15 40 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccccc1 ZINC000217806705 CG For-Sale Unstable DRD2 28 43 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccccc1 ZINC000217806705 CG For-Sale Unstable SLC6A1 34 42 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccccc1 ZINC000217806705 CG For-Sale Unstable GRIN2B 15 40 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccccc1 ZINC000217806705 CG For-Sale Unstable HCRTR1 24 53 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccccc1 ZINC000217806705 CG For-Sale Unstable PREP 34 50 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccccc1 ZINC000217806705 CG For-Sale Unstable HCRTR2 17 53 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccccc1 ZINC000217806705 CG For-Sale Unstable CACNA1I 55 34 O=C([C@@H]1C[C@@H]1c1ccc(Br)cc1)N1CCCC1 ZINC000217806706 CG On-Demand Unstable SLC6A1 15 47 O=C([C@@H]1C[C@@H]1c1ccc(Br)cc1)N1CCCC1 ZINC000217806706 CG On-Demand Unstable PRCP 15 44 O=C([C@@H]1C[C@@H]1c1ccc(Br)cc1)N1CCCC1 ZINC000217806706 CG On-Demand Unstable PREP 46 50 N[C@@H](C(=O)N[C@@H]1CCN2CCCC[C@@H]12)c1ccccc1 ZINC000217806720 CD For-Sale Unstable SIGMAR1 15 42 N[C@@H](C(=O)N[C@@H]1CCN2CCCC[C@@H]12)c1ccccc1 ZINC000217806720 CD For-Sale Unstable SLC18A3 72 38 N[C@@H](C(=O)N[C@@H]1CCN2CCCC[C@@H]12)c1ccccc1 ZINC000217806720 CD For-Sale Unstable METAP2 0 41 CO[C@@H](CC(=O)O)c1ccc(OCc2ccccc2C)cc1 ZINC000217806724 DH In-Stock Unstable HMGCR 42 44 CO[C@@H](CC(=O)O)c1ccc(OCc2ccccc2C)cc1 ZINC000217806724 DH In-Stock Unstable PTGER4 21 45 CO[C@@H](CC(=O)O)c1ccc(OCc2ccccc2C)cc1 ZINC000217806724 DH In-Stock Unstable FFAR1 61 50 CO[C@@H](CC(=O)O)c1ccc(OCc2ccccc2C)cc1 ZINC000217806724 DH In-Stock Unstable FFAR4 48 41 C[C@H](N)c1ccc(NC(=O)N2C[C@H](C)C[C@@H](C)C2)cc1 ZINC000217806754 CG For-Sale Unstable DPP4 16 44 C[C@H](N)c1ccc(NC(=O)N2C[C@H](C)C[C@@H](C)C2)cc1 ZINC000217806754 CG For-Sale Unstable EPHX2 20 43 O=C(N/C=C/c1ccccc1Cl)NCCN1CCNCC1 ZINC000217806771 DD For-Sale Unstable DRD4 45 38 O=C(N/C=C/c1ccccc1Cl)NCCN1CCNCC1 ZINC000217806771 DD For-Sale Unstable DRD3 28 41 O=C(N/C=C/c1ccccc1Cl)NCCN1CCNCC1 ZINC000217806771 DD For-Sale Unstable PLD2 45 33 N[C@H](C(=O)N[C@@H]1CCN2CCCC[C@@H]12)c1ccccc1 ZINC000217806794 CD On-Demand Unstable VACHT_TETCF 0 42 N[C@H](C(=O)N[C@@H]1CCN2CCCC[C@@H]12)c1ccccc1 ZINC000217806794 CD On-Demand Unstable SIGMAR1 0 42 N[C@H](C(=O)N[C@@H]1CCN2CCCC[C@@H]12)c1ccccc1 ZINC000217806794 CD On-Demand Unstable SLC18A3 60 38 N[C@H](C(=O)N[C@@H]1CCN2CCCC[C@@H]12)c1ccccc1 ZINC000217806794 CD On-Demand Unstable METAP2 0 41 O=C(NCC1CCNCC1)C1CS(=O)(=O)C1 ZINC000217806806 BB For-Sale Unstable F2R 17 48 CO[C@H](CC(=O)O)c1ccc(OCc2ccccc2C)cc1 ZINC000217806808 DH In-Stock Unstable HMGCR 42 44 CO[C@H](CC(=O)O)c1ccc(OCc2ccccc2C)cc1 ZINC000217806808 DH In-Stock Unstable PTGER4 21 45 CO[C@H](CC(=O)O)c1ccc(OCc2ccccc2C)cc1 ZINC000217806808 DH In-Stock Unstable FFAR1 61 50 CO[C@H](CC(=O)O)c1ccc(OCc2ccccc2C)cc1 ZINC000217806808 DH In-Stock Unstable FFAR4 48 41 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccccn1 ZINC000217806817 CE For-Sale Unstable HCRTR1 24 41 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccccn1 ZINC000217806817 CE For-Sale Unstable GRM4 53 39 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccccn1 ZINC000217806817 CE For-Sale Unstable HCRTR2 21 41 N[C@@H](C(=O)N[C@H]1CCN2CCCC[C@@H]12)c1ccccc1 ZINC000217806864 CD For-Sale Unstable VACHT_TETCF 0 42 N[C@@H](C(=O)N[C@H]1CCN2CCCC[C@@H]12)c1ccccc1 ZINC000217806864 CD For-Sale Unstable SIGMAR1 15 42 N[C@@H](C(=O)N[C@H]1CCN2CCCC[C@@H]12)c1ccccc1 ZINC000217806864 CD For-Sale Unstable SLC18A3 72 38 CCn1ccnc1CN[C@@H]1CCN(C(=O)OC(C)(C)C)C1 ZINC000217806883 CE On-Demand Unstable GPR119 35 42 O=S(=O)(CCCCO)Nc1ccc2c(c1)CCC2 ZINC000217806884 CD For-Sale Unstable MLNR 0 40 Cc1ccc(CNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217806886 DI For-Sale Unstable ANPEP 16 40 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccccn1 ZINC000217806898 CE For-Sale Unstable HCRTR1 24 41 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccccn1 ZINC000217806898 CE For-Sale Unstable GRM4 53 39 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccccn1 ZINC000217806898 CE For-Sale Unstable HCRTR2 21 41 O[C@@H](CCI)c1cccc(Cl)c1 ZINC000217806918 CG For-Sale Unstable ADRB1 18 41 O[C@@H](CCI)c1cccc(Cl)c1 ZINC000217806918 CG For-Sale Unstable ADRB3 29 41 N[C@H](C(=O)N[C@H]1CCN2CCCC[C@@H]12)c1ccccc1 ZINC000217806924 CD On-Demand Unstable VACHT_TETCF 0 42 N[C@H](C(=O)N[C@H]1CCN2CCCC[C@@H]12)c1ccccc1 ZINC000217806924 CD On-Demand Unstable SIGMAR1 0 42 N[C@H](C(=O)N[C@H]1CCN2CCCC[C@@H]12)c1ccccc1 ZINC000217806924 CD On-Demand Unstable SLC18A3 60 38 N[C@H](C(=O)N[C@H]1CCN2CCCC[C@@H]12)c1ccccc1 ZINC000217806924 CD On-Demand Unstable METAP2 0 41 CCCO[C@@H](CC(=O)O)c1ccc(OCc2ccccc2C)cc1 ZINC000217806940 EJ In-Stock Unstable HMGCR 31 43 CCCO[C@@H](CC(=O)O)c1ccc(OCc2ccccc2C)cc1 ZINC000217806940 EJ In-Stock Unstable PTGER4 26 42 CCCO[C@@H](CC(=O)O)c1ccc(OCc2ccccc2C)cc1 ZINC000217806940 EJ In-Stock Unstable ACACA 39 41 CCCO[C@@H](CC(=O)O)c1ccc(OCc2ccccc2C)cc1 ZINC000217806940 EJ In-Stock Unstable ACACB 22 41 CCCO[C@@H](CC(=O)O)c1ccc(OCc2ccccc2C)cc1 ZINC000217806940 EJ In-Stock Unstable PLA2G4B 56 34 CCCO[C@@H](CC(=O)O)c1ccc(OCc2ccccc2C)cc1 ZINC000217806940 EJ In-Stock Unstable FFAR1 51 55 CCCO[C@@H](CC(=O)O)c1ccc(OCc2ccccc2C)cc1 ZINC000217806940 EJ In-Stock Unstable FFAR4 42 38 CCn1ccnc1CN[C@H]1CCN(C(=O)OC(C)(C)C)C1 ZINC000217806953 CE On-Demand Unstable GPR119 35 42 CCCO[C@H](CC(=O)O)c1ccc(OCc2ccccc2C)cc1 ZINC000217807005 EJ In-Stock Unstable HMGCR 31 43 CCCO[C@H](CC(=O)O)c1ccc(OCc2ccccc2C)cc1 ZINC000217807005 EJ In-Stock Unstable PTGER4 26 42 CCCO[C@H](CC(=O)O)c1ccc(OCc2ccccc2C)cc1 ZINC000217807005 EJ In-Stock Unstable ACACA 39 41 CCCO[C@H](CC(=O)O)c1ccc(OCc2ccccc2C)cc1 ZINC000217807005 EJ In-Stock Unstable ACACB 22 41 CCCO[C@H](CC(=O)O)c1ccc(OCc2ccccc2C)cc1 ZINC000217807005 EJ In-Stock Unstable PLA2G4B 66 34 CCCO[C@H](CC(=O)O)c1ccc(OCc2ccccc2C)cc1 ZINC000217807005 EJ In-Stock Unstable FFAR1 67 83 CCCO[C@H](CC(=O)O)c1ccc(OCc2ccccc2C)cc1 ZINC000217807005 EJ In-Stock Unstable FFAR4 42 38 Cc1nc2cc(CNC(=O)CN3CCc4ccccc4C3)ccc2n1C ZINC000217807060 EF In-Stock Unstable HTR7 21 41 Cc1nc2cc(CNC(=O)CN3CCc4ccccc4C3)ccc2n1C ZINC000217807060 EF In-Stock Unstable ABCB1B 61 39 Cc1nc2cc(CNC(=O)CN3CCc4ccccc4C3)ccc2n1C ZINC000217807060 EF In-Stock Unstable ABCB1 0 44 Cc1nc2cc(CNC(=O)CN3CCc4ccccc4C3)ccc2n1C ZINC000217807060 EF In-Stock Unstable NOD2 44 39 O=C(NC[C@H]1CCCN1c1ccccc1)c1cnccn1 ZINC000217807065 CD For-Sale Unstable PSMB5 48 37 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cnccn1 ZINC000217807149 CD For-Sale Unstable PSMB5 48 37 O=C(N/C=C/c1ccccc1Cl)NCCCN1CCOCC1 ZINC000217807195 DE For-Sale Unstable HTR1A 19 40 O=C(N/C=C/c1ccccc1Cl)NCCCN1CCOCC1 ZINC000217807195 DE For-Sale Unstable DRD2 25 46 O=C(N/C=C/c1ccccc1Cl)NCCCN1CCOCC1 ZINC000217807195 DE For-Sale Unstable DRD3 47 46 O=C(N/C=C/c1ccccc1Cl)NCCCN1CCOCC1 ZINC000217807195 DE For-Sale Unstable TACR2 28 41 O=C(N/C=C/c1ccccc1Cl)NCCCN1CCOCC1 ZINC000217807195 DE For-Sale Unstable EPHX2 25 44 C[C@@H](c1ccc(Cl)cc1)N(C)C[C@@H](O)CN ZINC000217807244 BD On-Demand Unstable AOC3 23 50 Cc1nc(CCNC(=O)c2ccc(Br)c(Cl)c2)no1 ZINC000217807306 EF For-Sale Unstable KCNQ1 0 43 CC1(C)[C@H]2CC[C@@]1(C)[C@@H](NC(=O)c1cccs1)C2 ZINC000217807343 CH On-Demand Unstable OXTR 27 51 C[C@H](c1ccc(Cl)cc1)N(C)C[C@@H](O)CN ZINC000217807344 BD On-Demand Unstable AOC3 23 50 CNC[C@H](O)CN(C)[C@@H](C)c1ccc(Cl)cc1 ZINC000217807416 CD For-Sale Unstable UTS2 42 34 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccccc1F ZINC000217807444 CG For-Sale Unstable DRD2 31 40 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccccc1F ZINC000217807444 CG For-Sale Unstable SLC6A1 58 42 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccccc1F ZINC000217807444 CG For-Sale Unstable HCRTR1 37 44 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccccc1F ZINC000217807444 CG For-Sale Unstable HCRTR2 28 44 O[C@@H]1CCC[C@@H]1N[C@@H]1CCc2ccccc21 ZINC000217807454 BE On-Demand Unstable KCNN3 15 40 O[C@@H]1CCC[C@@H]1N[C@@H]1CCc2ccccc21 ZINC000217807454 BE On-Demand Unstable TSPAN17 0 40 CC(C)C[C@@H]1CN(c2cnc3ccccc3n2)CCN1 ZINC000217807512 CE For-Sale Unstable PRKCQ 19 51 O[C@@H]1CCC[C@H]1N[C@@H]1CCc2ccccc21 ZINC000217807521 BE On-Demand Unstable KCNN3 15 40 O[C@@H]1CCC[C@H]1N[C@@H]1CCc2ccccc21 ZINC000217807521 BE On-Demand Unstable TSPAN17 0 40 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1F ZINC000217807554 CG For-Sale Unstable DRD2 31 40 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1F ZINC000217807554 CG For-Sale Unstable SLC6A1 58 42 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1F ZINC000217807554 CG For-Sale Unstable HCRTR1 37 44 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1F ZINC000217807554 CG For-Sale Unstable HCRTR2 28 44 CC(C)C[C@H]1CN(c2cnc3ccccc3n2)CCN1 ZINC000217807583 CE For-Sale Unstable PRKCQ 19 51 Cc1csc(NC(=O)N/C=C/c2ccccc2Cl)n1 ZINC000217807603 CH For-Sale Unstable UL26 17 40 Cc1csc(NC(=O)N/C=C/c2ccccc2Cl)n1 ZINC000217807603 CH For-Sale Unstable GCK 18 43 C[C@H](N)c1cccc(NC(=O)N2[C@@H](C)CCC[C@@H]2C)c1 ZINC000217807606 CH For-Sale Unstable LIMK2 25 40 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(F)cc1 ZINC000217807644 CG For-Sale Unstable DRD2 48 36 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(F)cc1 ZINC000217807644 CG For-Sale Unstable DRD4 17 42 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(F)cc1 ZINC000217807644 CG For-Sale Unstable HCRTR1 34 57 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(F)cc1 ZINC000217807644 CG For-Sale Unstable CCR3 26 47 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(F)cc1 ZINC000217807644 CG For-Sale Unstable PLA2G4A 75 37 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(F)cc1 ZINC000217807644 CG For-Sale Unstable PLD1 68 41 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(F)cc1 ZINC000217807644 CG For-Sale Unstable PREP 16 43 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(F)cc1 ZINC000217807644 CG For-Sale Unstable SSTR3 19 40 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(F)cc1 ZINC000217807644 CG For-Sale Unstable PLD2 65 37 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(F)cc1 ZINC000217807644 CG For-Sale Unstable HCRTR2 22 57 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(F)cc1 ZINC000217807644 CG For-Sale Unstable ACKR3 65 36 C[C@H](N)c1ccc(NC(=O)N2[C@@H](C)CCC[C@@H]2C)cc1 ZINC000217807720 CH For-Sale Unstable HRH3 0 40 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(F)cc1 ZINC000217807729 CG For-Sale Unstable DRD2 48 36 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(F)cc1 ZINC000217807729 CG For-Sale Unstable DRD4 17 42 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(F)cc1 ZINC000217807729 CG For-Sale Unstable HCRTR1 34 57 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(F)cc1 ZINC000217807729 CG For-Sale Unstable CCR3 26 47 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(F)cc1 ZINC000217807729 CG For-Sale Unstable PLA2G4A 75 37 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(F)cc1 ZINC000217807729 CG For-Sale Unstable PLD1 68 41 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(F)cc1 ZINC000217807729 CG For-Sale Unstable PREP 16 43 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(F)cc1 ZINC000217807729 CG For-Sale Unstable SSTR3 19 40 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(F)cc1 ZINC000217807729 CG For-Sale Unstable PLD2 65 37 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(F)cc1 ZINC000217807729 CG For-Sale Unstable HCRTR2 22 57 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(F)cc1 ZINC000217807729 CG For-Sale Unstable ACKR3 65 36 C[C@@H](c1ccccc1Cl)N(C)C[C@@H](O)CN ZINC000217807732 BD On-Demand Unstable AOC3 18 54 COc1cccc(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217807809 DI For-Sale Unstable PTGER3 27 49 COc1cccc(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217807809 DI For-Sale Unstable MTNR1A 24 45 COc1cccc(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217807809 DI For-Sale Unstable MTNR1B 30 45 COc1cccc(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217807809 DI For-Sale Unstable TAAR1 38 50 COc1cccc(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217807809 DI For-Sale Unstable AKR1C3 15 41 COc1cccc(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217807809 DI For-Sale Unstable KCNK3 75 47 COc1cccc(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217807809 DI For-Sale Unstable KCNK9 59 38 C[C@H](c1ccccc1Cl)N(C)C[C@@H](O)CN ZINC000217807830 BD On-Demand Unstable AOC3 18 54 Nc1cc(C(=O)N[C@@H]2CCN3CCCC[C@@H]23)ccc1Cl ZINC000217807845 CE For-Sale Unstable HTR4 27 40 Nc1cc(C(=O)N[C@@H]2CCN3CCCC[C@@H]23)ccc1Cl ZINC000217807845 CE For-Sale Unstable SSTR3 29 40 Nc1cc(C(=O)N[C@@H]2CCN3CCCC[C@@H]23)ccc1Cl ZINC000217807845 CE For-Sale Unstable L3MBTL3 55 39 Cc1cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c(C)o1 ZINC000217807852 CG In-Stock Unstable DRD2 30 41 Cc1cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c(C)o1 ZINC000217807852 CG In-Stock Unstable HCRTR1 28 41 Cc1cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c(C)o1 ZINC000217807852 CG In-Stock Unstable HCRTR2 26 41 COCc1cc(=O)c(O)c([C@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2cc(OC)c(OC)c(OC)c2)o1 ZINC000217807866 KI In-Stock Unstable RORC 41 33 O=C(Cc1ccc(O)c(Cl)c1)N[C@@H]1CS(=O)(=O)C[C@H]1O ZINC000217807867 DB In-Stock Unstable NCE103 34 50 O=C(Cc1ccc(O)c(Cl)c1)N[C@@H]1CS(=O)(=O)C[C@H]1O ZINC000217807867 DB In-Stock Unstable P96878_MYCTU 21 48 O=C(Cc1ccc(O)c(Cl)c1)N[C@@H]1CS(=O)(=O)C[C@H]1O ZINC000217807867 DB In-Stock Unstable CAN2 0 50 O=C(N/C=C/c1ccccc1Cl)Nc1cc(Cl)ccc1O ZINC000217807894 DI For-Sale Anodyne KCNMA1 32 50 Nc1cc(C(=O)N[C@H]2CCN3CCCC[C@@H]23)ccc1Cl ZINC000217807907 CE For-Sale Unstable HTR4 27 40 Nc1cc(C(=O)N[C@H]2CCN3CCCC[C@@H]23)ccc1Cl ZINC000217807907 CE For-Sale Unstable SSTR3 29 40 Nc1cc(C(=O)N[C@H]2CCN3CCCC[C@@H]23)ccc1Cl ZINC000217807907 CE For-Sale Unstable L3MBTL3 55 39 COCc1cc(=O)c(O)c([C@@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2cc(OC)c(OC)c(OC)c2)o1 ZINC000217807920 KI In-Stock Unstable RORC 41 33 Cc1cc(C(=O)NC[C@H]2CCCN2c2ccccc2)c(C)o1 ZINC000217807922 CG In-Stock Unstable DRD2 30 41 Cc1cc(C(=O)NC[C@H]2CCCN2c2ccccc2)c(C)o1 ZINC000217807922 CG In-Stock Unstable HCRTR1 28 41 Cc1cc(C(=O)NC[C@H]2CCCN2c2ccccc2)c(C)o1 ZINC000217807922 CG In-Stock Unstable HCRTR2 26 41 COC(=O)C[C@H](c1ccc2c(c1)OCO2)c1c(O)cc(C)n(CCc2ccc(O)cc2)c1=O ZINC000217808017 JG In-Stock Unstable RORC 45 44 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217808022 CD On-Demand Unstable ACE 60 45 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217808022 CD On-Demand Unstable OPRM1 62 48 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217808022 CD On-Demand Unstable OPRD1 53 48 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217808022 CD On-Demand Unstable OPRK1 29 41 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217808022 CD On-Demand Unstable MME 56 42 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217808022 CD On-Demand Unstable VACHT_TETCF 0 40 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217808022 CD On-Demand Unstable SLC15A1 0 46 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217808022 CD On-Demand Unstable YARS 64 42 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217808022 CD On-Demand Unstable DPP7 55 37 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217808022 CD On-Demand Unstable POL 0 46 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217808022 CD On-Demand Unstable AMP1_PLAFQ 44 37 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217808022 CD On-Demand Unstable DPP8 26 44 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217808022 CD On-Demand Unstable SLC15A2 0 45 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217808022 CD On-Demand Unstable VM1B1_BOTAS 0 40 O=C(N/C=C/c1ccccc1Cl)Nc1nccs1 ZINC000217808076 CH For-Sale Anodyne MAP1 119 40 CC1(C)[C@H]2CC[C@@]1(C)[C@@H](NC(=O)Oc1ccccc1)C2 ZINC000217808095 CH For-Sale Unstable FAAH 26 43 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217808104 CD On-Demand Unstable ACE 60 45 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217808104 CD On-Demand Unstable OPRM1 62 48 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217808104 CD On-Demand Unstable OPRD1 53 48 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217808104 CD On-Demand Unstable OPRK1 29 41 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217808104 CD On-Demand Unstable MME 56 42 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217808104 CD On-Demand Unstable VACHT_TETCF 0 40 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217808104 CD On-Demand Unstable SLC15A1 0 46 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217808104 CD On-Demand Unstable YARS 64 42 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217808104 CD On-Demand Unstable DPP7 55 37 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217808104 CD On-Demand Unstable POL 0 46 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217808104 CD On-Demand Unstable AMP1_PLAFQ 44 37 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217808104 CD On-Demand Unstable DPP8 26 44 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217808104 CD On-Demand Unstable SLC15A2 0 45 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217808104 CD On-Demand Unstable VM1B1_BOTAS 0 40 COC(=O)C[C@@H](c1ccc2c(c1)OCO2)c1c(O)cc(C)n(CCc2ccc(O)cc2)c1=O ZINC000217808107 JG In-Stock Unstable RORC 45 44 C[C@@H](c1cccc(Cl)c1)N(C)C[C@@H](O)CN ZINC000217808150 BD On-Demand Unstable AOC3 34 47 CSc1cccc(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217808168 DJ For-Sale Unstable KCNK3 44 37 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217808192 CD On-Demand Unstable ACE 60 45 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217808192 CD On-Demand Unstable OPRM1 62 48 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217808192 CD On-Demand Unstable OPRD1 53 48 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217808192 CD On-Demand Unstable OPRK1 29 41 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217808192 CD On-Demand Unstable MME 56 42 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217808192 CD On-Demand Unstable VACHT_TETCF 0 40 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217808192 CD On-Demand Unstable SLC15A1 0 46 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217808192 CD On-Demand Unstable YARS 64 42 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217808192 CD On-Demand Unstable DPP7 55 37 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217808192 CD On-Demand Unstable POL 0 46 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217808192 CD On-Demand Unstable AMP1_PLAFQ 44 37 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217808192 CD On-Demand Unstable DPP8 26 44 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217808192 CD On-Demand Unstable SLC15A2 0 45 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217808192 CD On-Demand Unstable VM1B1_BOTAS 0 40 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](CC(C)C)C(=O)Nc3n[nH]c(C(C)C)n3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217808209 KJ In-Stock Unstable TUBA1A 17 61 C[C@H](c1cccc(Cl)c1)N(C)C[C@@H](O)CN ZINC000217808214 BD On-Demand Unstable AOC3 34 47 O=C(N/C=C/c1ccccc1Cl)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217808258 JH For-Sale Unstable LPL 51 44 O=C(N/C=C/c1ccccc1Cl)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217808258 JH For-Sale Unstable LIPG 20 44 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217808269 CD On-Demand Unstable ACE 60 45 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217808269 CD On-Demand Unstable OPRM1 62 48 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217808269 CD On-Demand Unstable OPRD1 53 48 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217808269 CD On-Demand Unstable OPRK1 29 41 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217808269 CD On-Demand Unstable MME 56 42 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217808269 CD On-Demand Unstable VACHT_TETCF 0 40 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217808269 CD On-Demand Unstable SLC15A1 0 46 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217808269 CD On-Demand Unstable YARS 64 42 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217808269 CD On-Demand Unstable DPP7 55 37 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217808269 CD On-Demand Unstable POL 0 46 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217808269 CD On-Demand Unstable AMP1_PLAFQ 44 37 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217808269 CD On-Demand Unstable DPP8 26 44 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217808269 CD On-Demand Unstable SLC15A2 0 45 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217808269 CD On-Demand Unstable VM1B1_BOTAS 0 40 CNC[C@H](O)CN(C)[C@@H](C)c1cccc(Cl)c1 ZINC000217808312 CD For-Sale Unstable ADRB1 20 41 CNC[C@H](O)CN(C)[C@@H](C)c1cccc(Cl)c1 ZINC000217808312 CD For-Sale Unstable ADRB3 32 41 CC[C@@H](C)[C@@H](N)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217808324 CD For-Sale Unstable TPP2 38 40 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217808362 FE For-Sale Unstable CA2 110 55 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217808362 FE For-Sale Unstable CA6 17 40 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217808362 FE For-Sale Unstable CA1 96 55 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217808362 FE For-Sale Unstable CA7 52 54 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217808362 FE For-Sale Unstable CA13 25 40 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217808362 FE For-Sale Unstable CA5B 61 54 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217808362 FE For-Sale Unstable CA4 71 55 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217808362 FE For-Sale Unstable CA5A 65 54 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217808362 FE For-Sale Unstable CA14 45 48 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217808362 FE For-Sale Unstable CA12 75 53 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217808362 FE For-Sale Unstable CA9 82 54 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217808362 FE For-Sale Unstable CYNT 27 43 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217808362 FE For-Sale Unstable NCE103 37 40 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217808362 FE For-Sale Unstable MTCA1 48 52 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217808362 FE For-Sale Unstable P96878_MYCTU 62 52 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217808362 FE For-Sale Unstable NAMPT 55 40 CC[C@H](C)[C@@H](N)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217808403 CD For-Sale Unstable TPP2 38 40 C[C@@H](c1cccc(Cl)c1)N(C)C[C@@H](O)CNC1CC1 ZINC000217808410 CE For-Sale Unstable ADRB1 17 40 C[C@@H](c1cccc(Cl)c1)N(C)C[C@@H](O)CNC1CC1 ZINC000217808410 CE For-Sale Unstable ADRB3 38 42 N#Cc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217808417 DF For-Sale Unstable DPP4 20 49 N#Cc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217808417 DF For-Sale Unstable ITK 23 40 N#Cc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217808417 DF For-Sale Unstable PREP 22 41 N#Cc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217808417 DF For-Sale Unstable CTRB_BOVIN 45 34 O=C(N/C=C/c1ccccc1Cl)Nc1cccnc1Cl ZINC000217808465 DI For-Sale Anodyne G2YM83_BOTF4 58 33 C[C@H](c1cccc(Cl)c1)N(C)C[C@@H](O)CNC1CC1 ZINC000217808499 CE For-Sale Unstable ADRB1 17 40 C[C@H](c1cccc(Cl)c1)N(C)C[C@@H](O)CNC1CC1 ZINC000217808499 CE For-Sale Unstable ADRB3 38 42 CC[C@@H](C)[C@H](N)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217808507 CD For-Sale Unstable TPP2 38 40 N#Cc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217808510 DF For-Sale Unstable DPP4 20 49 N#Cc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217808510 DF For-Sale Unstable ITK 23 40 N#Cc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217808510 DF For-Sale Unstable PREP 22 41 N#Cc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217808510 DF For-Sale Unstable CTRB_BOVIN 45 34 CC[C@H](C)[C@H](N)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217808575 CD On-Demand Unstable TPP2 38 40 O=C(CCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217808619 DG For-Sale Unstable SLC18A2 44 40 O=C(CCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217808619 DG For-Sale Unstable SIGMAR1 24 40 O=C(CCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217808619 DG For-Sale Unstable PREP 64 38 c1cnc2c(N[C@@H]3CC[C@@H]4CCCC[C@H]4C3)cccc2c1 ZINC000217808677 CK For-Sale Unstable NFKBIA 0 40 O=C(CCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217808690 DG For-Sale Unstable SLC18A2 44 40 O=C(CCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217808690 DG For-Sale Unstable SIGMAR1 24 40 O=C(CCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217808690 DG For-Sale Unstable PREP 64 38 N[C@@H](CC(=O)N[C@@H]1CCN2CCCC[C@@H]12)c1ccccc1 ZINC000217808706 CD For-Sale Unstable SIGMAR1 22 48 N[C@@H](CC(=O)N[C@@H]1CCN2CCCC[C@@H]12)c1ccccc1 ZINC000217808706 CD For-Sale Unstable SLC18A3 62 36 N[C@@H](CC(=O)N[C@@H]1CCN2CCCC[C@@H]12)c1ccccc1 ZINC000217808706 CD For-Sale Unstable METAP2 0 40 CCCCCC(=O)N[C@H]1CCC[C@H]1NC(=O)CCCCC ZINC000217808731 CG On-Demand Unstable LUXR 39 51 CCCCCC(=O)N[C@H]1CCC[C@H]1NC(=O)CCCCC ZINC000217808731 CG On-Demand Unstable TRAR 17 50 CCCCCC(=O)N[C@H]1CCC[C@H]1NC(=O)CCCCC ZINC000217808731 CG On-Demand Unstable LASR 70 50 CCCCCC(=O)N[C@H]1CCC[C@H]1NC(=O)CCCCC ZINC000217808731 CG On-Demand Unstable NOD1 43 37 CCCCCC(=O)N[C@H]1CCC[C@H]1NC(=O)CCCCC ZINC000217808731 CG On-Demand Unstable CQSS 56 34 c1cnc2c(N[C@H]3CC[C@@H]4CCCC[C@H]4C3)cccc2c1 ZINC000217808777 CK For-Sale Unstable NFKBIA 0 40 N[C@H](CC(=O)N[C@@H]1CCN2CCCC[C@@H]12)c1ccccc1 ZINC000217808781 CD On-Demand Unstable VACHT_TETCF 0 40 N[C@H](CC(=O)N[C@@H]1CCN2CCCC[C@@H]12)c1ccccc1 ZINC000217808781 CD On-Demand Unstable SIGMAR1 0 48 N[C@H](CC(=O)N[C@@H]1CCN2CCCC[C@@H]12)c1ccccc1 ZINC000217808781 CD On-Demand Unstable METAP2 0 40 COc1ccc([C@@H]2CC(=O)Oc3ccc4c(=O)c(-c5ccc(O)cc5)coc4c32)cc1O ZINC000217808792 II In-Stock Unstable ALDH2 97 42 COc1ccc([C@@H]2CC(=O)Oc3ccc4c(=O)c(-c5ccc(O)cc5)coc4c32)cc1O ZINC000217808792 II In-Stock Unstable IL2 24 41 CCCCCC(=O)N[C@H]1CCC[C@@H]1NC(=O)CCCCC ZINC000217808809 CG On-Demand Unstable LUXR 39 51 CCCCCC(=O)N[C@H]1CCC[C@@H]1NC(=O)CCCCC ZINC000217808809 CG On-Demand Unstable TRAR 17 50 CCCCCC(=O)N[C@H]1CCC[C@@H]1NC(=O)CCCCC ZINC000217808809 CG On-Demand Unstable LASR 70 50 CCCCCC(=O)N[C@H]1CCC[C@@H]1NC(=O)CCCCC ZINC000217808809 CG On-Demand Unstable NOD1 43 37 CCCCCC(=O)N[C@H]1CCC[C@@H]1NC(=O)CCCCC ZINC000217808809 CG On-Demand Unstable CQSS 56 34 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217808831 DG For-Sale Unstable HTR1A 21 52 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217808831 DG For-Sale Unstable DRD2 43 50 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217808831 DG For-Sale Unstable DRD4 44 34 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217808831 DG For-Sale Unstable HTR2A 15 41 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217808831 DG For-Sale Unstable DRD3 40 43 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217808831 DG For-Sale Unstable F10 15 44 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217808831 DG For-Sale Unstable GRIN2B 19 41 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217808831 DG For-Sale Unstable ELANE 15 42 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217808831 DG For-Sale Unstable HCRTR1 24 44 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217808831 DG For-Sale Unstable SIGMAR1 17 43 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217808831 DG For-Sale Unstable PLD1 22 42 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217808831 DG For-Sale Unstable PREP 18 43 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217808831 DG For-Sale Unstable CHRNA10 47 38 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217808831 DG For-Sale Unstable HCRTR2 19 44 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217808831 DG For-Sale Unstable MMP1 31 42 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217808831 DG For-Sale Unstable MCHR1 22 56 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217808831 DG For-Sale Unstable CACNA1I 52 33 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217808831 DG For-Sale Unstable NOD2 25 41 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217808831 DG For-Sale Unstable ACKR3 67 36 COc1ccc(-c2noc(CCC(=O)N3CCN(CCN4CCCC4)CC3)n2)cc1 ZINC000217808833 HD On-Demand Unstable HRH3 39 41 COc1ccc(-c2noc(CCC(=O)N3CCN(CCN4CCCC4)CC3)n2)cc1 ZINC000217808833 HD On-Demand Unstable CPT1A 30 43 C[C@@H](CO)S(=O)(=O)Nc1ccc2c(c1)CCC2 ZINC000217808834 CD For-Sale Unstable MLNR 0 40 O=C(COc1ccccc1)N1CCC[C@H](Cc2nc(C3CC3)no2)C1 ZINC000217808848 EF In-Stock Unstable COLA 156 49 O=C(COc1ccccc1)N1CCC[C@H](Cc2nc(C3CC3)no2)C1 ZINC000217808848 EF In-Stock Unstable CPT1A 128 49 O=C(COc1ccccc1)N1CCC[C@H](Cc2nc(C3CC3)no2)C1 ZINC000217808848 EF In-Stock Unstable CPT2 47 40 CC[C@@H](CCO)NCC(=O)N1CCCC1 ZINC000217808850 BC For-Sale Unstable RIR1_HHV11 47 36 N[C@@H](CC(=O)N[C@H]1CCN2CCCC[C@@H]12)c1ccccc1 ZINC000217808869 CD For-Sale Unstable SIGMAR1 22 48 N[C@@H](CC(=O)N[C@H]1CCN2CCCC[C@@H]12)c1ccccc1 ZINC000217808869 CD For-Sale Unstable SLC18A3 62 36 N[C@@H](CC(=O)N[C@H]1CCN2CCCC[C@@H]12)c1ccccc1 ZINC000217808869 CD For-Sale Unstable METAP2 0 40 COc1ccc([C@H]2CC(=O)Oc3ccc4c(=O)c(-c5ccc(O)cc5)coc4c32)cc1O ZINC000217808874 II In-Stock Unstable ALDH2 97 42 COc1ccc([C@H]2CC(=O)Oc3ccc4c(=O)c(-c5ccc(O)cc5)coc4c32)cc1O ZINC000217808874 II In-Stock Unstable IL2 24 41 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217808908 DG For-Sale Unstable HTR1A 21 52 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217808908 DG For-Sale Unstable DRD2 43 50 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217808908 DG For-Sale Unstable DRD4 44 34 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217808908 DG For-Sale Unstable HTR2A 15 41 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217808908 DG For-Sale Unstable DRD3 40 43 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217808908 DG For-Sale Unstable F10 15 44 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217808908 DG For-Sale Unstable GRIN2B 19 41 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217808908 DG For-Sale Unstable ELANE 15 42 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217808908 DG For-Sale Unstable HCRTR1 24 44 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217808908 DG For-Sale Unstable SIGMAR1 17 43 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217808908 DG For-Sale Unstable PLD1 22 42 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217808908 DG For-Sale Unstable PREP 18 43 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217808908 DG For-Sale Unstable CHRNA10 47 38 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217808908 DG For-Sale Unstable HCRTR2 19 44 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217808908 DG For-Sale Unstable MMP1 31 42 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217808908 DG For-Sale Unstable MCHR1 22 56 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217808908 DG For-Sale Unstable CACNA1I 52 33 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217808908 DG For-Sale Unstable NOD2 25 41 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217808908 DG For-Sale Unstable ACKR3 67 36 O=C(COc1ccccc1)N1CCC[C@@H](Cc2nc(C3CC3)no2)C1 ZINC000217808914 EF In-Stock Unstable COLA 156 49 O=C(COc1ccccc1)N1CCC[C@@H](Cc2nc(C3CC3)no2)C1 ZINC000217808914 EF In-Stock Unstable CPT1A 128 49 O=C(COc1ccccc1)N1CCC[C@@H](Cc2nc(C3CC3)no2)C1 ZINC000217808914 EF In-Stock Unstable CPT2 47 40 CC[C@H](CCO)NCC(=O)N1CCCC1 ZINC000217808915 BC For-Sale Unstable RIR1_HHV11 47 36 C[C@H](CO)S(=O)(=O)Nc1ccc2c(c1)CCC2 ZINC000217808928 CD For-Sale Unstable MLNR 0 40 Cc1cc(NC(=O)c2cc(-c3ccccc3C)nc3c2cnn3C(C)C)ccn1 ZINC000217808936 GJ On-Demand Unstable EZH2 19 40 N[C@H](CC(=O)N[C@H]1CCN2CCCC[C@@H]12)c1ccccc1 ZINC000217808969 CD On-Demand Unstable VACHT_TETCF 0 40 N[C@H](CC(=O)N[C@H]1CCN2CCCC[C@@H]12)c1ccccc1 ZINC000217808969 CD On-Demand Unstable SIGMAR1 0 48 N[C@H](CC(=O)N[C@H]1CCN2CCCC[C@@H]12)c1ccccc1 ZINC000217808969 CD On-Demand Unstable METAP2 0 40 O=C(Cn1cnc(-c2ccccc2)c1)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217808981 FF In-Stock Unstable CPT1A 50 39 O=C(COc1ccc(Cl)cc1Cl)N1CCC[C@H](Cc2nc(C3CC3)no2)C1 ZINC000217809035 HI In-Stock Unstable COLA 24 40 O=C(COc1ccc(Cl)cc1Cl)N1CCC[C@H](Cc2nc(C3CC3)no2)C1 ZINC000217809035 HI In-Stock Unstable CPT1A 23 40 O=C(COc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217809037 DF For-Sale Unstable COLA 119 42 O=C(COc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217809037 DF For-Sale Unstable CPT1A 111 39 O=C(COc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217809037 DF For-Sale Unstable CPT2 45 37 O=C(COc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217809037 DF For-Sale Unstable CHRNA10 61 43 Cc1cc(NC(=O)c2cc(-c3ccc(C)s3)nc3c2cnn3C(C)C)ccn1 ZINC000217809057 GK On-Demand Unstable EZH2 19 41 CSCC[C@@H](CO)NC(=O)CC[C@@H]1NC(=O)N(Cc2ccc3c(c2)OCO3)C1=O ZINC000217809098 HC In-Stock Unstable SSTR3 98 33 CSCC[C@@H](CO)NC(=O)CC[C@@H]1NC(=O)N(Cc2ccc3c(c2)OCO3)C1=O ZINC000217809098 HC In-Stock Unstable MCHR1 22 40 CC(C)C[C@@H](N)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217809102 CD For-Sale Unstable AMPX_VIBPR 0 40 O=C(COc1ccc(Cl)cc1Cl)N1CCC[C@@H](Cc2nc(C3CC3)no2)C1 ZINC000217809127 HI In-Stock Unstable COLA 24 40 O=C(COc1ccc(Cl)cc1Cl)N1CCC[C@@H](Cc2nc(C3CC3)no2)C1 ZINC000217809127 HI In-Stock Unstable CPT1A 23 40 O=C(COc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217809136 DF For-Sale Unstable COLA 119 42 O=C(COc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217809136 DF For-Sale Unstable CPT1A 111 39 O=C(COc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217809136 DF For-Sale Unstable CPT2 45 37 O=C(COc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217809136 DF For-Sale Unstable CHRNA10 61 43 CC(C)NC[C@H](O)CN(C)C(=O)OC(C)(C)C ZINC000217809150 BD In-Stock Unstable ADRB2 32 44 CC(C)C[C@H](N)C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217809163 CD On-Demand Unstable AMPX_VIBPR 0 40 Cn1c(=O)n(CCC(=O)Nc2cc(Br)ccc2N2CCOCC2)c2ccccc21 ZINC000217809202 JF On-Demand Unstable PRKDC 82 36 CC(C)NC[C@@H](O)CN(C)C(=O)OC(C)(C)C ZINC000217809226 BD In-Stock Unstable ADRB2 32 44 CC(C)C[C@@H](N)C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217809256 CD For-Sale Unstable AMPX_VIBPR 0 40 COc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217809258 DG For-Sale Unstable HTR1A 35 52 COc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217809258 DG For-Sale Unstable DRD2 60 59 COc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217809258 DG For-Sale Unstable DRD4 29 46 COc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217809258 DG For-Sale Unstable SLC6A1 29 40 COc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217809258 DG For-Sale Unstable DRD3 52 49 COc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217809258 DG For-Sale Unstable HTR4 46 39 COc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217809258 DG For-Sale Unstable HCRTR1 37 41 COc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217809258 DG For-Sale Unstable KCNA3 56 45 COc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217809258 DG For-Sale Unstable PREP 16 40 COc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217809258 DG For-Sale Unstable HCRTR2 26 41 COc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217809258 DG For-Sale Unstable HCN1 86 46 COc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217809258 DG For-Sale Unstable HCN4 60 44 COc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217809258 DG For-Sale Unstable ACKR3 74 38 COc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217809258 DG For-Sale Unstable KCNK3 34 40 COc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217809258 DG For-Sale Unstable KCNK9 26 40 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc(OC)c2OC(C)C)CC(=O)O4)cc1O ZINC000217809289 KK In-Stock Unstable AKR1B1 0 44 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc(OC)c2OC(C)C)CC(=O)O4)cc1O ZINC000217809289 KK In-Stock Unstable CYP1B1 65 36 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc(OC)c2OC(C)C)CC(=O)O4)cc1O ZINC000217809289 KK In-Stock Unstable CYP1A1 43 43 CC(C)(C)NC[C@H](O)CNC(=O)OC(C)(C)C ZINC000217809335 BD For-Sale Unstable ADRB2 50 44 CC(C)(C)NC[C@H](O)CNC(=O)OC(C)(C)C ZINC000217809335 BD For-Sale Unstable ADRB1 31 43 CC(C)(C)NC[C@H](O)CNC(=O)OC(C)(C)C ZINC000217809335 BD For-Sale Unstable PAPA1_CARPA 43 34 CC(C)(C)NC[C@H](O)CNC(=O)OC(C)(C)C ZINC000217809335 BD For-Sale Unstable CTSK 23 45 CC(C)C[C@H](N)C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217809336 CD On-Demand Unstable AMPX_VIBPR 0 40 COc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217809337 DG For-Sale Unstable HTR1A 35 52 COc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217809337 DG For-Sale Unstable DRD2 60 59 COc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217809337 DG For-Sale Unstable DRD4 29 46 COc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217809337 DG For-Sale Unstable SLC6A1 29 40 COc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217809337 DG For-Sale Unstable DRD3 52 49 COc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217809337 DG For-Sale Unstable HTR4 46 39 COc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217809337 DG For-Sale Unstable HCRTR1 37 41 COc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217809337 DG For-Sale Unstable KCNA3 56 45 COc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217809337 DG For-Sale Unstable PREP 16 40 COc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217809337 DG For-Sale Unstable HCRTR2 26 41 COc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217809337 DG For-Sale Unstable HCN1 86 46 COc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217809337 DG For-Sale Unstable HCN4 60 44 COc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217809337 DG For-Sale Unstable ACKR3 74 38 COc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217809337 DG For-Sale Unstable KCNK3 34 40 COc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217809337 DG For-Sale Unstable KCNK9 26 40 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc(OC)c2OC(C)C)CC(=O)O4)cc1O ZINC000217809378 KK In-Stock Unstable AKR1B1 0 44 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc(OC)c2OC(C)C)CC(=O)O4)cc1O ZINC000217809378 KK In-Stock Unstable CYP1B1 65 36 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc(OC)c2OC(C)C)CC(=O)O4)cc1O ZINC000217809378 KK In-Stock Unstable CYP1A1 43 43 CC(C)(C)NC[C@@H](O)CNC(=O)OC(C)(C)C ZINC000217809412 BD For-Sale Unstable ADRB2 50 44 CC(C)(C)NC[C@@H](O)CNC(=O)OC(C)(C)C ZINC000217809412 BD For-Sale Unstable ADRB1 31 43 CC(C)(C)NC[C@@H](O)CNC(=O)OC(C)(C)C ZINC000217809412 BD For-Sale Unstable PAPA1_CARPA 43 34 CC(C)(C)NC[C@@H](O)CNC(=O)OC(C)(C)C ZINC000217809412 BD For-Sale Unstable CTSK 23 45 CN[C@@H](C)c1ccc(NC(=O)N[C@@H]2CCC[C@@H](C)C2)cc1 ZINC000217809418 CH For-Sale Unstable EPHX2 45 40 COc1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217809466 DG For-Sale Unstable HTR1A 23 56 COc1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217809466 DG For-Sale Unstable DRD2 43 48 COc1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217809466 DG For-Sale Unstable DRD4 61 47 COc1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217809466 DG For-Sale Unstable DRD3 37 56 COc1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217809466 DG For-Sale Unstable OPRD1 17 43 COc1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217809466 DG For-Sale Unstable HCRTR1 17 42 COc1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217809466 DG For-Sale Unstable NQO2 16 40 COc1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217809466 DG For-Sale Unstable SIGMAR1 15 43 COc1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217809466 DG For-Sale Unstable MMP13 15 45 COc1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217809466 DG For-Sale Unstable CCR3 24 45 COc1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217809466 DG For-Sale Unstable PREP 26 41 COc1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217809466 DG For-Sale Unstable MTNR1A 52 42 COc1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217809466 DG For-Sale Unstable MTNR1B 56 47 COc1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217809466 DG For-Sale Unstable CHRNA10 68 45 COc1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217809466 DG For-Sale Unstable MCHR1 25 48 COc1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217809466 DG For-Sale Unstable CACNA1I 50 39 COc1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217809466 DG For-Sale Unstable ACKR3 72 40 COc1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217809466 DG For-Sale Unstable KCNK3 17 45 Cn1c(=O)n(C)c2cc(NC(=O)CC[C@@H]3NC(=O)c4ccccc4NC3=O)ccc21 ZINC000217809469 HD In-Stock Unstable BRPF1 0 41 CC(C)[C@@H]1CN(c2cnc3cc(F)c(F)cc3n2)CCN1 ZINC000217809476 CE For-Sale Unstable PRKCQ 24 42 CN[C@@H](C)c1ccc(NC(=O)N[C@H]2CCC[C@@H](C)C2)cc1 ZINC000217809495 CH For-Sale Unstable EPHX2 45 40 O=C(NCC1(c2ccccc2)CCCC1)c1cnc[nH]1 ZINC000217809530 CF In-Stock Unstable KCNA3 43 45 O=C(NCC1(c2ccccc2)CCCC1)c1cnc[nH]1 ZINC000217809530 CF In-Stock Unstable ACAT 0 54 CC(C)[C@H]1CN(c2cnc3cc(F)c(F)cc3n2)CCN1 ZINC000217809545 CE On-Demand Unstable PRKCQ 24 42 COc1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217809546 DG For-Sale Unstable HTR1A 23 56 COc1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217809546 DG For-Sale Unstable DRD2 43 48 COc1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217809546 DG For-Sale Unstable DRD4 61 47 COc1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217809546 DG For-Sale Unstable DRD3 37 56 COc1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217809546 DG For-Sale Unstable OPRD1 17 43 COc1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217809546 DG For-Sale Unstable HCRTR1 17 42 COc1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217809546 DG For-Sale Unstable NQO2 16 40 COc1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217809546 DG For-Sale Unstable SIGMAR1 15 43 COc1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217809546 DG For-Sale Unstable MMP13 15 45 COc1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217809546 DG For-Sale Unstable CCR3 24 45 COc1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217809546 DG For-Sale Unstable PREP 26 41 COc1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217809546 DG For-Sale Unstable MTNR1A 52 42 COc1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217809546 DG For-Sale Unstable MTNR1B 56 47 COc1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217809546 DG For-Sale Unstable CHRNA10 68 45 COc1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217809546 DG For-Sale Unstable MCHR1 25 48 COc1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217809546 DG For-Sale Unstable CACNA1I 50 39 COc1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217809546 DG For-Sale Unstable ACKR3 72 40 COc1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217809546 DG For-Sale Unstable KCNK3 17 45 COC(=O)[C@@H]1Cc2ccccc2CN1C(=O)c1cc(-c2ccccc2C)nc2c1cnn2C(C)C ZINC000217809562 JJ On-Demand Unstable OPRM1 23 44 COC(=O)[C@@H]1Cc2ccccc2CN1C(=O)c1cc(-c2ccccc2C)nc2c1cnn2C(C)C ZINC000217809562 JJ On-Demand Unstable OPRD1 66 35 COC(=O)[C@@H]1Cc2ccccc2CN1C(=O)c1cc(-c2ccccc2C)nc2c1cnn2C(C)C ZINC000217809562 JJ On-Demand Unstable CFTR 57 35 COC(=O)[C@@H]1Cc2ccccc2CN1C(=O)c1cc(-c2ccccc2C)nc2c1cnn2C(C)C ZINC000217809562 JJ On-Demand Unstable BCL2 0 40 COC(=O)COc1ccc2occ(-c3cc4ccccc4o3)c2c1 ZINC000217809597 DI In-Stock Unstable ALDH2 55 38 CN[C@@H](C)c1cccc(NC(=O)N[C@@H]2CCC[C@@H](C)C2)c1 ZINC000217809603 CH For-Sale Unstable EPHX2 31 44 COC(=O)[C@H]1Cc2ccccc2CN1C(=O)c1cc(-c2ccccc2C)nc2c1cnn2C(C)C ZINC000217809634 JJ On-Demand Unstable OPRM1 23 44 COC(=O)[C@H]1Cc2ccccc2CN1C(=O)c1cc(-c2ccccc2C)nc2c1cnn2C(C)C ZINC000217809634 JJ On-Demand Unstable OPRD1 66 35 COC(=O)[C@H]1Cc2ccccc2CN1C(=O)c1cc(-c2ccccc2C)nc2c1cnn2C(C)C ZINC000217809634 JJ On-Demand Unstable CFTR 57 35 COC(=O)[C@H]1Cc2ccccc2CN1C(=O)c1cc(-c2ccccc2C)nc2c1cnn2C(C)C ZINC000217809634 JJ On-Demand Unstable BCL2 0 40 Cn1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1=O ZINC000217809644 DD In-Stock Unstable HCRTR1 30 42 Cn1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1=O ZINC000217809644 DD In-Stock Unstable HCRTR2 28 42 Cn1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1=O ZINC000217809644 DD In-Stock Unstable HCN1 42 30 Cc1cc(C(=O)N[C@@H]2CCN3CCCC[C@@H]23)ccc1N ZINC000217809649 CD On-Demand Unstable SIGMAR1 0 43 Cc1cc(C(=O)N[C@@H]2CCN3CCCC[C@@H]23)ccc1N ZINC000217809649 CD On-Demand Unstable L3MBTL3 64 37 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)Nc3ccc(O)cc3)[C@H]21 ZINC000217809676 JH In-Stock Unstable TSHR 65 36 CN[C@@H](C)c1cccc(NC(=O)N[C@H]2CCC[C@@H](C)C2)c1 ZINC000217809686 CH For-Sale Unstable EPHX2 31 44 C[C@@H](CNC(=O)[C@@H]1CCC[C@@H]1C(=O)O)N(C)C1CC1 ZINC000217809707 CD For-Sale Unstable ACE 23 43 Cn1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1=O ZINC000217809708 DD In-Stock Unstable HCRTR1 30 42 Cn1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1=O ZINC000217809708 DD In-Stock Unstable HCRTR2 28 42 Cn1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1=O ZINC000217809708 DD In-Stock Unstable HCN1 42 30 Cc1cc(C(=O)N[C@H]2CCN3CCCC[C@@H]23)ccc1N ZINC000217809729 CD On-Demand Unstable SIGMAR1 0 43 Cc1cc(C(=O)N[C@H]2CCN3CCCC[C@@H]23)ccc1N ZINC000217809729 CD On-Demand Unstable L3MBTL3 64 37 CCCCCNC(=O)N/C=C/c1ccccc1Cl ZINC000217809749 CH For-Sale Unstable EPHX2 25 42 CCCCCNC(=O)N/C=C/c1ccccc1Cl ZINC000217809749 CH For-Sale Unstable ASAH1 60 37 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)Nc3ccc(O)cc3)[C@@H]21 ZINC000217809752 JH In-Stock Unstable TSHR 65 36 C[C@H](N)c1cccc(NC(=O)N[C@@H]2CCC[C@@H](C)C2)c1 ZINC000217809771 CG For-Sale Unstable EPHX2 35 48 COc1ccc(O)c(C(=O)Nc2nc3c(OC)cccc3s2)c1 ZINC000217809772 EG On-Demand Unstable ACE 17 40 COc1ccc(O)c(C(=O)Nc2nc3c(OC)cccc3s2)c1 ZINC000217809772 EG On-Demand Unstable ADORA2B 28 41 COc1ccc(O)c(C(=O)Nc2nc3c(OC)cccc3s2)c1 ZINC000217809772 EG On-Demand Unstable TRPV1 20 40 COc1ccc(O)c(C(=O)Nc2nc3c(OC)cccc3s2)c1 ZINC000217809772 EG On-Demand Unstable CSNK1D 33 44 COc1ccc(O)c(C(=O)Nc2nc3c(OC)cccc3s2)c1 ZINC000217809772 EG On-Demand Unstable LUCI_LUCLA 16 40 COc1ccc(O)c(C(=O)Nc2nc3c(OC)cccc3s2)c1 ZINC000217809772 EG On-Demand Unstable KCNK3 41 41 COc1ccc(O)c(C(=O)Nc2nc3c(OC)cccc3s2)c1 ZINC000217809772 EG On-Demand Unstable KCNK9 41 41 O=C(Cc1cccs1)N1CCC[C@H](Cc2nc(C3CC3)no2)C1 ZINC000217809776 EG In-Stock Unstable ETHR 45 51 C[C@H](CNC(=O)[C@@H]1CCC[C@@H]1C(=O)O)N(C)C1CC1 ZINC000217809813 CD For-Sale Unstable ACE 23 43 O=C(N/C=C/c1ccccc1Cl)Nc1ccccc1 ZINC000217809826 CI For-Sale Anodyne EPHX1 0 48 O=C(N/C=C/c1ccccc1Cl)Nc1ccccc1 ZINC000217809826 CI For-Sale Anodyne LPL 43 34 O=C(N/C=C/c1ccccc1Cl)Nc1ccccc1 ZINC000217809826 CI For-Sale Anodyne SMO 16 43 O=C(N/C=C/c1ccccc1Cl)Nc1ccccc1 ZINC000217809826 CI For-Sale Anodyne P95276_MYCTO 0 48 O=C(N/C=C/c1ccccc1Cl)Nc1ccccc1 ZINC000217809826 CI For-Sale Anodyne KCNK3 21 40 COc1nn(C)cc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217809831 DD For-Sale Unstable DRD2 40 45 COc1nn(C)cc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217809831 DD For-Sale Unstable DRD3 22 44 COc1nn(C)cc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217809831 DD For-Sale Unstable ACKR3 53 33 C[C@H](N)c1cccc(NC(=O)N[C@H]2CCC[C@@H](C)C2)c1 ZINC000217809848 CG For-Sale Unstable EPHX2 35 48 O=C(Cc1cccs1)N1CCC[C@@H](Cc2nc(C3CC3)no2)C1 ZINC000217809853 EG In-Stock Unstable ETHR 45 51 COc1nn(C)cc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217809903 DD For-Sale Unstable DRD2 40 45 COc1nn(C)cc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217809903 DD For-Sale Unstable DRD3 22 44 COc1nn(C)cc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217809903 DD For-Sale Unstable ACKR3 53 33 CCOC(=O)[C@@H]1CCCN(C(=O)N/C=C/c2ccccc2Cl)C1 ZINC000217809947 EG For-Sale Unstable SLC6A1 88 39 CCOC(=O)[C@@H]1CCCN(C(=O)N/C=C/c2ccccc2Cl)C1 ZINC000217809947 EG For-Sale Unstable FDFT1 29 43 C[C@H](N)c1ccc(NC(=O)N[C@@H]2CCC[C@@H](C)C2)cc1 ZINC000217809951 CG For-Sale Unstable EPHX2 50 43 CC(=O)NCCCc1ccc(-c2csc(NC(=O)c3c(C)nn(C)c3C)n2)cc1 ZINC000217809962 HG On-Demand Unstable ROCK1 20 41 CC(=O)NCCCc1ccc(-c2csc(NC(=O)c3c(C)nn(C)c3C)n2)cc1 ZINC000217809962 HG On-Demand Unstable SPHK2 41 34 O=C(CCc1ccccc1)N1CCC[C@H](Cc2nc(C3CC3)no2)C1 ZINC000217809963 EG In-Stock Unstable PREP 43 38 O=C(CCc1ccccc1)N1CCC[C@H](Cc2nc(C3CC3)no2)C1 ZINC000217809963 EG In-Stock Unstable ETHR 45 36 C[C@H](CNC(=O)[C@H]1CCC[C@@H]1C(=O)O)N(C)C1CC1 ZINC000217809990 CD For-Sale Unstable ACE 23 43 O=C(CCc1ccccc1)N1CCC[C@@H](Cc2nc(C3CC3)no2)C1 ZINC000217810018 EG In-Stock Unstable PREP 43 38 O=C(CCc1ccccc1)N1CCC[C@@H](Cc2nc(C3CC3)no2)C1 ZINC000217810018 EG In-Stock Unstable ETHR 45 36 O=C(CCC1CCCCC1)NC[C@H]1CCCN1c1ccccc1 ZINC000217810019 DI For-Sale Unstable CHRM4 21 46 O=C(CCC1CCCCC1)NC[C@H]1CCCN1c1ccccc1 ZINC000217810019 DI For-Sale Unstable CHRM5 20 46 O=C(CCC1CCCCC1)NC[C@H]1CCCN1c1ccccc1 ZINC000217810019 DI For-Sale Unstable PREP 20 42 C[C@H](N)c1ccc(NC(=O)N[C@H]2CCC[C@@H](C)C2)cc1 ZINC000217810027 CG For-Sale Unstable EPHX2 50 43 CCOC(=O)[C@H]1CCCN(C(=O)N/C=C/c2ccccc2Cl)C1 ZINC000217810034 EG For-Sale Unstable SLC6A1 88 39 CCOC(=O)[C@H]1CCCN(C(=O)N/C=C/c2ccccc2Cl)C1 ZINC000217810034 EG For-Sale Unstable FDFT1 29 43 COC(=O)C[C@H](c1ccc(OC)c(OC)c1)c1c(O)c2ccccc2oc1=O ZINC000217810041 GG In-Stock Unstable TNF 22 41 COC(=O)C[C@H](c1ccc(OC)c(OC)c1)c1c(O)c2ccccc2oc1=O ZINC000217810041 GG In-Stock Unstable NQO1 65 54 C[C@@H](O)[C@@H](C)Sc1ccc(S(=O)(=O)N(C)C)cc1[N+](=O)[O-] ZINC000217810078 ED On-Demand Unstable COLA 66 36 O=C(CCC1CCCCC1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217810100 DI For-Sale Unstable CHRM4 21 46 O=C(CCC1CCCCC1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217810100 DI For-Sale Unstable CHRM5 20 46 O=C(CCC1CCCCC1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217810100 DI For-Sale Unstable PREP 20 42 COC(=O)C[C@@H](c1ccc(OC)c(OC)c1)c1c(O)c2ccccc2oc1=O ZINC000217810113 GG In-Stock Unstable TNF 22 41 COC(=O)C[C@@H](c1ccc(OC)c(OC)c1)c1c(O)c2ccccc2oc1=O ZINC000217810113 GG In-Stock Unstable NQO1 65 54 O=C(O)Cc1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217810136 EH For-Sale Unstable SMO 16 51 C[C@H](O)[C@@H](C)Sc1ccc(S(=O)(=O)N(C)C)cc1[N+](=O)[O-] ZINC000217810148 ED On-Demand Unstable COLA 66 36 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1 ZINC000217810235 DH For-Sale Unstable DRD2 30 45 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1 ZINC000217810235 DH For-Sale Unstable DRD4 24 44 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1 ZINC000217810235 DH For-Sale Unstable SLC6A1 15 42 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1 ZINC000217810235 DH For-Sale Unstable HRH1 24 41 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1 ZINC000217810235 DH For-Sale Unstable DRD3 21 44 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1 ZINC000217810235 DH For-Sale Unstable F10 22 42 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1 ZINC000217810235 DH For-Sale Unstable CCR1 33 40 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1 ZINC000217810235 DH For-Sale Unstable PLD1 44 39 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1 ZINC000217810235 DH For-Sale Unstable PREP 17 43 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1 ZINC000217810235 DH For-Sale Unstable CACNA1I 62 36 C[C@H](Sc1ccc(S(=O)(=O)N(C)C)cc1[N+](=O)[O-])[C@@H](C)O ZINC000217810246 ED On-Demand Unstable COLA 66 36 CC(=O)NCCCc1ccc(-c2csc(NC(=O)CCc3nc(-c4ccncc4)no3)n2)cc1 ZINC000217810265 JH On-Demand Unstable ROCK1 23 46 CC(=O)NCCCc1ccc(-c2csc(NC(=O)CCc3nc(-c4ccncc4)no3)n2)cc1 ZINC000217810265 JH On-Demand Unstable ROCK2 16 41 CC(=O)NCCCc1ccc(-c2csc(NC(=O)CCc3nc(-c4ccncc4)no3)n2)cc1 ZINC000217810265 JH On-Demand Unstable HDAC9 15 42 CC(=O)NCCCc1ccc(-c2csc(NC(=O)CCc3nc(-c4ccncc4)no3)n2)cc1 ZINC000217810265 JH On-Demand Unstable HCAR2 20 40 CN(CC(=O)NCc1nnnn1-c1ccccc1)Cc1ccncc1 ZINC000217810270 EC In-Stock Unstable DAGLA 18 42 C[C@H](O)[C@H](C)Sc1ccc(S(=O)(=O)N(C)C)cc1[N+](=O)[O-] ZINC000217810324 ED On-Demand Unstable COLA 66 36 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1 ZINC000217810326 DH For-Sale Unstable DRD2 30 45 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1 ZINC000217810326 DH For-Sale Unstable DRD4 24 44 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1 ZINC000217810326 DH For-Sale Unstable SLC6A1 15 42 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1 ZINC000217810326 DH For-Sale Unstable HRH1 24 41 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1 ZINC000217810326 DH For-Sale Unstable DRD3 21 44 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1 ZINC000217810326 DH For-Sale Unstable F10 22 42 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1 ZINC000217810326 DH For-Sale Unstable CCR1 33 40 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1 ZINC000217810326 DH For-Sale Unstable PLD1 44 39 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1 ZINC000217810326 DH For-Sale Unstable PREP 17 43 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1 ZINC000217810326 DH For-Sale Unstable CACNA1I 62 36 Cc1ccccc1[C@H](CC(=O)O)NC(=O)c1ccnc(Cl)c1 ZINC000217810338 DF Annotated Unstable MME 0 45 Cc1ccccc1[C@H](CC(=O)O)NC(=O)c1ccnc(Cl)c1 ZINC000217810338 DF Annotated Unstable UTS2 61 38 Cc1ccccc1[C@H](CC(=O)O)NC(=O)c1ccnc(Cl)c1 ZINC000217810338 DF Annotated Unstable CTSA 119 52 CCCCCO[C@]1(C(F)(F)F)Oc2ccccc2C=C1C(=O)O ZINC000217810388 EI In-Stock Unstable PLA2G4B 44 33 COc1cc2c(cc1OC)CN(Cc1oc(CN3CCOCC3)cc(=O)c1O)CC2 ZINC000217810395 HD In-Stock Unstable ABCB1B 62 36 COc1cc2c(cc1OC)CN(Cc1oc(CN3CCOCC3)cc(=O)c1O)CC2 ZINC000217810395 HD In-Stock Unstable ABCB1 22 47 CCCCCO[C@@]1(C(F)(F)F)Oc2ccccc2C=C1C(=O)O ZINC000217810459 EI In-Stock Unstable PLA2G4B 44 33 CO[C@@H]1[C@H]2CC[C@@H]1CN(C(=O)CCC(=O)c1ccc(F)cc1)C2 ZINC000217810461 DF In-Stock Unstable HRH3 0 51 Cc1onc(-c2ccccc2Cl)c1C(=O)N1CCC[C@H](Cc2nc(C3CC3)no2)C1 ZINC000217810485 IJ In-Stock Unstable GPBAR1 28 40 COc1cn(CC(=O)N2CCc3ccccc3C2)c(C)cc1=O ZINC000217810518 DD In-Stock Unstable ABCB1B 40 33 Cc1onc(-c2ccccc2Cl)c1C(=O)N1CCC[C@@H](Cc2nc(C3CC3)no2)C1 ZINC000217810569 IJ In-Stock Unstable GPBAR1 28 40 CC(C)(C)OC(=O)N[C@H](O)CCC(=O)O ZINC000217810632 BC For-Sale Unstable PAPA1_CARPA 49 44 CC(C)(C)OC(=O)N[C@H](O)CCC(=O)O ZINC000217810632 BC For-Sale Unstable CTSK 25 47 CC(C)(C)OC(=O)N[C@H](O)CCC(=O)O ZINC000217810632 BC For-Sale Unstable PGA5 44 39 CC(C)(C)OC(=O)N[C@H](O)CCC(=O)O ZINC000217810632 BC For-Sale Unstable POLG_HCV1 25 50 CC(C)(C)OC(=O)N[C@H](O)CCC(=O)O ZINC000217810632 BC For-Sale Unstable POL 0 45 CC(C)(C)OC(=O)N[C@H](O)CCC(=O)O ZINC000217810632 BC For-Sale Unstable SSPA 0 43 O=C(NC[C@H]1CCCN1c1ccccc1)c1cc2ccccc2o1 ZINC000217810665 DH For-Sale Unstable DRD3 15 41 CC(C)(C)OC(=O)N[C@@H](O)CCC(=O)O ZINC000217810718 BC For-Sale Unstable PAPA1_CARPA 49 44 CC(C)(C)OC(=O)N[C@@H](O)CCC(=O)O ZINC000217810718 BC For-Sale Unstable CTSK 25 47 CC(C)(C)OC(=O)N[C@@H](O)CCC(=O)O ZINC000217810718 BC For-Sale Unstable PGA5 44 39 CC(C)(C)OC(=O)N[C@@H](O)CCC(=O)O ZINC000217810718 BC For-Sale Unstable POLG_HCV1 25 50 CC(C)(C)OC(=O)N[C@@H](O)CCC(=O)O ZINC000217810718 BC For-Sale Unstable POL 0 45 CC(C)(C)OC(=O)N[C@@H](O)CCC(=O)O ZINC000217810718 BC For-Sale Unstable SSPA 0 43 NC(=O)[C@@H]1CCCN(C(=O)CN2CCC[C@H](C(=O)O)C2)C1 ZINC000217810743 CB For-Sale Unstable SLC6A1 151 42 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cc2ccccc2o1 ZINC000217810746 DH For-Sale Unstable DRD3 15 41 CC1(C)CC(NC(=O)N/C=C/c2ccccc2Cl)CC(C)(C)N1 ZINC000217810753 EH For-Sale Unstable VATB 0 43 CC1(C)CC(NC(=O)N/C=C/c2ccccc2Cl)CC(C)(C)N1 ZINC000217810753 EH For-Sale Unstable ENV 33 42 CC1(C)CC(NC(=O)N/C=C/c2ccccc2Cl)CC(C)(C)N1 ZINC000217810753 EH For-Sale Unstable EZH2 54 41 CC1(C)CC(NC(=O)N/C=C/c2ccccc2Cl)CC(C)(C)N1 ZINC000217810753 EH For-Sale Unstable HIV1_ENV 0 44 COc1ccccc1-c1n[nH]cc1C(=O)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217810824 FG In-Stock Unstable HTR4 21 49 COc1ccccc1-c1n[nH]cc1C(=O)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217810824 FG In-Stock Unstable HCN1 74 36 COc1ccccc1-c1n[nH]cc1C(=O)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217810824 FG In-Stock Unstable HCN4 54 36 Cc1ccc(O)c(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217810853 DI For-Sale Unstable KCNMA1 18 41 COc1ccc(N(Cc2ccccc2)C(=O)CCn2c(=O)n(C)c3ccccc32)cc1 ZINC000217810942 HH On-Demand Unstable CMA1 19 40 O=C(N/C=C/c1ccccc1Cl)N1CCN(CCO)CC1 ZINC000217810948 DD For-Sale Unstable DRD3 21 40 CO[C@@H]1CCOC[C@H]1Nc1ccnc2ccc(Cl)cc12 ZINC000217811018 CG In-Stock Unstable HRP1_PLAFA 67 36 CO[C@@H]1CCOC[C@H]1Nc1ccnc2ccc(Cl)cc12 ZINC000217811018 CG In-Stock Unstable HNMT 45 31 CN(C)c1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217811028 DG For-Sale Unstable DRD3 15 40 CN(C)c1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217811028 DG For-Sale Unstable ACKR3 54 35 C[C@@H]1CCCN(C(=O)N/C=C/c2ccccc2Cl)C1 ZINC000217811046 CH For-Sale Unstable SLC6A1 46 37 COc1ccc(-c2nnc(S[C@@H](C(N)=O)c3ccc(F)cc3)n2Cc2ccco2)cc1 ZINC000217811075 II On-Demand Unstable HCRTR2 22 51 CN(C)c1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217811102 DG For-Sale Unstable DRD3 15 40 CN(C)c1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217811102 DG For-Sale Unstable ACKR3 54 35 C[C@H]1CCCN(C(=O)N/C=C/c2ccccc2Cl)C1 ZINC000217811115 CH For-Sale Unstable SLC6A1 46 37 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)Nc1cc(Cl)ccc1O)C(=O)OC2 ZINC000217811119 JJ In-Stock Unstable IMPDH1 0 68 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)Nc1cc(Cl)ccc1O)C(=O)OC2 ZINC000217811119 JJ In-Stock Unstable IMPDH2 0 68 C[C@H](N)c1cccc(NC(=O)N2C[C@@H](C)OC[C@@H]2C)c1 ZINC000217811121 CE For-Sale Unstable LIMK2 32 40 COc1ccc(-c2nnc(S[C@H](C(N)=O)c3ccc(F)cc3)n2Cc2ccco2)cc1 ZINC000217811155 II On-Demand Unstable HCRTR2 22 51 C[C@H]1CN(C(=O)Nc2cccc([C@H](C)N)c2)[C@@H](C)CO1 ZINC000217811206 CE For-Sale Unstable LIMK2 32 40 CN(C)c1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217811241 DG For-Sale Unstable HCRTR1 15 42 CN(C)c1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217811241 DG For-Sale Unstable PREP 21 41 CN(C)c1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217811241 DG For-Sale Unstable CACNA1I 45 37 CN(C)c1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217811241 DG For-Sale Unstable ACKR3 62 34 CN(C)c1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217811317 DG For-Sale Unstable HCRTR1 15 42 CN(C)c1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217811317 DG For-Sale Unstable PREP 21 41 CN(C)c1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217811317 DG For-Sale Unstable CACNA1I 45 37 CN(C)c1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217811317 DG For-Sale Unstable ACKR3 62 34 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)Nc3ccc4cc[nH]c4c3)[C@H]21 ZINC000217811335 JH In-Stock Unstable TSHR 50 33 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)Nc3ccc4cc[nH]c4c3)[C@H]21 ZINC000217811335 JH In-Stock Unstable ENPP1 60 33 CCN(Cc1ccccc1)C(=O)N/C=C/c1ccccc1Cl ZINC000217811338 DJ For-Sale Unstable TSPO 20 42 COc1ccc(-c2nnc(S[C@@H]3CCCCNC3=O)n2-c2ccc(Cl)cc2)cc1 ZINC000217811391 II On-Demand Unstable VCP 62 39 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc2c(c1)OCO2 ZINC000217811417 DF In-Stock Unstable NOS2 83 39 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)Nc3ccc4cc[nH]c4c3)[C@@H]21 ZINC000217811421 JH In-Stock Unstable TSHR 50 33 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)Nc3ccc4cc[nH]c4c3)[C@@H]21 ZINC000217811421 JH In-Stock Unstable ENPP1 60 33 COc1ccc(-c2nnc(S[C@H]3CCCCNC3=O)n2-c2ccc(Cl)cc2)cc1 ZINC000217811468 II On-Demand Unstable VCP 62 39 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc2c(c1)OCO2 ZINC000217811498 DF In-Stock Unstable NOS2 83 39 CCCCCCCCOc1ccc([C@H](CC(=O)OC)C2=C(O)C(=O)c3ccccc3C2=O)cc1 ZINC000217811552 JK In-Stock Unstable THRA 40 36 CCCCCCCCOc1ccc([C@H](CC(=O)OC)C2=C(O)C(=O)c3ccccc3C2=O)cc1 ZINC000217811552 JK In-Stock Unstable PLA2G4B 98 40 CCCCCCCCOc1ccc([C@H](CC(=O)OC)C2=C(O)C(=O)c3ccccc3C2=O)cc1 ZINC000217811552 JK In-Stock Unstable FAAH 23 44 COc1ccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217811591 DG For-Sale Unstable HTR1A 15 43 COc1ccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217811591 DG For-Sale Unstable DRD2 40 41 COc1ccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217811591 DG For-Sale Unstable HRH1 22 41 COc1ccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217811591 DG For-Sale Unstable DRD3 23 42 COc1ccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217811591 DG For-Sale Unstable SIGMAR1 30 51 COc1ccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217811591 DG For-Sale Unstable MMP13 45 40 COc1ccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217811591 DG For-Sale Unstable CCR3 26 40 COc1ccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217811591 DG For-Sale Unstable NOS2 24 42 COc1ccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217811591 DG For-Sale Unstable MTNR1A 51 36 COc1ccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217811591 DG For-Sale Unstable MTNR1B 46 36 COc1ccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217811591 DG For-Sale Unstable MMP3 42 38 COc1ccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217811591 DG For-Sale Unstable MMP8 22 40 COc1ccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217811591 DG For-Sale Unstable MMP12 17 40 COc1ccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217811591 DG For-Sale Unstable CHRNA10 43 37 COc1ccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217811591 DG For-Sale Unstable CA9 16 40 COc1ccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217811591 DG For-Sale Unstable MMP1 49 38 COc1ccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217811591 DG For-Sale Unstable MCHR1 28 43 COc1ccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217811591 DG For-Sale Unstable MBTPS1 49 35 COc1ccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217811591 DG For-Sale Unstable ACKR3 51 33 CC[C@@H]1CCCCN1C(=O)N/C=C/c1ccccc1Cl ZINC000217811622 CI For-Sale Unstable ABHD11 0 41 CCCCCCCCOc1ccc([C@@H](CC(=O)OC)C2=C(O)C(=O)c3ccccc3C2=O)cc1 ZINC000217811636 JK In-Stock Unstable THRA 40 36 CCCCCCCCOc1ccc([C@@H](CC(=O)OC)C2=C(O)C(=O)c3ccccc3C2=O)cc1 ZINC000217811636 JK In-Stock Unstable PLA2G4B 98 40 CCCCCCCCOc1ccc([C@@H](CC(=O)OC)C2=C(O)C(=O)c3ccccc3C2=O)cc1 ZINC000217811636 JK In-Stock Unstable FAAH 23 44 COc1ccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217811675 DG For-Sale Unstable HTR1A 15 43 COc1ccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217811675 DG For-Sale Unstable DRD2 40 41 COc1ccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217811675 DG For-Sale Unstable HRH1 22 41 COc1ccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217811675 DG For-Sale Unstable DRD3 23 42 COc1ccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217811675 DG For-Sale Unstable SIGMAR1 30 51 COc1ccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217811675 DG For-Sale Unstable MMP13 45 40 COc1ccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217811675 DG For-Sale Unstable CCR3 26 40 COc1ccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217811675 DG For-Sale Unstable NOS2 24 42 COc1ccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217811675 DG For-Sale Unstable MTNR1A 51 36 COc1ccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217811675 DG For-Sale Unstable MTNR1B 46 36 COc1ccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217811675 DG For-Sale Unstable MMP3 42 38 COc1ccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217811675 DG For-Sale Unstable MMP8 22 40 COc1ccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217811675 DG For-Sale Unstable MMP12 17 40 COc1ccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217811675 DG For-Sale Unstable CHRNA10 43 37 COc1ccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217811675 DG For-Sale Unstable CA9 16 40 COc1ccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217811675 DG For-Sale Unstable MMP1 49 38 COc1ccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217811675 DG For-Sale Unstable MCHR1 28 43 COc1ccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217811675 DG For-Sale Unstable MBTPS1 49 35 COc1ccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217811675 DG For-Sale Unstable ACKR3 51 33 C[C@@H](Cc1cccc(Cl)c1)NC(=O)[C@@H]1C[C@@H](O)CN1 ZINC000217811687 CD For-Sale Unstable CTSC 24 43 CC[C@H]1CCCCN1C(=O)N/C=C/c1ccccc1Cl ZINC000217811698 CI For-Sale Unstable ABHD11 0 41 COc1ccc([C@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c(OC)c1OC ZINC000217811742 KH In-Stock Unstable CYP1B1 68 43 COc1ccc([C@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c(OC)c1OC ZINC000217811742 KH In-Stock Unstable CYP1A1 50 43 COc1ccc([C@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c(OC)c1OC ZINC000217811742 KH In-Stock Unstable CYP1A2 42 43 CSc1ccc(-c2csc(NC(=O)c3cc(-c4ccco4)on3)n2)cc1 ZINC000217811746 GK On-Demand Unstable MPL 65 38 C[C@H](Cc1cccc(Cl)c1)NC(=O)[C@@H]1C[C@@H](O)CN1 ZINC000217811764 CD For-Sale Unstable CTSC 24 43 CCOc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217811788 DG For-Sale Unstable DRD2 41 43 CCOc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217811788 DG For-Sale Unstable DRD3 18 41 CCOc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217811788 DG For-Sale Unstable HTR4 43 33 CCOc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217811788 DG For-Sale Unstable HCRTR1 34 40 CCOc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217811788 DG For-Sale Unstable KCNA3 43 45 CCOc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217811788 DG For-Sale Unstable HCRTR2 26 40 CCOc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217811788 DG For-Sale Unstable HCN1 100 49 CCOc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217811788 DG For-Sale Unstable HCN4 73 49 CCOc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217811788 DG For-Sale Unstable ACKR3 63 34 CCOc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217811788 DG For-Sale Unstable KCNK3 32 41 CCOc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217811788 DG For-Sale Unstable KCNK9 24 41 COc1cccc(CN2CCN(C(=O)Cn3nc(C)cc3N)CC2=O)c1 ZINC000217811795 FC In-Stock Unstable FPR2 23 44 COc1ccc([C@@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c(OC)c1OC ZINC000217811814 KH In-Stock Unstable CYP1B1 68 43 COc1ccc([C@@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c(OC)c1OC ZINC000217811814 KH In-Stock Unstable CYP1A1 50 43 COc1ccc([C@@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c(OC)c1OC ZINC000217811814 KH In-Stock Unstable CYP1A2 42 43 C[C@@H](Cc1cccc(Cl)c1)NC(=O)[C@H]1C[C@@H](O)CN1 ZINC000217811836 CD For-Sale Unstable CTSC 24 43 C[C@@H](Cc1cccc(Cl)c1)NC(=O)[C@H]1C[C@@H](O)CN1 ZINC000217811836 CD For-Sale Unstable LMGT2 0 44 CNC(=O)[C@@H]1CCCCN1[C@@H](C)c1ccc(OC)cc1O ZINC000217811842 CE For-Sale Unstable MMP13 16 43 CNC(=O)[C@@H]1CCCCN1[C@@H](C)c1ccc(OC)cc1O ZINC000217811842 CE For-Sale Unstable MMP3 22 43 CNC(=O)[C@@H]1CCCCN1[C@@H](C)c1ccc(OC)cc1O ZINC000217811842 CE For-Sale Unstable MMP7 21 41 CNC(=O)[C@@H]1CCCCN1[C@@H](C)c1ccc(OC)cc1O ZINC000217811842 CE For-Sale Unstable MMP1 20 43 C[C@H]1CCCC[C@H]1OC[C@@H](O)CN[C@H](C)c1ccccn1 ZINC000217811872 CF For-Sale Unstable ADRB2 47 43 C[C@H]1CCCC[C@H]1OC[C@@H](O)CN[C@H](C)c1ccccn1 ZINC000217811872 CF For-Sale Unstable ADRB1 26 40 CCOc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217811883 DG For-Sale Unstable DRD2 41 43 CCOc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217811883 DG For-Sale Unstable DRD3 18 41 CCOc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217811883 DG For-Sale Unstable HTR4 43 33 CCOc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217811883 DG For-Sale Unstable HCRTR1 34 40 CCOc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217811883 DG For-Sale Unstable KCNA3 43 45 CCOc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217811883 DG For-Sale Unstable HCRTR2 26 40 CCOc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217811883 DG For-Sale Unstable HCN1 100 49 CCOc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217811883 DG For-Sale Unstable HCN4 73 49 CCOc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217811883 DG For-Sale Unstable ACKR3 63 34 CCOc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217811883 DG For-Sale Unstable KCNK3 32 41 CCOc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217811883 DG For-Sale Unstable KCNK9 24 41 C[C@H](Cc1cccc(Cl)c1)NC(=O)[C@H]1C[C@@H](O)CN1 ZINC000217811920 CD For-Sale Unstable CTSC 24 43 O=C(Cc1cc2c(cc1Cl)OCCO2)NCCc1ccncc1 ZINC000217811931 EE In-Stock Unstable CA5B 18 47 O=C(Cc1cc2c(cc1Cl)OCCO2)NCCc1ccncc1 ZINC000217811931 EE In-Stock Unstable CA5A 15 47 O=C(Cc1cc2c(cc1Cl)OCCO2)NCCc1ccncc1 ZINC000217811931 EE In-Stock Unstable NCE103 25 45 O=C(Cc1cc2c(cc1Cl)OCCO2)NCCc1ccncc1 ZINC000217811931 EE In-Stock Unstable P96878_MYCTU 19 45 O=C(Cc1cc2c(cc1Cl)OCCO2)NCCc1ccncc1 ZINC000217811931 EE In-Stock Unstable CAN2 0 45 Cc1ccc(-c2csc(NC(=O)c3cc(-c4ccco4)on3)n2)s1 ZINC000217811948 FJ On-Demand Unstable MPL 41 33 C[C@H](NC[C@H](O)CO[C@@H]1CCCC[C@@H]1C)c1ccccn1 ZINC000217811950 CF For-Sale Unstable ADRB2 47 43 C[C@H](NC[C@H](O)CO[C@@H]1CCCC[C@@H]1C)c1ccccn1 ZINC000217811950 CF For-Sale Unstable ADRB1 26 40 O=C(CSc1ccc(F)cc1)N1CCC[C@H](Cc2nc(C3CC3)no2)C1 ZINC000217811969 GH In-Stock Unstable CCR3 49 34 CCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217811990 DG For-Sale Unstable AVPR1A 18 42 CCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217811990 DG For-Sale Unstable GRIN2B 19 45 CCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217811990 DG For-Sale Unstable HCRTR1 17 42 CCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217811990 DG For-Sale Unstable ITGA4 43 32 CCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217811990 DG For-Sale Unstable CHRNA10 55 42 CCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217811990 DG For-Sale Unstable CACNA1I 57 34 CCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217811990 DG For-Sale Unstable HCN1 45 33 CCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217811990 DG For-Sale Unstable HCN4 42 33 CCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217811990 DG For-Sale Unstable NOD2 32 42 CCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217811990 DG For-Sale Unstable ACKR3 57 34 C=C(C)COc1cccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c1 ZINC000217812023 KK In-Stock Unstable AKR1B1 0 41 C=C(C)COc1cccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c1 ZINC000217812023 KK In-Stock Unstable CYP1B1 40 33 C=C(C)COc1cccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c1 ZINC000217812023 KK In-Stock Unstable CYP1A1 31 41 COc1ccc(NC(=O)N/C=C/c2ccccc2Cl)c(OC)c1 ZINC000217812024 EI For-Sale Unstable CYP1B1 41 46 COc1ccc(NC(=O)N/C=C/c2ccccc2Cl)c(OC)c1 ZINC000217812024 EI For-Sale Unstable GRM4 16 40 COc1ccc(NC(=O)N/C=C/c2ccccc2Cl)c(OC)c1 ZINC000217812024 EI For-Sale Unstable MTNR1A 20 45 COc1ccc(NC(=O)N/C=C/c2ccccc2Cl)c(OC)c1 ZINC000217812024 EI For-Sale Unstable MTNR1B 20 45 COc1ccc(NC(=O)N/C=C/c2ccccc2Cl)c(OC)c1 ZINC000217812024 EI For-Sale Unstable AKR1C2 45 34 COc1ccc(NC(=O)N/C=C/c2ccccc2Cl)c(OC)c1 ZINC000217812024 EI For-Sale Unstable CYSP_PLAFA 47 42 O=C(CSc1ccc(F)cc1)N1CCC[C@@H](Cc2nc(C3CC3)no2)C1 ZINC000217812053 GH In-Stock Unstable CCR3 52 34 CCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217812066 DG For-Sale Unstable AVPR1A 18 42 CCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217812066 DG For-Sale Unstable GRIN2B 19 45 CCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217812066 DG For-Sale Unstable HCRTR1 17 42 CCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217812066 DG For-Sale Unstable ITGA4 43 32 CCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217812066 DG For-Sale Unstable CHRNA10 55 42 CCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217812066 DG For-Sale Unstable CACNA1I 57 34 CCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217812066 DG For-Sale Unstable HCN1 45 33 CCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217812066 DG For-Sale Unstable HCN4 42 33 CCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217812066 DG For-Sale Unstable NOD2 32 42 CCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217812066 DG For-Sale Unstable ACKR3 57 34 C=C(C)COc1cccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c1 ZINC000217812123 KK In-Stock Unstable AKR1B1 0 41 C=C(C)COc1cccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c1 ZINC000217812123 KK In-Stock Unstable CYP1B1 40 33 C=C(C)COc1cccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)c1 ZINC000217812123 KK In-Stock Unstable CYP1A1 31 41 O=C(NCCOCC1CC1)c1ccc(Br)c(Cl)c1 ZINC000217812126 EG On-Demand Unstable CACNA1I 43 33 COc1cccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217812176 DG For-Sale Unstable HTR1A 19 45 COc1cccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217812176 DG For-Sale Unstable DRD2 44 44 COc1cccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217812176 DG For-Sale Unstable DRD4 46 36 COc1cccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217812176 DG For-Sale Unstable DRD3 28 44 COc1cccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217812176 DG For-Sale Unstable OPRK1 15 40 COc1cccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217812176 DG For-Sale Unstable SLC18A2 39 42 COc1cccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217812176 DG For-Sale Unstable TACR1 15 44 COc1cccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217812176 DG For-Sale Unstable SIGMAR1 31 54 COc1cccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217812176 DG For-Sale Unstable CCR3 21 42 COc1cccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217812176 DG For-Sale Unstable MTNR1A 73 42 COc1cccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217812176 DG For-Sale Unstable MTNR1B 76 42 COc1cccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217812176 DG For-Sale Unstable CHRNA10 64 44 COc1cccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217812176 DG For-Sale Unstable MCHR1 21 43 COc1cccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217812176 DG For-Sale Unstable ACKR3 68 36 CC(=O)NCCCc1ccc(-c2csc(NC(=O)c3cc(-c4ccco4)on3)n2)cc1 ZINC000217812197 II On-Demand Unstable ROCK1 20 40 CC(=O)NCCCc1ccc(-c2csc(NC(=O)c3cc(-c4ccco4)on3)n2)cc1 ZINC000217812197 II On-Demand Unstable HDAC10 17 43 CNC(=O)[C@@H]1CCCCN1[C@@H](C)Cc1ccc(O)cc1 ZINC000217812240 CD For-Sale Unstable OPRM1 42 43 CNC(=O)[C@@H]1CCCCN1[C@@H](C)Cc1ccc(O)cc1 ZINC000217812240 CD For-Sale Unstable OPRD1 23 43 CNC(=O)[C@@H]1CCCCN1[C@@H](C)Cc1ccc(O)cc1 ZINC000217812240 CD For-Sale Unstable OPRK1 0 40 CNC(=O)[C@@H]1CCCCN1[C@@H](C)Cc1ccc(O)cc1 ZINC000217812240 CD For-Sale Unstable NTSR1 91 35 CNC(=O)[C@@H]1CCCCN1[C@@H](C)Cc1ccc(O)cc1 ZINC000217812240 CD For-Sale Unstable NTSR2 67 33 CNC(=O)[C@@H]1CCCCN1[C@@H](C)Cc1ccc(O)cc1 ZINC000217812240 CD For-Sale Unstable HLA-A 49 34 CNC(=O)[C@@H]1CCCCN1[C@@H](C)Cc1ccc(O)cc1 ZINC000217812240 CD For-Sale Unstable LGMN 65 34 CNC(=O)[C@@H]1CCCCN1[C@@H](C)Cc1ccc(O)cc1 ZINC000217812240 CD For-Sale Unstable SORT1 43 32 CNC(=O)[C@@H]1CCCCN1[C@@H](C)Cc1ccc(O)cc1 ZINC000217812240 CD For-Sale Unstable YARS 62 33 CNC(=O)[C@@H]1CCCCN1[C@@H](C)Cc1ccc(O)cc1 ZINC000217812240 CD For-Sale Unstable MARS 46 33 CNC(=O)[C@@H]1CCCCN1[C@@H](C)Cc1ccc(O)cc1 ZINC000217812240 CD For-Sale Unstable XIAP 40 43 COc1cccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217812246 DG For-Sale Unstable HTR1A 19 45 COc1cccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217812246 DG For-Sale Unstable DRD2 44 44 COc1cccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217812246 DG For-Sale Unstable DRD4 46 36 COc1cccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217812246 DG For-Sale Unstable DRD3 28 44 COc1cccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217812246 DG For-Sale Unstable OPRK1 15 40 COc1cccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217812246 DG For-Sale Unstable SLC18A2 39 42 COc1cccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217812246 DG For-Sale Unstable TACR1 15 44 COc1cccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217812246 DG For-Sale Unstable SIGMAR1 31 54 COc1cccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217812246 DG For-Sale Unstable CCR3 21 42 COc1cccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217812246 DG For-Sale Unstable MTNR1A 73 42 COc1cccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217812246 DG For-Sale Unstable MTNR1B 76 42 COc1cccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217812246 DG For-Sale Unstable CHRNA10 64 44 COc1cccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217812246 DG For-Sale Unstable MCHR1 21 43 COc1cccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217812246 DG For-Sale Unstable ACKR3 68 36 CC(=O)NCCCc1ccc(-c2csc(NC(=O)c3cccc(C[S@@](C)=O)c3)n2)cc1 ZINC000217812304 JI On-Demand Unstable ROCK1 21 43 CC(=O)NCCCc1ccc(-c2csc(NC(=O)c3cccc(C[S@@](C)=O)c3)n2)cc1 ZINC000217812304 JI On-Demand Unstable ROCK2 17 44 CC(=O)NCCCc1ccc(-c2csc(NC(=O)c3cccc(C[S@@](C)=O)c3)n2)cc1 ZINC000217812304 JI On-Demand Unstable AOC3 15 52 CC(=O)NCCCc1ccc(-c2csc(NC(=O)c3cccc(C[S@](C)=O)c3)n2)cc1 ZINC000217812370 JI On-Demand Unstable ROCK1 21 43 CC(=O)NCCCc1ccc(-c2csc(NC(=O)c3cccc(C[S@](C)=O)c3)n2)cc1 ZINC000217812370 JI On-Demand Unstable ROCK2 17 44 CC(=O)NCCCc1ccc(-c2csc(NC(=O)c3cccc(C[S@](C)=O)c3)n2)cc1 ZINC000217812370 JI On-Demand Unstable AOC3 15 52 C[C@@H](c1ccccc1F)N(C)C[C@@H](N)c1ccccc1 ZINC000217812434 CH For-Sale Unstable AOC3 24 40 C[C@@H]1CCCC[C@@H]1OC[C@@H](O)CNC(C)(C)CC(C)(C)C ZINC000217812441 CH For-Sale Unstable ADRB2 45 39 CNC(=O)[C@@H]1CCCCN1[C@@H](C)CCc1ccc(O)cc1 ZINC000217812453 CE For-Sale Unstable ACE 33 47 CNC(=O)[C@@H]1CCCCN1[C@@H](C)CCc1ccc(O)cc1 ZINC000217812453 CE For-Sale Unstable FKBP1A 50 37 CNC(=O)[C@@H]1CCCCN1[C@@H](C)CCc1ccc(O)cc1 ZINC000217812453 CE For-Sale Unstable OPRM1 26 40 CNC(=O)[C@@H]1CCCCN1[C@@H](C)CCc1ccc(O)cc1 ZINC000217812453 CE For-Sale Unstable NTSR1 80 34 CNC(=O)[C@@H]1CCCCN1[C@@H](C)CCc1ccc(O)cc1 ZINC000217812453 CE For-Sale Unstable NTSR2 70 33 CNC(=O)[C@@H]1CCCCN1[C@@H](C)CCc1ccc(O)cc1 ZINC000217812453 CE For-Sale Unstable HLA-A 47 32 CNC(=O)[C@@H]1CCCCN1[C@@H](C)CCc1ccc(O)cc1 ZINC000217812453 CE For-Sale Unstable LGMN 59 33 CNC(=O)[C@@H]1CCCCN1[C@@H](C)CCc1ccc(O)cc1 ZINC000217812453 CE For-Sale Unstable XIAP 48 38 CNC(=O)[C@@H]1CCCCN1[C@@H](C)CCc1ccc(O)cc1 ZINC000217812453 CE For-Sale Unstable BIRC2 63 41 CC(=O)NCCCc1ccc(-c2csc(NC(=O)c3cc(-c4ccc(Cl)cc4)n[nH]3)n2)cc1 ZINC000217812483 JK On-Demand Unstable MPL 23 42 CC(=O)NCCCc1ccc(-c2csc(NC(=O)c3cc(-c4ccc(Cl)cc4)n[nH]3)n2)cc1 ZINC000217812483 JK On-Demand Unstable ROCK1 21 41 CC(=O)NCCCc1ccc(-c2csc(NC(=O)c3cc(-c4ccc(Cl)cc4)n[nH]3)n2)cc1 ZINC000217812483 JK On-Demand Unstable SPHK2 41 36 CC(=O)NCCCc1ccc(-c2csc(NC(=O)c3cc(-c4ccc(Cl)cc4)n[nH]3)n2)cc1 ZINC000217812483 JK On-Demand Unstable ROCK2 16 41 CC(=O)NCCCc1ccc(-c2csc(NC(=O)c3cc(-c4ccc(Cl)cc4)n[nH]3)n2)cc1 ZINC000217812483 JK On-Demand Unstable ALPL 66 38 CC(=O)NCCCc1ccc(-c2csc(NC(=O)c3cc(-c4ccc(Cl)cc4)n[nH]3)n2)cc1 ZINC000217812483 JK On-Demand Unstable U38 0 44 C[C@H](c1ccccc1F)N(C)C[C@@H](N)c1ccccc1 ZINC000217812513 CH For-Sale Unstable AOC3 24 40 Cc1nc2ccccc2nc1N1CCN[C@H](C(C)C)C1 ZINC000217812524 CE For-Sale Unstable PRKCQ 43 35 C[C@H]1CCCC[C@@H]1OC[C@@H](O)CNC(C)(C)CC(C)(C)C ZINC000217812530 CH For-Sale Unstable ADRB2 45 39 Cc1cccc(OCC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217812540 DG For-Sale Unstable CCKAR 52 34 Cc1cccc(OCC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217812540 DG For-Sale Unstable COLA 72 36 Cc1cccc(OCC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217812540 DG For-Sale Unstable CPT1A 68 36 Cc1cccc(OCC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217812540 DG For-Sale Unstable FAAH 16 41 Cc1cccc(OCC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217812540 DG For-Sale Unstable CHRNA10 61 37 CNC(=O)[C@@H]1CCCCN1[C@@H](C)c1ccccc1O ZINC000217812570 CE For-Sale Unstable XPNPEP1 0 40 CNC(=O)[C@@H]1CCCCN1[C@@H](C)c1ccccc1O ZINC000217812570 CE For-Sale Unstable XPNPEP2 0 40 CNC(=O)[C@@H]1CCCCN1[C@@H](C)c1ccccc1O ZINC000217812570 CE For-Sale Unstable XIAP 40 34 CC(=O)NCCCc1ccc(-c2csc(NC(=O)c3cc(-c4ccc(C)cc4)n[nH]3)n2)cc1 ZINC000217812586 JJ On-Demand Unstable ROCK1 22 42 CC(=O)NCCCc1ccc(-c2csc(NC(=O)c3cc(-c4ccc(C)cc4)n[nH]3)n2)cc1 ZINC000217812586 JJ On-Demand Unstable ROCK2 18 42 CC(=O)NCCCc1ccc(-c2csc(NC(=O)c3cc(-c4ccc(C)cc4)n[nH]3)n2)cc1 ZINC000217812586 JJ On-Demand Unstable HDAC9 15 45 CC(=O)NCCCc1ccc(-c2csc(NC(=O)c3cc(-c4ccc(C)cc4)n[nH]3)n2)cc1 ZINC000217812586 JJ On-Demand Unstable ALPL 43 31 Cc1nc2ccccc2nc1N1CCN[C@@H](C(C)C)C1 ZINC000217812593 CE On-Demand Unstable PRKCQ 43 35 Cc1cccc(OCC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217812608 DG For-Sale Unstable CCKAR 52 34 Cc1cccc(OCC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217812608 DG For-Sale Unstable COLA 72 36 Cc1cccc(OCC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217812608 DG For-Sale Unstable CPT1A 68 36 Cc1cccc(OCC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217812608 DG For-Sale Unstable FAAH 16 41 Cc1cccc(OCC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217812608 DG For-Sale Unstable CHRNA10 61 37 C[C@@H]1CCCC[C@H]1OC[C@@H](O)CNC(C)(C)CC(C)(C)C ZINC000217812614 CH For-Sale Unstable ADRB2 45 39 CC(C)CCNC(=O)CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12 ZINC000217812621 HH In-Stock Unstable TOP1 0 41 CCOC(=O)[C@@H](Oc1ccc(C)cc1)c1ccccc1 ZINC000217812640 CH For-Sale Unstable PPARA 24 48 C[C@H]1CCCC[C@H]1OC[C@@H](O)CNC(C)(C)CC(C)(C)C ZINC000217812682 CH For-Sale Unstable ADRB2 45 39 CC(C)CCNC(=O)CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12 ZINC000217812704 HH In-Stock Unstable TOP1 0 41 CSc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217812716 EH For-Sale Unstable DRD2 31 40 CSc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217812716 EH For-Sale Unstable HCRTR1 34 41 CSc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217812716 EH For-Sale Unstable PREP 18 40 CSc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217812716 EH For-Sale Unstable HCRTR2 26 41 CSc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217812716 EH For-Sale Unstable HCN1 54 32 CSc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217812716 EH For-Sale Unstable HCN4 40 30 CCOC(=O)[C@H](Oc1ccc(C)cc1)c1ccccc1 ZINC000217812720 CH For-Sale Unstable PPARA 24 48 C[C@H](Cc1ccc(Br)cc1)NC(=O)[C@@H]1C[C@@H](O)CN1 ZINC000217812751 ED In-Stock Unstable CTSC 30 41 C[C@@H]1CCC[C@H](OC[C@@H](O)CNC(C)(C)CC(C)(C)C)C1 ZINC000217812761 CH For-Sale Unstable ADRB2 30 49 C[C@@H]1CCC[C@H](OC[C@@H](O)CNC(C)(C)CC(C)(C)C)C1 ZINC000217812761 CH For-Sale Unstable ADRB1 0 49 CSc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217812797 EH For-Sale Unstable DRD2 31 40 CSc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217812797 EH For-Sale Unstable HCRTR1 34 41 CSc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217812797 EH For-Sale Unstable PREP 18 40 CSc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217812797 EH For-Sale Unstable HCRTR2 26 41 CSc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217812797 EH For-Sale Unstable HCN1 54 32 CSc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217812797 EH For-Sale Unstable HCN4 40 30 CC(C)CNC(=O)c1ccc(NC(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc1 ZINC000217812803 HF In-Stock Unstable CHRNA4 28 46 CC(C)CNC(=O)c1ccc(NC(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc1 ZINC000217812803 HF In-Stock Unstable F3 83 37 CCOC(=O)[C@H](Oc1cccc(Br)c1)c1ccccc1 ZINC000217812822 EI On-Demand Unstable F9 19 40 CCOC(=O)[C@H](Oc1cccc(Br)c1)c1ccccc1 ZINC000217812822 EI On-Demand Unstable PDS 53 44 C[C@@H](Cc1ccc(Br)cc1)NC(=O)[C@H]1C[C@@H](O)CN1 ZINC000217812828 ED On-Demand Unstable CTSC 30 41 C[C@H]1CCC[C@H](OC[C@@H](O)CNC(C)(C)CC(C)(C)C)C1 ZINC000217812834 CH For-Sale Unstable ADRB2 30 49 C[C@H]1CCC[C@H](OC[C@@H](O)CNC(C)(C)CC(C)(C)C)C1 ZINC000217812834 CH For-Sale Unstable ADRB1 0 49 C[C@H](Cc1ccc(Br)cc1)NC(=O)[C@H]1C[C@@H](O)CN1 ZINC000217812898 ED In-Stock Unstable CTSC 30 41 CSc1ncccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217812901 EG For-Sale Unstable HCRTR1 35 44 CSc1ncccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217812901 EG For-Sale Unstable HCRTR2 28 44 C[C@@H]1CCC[C@@H](OC[C@@H](O)CNC(C)(C)CC(C)(C)C)C1 ZINC000217812905 CH For-Sale Unstable ADRB2 30 49 C[C@@H]1CCC[C@@H](OC[C@@H](O)CNC(C)(C)CC(C)(C)C)C1 ZINC000217812905 CH For-Sale Unstable ADRB1 0 49 CSc1ncccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217812992 EG For-Sale Unstable HCRTR1 35 44 CSc1ncccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217812992 EG For-Sale Unstable HCRTR2 28 44 C[C@H]1CCC[C@@H](OC[C@@H](O)CNC(C)(C)CC(C)(C)C)C1 ZINC000217812993 CH For-Sale Unstable ADRB2 30 49 C[C@H]1CCC[C@@H](OC[C@@H](O)CNC(C)(C)CC(C)(C)C)C1 ZINC000217812993 CH For-Sale Unstable ADRB1 0 49 CC(C)[C@@H]1CN(c2cnc3cc(C(F)(F)F)ccc3n2)CCN1 ZINC000217813094 DG For-Sale Unstable PRKCQ 19 41 COc1ccc([C@@H]2CC(=O)Oc3ccc4c(c32)OC(C)(C)CC4=O)c(OC)c1OC ZINC000217813114 HH In-Stock Unstable MT-ND4 50 30 O=C(COc1ccc(F)cc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217813118 EF For-Sale Unstable HCRTR1 15 41 O=C(COc1ccc(F)cc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217813118 EF For-Sale Unstable COLA 65 39 O=C(COc1ccc(F)cc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217813118 EF For-Sale Unstable CPT1A 61 39 CCOC(=O)[C@@H](Oc1cccc(Cl)c1)c1ccccc1 ZINC000217813124 CI For-Sale Unstable PPARA 18 42 CCOC(=O)[C@@H](Oc1cccc(Cl)c1)c1ccccc1 ZINC000217813124 CI For-Sale Unstable PDS 79 47 CC(C)[C@H]1CN(c2cnc3cc(C(F)(F)F)ccc3n2)CCN1 ZINC000217813165 DG For-Sale Unstable PRKCQ 19 41 O=C(COc1ccc(F)cc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217813189 EF For-Sale Unstable HCRTR1 18 45 O=C(COc1ccc(F)cc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217813189 EF For-Sale Unstable COLA 65 39 O=C(COc1ccc(F)cc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217813189 EF For-Sale Unstable CPT1A 61 39 COc1ccc([C@H]2CC(=O)Oc3ccc4c(c32)OC(C)(C)CC4=O)c(OC)c1OC ZINC000217813195 HH In-Stock Unstable MT-ND4 50 30 CCOC(=O)[C@H](Oc1cccc(Cl)c1)c1ccccc1 ZINC000217813215 CI For-Sale Unstable PPARA 18 42 CCOC(=O)[C@H](Oc1cccc(Cl)c1)c1ccccc1 ZINC000217813215 CI For-Sale Unstable PDS 79 47 C[C@@H]1CCCC[C@@H]1NC(=O)N/C=C/c1ccccc1Cl ZINC000217813233 CI For-Sale Unstable PDE7A 0 41 N#Cc1ccc(C(=O)N2CCC[C@H](Cc3nc(C4CC4)no3)C2)cc1 ZINC000217813272 EF In-Stock Unstable GRM3 15 45 O=C(Cc1ccc(Cl)cc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217813295 EH For-Sale Unstable DRD2 22 40 O=C(Cc1ccc(Cl)cc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217813295 EH For-Sale Unstable KCNQ2 19 44 O=C(Cc1ccc(Cl)cc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217813295 EH For-Sale Unstable SIGMAR1 25 49 O=C1C[C@H](N2CCc3c([nH]c4ccccc34)[C@@H]2c2ccccc2)C(=O)N1c1ccccc1 ZINC000217813296 HI In-Stock Unstable PDE5A 54 45 O=C1C[C@H](N2CCc3c([nH]c4ccccc34)[C@@H]2c2ccccc2)C(=O)N1c1ccccc1 ZINC000217813296 HI In-Stock Unstable DRD5 15 41 O=C1C[C@H](N2CCc3c([nH]c4ccccc34)[C@@H]2c2ccccc2)C(=O)N1c1ccccc1 ZINC000217813296 HI In-Stock Unstable ME1 0 43 O=C1C[C@H](N2CCc3c([nH]c4ccccc34)[C@@H]2c2ccccc2)C(=O)N1c1ccccc1 ZINC000217813296 HI In-Stock Unstable PDE11A 92 40 O=C1C[C@H](N2CCc3c([nH]c4ccccc34)[C@@H]2c2ccccc2)C(=O)N1c1ccccc1 ZINC000217813296 HI In-Stock Unstable KIF11 22 42 C[C@H]1CCCC[C@@H]1NC(=O)N/C=C/c1ccccc1Cl ZINC000217813303 CI For-Sale Unstable PDE7A 0 41 CC(C)n1c(CCNC(=O)CCCC[C@@H]2SC[C@@H]3NC(=O)N[C@H]23)nc2ccccc21 ZINC000217813312 IG In-Stock Unstable PLCD1 0 43 CC(C)n1c(CCNC(=O)CCCC[C@@H]2SC[C@@H]3NC(=O)N[C@H]23)nc2ccccc21 ZINC000217813312 IG In-Stock Unstable AGAL_COFAR 0 50 CC(C)n1c(CCNC(=O)CCCC[C@@H]2SC[C@@H]3NC(=O)N[C@H]23)nc2ccccc21 ZINC000217813312 IG In-Stock Unstable HSPA8 0 41 CC(C)n1c(CCNC(=O)CCCC[C@@H]2SC[C@@H]3NC(=O)N[C@H]23)nc2ccccc21 ZINC000217813312 IG In-Stock Unstable CYTH3 0 43 CC(C)n1c(CCNC(=O)CCCC[C@@H]2SC[C@@H]3NC(=O)N[C@H]23)nc2ccccc21 ZINC000217813312 IG In-Stock Unstable HLCS 0 41 CC(C)n1c(CCNC(=O)CCCC[C@@H]2SC[C@@H]3NC(=O)N[C@H]23)nc2ccccc21 ZINC000217813312 IG In-Stock Unstable GIGYF2 0 42 CC(C)n1c(CCNC(=O)CCCC[C@@H]2SC[C@@H]3NC(=O)N[C@H]23)nc2ccccc21 ZINC000217813312 IG In-Stock Unstable BIRA 0 42 CC(C)C[C@@H](C)OC[C@@H](O)CN[C@H](c1cccs1)C(C)C ZINC000217813315 DH For-Sale Unstable ADRB2 23 47 CCCS(=O)(=O)CCSc1nnnn1-c1ccc(O)cc1 ZINC000217813319 ED On-Demand Unstable CELA2A 29 40 N#Cc1ccc(C(=O)N2CCC[C@@H](Cc3nc(C4CC4)no3)C2)cc1 ZINC000217813346 EF In-Stock Unstable GRM3 15 45 CC(C)C[C@H](C)OC[C@@H](O)CN[C@H](c1cccs1)C(C)C ZINC000217813389 DH For-Sale Unstable ADRB2 23 47 C[C@@H]1CCCC[C@H]1NC(=O)N/C=C/c1ccccc1Cl ZINC000217813391 CI For-Sale Unstable PDE7A 0 41 O=C(Cc1ccc(Cl)cc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217813401 EH For-Sale Unstable DRD2 22 40 O=C(Cc1ccc(Cl)cc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217813401 EH For-Sale Unstable KCNQ2 19 44 O=C(Cc1ccc(Cl)cc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217813401 EH For-Sale Unstable SIGMAR1 25 49 O=C1C[C@H](N2CCc3c([nH]c4ccccc34)[C@@H]2c2ccccc2)C(=O)N1c1cccc(F)c1 ZINC000217813405 IJ In-Stock Unstable PDE5A 53 42 O=C1C[C@H](N2CCc3c([nH]c4ccccc34)[C@@H]2c2ccccc2)C(=O)N1c1cccc(F)c1 ZINC000217813405 IJ In-Stock Unstable ME1 0 41 O=C1C[C@H](N2CCc3c([nH]c4ccccc34)[C@@H]2c2ccccc2)C(=O)N1c1cccc(F)c1 ZINC000217813405 IJ In-Stock Unstable PDE11A 93 39 O=C1C[C@H](N2CCc3c([nH]c4ccccc34)[C@@H]2c2ccccc2)C(=O)N1c1cccc(F)c1 ZINC000217813405 IJ In-Stock Unstable KIF11 24 42 CC(C)C[C@@H](C)OC[C@H](O)CN[C@H](c1cccs1)C(C)C ZINC000217813481 DH For-Sale Unstable ADRB2 23 47 C[C@H]1CCCC[C@H]1NC(=O)N/C=C/c1ccccc1Cl ZINC000217813496 CI For-Sale Unstable PDE7A 0 41 CCOC(=O)[C@@H](Oc1cccc(F)c1)c1ccccc1 ZINC000217813511 CH For-Sale Unstable PPARA 15 42 CCOC(=O)[C@@H](Oc1cccc(F)c1)c1ccccc1 ZINC000217813511 CH For-Sale Unstable PDS 48 43 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(F)cc1Cl ZINC000217813520 EH For-Sale Unstable DRD2 35 40 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(F)cc1Cl ZINC000217813520 EH For-Sale Unstable SLC6A1 46 41 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(F)cc1Cl ZINC000217813520 EH For-Sale Unstable HCRTR1 30 43 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(F)cc1Cl ZINC000217813520 EH For-Sale Unstable P2RX7 51 42 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(F)cc1Cl ZINC000217813520 EH For-Sale Unstable PYGL 27 42 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(F)cc1Cl ZINC000217813520 EH For-Sale Unstable HCRTR2 21 43 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(F)cc1Cl ZINC000217813520 EH For-Sale Unstable ACKR3 56 32 CC(C)C[C@H](C)OC[C@H](O)CN[C@H](c1cccs1)C(C)C ZINC000217813561 DH For-Sale Unstable ADRB2 23 47 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(F)cc1Cl ZINC000217813597 EH For-Sale Unstable DRD2 35 40 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(F)cc1Cl ZINC000217813597 EH For-Sale Unstable SLC6A1 46 41 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(F)cc1Cl ZINC000217813597 EH For-Sale Unstable HCRTR1 30 43 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(F)cc1Cl ZINC000217813597 EH For-Sale Unstable P2RX7 51 42 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(F)cc1Cl ZINC000217813597 EH For-Sale Unstable PYGL 27 42 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(F)cc1Cl ZINC000217813597 EH For-Sale Unstable HCRTR2 21 43 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(F)cc1Cl ZINC000217813597 EH For-Sale Unstable ACKR3 56 32 CCOC(=O)[C@H](Oc1cccc(F)c1)c1ccccc1 ZINC000217813608 CH For-Sale Unstable PPARA 15 42 CCOC(=O)[C@H](Oc1cccc(F)c1)c1ccccc1 ZINC000217813608 CH For-Sale Unstable PDS 48 43 COc1ccc(-c2c(C(=O)O)cnn2C(C)(C)C)cc1 ZINC000217813654 CG On-Demand Unstable AKR1C2 50 37 O=C(NC[C@H]1CCCN1c1ccccc1)c1c(F)cccc1Cl ZINC000217813697 EH For-Sale Unstable SLC6A1 43 37 O=C(NC[C@@H]1CCCN1c1ccccc1)c1c(F)cccc1Cl ZINC000217813761 EH For-Sale Unstable SLC6A1 43 37 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)N2CCc3[nH]c4ccccc4c3C2)[C@@H](C)O)cc1 ZINC000217813816 IE On-Demand Unstable MMP13 18 40 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)N2CCc3[nH]c4ccccc4c3C2)[C@@H](C)O)cc1 ZINC000217813816 IE On-Demand Unstable MMP2 19 40 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)N2CCc3[nH]c4ccccc4c3C2)[C@@H](C)O)cc1 ZINC000217813816 IE On-Demand Unstable ADAMTS4 53 34 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(Nc2ccccc2)cc1 ZINC000217813867 FK For-Sale Anodyne EPHX1 0 43 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(Nc2ccccc2)cc1 ZINC000217813867 FK For-Sale Anodyne SMO 17 43 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(Nc2ccccc2)cc1 ZINC000217813867 FK For-Sale Anodyne P95276_MYCTO 0 43 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCc3[nH]c4ccccc4c3C2)[C@@H](C)O)cc1 ZINC000217813887 IE On-Demand Unstable MMP13 18 40 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCc3[nH]c4ccccc4c3C2)[C@@H](C)O)cc1 ZINC000217813887 IE On-Demand Unstable MMP2 19 40 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCc3[nH]c4ccccc4c3C2)[C@@H](C)O)cc1 ZINC000217813887 IE On-Demand Unstable ADAMTS4 53 34 Cc1cc(C(=O)N2CCCN(Cc3cccnc3)CC2)cc(=O)[nH]1 ZINC000217813946 ED In-Stock Unstable FAAH 20 40 Cc1cc(C(=O)N2CCCN(Cc3cccnc3)CC2)cc(=O)[nH]1 ZINC000217813946 ED In-Stock Unstable PARP1 20 40 Cc1cc(C(=O)N2CCCN(Cc3cccnc3)CC2)cc(=O)[nH]1 ZINC000217813946 ED In-Stock Unstable MGLL 0 40 Cc1cc(C(=O)N2CCCN(Cc3cccnc3)CC2)cc(=O)[nH]1 ZINC000217813946 ED In-Stock Unstable CCR8 23 40 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)N2CCc3[nH]c4ccccc4c3C2)[C@H](C)O)cc1 ZINC000217813968 IE On-Demand Unstable MMP13 18 40 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)N2CCc3[nH]c4ccccc4c3C2)[C@H](C)O)cc1 ZINC000217813968 IE On-Demand Unstable MMP2 19 40 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)N2CCc3[nH]c4ccccc4c3C2)[C@H](C)O)cc1 ZINC000217813968 IE On-Demand Unstable ADAMTS4 53 34 O=C1C[C@@H]2CC[C@H](C1)N2CCc1cccc(Cl)c1 ZINC000217814002 CG On-Demand Unstable CACNA1C 27 47 O=C1C[C@@H]2CC[C@H](C1)N2CCc1cccc(Cl)c1 ZINC000217814002 CG On-Demand Unstable CACNA1D 84 52 O=C1C[C@@H]2CC[C@H](C1)N2CCc1cccc(Cl)c1 ZINC000217814002 CG On-Demand Unstable Q8WSF8_APLCA 17 40 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCc3[nH]c4ccccc4c3C2)[C@H](C)O)cc1 ZINC000217814015 IE On-Demand Unstable MMP13 18 40 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCc3[nH]c4ccccc4c3C2)[C@H](C)O)cc1 ZINC000217814015 IE On-Demand Unstable MMP2 19 40 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCc3[nH]c4ccccc4c3C2)[C@H](C)O)cc1 ZINC000217814015 IE On-Demand Unstable ADAMTS4 53 34 CCOC(=O)[C@H](Oc1ccc(F)cc1Cl)c1ccccc1 ZINC000217814032 DI On-Demand Unstable AGTR1B 0 43 Cc1cccc(NC(=O)N/C=C/c2ccccc2Cl)n1 ZINC000217814110 CH For-Sale Unstable GRM5 18 48 Cc1cccc(NC(=O)N/C=C/c2ccccc2Cl)n1 ZINC000217814110 CH For-Sale Unstable SORT1 17 46 O=C(c1cc(C2CC2)on1)N1CCC[C@H](Cc2nc(C3CC3)no2)C1 ZINC000217814121 EF In-Stock Unstable S1PR3 0 41 O=C(c1cc(C2CC2)on1)N1CCC[C@@H](Cc2nc(C3CC3)no2)C1 ZINC000217814188 EF In-Stock Unstable S1PR3 0 41 O=C(Nc1nc2c(s1)CCCC2)c1nn(-c2ccccc2)cc1O ZINC000217814244 EG On-Demand Unstable SLC27A1 31 52 COc1ccc(CCN2C(=O)N[C@@H](CC(=O)N[C@H](CO)c3ccccc3)C2=O)cc1 ZINC000217814245 HD In-Stock Unstable GPR88 0 47 CC(C)Oc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217814248 EH For-Sale Unstable PREP 15 41 CC(C)Oc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217814248 EH For-Sale Unstable CACNA1I 45 32 O=C(N/C=C/c1ccccc1Cl)Nc1ccccn1 ZINC000217814310 CH For-Sale Anodyne TYK2 48 34 CC(C)Oc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217814330 EH For-Sale Unstable PREP 15 41 CC(C)Oc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217814330 EH For-Sale Unstable CACNA1I 45 32 CC(C)(C)OC(=O)Nc1ccc2c(c1)C(=O)c1ccccc1-2 ZINC000217814346 CI For-Sale Unstable CASP2 16 40 O=C(N/C=C/c1ccccc1Cl)Nc1cccnc1 ZINC000217814391 CH For-Sale Anodyne NAMPT 33 46 COc1cc(OC)cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217814428 EG For-Sale Unstable HTR1A 17 48 COc1cc(OC)cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217814428 EG For-Sale Unstable DRD2 41 43 COc1cc(OC)cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217814428 EG For-Sale Unstable DRD4 48 37 COc1cc(OC)cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217814428 EG For-Sale Unstable DRD3 35 45 COc1cc(OC)cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217814428 EG For-Sale Unstable PREP 18 40 COc1cc(OC)cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217814428 EG For-Sale Unstable CHRNA10 47 41 COc1cc(OC)cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217814428 EG For-Sale Unstable MCHR1 19 49 COc1cc(OC)cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217814428 EG For-Sale Unstable CACNA1I 64 35 COc1cc(OC)cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217814428 EG For-Sale Unstable ACKR3 71 37 COc1ccc2cc(C(=O)N3CCC[C@H](Cc4nc(C5CC5)no4)C3)[nH]c2c1 ZINC000217814472 GH In-Stock Unstable GRIN2B 24 49 COc1ccc2cc(C(=O)N3CCC[C@H](Cc4nc(C5CC5)no4)C3)[nH]c2c1 ZINC000217814472 GH In-Stock Unstable FPR2 26 41 COc1ccc2cc(C(=O)N3CCC[C@H](Cc4nc(C5CC5)no4)C3)[nH]c2c1 ZINC000217814472 GH In-Stock Unstable AKR1C3 0 40 COc1cc(OC)cc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217814512 EG For-Sale Unstable HTR1A 17 48 COc1cc(OC)cc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217814512 EG For-Sale Unstable DRD2 41 43 COc1cc(OC)cc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217814512 EG For-Sale Unstable DRD4 48 37 COc1cc(OC)cc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217814512 EG For-Sale Unstable DRD3 35 45 COc1cc(OC)cc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217814512 EG For-Sale Unstable PREP 18 40 COc1cc(OC)cc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217814512 EG For-Sale Unstable CHRNA10 47 41 COc1cc(OC)cc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217814512 EG For-Sale Unstable MCHR1 19 49 COc1cc(OC)cc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217814512 EG For-Sale Unstable CACNA1I 64 35 COc1cc(OC)cc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217814512 EG For-Sale Unstable ACKR3 71 37 COc1ccc2cc(C(=O)N3CCC[C@@H](Cc4nc(C5CC5)no4)C3)[nH]c2c1 ZINC000217814543 GH In-Stock Unstable GRIN2B 24 49 COc1ccc2cc(C(=O)N3CCC[C@@H](Cc4nc(C5CC5)no4)C3)[nH]c2c1 ZINC000217814543 GH In-Stock Unstable FPR2 26 41 COc1ccc2cc(C(=O)N3CCC[C@@H](Cc4nc(C5CC5)no4)C3)[nH]c2c1 ZINC000217814543 GH In-Stock Unstable AKR1C3 0 40 CNC(=O)Cc1c(C)n[nH]c1N ZINC000217814546 AB In-Stock Unstable HAO2 60 35 CC[C@@H](C)[C@@H]1CN(c2cnc3ccccc3n2)CCN1 ZINC000217814593 CE For-Sale Unstable SORD 17 45 COc1cccc(OC)c1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217814627 EG For-Sale Unstable HTR1A 46 48 COc1cccc(OC)c1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217814627 EG For-Sale Unstable DRD2 64 69 COc1cccc(OC)c1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217814627 EG For-Sale Unstable DRD1 20 41 COc1cccc(OC)c1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217814627 EG For-Sale Unstable DRD4 32 41 COc1cccc(OC)c1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217814627 EG For-Sale Unstable DRD3 54 53 COc1cccc(OC)c1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217814627 EG For-Sale Unstable KCNA3 42 34 COc1cccc(OC)c1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217814627 EG For-Sale Unstable HCN1 53 36 COc1cccc(OC)c1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217814627 EG For-Sale Unstable HCN4 41 34 COc1cccc(OC)c1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217814627 EG For-Sale Unstable ACKR3 77 39 CC[C@H](C)[C@@H]1CN(c2cnc3ccccc3n2)CCN1 ZINC000217814678 CE For-Sale Unstable SORD 17 45 COc1ccc(CN2C(=O)N[C@@H](CC(=O)NCCc3ccc(O)cc3)C2=O)cc1 ZINC000217814710 GD In-Stock Unstable ADRB1 22 40 COc1ccc(CN2C(=O)N[C@@H](CC(=O)NCCc3ccc(O)cc3)C2=O)cc1 ZINC000217814710 GD In-Stock Unstable ADRB3 19 40 COc1ccc(CN2C(=O)N[C@@H](CC(=O)NCCc3ccc(O)cc3)C2=O)cc1 ZINC000217814710 GD In-Stock Unstable PROKR1 62 38 COc1cccc(OC)c1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217814716 EG For-Sale Unstable HTR1A 46 48 COc1cccc(OC)c1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217814716 EG For-Sale Unstable DRD2 64 69 COc1cccc(OC)c1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217814716 EG For-Sale Unstable DRD1 20 41 COc1cccc(OC)c1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217814716 EG For-Sale Unstable DRD4 32 41 COc1cccc(OC)c1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217814716 EG For-Sale Unstable DRD3 54 53 COc1cccc(OC)c1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217814716 EG For-Sale Unstable KCNA3 42 34 COc1cccc(OC)c1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217814716 EG For-Sale Unstable HCN1 53 36 COc1cccc(OC)c1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217814716 EG For-Sale Unstable HCN4 41 34 COc1cccc(OC)c1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217814716 EG For-Sale Unstable ACKR3 77 39 CC[C@@H](C)[C@H]1CN(c2cnc3ccccc3n2)CCN1 ZINC000217814759 CE For-Sale Unstable SORD 17 45 Cn1ncc(C(N)=O)c1-c1ccc(F)cc1 ZINC000217814801 BD For-Sale Unstable CDC7 22 40 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217814831 EG For-Sale Unstable HTR1A 29 48 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217814831 EG For-Sale Unstable DRD2 55 50 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217814831 EG For-Sale Unstable DRD4 42 32 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217814831 EG For-Sale Unstable ACHE 17 49 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217814831 EG For-Sale Unstable DRD3 49 45 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217814831 EG For-Sale Unstable CYSLTR1 64 39 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217814831 EG For-Sale Unstable F10 17 42 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217814831 EG For-Sale Unstable PDE4A 16 46 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217814831 EG For-Sale Unstable AGTR2 42 33 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217814831 EG For-Sale Unstable PDE4D 15 42 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217814831 EG For-Sale Unstable CPT1A 43 30 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217814831 EG For-Sale Unstable CHRNA10 43 36 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217814831 EG For-Sale Unstable MCHR1 24 46 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217814831 EG For-Sale Unstable CACNA1I 54 35 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217814831 EG For-Sale Unstable ACKR3 90 49 CC[C@@H](CCO)NC[C@@H](O)COCC(C)C ZINC000217814837 BC On-Demand Unstable ADRB2 0 59 CC[C@H](C)[C@H]1CN(c2cnc3ccccc3n2)CCN1 ZINC000217814846 CE For-Sale Unstable SORD 17 45 CC[C@H](CCO)NC[C@@H](O)COCC(C)C ZINC000217814902 BC On-Demand Unstable ADRB2 0 59 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217814912 EG For-Sale Unstable HTR1A 29 48 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217814912 EG For-Sale Unstable DRD2 55 50 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217814912 EG For-Sale Unstable DRD4 42 32 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217814912 EG For-Sale Unstable ACHE 17 49 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217814912 EG For-Sale Unstable DRD3 49 45 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217814912 EG For-Sale Unstable CYSLTR1 64 39 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217814912 EG For-Sale Unstable F10 17 42 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217814912 EG For-Sale Unstable PDE4A 16 46 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217814912 EG For-Sale Unstable AGTR2 42 33 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217814912 EG For-Sale Unstable PDE4D 15 42 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217814912 EG For-Sale Unstable CPT1A 43 30 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217814912 EG For-Sale Unstable CHRNA10 43 36 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217814912 EG For-Sale Unstable MCHR1 24 46 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217814912 EG For-Sale Unstable CACNA1I 54 35 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217814912 EG For-Sale Unstable ACKR3 90 49 CC[C@@H](CCO)NC[C@H](O)COCC(C)C ZINC000217814972 BC On-Demand Unstable ADRB2 0 59 COc1cccc(OCC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217815009 EF For-Sale Unstable DRD4 43 33 COc1cccc(OCC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217815009 EF For-Sale Unstable COLA 74 37 COc1cccc(OCC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217815009 EF For-Sale Unstable CPT1A 67 37 COc1cccc(OCC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217815009 EF For-Sale Unstable MTNR1A 57 36 COc1cccc(OCC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217815009 EF For-Sale Unstable MTNR1B 49 41 COc1cccc(OCC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217815009 EF For-Sale Unstable CHRNA10 57 48 COc1cccc(OCC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217815009 EF For-Sale Unstable MCHR1 16 41 COc1cccc(OCC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217815009 EF For-Sale Unstable ACKR3 66 35 CC[C@H](CCO)NC[C@H](O)COCC(C)C ZINC000217815036 BC On-Demand Unstable ADRB2 0 59 C[C@@H](N)[C@H](c1cccc(Br)c1)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217815050 FI For-Sale Unstable MBTD1 0 44 CCOC(=O)[C@H](Oc1ccccc1CC)c1ccccc1 ZINC000217815065 CH On-Demand Unstable F9 26 42 CCOC(=O)[C@H](Oc1ccccc1CC)c1ccccc1 ZINC000217815065 CH On-Demand Unstable GUAB 0 40 CNC(=O)Cc1c(-c2ccccc2)n[nH]c1N ZINC000217815077 BC In-Stock Unstable HAO2 62 33 COc1cccc(OCC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217815080 EF For-Sale Unstable DRD4 43 33 COc1cccc(OCC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217815080 EF For-Sale Unstable COLA 74 37 COc1cccc(OCC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217815080 EF For-Sale Unstable CPT1A 67 37 COc1cccc(OCC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217815080 EF For-Sale Unstable MTNR1A 57 36 COc1cccc(OCC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217815080 EF For-Sale Unstable MTNR1B 49 41 COc1cccc(OCC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217815080 EF For-Sale Unstable CHRNA10 57 48 COc1cccc(OCC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217815080 EF For-Sale Unstable MCHR1 16 41 COc1cccc(OCC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217815080 EF For-Sale Unstable ACKR3 66 35 C[C@H](N)[C@H](c1cccc(Br)c1)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217815124 FI For-Sale Unstable MBTD1 0 44 CC(=O)Nc1cccc(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217815190 EI For-Sale Unstable TYK2 23 40 CC(=O)Nc1cccc(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217815190 EI For-Sale Unstable IMDH_CRYPV 43 37 CC(=O)Nc1cccc(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217815190 EI For-Sale Unstable KCNK3 105 44 CC(=O)Nc1cccc(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217815190 EI For-Sale Unstable KCNK9 67 37 CCSc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217815191 EI For-Sale Unstable HCRTR1 30 40 CCSc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217815191 EI For-Sale Unstable HCRTR2 24 40 CCSc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217815191 EI For-Sale Unstable HCN1 63 31 CCSc1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217815191 EI For-Sale Unstable HCN4 48 31 C[C@@H](N)[C@@H](c1cccc(Br)c1)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217815210 FI For-Sale Unstable MBTD1 0 44 C[C@@H]1CN(C)CCN1C(=O)c1ccc(Br)c(Cl)c1 ZINC000217815256 EF On-Demand Unstable SLC6A7 0 41 CCN(CCOc1cccc(/C=C\C(=O)O)c1)CC(C)C ZINC000217815259 CG For-Sale Unstable AKR1C3 28 40 CCSc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217815269 EI For-Sale Unstable HCRTR1 30 40 CCSc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217815269 EI For-Sale Unstable HCRTR2 24 40 CCSc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217815269 EI For-Sale Unstable HCN1 63 31 CCSc1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217815269 EI For-Sale Unstable HCN4 48 31 C[C@H](N)[C@@H](c1cccc(Br)c1)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217815282 FI For-Sale Unstable MBTD1 0 44 C[C@H]1CN(C)CCN1C(=O)c1ccc(Br)c(Cl)c1 ZINC000217815322 EF On-Demand Unstable SLC6A7 0 41 O=C(NCc1ccccn1)[C@@H]1CC[C@@H](CNS(=O)(=O)c2ccc(F)cc2)CC1 ZINC000217815329 HF In-Stock Unstable NPY2R 84 47 O=C(NCc1ccccn1)[C@@H]1CC[C@@H](CNS(=O)(=O)c2ccc(F)cc2)CC1 ZINC000217815329 HF In-Stock Unstable NPY5R 28 47 O=C(NCc1ccccn1)[C@@H]1CC[C@@H](CNS(=O)(=O)c2ccc(F)cc2)CC1 ZINC000217815329 HF In-Stock Unstable GPR39 0 42 O=C(CSc1ccc(F)cc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217815387 EH For-Sale Unstable HCRTR1 17 40 Cc1ccc(Br)c(C(=O)N2CCN(C)C[C@@H]2C)c1 ZINC000217815443 DF On-Demand Unstable HCRTR1 43 36 O=C(CSc1ccc(F)cc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217815479 EH For-Sale Unstable HCRTR1 17 40 Cc1ccc(Br)c(C(=O)N2CCN(C)C[C@H]2C)c1 ZINC000217815525 DF On-Demand Unstable HCRTR1 43 36 Nc1[nH]nc(-c2ccccc2)c1CC(=O)N1CCOCC1 ZINC000217815557 CD In-Stock Unstable AKR1C3 23 40 CCCN(CCOc1ccc(/C=C\C(=O)O)cc1)C1CC1 ZINC000217815586 CG On-Demand Unstable PLA2G4B 51 32 C[C@@H]1CCC[C@H](OC[C@@H](O)CNC(C2CC2)C2CC2)C1 ZINC000217815589 CF For-Sale Unstable ADRB2 0 40 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cc(-c2ccccc2)on1 ZINC000217815598 EH For-Sale Unstable HDAC10 17 47 O=C(Cc1cccc(C(F)(F)F)c1)N1CCC[C@H](Cc2nc(C3CC3)no2)C1 ZINC000217815601 GH In-Stock Unstable CCR2 43 36 O=C(Cc1cccc(C(F)(F)F)c1)N1CCC[C@H](Cc2nc(C3CC3)no2)C1 ZINC000217815601 GH In-Stock Unstable ETHR 40 38 O=C(NC[C@H]1CCCN1c1ccccc1)c1cc(-c2ccccc2)on1 ZINC000217815671 EH For-Sale Unstable HDAC10 17 47 O=C(Cc1cccc(C(F)(F)F)c1)N1CCC[C@@H](Cc2nc(C3CC3)no2)C1 ZINC000217815674 GH In-Stock Unstable CCR2 43 36 O=C(Cc1cccc(C(F)(F)F)c1)N1CCC[C@@H](Cc2nc(C3CC3)no2)C1 ZINC000217815674 GH In-Stock Unstable ETHR 40 38 C[C@H]1CCC[C@H](OC[C@@H](O)CNC(C2CC2)C2CC2)C1 ZINC000217815675 CF For-Sale Unstable ADRB2 0 40 O=C(Cn1nnc(-c2ccc(Cl)cc2)n1)Nc1ccccc1C(=O)N1CCCC1 ZINC000217815740 HF On-Demand Unstable F10 17 46 O=C(Cn1nnc(-c2ccc(Cl)cc2)n1)Nc1ccccc1C(=O)N1CCCC1 ZINC000217815740 HF On-Demand Unstable KCNQ2 22 40 O=C(Cn1nnc(-c2ccc(Cl)cc2)n1)Nc1ccccc1C(=O)N1CCCC1 ZINC000217815740 HF On-Demand Unstable NPSR1 15 45 O=C(Cn1nnc(-c2ccc(Cl)cc2)n1)Nc1ccccc1C(=O)N1CCCC1 ZINC000217815740 HF On-Demand Unstable SCARB1 41 41 CC(C)(C)OC(=O)N1CCC[C@@H]1[C@H](O)c1cccs1 ZINC000217815750 CG For-Sale Unstable PREP 15 42 C[C@@H]1CCC[C@@H](OC[C@@H](O)CNC(C2CC2)C2CC2)C1 ZINC000217815761 CF For-Sale Unstable ADRB2 0 40 O=C(NC[C@H]1CCCN1c1ccccc1)c1cccc(C(F)(F)F)c1 ZINC000217815779 EI For-Sale Unstable DRD2 25 43 O=C(NC[C@H]1CCCN1c1ccccc1)c1cccc(C(F)(F)F)c1 ZINC000217815779 EI For-Sale Unstable KCNJ11 20 41 O=C(NC[C@H]1CCCN1c1ccccc1)c1cccc(C(F)(F)F)c1 ZINC000217815779 EI For-Sale Unstable CCR2 118 57 O=C(NC[C@H]1CCCN1c1ccccc1)c1cccc(C(F)(F)F)c1 ZINC000217815779 EI For-Sale Unstable CHRNA10 18 42 O=C(NC[C@H]1CCCN1c1ccccc1)c1cccc(C(F)(F)F)c1 ZINC000217815779 EI For-Sale Unstable CACNA1I 54 45 O=C(NC[C@H]1CCCN1c1ccccc1)c1cccc(C(F)(F)F)c1 ZINC000217815779 EI For-Sale Unstable AKR1C3 17 40 O=C(NC[C@H]1CCCN1c1ccccc1)c1cccc(C(F)(F)F)c1 ZINC000217815779 EI For-Sale Unstable LIPG 45 36 O=C(NC[C@H]1CCCN1c1ccccc1)c1cccc(C(F)(F)F)c1 ZINC000217815779 EI For-Sale Unstable SFRP1 73 37 O=C(NC[C@H]1CCCN1c1ccccc1)c1cccc(C(F)(F)F)c1 ZINC000217815779 EI For-Sale Unstable WNT3 42 31 COC(=O)C[C@H](c1ccc(OC)c(OC)c1)c1oc(CN2CCCCC2)cc(=O)c1O ZINC000217815782 IG In-Stock Unstable TNF 21 40 CC(C)(C)OC(=O)N1CCC[C@@H]1[C@@H](O)c1cccs1 ZINC000217815822 CG For-Sale Unstable PREP 15 42 C[C@H]1CCC[C@@H](OC[C@@H](O)CNC(C2CC2)C2CC2)C1 ZINC000217815829 CF For-Sale Unstable ADRB2 0 40 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cccc(C(F)(F)F)c1 ZINC000217815867 EI For-Sale Unstable DRD2 25 43 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cccc(C(F)(F)F)c1 ZINC000217815867 EI For-Sale Unstable KCNJ11 20 41 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cccc(C(F)(F)F)c1 ZINC000217815867 EI For-Sale Unstable CCR2 118 57 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cccc(C(F)(F)F)c1 ZINC000217815867 EI For-Sale Unstable CHRNA10 18 42 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cccc(C(F)(F)F)c1 ZINC000217815867 EI For-Sale Unstable CACNA1I 54 45 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cccc(C(F)(F)F)c1 ZINC000217815867 EI For-Sale Unstable AKR1C3 17 40 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cccc(C(F)(F)F)c1 ZINC000217815867 EI For-Sale Unstable LIPG 45 36 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cccc(C(F)(F)F)c1 ZINC000217815867 EI For-Sale Unstable SFRP1 73 37 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cccc(C(F)(F)F)c1 ZINC000217815867 EI For-Sale Unstable WNT3 42 31 COC(=O)C[C@@H](c1ccc(OC)c(OC)c1)c1oc(CN2CCCCC2)cc(=O)c1O ZINC000217815875 IG In-Stock Unstable TNF 21 40 CCc1ccc(C(=O)[C@@H]2C[C@@H]2C(=O)O)cc1 ZINC000217815957 BE In-Stock Unstable GRIK2 74 49 O=C(OCc1ccccc1)N1CCC[C@H](Cc2nc(C3CC3)no2)C1 ZINC000217815992 EH In-Stock Unstable GRIN2B 31 44 O=C(OCc1ccccc1)N1CCC[C@H](Cc2nc(C3CC3)no2)C1 ZINC000217815992 EH In-Stock Unstable PREP 30 42 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(C(F)(F)F)cc1 ZINC000217815994 EI For-Sale Unstable PLA2G4A 43 31 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(C(F)(F)F)cc1 ZINC000217815994 EI For-Sale Unstable PREP 16 41 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(C(F)(F)F)cc1 ZINC000217815994 EI For-Sale Unstable MTTP 50 38 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(C(F)(F)F)cc1 ZINC000217815994 EI For-Sale Unstable CCR2 62 44 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(C(F)(F)F)cc1 ZINC000217815994 EI For-Sale Unstable SLC6A5 29 40 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(C(F)(F)F)cc1 ZINC000217815994 EI For-Sale Unstable EPHX2 23 45 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(C(F)(F)F)cc1 ZINC000217815994 EI For-Sale Unstable MCHR1 22 47 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(C(F)(F)F)cc1 ZINC000217815994 EI For-Sale Unstable CACNA1I 46 39 CCc1ccc(C(=O)[C@H]2C[C@@H]2C(=O)O)cc1 ZINC000217816039 BE In-Stock Unstable GRIK2 74 49 CN(Cc1cccs1)Cc1ccccc1/C=C\C(=O)O ZINC000217816040 CG For-Sale Unstable PTGER2 53 45 CN(Cc1cccs1)Cc1ccccc1/C=C\C(=O)O ZINC000217816040 CG For-Sale Unstable PTGER3 23 42 O=C(OCc1ccccc1)N1CCC[C@@H](Cc2nc(C3CC3)no2)C1 ZINC000217816063 EH In-Stock Unstable GRIN2B 31 44 O=C(OCc1ccccc1)N1CCC[C@@H](Cc2nc(C3CC3)no2)C1 ZINC000217816063 EH In-Stock Unstable PREP 30 42 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(C(F)(F)F)cc1 ZINC000217816077 EI For-Sale Unstable PLA2G4A 43 31 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(C(F)(F)F)cc1 ZINC000217816077 EI For-Sale Unstable PREP 16 41 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(C(F)(F)F)cc1 ZINC000217816077 EI For-Sale Unstable MTTP 50 38 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(C(F)(F)F)cc1 ZINC000217816077 EI For-Sale Unstable CCR2 62 44 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(C(F)(F)F)cc1 ZINC000217816077 EI For-Sale Unstable SLC6A5 29 40 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(C(F)(F)F)cc1 ZINC000217816077 EI For-Sale Unstable EPHX2 23 45 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(C(F)(F)F)cc1 ZINC000217816077 EI For-Sale Unstable MCHR1 22 47 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(C(F)(F)F)cc1 ZINC000217816077 EI For-Sale Unstable CACNA1I 46 39 CCc1ccc(C(=O)[C@@H]2C[C@H]2C(=O)O)cc1 ZINC000217816134 BE In-Stock Unstable GRIK2 74 49 O=C(c1ccc(Br)c(Cl)c1)N1CCCS(=O)(=O)CC1 ZINC000217816157 FE On-Demand Unstable L3MBTL3 45 36 Cc1ccc(Cn2nccc2NC(=O)c2cnn(-c3ccc(Cl)cc3)c2C(F)(F)F)cc1 ZINC000217816161 JK On-Demand Unstable MST1R 49 37 Cn1ccnc1CN1CCN(Cc2cccnc2)C[C@@H](C(=O)O)C1 ZINC000217816162 EC In-Stock Unstable DRD4 15 44 Cn1ccnc1CN1CCN(Cc2cccnc2)C[C@@H](C(=O)O)C1 ZINC000217816162 EC In-Stock Unstable SLC6A1 58 32 Cn1ccnc1CN1CCN(Cc2cccnc2)C[C@@H](C(=O)O)C1 ZINC000217816162 EC In-Stock Unstable S1PR1 29 40 C[C@@H](c1ccc(Cl)cc1)N(C)[C@H](C)C(N)=S ZINC000217816169 CG For-Sale Unstable UTS2 41 32 O=C(NC[C@H]1CCCN1c1ccccc1)c1cc(=O)c2ccccc2o1 ZINC000217816203 EG For-Sale Unstable DRD2 29 40 O=C(NC[C@H]1CCCN1c1ccccc1)c1cc(=O)c2ccccc2o1 ZINC000217816203 EG For-Sale Unstable KCNH2 15 46 O=C(NC[C@H]1CCCN1c1ccccc1)c1cc(=O)c2ccccc2o1 ZINC000217816203 EG For-Sale Unstable BCHE 31 44 CCc1ccc(C(=O)[C@H]2C[C@H]2C(=O)O)cc1 ZINC000217816225 BE In-Stock Unstable GRIK2 74 49 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cc(=O)c2ccccc2o1 ZINC000217816280 EG For-Sale Unstable DRD2 29 40 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cc(=O)c2ccccc2o1 ZINC000217816280 EG For-Sale Unstable KCNH2 15 46 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cc(=O)c2ccccc2o1 ZINC000217816280 EG For-Sale Unstable BCHE 31 44 CC[C@@H]1CN(Cc2ccc(F)c(/C=C\C(=O)O)c2)CCO1 ZINC000217816318 CF For-Sale Unstable DRD4 20 46 Cc1ccc(Cn2nccc2NC(=O)C2CCN(c3nc4ccccc4o3)CC2)cc1 ZINC000217816345 HI On-Demand Unstable PTGES 38 42 CN1CCN(C)[C@@H](CNC(=O)c2ccc(Br)c(Cl)c2)C1 ZINC000217816366 FE On-Demand Unstable UTS2R 25 40 CN1CCN(C)[C@@H](CNC(=O)c2ccc(Br)c(Cl)c2)C1 ZINC000217816366 FE On-Demand Unstable CACNA1I 71 47 CC[C@H]1CN(Cc2ccc(F)c(/C=C\C(=O)O)c2)CCO1 ZINC000217816378 CF For-Sale Unstable DRD4 20 46 O=C(NC[C@H]1CCCN1c1ccccc1)c1cc2ccccc2oc1=O ZINC000217816393 EG For-Sale Unstable DRD2 30 40 O=C(NC[C@H]1CCCN1c1ccccc1)c1cc2ccccc2oc1=O ZINC000217816393 EG For-Sale Unstable MAOB 15 54 O=C(N/C=C/c1ccccc1Cl)Nc1ccccc1N1CCOCC1 ZINC000217816410 FH For-Sale Unstable CSF1R 0 48 O=C(N/C=C/c1ccccc1Cl)Nc1ccccc1N1CCOCC1 ZINC000217816410 FH For-Sale Unstable AKR1C3 24 51 CN(C)C1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217816460 CE For-Sale Unstable SIGMAR1 31 48 CN(C)C1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217816460 CE For-Sale Unstable PTGER3 16 48 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cc2ccccc2oc1=O ZINC000217816475 EG For-Sale Unstable DRD2 30 40 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cc2ccccc2oc1=O ZINC000217816475 EG For-Sale Unstable MAOB 15 54 CN1CCN(c2ccc(NC(=O)N/C=C/c3ccccc3Cl)cc2)CC1 ZINC000217816486 FH For-Sale Unstable HCK 28 46 CN(C)C1CCN(Cc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217816553 CE For-Sale Unstable DRD2 15 40 CN(C)C1CCN(Cc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217816553 CE For-Sale Unstable DRD4 42 40 CN(C)C1CCN(Cc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217816553 CE For-Sale Unstable ACHE 28 43 CN(C)C1CCN(Cc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217816553 CE For-Sale Unstable HRH3 15 40 CN(C)C1CCN(Cc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217816553 CE For-Sale Unstable SIGMAR1 45 63 CC(C)C[C@H](NC(=O)c1cccc2c1ccn2C)C(=O)O ZINC000217816572 CE In-Stock Unstable MME 21 42 CC(C)C[C@H](NC(=O)c1cccc2c1ccn2C)C(=O)O ZINC000217816572 CE In-Stock Unstable EDNRA 34 44 CC(C)C[C@H](NC(=O)c1cccc2c1ccn2C)C(=O)O ZINC000217816572 CE In-Stock Unstable CCKAR 28 45 CC(C)C[C@H](NC(=O)c1cccc2c1ccn2C)C(=O)O ZINC000217816572 CE In-Stock Unstable FPR1 54 37 CC(C)C[C@H](NC(=O)c1cccc2c1ccn2C)C(=O)O ZINC000217816572 CE In-Stock Unstable NPR 47 35 O=C(/C=C/c1ccc2c(c1)OCO2)NC[C@H]1CCCN1c1ccccc1 ZINC000217816605 FG For-Sale Unstable NOS2 85 39 O=C(/C=C/c1ccc2c(c1)OCO2)NC[C@H]1CCCN1c1ccccc1 ZINC000217816605 FG For-Sale Unstable HDAC1 23 44 O=C(/C=C/c1ccc2c(c1)OCO2)NC[C@H]1CCCN1c1ccccc1 ZINC000217816605 FG For-Sale Unstable HDAC6 20 44 O=C(/C=C/c1ccc2c(c1)OCO2)NC[C@H]1CCCN1c1ccccc1 ZINC000217816605 FG For-Sale Unstable DYRK2 46 35 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(N2CCCCC2)cc1 ZINC000217816609 FK For-Sale Unstable LPL 44 36 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(N2CCCCC2)cc1 ZINC000217816609 FK For-Sale Unstable KCNQ2 28 42 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(N2CCCCC2)cc1 ZINC000217816609 FK For-Sale Unstable PRNP 41 36 O=C(O)/C=C\c1ccc(OCCN2CCCC2=O)cc1 ZINC000217816632 CD For-Sale Unstable HRH3 19 47 O=C(O)/C=C\c1ccc(OCCN2CCCC2=O)cc1 ZINC000217816632 CD For-Sale Unstable PSMB2 46 36 O=C(O)/C=C\c1ccc(OCCN2CCCC2=O)cc1 ZINC000217816632 CD For-Sale Unstable PSMB1 40 36 CCCc1ccc(C(=O)[C@@H]2C[C@@H]2C(=O)O)cc1 ZINC000217816656 BF In-Stock Unstable GRIK2 63 51 O=C(NCCN1CCSCC1)c1ccc(Br)c(Cl)c1 ZINC000217816686 FF On-Demand Unstable DRD4 55 44 O=C(NCCN1CCSCC1)c1ccc(Br)c(Cl)c1 ZINC000217816686 FF On-Demand Unstable DRD3 33 41 O=C(NCCN1CCSCC1)c1ccc(Br)c(Cl)c1 ZINC000217816686 FF On-Demand Unstable PLD1 45 44 O=C(NCCN1CCSCC1)c1ccc(Br)c(Cl)c1 ZINC000217816686 FF On-Demand Unstable PLD2 79 44 O=C(/C=C/c1ccc2c(c1)OCO2)NC[C@@H]1CCCN1c1ccccc1 ZINC000217816689 FG For-Sale Unstable NOS2 85 39 O=C(/C=C/c1ccc2c(c1)OCO2)NC[C@@H]1CCCN1c1ccccc1 ZINC000217816689 FG For-Sale Unstable HDAC1 23 44 O=C(/C=C/c1ccc2c(c1)OCO2)NC[C@@H]1CCCN1c1ccccc1 ZINC000217816689 FG For-Sale Unstable HDAC6 20 44 O=C(/C=C/c1ccc2c(c1)OCO2)NC[C@@H]1CCCN1c1ccccc1 ZINC000217816689 FG For-Sale Unstable DYRK2 46 35 COc1ccc(/C=C\C(=O)O)cc1CN1CCCC1=O ZINC000217816727 CD For-Sale Unstable PTGER2 0 44 CCCc1ccc(C(=O)[C@H]2C[C@@H]2C(=O)O)cc1 ZINC000217816751 BF In-Stock Unstable GRIK2 63 51 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccccc2Cl)CC(=O)O4)cc1O ZINC000217816768 JJ In-Stock Unstable AKR1B1 0 46 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccccc2Cl)CC(=O)O4)cc1O ZINC000217816768 JJ In-Stock Unstable CYP1B1 62 39 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccccc2Cl)CC(=O)O4)cc1O ZINC000217816768 JJ In-Stock Unstable CYP1A1 48 46 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccccc2Cl)CC(=O)O4)cc1O ZINC000217816768 JJ In-Stock Unstable CYP1A2 41 39 C[C@@H](c1ccc(Cl)cc1)N(C)[C@H](C)C(=O)N1CCNCC1 ZINC000217816785 DE For-Sale Unstable CCR1 42 37 C[C@@H](c1ccc(Cl)cc1)N(C)[C@H](C)C(=O)N1CCNCC1 ZINC000217816785 DE For-Sale Unstable UTS2 43 33 O=C(O)/C=C\c1cccc(Cn2cnc3ccccc32)c1 ZINC000217816804 CG For-Sale Unstable PTGER2 26 40 O=C(O)/C=C\c1cccc(Cn2cnc3ccccc32)c1 ZINC000217816804 CG For-Sale Unstable HDAC8 45 46 O=C(O)/C=C\c1cccc(Cn2cnc3ccccc32)c1 ZINC000217816804 CG For-Sale Unstable HDAC1 21 46 O=C(O)/C=C\c1cccc(Cn2cnc3ccccc32)c1 ZINC000217816804 CG For-Sale Unstable HDAC6 39 46 O=C(O)/C=C\c1cccc(Cn2cnc3ccccc32)c1 ZINC000217816804 CG For-Sale Unstable PKM 18 41 O=C(O)/C=C\c1cccc(Cn2cnc3ccccc32)c1 ZINC000217816804 CG For-Sale Unstable NR1I2 54 42 O=C(O)/C=C\c1cccc(Cn2cnc3ccccc32)c1 ZINC000217816804 CG For-Sale Unstable RHOA 0 47 Cc1ccc(Br)c(C(=O)NCCN2CCSCC2)c1 ZINC000217816812 EF On-Demand Unstable DRD2 19 51 Cc1ccc(Br)c(C(=O)NCCN2CCSCC2)c1 ZINC000217816812 EF On-Demand Unstable DRD4 46 40 Cc1ccc(Br)c(C(=O)NCCN2CCSCC2)c1 ZINC000217816812 EF On-Demand Unstable HTR2C 32 43 Cc1ccc(Br)c(C(=O)NCCN2CCSCC2)c1 ZINC000217816812 EF On-Demand Unstable DRD3 29 51 Cc1ccc(Br)c(C(=O)NCCN2CCSCC2)c1 ZINC000217816812 EF On-Demand Unstable PLD2 46 35 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccccc2Cl)CC(=O)O4)cc1O ZINC000217816849 JJ In-Stock Unstable AKR1B1 0 46 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccccc2Cl)CC(=O)O4)cc1O ZINC000217816849 JJ In-Stock Unstable CYP1B1 62 39 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccccc2Cl)CC(=O)O4)cc1O ZINC000217816849 JJ In-Stock Unstable CYP1A1 48 46 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccccc2Cl)CC(=O)O4)cc1O ZINC000217816849 JJ In-Stock Unstable CYP1A2 41 39 CCCc1ccc(C(=O)[C@@H]2C[C@H]2C(=O)O)cc1 ZINC000217816850 BF In-Stock Unstable GRIK2 63 51 CCCc1ccc(C(=O)[C@H]2C[C@H]2C(=O)O)cc1 ZINC000217816910 BF In-Stock Unstable GRIK2 63 51 C[C@@H](c1ccccc1Cl)N(C)[C@H](C)C(=O)N1CCNCC1 ZINC000217816969 DE For-Sale Unstable FDFT1 0 41 CCCCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217816977 FI For-Sale Unstable DRD2 31 42 CCCCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217816977 FI For-Sale Unstable DRD3 27 42 CCCCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217816977 FI For-Sale Unstable AVPR1A 18 43 CCCCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217816977 FI For-Sale Unstable P2RY12 89 34 CCCCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217816977 FI For-Sale Unstable GRIN2B 20 47 CCCCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217816977 FI For-Sale Unstable LTA4H 42 39 CCCCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217816977 FI For-Sale Unstable HCRTR1 16 41 CCCCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217816977 FI For-Sale Unstable CYSLTR2 49 37 CCCCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217816977 FI For-Sale Unstable HRH3 42 38 CCCCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217816977 FI For-Sale Unstable PLA2G4A 24 40 CCCCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217816977 FI For-Sale Unstable ITGA4 42 31 CCCCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217816977 FI For-Sale Unstable PLA2G4B 90 40 CCCCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217816977 FI For-Sale Unstable CHRNA10 47 40 CCCCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217816977 FI For-Sale Unstable ACKR3 48 33 COc1ccc(-c2noc(CCC(=O)N3CCN([C@@H](C#N)c4ccccc4)CC3)n2)cc1 ZINC000217816978 IG On-Demand Unstable PTAFR 54 52 COc1ccc(-c2noc(CCC(=O)N3CCN([C@@H](C#N)c4ccccc4)CC3)n2)cc1 ZINC000217816978 IG On-Demand Unstable COLA 25 41 COc1ccc(-c2noc(CCC(=O)N3CCN([C@@H](C#N)c4ccccc4)CC3)n2)cc1 ZINC000217816978 IG On-Demand Unstable CPT1A 20 41 CCCC[C@H]1N=C(N)S[C@H]1C ZINC000217816982 AD For-Sale Unstable NOS2 16 49 CCOC(=O)[C@@H](Oc1cccc(C)c1C)c1ccccc1 ZINC000217816983 CH For-Sale Unstable F9 26 43 O=C(N/C=C/c1ccccc1Cl)Nc1cccc2ccccc12 ZINC000217817044 DK For-Sale Anodyne CXCL8 42 37 O=C(N/C=C/c1ccccc1Cl)Nc1cccc2ccccc12 ZINC000217817044 DK For-Sale Anodyne TRPV1 36 49 COC(=O)[C@@H]1C[C@@H]1C(=O)c1ccc(C)cc1 ZINC000217817057 BD In-Stock Unstable SLC6A1 40 40 COC(=O)[C@@H]1C[C@@H]1C(=O)c1ccc(C)cc1 ZINC000217817057 BD In-Stock Unstable SLC6A3 18 40 CCOC(=O)[C@H](Oc1cccc(C)c1C)c1ccccc1 ZINC000217817062 CH For-Sale Unstable F9 26 43 COc1ccc(-c2noc(CCC(=O)N3CCN([C@H](C#N)c4ccccc4)CC3)n2)cc1 ZINC000217817063 IG On-Demand Unstable PTAFR 54 52 COc1ccc(-c2noc(CCC(=O)N3CCN([C@H](C#N)c4ccccc4)CC3)n2)cc1 ZINC000217817063 IG On-Demand Unstable COLA 25 41 COc1ccc(-c2noc(CCC(=O)N3CCN([C@H](C#N)c4ccccc4)CC3)n2)cc1 ZINC000217817063 IG On-Demand Unstable CPT1A 20 41 CCCCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217817067 FI For-Sale Unstable DRD2 31 42 CCCCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217817067 FI For-Sale Unstable DRD3 27 42 CCCCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217817067 FI For-Sale Unstable AVPR1A 18 43 CCCCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217817067 FI For-Sale Unstable P2RY12 89 34 CCCCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217817067 FI For-Sale Unstable GRIN2B 20 47 CCCCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217817067 FI For-Sale Unstable LTA4H 42 39 CCCCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217817067 FI For-Sale Unstable HCRTR1 16 41 CCCCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217817067 FI For-Sale Unstable CYSLTR2 49 37 CCCCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217817067 FI For-Sale Unstable HRH3 42 38 CCCCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217817067 FI For-Sale Unstable PLA2G4A 24 40 CCCCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217817067 FI For-Sale Unstable ITGA4 42 31 CCCCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217817067 FI For-Sale Unstable PLA2G4B 90 40 CCCCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217817067 FI For-Sale Unstable CHRNA10 47 40 CCCCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217817067 FI For-Sale Unstable ACKR3 48 33 CCCC[C@@H]1N=C(N)S[C@H]1C ZINC000217817074 AD For-Sale Unstable NOS2 16 49 COC(=O)[C@H]1C[C@@H]1C(=O)c1ccc(C)cc1 ZINC000217817149 BD In-Stock Unstable SLC6A1 40 40 COC(=O)[C@H]1C[C@@H]1C(=O)c1ccc(C)cc1 ZINC000217817149 BD In-Stock Unstable SLC6A3 18 40 CCCC[C@H]1N=C(N)S[C@@H]1C ZINC000217817150 AD For-Sale Unstable NOS2 0 49 CCOc1ccc(OCC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217817159 FG For-Sale Unstable COLA 60 39 CCOc1ccc(OCC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217817159 FG For-Sale Unstable CPT1A 58 39 CCOc1ccc(OCC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217817159 FG For-Sale Unstable CHRNA10 40 39 COC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217817166 EH For-Sale Unstable ACR 47 39 OC1(c2ccccc2)CCN(c2ccccn2)CC1 ZINC000217817207 CF On-Demand Unstable DRD4 31 43 OC1(c2ccccc2)CCN(c2ccccn2)CC1 ZINC000217817207 CF On-Demand Unstable OPRK1 16 55 OC1(c2ccccc2)CCN(c2ccccn2)CC1 ZINC000217817207 CF On-Demand Unstable OPRL1 26 55 OC1(c2ccccc2)CCN(c2ccccn2)CC1 ZINC000217817207 CF On-Demand Unstable EBP 29 47 OC1(c2ccccc2)CCN(c2ccccn2)CC1 ZINC000217817207 CF On-Demand Unstable SORD 44 39 Cc1ccn2c(C(=O)N3CCC[C@@H](COc4cccc(F)c4)C3)nnc2n1 ZINC000217817211 FF In-Stock Unstable CHRNA10 46 42 CCCC[C@@H]1N=C(N)S[C@@H]1C ZINC000217817224 AD For-Sale Unstable NOS2 0 49 CCOc1ccc(OCC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217817226 FG For-Sale Unstable COLA 60 39 CCOc1ccc(OCC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217817226 FG For-Sale Unstable CPT1A 58 39 CCOc1ccc(OCC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217817226 FG For-Sale Unstable CHRNA10 40 39 COC(=O)[C@@H]1C[C@H]1C(=O)c1ccc(C)cc1 ZINC000217817230 BD In-Stock Unstable SLC6A1 40 40 COC(=O)[C@@H]1C[C@H]1C(=O)c1ccc(C)cc1 ZINC000217817230 BD In-Stock Unstable SLC6A3 18 40 Cc1ccn2c(C(=O)N3CCC[C@H](COc4cccc(F)c4)C3)nnc2n1 ZINC000217817257 FF In-Stock Unstable CHRNA10 46 42 COc1ccc(/C=C\C(=O)O)cc1Cn1c(C)csc1=O ZINC000217817262 DE For-Sale Unstable AKR1C3 37 41 COC(=O)[C@H]1C[C@H]1C(=O)c1ccc(C)cc1 ZINC000217817281 BD In-Stock Unstable SLC6A1 40 40 COC(=O)[C@H]1C[C@H]1C(=O)c1ccc(C)cc1 ZINC000217817281 BD In-Stock Unstable SLC6A3 18 40 Cc1ccc2cccnc2c1NO ZINC000217817286 AE For-Sale Unstable C0L093_TOBAC 63 36 O=C(N/C=C/c1ccccc1Cl)Nc1ccc2ccccc2c1 ZINC000217817302 DK For-Sale Anodyne UL80 51 40 O=C(N/C=C/c1ccccc1Cl)Nc1ccc2ccccc2c1 ZINC000217817302 DK For-Sale Anodyne IMDH_CRYPV 50 40 COc1cc2ncn(CC(=O)N[C@H](CO)c3ccccc3)c(=O)c2cc1OC ZINC000217817310 GD In-Stock Unstable KDR 50 39 COc1cc2ncn(CC(=O)N[C@H](CO)c3ccccc3)c(=O)c2cc1OC ZINC000217817310 GD In-Stock Unstable SOAT1 0 40 COc1cc2ncn(CC(=O)N[C@H](CO)c3ccccc3)c(=O)c2cc1OC ZINC000217817310 GD In-Stock Unstable PDGFRA 42 36 COc1cc2ncn(CC(=O)N[C@H](CO)c3ccccc3)c(=O)c2cc1OC ZINC000217817310 GD In-Stock Unstable ENPP1 50 30 COc1cc2ncn(CC(=O)N[C@H](CO)c3ccccc3)c(=O)c2cc1OC ZINC000217817310 GD In-Stock Unstable GPR88 0 40 CS(=O)(=O)N1CCC(C(=O)NC[C@@H]2CCCN2c2ccccc2)CC1 ZINC000217817342 FD For-Sale Unstable EPHX2 41 43 O=C(N[C@@H]1CCN2CCC[C@@H]12)c1ccc(Br)c(Cl)c1 ZINC000217817379 EG For-Sale Unstable CHRNA7 17 42 CCc1ccc(C(=O)[C@@H]2C[C@@H]2C(=O)OC)cc1 ZINC000217817381 BE In-Stock Unstable SLC6A1 0 44 COc1ccc2cc(NC(=O)[C@H](C)Nc3ccc4c(cc3=O)[C@@H](NC(C)=O)CCc3cc(OC)c(OC)c(OC)c3-4)cnc2c1 ZINC000217817384 KJ In-Stock Unstable TUBA1A 17 60 CS(=O)(=O)N1CCC(C(=O)NC[C@H]2CCCN2c2ccccc2)CC1 ZINC000217817408 FD For-Sale Unstable EPHX2 41 43 O=C(N[C@H]1CCN2CCC[C@@H]12)c1ccc(Br)c(Cl)c1 ZINC000217817446 EG For-Sale Unstable CHRNA7 17 42 CCc1ccc(C(=O)[C@H]2C[C@@H]2C(=O)OC)cc1 ZINC000217817472 BE In-Stock Unstable SLC6A1 0 44 CC1(C)[C@H]2CC[C@]1(C)[C@@H](OC(=O)C[N+]1(CC(=O)O[C@@H]3C[C@H]4CC[C@]3(C)C4(C)C)CCOCC1)C2 ZINC000217817474 JI In-Stock Unstable ELANE 0 43 COC(=O)C[C@H](c1ccc2c(c1)n(C)c(=O)n2C)c1c(O)c2ccccc2oc1=O ZINC000217817480 HE In-Stock Unstable NQO1 47 48 O=C(Nc1ccccc1)N1CCC[C@H](Cc2nc(C3CC3)no2)C1 ZINC000217817487 EG In-Stock Unstable SMO 42 41 Cc1ccc2cccc(NO)c2n1 ZINC000217817530 AE For-Sale Unstable RELA 19 47 O=C(Nc1ccccc1)N1CCC[C@@H](Cc2nc(C3CC3)no2)C1 ZINC000217817538 EG In-Stock Unstable SMO 42 41 CC(C)(Oc1ccc(Cl)cc1)C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217817548 FI For-Sale Unstable DRD2 17 43 CC(C)(Oc1ccc(Cl)cc1)C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217817548 FI For-Sale Unstable HRH1 16 43 CC(C)(Oc1ccc(Cl)cc1)C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217817548 FI For-Sale Unstable APP 40 38 CC(C)(Oc1ccc(Cl)cc1)C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217817548 FI For-Sale Unstable CACNA1I 49 34 Cc1cc(=O)n(Cc2cccc(/C=C\C(=O)O)c2)cn1 ZINC000217817549 CD For-Sale Unstable PTGER2 24 42 CCc1ccc(C(=O)[C@@H]2C[C@H]2C(=O)OC)cc1 ZINC000217817560 BE In-Stock Unstable SLC6A1 0 44 COC(=O)C[C@@H](c1ccc2c(c1)n(C)c(=O)n2C)c1c(O)c2ccccc2oc1=O ZINC000217817561 HE In-Stock Unstable NQO1 47 48 CC[C@@H](C)c1ccccc1OCC(=O)N1CCN(c2cccc(O)c2)CC1 ZINC000217817591 FH On-Demand Unstable HTR1B 15 40 CC(C)(Oc1ccc(Cl)cc1)C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217817604 FI For-Sale Unstable DRD2 17 43 CC(C)(Oc1ccc(Cl)cc1)C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217817604 FI For-Sale Unstable HRH1 16 43 CC(C)(Oc1ccc(Cl)cc1)C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217817604 FI For-Sale Unstable APP 40 38 CC(C)(Oc1ccc(Cl)cc1)C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217817604 FI For-Sale Unstable CACNA1I 49 34 CCc1ccc(C(=O)[C@H]2C[C@H]2C(=O)OC)cc1 ZINC000217817623 BE In-Stock Unstable SLC6A1 0 44 COCCCOCc1cc(/C=C\C(=O)O)ccc1OC ZINC000217817629 CE For-Sale Unstable APP 20 40 COCCCOCc1cc(/C=C\C(=O)O)ccc1OC ZINC000217817629 CE For-Sale Unstable AKR1C3 30 40 O=C(CCSc1ccc2c(c1)OCCO2)N1CCC[C@@H]1c1ccccn1 ZINC000217817642 FH In-Stock Unstable COLA 112 42 O=C(CCSc1ccc2c(c1)OCCO2)N1CCC[C@@H]1c1ccccn1 ZINC000217817642 FH In-Stock Unstable CPT1A 96 42 O=C(Cc1cccs1)NCC1C[C@@H]2CC[C@H](C1)N2 ZINC000217817647 CD For-Sale Unstable CA5B 33 43 O=C(Cc1cccs1)NCC1C[C@@H]2CC[C@H](C1)N2 ZINC000217817647 CD For-Sale Unstable CA5A 32 43 O=C(Cc1cccs1)NCC1C[C@@H]2CC[C@H](C1)N2 ZINC000217817647 CD For-Sale Unstable GLRA1 21 43 CC[C@H](C)c1ccccc1OCC(=O)N1CCN(c2cccc(O)c2)CC1 ZINC000217817649 FH On-Demand Unstable HTR1B 15 40 CCOC(=O)c1sc(N)nc1-c1cn(C)cn1 ZINC000217817657 CD For-Sale Unstable DHODH 25 40 COCCCOCc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217817714 CE For-Sale Unstable PTGER3 18 46 COCCCOCc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217817714 CE For-Sale Unstable AKR1B10 35 43 COC(=O)[C@@H]1C[C@@H]1C(=O)c1ccc(C(C)C)cc1 ZINC000217817720 BF In-Stock Unstable SLC6A1 27 40 COC(=O)[C@@H]1C[C@@H]1C(=O)c1ccc(C(C)C)cc1 ZINC000217817720 BF In-Stock Unstable SLC6A3 17 40 O=C(CCSc1ccc2c(c1)OCCO2)N1CCC[C@H]1c1ccccn1 ZINC000217817732 FH In-Stock Unstable COLA 112 42 O=C(CCSc1ccc2c(c1)OCCO2)N1CCC[C@H]1c1ccccn1 ZINC000217817732 FH In-Stock Unstable CPT1A 96 42 N#Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217817787 CG For-Sale Unstable MAOB 21 56 N#Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217817787 CG For-Sale Unstable PTGER2 31 43 N#Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217817787 CG For-Sale Unstable PTGER4 0 45 N#Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217817787 CG For-Sale Unstable FFAR1 33 45 N#Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217817787 CG For-Sale Unstable AKR1C3 30 41 CCOc1ccc(C(=O)N2CCC(NC(=O)CCc3ncc(-c4ccc(C)cc4)o3)CC2)cc1 ZINC000217817790 JI On-Demand Unstable SSTR5 43 35 CSC(=S)NCCCN ZINC000217817792 AC For-Sale Unstable PAO 45 36 COC(=O)[C@H]1C[C@@H]1C(=O)c1ccc(C(C)C)cc1 ZINC000217817801 BF In-Stock Unstable SLC6A1 27 40 COC(=O)[C@H]1C[C@@H]1C(=O)c1ccc(C(C)C)cc1 ZINC000217817801 BF In-Stock Unstable SLC6A3 17 40 O=C(O)c1cnn(C2CCCCC2)c1-c1ccc(F)cc1 ZINC000217817807 CH For-Sale Unstable MAPK14 15 42 N#Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217817865 CG For-Sale Unstable MAOA 15 41 N#Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217817865 CG For-Sale Unstable MAOB 66 56 N#Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217817865 CG For-Sale Unstable PTGER2 38 47 N#Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217817865 CG For-Sale Unstable EDNRA 0 41 N#Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217817865 CG For-Sale Unstable PTGER4 32 46 N#Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217817865 CG For-Sale Unstable PTGER3 20 46 N#Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217817865 CG For-Sale Unstable GYS1 43 31 N#Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217817865 CG For-Sale Unstable 17HSDCL 0 40 N#Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217817865 CG For-Sale Unstable FFAR1 58 54 N#Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217817865 CG For-Sale Unstable AKR1C3 34 44 N#Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217817865 CG For-Sale Unstable YOPH 0 40 N#Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217817865 CG For-Sale Unstable FFAR4 25 42 COC(=O)[C@@H]1C[C@H]1C(=O)c1ccc(C(C)C)cc1 ZINC000217817882 BF In-Stock Unstable SLC6A1 27 40 COC(=O)[C@@H]1C[C@H]1C(=O)c1ccc(C(C)C)cc1 ZINC000217817882 BF In-Stock Unstable SLC6A3 17 40 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cc(-c4ccco4)on3)CC2)cc1 ZINC000217817901 HG On-Demand Unstable AVPR1A 18 41 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cc(-c4ccco4)on3)CC2)cc1 ZINC000217817901 HG On-Demand Unstable SSTR5 47 37 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cc(-c4ccco4)on3)CC2)cc1 ZINC000217817901 HG On-Demand Unstable PDK1 41 35 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cc(-c4ccco4)on3)CC2)cc1 ZINC000217817901 HG On-Demand Unstable HPGDS 34 41 O=C(O)/C=C\c1ccccc1COc1cccc(Cl)c1 ZINC000217817941 CI For-Sale Unstable MAOB 28 41 O=C(O)/C=C\c1ccccc1COc1cccc(Cl)c1 ZINC000217817941 CI For-Sale Unstable PTGER2 22 46 O=C(O)/C=C\c1ccccc1COc1cccc(Cl)c1 ZINC000217817941 CI For-Sale Unstable PTGER4 34 55 O=C(O)/C=C\c1ccccc1COc1cccc(Cl)c1 ZINC000217817941 CI For-Sale Unstable PTGER3 34 56 O=C(O)/C=C\c1ccccc1COc1cccc(Cl)c1 ZINC000217817941 CI For-Sale Unstable CDC25B 23 42 O=C(O)/C=C\c1ccccc1COc1cccc(Cl)c1 ZINC000217817941 CI For-Sale Unstable PTGDR 0 56 O=C(O)/C=C\c1ccccc1COc1cccc(Cl)c1 ZINC000217817941 CI For-Sale Unstable PDS 37 44 O=C(NC[C@H]1CCCN1c1ccccc1)C1c2ccccc2Oc2ccccc21 ZINC000217817943 GJ For-Sale Unstable TK 46 44 O=C(NC[C@H]1CCCN1c1ccccc1)C1c2ccccc2Oc2ccccc21 ZINC000217817943 GJ For-Sale Unstable GRM8 41 38 COC(=O)[C@H]1C[C@H]1C(=O)c1ccc(C(C)C)cc1 ZINC000217817961 BF In-Stock Unstable SLC6A1 27 40 COC(=O)[C@H]1C[C@H]1C(=O)c1ccc(C(C)C)cc1 ZINC000217817961 BF In-Stock Unstable SLC6A3 17 40 O=C1NCCCC[C@@H]1N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000217817964 CD For-Sale Unstable DRD2 15 46 O=C1NCCCC[C@@H]1N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000217817964 CD For-Sale Unstable DRD4 44 46 O=C1NCCCC[C@@H]1N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000217817964 CD For-Sale Unstable ACHE 31 40 O=C1NCCCC[C@@H]1N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000217817964 CD For-Sale Unstable DRD3 26 41 O=C1NCCCC[C@@H]1N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000217817964 CD For-Sale Unstable CHRM3 16 41 O=C1NCCCC[C@@H]1N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000217817964 CD For-Sale Unstable SIGMAR1 49 47 O=C1NCCCC[C@@H]1N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000217817964 CD For-Sale Unstable CCR3 18 42 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cnc4onc(C(C)C)c4c3)CC2)cc1 ZINC000217817998 IH On-Demand Unstable SSTR5 53 41 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cnc4onc(C(C)C)c4c3)CC2)cc1 ZINC000217817998 IH On-Demand Unstable SLC6A5 33 41 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cnc4onc(C(C)C)c4c3)CC2)cc1 ZINC000217817998 IH On-Demand Unstable EPHX2 16 40 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cnc4onc(C(C)C)c4c3)CC2)cc1 ZINC000217817998 IH On-Demand Unstable PLAU 18 41 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cnc4onc(C(C)C)c4c3)CC2)cc1 ZINC000217817998 IH On-Demand Unstable MCHR1 24 43 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cnc4onc(C(C)C)c4c3)CC2)cc1 ZINC000217817998 IH On-Demand Unstable HPGDS 36 40 O=C(O)/C=C\c1cccc(OCCOC2CCCCC2)c1 ZINC000217818015 CH For-Sale Unstable NR1H4 26 41 O=C(NC[C@@H]1CCCN1c1ccccc1)C1c2ccccc2Oc2ccccc21 ZINC000217818016 GJ For-Sale Unstable TK 46 44 O=C(NC[C@@H]1CCCN1c1ccccc1)C1c2ccccc2Oc2ccccc21 ZINC000217818016 GJ For-Sale Unstable GRM8 41 38 COc1cccc2ccn(CCC(=O)Nc3ccc4cc[nH]c4c3)c12 ZINC000217818029 EI In-Stock Unstable ENPP1 67 40 O=C1NCCCC[C@@H]1N[C@H]1CCN(Cc2ccccc2)C1 ZINC000217818045 CD For-Sale Unstable DRD2 15 46 O=C1NCCCC[C@@H]1N[C@H]1CCN(Cc2ccccc2)C1 ZINC000217818045 CD For-Sale Unstable DRD4 44 46 O=C1NCCCC[C@@H]1N[C@H]1CCN(Cc2ccccc2)C1 ZINC000217818045 CD For-Sale Unstable ACHE 31 40 O=C1NCCCC[C@@H]1N[C@H]1CCN(Cc2ccccc2)C1 ZINC000217818045 CD For-Sale Unstable DRD3 26 41 O=C1NCCCC[C@@H]1N[C@H]1CCN(Cc2ccccc2)C1 ZINC000217818045 CD For-Sale Unstable CHRM3 16 41 O=C1NCCCC[C@@H]1N[C@H]1CCN(Cc2ccccc2)C1 ZINC000217818045 CD For-Sale Unstable SIGMAR1 49 47 O=C1NCCCC[C@@H]1N[C@H]1CCN(Cc2ccccc2)C1 ZINC000217818045 CD For-Sale Unstable CCR3 18 42 CCCc1ccc(C(=O)[C@@H]2C[C@@H]2C(=O)OC)cc1 ZINC000217818063 BF In-Stock Unstable SLC6A1 0 46 CCCc1ccc(C(=O)[C@@H]2C[C@@H]2C(=O)OC)cc1 ZINC000217818063 BF In-Stock Unstable GRIK2 16 41 O=C(O)/C=C\c1ccc(OCCOC2CCCCC2)cc1 ZINC000217818108 CH For-Sale Unstable ADRB1 15 43 O=C(O)/C=C\c1ccc(OCCOC2CCCCC2)cc1 ZINC000217818108 CH For-Sale Unstable HPGD 20 55 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cc(-c4cccs4)on3)CC2)cc1 ZINC000217818127 IH On-Demand Unstable AVPR1A 18 41 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cc(-c4cccs4)on3)CC2)cc1 ZINC000217818127 IH On-Demand Unstable CNR2 19 46 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cc(-c4cccs4)on3)CC2)cc1 ZINC000217818127 IH On-Demand Unstable SSTR5 48 38 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cc(-c4cccs4)on3)CC2)cc1 ZINC000217818127 IH On-Demand Unstable SLC6A5 36 40 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cc(-c4cccs4)on3)CC2)cc1 ZINC000217818127 IH On-Demand Unstable PDK1 40 33 CCOc1ccc(C(=O)N2CCC(NC(=O)c3cc(-c4cccs4)on3)CC2)cc1 ZINC000217818127 IH On-Demand Unstable ETHR 50 37 O=C(Nc1ccc(C(F)(F)F)cc1)N1CCC[C@H](Cc2nc(C3CC3)no2)C1 ZINC000217818140 GI In-Stock Unstable EPHX2 37 45 O=C(Nc1ccc(C(F)(F)F)cc1)N1CCC[C@H](Cc2nc(C3CC3)no2)C1 ZINC000217818140 GI In-Stock Unstable TRPM8 45 39 CCOC(=O)c1c[nH]c(=O)c2c1OC(=O)C[C@@H]2c1ccccc1OC ZINC000217818141 EE In-Stock Unstable DHFR-TS 0 44 CCCc1ccc(C(=O)[C@H]2C[C@@H]2C(=O)OC)cc1 ZINC000217818144 BF In-Stock Unstable SLC6A1 0 46 CCCc1ccc(C(=O)[C@H]2C[C@@H]2C(=O)OC)cc1 ZINC000217818144 BF In-Stock Unstable GRIK2 16 41 CN(C)S(=O)(=O)c1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217818154 GE For-Sale Unstable CA2 15 42 CN(C)S(=O)(=O)c1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217818154 GE For-Sale Unstable NPY2R 15 40 CN(C)S(=O)(=O)c1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217818154 GE For-Sale Unstable LIMK2 42 37 CC1(C)C[C@H]2C[C@@](C)(CN2C(=O)N/C=C/c2ccccc2Cl)C1 ZINC000217818203 EJ For-Sale Unstable AVPR2 17 47 CC1(C)C[C@H]2C[C@@](C)(CN2C(=O)N/C=C/c2ccccc2Cl)C1 ZINC000217818203 EJ For-Sale Unstable AVPR1A 38 44 CCCc1ccc(C(=O)[C@@H]2C[C@H]2C(=O)OC)cc1 ZINC000217818223 BF In-Stock Unstable SLC6A1 0 46 CCCc1ccc(C(=O)[C@@H]2C[C@H]2C(=O)OC)cc1 ZINC000217818223 BF In-Stock Unstable GRIK2 16 41 CCOC(=O)c1c[nH]c(=O)c2c1OC(=O)C[C@H]2c1ccccc1OC ZINC000217818230 EE In-Stock Unstable DHFR-TS 0 44 O=C(Nc1ccc(C(F)(F)F)cc1)N1CCC[C@@H](Cc2nc(C3CC3)no2)C1 ZINC000217818231 GI In-Stock Unstable EPHX2 37 45 O=C(Nc1ccc(C(F)(F)F)cc1)N1CCC[C@@H](Cc2nc(C3CC3)no2)C1 ZINC000217818231 GI In-Stock Unstable TRPM8 45 39 CN(C)S(=O)(=O)c1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217818232 GE For-Sale Unstable CA2 15 42 CN(C)S(=O)(=O)c1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217818232 GE For-Sale Unstable NPY2R 15 40 CN(C)S(=O)(=O)c1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217818232 GE For-Sale Unstable LIMK2 42 37 CCOc1ccc(C(=O)N2CCC(NC(=O)c3occc3COc3ccccc3)CC2)cc1 ZINC000217818240 II On-Demand Unstable DRD4 15 40 CCOc1ccc(C(=O)N2CCC(NC(=O)c3occc3COc3ccccc3)CC2)cc1 ZINC000217818240 II On-Demand Unstable AVPR1A 23 44 CCOc1ccc(C(=O)N2CCC(NC(=O)c3occc3COc3ccccc3)CC2)cc1 ZINC000217818240 II On-Demand Unstable SSTR5 45 36 CCOc1ccc(C(=O)N2CCC(NC(=O)c3occc3COc3ccccc3)CC2)cc1 ZINC000217818240 II On-Demand Unstable ADAM17 65 38 CCOc1ccc(C(=O)N2CCC(NC(=O)c3occc3COc3ccccc3)CC2)cc1 ZINC000217818240 II On-Demand Unstable SLC6A5 37 43 CCOc1ccc(C(=O)N2CCC(NC(=O)c3occc3COc3ccccc3)CC2)cc1 ZINC000217818240 II On-Demand Unstable EPHX2 16 40 CCOc1ccc(C(=O)N2CCC(NC(=O)c3occc3COc3ccccc3)CC2)cc1 ZINC000217818240 II On-Demand Unstable HPGDS 32 40 Cc1cc(C(N)=O)ccc1N[C@H]1C[C@H](C)CC[C@H]1C(C)C ZINC000217818246 CH For-Sale Unstable TRPM8 17 51 CCCc1ccc(C(=O)[C@H]2C[C@H]2C(=O)OC)cc1 ZINC000217818303 BF In-Stock Unstable SLC6A1 0 46 CCCc1ccc(C(=O)[C@H]2C[C@H]2C(=O)OC)cc1 ZINC000217818303 BF In-Stock Unstable GRIK2 16 41 Cc1ccccc1NC(=O)N1CCC[C@H](Cc2nc(C3CC3)no2)C1 ZINC000217818327 EH In-Stock Unstable SMO 32 45 Cc1cc(C(N)=O)ccc1N[C@H]1C[C@@H](C)CC[C@H]1C(C)C ZINC000217818328 CH For-Sale Unstable TRPM8 17 51 COC(=O)C[C@@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc2c(c1)OCO2 ZINC000217818329 GF In-Stock Unstable EDNRB 66 35 COC(=O)C[C@@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc2c(c1)OCO2 ZINC000217818329 GF In-Stock Unstable EDNRA 65 39 COC(=O)C[C@@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc2c(c1)OCO2 ZINC000217818329 GF In-Stock Unstable BMP1 40 38 COC(=O)C[C@@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc2c(c1)OCO2 ZINC000217818329 GF In-Stock Unstable RORC 33 41 COc1ccc(Br)c(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217818348 GH For-Sale Unstable DRD2 42 49 COc1ccc(Br)c(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217818348 GH For-Sale Unstable DRD4 40 31 COc1ccc(Br)c(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217818348 GH For-Sale Unstable DRD3 34 51 COc1ccc(Br)c(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217818348 GH For-Sale Unstable SIGMAR1 16 51 COc1ccc(Br)c(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217818348 GH For-Sale Unstable MTNR1A 43 35 COc1ccc(Br)c(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217818348 GH For-Sale Unstable MTNR1B 43 35 COc1ccc(Br)c(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217818348 GH For-Sale Unstable CHRNA10 53 40 COc1ccc(Br)c(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217818348 GH For-Sale Unstable AKR1C2 41 34 COc1ccc(Br)c(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217818348 GH For-Sale Unstable ACKR3 66 35 CCOc1ccc(C(=O)N2CCC(NC(=O)CCc3ncc(-c4ccccc4)o3)CC2)cc1 ZINC000217818350 II On-Demand Unstable AVPR1A 19 42 CCOc1ccc(C(=O)N2CCC(NC(=O)CCc3ncc(-c4ccccc4)o3)CC2)cc1 ZINC000217818350 II On-Demand Unstable SSTR5 42 38 CCOc1ccc(C(=O)N2CCC(NC(=O)CCc3ncc(-c4ccccc4)o3)CC2)cc1 ZINC000217818350 II On-Demand Unstable TNKS 54 30 CCOc1ccc(C(=O)N2CCC(NC(=O)CCc3ncc(-c4ccccc4)o3)CC2)cc1 ZINC000217818350 II On-Demand Unstable ADIPOR1 0 41 CCOc1ccc(C(=O)N2CCC(NC(=O)CCc3ncc(-c4ccccc4)o3)CC2)cc1 ZINC000217818350 II On-Demand Unstable ADIPOR2 0 41 CN(C)c1cccc(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217818384 DI For-Sale Unstable KCNK3 44 42 COC(=O)C[C@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc2c(c1)OCO2 ZINC000217818396 GF In-Stock Unstable EDNRB 66 35 COC(=O)C[C@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc2c(c1)OCO2 ZINC000217818396 GF In-Stock Unstable EDNRA 65 39 COC(=O)C[C@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc2c(c1)OCO2 ZINC000217818396 GF In-Stock Unstable BMP1 40 38 COC(=O)C[C@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc2c(c1)OCO2 ZINC000217818396 GF In-Stock Unstable RORC 33 41 Cc1ccccc1NC(=O)N1CCC[C@@H](Cc2nc(C3CC3)no2)C1 ZINC000217818402 EH In-Stock Unstable SMO 32 45 COc1ccc(Br)c(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217818436 GH For-Sale Unstable DRD2 42 49 COc1ccc(Br)c(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217818436 GH For-Sale Unstable DRD4 40 31 COc1ccc(Br)c(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217818436 GH For-Sale Unstable DRD3 34 51 COc1ccc(Br)c(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217818436 GH For-Sale Unstable SIGMAR1 16 51 COc1ccc(Br)c(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217818436 GH For-Sale Unstable MTNR1A 43 35 COc1ccc(Br)c(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217818436 GH For-Sale Unstable MTNR1B 43 35 COc1ccc(Br)c(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217818436 GH For-Sale Unstable CHRNA10 53 40 COc1ccc(Br)c(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217818436 GH For-Sale Unstable AKR1C2 41 34 COc1ccc(Br)c(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217818436 GH For-Sale Unstable ACKR3 66 35 CCN(CCOc1ccc(/C=C\C(=O)O)cc1)CC(C)C ZINC000217818455 CG On-Demand Unstable ERG2 17 43 CCOc1ccc(C(=O)N2CCC(NC(=O)CCc3ncc(-c4ccccc4Cl)o3)CC2)cc1 ZINC000217818467 JJ On-Demand Unstable AVPR1A 18 40 CN1CCc2nc(NC(=O)N/C=C/c3ccccc3Cl)sc2C1 ZINC000217818482 EH For-Sale Unstable F10 28 49 CCCCOc1ccc(NC(=O)N2CCC[C@H](Cc3nc(C4CC4)no3)C2)cc1 ZINC000217818507 GJ In-Stock Unstable PDGFRB 43 37 CCCCOc1ccc(NC(=O)N2CCC[C@H](Cc3nc(C4CC4)no3)C2)cc1 ZINC000217818507 GJ In-Stock Unstable HRH3 27 42 Cc1onc(-c2ccccc2Cl)c1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217818526 GJ For-Sale Unstable GPBAR1 37 47 CCN(CCOc1cccc(/C=C\C(=O)O)c1)C(C)C ZINC000217818566 CF For-Sale Unstable NR1H4 45 38 CCN(CCOc1cccc(/C=C\C(=O)O)c1)C(C)C ZINC000217818566 CF For-Sale Unstable AKR1C3 40 40 CCCCOc1ccc(NC(=O)N2CCC[C@@H](Cc3nc(C4CC4)no3)C2)cc1 ZINC000217818582 GJ In-Stock Unstable PDGFRB 47 37 CCCCOc1ccc(NC(=O)N2CCC[C@@H](Cc3nc(C4CC4)no3)C2)cc1 ZINC000217818582 GJ In-Stock Unstable HRH3 27 42 CCCCOc1ccc(NC(=O)N2CCC[C@@H](Cc3nc(C4CC4)no3)C2)cc1 ZINC000217818582 GJ In-Stock Unstable EPHX2 19 44 CCOc1ccc(C(=O)N2CCC(NC(=O)CCc3ncc(-c4ccc(Cl)cc4)o3)CC2)cc1 ZINC000217818593 JJ On-Demand Unstable SSTR5 40 35 O=C(N/C=C/c1ccccc1Cl)Nc1ccc2nc[nH]c2c1 ZINC000217818600 DI For-Sale Anodyne NR2E3 59 33 Cc1onc(-c2ccccc2Cl)c1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217818603 GJ For-Sale Unstable GPBAR1 37 47 CCN(CCOc1ccc(/C=C\C(=O)O)cc1)C(C)C ZINC000217818675 CF On-Demand Unstable AHR 20 42 CCN(CCOc1ccc(/C=C\C(=O)O)cc1)C(C)C ZINC000217818675 CF On-Demand Unstable PLA2G4B 44 31 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCOCC2)cc1 ZINC000217818695 IE For-Sale Unstable TGM2 64 46 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCOCC2)cc1 ZINC000217818695 IE For-Sale Unstable F13A1 56 39 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCOCC2)cc1 ZINC000217818695 IE For-Sale Unstable NAMPT 39 42 CCOc1ccc(C(=O)N2CCC(NC(=O)CCc3ncc(-c4ccc(F)cc4F)o3)CC2)cc1 ZINC000217818701 JI On-Demand Unstable SSTR5 43 36 O=C(O)/C=C\c1ccccc1-n1cc(I)cn1 ZINC000217818733 EF For-Sale Anodyne PTGER2 36 42 O=C(O)/C=C\c1ccccc1-n1cc(I)cn1 ZINC000217818733 EF For-Sale Anodyne PTGER4 0 42 O=C(O)/C=C\c1ccccc1-n1cc(I)cn1 ZINC000217818733 EF For-Sale Anodyne PTGER3 16 42 C=CC[C@@](C)(NNC(=O)c1ccccc1)c1ccccc1 ZINC000217818768 CG For-Sale Unstable ECR 43 41 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCOCC2)cc1 ZINC000217818769 IE For-Sale Unstable TGM2 64 46 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCOCC2)cc1 ZINC000217818769 IE For-Sale Unstable F13A1 56 39 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCOCC2)cc1 ZINC000217818769 IE For-Sale Unstable NAMPT 39 42 NC(=O)c1ccccc1NC(=O)N/C=C/c1ccccc1Cl ZINC000217818791 DG For-Sale Unstable PAGA 0 45 O=C(C[C@H](c1ccc2c(c1)OCO2)c1c(O)nc2ccccn2c1=O)NCCc1ccc(O)c(O)c1 ZINC000217818794 JE In-Stock Unstable NOS2 75 36 C[C@@H](CNC(=O)c1ccc(Cl)c([N+](=O)[O-])c1)N(C)C1CC1 ZINC000217818801 DE On-Demand Unstable TAAR1 15 43 CCOc1ccc(C(=O)N2CCC(NC(=O)CCc3ncc(-c4ccccc4F)o3)CC2)cc1 ZINC000217818807 JI On-Demand Unstable AVPR1A 18 40 CCCCN(C1CC1)[C@H](c1cccc(Cl)c1)[C@@H](N)CC ZINC000217818816 CI For-Sale Unstable OPRL1 0 45 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(OC(F)(F)F)cc1 ZINC000217818856 FH For-Sale Unstable GCGR 37 40 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(OC(F)(F)F)cc1 ZINC000217818856 FH For-Sale Unstable GRIN2B 40 40 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(OC(F)(F)F)cc1 ZINC000217818856 FH For-Sale Unstable TRPV1 17 52 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(OC(F)(F)F)cc1 ZINC000217818856 FH For-Sale Unstable ITGA4 41 30 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(OC(F)(F)F)cc1 ZINC000217818856 FH For-Sale Unstable EPHX2 40 38 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(OC(F)(F)F)cc1 ZINC000217818856 FH For-Sale Unstable NOD2 24 43 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(OC(F)(F)F)cc1 ZINC000217818856 FH For-Sale Unstable ACKR3 56 32 O=C(C[C@@H](c1ccc2c(c1)OCO2)c1c(O)nc2ccccn2c1=O)NCCc1ccc(O)c(O)c1 ZINC000217818860 JE In-Stock Unstable NOS2 75 36 C[C@H](CNC(=O)c1ccc(Cl)c([N+](=O)[O-])c1)N(C)C1CC1 ZINC000217818879 DE On-Demand Unstable TAAR1 15 43 CCCCN(C1CC1)[C@@H](c1cccc(Cl)c1)[C@@H](N)CC ZINC000217818898 CI For-Sale Unstable OPRL1 0 45 CCOc1ccc(C(=O)N2CCC(NC(=O)CSc3ccc(C(C)(C)C)cc3)CC2)cc1 ZINC000217818909 JJ On-Demand Unstable AVPR1A 20 45 CCOc1ccc(C(=O)N2CCC(NC(=O)CSc3ccc(C(C)(C)C)cc3)CC2)cc1 ZINC000217818909 JJ On-Demand Unstable SSTR5 45 39 CCOc1ccc(C(=O)N2CCC(NC(=O)CSc3ccc(C(C)(C)C)cc3)CC2)cc1 ZINC000217818909 JJ On-Demand Unstable SLC6A5 36 43 CCOc1ccc(C(=O)N2CCC(NC(=O)CSc3ccc(C(C)(C)C)cc3)CC2)cc1 ZINC000217818909 JJ On-Demand Unstable EPHX2 33 40 CCOc1ccc(C(=O)N2CCC(NC(=O)CSc3ccc(C(C)(C)C)cc3)CC2)cc1 ZINC000217818909 JJ On-Demand Unstable L3MBTL3 45 34 CCOc1ccc(C(=O)N2CCC(NC(=O)CSc3ccc(C(C)(C)C)cc3)CC2)cc1 ZINC000217818909 JJ On-Demand Unstable LUXN 0 41 CCOc1ccc(C(=O)N2CCC(NC(=O)CSc3ccc(C(C)(C)C)cc3)CC2)cc1 ZINC000217818909 JJ On-Demand Unstable ADIPOR1 0 41 CCOc1ccc(C(=O)N2CCC(NC(=O)CSc3ccc(C(C)(C)C)cc3)CC2)cc1 ZINC000217818909 JJ On-Demand Unstable ADIPOR2 0 41 O=C(O)/C=C\c1ccccc1CN1CCN(CCO)CC1 ZINC000217818917 CC For-Sale Unstable PTGER2 40 48 O=C(O)/C=C\c1ccccc1CN1CCN(CCO)CC1 ZINC000217818917 CC For-Sale Unstable PTGER4 0 48 O=C(O)/C=C\c1ccccc1CN1CCN(CCO)CC1 ZINC000217818917 CC For-Sale Unstable PTGER3 17 48 CCN(CCO)C(=S)SC ZINC000217818918 AC For-Sale Unstable CAH2 0 41 CCN(CCO)C(=S)SC ZINC000217818918 AC For-Sale Unstable CAH1 0 41 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(OC(F)(F)F)cc1 ZINC000217818925 FH For-Sale Unstable GCGR 37 40 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(OC(F)(F)F)cc1 ZINC000217818925 FH For-Sale Unstable GRIN2B 40 40 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(OC(F)(F)F)cc1 ZINC000217818925 FH For-Sale Unstable TRPV1 17 52 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(OC(F)(F)F)cc1 ZINC000217818925 FH For-Sale Unstable ITGA4 41 30 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(OC(F)(F)F)cc1 ZINC000217818925 FH For-Sale Unstable EPHX2 40 38 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(OC(F)(F)F)cc1 ZINC000217818925 FH For-Sale Unstable NOD2 24 43 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(OC(F)(F)F)cc1 ZINC000217818925 FH For-Sale Unstable ACKR3 56 32 COC(=O)C[C@H](c1cc(OC)c2c(c1)OCO2)c1c(O)cc(C)n(CC(=O)O)c1=O ZINC000217818973 HD In-Stock Unstable RORC 42 40 O=C(N/C=C/c1ccccc1Cl)Nc1cccc(Br)c1 ZINC000217818982 FJ For-Sale Anodyne KCNK3 45 40 Nc1nc(/C=C\c2cccc3ccccc23)cs1 ZINC000217819014 CI For-Sale Unstable CHAT 76 42 O=C(O)/C=C\c1ccc(CN2CCN(CCO)CC2)cc1 ZINC000217819016 CC For-Sale Unstable SIGMAR1 31 45 O=C(O)/C=C\c1ccc(CN2CCN(CCO)CC2)cc1 ZINC000217819016 CC For-Sale Unstable CACNA1G 16 41 COc1ccc(OC)c(-c2cc(C(=O)NC[C@@H]3CCCN3c3ccccc3)n(C)n2)c1 ZINC000217819026 HH For-Sale Unstable DRD2 34 41 COc1ccc(OC)c(-c2cc(C(=O)NC[C@@H]3CCCN3c3ccccc3)n(C)n2)c1 ZINC000217819026 HH For-Sale Unstable DRD3 18 41 COc1ccc(OC)c(-c2cc(C(=O)NC[C@@H]3CCCN3c3ccccc3)n(C)n2)c1 ZINC000217819026 HH For-Sale Unstable ACKR3 65 35 COC(=O)C[C@@H](c1cc(OC)c2c(c1)OCO2)c1c(O)cc(C)n(CC(=O)O)c1=O ZINC000217819064 HD In-Stock Unstable RORC 42 40 COC(=O)[C@@H]1C[C@@H]1C(=O)c1cccc2ccccc12 ZINC000217819071 CF In-Stock Unstable SLC6A1 19 48 COc1ccc(OC)c(-c2cc(C(=O)NC[C@H]3CCCN3c3ccccc3)n(C)n2)c1 ZINC000217819104 HH For-Sale Unstable DRD2 34 41 COc1ccc(OC)c(-c2cc(C(=O)NC[C@H]3CCCN3c3ccccc3)n(C)n2)c1 ZINC000217819104 HH For-Sale Unstable DRD3 18 41 COc1ccc(OC)c(-c2cc(C(=O)NC[C@H]3CCCN3c3ccccc3)n(C)n2)c1 ZINC000217819104 HH For-Sale Unstable ACKR3 65 35 O=C(O)/C=C\c1cccc(CN2CCN(CCO)CC2)c1 ZINC000217819125 CC For-Sale Unstable SIGMAR1 46 45 O=C(O)/C=C\c1cccc(CN2CCN(CCO)CC2)c1 ZINC000217819125 CC For-Sale Unstable HDAC1 15 42 O=C(O)/C=C\c1cccc(CN2CCN(CCO)CC2)c1 ZINC000217819125 CC For-Sale Unstable FAAH 20 40 O=C(O)/C=C\c1cccc(CN2CCN(CCO)CC2)c1 ZINC000217819125 CC For-Sale Unstable AKR1C3 40 38 COC(=O)[C@H]1C[C@@H]1C(=O)c1cccc2ccccc12 ZINC000217819148 CF In-Stock Unstable SLC6A1 19 48 CCOc1ccc(CCNC(=O)N/C=C/c2ccccc2Cl)cc1OCC ZINC000217819185 GJ For-Sale Unstable CAN2 0 40 COc1ccc(C(=O)/C=C\c2ccc(OC)cc2OC)c(F)c1 ZINC000217819200 DH On-Demand Mild CYP1B1 63 55 COc1ccc(C(=O)/C=C\c2ccc(OC)cc2OC)c(F)c1 ZINC000217819200 DH On-Demand Mild CYP1A1 51 55 COc1ccc(C(=O)/C=C\c2ccc(OC)cc2OC)c(F)c1 ZINC000217819200 DH On-Demand Mild TUBB1 29 40 COc1ccc(C(=O)/C=C\c2ccc(OC)cc2OC)c(F)c1 ZINC000217819200 DH On-Demand Mild CYP1A2 20 55 COc1ccc(C(=O)/C=C\c2ccc(OC)cc2OC)c(F)c1 ZINC000217819200 DH On-Demand Mild ABCG2 26 60 COc1ccc(C(=O)/C=C\c2ccc(OC)cc2OC)c(F)c1 ZINC000217819200 DH On-Demand Mild CYSP_PLAFA 90 71 COCC(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217819204 BD For-Sale Unstable SLC18A2 21 40 CN(Cc1cccc(/C=C\C(=O)O)c1)Cc1cccs1 ZINC000217819210 CG For-Sale Unstable HCAR2 28 42 CN(Cc1cccc(/C=C\C(=O)O)c1)Cc1cccs1 ZINC000217819210 CG For-Sale Unstable AKR1C3 40 39 O=C(CCN1CCS[C@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217819217 EI On-Demand Unstable DRD2 30 42 O=C(CCN1CCS[C@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217819217 EI On-Demand Unstable HTR2A 24 45 O=C(CCN1CCS[C@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217819217 EI On-Demand Unstable SLC6A1 69 34 O=C(CCN1CCS[C@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217819217 EI On-Demand Unstable SIGMAR1 15 49 O=C(CCN1CCS[C@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217819217 EI On-Demand Unstable SLC18A3 20 49 O=C(CCN1CCS[C@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217819217 EI On-Demand Unstable CYP2J2 48 34 COC(=O)[C@@H]1C[C@H]1C(=O)c1cccc2ccccc12 ZINC000217819219 CF In-Stock Unstable SLC6A1 19 48 Cc1nn(C)c(C)c1C(=O)Nc1ccnn1Cc1cccc(Cl)c1Cl ZINC000217819265 GH On-Demand Unstable P2RX7 22 42 CC(C)(C)c1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217819280 EK For-Sale Unstable TRPV1 22 43 CC(C)(C)c1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217819280 EK For-Sale Unstable IMDH_CRYPV 51 35 O=C(CCN1CCS[C@@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217819288 EI On-Demand Unstable DRD2 30 42 O=C(CCN1CCS[C@@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217819288 EI On-Demand Unstable HTR2A 24 45 O=C(CCN1CCS[C@@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217819288 EI On-Demand Unstable SLC6A1 69 34 O=C(CCN1CCS[C@@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217819288 EI On-Demand Unstable SIGMAR1 15 49 O=C(CCN1CCS[C@@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217819288 EI On-Demand Unstable SLC18A3 20 49 O=C(CCN1CCS[C@@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217819288 EI On-Demand Unstable CYP2J2 48 34 COCC(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217819291 BD For-Sale Unstable SLC18A2 21 40 COC(=O)[C@H]1C[C@H]1C(=O)c1cccc2ccccc12 ZINC000217819296 CF In-Stock Unstable SLC6A1 19 48 CCCCCCCCCCCCC/C=C/[C@@H](O)[C@H](CN[C@@H]1C=C(CO)[C@H](O)[C@@H](O)[C@H]1O)NC(=O)CCCCCCCCCCCCCCC ZINC000217819342 KK Annotated Unstable SELP 34 46 O=C(Cc1ccc(Cl)cc1)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217819351 EF In-Stock Unstable CHRNA4 43 55 Clc1ccc2c(c1Br)CCNC2 ZINC000217819353 BF For-Sale Unstable PNMT 46 52 Cc1ccccc1-c1nnc(S[C@@H](C(N)=O)c2ccc(F)cc2)n1Cc1ccco1 ZINC000217819407 HI On-Demand Unstable HCRTR2 25 56 CN(Cc1ccc(F)c(/C=C\C(=O)O)c1)Cc1cccs1 ZINC000217819445 DH For-Sale Unstable PTGER2 21 41 Clc1c(Br)ccc2c1CCNC2 ZINC000217819455 BF For-Sale Unstable PNMT 43 47 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)NCCc3ccccc3)[C@H]21 ZINC000217819463 JG In-Stock Unstable TSHR 43 34 Cc1ccccc1-c1nnc(S[C@H](C(N)=O)c2ccc(F)cc2)n1Cc1ccco1 ZINC000217819478 HI On-Demand Unstable HCRTR2 25 56 Clc1cc2c(cc1Br)CCNC2 ZINC000217819518 BF For-Sale Unstable PNMT 40 50 CN(C)C1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217819522 CE For-Sale Unstable DRD2 23 42 CN(C)C1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217819522 CE For-Sale Unstable DRD4 53 43 CN(C)C1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217819522 CE For-Sale Unstable ACHE 41 49 CN(C)C1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217819522 CE For-Sale Unstable DRD3 15 40 CN(C)C1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217819522 CE For-Sale Unstable CHRM3 25 42 CN(C)C1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217819522 CE For-Sale Unstable SIGMAR1 55 62 CN(C)C1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217819522 CE For-Sale Unstable CCR3 32 44 CN(C)C1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217819522 CE For-Sale Unstable MCHR1 34 40 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)NCCc3ccccc3)[C@@H]21 ZINC000217819535 JG In-Stock Unstable TSHR 43 34 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(NS(=O)(=O)c2cccc(F)c2)cc1 ZINC000217819585 JI For-Sale Unstable SFRP1 71 33 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(NS(=O)(=O)c2cccc(F)c2)cc1 ZINC000217819585 JI For-Sale Unstable LIMK2 39 40 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(NS(=O)(=O)c2cccc(F)c2)cc1 ZINC000217819585 JI For-Sale Unstable WNT3 55 31 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(NS(=O)(=O)c2cccc(F)c2)cc1 ZINC000217819585 JI For-Sale Unstable ACKR3 56 33 COc1ccc(O)c(C(=O)Nc2ccc(-c3csc(C)n3)cc2)c1 ZINC000217819586 EI On-Demand Unstable F10 0 55 COc1ccc(O)c(C(=O)Nc2ccc(-c3csc(C)n3)cc2)c1 ZINC000217819586 EI On-Demand Unstable SCN10A 49 38 COc1ccc(O)c(C(=O)Nc2ccc(-c3csc(C)n3)cc2)c1 ZINC000217819586 EI On-Demand Unstable U38 0 55 COc1ccc(O)c(C(=O)Nc2ccc(-c3csc(C)n3)cc2)c1 ZINC000217819586 EI On-Demand Unstable Q25615_ONCVO 68 37 C[C@@H](C1CC1)N(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217819639 CF For-Sale Unstable NR1H4 46 35 C[C@@H](c1ccc(Cl)cc1)N(C)[C@@H](C(=O)O)c1ccccc1 ZINC000217819644 DI For-Sale Unstable SLC6A9 0 42 C[C@@H](c1ccc(Cl)cc1)N(C)[C@@H](C(=O)O)c1ccccc1 ZINC000217819644 DI For-Sale Unstable UTS2 53 42 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(NS(=O)(=O)c2cccc(F)c2)cc1 ZINC000217819676 JI For-Sale Unstable SFRP1 71 33 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(NS(=O)(=O)c2cccc(F)c2)cc1 ZINC000217819676 JI For-Sale Unstable LIMK2 39 40 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(NS(=O)(=O)c2cccc(F)c2)cc1 ZINC000217819676 JI For-Sale Unstable WNT3 55 31 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(NS(=O)(=O)c2cccc(F)c2)cc1 ZINC000217819676 JI For-Sale Unstable ACKR3 56 33 O=C(N/C=C/c1ccccc1Cl)Nc1ccc2cn[nH]c2c1 ZINC000217819688 DI For-Sale Anodyne MAOB 20 42 O=C(N/C=C/c1ccccc1Cl)Nc1ccc2cn[nH]c2c1 ZINC000217819688 DI For-Sale Anodyne NR2E3 52 33 C[C@H](C1CC1)N(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217819710 CF For-Sale Unstable NR1H4 46 35 CC[C@@H](C)N(C)CCN[C@@H]1CCc2cccnc21 ZINC000217819716 BE On-Demand Unstable CXCR4 40 38 C[C@H](c1ccc(Cl)cc1)N(C)[C@@H](C(=O)O)c1ccccc1 ZINC000217819728 DI For-Sale Unstable SLC6A9 0 42 C[C@H](c1ccc(Cl)cc1)N(C)[C@@H](C(=O)O)c1ccccc1 ZINC000217819728 DI For-Sale Unstable UTS2 53 42 CC[C@H](C)N(C)CCN[C@@H]1CCc2cccnc21 ZINC000217819793 BE On-Demand Unstable CXCR4 40 38 O=C(CNS(=O)(=O)c1cccc(Cl)c1)NC[C@H]1CCCN1c1ccccc1 ZINC000217819796 HE For-Sale Unstable DRD2 15 40 O=C(CNS(=O)(=O)c1cccc(Cl)c1)NC[C@H]1CCCN1c1ccccc1 ZINC000217819796 HE For-Sale Unstable FBP1 18 45 O=C(CNS(=O)(=O)c1cccc(Cl)c1)NC[C@H]1CCCN1c1ccccc1 ZINC000217819796 HE For-Sale Unstable ADAMTS5 22 40 O=C(CNS(=O)(=O)c1cccc(Cl)c1)NC[C@H]1CCCN1c1ccccc1 ZINC000217819796 HE For-Sale Unstable SFRP1 62 36 CC[C@@H]1CCCC[C@@H]1NC(=O)C[C@@H](N)c1ccccc1 ZINC000217819805 CG On-Demand Unstable AMY2 45 32 NC(=O)c1ccc(N2CCCC2)c(NC(=O)Cn2nnc(-c3ccc(Cl)cc3)n2)c1 ZINC000217819808 IE On-Demand Unstable CNR1 51 31 NC(=O)c1ccc(N2CCCC2)c(NC(=O)Cn2nnc(-c3ccc(Cl)cc3)n2)c1 ZINC000217819808 IE On-Demand Unstable KCNQ2 43 44 NC(=O)c1ccc(N2CCCC2)c(NC(=O)Cn2nnc(-c3ccc(Cl)cc3)n2)c1 ZINC000217819808 IE On-Demand Unstable SCARB1 37 40 O=C(CNS(=O)(=O)c1cccc(Cl)c1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217819866 HE For-Sale Unstable DRD2 15 40 O=C(CNS(=O)(=O)c1cccc(Cl)c1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217819866 HE For-Sale Unstable FBP1 18 45 O=C(CNS(=O)(=O)c1cccc(Cl)c1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217819866 HE For-Sale Unstable ADAMTS5 22 40 O=C(CNS(=O)(=O)c1cccc(Cl)c1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217819866 HE For-Sale Unstable SFRP1 62 36 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217819884 GF For-Sale Unstable CA2 104 62 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217819884 GF For-Sale Unstable CA6 25 41 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217819884 GF For-Sale Unstable CA1 95 62 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217819884 GF For-Sale Unstable CA7 51 56 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217819884 GF For-Sale Unstable CA13 22 41 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217819884 GF For-Sale Unstable CA5B 62 56 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217819884 GF For-Sale Unstable CA4 67 57 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217819884 GF For-Sale Unstable CA5A 64 56 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217819884 GF For-Sale Unstable CA14 43 53 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217819884 GF For-Sale Unstable CA12 74 62 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217819884 GF For-Sale Unstable CA9 81 62 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217819884 GF For-Sale Unstable CYNT 26 45 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217819884 GF For-Sale Unstable NCE103 44 54 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217819884 GF For-Sale Unstable LIG1 0 45 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217819884 GF For-Sale Unstable MTCA1 43 39 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217819884 GF For-Sale Unstable P96878_MYCTU 62 51 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217819884 GF For-Sale Unstable CA 0 40 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217819884 GF For-Sale Unstable CAN2 0 51 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217819884 GF For-Sale Unstable A6YCJ1_9METZ 25 50 CC[C@H]1CCCC[C@@H]1NC(=O)C[C@@H](N)c1ccccc1 ZINC000217819891 CG For-Sale Unstable AMY2 45 32 O=C(C[C@@H]1NC(=O)N(Cc2ccccc2)C1=O)NCCc1ccc(O)cc1 ZINC000217819916 FD In-Stock Unstable NCE103 22 45 O=C(C[C@@H]1NC(=O)N(Cc2ccccc2)C1=O)NCCc1ccc(O)cc1 ZINC000217819916 FD In-Stock Unstable P96878_MYCTU 17 45 O=C(C[C@@H]1NC(=O)N(Cc2ccccc2)C1=O)NCCc1ccc(O)cc1 ZINC000217819916 FD In-Stock Unstable CAN2 0 45 O=C(CNS(=O)(=O)c1cccc(F)c1)NC[C@H]1CCCN1c1ccccc1 ZINC000217819957 GD For-Sale Unstable HTR6 34 42 O=C(CNS(=O)(=O)c1cccc(F)c1)NC[C@H]1CCCN1c1ccccc1 ZINC000217819957 GD For-Sale Unstable SFRP1 104 35 O=C(CNS(=O)(=O)c1cccc(F)c1)NC[C@H]1CCCN1c1ccccc1 ZINC000217819957 GD For-Sale Unstable WNT3 72 34 O=C(N/C=C/c1ccccc1Cl)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217819975 HK For-Sale Anodyne JUN 22 43 O=C(N/C=C/c1ccccc1Cl)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217819975 HK For-Sale Anodyne PTPA 0 45 CC[C@@H]1CCCC[C@H]1NC(=O)C[C@@H](N)c1ccccc1 ZINC000217819979 CG On-Demand Unstable AMY2 45 32 COc1ccc(CN2CCCC2=O)cc1/C=C\C(=O)O ZINC000217819993 CD For-Sale Unstable PTGER2 34 58 COc1ccc(CN2CCCC2=O)cc1/C=C\C(=O)O ZINC000217819993 CD For-Sale Unstable PTGER4 15 41 COc1ccc(CN2CCCC2=O)cc1/C=C\C(=O)O ZINC000217819993 CD For-Sale Unstable PTGER3 16 58 COCCNC(=O)CCCCCN1C(=O)c2ccccc2N2C(=O)c3c(ccc(OC)c3OC)[C@H]12 ZINC000217820024 JG In-Stock Unstable HTR7 25 40 O=C(CNS(=O)(=O)c1cccc(F)c1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217820060 GD For-Sale Unstable HTR6 34 42 O=C(CNS(=O)(=O)c1cccc(F)c1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217820060 GD For-Sale Unstable SFRP1 104 35 O=C(CNS(=O)(=O)c1cccc(F)c1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217820060 GD For-Sale Unstable WNT3 72 34 CCc1ccccc1NC(=O)N/C=C/c1ccccc1Cl ZINC000217820068 DJ For-Sale Unstable CXCL8 55 39 CC[C@H]1CCCC[C@H]1NC(=O)C[C@@H](N)c1ccccc1 ZINC000217820076 CG For-Sale Unstable AMY2 45 32 COCCNC(=O)CCCCCN1C(=O)c2ccccc2N2C(=O)c3c(ccc(OC)c3OC)[C@@H]12 ZINC000217820103 JG In-Stock Unstable HTR7 25 40 COC(=O)[C@@H](C)N(C)[C@@H](C)c1ccc(Cl)cc1 ZINC000217820144 CF For-Sale Unstable UTS2 55 42 COc1cc(Cl)c(C(=O)O)c(OC)c1OC ZINC000217820172 BE For-Sale Unstable ALS 77 40 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](CC(C)C)CC(=O)O4)cc1O ZINC000217820208 HI In-Stock Unstable AKR1B1 0 48 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](CC(C)C)CC(=O)O4)cc1O ZINC000217820208 HI In-Stock Unstable CYP1B1 56 35 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](CC(C)C)CC(=O)O4)cc1O ZINC000217820208 HI In-Stock Unstable CYP1A1 42 48 C[C@@H](c1ccccc1Cl)N(C)[C@@H](C(=O)O)c1ccccc1 ZINC000217820294 DI For-Sale Unstable CXCL8 45 44 C[C@@H](c1ccccc1Cl)N(C)[C@@H](C(=O)O)c1ccccc1 ZINC000217820294 DI For-Sale Unstable AOC3 15 40 NC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217820295 DG For-Sale Unstable SMO 16 40 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](CC(C)C)CC(=O)O4)cc1O ZINC000217820297 HI In-Stock Unstable AKR1B1 0 48 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](CC(C)C)CC(=O)O4)cc1O ZINC000217820297 HI In-Stock Unstable CYP1B1 56 35 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](CC(C)C)CC(=O)O4)cc1O ZINC000217820297 HI In-Stock Unstable CYP1A1 42 48 O=C(Cn1nnc(-c2ccc(Cl)cc2)n1)N[C@@H]1CCSc2c(F)cccc21 ZINC000217820323 HG On-Demand Unstable SCARB1 46 42 CC(C)(C)c1ccc(S(=O)(=O)NCC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217820349 IG For-Sale Unstable ADAMTS5 36 42 CC(C)(C)c1ccc(S(=O)(=O)NCC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217820349 IG For-Sale Unstable SFRP1 115 35 CC(C)(C)c1ccc(S(=O)(=O)NCC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217820349 IG For-Sale Unstable WNT3 82 35 COc1cc(CC(=O)O)c(O)c(Cl)c1OC ZINC000217820360 BD For-Sale Unstable TUBB1 40 35 C[C@H](c1ccccc1Cl)N(C)[C@@H](C(=O)O)c1ccccc1 ZINC000217820385 DI For-Sale Unstable CXCL8 45 44 C[C@H](c1ccccc1Cl)N(C)[C@@H](C(=O)O)c1ccccc1 ZINC000217820385 DI For-Sale Unstable AOC3 15 40 O=C(Cn1nnc(-c2ccc(Cl)cc2)n1)N[C@H]1CCSc2c(F)cccc21 ZINC000217820394 HG On-Demand Unstable SCARB1 46 42 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(F)c(Cl)c1 ZINC000217820400 EJ For-Sale Anodyne P95276_MYCTO 0 44 CC(C)(C)c1ccc(S(=O)(=O)NCC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217820433 IG For-Sale Unstable ADAMTS5 36 42 CC(C)(C)c1ccc(S(=O)(=O)NCC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217820433 IG For-Sale Unstable SFRP1 115 35 CC(C)(C)c1ccc(S(=O)(=O)NCC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217820433 IG For-Sale Unstable WNT3 82 35 CCN(CC)c1ccc(NC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217820497 EJ For-Sale Unstable GHSR 20 47 C[C@@H](c1ccccc1Cl)N(C)[C@H](C)C(=O)O ZINC000217820524 BF For-Sale Unstable CXCL8 51 44 O=C1C[C@H](N2Cc3[nH]c4ccccc4c3[C@@H](c3ccccc3)C2)C(=O)N1c1ccccc1 ZINC000217820531 HI In-Stock Unstable ME1 0 44 O=C1C[C@H](N2Cc3[nH]c4ccccc4c3[C@@H](c3ccccc3)C2)C(=O)N1c1ccccc1 ZINC000217820531 HI In-Stock Unstable PDE11A 48 33 COc1cc(OC)c(C(=O)O)c(Cl)c1OC ZINC000217820575 BE For-Sale Unstable ALS 70 37 O=C(N/C=C/c1ccccc1Cl)NCc1ccc(F)cc1 ZINC000217820590 DH For-Sale Unstable AMP1_PLAFQ 16 42 O=C(Nc1cnccc1Cl)c1cccc(Cl)c1F ZINC000217820615 CH For-Sale Anodyne TRPV1 25 42 O=C(Nc1cnccc1Cl)c1cccc(Cl)c1F ZINC000217820615 CH For-Sale Anodyne PIM1 15 40 O=C(Nc1cnccc1Cl)c1cccc(Cl)c1F ZINC000217820615 CH For-Sale Anodyne JAK1 0 44 O=C(Nc1cnccc1Cl)c1cccc(Cl)c1F ZINC000217820615 CH For-Sale Anodyne GRM4 43 45 O=C(Nc1cnccc1Cl)c1cccc(Cl)c1F ZINC000217820615 CH For-Sale Anodyne TYK2 30 44 O=C(Nc1cnccc1Cl)c1cccc(Cl)c1F ZINC000217820615 CH For-Sale Anodyne PIM2 17 40 O=C(Nc1cnccc1Cl)c1cccc(Cl)c1F ZINC000217820615 CH For-Sale Anodyne EPHB3 58 43 O=C(Nc1cnccc1Cl)c1cccc(Cl)c1F ZINC000217820615 CH For-Sale Anodyne NR2E3 43 33 O=C(Nc1cnccc1Cl)c1cccc(Cl)c1F ZINC000217820615 CH For-Sale Anodyne KCNK3 16 40 O=C(Nc1cnccc1Cl)c1cccc(Cl)c1F ZINC000217820615 CH For-Sale Anodyne G2YM83_BOTF4 69 35 COc1ccc(Cn2c(C)csc2=O)cc1/C=C\C(=O)O ZINC000217820617 DE For-Sale Unstable PTGER2 36 40 COc1ccc(Cn2c(C)csc2=O)cc1/C=C\C(=O)O ZINC000217820617 DE For-Sale Unstable PTGER4 0 40 COc1ccc(Cn2c(C)csc2=O)cc1/C=C\C(=O)O ZINC000217820617 DE For-Sale Unstable PTGER3 18 40 COc1cccc(C(=O)NCCC(=O)N2CCC[C@@H]2c2ccccn2)c1 ZINC000217820644 FF In-Stock Unstable HTR1A 22 55 COc1cccc(C(=O)NCCC(=O)N2CCC[C@@H]2c2ccccn2)c1 ZINC000217820644 FF In-Stock Unstable DRD2 23 46 COc1cccc(C(=O)NCCC(=O)N2CCC[C@@H]2c2ccccn2)c1 ZINC000217820644 FF In-Stock Unstable DRD4 60 48 COc1cccc(C(=O)NCCC(=O)N2CCC[C@@H]2c2ccccn2)c1 ZINC000217820644 FF In-Stock Unstable DRD3 32 47 COc1cccc(C(=O)NCCC(=O)N2CCC[C@@H]2c2ccccn2)c1 ZINC000217820644 FF In-Stock Unstable CPT1A 122 49 COc1cccc(C(=O)NCCC(=O)N2CCC[C@@H]2c2ccccn2)c1 ZINC000217820644 FF In-Stock Unstable CPT2 40 36 COc1cccc(C(=O)NCCC(=O)N2CCC[C@@H]2c2ccccn2)c1 ZINC000217820644 FF In-Stock Unstable FAP 0 55 COc1cccc(C(=O)NCCC(=O)N2CCC[C@@H]2c2ccccn2)c1 ZINC000217820644 FF In-Stock Unstable ALPHA-1A 0 41 COc1cccc(C(=O)NCCC(=O)N2CCC[C@@H]2c2ccccn2)c1 ZINC000217820644 FF In-Stock Unstable ACKR3 64 33 COc1cccc(C(=O)NCCC(=O)N2CCC[C@@H]2c2ccccn2)c1 ZINC000217820644 FF In-Stock Unstable BRPF1 0 40 COc1cc(Cl)c(OCC(=O)O)cc1OC ZINC000217820680 BD For-Sale Unstable PPARD 28 41 COc1cc(Cl)c(OCC(=O)O)cc1OC ZINC000217820680 BD For-Sale Unstable PTGDR2 45 42 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2Cl)CC1 ZINC000217820687 FH For-Sale Unstable DRD1 38 40 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2Cl)CC1 ZINC000217820687 FH For-Sale Unstable DRD3 34 41 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2Cl)CC1 ZINC000217820687 FH For-Sale Unstable PDK2 0 41 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2Cl)CC1 ZINC000217820687 FH For-Sale Unstable TACR3 0 45 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2Cl)CC1 ZINC000217820687 FH For-Sale Unstable PDK3 0 41 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2Cl)CC1 ZINC000217820687 FH For-Sale Unstable PDK4 0 41 COc1cccc(C(=O)NCCC(=O)N2CCC[C@H]2c2ccccn2)c1 ZINC000217820728 FF In-Stock Unstable HTR1A 22 55 COc1cccc(C(=O)NCCC(=O)N2CCC[C@H]2c2ccccn2)c1 ZINC000217820728 FF In-Stock Unstable DRD2 23 46 COc1cccc(C(=O)NCCC(=O)N2CCC[C@H]2c2ccccn2)c1 ZINC000217820728 FF In-Stock Unstable DRD4 60 48 COc1cccc(C(=O)NCCC(=O)N2CCC[C@H]2c2ccccn2)c1 ZINC000217820728 FF In-Stock Unstable DRD3 32 47 COc1cccc(C(=O)NCCC(=O)N2CCC[C@H]2c2ccccn2)c1 ZINC000217820728 FF In-Stock Unstable CPT1A 122 49 COc1cccc(C(=O)NCCC(=O)N2CCC[C@H]2c2ccccn2)c1 ZINC000217820728 FF In-Stock Unstable CPT2 40 36 COc1cccc(C(=O)NCCC(=O)N2CCC[C@H]2c2ccccn2)c1 ZINC000217820728 FF In-Stock Unstable FAP 0 55 COc1cccc(C(=O)NCCC(=O)N2CCC[C@H]2c2ccccn2)c1 ZINC000217820728 FF In-Stock Unstable ALPHA-1A 0 41 COc1cccc(C(=O)NCCC(=O)N2CCC[C@H]2c2ccccn2)c1 ZINC000217820728 FF In-Stock Unstable ACKR3 64 33 COc1cccc(C(=O)NCCC(=O)N2CCC[C@H]2c2ccccn2)c1 ZINC000217820728 FF In-Stock Unstable BRPF1 0 40 O=C1C[C@H](N2Cc3[nH]c4ccccc4c3[C@@H](c3ccccc3)C2)C(=O)N1c1ccc2c(c1)OCCO2 ZINC000217820767 JI In-Stock Unstable PDE5A 37 41 O=C1C[C@H](N2Cc3[nH]c4ccccc4c3[C@@H](c3ccccc3)C2)C(=O)N1c1ccc2c(c1)OCCO2 ZINC000217820767 JI In-Stock Unstable PDE11A 85 38 O=C(CCN1CC[C@@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820803 CH On-Demand Unstable HTR1A 22 59 O=C(CCN1CC[C@@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820803 CH On-Demand Unstable DRD2 47 76 O=C(CCN1CC[C@@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820803 CH On-Demand Unstable DRD1 19 45 O=C(CCN1CC[C@@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820803 CH On-Demand Unstable DRD4 46 59 O=C(CCN1CC[C@@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820803 CH On-Demand Unstable HTR2A 48 54 O=C(CCN1CC[C@@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820803 CH On-Demand Unstable HTR2C 27 57 O=C(CCN1CC[C@@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820803 CH On-Demand Unstable SLC6A1 127 39 O=C(CCN1CC[C@@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820803 CH On-Demand Unstable SLC6A4 22 52 O=C(CCN1CC[C@@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820803 CH On-Demand Unstable ADRA1A 18 46 O=C(CCN1CC[C@@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820803 CH On-Demand Unstable HRH1 29 59 O=C(CCN1CC[C@@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820803 CH On-Demand Unstable ADRA1B 20 46 O=C(CCN1CC[C@@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820803 CH On-Demand Unstable DRD3 18 57 O=C(CCN1CC[C@@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820803 CH On-Demand Unstable SLC6A3 29 52 O=C(CCN1CC[C@@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820803 CH On-Demand Unstable DRD5 15 50 O=C(CCN1CC[C@@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820803 CH On-Demand Unstable HTR7 22 45 O=C(CCN1CC[C@@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820803 CH On-Demand Unstable SIGMAR1 46 71 O=C(CCN1CC[C@@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820803 CH On-Demand Unstable HSD11B1 19 40 O=C(CCN1CC[C@@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820803 CH On-Demand Unstable PRCP 33 51 O=C(CCN1CC[C@@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820803 CH On-Demand Unstable CCR3 38 43 O=C(CCN1CC[C@@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820803 CH On-Demand Unstable CCR5 65 35 O=C(CCN1CC[C@@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820803 CH On-Demand Unstable PLD1 44 37 O=C(CCN1CC[C@@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820803 CH On-Demand Unstable SLC18A3 79 59 O=C(CCN1CC[C@@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820803 CH On-Demand Unstable CCR2 16 45 O=C(CCN1CC[C@@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820803 CH On-Demand Unstable PLD2 43 37 O=C(CCN1CC[C@@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820803 CH On-Demand Unstable MCHR1 23 51 O=C(CCN1CC[C@@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820803 CH On-Demand Unstable CYP2J2 57 41 COC(=O)[C@@H]1C[C@@H]1C(=O)c1ccc(OC)c2ccccc12 ZINC000217820814 CF In-Stock Unstable AGTR2 45 33 O=C1C[C@H](N2Cc3[nH]c4ccccc4c3[C@@H](c3ccccc3)C2)C(=O)N1c1ccc2c(c1)OCO2 ZINC000217820860 JI In-Stock Unstable PDE5A 55 46 O=C1C[C@H](N2Cc3[nH]c4ccccc4c3[C@@H](c3ccccc3)C2)C(=O)N1c1ccc2c(c1)OCO2 ZINC000217820860 JI In-Stock Unstable PDE11A 94 43 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1cc(F)ccc1N ZINC000217820867 CH For-Sale Unstable TRPM8 19 56 O=C(CCN1CC[C@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820873 CH On-Demand Unstable HTR1A 22 59 O=C(CCN1CC[C@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820873 CH On-Demand Unstable DRD2 47 76 O=C(CCN1CC[C@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820873 CH On-Demand Unstable DRD1 19 45 O=C(CCN1CC[C@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820873 CH On-Demand Unstable DRD4 46 59 O=C(CCN1CC[C@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820873 CH On-Demand Unstable HTR2A 48 54 O=C(CCN1CC[C@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820873 CH On-Demand Unstable HTR2C 27 57 O=C(CCN1CC[C@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820873 CH On-Demand Unstable SLC6A1 127 39 O=C(CCN1CC[C@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820873 CH On-Demand Unstable SLC6A4 22 52 O=C(CCN1CC[C@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820873 CH On-Demand Unstable ADRA1A 18 46 O=C(CCN1CC[C@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820873 CH On-Demand Unstable HRH1 29 59 O=C(CCN1CC[C@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820873 CH On-Demand Unstable ADRA1B 20 46 O=C(CCN1CC[C@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820873 CH On-Demand Unstable DRD3 18 57 O=C(CCN1CC[C@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820873 CH On-Demand Unstable SLC6A3 29 52 O=C(CCN1CC[C@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820873 CH On-Demand Unstable DRD5 15 50 O=C(CCN1CC[C@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820873 CH On-Demand Unstable HTR7 22 45 O=C(CCN1CC[C@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820873 CH On-Demand Unstable SIGMAR1 46 71 O=C(CCN1CC[C@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820873 CH On-Demand Unstable HSD11B1 19 40 O=C(CCN1CC[C@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820873 CH On-Demand Unstable PRCP 33 51 O=C(CCN1CC[C@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820873 CH On-Demand Unstable CCR3 38 43 O=C(CCN1CC[C@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820873 CH On-Demand Unstable CCR5 65 35 O=C(CCN1CC[C@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820873 CH On-Demand Unstable PLD1 44 37 O=C(CCN1CC[C@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820873 CH On-Demand Unstable SLC18A3 79 59 O=C(CCN1CC[C@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820873 CH On-Demand Unstable CCR2 16 45 O=C(CCN1CC[C@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820873 CH On-Demand Unstable PLD2 43 37 O=C(CCN1CC[C@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820873 CH On-Demand Unstable MCHR1 23 51 O=C(CCN1CC[C@H](c2ccccc2)C1)c1ccc(F)cc1 ZINC000217820873 CH On-Demand Unstable CYP2J2 57 41 COC(=O)[C@H]1C[C@@H]1C(=O)c1ccc(OC)c2ccccc12 ZINC000217820902 CF In-Stock Unstable AGTR2 45 33 COC(=O)[C@@H](C)N(C)[C@@H](C)c1ccccc1Cl ZINC000217820920 CF For-Sale Unstable CXCL8 42 35 Cc1nn(Cc2ccccc2/C=C\C(=O)O)c(C)c1C ZINC000217820928 CF For-Sale Unstable PTGER2 45 46 Cc1nn(Cc2ccccc2/C=C\C(=O)O)c(C)c1C ZINC000217820928 CF For-Sale Unstable PTGER4 22 46 Cc1nn(Cc2ccccc2/C=C\C(=O)O)c(C)c1C ZINC000217820928 CF For-Sale Unstable PTGER3 18 46 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1cc(F)ccc1N ZINC000217820948 CH For-Sale Unstable TRPM8 19 56 COC(=O)[C@@H]1C[C@H]1C(=O)c1ccc(OC)c2ccccc12 ZINC000217820960 CF In-Stock Unstable AGTR2 45 33 COC(=O)C[C@H](c1ccc2c(c1)OCO2)c1c(O)c2ccccc2oc1=O ZINC000217820995 FF In-Stock Unstable NQO1 53 37 O=C(/C=C\c1cccc2ccccc12)CCl ZINC000217821001 BH For-Sale Unstable CHAT 79 44 O=C(Nc1ccc(OC(F)F)c(Cl)c1)c1c[nH]nc1-c1ccc(Cl)cc1 ZINC000217821011 GK On-Demand Anodyne GRM4 44 44 O=C(Nc1ccc(OC(F)F)c(Cl)c1)c1c[nH]nc1-c1ccc(Cl)cc1 ZINC000217821011 GK On-Demand Anodyne NR2E3 62 35 O=C(Nc1ccc(OC(F)F)c(Cl)c1)c1c[nH]nc1-c1ccc(Cl)cc1 ZINC000217821011 GK On-Demand Anodyne Q25615_ONCVO 30 41 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)c1cc(F)ccc1N ZINC000217821013 CH For-Sale Unstable TRPM8 19 56 O=C(O)/C=C\c1ccc(COc2cccc(Cl)c2)cc1 ZINC000217821019 CI For-Sale Unstable MAOB 56 45 O=C(O)/C=C\c1ccc(COc2cccc(Cl)c2)cc1 ZINC000217821019 CI For-Sale Unstable PTGER2 17 53 O=C(O)/C=C\c1ccc(COc2cccc(Cl)c2)cc1 ZINC000217821019 CI For-Sale Unstable PTGER1 43 37 O=C(O)/C=C\c1ccc(COc2cccc(Cl)c2)cc1 ZINC000217821019 CI For-Sale Unstable PTGER4 27 53 O=C(O)/C=C\c1ccc(COc2cccc(Cl)c2)cc1 ZINC000217821019 CI For-Sale Unstable PTPN2 0 42 O=C(O)/C=C\c1ccc(COc2cccc(Cl)c2)cc1 ZINC000217821019 CI For-Sale Unstable PTGER3 27 53 O=C(O)/C=C\c1ccc(COc2cccc(Cl)c2)cc1 ZINC000217821019 CI For-Sale Unstable CDC25B 22 42 O=C(O)/C=C\c1ccc(COc2cccc(Cl)c2)cc1 ZINC000217821019 CI For-Sale Unstable PTGDR 0 48 O=C(O)/C=C\c1ccc(COc2cccc(Cl)c2)cc1 ZINC000217821019 CI For-Sale Unstable 17HSDCL 0 40 O=C(O)/C=C\c1ccc(COc2cccc(Cl)c2)cc1 ZINC000217821019 CI For-Sale Unstable FFAR1 40 43 O=C(O)/C=C\c1ccc(COc2cccc(Cl)c2)cc1 ZINC000217821019 CI For-Sale Unstable AKR1C3 36 50 O=C(O)/C=C\c1ccc(COc2cccc(Cl)c2)cc1 ZINC000217821019 CI For-Sale Unstable PDS 45 40 COC(=O)[C@H]1C[C@H]1C(=O)c1ccc(OC)c2ccccc12 ZINC000217821049 CF In-Stock Unstable AGTR2 45 33 O=C(N/C=C/c1ccccc1Cl)NC1CCCCCC1 ZINC000217821065 CI For-Sale Unstable EPHX2 36 48 COc1cc(C(=O)Nc2cnccc2Cl)ccc1F ZINC000217821078 CG For-Sale Unstable MAOB 18 40 COc1cc(C(=O)Nc2cnccc2Cl)ccc1F ZINC000217821078 CG For-Sale Unstable F10 45 44 COc1cc(C(=O)Nc2cnccc2Cl)ccc1F ZINC000217821078 CG For-Sale Unstable PDE4B 15 44 COc1cc(C(=O)Nc2cnccc2Cl)ccc1F ZINC000217821078 CG For-Sale Unstable PDE4D 17 53 COc1cc(C(=O)Nc2cnccc2Cl)ccc1F ZINC000217821078 CG For-Sale Unstable COLA 82 38 COc1cc(C(=O)Nc2cnccc2Cl)ccc1F ZINC000217821078 CG For-Sale Unstable CPT1A 82 36 COc1cc(C(=O)Nc2cnccc2Cl)ccc1F ZINC000217821078 CG For-Sale Unstable CPT2 45 35 COc1cc(C(=O)Nc2cnccc2Cl)ccc1F ZINC000217821078 CG For-Sale Unstable PYGL 20 43 COc1cc(C(=O)Nc2cnccc2Cl)ccc1F ZINC000217821078 CG For-Sale Unstable KDR 42 37 COc1cc(C(=O)Nc2cnccc2Cl)ccc1F ZINC000217821078 CG For-Sale Unstable GRM4 38 51 COc1cc(C(=O)Nc2cnccc2Cl)ccc1F ZINC000217821078 CG For-Sale Unstable ROCK2 40 41 COc1cc(C(=O)Nc2cnccc2Cl)ccc1F ZINC000217821078 CG For-Sale Unstable ABCB1 0 53 COc1cc(C(=O)Nc2cnccc2Cl)ccc1F ZINC000217821078 CG For-Sale Unstable CPT1B 68 36 COc1cc(C(=O)Nc2cnccc2Cl)ccc1F ZINC000217821078 CG For-Sale Unstable CSF1R 42 39 COc1cc(C(=O)Nc2cnccc2Cl)ccc1F ZINC000217821078 CG For-Sale Unstable FABH 0 44 COc1cc(C(=O)Nc2cnccc2Cl)ccc1F ZINC000217821078 CG For-Sale Unstable Q8MMZ8_EIMTE 0 46 COc1cc(C(=O)Nc2cnccc2Cl)ccc1F ZINC000217821078 CG For-Sale Unstable TAAR1 29 50 COc1cc(C(=O)Nc2cnccc2Cl)ccc1F ZINC000217821078 CG For-Sale Unstable SCD1 33 43 COc1cc(C(=O)Nc2cnccc2Cl)ccc1F ZINC000217821078 CG For-Sale Unstable SCD 24 43 COc1cc(C(=O)Nc2cnccc2Cl)ccc1F ZINC000217821078 CG For-Sale Unstable SMO 18 41 COc1cc(C(=O)Nc2cnccc2Cl)ccc1F ZINC000217821078 CG For-Sale Unstable GLMU 0 41 COc1cc(C(=O)Nc2cnccc2Cl)ccc1F ZINC000217821078 CG For-Sale Unstable KCNK3 48 36 COC(=O)C[C@@H](c1ccc2c(c1)OCO2)c1c(O)c2ccccc2oc1=O ZINC000217821081 FF In-Stock Unstable NQO1 53 37 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)c1cc(F)ccc1N ZINC000217821086 CH For-Sale Unstable TRPM8 19 56 O=C(O)/C=C\c1ccc(COc2cccc(Cl)c2)c(F)c1 ZINC000217821091 DI For-Sale Unstable MAOB 25 41 O=C(O)/C=C\c1ccc(COc2cccc(Cl)c2)c(F)c1 ZINC000217821091 DI For-Sale Unstable PTGER2 35 43 O=C(O)/C=C\c1ccc(COc2cccc(Cl)c2)c(F)c1 ZINC000217821091 DI For-Sale Unstable PTGER1 37 43 O=C(O)/C=C\c1ccc(COc2cccc(Cl)c2)c(F)c1 ZINC000217821091 DI For-Sale Unstable PTGER4 19 41 O=C(O)/C=C\c1ccc(COc2cccc(Cl)c2)c(F)c1 ZINC000217821091 DI For-Sale Unstable PTGER3 17 41 O=C(O)/C=C\c1ccc(COc2cccc(Cl)c2)c(F)c1 ZINC000217821091 DI For-Sale Unstable CDC25B 25 49 O=C(O)/C=C\c1ccc(COc2cccc(Cl)c2)c(F)c1 ZINC000217821091 DI For-Sale Unstable AKR1C3 31 45 O=C(Nc1ccc(OC(F)F)c(Cl)c1)c1c[nH]nc1-c1ccc(F)cc1 ZINC000217821130 GJ On-Demand Anodyne GRM4 48 44 O=C(Nc1ccc(OC(F)F)c(Cl)c1)c1c[nH]nc1-c1ccc(F)cc1 ZINC000217821130 GJ On-Demand Anodyne NR2E3 62 35 COC(=O)[C@@H]1C[C@@H]1C(=O)c1ccc(OC)cc1 ZINC000217821136 BD In-Stock Unstable SLC6A1 28 41 C[C@@H](CCO)NCc1cccc(OC(F)(F)F)c1 ZINC000217821165 CE On-Demand Unstable CETP 0 43 O=C(O)/C=C\c1cccc(COc2cccc(Cl)c2)c1 ZINC000217821167 CI For-Sale Unstable MAOB 73 49 O=C(O)/C=C\c1cccc(COc2cccc(Cl)c2)c1 ZINC000217821167 CI For-Sale Unstable PTGER2 17 53 O=C(O)/C=C\c1cccc(COc2cccc(Cl)c2)c1 ZINC000217821167 CI For-Sale Unstable CYSLTR1 22 40 O=C(O)/C=C\c1cccc(COc2cccc(Cl)c2)c1 ZINC000217821167 CI For-Sale Unstable PTGER1 42 37 O=C(O)/C=C\c1cccc(COc2cccc(Cl)c2)c1 ZINC000217821167 CI For-Sale Unstable PTGER4 27 53 O=C(O)/C=C\c1cccc(COc2cccc(Cl)c2)c1 ZINC000217821167 CI For-Sale Unstable PTGER3 25 53 O=C(O)/C=C\c1cccc(COc2cccc(Cl)c2)c1 ZINC000217821167 CI For-Sale Unstable LTB4R 15 43 O=C(O)/C=C\c1cccc(COc2cccc(Cl)c2)c1 ZINC000217821167 CI For-Sale Unstable CDC25B 0 44 O=C(O)/C=C\c1cccc(COc2cccc(Cl)c2)c1 ZINC000217821167 CI For-Sale Unstable NR1H4 45 41 O=C(O)/C=C\c1cccc(COc2cccc(Cl)c2)c1 ZINC000217821167 CI For-Sale Unstable 17HSDCL 0 40 O=C(O)/C=C\c1cccc(COc2cccc(Cl)c2)c1 ZINC000217821167 CI For-Sale Unstable FFAR1 50 43 O=C(O)/C=C\c1cccc(COc2cccc(Cl)c2)c1 ZINC000217821167 CI For-Sale Unstable AKR1C3 40 48 O=C(O)/C=C\c1cccc(COc2cccc(Cl)c2)c1 ZINC000217821167 CI For-Sale Unstable ADCYAP1R1 33 40 O=C(O)/C=C\c1cccc(COc2cccc(Cl)c2)c1 ZINC000217821167 CI For-Sale Unstable TUBA4A 0 42 O=C(O)/C=C\c1cccc(COc2cccc(Cl)c2)c1 ZINC000217821167 CI For-Sale Unstable PDS 64 42 Cc1ccc(C)c(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217821178 DJ For-Sale Unstable CXCL8 41 32 COC(=O)C[C@@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(OC)c(O)c1 ZINC000217821188 GF In-Stock Unstable TNF 21 42 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)[C@@H]1CCCN1 ZINC000217821192 CE For-Sale Unstable TRPM8 19 49 Cc1cc(Cl)cc(C(=O)Nc2cnccc2Cl)c1 ZINC000217821205 CH For-Sale Unstable SCN10A 42 44 Cc1cc(Cl)cc(C(=O)Nc2cnccc2Cl)c1 ZINC000217821205 CH For-Sale Unstable CSF1R 23 52 Cc1cc(Cl)cc(C(=O)Nc2cnccc2Cl)c1 ZINC000217821205 CH For-Sale Unstable KCNK3 53 43 Cc1cc(Cl)cc(C(=O)Nc2cnccc2Cl)c1 ZINC000217821205 CH For-Sale Unstable KCNK9 33 43 COC(=O)[C@H]1C[C@@H]1C(=O)c1ccc(OC)cc1 ZINC000217821219 BD In-Stock Unstable SLC6A1 28 41 C[C@H](CCO)NCc1cccc(OC(F)(F)F)c1 ZINC000217821243 CE On-Demand Unstable CETP 0 43 COc1ccc(/C=C\C(=O)O)cc1COC1CCCCC1 ZINC000217821247 CH For-Sale Unstable PTGER2 0 42 COc1ccc(/C=C\C(=O)O)cc1COC1CCCCC1 ZINC000217821247 CH For-Sale Unstable AKR1C3 23 40 COc1cc(CNC(=O)COc2ccccc2)ccc1OC(C)C ZINC000217821255 EG In-Stock Unstable TSHR 47 33 COc1cc(CNC(=O)COc2ccccc2)ccc1OC(C)C ZINC000217821255 EG In-Stock Unstable PPARA 18 41 COc1cc(CNC(=O)COc2ccccc2)ccc1OC(C)C ZINC000217821255 EG In-Stock Unstable ADORA2B 0 42 COc1cc(CNC(=O)COc2ccccc2)ccc1OC(C)C ZINC000217821255 EG In-Stock Unstable HCRTR1 22 41 COc1cc(CNC(=O)COc2ccccc2)ccc1OC(C)C ZINC000217821255 EG In-Stock Unstable TRPV1 31 42 COc1cc(CNC(=O)COc2ccccc2)ccc1OC(C)C ZINC000217821255 EG In-Stock Unstable PTGER3 35 40 COc1cc(CNC(=O)COc2ccccc2)ccc1OC(C)C ZINC000217821255 EG In-Stock Unstable ROCK2 15 41 COc1cc(CNC(=O)COc2ccccc2)ccc1OC(C)C ZINC000217821255 EG In-Stock Unstable PDE6A 41 32 COc1cc(CNC(=O)COc2ccccc2)ccc1OC(C)C ZINC000217821255 EG In-Stock Unstable ABCB1 22 41 COc1cc(CNC(=O)COc2ccccc2)ccc1OC(C)C ZINC000217821255 EG In-Stock Unstable TTR 0 40 COc1cc(CNC(=O)COc2ccccc2)ccc1OC(C)C ZINC000217821255 EG In-Stock Unstable MT-ND1 24 42 COc1cc(CNC(=O)COc2ccccc2)ccc1OC(C)C ZINC000217821255 EG In-Stock Unstable HCRTR2 28 40 COc1cc(CNC(=O)COc2ccccc2)ccc1OC(C)C ZINC000217821255 EG In-Stock Unstable ABCG2 19 41 COc1cc(CNC(=O)COc2ccccc2)ccc1OC(C)C ZINC000217821255 EG In-Stock Unstable DRTS_TRYCR 47 32 COc1cc(CNC(=O)COc2ccccc2)ccc1OC(C)C ZINC000217821255 EG In-Stock Unstable BLAIMP-1 0 42 COc1cc(CNC(=O)COc2ccccc2)ccc1OC(C)C ZINC000217821255 EG In-Stock Unstable PDS 55 38 COC(=O)C[C@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(OC)c(O)c1 ZINC000217821269 GF In-Stock Unstable TNF 21 42 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)[C@@H]1CCCN1 ZINC000217821271 CE For-Sale Unstable TRPM8 19 49 O=C(CCNS(=O)(=O)c1cccc(Cl)c1)NC[C@H]1CCCN1c1ccccc1 ZINC000217821290 HF For-Sale Unstable HTR7 18 42 O=C(CCNS(=O)(=O)c1cccc(Cl)c1)NC[C@H]1CCCN1c1ccccc1 ZINC000217821290 HF For-Sale Unstable ADAMTS5 20 41 O=C(CCNS(=O)(=O)c1cccc(Cl)c1)NC[C@H]1CCCN1c1ccccc1 ZINC000217821290 HF For-Sale Unstable SFRP1 40 35 COC(=O)[C@@H]1C[C@H]1C(=O)c1ccc(OC)cc1 ZINC000217821293 BD In-Stock Unstable SLC6A1 28 41 C[C@@H](c1cccc(Cl)c1)N(C)[C@H](C)C(=O)O ZINC000217821298 BF For-Sale Unstable ADRB1 21 41 C[C@@H](c1cccc(Cl)c1)N(C)[C@H](C)C(=O)O ZINC000217821298 BF For-Sale Unstable ADRB3 33 41 O=C(N/C=C/c1ccccc1Cl)Nc1cc(Cl)cc(Cl)c1 ZINC000217821303 EK For-Sale Anodyne PPIA 16 43 CSCCOc1ccc(OCc2ccccc2)cc1 ZINC000217821310 CI On-Demand Unstable MAOB 34 41 CSCCOc1ccc(OCc2ccccc2)cc1 ZINC000217821310 CI On-Demand Unstable LTA4H 50 43 CSCCOc1ccc(OCc2ccccc2)cc1 ZINC000217821310 CI On-Demand Unstable SCN2A 15 43 CSCCOc1ccc(OCc2ccccc2)cc1 ZINC000217821310 CI On-Demand Unstable ESRRG 39 40 CSCCOc1ccc(OCc2ccccc2)cc1 ZINC000217821310 CI On-Demand Unstable TAAR1 22 51 CSCCOc1ccc(OCc2ccccc2)cc1 ZINC000217821310 CI On-Demand Unstable FFAR1 32 46 CSCCOc1ccc(OCc2ccccc2)cc1 ZINC000217821310 CI On-Demand Unstable PIR 0 41 Cc1ccccc1OC1CCN(C(=O)c2ccc(C#CC(C)(C)O)cc2)CC1 ZINC000217821320 GH In-Stock Unstable L3MBTL3 50 34 CC(=O)c1cccc(S(=O)(=O)N2CCC[C@H](Cc3nc(C4CC4)no3)C2)c1 ZINC000217821329 GF In-Stock Unstable AKR1C3 55 37 O=C(O)/C=C\c1ccc(OCCOC2CCCC2)cc1 ZINC000217821337 CG For-Sale Unstable ADRB1 15 44 O=C(O)/C=C\c1ccc(OCCOC2CCCC2)cc1 ZINC000217821337 CG For-Sale Unstable HPGD 22 53 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@@H](C)O)cc1 ZINC000217821347 HE On-Demand Unstable CA2 25 41 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@@H](C)O)cc1 ZINC000217821347 HE On-Demand Unstable CA1 22 41 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@@H](C)O)cc1 ZINC000217821347 HE On-Demand Unstable MMP13 37 47 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@@H](C)O)cc1 ZINC000217821347 HE On-Demand Unstable MMP2 20 47 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@@H](C)O)cc1 ZINC000217821347 HE On-Demand Unstable MMP12 63 45 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@@H](C)O)cc1 ZINC000217821347 HE On-Demand Unstable CA12 21 41 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@@H](C)O)cc1 ZINC000217821347 HE On-Demand Unstable MMP7 19 45 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@@H](C)O)cc1 ZINC000217821347 HE On-Demand Unstable ADAMTS4 51 36 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@@H](C)O)cc1 ZINC000217821347 HE On-Demand Unstable CA9 21 41 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@@H](C)O)cc1 ZINC000217821347 HE On-Demand Unstable LEF 64 45 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@@H](C)O)cc1 ZINC000217821347 HE On-Demand Unstable IDO1 29 51 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)[C@@H]1CCCN1 ZINC000217821358 CE For-Sale Unstable TRPM8 19 49 COC(=O)[C@H]1C[C@H]1C(=O)c1ccc(OC)cc1 ZINC000217821361 BD In-Stock Unstable SLC6A1 28 41 O=C(CCNS(=O)(=O)c1cccc(Cl)c1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217821372 HF For-Sale Unstable HTR7 18 42 O=C(CCNS(=O)(=O)c1cccc(Cl)c1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217821372 HF For-Sale Unstable ADAMTS5 20 41 O=C(CCNS(=O)(=O)c1cccc(Cl)c1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217821372 HF For-Sale Unstable SFRP1 40 35 O=C(COc1ccccc1)NCCCc1ccccc1Cl ZINC000217821378 DG In-Stock Unstable CYSP_TRYCR 0 40 O=C(COc1ccccc1)NCCCc1ccccc1Cl ZINC000217821378 DG In-Stock Unstable MTNR1A 40 41 O=C(COc1ccccc1)NCCCc1ccccc1Cl ZINC000217821378 DG In-Stock Unstable MTNR1B 53 38 O=C(COc1ccccc1)NCCCc1ccccc1Cl ZINC000217821378 DG In-Stock Unstable CRTM 49 43 CC(=O)c1cccc(S(=O)(=O)N2CCC[C@@H](Cc3nc(C4CC4)no3)C2)c1 ZINC000217821416 GF In-Stock Unstable AKR1C3 55 37 CCOc1ccccc1NC(=O)N/C=C/c1ccccc1Cl ZINC000217821419 DJ For-Sale Unstable CXCL8 51 33 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@@H](C)O)cc1 ZINC000217821424 HE On-Demand Unstable CA2 25 41 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@@H](C)O)cc1 ZINC000217821424 HE On-Demand Unstable CA1 22 41 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@@H](C)O)cc1 ZINC000217821424 HE On-Demand Unstable MMP13 37 47 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@@H](C)O)cc1 ZINC000217821424 HE On-Demand Unstable MMP2 20 47 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@@H](C)O)cc1 ZINC000217821424 HE On-Demand Unstable MMP12 63 45 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@@H](C)O)cc1 ZINC000217821424 HE On-Demand Unstable CA12 21 41 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@@H](C)O)cc1 ZINC000217821424 HE On-Demand Unstable MMP7 19 45 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@@H](C)O)cc1 ZINC000217821424 HE On-Demand Unstable ADAMTS4 51 36 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@@H](C)O)cc1 ZINC000217821424 HE On-Demand Unstable CA9 21 41 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@@H](C)O)cc1 ZINC000217821424 HE On-Demand Unstable LEF 64 45 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@@H](C)O)cc1 ZINC000217821424 HE On-Demand Unstable IDO1 29 51 O=C(O)/C=C\c1ccc(OCCN2CCC(O)CC2)cc1 ZINC000217821456 CD For-Sale Unstable ESR1 64 41 O=C(O)/C=C\c1ccc(OCCN2CCC(O)CC2)cc1 ZINC000217821456 CD For-Sale Unstable HRH2 28 40 O=C(O)/C=C\c1ccc(OCCN2CCC(O)CC2)cc1 ZINC000217821456 CD For-Sale Unstable HRH1 19 40 O=C(O)/C=C\c1ccc(OCCN2CCC(O)CC2)cc1 ZINC000217821456 CD For-Sale Unstable ESR2 43 41 O=C(O)/C=C\c1ccc(OCCN2CCC(O)CC2)cc1 ZINC000217821456 CD For-Sale Unstable LTA4H 66 50 O=C(O)/C=C\c1ccc(OCCN2CCC(O)CC2)cc1 ZINC000217821456 CD For-Sale Unstable HRH3 50 51 O=C(O)/C=C\c1ccc(OCCN2CCC(O)CC2)cc1 ZINC000217821456 CD For-Sale Unstable SIGMAR1 19 44 O=C(O)/C=C\c1ccc(OCCN2CCC(O)CC2)cc1 ZINC000217821456 CD For-Sale Unstable PSMB2 53 42 O=C(O)/C=C\c1ccc(OCCN2CCC(O)CC2)cc1 ZINC000217821456 CD For-Sale Unstable PSMB5 18 42 O=C(O)/C=C\c1ccc(OCCN2CCC(O)CC2)cc1 ZINC000217821456 CD For-Sale Unstable PSMB1 47 42 O=C(O)/C=C\c1ccc(OCCN2CCC(O)CC2)cc1 ZINC000217821456 CD For-Sale Unstable MEN1 47 34 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)C1CCNCC1 ZINC000217821469 CF On-Demand Unstable TRPM8 20 51 CCOc1ccc(C(=O)[C@@H]2C[C@@H]2C(=O)OC)cc1 ZINC000217821472 BE In-Stock Unstable SLC6A1 0 45 Cc1cccc(S(=O)(=O)Nc2ccc(C(=O)NC[C@@H]3CCCN3c3ccccc3)cc2)c1 ZINC000217821477 II For-Sale Unstable F2 18 41 Cc1cccc(S(=O)(=O)Nc2ccc(C(=O)NC[C@@H]3CCCN3c3ccccc3)cc2)c1 ZINC000217821477 II For-Sale Unstable ST14 46 32 Cc1cccc(S(=O)(=O)Nc2ccc(C(=O)NC[C@@H]3CCCN3c3ccccc3)cc2)c1 ZINC000217821477 II For-Sale Unstable SFRP1 40 32 Cc1cccc(S(=O)(=O)Nc2ccc(C(=O)NC[C@@H]3CCCN3c3ccccc3)cc2)c1 ZINC000217821477 II For-Sale Unstable LIMK2 38 41 O=C(COc1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217821488 DG In-Stock Unstable ADRB1 24 41 O=C(COc1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217821488 DG In-Stock Unstable SCNN1A 66 41 O=C(COc1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217821488 DG In-Stock Unstable ADRB3 29 41 O=C(COc1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217821488 DG In-Stock Unstable SDH1 0 43 O=C(COc1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217821488 DG In-Stock Unstable SCN2A 22 40 O=C(COc1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217821488 DG In-Stock Unstable HDAC8 17 43 O=C(COc1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217821488 DG In-Stock Unstable MTNR1B 30 40 O=C(COc1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217821488 DG In-Stock Unstable PLA2G4B 37 41 O=C(COc1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217821488 DG In-Stock Unstable FAAH 43 44 O=C(COc1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217821488 DG In-Stock Unstable SCN5A 0 46 O=C(COc1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217821488 DG In-Stock Unstable SLC6A5 20 42 O=C(COc1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217821488 DG In-Stock Unstable C5AR1 17 40 O=C(COc1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217821488 DG In-Stock Unstable ADAMTS4 15 43 O=C(COc1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217821488 DG In-Stock Unstable ADAMTS5 19 67 O=C(COc1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217821488 DG In-Stock Unstable AMP1_PLAFQ 35 40 O=C(COc1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217821488 DG In-Stock Unstable FFAR1 38 43 O=C(COc1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217821488 DG In-Stock Unstable NCE103 32 42 O=C(COc1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217821488 DG In-Stock Unstable FFAR4 43 43 O=C(COc1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217821488 DG In-Stock Unstable CRTM 78 53 O=C(COc1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217821488 DG In-Stock Unstable P96878_MYCTU 17 42 O=C(COc1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217821488 DG In-Stock Unstable CAN2 0 42 O=C(COc1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217821488 DG In-Stock Unstable PDS 54 40 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@H](C)O)cc1 ZINC000217821502 HE On-Demand Unstable CA2 25 41 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@H](C)O)cc1 ZINC000217821502 HE On-Demand Unstable CA1 22 41 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@H](C)O)cc1 ZINC000217821502 HE On-Demand Unstable MMP13 37 47 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@H](C)O)cc1 ZINC000217821502 HE On-Demand Unstable MMP2 20 47 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@H](C)O)cc1 ZINC000217821502 HE On-Demand Unstable MMP12 63 45 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@H](C)O)cc1 ZINC000217821502 HE On-Demand Unstable CA12 21 41 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@H](C)O)cc1 ZINC000217821502 HE On-Demand Unstable MMP7 19 45 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@H](C)O)cc1 ZINC000217821502 HE On-Demand Unstable ADAMTS4 51 36 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@H](C)O)cc1 ZINC000217821502 HE On-Demand Unstable CA9 21 41 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@H](C)O)cc1 ZINC000217821502 HE On-Demand Unstable LEF 64 45 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@H](C)O)cc1 ZINC000217821502 HE On-Demand Unstable IDO1 29 51 Cc1cc(C)cc(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217821540 DJ For-Sale Unstable LPL 42 33 CCOc1ccc(C(=O)[C@H]2C[C@@H]2C(=O)OC)cc1 ZINC000217821546 BE In-Stock Unstable SLC6A1 0 45 Cc1cccc(S(=O)(=O)Nc2ccc(C(=O)NC[C@H]3CCCN3c3ccccc3)cc2)c1 ZINC000217821547 II For-Sale Unstable F2 18 41 Cc1cccc(S(=O)(=O)Nc2ccc(C(=O)NC[C@H]3CCCN3c3ccccc3)cc2)c1 ZINC000217821547 II For-Sale Unstable ST14 46 32 Cc1cccc(S(=O)(=O)Nc2ccc(C(=O)NC[C@H]3CCCN3c3ccccc3)cc2)c1 ZINC000217821547 II For-Sale Unstable SFRP1 40 32 Cc1cccc(S(=O)(=O)Nc2ccc(C(=O)NC[C@H]3CCCN3c3ccccc3)cc2)c1 ZINC000217821547 II For-Sale Unstable LIMK2 38 41 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)C1CCNCC1 ZINC000217821555 CF On-Demand Unstable TRPM8 20 51 CCN(Cc1cc(/C=C\C(=O)O)ccc1OC)CC(C)C ZINC000217821579 CG For-Sale Unstable TUBB1 42 37 CCN(Cc1cc(/C=C\C(=O)O)ccc1OC)CC(C)C ZINC000217821579 CG For-Sale Unstable AKR1C3 31 42 O=C(COc1ccccc1)NCCCc1ccc(F)cc1 ZINC000217821593 CF In-Stock Unstable HRH2 29 40 O=C(COc1ccccc1)NCCCc1ccc(F)cc1 ZINC000217821593 CF In-Stock Unstable ADRB3 29 41 O=C(COc1ccccc1)NCCCc1ccc(F)cc1 ZINC000217821593 CF In-Stock Unstable SDH1 0 43 O=C(COc1ccccc1)NCCCc1ccc(F)cc1 ZINC000217821593 CF In-Stock Unstable CYSP_TRYCR 0 40 O=C(COc1ccccc1)NCCCc1ccc(F)cc1 ZINC000217821593 CF In-Stock Unstable SCN2A 16 40 O=C(COc1ccccc1)NCCCc1ccc(F)cc1 ZINC000217821593 CF In-Stock Unstable HDAC8 18 43 O=C(COc1ccccc1)NCCCc1ccc(F)cc1 ZINC000217821593 CF In-Stock Unstable MTNR1B 32 40 O=C(COc1ccccc1)NCCCc1ccc(F)cc1 ZINC000217821593 CF In-Stock Unstable PLA2G4B 37 41 O=C(COc1ccccc1)NCCCc1ccc(F)cc1 ZINC000217821593 CF In-Stock Unstable FAAH 50 44 O=C(COc1ccccc1)NCCCc1ccc(F)cc1 ZINC000217821593 CF In-Stock Unstable AMP1_PLAFQ 28 40 O=C(COc1ccccc1)NCCCc1ccc(F)cc1 ZINC000217821593 CF In-Stock Unstable TAAR1 15 42 O=C(COc1ccccc1)NCCCc1ccc(F)cc1 ZINC000217821593 CF In-Stock Unstable FFAR1 38 43 O=C(COc1ccccc1)NCCCc1ccc(F)cc1 ZINC000217821593 CF In-Stock Unstable FFAR4 43 43 O=C(COc1ccccc1)NCCCc1ccc(F)cc1 ZINC000217821593 CF In-Stock Unstable CRTM 70 51 O=C(COc1ccccc1)NCCCc1ccc(F)cc1 ZINC000217821593 CF In-Stock Unstable PDS 24 40 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@H](C)O)cc1 ZINC000217821594 HE On-Demand Unstable CA2 25 41 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@H](C)O)cc1 ZINC000217821594 HE On-Demand Unstable CA1 22 41 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@H](C)O)cc1 ZINC000217821594 HE On-Demand Unstable MMP13 37 47 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@H](C)O)cc1 ZINC000217821594 HE On-Demand Unstable MMP2 20 47 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@H](C)O)cc1 ZINC000217821594 HE On-Demand Unstable MMP12 63 45 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@H](C)O)cc1 ZINC000217821594 HE On-Demand Unstable CA12 21 41 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@H](C)O)cc1 ZINC000217821594 HE On-Demand Unstable MMP7 19 45 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@H](C)O)cc1 ZINC000217821594 HE On-Demand Unstable ADAMTS4 51 36 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@H](C)O)cc1 ZINC000217821594 HE On-Demand Unstable CA9 21 41 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@H](C)O)cc1 ZINC000217821594 HE On-Demand Unstable LEF 64 45 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(F)c(Cl)c2)[C@H](C)O)cc1 ZINC000217821594 HE On-Demand Unstable IDO1 29 51 CCOc1ccc(C(=O)[C@@H]2C[C@H]2C(=O)OC)cc1 ZINC000217821634 BE In-Stock Unstable SLC6A1 0 45 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)C1CCNCC1 ZINC000217821636 CF For-Sale Unstable TRPM8 18 50 CC[C@@H](N)CN1C[C@H](C)O[C@@H](C)C1 ZINC000217821643 AC For-Sale Unstable ZM.86993 0 44 COc1ccc(OCCNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217821654 EH For-Sale Unstable HRH2 22 40 COc1ccc(OCCNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217821654 EH For-Sale Unstable MTNR1A 37 45 COc1ccc(OCCNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217821654 EH For-Sale Unstable MTNR1B 30 45 COc1ccccc1CCCNC(=O)COc1ccccc1 ZINC000217821696 CF In-Stock Unstable HTR1A 16 43 COc1ccccc1CCCNC(=O)COc1ccccc1 ZINC000217821696 CF In-Stock Unstable DRD2 21 41 COc1ccccc1CCCNC(=O)COc1ccccc1 ZINC000217821696 CF In-Stock Unstable ADRA1D 15 43 COc1ccccc1CCCNC(=O)COc1ccccc1 ZINC000217821696 CF In-Stock Unstable TSPO 43 36 COc1ccccc1CCCNC(=O)COc1ccccc1 ZINC000217821696 CF In-Stock Unstable MTNR1A 79 49 COc1ccccc1CCCNC(=O)COc1ccccc1 ZINC000217821696 CF In-Stock Unstable MTNR1B 71 49 COc1ccccc1CCCNC(=O)COc1ccccc1 ZINC000217821696 CF In-Stock Unstable PLA2G4B 50 34 COc1ccccc1CCCNC(=O)COc1ccccc1 ZINC000217821696 CF In-Stock Unstable FAAH 18 44 COc1ccccc1CCCNC(=O)COc1ccccc1 ZINC000217821696 CF In-Stock Unstable CRTM 45 41 COc1ccccc1CCCNC(=O)COc1ccccc1 ZINC000217821696 CF In-Stock Unstable MBTPS1 41 40 CN(C(=O)COc1ccc(Oc2ccccc2)cc1)C1CCCC1 ZINC000217821704 EI On-Demand Unstable ALOX5 25 43 CN(C(=O)COc1ccc(Oc2ccccc2)cc1)C1CCCC1 ZINC000217821704 EI On-Demand Unstable SRD5A2 22 40 CN(C(=O)COc1ccc(Oc2ccccc2)cc1)C1CCCC1 ZINC000217821704 EI On-Demand Unstable LTA4H 69 45 CN(C(=O)COc1ccc(Oc2ccccc2)cc1)C1CCCC1 ZINC000217821704 EI On-Demand Unstable CCR5 15 42 CN(C(=O)COc1ccc(Oc2ccccc2)cc1)C1CCCC1 ZINC000217821704 EI On-Demand Unstable COLA 141 48 CN(C(=O)COc1ccc(Oc2ccccc2)cc1)C1CCCC1 ZINC000217821704 EI On-Demand Unstable CPT1A 129 43 CN(C(=O)COc1ccc(Oc2ccccc2)cc1)C1CCCC1 ZINC000217821704 EI On-Demand Unstable CPT2 51 43 CN(C(=O)COc1ccc(Oc2ccccc2)cc1)C1CCCC1 ZINC000217821704 EI On-Demand Unstable AMY2 44 32 CN(C(=O)COc1ccc(Oc2ccccc2)cc1)C1CCCC1 ZINC000217821704 EI On-Demand Unstable PLA2G4B 44 32 CN(C(=O)COc1ccc(Oc2ccccc2)cc1)C1CCCC1 ZINC000217821704 EI On-Demand Unstable NS5B 0 42 CN(C(=O)COc1ccc(Oc2ccccc2)cc1)C1CCCC1 ZINC000217821704 EI On-Demand Unstable LUXN 0 46 CCN(Cc1ccc(OC)c(/C=C\C(=O)O)c1)CC(C)C ZINC000217821705 CG For-Sale Unstable PTGER2 23 41 CCN(Cc1ccc(OC)c(/C=C\C(=O)O)c1)CC(C)C ZINC000217821705 CG For-Sale Unstable PTGER4 0 41 CC[C@H](N)CN1C[C@H](C)O[C@@H](C)C1 ZINC000217821719 AC For-Sale Unstable ZM.86993 0 44 COC(=O)[C@@H](C)N(C)[C@@H](C)c1cccc(Cl)c1 ZINC000217821720 CF For-Sale Unstable ADRB1 23 41 COC(=O)[C@@H](C)N(C)[C@@H](C)c1cccc(Cl)c1 ZINC000217821720 CF For-Sale Unstable ADRB3 37 41 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)C1CCNCC1 ZINC000217821722 CF For-Sale Unstable TRPM8 18 50 CCOc1ccc(C(=O)[C@H]2C[C@H]2C(=O)OC)cc1 ZINC000217821723 BE In-Stock Unstable SLC6A1 0 45 Cc1ncsc1CCNC(=O)C1CCN(C(=O)Cc2ccccc2)CC1 ZINC000217821730 FF In-Stock Unstable GPR183 0 40 COc1ccc(OC[C@@H](C)NC(=O)COc2ccccc2)cc1 ZINC000217821778 DF In-Stock Unstable ADRB2 19 41 COc1ccc(OC[C@@H](C)NC(=O)COc2ccccc2)cc1 ZINC000217821778 DF In-Stock Unstable ADRB1 23 41 COc1ccc(OC[C@@H](C)NC(=O)COc2ccccc2)cc1 ZINC000217821778 DF In-Stock Unstable ADRB3 29 42 COc1ccc(OC[C@@H](C)NC(=O)COc2ccccc2)cc1 ZINC000217821778 DF In-Stock Unstable SDH1 0 50 COc1ccc(OC[C@@H](C)NC(=O)COc2ccccc2)cc1 ZINC000217821778 DF In-Stock Unstable CASP3 17 41 COc1ccc(OC[C@@H](C)NC(=O)COc2ccccc2)cc1 ZINC000217821778 DF In-Stock Unstable ACACA 40 37 COc1ccc(OC[C@@H](C)NC(=O)COc2ccccc2)cc1 ZINC000217821778 DF In-Stock Unstable HDAC8 20 43 COc1ccc(OC[C@@H](C)NC(=O)COc2ccccc2)cc1 ZINC000217821778 DF In-Stock Unstable PLA2G4B 49 33 COc1ccc(OC[C@@H](C)NC(=O)COc2ccccc2)cc1 ZINC000217821778 DF In-Stock Unstable CAPN2 46 41 COc1ccc(OC[C@@H](C)NC(=O)COc2ccccc2)cc1 ZINC000217821778 DF In-Stock Unstable MMP1 29 41 COc1ccc(OC[C@@H](C)NC(=O)COc2ccccc2)cc1 ZINC000217821778 DF In-Stock Unstable DXR 23 41 COc1ccc(OC[C@@H](C)NC(=O)COc2ccccc2)cc1 ZINC000217821778 DF In-Stock Unstable FFAR1 19 42 COc1ccc(OC[C@@H](C)NC(=O)COc2ccccc2)cc1 ZINC000217821778 DF In-Stock Unstable ISPD 0 43 COc1ccc(OC[C@@H](C)NC(=O)COc2ccccc2)cc1 ZINC000217821778 DF In-Stock Unstable PDS 53 38 COc1ccc(OC[C@@H](C)NC(=O)COc2ccccc2)cc1 ZINC000217821778 DF In-Stock Unstable GPR88 0 43 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)Nc3nccs3)[C@H]21 ZINC000217821789 JF In-Stock Unstable MAP1 84 38 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)[C@@H]1CCCCN1 ZINC000217821795 CF For-Sale Unstable TRPM8 17 47 Cn1ccnc1[C@@H](NC(=O)Cn1nnc(-c2ccc(Cl)cc2)n1)c1cccc(F)c1 ZINC000217821810 IF On-Demand Unstable SCARB1 47 41 C=C[C@@H]1O[C@@H]1[C@H](NC(=O)OC(C)(C)C)C(C)C ZINC000217821816 BE For-Sale Unstable CTSK 22 46 O=C(CNS(=O)(=O)c1ccc(F)c(Cl)c1)NC[C@H]1CCCN1c1ccccc1 ZINC000217821825 IF For-Sale Unstable APP 43 35 O=C(CNS(=O)(=O)c1ccc(F)c(Cl)c1)NC[C@H]1CCCN1c1ccccc1 ZINC000217821825 IF For-Sale Unstable SFRP1 81 34 O=C(CNS(=O)(=O)c1ccc(F)c(Cl)c1)NC[C@H]1CCCN1c1ccccc1 ZINC000217821825 IF For-Sale Unstable WNT3 55 33 Cc1nonc1CC(=O)NCc1cc(-c2ccccc2)n[nH]1 ZINC000217821841 CD In-Stock Unstable P2RX7 29 41 Cc1nonc1CC(=O)NCc1cc(-c2ccccc2)n[nH]1 ZINC000217821841 CD In-Stock Unstable HAO2 56 32 COc1ccc(OC[C@H](C)NC(=O)COc2ccccc2)cc1 ZINC000217821854 DF In-Stock Unstable ADRB2 19 41 COc1ccc(OC[C@H](C)NC(=O)COc2ccccc2)cc1 ZINC000217821854 DF In-Stock Unstable ADRB1 23 41 COc1ccc(OC[C@H](C)NC(=O)COc2ccccc2)cc1 ZINC000217821854 DF In-Stock Unstable ADRB3 29 42 COc1ccc(OC[C@H](C)NC(=O)COc2ccccc2)cc1 ZINC000217821854 DF In-Stock Unstable SDH1 0 50 COc1ccc(OC[C@H](C)NC(=O)COc2ccccc2)cc1 ZINC000217821854 DF In-Stock Unstable CASP3 17 41 COc1ccc(OC[C@H](C)NC(=O)COc2ccccc2)cc1 ZINC000217821854 DF In-Stock Unstable ACACA 40 37 COc1ccc(OC[C@H](C)NC(=O)COc2ccccc2)cc1 ZINC000217821854 DF In-Stock Unstable HDAC8 20 43 COc1ccc(OC[C@H](C)NC(=O)COc2ccccc2)cc1 ZINC000217821854 DF In-Stock Unstable PLA2G4B 49 33 COc1ccc(OC[C@H](C)NC(=O)COc2ccccc2)cc1 ZINC000217821854 DF In-Stock Unstable CAPN2 46 41 COc1ccc(OC[C@H](C)NC(=O)COc2ccccc2)cc1 ZINC000217821854 DF In-Stock Unstable MMP1 29 41 COc1ccc(OC[C@H](C)NC(=O)COc2ccccc2)cc1 ZINC000217821854 DF In-Stock Unstable DXR 23 41 COc1ccc(OC[C@H](C)NC(=O)COc2ccccc2)cc1 ZINC000217821854 DF In-Stock Unstable FFAR1 19 42 COc1ccc(OC[C@H](C)NC(=O)COc2ccccc2)cc1 ZINC000217821854 DF In-Stock Unstable ISPD 0 43 COc1ccc(OC[C@H](C)NC(=O)COc2ccccc2)cc1 ZINC000217821854 DF In-Stock Unstable PDS 53 38 COc1ccc(OC[C@H](C)NC(=O)COc2ccccc2)cc1 ZINC000217821854 DF In-Stock Unstable GPR88 0 43 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)Nc3nccs3)[C@@H]21 ZINC000217821867 JF In-Stock Unstable MAP1 84 38 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)[C@@H]1CCCCN1 ZINC000217821879 CF For-Sale Unstable TRPM8 17 47 Cn1ccnc1[C@H](NC(=O)Cn1nnc(-c2ccc(Cl)cc2)n1)c1cccc(F)c1 ZINC000217821887 IF On-Demand Unstable SCARB1 47 41 CC(=O)NCCNC(=O)N/C=C/c1ccccc1Cl ZINC000217821888 CD For-Sale Unstable MTNR1A 25 48 CC(=O)NCCNC(=O)N/C=C/c1ccccc1Cl ZINC000217821888 CD For-Sale Unstable MTNR1B 21 48 C=C[C@@H]1O[C@H]1[C@@H](NC(=O)OC(C)(C)C)C(C)C ZINC000217821895 BE For-Sale Unstable CTSK 22 46 O=C(CNS(=O)(=O)c1ccc(F)c(Cl)c1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217821912 IF For-Sale Unstable APP 43 35 O=C(CNS(=O)(=O)c1ccc(F)c(Cl)c1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217821912 IF For-Sale Unstable SFRP1 81 34 O=C(CNS(=O)(=O)c1ccc(F)c(Cl)c1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217821912 IF For-Sale Unstable WNT3 55 33 O=S(=O)(c1c(F)cccc1F)N1CCC[C@H](Cc2nc(C3CC3)no2)C1 ZINC000217821944 GF In-Stock Unstable PKM 23 40 CCN(Cc1cc(/C=C\C(=O)O)ccc1OC)C(C)C ZINC000217821947 CG For-Sale Unstable PTGER2 0 41 CCN(Cc1cc(/C=C\C(=O)O)ccc1OC)C(C)C ZINC000217821947 CG For-Sale Unstable TUBB1 52 38 CCN(Cc1cc(/C=C\C(=O)O)ccc1OC)C(C)C ZINC000217821947 CG For-Sale Unstable AKR1C3 31 42 CCN(Cc1cc(/C=C\C(=O)O)ccc1OC)C(C)C ZINC000217821947 CG For-Sale Unstable ABCG2 15 40 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)[C@@H]1CCCCN1 ZINC000217821960 CF For-Sale Unstable TRPM8 17 47 CC(C)Oc1cccc(CCCNC(=O)COc2ccccc2)c1 ZINC000217821965 EH In-Stock Unstable ACHE 0 41 CC(C)Oc1cccc(CCCNC(=O)COc2ccccc2)c1 ZINC000217821965 EH In-Stock Unstable ANPEP 24 43 CC(C)Oc1cccc(CCCNC(=O)COc2ccccc2)c1 ZINC000217821965 EH In-Stock Unstable SDH1 0 40 CC(C)Oc1cccc(CCCNC(=O)COc2ccccc2)c1 ZINC000217821965 EH In-Stock Unstable FDFT1 26 58 CC(C)Oc1cccc(CCCNC(=O)COc2ccccc2)c1 ZINC000217821965 EH In-Stock Unstable HDAC8 16 42 CC(C)Oc1cccc(CCCNC(=O)COc2ccccc2)c1 ZINC000217821965 EH In-Stock Unstable MTNR1A 56 46 CC(C)Oc1cccc(CCCNC(=O)COc2ccccc2)c1 ZINC000217821965 EH In-Stock Unstable MTNR1B 65 46 CC(C)Oc1cccc(CCCNC(=O)COc2ccccc2)c1 ZINC000217821965 EH In-Stock Unstable FAAH 36 46 CC(C)Oc1cccc(CCCNC(=O)COc2ccccc2)c1 ZINC000217821965 EH In-Stock Unstable PAM 0 40 CC(C)Oc1cccc(CCCNC(=O)COc2ccccc2)c1 ZINC000217821965 EH In-Stock Unstable FURIN 43 35 CC(C)Oc1cccc(CCCNC(=O)COc2ccccc2)c1 ZINC000217821965 EH In-Stock Unstable CAPN2 29 41 CC(C)Oc1cccc(CCCNC(=O)COc2ccccc2)c1 ZINC000217821965 EH In-Stock Unstable PLM2_PLAFA 22 40 CC(C)Oc1cccc(CCCNC(=O)COc2ccccc2)c1 ZINC000217821965 EH In-Stock Unstable TSPAN17 0 43 CC(C)Oc1cccc(CCCNC(=O)COc2ccccc2)c1 ZINC000217821965 EH In-Stock Unstable AMP1_PLAFQ 51 49 CC(C)Oc1cccc(CCCNC(=O)COc2ccccc2)c1 ZINC000217821965 EH In-Stock Unstable POLG_WNV 47 37 CC(C)Oc1cccc(CCCNC(=O)COc2ccccc2)c1 ZINC000217821965 EH In-Stock Unstable CRTM 95 58 CC(C)Oc1cccc(CCCNC(=O)COc2ccccc2)c1 ZINC000217821965 EH In-Stock Unstable PTGES 28 41 CC(C)Oc1cccc(CCCNC(=O)COc2ccccc2)c1 ZINC000217821965 EH In-Stock Unstable CRTH2 0 44 CC(C)Oc1cccc(CCCNC(=O)COc2ccccc2)c1 ZINC000217821965 EH In-Stock Unstable CAN2 0 40 CC(C)Oc1cccc(CCCNC(=O)COc2ccccc2)c1 ZINC000217821965 EH In-Stock Unstable PDS 73 43 CC(C)Oc1cccc(CCCNC(=O)COc2ccccc2)c1 ZINC000217821965 EH In-Stock Unstable LMGT2 0 42 CCN(C(=O)N/C=C/c1ccccc1Cl)C(C)(C)C ZINC000217821981 CI For-Sale Unstable ECR 56 37 CCN(C(=O)N/C=C/c1ccccc1Cl)C(C)(C)C ZINC000217821981 CI For-Sale Unstable E3UJZ5_SPOLI 43 34 C=C[C@@H]1O[C@H]1[C@H](NC(=O)OC(C)(C)C)C(C)C ZINC000217821985 BE For-Sale Unstable CTSK 22 46 COc1cc([C@@H](C)N(C)[C@@H](C)CC(C)C)ccc1O ZINC000217821989 CH For-Sale Unstable FOLH1 43 48 O=C(CCNS(=O)(=O)c1ccc(F)c(Cl)c1)NC[C@H]1CCCN1c1ccccc1 ZINC000217822017 IF For-Sale Unstable TBXA2R 43 35 O=C(CCNS(=O)(=O)c1ccc(F)c(Cl)c1)NC[C@H]1CCCN1c1ccccc1 ZINC000217822017 IF For-Sale Unstable HTR7 16 40 O=C(CCNS(=O)(=O)c1ccc(F)c(Cl)c1)NC[C@H]1CCCN1c1ccccc1 ZINC000217822017 IF For-Sale Unstable APP 42 35 O=C(CCNS(=O)(=O)c1ccc(F)c(Cl)c1)NC[C@H]1CCCN1c1ccccc1 ZINC000217822017 IF For-Sale Unstable SFRP1 59 33 O=S(=O)(c1c(F)cccc1F)N1CCC[C@@H](Cc2nc(C3CC3)no2)C1 ZINC000217822024 GF In-Stock Unstable PKM 23 40 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)[C@@H]1CCCCN1 ZINC000217822038 CF For-Sale Unstable TRPM8 17 47 CCN(Cc1ccc(OC)c(/C=C\C(=O)O)c1)C(C)C ZINC000217822059 CG For-Sale Unstable PTGER2 35 43 CCN(Cc1ccc(OC)c(/C=C\C(=O)O)c1)C(C)C ZINC000217822059 CG For-Sale Unstable PTGER4 0 43 CCN(Cc1ccc(OC)c(/C=C\C(=O)O)c1)C(C)C ZINC000217822059 CG For-Sale Unstable PTGER3 17 43 CC(C)Oc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822076 EH In-Stock Unstable ALOX5 17 40 CC(C)Oc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822076 EH In-Stock Unstable PPARG 20 44 CC(C)Oc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822076 EH In-Stock Unstable PPARA 20 44 CC(C)Oc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822076 EH In-Stock Unstable ADRB3 41 38 CC(C)Oc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822076 EH In-Stock Unstable ANPEP 18 43 CC(C)Oc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822076 EH In-Stock Unstable SDH1 0 41 CC(C)Oc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822076 EH In-Stock Unstable FDFT1 17 45 CC(C)Oc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822076 EH In-Stock Unstable ACACA 41 38 CC(C)Oc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822076 EH In-Stock Unstable SCN2A 23 42 CC(C)Oc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822076 EH In-Stock Unstable HDAC8 15 47 CC(C)Oc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822076 EH In-Stock Unstable MTNR1A 42 40 CC(C)Oc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822076 EH In-Stock Unstable MTNR1B 43 42 CC(C)Oc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822076 EH In-Stock Unstable MMP8 15 43 CC(C)Oc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822076 EH In-Stock Unstable PLA2G4B 64 41 CC(C)Oc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822076 EH In-Stock Unstable FAAH 44 44 CC(C)Oc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822076 EH In-Stock Unstable CAPN2 0 43 CC(C)Oc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822076 EH In-Stock Unstable AMP1_PLAFQ 33 43 CC(C)Oc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822076 EH In-Stock Unstable FFAR1 40 38 CC(C)Oc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822076 EH In-Stock Unstable CRTM 62 47 O=C(N/C=C/c1ccccc1Cl)NC12CC3CC(CC(C3)C1)C2 ZINC000217822079 EJ For-Sale Unstable EPHX2 101 50 O=C(CCNS(=O)(=O)c1ccc(F)c(Cl)c1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217822096 IF For-Sale Unstable TBXA2R 43 35 O=C(CCNS(=O)(=O)c1ccc(F)c(Cl)c1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217822096 IF For-Sale Unstable HTR7 16 40 O=C(CCNS(=O)(=O)c1ccc(F)c(Cl)c1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217822096 IF For-Sale Unstable APP 42 35 O=C(CCNS(=O)(=O)c1ccc(F)c(Cl)c1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217822096 IF For-Sale Unstable SFRP1 59 33 C[C@@H](c1ccccc1F)N(C)[C@H](C)C(=O)O ZINC000217822099 BE For-Sale Unstable CES2 20 40 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)[C@@H]1CCCNC1 ZINC000217822129 CF On-Demand Unstable TRPM8 18 47 O=S(=O)(c1cccc(C(F)(F)F)c1)N1CCC[C@H](Cc2nc(C3CC3)no2)C1 ZINC000217822136 HH In-Stock Unstable CACNA1B 47 35 CCc1ccc(C[C@@H]2C[C@@H]2C(=O)O)cc1 ZINC000217822179 BF In-Stock Unstable GRIK2 25 44 CCCN(Cc1ccc(OC)c(/C=C\C(=O)O)c1)C1CC1 ZINC000217822182 CG For-Sale Unstable PTGER2 29 40 CCCN(Cc1ccc(OC)c(/C=C\C(=O)O)c1)C1CC1 ZINC000217822182 CG For-Sale Unstable PTGER4 0 40 O=C(N/C=C/c1ccccc1Cl)Nc1cccc2cccnc12 ZINC000217822188 DJ For-Sale Anodyne PFHDAC1 0 41 CCOc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822196 DG In-Stock Unstable ALOX5 19 46 CCOc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822196 DG In-Stock Unstable LTA4H 44 41 CCOc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822196 DG In-Stock Unstable SDH1 0 44 CCOc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822196 DG In-Stock Unstable FDFT1 18 47 CCOc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822196 DG In-Stock Unstable CYSP_TRYCR 0 40 CCOc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822196 DG In-Stock Unstable SCN2A 42 55 CCOc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822196 DG In-Stock Unstable PLA2G4A 36 40 CCOc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822196 DG In-Stock Unstable HDAC8 18 47 CCOc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822196 DG In-Stock Unstable MTNR1A 58 42 CCOc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822196 DG In-Stock Unstable MTNR1B 51 44 CCOc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822196 DG In-Stock Unstable MMP3 21 43 CCOc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822196 DG In-Stock Unstable PLA2G4B 80 43 CCOc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822196 DG In-Stock Unstable FAAH 53 43 CCOc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822196 DG In-Stock Unstable S1PR1 17 40 CCOc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822196 DG In-Stock Unstable AMP1_PLAFQ 29 42 CCOc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822196 DG In-Stock Unstable FFAR1 43 41 CCOc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822196 DG In-Stock Unstable FFAR4 45 37 CCOc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822196 DG In-Stock Unstable CRTM 72 50 CCOc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822196 DG In-Stock Unstable PDS 68 44 CCOc1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217822196 DG In-Stock Unstable CES1D 45 33 O=C(CCNS(=O)(=O)c1cccc(F)c1)NC[C@H]1CCCN1c1ccccc1 ZINC000217822213 HE For-Sale Unstable SFRP1 88 34 O=C(CCNS(=O)(=O)c1cccc(F)c1)NC[C@H]1CCCN1c1ccccc1 ZINC000217822213 HE For-Sale Unstable WNT3 58 32 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)[C@@H]1CCCNC1 ZINC000217822215 CF On-Demand Unstable TRPM8 18 47 O=S(=O)(c1cccc(C(F)(F)F)c1)N1CCC[C@@H](Cc2nc(C3CC3)no2)C1 ZINC000217822223 HH In-Stock Unstable CACNA1B 47 35 CCc1ccc(C[C@H]2C[C@@H]2C(=O)O)cc1 ZINC000217822263 BF In-Stock Unstable GRIK2 25 44 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)[C@@H]1CCCNC1 ZINC000217822292 CF For-Sale Unstable TRPM8 17 46 O=C(CCNS(=O)(=O)c1cccc(F)c1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217822297 HE For-Sale Unstable SFRP1 88 34 O=C(CCNS(=O)(=O)c1cccc(F)c1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217822297 HE For-Sale Unstable WNT3 58 32 CCCOc1ccccc1CCCNC(=O)COc1ccccc1 ZINC000217822302 EH In-Stock Unstable LTB4R 40 36 CCCOc1ccccc1CCCNC(=O)COc1ccccc1 ZINC000217822302 EH In-Stock Unstable MTNR1A 57 44 CCCOc1ccccc1CCCNC(=O)COc1ccccc1 ZINC000217822302 EH In-Stock Unstable MTNR1B 67 46 CCCOc1ccccc1CCCNC(=O)COc1ccccc1 ZINC000217822302 EH In-Stock Unstable PLA2G4B 80 37 CCCOc1ccccc1CCCNC(=O)COc1ccccc1 ZINC000217822302 EH In-Stock Unstable CRTM 43 39 CCc1ccc(C[C@@H]2C[C@H]2C(=O)O)cc1 ZINC000217822357 BF In-Stock Unstable GRIK2 25 44 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)[C@@H]1CCCNC1 ZINC000217822371 CF For-Sale Unstable TRPM8 17 46 C[C@@H]1Cc2ccccc2N1C(=O)N/C=C/c1ccccc1Cl ZINC000217822391 DI For-Sale Unstable DRD4 27 47 C[C@@H]1Cc2ccccc2N1C(=O)N/C=C/c1ccccc1Cl ZINC000217822391 DI For-Sale Unstable TPP2 45 34 CCCCCN(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217822396 CG For-Sale Unstable THRA 61 46 CCCCCN(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217822396 CG For-Sale Unstable FDPS 33 43 CCCCCN(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217822396 CG For-Sale Unstable ACHE 0 45 CCCCCN(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217822396 CG For-Sale Unstable THRB 30 46 CCCCCN(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217822396 CG For-Sale Unstable LTB4R 22 42 CCCCCN(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217822396 CG For-Sale Unstable PLA2G4B 85 42 CCCCCN(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217822396 CG For-Sale Unstable LSS 48 34 CCCCCN(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217822396 CG For-Sale Unstable AKR1C3 26 42 CC1CCN(c2ccc([C@@H](C)NC(=O)COc3ccccc3)cc2)CC1 ZINC000217822419 FI In-Stock Unstable ACACA 50 40 CC1CCN(c2ccc([C@@H](C)NC(=O)COc3ccccc3)cc2)CC1 ZINC000217822419 FI In-Stock Unstable PRCP 15 42 CC1CCN(c2ccc([C@@H](C)NC(=O)COc3ccccc3)cc2)CC1 ZINC000217822419 FI In-Stock Unstable ACACB 27 40 CC1CCN(c2ccc([C@@H](C)NC(=O)COc3ccccc3)cc2)CC1 ZINC000217822419 FI In-Stock Unstable COLA 65 35 CC1CCN(c2ccc([C@@H](C)NC(=O)COc3ccccc3)cc2)CC1 ZINC000217822419 FI In-Stock Unstable CPT1A 61 35 CC1CCN(c2ccc([C@@H](C)NC(=O)COc3ccccc3)cc2)CC1 ZINC000217822419 FI In-Stock Unstable CAPN2 43 39 CCc1ccc(C[C@H]2C[C@H]2C(=O)O)cc1 ZINC000217822450 BF In-Stock Unstable GRIK2 25 44 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1ccc(CN)cc1 ZINC000217822469 CG On-Demand Unstable TRPM8 23 71 C[C@H]1Cc2ccccc2N1C(=O)N/C=C/c1ccccc1Cl ZINC000217822478 DI For-Sale Unstable DRD4 27 47 C[C@H]1Cc2ccccc2N1C(=O)N/C=C/c1ccccc1Cl ZINC000217822478 DI For-Sale Unstable TPP2 45 34 CC1CCN(c2ccc([C@H](C)NC(=O)COc3ccccc3)cc2)CC1 ZINC000217822513 FI In-Stock Unstable ACACA 50 40 CC1CCN(c2ccc([C@H](C)NC(=O)COc3ccccc3)cc2)CC1 ZINC000217822513 FI In-Stock Unstable PRCP 15 42 CC1CCN(c2ccc([C@H](C)NC(=O)COc3ccccc3)cc2)CC1 ZINC000217822513 FI In-Stock Unstable ACACB 27 40 CC1CCN(c2ccc([C@H](C)NC(=O)COc3ccccc3)cc2)CC1 ZINC000217822513 FI In-Stock Unstable COLA 65 35 CC1CCN(c2ccc([C@H](C)NC(=O)COc3ccccc3)cc2)CC1 ZINC000217822513 FI In-Stock Unstable CPT1A 61 35 CC1CCN(c2ccc([C@H](C)NC(=O)COc3ccccc3)cc2)CC1 ZINC000217822513 FI In-Stock Unstable CAPN2 43 39 CCCCCN(C)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217822514 CG For-Sale Unstable THRA 75 41 CCCCCN(C)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217822514 CG For-Sale Unstable FDPS 32 42 CCCCCN(C)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217822514 CG For-Sale Unstable LTA4H 22 47 CCCCCN(C)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217822514 CG For-Sale Unstable THRB 36 41 CCCCCN(C)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217822514 CG For-Sale Unstable SHC 31 41 CCCCCN(C)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217822514 CG For-Sale Unstable PLA2G4B 93 40 CCCCCN(C)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217822514 CG For-Sale Unstable LSS 57 41 CCCCCN(C)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217822514 CG For-Sale Unstable FAAH 23 41 CCCCCN(C)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217822514 CG For-Sale Unstable AKR1C3 0 43 CCCCCN(C)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217822514 CG For-Sale Unstable NORA 0 49 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1ccc(CN)cc1 ZINC000217822544 CG On-Demand Unstable TRPM8 23 71 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)c1ccc(CN)cc1 ZINC000217822611 CG For-Sale Unstable TRPM8 23 71 CN(Cc1ccsc1)Cc1ccccc1/C=C\C(=O)O ZINC000217822623 CG For-Sale Unstable PTGER2 54 44 CN(Cc1ccsc1)Cc1ccccc1/C=C\C(=O)O ZINC000217822623 CG For-Sale Unstable PTGER4 26 40 CN(Cc1ccsc1)Cc1ccccc1/C=C\C(=O)O ZINC000217822623 CG For-Sale Unstable PTGER3 21 45 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)COc3ccccc3)cc2)C1 ZINC000217822644 FI In-Stock Unstable HRH3 0 41 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)COc3ccccc3)cc2)C1 ZINC000217822644 FI In-Stock Unstable COLA 80 35 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)COc3ccccc3)cc2)C1 ZINC000217822644 FI In-Stock Unstable CPT1A 72 35 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)COc3ccccc3)cc2)C1 ZINC000217822644 FI In-Stock Unstable CAPN2 41 39 COC(=O)C[C@@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(OCC(=O)O)c(OC)c1 ZINC000217822664 IF In-Stock Unstable TNF 22 43 O=C(N/C=C/c1ccccc1Cl)N1CCN(c2ncccn2)CC1 ZINC000217822686 EF For-Sale Unstable SLC6A7 0 46 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)c1ccc(CN)cc1 ZINC000217822688 CG For-Sale Unstable TRPM8 23 71 C=C(CN[C@@H](CC)CCO)c1ccccc1 ZINC000217822705 BE For-Sale Unstable AOC3 49 50 C[C@H](NC(=O)COc1ccccc1)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217822722 FI In-Stock Unstable HRH3 0 41 C[C@H](NC(=O)COc1ccccc1)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217822722 FI In-Stock Unstable COLA 80 35 C[C@H](NC(=O)COc1ccccc1)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217822722 FI In-Stock Unstable CPT1A 72 35 C[C@H](NC(=O)COc1ccccc1)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217822722 FI In-Stock Unstable CAPN2 41 39 COC(=O)C[C@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(OCC(=O)O)c(OC)c1 ZINC000217822736 IF In-Stock Unstable TNF 22 43 C[C@@H]1CCCN1[C@@](C)(C(=O)O)c1ccccc1 ZINC000217822748 BE For-Sale Unstable CHRM3 54 45 C[C@@H]1CCCN1[C@@](C)(C(=O)O)c1ccccc1 ZINC000217822748 BE For-Sale Unstable HRH3 0 44 C[C@@H]1CCCN1[C@@](C)(C(=O)O)c1ccccc1 ZINC000217822748 BE For-Sale Unstable AMY2 46 32 C[C@@H]1CCCN1[C@@](C)(C(=O)O)c1ccccc1 ZINC000217822748 BE For-Sale Unstable CYP2J2 47 35 C=C(CN[C@H](CC)CCO)c1ccccc1 ZINC000217822773 BE For-Sale Unstable AOC3 49 50 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)CN ZINC000217822796 BD On-Demand Unstable TRPM8 22 55 Cc1cccc(N2CCN(C(=O)N/C=C/c3ccccc3Cl)CC2)c1 ZINC000217822800 FI For-Sale Unstable CCR1 22 43 C[C@H]1CCCN1[C@@](C)(C(=O)O)c1ccccc1 ZINC000217822830 BE For-Sale Unstable CHRM3 54 45 C[C@H]1CCCN1[C@@](C)(C(=O)O)c1ccccc1 ZINC000217822830 BE For-Sale Unstable HRH3 0 44 C[C@H]1CCCN1[C@@](C)(C(=O)O)c1ccccc1 ZINC000217822830 BE For-Sale Unstable AMY2 46 32 C[C@H]1CCCN1[C@@](C)(C(=O)O)c1ccccc1 ZINC000217822830 BE For-Sale Unstable CYP2J2 47 35 Cc1ccc2c(c1)[C@@H](NC(=O)COc1ccccc1)CC(C)(C)O2 ZINC000217822840 EH In-Stock Unstable PBPX 0 41 Cc1ccc2c(c1)[C@@H](NC(=O)COc1ccccc1)CC(C)(C)O2 ZINC000217822840 EH In-Stock Unstable LUXN 0 40 COc1ccc(CNC(=O)CNc2ccc3c(cc2=O)[C@@H](NC(C)=O)CCc2cc(OC)c(OC)c(OC)c2-3)cc1OC ZINC000217822845 KH In-Stock Unstable TUBA1A 19 70 COc1ccc(CNC(=O)CNc2ccc3c(cc2=O)[C@@H](NC(C)=O)CCc2cc(OC)c(OC)c(OC)c2-3)cc1OC ZINC000217822845 KH In-Stock Unstable TPPP 0 69 O=C(NC[C@@H]1CCCCO1)c1cc(=O)n(-c2ccccc2)[nH]1 ZINC000217822852 DD In-Stock Unstable CTSA 59 43 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)CN ZINC000217822878 BD On-Demand Unstable TRPM8 22 55 CCOC(=O)N1CCC(NC(=O)N/C=C/c2ccccc2Cl)CC1 ZINC000217822908 FG For-Sale Unstable EPHX2 39 41 CCOC(=O)N1CCC(NC(=O)N/C=C/c2ccccc2Cl)CC1 ZINC000217822908 FG For-Sale Unstable CCR8 35 42 Cc1ccc2c(c1)[C@H](NC(=O)COc1ccccc1)CC(C)(C)O2 ZINC000217822925 EH In-Stock Unstable PBPX 0 41 Cc1ccc2c(c1)[C@H](NC(=O)COc1ccccc1)CC(C)(C)O2 ZINC000217822925 EH In-Stock Unstable LUXN 0 40 O=C(NC[C@H]1CCCCO1)c1cc(=O)n(-c2ccccc2)[nH]1 ZINC000217822940 DD In-Stock Unstable CTSA 59 43 COc1ccc(/C=C\C(=O)O)cc1CN(C)[C@@H](C)C1CC1 ZINC000217822944 CG For-Sale Unstable AKR1C3 38 41 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)CN ZINC000217822955 BD For-Sale Unstable TRPM8 22 55 CC(C)(C)c1ccc(S(=O)(=O)NCCC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217822993 IG For-Sale Unstable ADAMTS5 34 43 CC(C)(C)c1ccc(S(=O)(=O)NCCC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217822993 IG For-Sale Unstable SFRP1 98 34 CC(C)(C)c1ccc(S(=O)(=O)NCCC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217822993 IG For-Sale Unstable WNT3 68 33 O=C(N/C=C/c1ccccc1Cl)N1CCN(c2cccc(Cl)c2)CC1 ZINC000217823004 GI For-Sale Unstable HTR1A 17 45 O=C(N/C=C/c1ccccc1Cl)N1CCN(c2cccc(Cl)c2)CC1 ZINC000217823004 GI For-Sale Unstable RBP4 17 40 COc1ccc(/C=C\C(=O)O)cc1CN(C)[C@H](C)C1CC1 ZINC000217823015 CG For-Sale Unstable AKR1C3 38 41 Cc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)COc1ccccc1 ZINC000217823027 EH In-Stock Unstable PBPX 0 42 Cc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)COc1ccccc1 ZINC000217823027 EH In-Stock Unstable LUXN 0 41 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)CN ZINC000217823028 BD For-Sale Unstable TRPM8 22 55 CC(C)(C)c1ccc(S(=O)(=O)NCCC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217823069 IG For-Sale Unstable ADAMTS5 34 43 CC(C)(C)c1ccc(S(=O)(=O)NCCC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217823069 IG For-Sale Unstable SFRP1 98 34 CC(C)(C)c1ccc(S(=O)(=O)NCCC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217823069 IG For-Sale Unstable WNT3 68 33 O=C(O)CCCCCNC(=O)[C@@H]1C[C@@H]2CCCC[C@@H]2N1 ZINC000217823075 CD On-Demand Unstable EPHX2 0 40 CC(=O)[C@@H](C)N(C)[C@@H](C)c1ccc(Cl)cc1 ZINC000217823081 BG For-Sale Unstable UTS2 50 38 Cc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)COc1ccccc1 ZINC000217823089 EH In-Stock Unstable PBPX 0 42 Cc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)COc1ccccc1 ZINC000217823089 EH In-Stock Unstable LUXN 0 41 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1cccc(N)c1 ZINC000217823109 CG On-Demand Unstable TRPM8 0 75 O=C(O)/C=C\c1ccccc1CN1CCCCCC1=O ZINC000217823111 CF For-Sale Unstable PTGER2 44 50 O=C(O)/C=C\c1ccccc1CN1CCCCCC1=O ZINC000217823111 CF For-Sale Unstable PTGER4 23 48 O=C(O)/C=C\c1ccccc1CN1CCCCCC1=O ZINC000217823111 CF For-Sale Unstable PTGER3 19 50 Cc1ccc2nc(-c3ccc(NC(=O)N/C=C/c4ccccc4Cl)cc3)sc2c1 ZINC000217823120 HK For-Sale Unstable CSNK1D 25 41 Cc1ccc2nc(-c3ccc(NC(=O)N/C=C/c4ccccc4Cl)cc3)sc2c1 ZINC000217823120 HK For-Sale Unstable APP 25 52 Cc1ccc2nc(-c3ccc(NC(=O)N/C=C/c4ccccc4Cl)cc3)sc2c1 ZINC000217823120 HK For-Sale Unstable NR2E3 45 33 COC(=O)c1ccccc1S(=O)(=O)NCC(F)(F)F ZINC000217823153 CD For-Sale Unstable PRTN3 45 32 COC(=O)c1ccccc1S(=O)(=O)NCC(F)(F)F ZINC000217823153 CD For-Sale Unstable ILV2 0 40 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1cccc(N)c1 ZINC000217823174 CG On-Demand Unstable TRPM8 23 75 O=C(O)CCCCCNC(=O)[C@@H]1C[C@H]2CCCC[C@@H]2N1 ZINC000217823187 CD On-Demand Unstable EPHX2 0 40 COc1ccc2c(c1)[C@@H](NC(=O)COc1ccccc1)CC(C)(C)O2 ZINC000217823202 EG In-Stock Unstable TRAR 36 40 COc1ccc2c(c1)[C@@H](NC(=O)COc1ccccc1)CC(C)(C)O2 ZINC000217823202 EG In-Stock Unstable PBPX 0 41 COc1ccc2c(c1)[C@@H](NC(=O)COc1ccccc1)CC(C)(C)O2 ZINC000217823202 EG In-Stock Unstable LUXN 0 42 CCN1CCN(Cc2ccc(OCC(N)=O)cc2)C[C@@H](O)C1 ZINC000217823223 DC In-Stock Unstable HRH3 18 43 O=C(N/C=C/c1ccccc1Cl)Nc1ccc2c(c1)OCO2 ZINC000217823237 DH For-Sale Unstable KCNQ2 15 52 O=C(N/C=C/c1ccccc1Cl)Nc1ccc2c(c1)OCO2 ZINC000217823237 DH For-Sale Unstable CCR2 0 50 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)c1cccc(N)c1 ZINC000217823260 CG For-Sale Unstable TRPM8 21 65 COc1ccc2c(c1)[C@H](NC(=O)COc1ccccc1)CC(C)(C)O2 ZINC000217823284 EG In-Stock Unstable TRAR 36 40 COc1ccc2c(c1)[C@H](NC(=O)COc1ccccc1)CC(C)(C)O2 ZINC000217823284 EG In-Stock Unstable PBPX 0 41 COc1ccc2c(c1)[C@H](NC(=O)COc1ccccc1)CC(C)(C)O2 ZINC000217823284 EG In-Stock Unstable LUXN 0 42 CC(C)NC(=O)CCCCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12 ZINC000217823317 HH In-Stock Unstable TOP1 0 40 O=C(O)[C@@H]1[C@H]2CN(C(=O)CCc3cccnc3)C[C@H]21 ZINC000217823336 CC In-Stock Unstable TBXAS1 40 47 O=C(O)[C@@H]1[C@H]2CN(C(=O)CCc3cccnc3)C[C@H]21 ZINC000217823336 CC In-Stock Unstable PTAFR 33 46 O=C(O)[C@@H]1[C@H]2CN(C(=O)CCc3cccnc3)C[C@H]21 ZINC000217823336 CC In-Stock Unstable C3AR1 57 50 O=C(O)[C@@H]1[C@H]2CN(C(=O)CCc3cccnc3)C[C@H]21 ZINC000217823336 CC In-Stock Unstable NAMPT 22 40 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)c1cccc(N)c1 ZINC000217823342 CG For-Sale Unstable TRPM8 21 65 O=C(NC[C@H]1CCCN1c1ccccc1)c1cccc(NS(=O)(=O)c2cccc(F)c2)c1 ZINC000217823402 JI For-Sale Unstable SFRP1 54 35 O=C(NC[C@H]1CCCN1c1ccccc1)c1cccc(NS(=O)(=O)c2cccc(F)c2)c1 ZINC000217823402 JI For-Sale Unstable LIMK2 32 42 O=C(NC[C@H]1CCCN1c1ccccc1)c1cccc(NS(=O)(=O)c2cccc(F)c2)c1 ZINC000217823402 JI For-Sale Unstable ACKR3 56 33 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)COc1ccccc1 ZINC000217823405 EG In-Stock Unstable TRPV1 0 45 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)COc1ccccc1 ZINC000217823405 EG In-Stock Unstable MTNR1A 46 33 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)COc1ccccc1 ZINC000217823405 EG In-Stock Unstable TRAR 42 40 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)COc1ccccc1 ZINC000217823405 EG In-Stock Unstable PBPX 0 41 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)COc1ccccc1 ZINC000217823405 EG In-Stock Unstable LUXN 0 43 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)COc1ccccc1 ZINC000217823405 EG In-Stock Unstable ISPD 0 40 CC(C)NC(=O)CCCCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12 ZINC000217823406 HH In-Stock Unstable TOP1 0 40 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1ccc(N)cc1 ZINC000217823416 CG For-Sale Unstable TRPM8 23 76 O=C(N/C=C/c1ccccc1Cl)Nc1cccc(F)c1 ZINC000217823461 CI For-Sale Anodyne KCNK3 52 44 O=C(O)[C@@H]1CCCN1C(=O)[C@@H]1C[C@@H]2CCCC[C@@H]2N1 ZINC000217823487 CC For-Sale Unstable ACE 24 49 O=C(O)[C@@H]1CCCN1C(=O)[C@@H]1C[C@@H]2CCCC[C@@H]2N1 ZINC000217823487 CC For-Sale Unstable MME 0 47 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)COc1ccccc1 ZINC000217823492 EG In-Stock Unstable TRPV1 0 45 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)COc1ccccc1 ZINC000217823492 EG In-Stock Unstable MTNR1A 46 33 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)COc1ccccc1 ZINC000217823492 EG In-Stock Unstable TRAR 42 40 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)COc1ccccc1 ZINC000217823492 EG In-Stock Unstable PBPX 0 41 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)COc1ccccc1 ZINC000217823492 EG In-Stock Unstable LUXN 0 43 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)COc1ccccc1 ZINC000217823492 EG In-Stock Unstable ISPD 0 40 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cccc(NS(=O)(=O)c2cccc(F)c2)c1 ZINC000217823496 JI For-Sale Unstable SFRP1 54 35 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cccc(NS(=O)(=O)c2cccc(F)c2)c1 ZINC000217823496 JI For-Sale Unstable LIMK2 32 42 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cccc(NS(=O)(=O)c2cccc(F)c2)c1 ZINC000217823496 JI For-Sale Unstable ACKR3 56 33 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1ccc(N)cc1 ZINC000217823506 CG For-Sale Unstable TRPM8 23 76 CC(=O)[C@@H](C)N(C)[C@@H](C)c1cccc(Cl)c1 ZINC000217823554 BG For-Sale Unstable PSBA 0 44 O=C(O)[C@H]1CCCN1C(=O)[C@@H]1C[C@@H]2CCCC[C@@H]2N1 ZINC000217823565 CC For-Sale Unstable ACE 24 49 O=C(O)[C@H]1CCCN1C(=O)[C@@H]1C[C@@H]2CCCC[C@@H]2N1 ZINC000217823565 CC For-Sale Unstable MME 0 47 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)c1ccc(N)cc1 ZINC000217823589 CG For-Sale Unstable TRPM8 23 76 COc1ccc(Br)cc1CCC(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217823594 HI For-Sale Unstable DRD2 36 44 COc1ccc(Br)cc1CCC(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217823594 HI For-Sale Unstable DRD3 17 46 COc1ccc(Br)cc1CCC(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217823594 HI For-Sale Unstable MBTPS1 48 34 COc1ccc(Br)cc1CCC(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217823594 HI For-Sale Unstable ACKR3 58 34 CC[C@@H](NC(=O)COc1ccccc1)c1ccc(C)c(C)c1 ZINC000217823609 CH In-Stock Unstable PTGER3 51 45 CC[C@@H](NC(=O)COc1ccccc1)c1ccc(C)c(C)c1 ZINC000217823609 CH In-Stock Unstable TACR3 43 37 CC[C@@H](NC(=O)COc1ccccc1)c1ccc(C)c(C)c1 ZINC000217823609 CH In-Stock Unstable ACE2 41 33 CC[C@@H](NC(=O)COc1ccccc1)c1ccc(C)c(C)c1 ZINC000217823609 CH In-Stock Unstable FFAR1 18 40 CC[C@@H](NC(=O)COc1ccccc1)c1ccc(C)c(C)c1 ZINC000217823609 CH In-Stock Unstable PDS 74 39 Cc1ccc(C[C@@H]2C[C@@H]2C(=O)O)cc1C ZINC000217823623 BF In-Stock Unstable GRIK2 31 40 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)c1ccc(N)cc1 ZINC000217823666 CG For-Sale Unstable TRPM8 23 76 COc1ccc(Br)cc1CCC(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217823680 HI For-Sale Unstable DRD2 36 44 COc1ccc(Br)cc1CCC(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217823680 HI For-Sale Unstable DRD3 17 46 COc1ccc(Br)cc1CCC(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217823680 HI For-Sale Unstable MBTPS1 48 34 COc1ccc(Br)cc1CCC(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217823680 HI For-Sale Unstable ACKR3 58 34 CC[C@H](NC(=O)COc1ccccc1)c1ccc(C)c(C)c1 ZINC000217823681 CH In-Stock Unstable PTGER3 51 45 CC[C@H](NC(=O)COc1ccccc1)c1ccc(C)c(C)c1 ZINC000217823681 CH In-Stock Unstable TACR3 43 37 CC[C@H](NC(=O)COc1ccccc1)c1ccc(C)c(C)c1 ZINC000217823681 CH In-Stock Unstable ACE2 41 33 CC[C@H](NC(=O)COc1ccccc1)c1ccc(C)c(C)c1 ZINC000217823681 CH In-Stock Unstable FFAR1 18 40 CC[C@H](NC(=O)COc1ccccc1)c1ccc(C)c(C)c1 ZINC000217823681 CH In-Stock Unstable PDS 74 39 O=C(N/C=C/c1ccccc1Cl)N1CCc2ccccc21 ZINC000217823688 CI For-Sale Unstable AVPR2 32 41 Cc1ccc(C[C@H]2C[C@@H]2C(=O)O)cc1C ZINC000217823701 BF In-Stock Unstable GRIK2 31 40 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)Cc1ccc(N)cc1 ZINC000217823764 CG On-Demand Unstable TRPM8 22 58 Cc1ccc(C[C@@H]2C[C@H]2C(=O)O)cc1C ZINC000217823780 BF In-Stock Unstable GRIK2 31 40 O=C(CCc1ccc(Br)cc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217823788 GI For-Sale Unstable TRAR 17 41 CC[C@@H](NC(=O)COc1ccccc1)c1ccc(C)cc1C ZINC000217823795 CH In-Stock Unstable RORC 18 43 CC[C@@H](NC(=O)COc1ccccc1)c1ccc(C)cc1C ZINC000217823795 CH In-Stock Unstable PDS 67 40 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(I)cc1 ZINC000217823809 GJ For-Sale Anodyne SMO 19 40 O=C(O)/C=C\c1ccccc1CN1C(=O)CCCCC1=O ZINC000217823810 CE For-Sale Unstable PTGER3 31 49 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)Cc1ccc(N)cc1 ZINC000217823841 CG On-Demand Unstable TRPM8 22 58 Cc1ccc(C[C@H]2C[C@H]2C(=O)O)cc1C ZINC000217823850 BF In-Stock Unstable GRIK2 31 40 O=C(CCc1ccc(Br)cc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217823855 GI For-Sale Unstable TRAR 17 41 CC[C@H](NC(=O)COc1ccccc1)c1ccc(C)cc1C ZINC000217823883 CH In-Stock Unstable RORC 18 43 CC[C@H](NC(=O)COc1ccccc1)c1ccc(C)cc1C ZINC000217823883 CH In-Stock Unstable PDS 67 40 COc1cc2c(cc1OC)CN(Cc1oc(CN3CCCCC3)cc(=O)c1O)CC2 ZINC000217823888 HF In-Stock Unstable ABCB1B 61 35 COc1cc2c(cc1OC)CN(Cc1oc(CN3CCCCC3)cc(=O)c1O)CC2 ZINC000217823888 HF In-Stock Unstable ABCB1 23 47 CC(=O)[C@@H](C)N(C)[C@@H](C)c1ccccc1F ZINC000217823898 BF For-Sale Unstable CES2 20 40 CSCCOc1ccc(Cl)cc1Br ZINC000217823916 CH On-Demand Unstable S1PR4 36 51 O=C(N/C=C/c1ccccc1Cl)NCCc1c[nH]c2ccccc12 ZINC000217823920 EI For-Sale Unstable ACHE 27 40 O=C(N/C=C/c1ccccc1Cl)NCCc1c[nH]c2ccccc12 ZINC000217823920 EI For-Sale Unstable TACR1 0 43 O=C(N/C=C/c1ccccc1Cl)NCCc1c[nH]c2ccccc12 ZINC000217823920 EI For-Sale Unstable MC4R 33 47 O=C(N/C=C/c1ccccc1Cl)NCCc1c[nH]c2ccccc12 ZINC000217823920 EI For-Sale Unstable CCKAR 31 42 O=C(N/C=C/c1ccccc1Cl)NCCc1c[nH]c2ccccc12 ZINC000217823920 EI For-Sale Unstable BCHE 15 41 O=C(N/C=C/c1ccccc1Cl)NCCc1c[nH]c2ccccc12 ZINC000217823920 EI For-Sale Unstable MPO 25 41 O=C(N/C=C/c1ccccc1Cl)NCCc1c[nH]c2ccccc12 ZINC000217823920 EI For-Sale Unstable BRS3 27 42 O=C(N/C=C/c1ccccc1Cl)NCCc1c[nH]c2ccccc12 ZINC000217823920 EI For-Sale Unstable NMBR 37 44 O=C(N/C=C/c1ccccc1Cl)NCCc1c[nH]c2ccccc12 ZINC000217823920 EI For-Sale Unstable SSTR3 17 40 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable ACHE 36 45 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable MME 22 40 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable EDNRB 46 34 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable EDNRA 37 40 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable TACR1 43 54 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable NQO2 28 42 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable TACR2 24 48 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable CCKAR 75 53 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable MPO 55 37 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable BRS3 28 53 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable NMBR 46 30 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable MC3R 54 38 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable MC5R 55 33 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable CA5B 25 40 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable CA5A 24 40 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable MTNR1A 34 48 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable MTNR1B 26 44 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable MMP2 24 44 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable MMP8 35 44 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable GRIA1 24 45 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable MMP14 68 44 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable GRPR 66 35 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable ECE1 51 39 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable MMP11 50 32 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable CCKBR 66 42 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable GHSR 57 41 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable ALOX15 31 51 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable MC1R 66 38 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable ADAM9 40 41 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable MMP1 23 50 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable NPR 29 40 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable SLC15A2 0 44 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable KISS1R 61 34 CS(=O)(=O)CC(=O)NCCc1c[nH]c2ccccc12 ZINC000217823921 CC On-Demand Unstable LASB 0 42 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)Cc1ccc(N)cc1 ZINC000217823937 CG For-Sale Unstable TRPM8 22 58 C[C@H](Cc1ccc(O)cc1)N1CCO[C@@H]2CCCC[C@@H]21 ZINC000217823957 CF For-Sale Unstable YARS 51 32 CCCOc1ccc(CCC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217823966 FI For-Sale Unstable LTA4H 53 41 CCCOc1ccc(CCC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217823966 FI For-Sale Unstable PLA2G4A 19 42 CCCOc1ccc(CCC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217823966 FI For-Sale Unstable PLA2G4B 46 37 CC[C@@H](NC(=O)COc1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217823980 EG In-Stock Unstable PTGER3 35 46 CC[C@@H](NC(=O)COc1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217823980 EG In-Stock Unstable TACR3 41 38 CC[C@@H](NC(=O)COc1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217823980 EG In-Stock Unstable MTNR1B 34 40 CC[C@@H](NC(=O)COc1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217823980 EG In-Stock Unstable PLA2G4B 40 40 CC[C@@H](NC(=O)COc1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217823980 EG In-Stock Unstable PAM 0 43 CC[C@@H](NC(=O)COc1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217823980 EG In-Stock Unstable HCRTR2 23 40 CC[C@@H](NC(=O)COc1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217823980 EG In-Stock Unstable ENPP1 57 34 CC[C@@H](NC(=O)COc1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217823980 EG In-Stock Unstable PDS 67 38 CC[C@@H](NC(=O)COc1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217823980 EG In-Stock Unstable GPR88 0 41 CCCc1ccc(C[C@@H]2C[C@@H]2C(=O)O)cc1 ZINC000217823995 BF In-Stock Unstable GRIK2 22 46 O=c1c(-c2c3cn[nH]c3nc3c2oc2cc(O)ccc23)coc2ccccc12 ZINC000217824009 FI In-Stock Bother ALDH2 59 32 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)Cc1ccc(N)cc1 ZINC000217824022 CG For-Sale Unstable TRPM8 22 58 CCCOc1ccc(CCC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217824026 FI For-Sale Unstable LTA4H 53 41 CCCOc1ccc(CCC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217824026 FI For-Sale Unstable PLA2G4A 19 42 CCCOc1ccc(CCC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217824026 FI For-Sale Unstable PLA2G4B 46 37 CC[C@H](NC(=O)COc1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217824062 EG In-Stock Unstable PTGER3 35 46 CC[C@H](NC(=O)COc1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217824062 EG In-Stock Unstable TACR3 41 38 CC[C@H](NC(=O)COc1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217824062 EG In-Stock Unstable MTNR1B 34 40 CC[C@H](NC(=O)COc1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217824062 EG In-Stock Unstable PLA2G4B 40 40 CC[C@H](NC(=O)COc1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217824062 EG In-Stock Unstable PAM 0 43 CC[C@H](NC(=O)COc1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217824062 EG In-Stock Unstable HCRTR2 23 40 CC[C@H](NC(=O)COc1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217824062 EG In-Stock Unstable ENPP1 57 34 CC[C@H](NC(=O)COc1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217824062 EG In-Stock Unstable PDS 67 38 CC[C@H](NC(=O)COc1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217824062 EG In-Stock Unstable GPR88 0 41 CCCc1ccc(C[C@H]2C[C@@H]2C(=O)O)cc1 ZINC000217824081 BF In-Stock Unstable GRIK2 22 46 Cc1nn(Cc2cccc(/C=C\C(=O)O)c2)c(C)c1C ZINC000217824093 CF For-Sale Unstable PTGER2 0 41 Cc1nn(Cc2cccc(/C=C\C(=O)O)c2)c(C)c1C ZINC000217824093 CF For-Sale Unstable HDAC8 37 44 Cc1nn(Cc2cccc(/C=C\C(=O)O)c2)c(C)c1C ZINC000217824093 CF For-Sale Unstable HDAC6 23 44 O=C(CCc1cccc(Cl)c1)NC[C@H]1CCCN1c1ccccc1 ZINC000217824124 EI In-Stock Unstable SIGMAR1 16 45 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)CCCCCN ZINC000217824131 CG For-Sale Unstable TRPM8 19 66 CC[C@@H](NC(=O)COc1ccccc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217824156 EF In-Stock Unstable CTSF 47 34 CC[C@@H](NC(=O)COc1ccccc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217824156 EF In-Stock Unstable TACR3 45 38 CC[C@@H](NC(=O)COc1ccccc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217824156 EF In-Stock Unstable PDS 45 38 CC[C@@H](NC(=O)COc1ccccc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217824156 EF In-Stock Unstable GPR88 0 40 CCCc1ccc(C[C@@H]2C[C@H]2C(=O)O)cc1 ZINC000217824158 BF In-Stock Unstable GRIK2 22 46 COc1ccc(COC2CCCCC2)cc1/C=C\C(=O)O ZINC000217824174 CH For-Sale Unstable PTGER2 32 44 COc1ccc(COC2CCCCC2)cc1/C=C\C(=O)O ZINC000217824174 CH For-Sale Unstable PTGER4 0 44 COc1ccc(COC2CCCCC2)cc1/C=C\C(=O)O ZINC000217824174 CH For-Sale Unstable PTGER3 15 44 O=C(CCc1cccc(Cl)c1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217824202 EI In-Stock Unstable SIGMAR1 16 45 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)CCCCCN ZINC000217824218 CG For-Sale Unstable TRPM8 19 66 COc1cc(C(=O)N2CCC([C@@H](C)O)CC2)ccc1F ZINC000217824220 CE On-Demand Unstable L3MBTL3 66 38 COc1cc(C(=O)N2CCC([C@@H](C)O)CC2)ccc1F ZINC000217824220 CE On-Demand Unstable HPGD 43 40 CC[C@H](NC(=O)COc1ccccc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217824231 EF In-Stock Unstable CTSF 47 34 CC[C@H](NC(=O)COc1ccccc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217824231 EF In-Stock Unstable TACR3 45 38 CC[C@H](NC(=O)COc1ccccc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217824231 EF In-Stock Unstable PDS 45 38 CC[C@H](NC(=O)COc1ccccc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217824231 EF In-Stock Unstable GPR88 0 40 CCCc1ccc(C[C@H]2C[C@H]2C(=O)O)cc1 ZINC000217824244 BF In-Stock Unstable GRIK2 22 46 O=C(O)/C=C\c1ccc(COC2CCCCC2)c(F)c1 ZINC000217824257 CH For-Sale Unstable AKR1C3 28 40 COc1cc(C(=O)N2CCC([C@H](C)O)CC2)ccc1F ZINC000217824293 CE On-Demand Unstable L3MBTL3 66 38 COc1cc(C(=O)N2CCC([C@H](C)O)CC2)ccc1F ZINC000217824293 CE On-Demand Unstable HPGD 43 40 O=C(O)[C@H]1C[C@@H](O)CN1C(=O)[C@@H]1C[C@@H]2CCCC[C@@H]2N1 ZINC000217824295 CB For-Sale Unstable MME 20 51 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)CCCCCN ZINC000217824304 CG For-Sale Unstable TRPM8 19 66 COc1ccc(/C=C\C(=O)O)cc1COC1CCCC1 ZINC000217824324 CG For-Sale Unstable PTGER2 0 43 COc1ccc(/C=C\C(=O)O)cc1COC1CCCC1 ZINC000217824324 CG For-Sale Unstable AKR1C3 23 41 COc1ccc(-c2noc(CNC(=O)COc3ccccc3)n2)c(OC)c1 ZINC000217824353 FE In-Stock Unstable COLA 40 38 COc1ccc(-c2noc(CNC(=O)COc3ccccc3)n2)c(OC)c1 ZINC000217824353 FE In-Stock Unstable MTNR1A 67 39 COc1ccc(-c2noc(CNC(=O)COc3ccccc3)n2)c(OC)c1 ZINC000217824353 FE In-Stock Unstable MTNR1B 57 39 COc1ccc(-c2noc(CNC(=O)COc3ccccc3)n2)c(OC)c1 ZINC000217824353 FE In-Stock Unstable MT-CYB 44 32 O=C(O)[C@H]1C[C@H](O)CN1C(=O)[C@@H]1C[C@@H]2CCCC[C@@H]2N1 ZINC000217824372 CB For-Sale Unstable MME 20 51 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)CCCCCN ZINC000217824392 CG For-Sale Unstable TRPM8 19 66 Cc1cc(Cl)cc(C(=O)N2CCC([C@@H](C)O)CC2)c1 ZINC000217824396 CF On-Demand Unstable L3MBTL3 54 36 COc1ccc(COC2CCCC2)cc1/C=C\C(=O)O ZINC000217824408 CG For-Sale Unstable PTGER2 34 45 COc1ccc(COC2CCCC2)cc1/C=C\C(=O)O ZINC000217824408 CG For-Sale Unstable PTGER4 0 45 COc1ccc(COC2CCCC2)cc1/C=C\C(=O)O ZINC000217824408 CG For-Sale Unstable PTGER3 16 45 O=C(O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H]1C[C@@H]2CCCC[C@@H]2N1 ZINC000217824450 CB For-Sale Unstable MME 20 51 Cc1cc(Cl)cc(C(=O)N2CCC([C@H](C)O)CC2)c1 ZINC000217824473 CF On-Demand Unstable L3MBTL3 54 36 O=C(O)/C=C\c1ccccc1COCc1ccccc1 ZINC000217824481 CH For-Sale Unstable PTGER2 30 58 O=C(O)/C=C\c1ccccc1COCc1ccccc1 ZINC000217824481 CH For-Sale Unstable PTGER4 42 58 O=C(O)/C=C\c1ccccc1COCc1ccccc1 ZINC000217824481 CH For-Sale Unstable PTGER3 34 58 O=C(O)/C=C\c1ccccc1COCc1ccccc1 ZINC000217824481 CH For-Sale Unstable CAPN2 40 37 O=C(O)/C=C\c1ccccc1COCc1ccccc1 ZINC000217824481 CH For-Sale Unstable PTGDR 0 57 O=C(O)/C=C\c1ccccc1COCc1ccccc1 ZINC000217824481 CH For-Sale Unstable HCAR2 0 40 COc1cccc(-c2noc(CN(C)C(=O)COc3ccccc3)n2)c1 ZINC000217824483 FF In-Stock Unstable FABP4 46 35 O=C(CCc1ccc(Cl)cc1Cl)NC[C@H]1CCCN1c1ccccc1 ZINC000217824489 GJ For-Sale Unstable MC4R 50 38 O=C(CCc1ccc(Cl)cc1Cl)NC[C@H]1CCCN1c1ccccc1 ZINC000217824489 GJ For-Sale Unstable P2RX7 36 40 O=C(CCc1ccc(Cl)cc1Cl)NC[C@H]1CCCN1c1ccccc1 ZINC000217824489 GJ For-Sale Unstable MC5R 29 43 O=C(CCc1ccc(Cl)cc1Cl)NC[C@H]1CCCN1c1ccccc1 ZINC000217824489 GJ For-Sale Unstable EPHX2 15 41 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)C1(N)CCCCC1 ZINC000217824510 CG For-Sale Unstable TRPM8 18 48 O=C(O)[C@@H]1C[C@H](O)CN1C(=O)[C@@H]1C[C@@H]2CCCC[C@@H]2N1 ZINC000217824526 CB For-Sale Unstable MME 20 51 CC1(C)[C@H]2CC[C@@]1(CS(=O)(=O)N1CCC[C@H](Cc3nc(C4CC4)no3)C1)C(=O)C2 ZINC000217824534 HF In-Stock Unstable CA5B 23 40 CC1(C)[C@H]2CC[C@@]1(CS(=O)(=O)N1CCC[C@H](Cc3nc(C4CC4)no3)C1)C(=O)C2 ZINC000217824534 HF In-Stock Unstable CA5A 25 40 CC1(C)[C@H]2CC[C@@]1(CS(=O)(=O)N1CCC[C@H](Cc3nc(C4CC4)no3)C1)C(=O)C2 ZINC000217824534 HF In-Stock Unstable CXCR3 15 46 CN(Cc1nc2cc(Cl)ccc2[nH]1)C(=O)C1(C(N)=O)CC1 ZINC000217824543 DD In-Stock Unstable CHEK2 45 36 CN(Cc1nc2cc(Cl)ccc2[nH]1)C(=O)C1(C(N)=O)CC1 ZINC000217824543 DD In-Stock Unstable PIN1 16 42 O=C(O)/C=C\c1ccc(COCc2ccccc2)c(F)c1 ZINC000217824550 CH For-Sale Unstable PTGER2 44 45 O=C(O)/C=C\c1ccc(COCc2ccccc2)c(F)c1 ZINC000217824550 CH For-Sale Unstable PTGER4 0 43 O=C(O)/C=C\c1ccc(COCc2ccccc2)c(F)c1 ZINC000217824550 CH For-Sale Unstable PTGER3 17 43 O=C(O)/C=C\c1ccc(COCc2ccccc2)c(F)c1 ZINC000217824550 CH For-Sale Unstable PTGDR 0 40 O=C(O)/C=C\c1ccc(COCc2ccccc2)c(F)c1 ZINC000217824550 CH For-Sale Unstable AKR1C3 36 52 O=C(O)/C=C\c1ccc(COCc2ccccc2)c(F)c1 ZINC000217824550 CH For-Sale Unstable AKR1B10 15 44 O=C(CCc1ccc(Cl)cc1Cl)NC[C@@H]1CCCN1c1ccccc1 ZINC000217824567 GJ For-Sale Unstable MC4R 50 38 O=C(CCc1ccc(Cl)cc1Cl)NC[C@@H]1CCCN1c1ccccc1 ZINC000217824567 GJ For-Sale Unstable P2RX7 36 40 O=C(CCc1ccc(Cl)cc1Cl)NC[C@@H]1CCCN1c1ccccc1 ZINC000217824567 GJ For-Sale Unstable MC5R 29 43 O=C(CCc1ccc(Cl)cc1Cl)NC[C@@H]1CCCN1c1ccccc1 ZINC000217824567 GJ For-Sale Unstable EPHX2 15 41 COc1cc(NC(=O)N/C=C/c2ccccc2Cl)c(OC)cc1Cl ZINC000217824573 FJ For-Sale Unstable CYSP_PLAFA 40 36 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)C1(N)CCCCC1 ZINC000217824581 CG For-Sale Unstable TRPM8 18 48 COc1ccc(-c2noc(CN(C)C(=O)COc3ccccc3)n2)c(OC)c1 ZINC000217824610 GF In-Stock Unstable TSPO 45 38 Fc1ccc(CN2CCNCC2)c(Cl)c1F ZINC000217824644 BE For-Sale Unstable CXCR4 21 43 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)C1(N)CCCCC1 ZINC000217824647 CG For-Sale Unstable TRPM8 18 48 COc1ccc(/C=C\C(=O)O)cc1CN1CCC(O)CC1 ZINC000217824667 CD For-Sale Unstable SIGMAR1 16 42 COc1ccc(/C=C\C(=O)O)cc1CN1CCC(O)CC1 ZINC000217824667 CD For-Sale Unstable CCR2 0 46 COc1ccc(/C=C\C(=O)O)cc1CN1CCC(O)CC1 ZINC000217824667 CD For-Sale Unstable AKR1C3 21 41 CC(C)c1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217824727 DH In-Stock Unstable ALOX5 19 41 CC(C)c1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217824727 DH In-Stock Unstable ANPEP 21 44 CC(C)c1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217824727 DH In-Stock Unstable SDH1 0 42 CC(C)c1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217824727 DH In-Stock Unstable FDFT1 18 45 CC(C)c1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217824727 DH In-Stock Unstable PTGER3 52 38 CC(C)c1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217824727 DH In-Stock Unstable SCN2A 25 40 CC(C)c1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217824727 DH In-Stock Unstable HDAC8 15 45 CC(C)c1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217824727 DH In-Stock Unstable MTNR1A 36 40 CC(C)c1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217824727 DH In-Stock Unstable MTNR1B 43 40 CC(C)c1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217824727 DH In-Stock Unstable PLA2G4B 51 39 CC(C)c1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217824727 DH In-Stock Unstable FAAH 45 42 CC(C)c1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217824727 DH In-Stock Unstable CASP1 20 41 CC(C)c1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217824727 DH In-Stock Unstable PLM2_PLAFA 30 40 CC(C)c1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217824727 DH In-Stock Unstable AMP1_PLAFQ 37 44 CC(C)c1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217824727 DH In-Stock Unstable FFAR1 42 37 CC(C)c1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217824727 DH In-Stock Unstable CRTM 68 48 CC(C)c1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217824727 DH In-Stock Unstable ACAT 0 46 CC(C)c1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217824727 DH In-Stock Unstable BLAIMP-1 0 43 CC(C)c1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217824727 DH In-Stock Unstable PDS 50 40 CC(C)c1ccc(CCCNC(=O)COc2ccccc2)cc1 ZINC000217824727 DH In-Stock Unstable CES1D 45 34 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)C1(N)CCCCC1 ZINC000217824733 CG For-Sale Unstable TRPM8 18 48 Fc1ccc(Cl)c(F)c1CN1CCNCC1 ZINC000217824743 BE For-Sale Unstable CXCR4 21 43 COc1ccc(CN2CCC(O)CC2)cc1/C=C\C(=O)O ZINC000217824793 CD For-Sale Unstable DRD2 23 41 COc1ccc(CN2CCC(O)CC2)cc1/C=C\C(=O)O ZINC000217824793 CD For-Sale Unstable DRD4 42 41 COc1ccc(CN2CCC(O)CC2)cc1/C=C\C(=O)O ZINC000217824793 CD For-Sale Unstable ACHE 30 44 COc1ccc(CN2CCC(O)CC2)cc1/C=C\C(=O)O ZINC000217824793 CD For-Sale Unstable HRH1 21 43 COc1ccc(CN2CCC(O)CC2)cc1/C=C\C(=O)O ZINC000217824793 CD For-Sale Unstable DRD3 25 40 COc1ccc(CN2CCC(O)CC2)cc1/C=C\C(=O)O ZINC000217824793 CD For-Sale Unstable PTGER2 29 42 COc1ccc(CN2CCC(O)CC2)cc1/C=C\C(=O)O ZINC000217824793 CD For-Sale Unstable PTGER4 17 42 COc1ccc(CN2CCC(O)CC2)cc1/C=C\C(=O)O ZINC000217824793 CD For-Sale Unstable SIGMAR1 39 47 COc1ccc(CN2CCC(O)CC2)cc1/C=C\C(=O)O ZINC000217824793 CD For-Sale Unstable PTGER3 15 42 COc1ccc(CN2CCC(O)CC2)cc1/C=C\C(=O)O ZINC000217824793 CD For-Sale Unstable SSTR5 68 40 COc1ccc(CN2CCC(O)CC2)cc1/C=C\C(=O)O ZINC000217824793 CD For-Sale Unstable CCR3 20 41 COc1ccc(CN2CCC(O)CC2)cc1/C=C\C(=O)O ZINC000217824793 CD For-Sale Unstable MCHR1 33 45 COc1ccc(CN2CCC(O)CC2)cc1/C=C\C(=O)O ZINC000217824793 CD For-Sale Unstable CACNA1G 16 41 COc1ccc(CN2CCC(O)CC2)cc1/C=C\C(=O)O ZINC000217824793 CD For-Sale Unstable CCR8 21 42 Cc1cccc(N2CCN(C(=O)N/C=C/c3ccccc3Cl)CC2)c1C ZINC000217824794 FI For-Sale Unstable HTR2A 30 42 Cc1cccc(N2CCN(C(=O)N/C=C/c3ccccc3Cl)CC2)c1C ZINC000217824794 FI For-Sale Unstable HTR2C 33 42 Cc1cccc(N2CCN(C(=O)N/C=C/c3ccccc3Cl)CC2)c1C ZINC000217824794 FI For-Sale Unstable SLC6A4 15 42 CCOC(=O)CC(=O)COc1ccc([C@@H](C)CC)cc1 ZINC000217824812 CG For-Sale Unstable PLA2G4B 78 35 C/C(=C/c1ccccc1)C(=O)CCl ZINC000217824822 AF For-Sale Unstable TLR4 33 45 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)CCN ZINC000217824837 BD For-Sale Unstable TRPM8 0 61 O=C(CCc1ccc(Cl)c(Cl)c1)NC[C@H]1CCCN1c1ccccc1 ZINC000217824854 GJ For-Sale Unstable OPRK1 22 41 O=C(CCc1ccc(Cl)c(Cl)c1)NC[C@H]1CCCN1c1ccccc1 ZINC000217824854 GJ For-Sale Unstable SIGMAR1 22 44 O=C(CCc1ccc(Cl)c(Cl)c1)NC[C@H]1CCCN1c1ccccc1 ZINC000217824854 GJ For-Sale Unstable CCR3 26 41 O=C(COc1ccccc1)NCCCN1CCCc2ccccc21 ZINC000217824863 DG In-Stock Unstable CYSLTR2 48 32 O=C(COc1ccccc1)NCCCN1CCCc2ccccc21 ZINC000217824863 DG In-Stock Unstable MTNR1C 0 40 COc1ccc(N2CCN(c3ccc(NC(C)=O)cc3)CC2)cc1 ZINC000217824872 EF For-Sale Unstable GYRB 27 47 COc1ccc(N2CCN(c3ccc(NC(C)=O)cc3)CC2)cc1 ZINC000217824872 EF For-Sale Unstable HTR1A 17 54 COc1ccc(N2CCN(c3ccc(NC(C)=O)cc3)CC2)cc1 ZINC000217824872 EF For-Sale Unstable TSHR 41 31 COc1ccc(N2CCN(c3ccc(NC(C)=O)cc3)CC2)cc1 ZINC000217824872 EF For-Sale Unstable DRD4 46 39 COc1ccc(N2CCN(c3ccc(NC(C)=O)cc3)CC2)cc1 ZINC000217824872 EF For-Sale Unstable HTR1B 18 44 COc1ccc(N2CCN(c3ccc(NC(C)=O)cc3)CC2)cc1 ZINC000217824872 EF For-Sale Unstable F10 21 51 COc1ccc(N2CCN(c3ccc(NC(C)=O)cc3)CC2)cc1 ZINC000217824872 EF For-Sale Unstable PDGFRB 40 38 COc1ccc(N2CCN(c3ccc(NC(C)=O)cc3)CC2)cc1 ZINC000217824872 EF For-Sale Unstable CA1 18 44 COc1ccc(N2CCN(c3ccc(NC(C)=O)cc3)CC2)cc1 ZINC000217824872 EF For-Sale Unstable MMP13 29 40 COc1ccc(N2CCN(c3ccc(NC(C)=O)cc3)CC2)cc1 ZINC000217824872 EF For-Sale Unstable PRNP 55 44 COc1ccc(N2CCN(c3ccc(NC(C)=O)cc3)CC2)cc1 ZINC000217824872 EF For-Sale Unstable JAK2 17 45 COc1ccc(N2CCN(c3ccc(NC(C)=O)cc3)CC2)cc1 ZINC000217824872 EF For-Sale Unstable MAPK1 16 42 COc1ccc(N2CCN(c3ccc(NC(C)=O)cc3)CC2)cc1 ZINC000217824872 EF For-Sale Unstable MTNR1A 44 51 COc1ccc(N2CCN(c3ccc(NC(C)=O)cc3)CC2)cc1 ZINC000217824872 EF For-Sale Unstable MTNR1B 47 51 COc1ccc(N2CCN(c3ccc(NC(C)=O)cc3)CC2)cc1 ZINC000217824872 EF For-Sale Unstable MMP2 18 45 COc1ccc(N2CCN(c3ccc(NC(C)=O)cc3)CC2)cc1 ZINC000217824872 EF For-Sale Unstable MMP3 25 40 COc1ccc(N2CCN(c3ccc(NC(C)=O)cc3)CC2)cc1 ZINC000217824872 EF For-Sale Unstable GALR2 40 34 COc1ccc(N2CCN(c3ccc(NC(C)=O)cc3)CC2)cc1 ZINC000217824872 EF For-Sale Unstable MMP9 27 45 COc1ccc(N2CCN(c3ccc(NC(C)=O)cc3)CC2)cc1 ZINC000217824872 EF For-Sale Unstable EPHX2 23 48 COc1ccc(N2CCN(c3ccc(NC(C)=O)cc3)CC2)cc1 ZINC000217824872 EF For-Sale Unstable ACR 51 44 COc1ccc(N2CCN(c3ccc(NC(C)=O)cc3)CC2)cc1 ZINC000217824872 EF For-Sale Unstable CA12 15 40 COc1ccc(N2CCN(c3ccc(NC(C)=O)cc3)CC2)cc1 ZINC000217824872 EF For-Sale Unstable CA9 17 40 COc1ccc(N2CCN(c3ccc(NC(C)=O)cc3)CC2)cc1 ZINC000217824872 EF For-Sale Unstable AKR1C3 28 41 COc1ccc(N2CCN(c3ccc(NC(C)=O)cc3)CC2)cc1 ZINC000217824872 EF For-Sale Unstable IDO1 22 51 COc1ccc(N2CCN(c3ccc(NC(C)=O)cc3)CC2)cc1 ZINC000217824872 EF For-Sale Unstable AKR1C2 50 41 COc1ccc(N2CCN(c3ccc(NC(C)=O)cc3)CC2)cc1 ZINC000217824872 EF For-Sale Unstable NOD2 17 40 COc1cc(O)c(C(C)(C)O)c(Cl)c1OC ZINC000217824877 BE For-Sale Unstable TUBB1 43 38 CCOC(=O)CC(=O)COc1ccc([C@H](C)CC)cc1 ZINC000217824899 CG For-Sale Unstable PLA2G4B 78 35 O=C(N/C=C/c1ccccc1Cl)N1CCN(c2ccccc2)CC1 ZINC000217824901 EH For-Sale Unstable AKR1C3 0 43 O=C(O)/C=C\c1ccc(CN2CCC(O)CC2)c(F)c1 ZINC000217824906 CD For-Sale Unstable SIGMAR1 17 40 O=C(O)/C=C\c1ccc(CN2CCC(O)CC2)c(F)c1 ZINC000217824906 CD For-Sale Unstable GPR183 0 40 CCC[C@@H](N)C(=O)N1C[C@H](C)O[C@@H](C)C1 ZINC000217824917 BC For-Sale Unstable DPP7 46 36 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)CCN ZINC000217824920 BD For-Sale Unstable TRPM8 0 61 O=C(NCc1ccccc1)OC[C@@H]1CCNC1 ZINC000217824934 BD For-Sale Unstable SLC6A2 0 42 O=C(NCc1ccccc1)OC[C@@H]1CCNC1 ZINC000217824934 BD For-Sale Unstable PDS 44 38 O=C(CCc1ccc(Cl)c(Cl)c1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217824935 GJ For-Sale Unstable OPRK1 22 41 O=C(CCc1ccc(Cl)c(Cl)c1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217824935 GJ For-Sale Unstable SIGMAR1 22 44 O=C(CCc1ccc(Cl)c(Cl)c1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217824935 GJ For-Sale Unstable CCR3 26 41 CCOc1ccc(CNC(=O)COc2ccccc2C)cc1OCC ZINC000217824985 EG In-Stock Unstable CETP 0 40 CCOc1ccc(CNC(=O)COc2ccccc2C)cc1OCC ZINC000217824985 EG In-Stock Unstable PDS 40 32 CCC[C@H](N)C(=O)N1C[C@H](C)O[C@@H](C)C1 ZINC000217824999 BC On-Demand Unstable DPP7 42 33 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)CCN ZINC000217825004 BD For-Sale Unstable TRPM8 0 61 CN1CCCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217825005 CD For-Sale Unstable SLC6A1 49 38 CN1CCCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217825005 CD For-Sale Unstable PTGER2 42 45 CN1CCCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217825005 CD For-Sale Unstable PTGER4 0 45 CN1CCCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217825005 CD For-Sale Unstable PTGER3 18 45 COc1ccc(CCC(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217825047 FG For-Sale Unstable HTR1A 15 41 COc1ccc(CCC(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217825047 FG For-Sale Unstable FKBP1A 18 40 COc1ccc(CCC(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217825047 FG For-Sale Unstable MTNR1A 74 39 COc1ccc(CCC(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217825047 FG For-Sale Unstable MTNR1B 72 39 COc1ccc(CCC(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217825047 FG For-Sale Unstable ACKR3 63 34 COc1ccc(CNC(=O)CCCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@H]23)cc1 ZINC000217825076 JH In-Stock Unstable HTR7 32 44 COc1ccc(CNC(=O)CCCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@H]23)cc1 ZINC000217825076 JH In-Stock Unstable SCN9A 0 51 COc1cc(CNC(=O)COc2ccccc2C)ccc1OC(C)C ZINC000217825080 EG In-Stock Unstable TRPV1 26 41 COc1cc(CNC(=O)COc2ccccc2C)ccc1OC(C)C ZINC000217825080 EG In-Stock Unstable DRTS_TRYCR 44 30 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)CCN ZINC000217825084 BD For-Sale Unstable TRPM8 0 61 Cc1cccc(C)c1NC(=O)N/C=C/c1ccccc1Cl ZINC000217825114 DJ For-Sale Unstable CXCL8 23 42 Cc1cccc(C)c1NC(=O)N/C=C/c1ccccc1Cl ZINC000217825114 DJ For-Sale Unstable ACAT 0 43 COc1ccc(CCC(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217825123 FG For-Sale Unstable HTR1A 15 41 COc1ccc(CCC(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217825123 FG For-Sale Unstable FKBP1A 18 40 COc1ccc(CCC(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217825123 FG For-Sale Unstable MTNR1A 74 39 COc1ccc(CCC(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217825123 FG For-Sale Unstable MTNR1B 72 39 COc1ccc(CCC(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217825123 FG For-Sale Unstable ACKR3 63 34 Cc1[nH]c(=O)[nH]c(=O)c1CC(=O)NCc1cc2cc(F)ccc2[nH]1 ZINC000217825132 EC In-Stock Unstable P2RX7 49 44 CN1CCCN(Cc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217825137 CD For-Sale Unstable HRH3 17 44 CN1CCCN(Cc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217825137 CD For-Sale Unstable SIGMAR1 30 44 COc1ccc(CNC(=O)CCCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@@H]23)cc1 ZINC000217825172 JH In-Stock Unstable HTR7 32 44 COc1ccc(CNC(=O)CCCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@@H]23)cc1 ZINC000217825172 JH In-Stock Unstable SCN9A 0 51 Cc1ccc(C(=O)N[C@H]2C[C@H](C)CC[C@H]2C(C)C)cc1N ZINC000217825173 CH For-Sale Unstable TRPM8 23 72 CC1(C)[C@H]2CC[C@@]1(C)[C@@H](OC(=O)CS(C)(=O)=O)C2 ZINC000217825197 CD For-Sale Unstable ELANE 17 47 Cc1ccccc1OCC(=O)NCCCc1ccccc1Cl ZINC000217825214 DH In-Stock Unstable CXCL8 44 37 Cc1ccccc1OCC(=O)NCCCc1ccccc1Cl ZINC000217825214 DH In-Stock Unstable P2RX7 16 41 Cc1ccccc1OCC(=O)NCCCc1ccccc1Cl ZINC000217825214 DH In-Stock Unstable CYSP_TRYCR 0 50 Cc1ccccc1OCC(=O)NCCCc1ccccc1Cl ZINC000217825214 DH In-Stock Unstable CETP 0 42 Cc1ccccc1OCC(=O)NCCCc1ccccc1Cl ZINC000217825214 DH In-Stock Unstable MTNR1B 43 37 COc1ccc([N+](=O)[O-])cc1NC(=O)N/C=C/c1ccccc1Cl ZINC000217825216 EI For-Sale Unstable PYGL 16 44 COc1ccc([N+](=O)[O-])cc1NC(=O)N/C=C/c1ccccc1Cl ZINC000217825216 EI For-Sale Unstable KCNMA1 28 54 CCOc1ccccc1CCC(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217825232 FH For-Sale Unstable MBTPS1 40 35 CCOc1ccccc1CCC(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217825232 FH For-Sale Unstable HCN1 45 35 CCOc1ccccc1CCC(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217825232 FH For-Sale Unstable HCN4 45 35 CC(=O)N[C@@H](CC(=O)N(C)Cc1c(C)nc2sc(C)cn12)c1ccc(Cl)cc1 ZINC000217825233 HH On-Demand Unstable UTS2 41 32 Cc1ccc(C(=O)N[C@H]2C[C@@H](C)CC[C@H]2C(C)C)cc1N ZINC000217825245 CH For-Sale Unstable TRPM8 23 72 COc1cc([C@H](C)N2CCO[C@@H]3CCCC[C@@H]32)ccc1O ZINC000217825285 CG For-Sale Unstable PNLIP 0 42 COc1cc([C@H](C)N2CCO[C@@H]3CCCC[C@@H]32)ccc1O ZINC000217825285 CG For-Sale Unstable SLC22A3 0 40 CC[C@@H](CCO)NC[C@@H](O)c1ccccc1 ZINC000217825293 BD On-Demand Unstable ADRB1 0 40 CC[C@@H](CCO)NC[C@@H](O)c1ccccc1 ZINC000217825293 BD On-Demand Unstable ADRB3 0 41 CC(=O)N[C@H](CC(=O)N(C)Cc1c(C)nc2sc(C)cn12)c1ccc(Cl)cc1 ZINC000217825299 HH On-Demand Unstable UTS2 41 32 CCOc1ccccc1CCC(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217825310 FH For-Sale Unstable MBTPS1 40 35 CCOc1ccccc1CCC(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217825310 FH For-Sale Unstable HCN1 45 35 CCOc1ccccc1CCC(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217825310 FH For-Sale Unstable HCN4 45 35 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)[C@@H](N)c1ccccc1 ZINC000217825330 CG For-Sale Unstable TRPM8 21 61 Cc1ccccc1OCC(=O)NCCCc1ccc(Cl)cc1 ZINC000217825338 DH In-Stock Unstable CYSP_TRYCR 0 50 Cc1ccccc1OCC(=O)NCCCc1ccc(Cl)cc1 ZINC000217825338 DH In-Stock Unstable CETP 0 43 Cc1ccccc1OCC(=O)NCCCc1ccc(Cl)cc1 ZINC000217825338 DH In-Stock Unstable MTNR1A 19 41 Cc1ccccc1OCC(=O)NCCCc1ccc(Cl)cc1 ZINC000217825338 DH In-Stock Unstable MTNR1B 24 42 Cc1ccccc1OCC(=O)NCCCc1ccc(Cl)cc1 ZINC000217825338 DH In-Stock Unstable SCN5A 0 40 Cc1ccccc1OCC(=O)NCCCc1ccc(Cl)cc1 ZINC000217825338 DH In-Stock Unstable CRTM 46 44 CCNc1nc(C)c(C(=O)N(C)Cc2cc(-c3ccccc3)on2)s1 ZINC000217825345 FH In-Stock Unstable TSPO 16 43 O=C(O)[C@@H]1C[C@@H]1Cc1cccnc1 ZINC000217825364 AD In-Stock Unstable NPY2R 42 34 O=C(O)[C@@H]1C[C@@H]1Cc1cccnc1 ZINC000217825364 AD In-Stock Unstable CHRNA7 39 42 O=C(O)[C@@H]1C[C@@H]1Cc1cccnc1 ZINC000217825364 AD In-Stock Unstable ACHP_LYMST 23 43 CC[C@H](CCO)NC[C@@H](O)c1ccccc1 ZINC000217825372 BD On-Demand Unstable ADRB1 0 40 CC[C@H](CCO)NC[C@@H](O)c1ccccc1 ZINC000217825372 BD On-Demand Unstable ADRB3 0 41 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)[C@@H](N)c1ccccc1 ZINC000217825391 CG For-Sale Unstable TRPM8 21 61 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)c3ccno3)C2)n1 ZINC000217825392 FG In-Stock Unstable HRH3 16 40 C[C@@H](c1cccc(Cl)c1)N(C)C[C@@](C)(O)c1ccccc1 ZINC000217825414 DI For-Sale Unstable AOC3 18 40 C[C@@H](c1cccc(Cl)c1)N(C)C[C@@](C)(O)c1ccccc1 ZINC000217825414 DI For-Sale Unstable VIPR1 38 40 CC(C)[C@H](NNC(=O)OC(C)(C)C)C(=O)O ZINC000217825422 BD For-Sale Unstable PGA5 44 39 Cc1ccccc1OCC(=O)NCCCc1ccc(F)cc1 ZINC000217825449 DG In-Stock Unstable CYSP_TRYCR 0 54 Cc1ccccc1OCC(=O)NCCCc1ccc(F)cc1 ZINC000217825449 DG In-Stock Unstable MTNR1B 27 40 Cc1ccccc1OCC(=O)NCCCc1ccc(F)cc1 ZINC000217825449 DG In-Stock Unstable LEF 51 40 Cc1ccccc1OCC(=O)NCCCc1ccc(F)cc1 ZINC000217825449 DG In-Stock Unstable CRTM 44 45 O=C(O)[C@H]1C[C@@H]1Cc1cccnc1 ZINC000217825450 AD In-Stock Unstable NPY2R 42 34 O=C(O)[C@H]1C[C@@H]1Cc1cccnc1 ZINC000217825450 AD In-Stock Unstable CHRNA7 39 42 O=C(O)[C@H]1C[C@@H]1Cc1cccnc1 ZINC000217825450 AD In-Stock Unstable ACHP_LYMST 23 43 CC[C@@H](CCO)NC[C@H](O)c1ccccc1 ZINC000217825451 BD On-Demand Unstable ADRB1 0 40 CC[C@@H](CCO)NC[C@H](O)c1ccccc1 ZINC000217825451 BD On-Demand Unstable ADRB3 0 41 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)c3ccno3)C2)n1 ZINC000217825472 FG In-Stock Unstable HRH3 16 40 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)[C@@H](N)c1ccccc1 ZINC000217825476 CG For-Sale Unstable TRPM8 21 61 CC(C)[C@@H](CO)NC(=O)[C@H](Cc1ccccc1)N1Cc2ccccc2C1=O ZINC000217825487 FE In-Stock Unstable MME 54 39 CC(C)[C@@H](CO)NC(=O)[C@H](Cc1ccccc1)N1Cc2ccccc2C1=O ZINC000217825487 FE In-Stock Unstable CAPN1 23 41 CC(C)[C@@H](CO)NC(=O)[C@H](Cc1ccccc1)N1Cc2ccccc2C1=O ZINC000217825487 FE In-Stock Unstable POL 0 41 CC(C)[C@@H](CO)NC(=O)[C@H](Cc1ccccc1)N1Cc2ccccc2C1=O ZINC000217825487 FE In-Stock Unstable DERP1 0 48 C[C@H](c1cccc(Cl)c1)N(C)C[C@@](C)(O)c1ccccc1 ZINC000217825514 DI For-Sale Unstable AOC3 18 40 C[C@H](c1cccc(Cl)c1)N(C)C[C@@](C)(O)c1ccccc1 ZINC000217825514 DI For-Sale Unstable VIPR1 38 40 CC[C@H](CCO)NC[C@H](O)c1ccccc1 ZINC000217825529 BD On-Demand Unstable ADRB1 0 40 CC[C@H](CCO)NC[C@H](O)c1ccccc1 ZINC000217825529 BD On-Demand Unstable ADRB3 0 41 O=C(O)[C@@H]1C[C@H]1Cc1cccnc1 ZINC000217825540 AD In-Stock Unstable NPY2R 42 34 O=C(O)[C@@H]1C[C@H]1Cc1cccnc1 ZINC000217825540 AD In-Stock Unstable CHRNA7 39 42 O=C(O)[C@@H]1C[C@H]1Cc1cccnc1 ZINC000217825540 AD In-Stock Unstable ACHP_LYMST 23 43 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)[C@@H](N)c1ccccc1 ZINC000217825552 CG For-Sale Unstable TRPM8 21 61 COc1ccccc1CCCNC(=O)COc1ccccc1C ZINC000217825555 DG In-Stock Unstable ADRA1D 15 40 COc1ccccc1CCCNC(=O)COc1ccccc1C ZINC000217825555 DG In-Stock Unstable CYSP_TRYCR 0 51 COc1ccccc1CCCNC(=O)COc1ccccc1C ZINC000217825555 DG In-Stock Unstable CETP 0 40 COc1ccccc1CCCNC(=O)COc1ccccc1C ZINC000217825555 DG In-Stock Unstable MTNR1A 60 43 COc1ccccc1CCCNC(=O)COc1ccccc1C ZINC000217825555 DG In-Stock Unstable MTNR1B 52 48 COc1ccccc1CCCNC(=O)COc1ccccc1C ZINC000217825555 DG In-Stock Unstable MBTPS1 41 33 COc1ccccc1CCCNC(=O)COc1ccccc1C ZINC000217825555 DG In-Stock Unstable MT-CYB 21 41 C[C@@H](O)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)O ZINC000217825558 CC For-Sale Unstable MME 42 46 C[C@@H](O)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)O ZINC000217825558 CC For-Sale Unstable ANPEP 50 35 C[C@@H](O)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)O ZINC000217825558 CC For-Sale Unstable PGA 49 38 C[C@@H](O)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)O ZINC000217825558 CC For-Sale Unstable POL 0 40 CS(=O)(=O)c1ccc(CNCc2ccc(O)c(F)c2)cc1 ZINC000217825574 DE On-Demand Unstable CA2 21 49 CS(=O)(=O)c1ccc(CNCc2ccc(O)c(F)c2)cc1 ZINC000217825574 DE On-Demand Unstable PTGS2 35 40 CS(=O)(=O)c1ccc(CNCc2ccc(O)c(F)c2)cc1 ZINC000217825574 DE On-Demand Unstable CA1 20 40 CS(=O)(=O)c1ccc(CNCc2ccc(O)c(F)c2)cc1 ZINC000217825574 DE On-Demand Unstable TRPV1 20 46 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217825599 ID In-Stock Unstable HTR1D 22 40 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217825599 ID In-Stock Unstable HTR1B 16 40 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217825599 ID In-Stock Unstable SSTR2 40 38 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217825599 ID In-Stock Unstable OPRM1 15 40 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217825599 ID In-Stock Unstable MME 27 40 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217825599 ID In-Stock Unstable EDNRA 38 40 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217825599 ID In-Stock Unstable TACR1 35 44 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217825599 ID In-Stock Unstable MC4R 44 37 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217825599 ID In-Stock Unstable TACR2 25 44 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217825599 ID In-Stock Unstable CCKAR 89 46 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217825599 ID In-Stock Unstable BRS3 27 44 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217825599 ID In-Stock Unstable MC3R 67 37 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217825599 ID In-Stock Unstable MC5R 58 35 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217825599 ID In-Stock Unstable GRPR 47 33 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217825599 ID In-Stock Unstable ECE1 51 41 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217825599 ID In-Stock Unstable HDAC2 15 41 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217825599 ID In-Stock Unstable HDAC3 15 41 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217825599 ID In-Stock Unstable SSTR3 52 38 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217825599 ID In-Stock Unstable MMP11 96 36 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217825599 ID In-Stock Unstable CCKBR 74 46 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217825599 ID In-Stock Unstable GHSR 69 40 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217825599 ID In-Stock Unstable MC1R 86 37 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217825599 ID In-Stock Unstable SLC15A2 0 40 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217825599 ID In-Stock Unstable KISS1R 68 33 COc1ccc(CCC(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1OC ZINC000217825607 GG For-Sale Unstable DRD2 38 41 COc1ccc(CCC(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1OC ZINC000217825607 GG For-Sale Unstable ACKR3 65 35 O=C(O)[C@H]1C[C@H]1Cc1cccnc1 ZINC000217825620 AD In-Stock Unstable NPY2R 42 34 O=C(O)[C@H]1C[C@H]1Cc1cccnc1 ZINC000217825620 AD In-Stock Unstable CHRNA7 39 42 O=C(O)[C@H]1C[C@H]1Cc1cccnc1 ZINC000217825620 AD In-Stock Unstable ACHP_LYMST 23 43 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)CCCCCCN ZINC000217825637 CG For-Sale Unstable TRPM8 0 66 C[C@H](O)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)O ZINC000217825651 CC For-Sale Unstable MME 42 46 C[C@H](O)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)O ZINC000217825651 CC For-Sale Unstable ANPEP 50 35 C[C@H](O)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)O ZINC000217825651 CC For-Sale Unstable PGA 49 38 C[C@H](O)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)O ZINC000217825651 CC For-Sale Unstable POL 0 40 COc1ccc(CCCNC(=O)COc2ccccc2C)cc1 ZINC000217825659 DG In-Stock Unstable BMP1 27 40 COc1ccc(CCCNC(=O)COc2ccccc2C)cc1 ZINC000217825659 DG In-Stock Unstable CYSP_TRYCR 0 52 COc1ccc(CCCNC(=O)COc2ccccc2C)cc1 ZINC000217825659 DG In-Stock Unstable CETP 0 40 COc1ccc(CCCNC(=O)COc2ccccc2C)cc1 ZINC000217825659 DG In-Stock Unstable SCN2A 19 45 COc1ccc(CCCNC(=O)COc2ccccc2C)cc1 ZINC000217825659 DG In-Stock Unstable HDAC8 15 46 COc1ccc(CCCNC(=O)COc2ccccc2C)cc1 ZINC000217825659 DG In-Stock Unstable MTNR1A 86 47 COc1ccc(CCCNC(=O)COc2ccccc2C)cc1 ZINC000217825659 DG In-Stock Unstable MTNR1B 67 47 COc1ccc(CCCNC(=O)COc2ccccc2C)cc1 ZINC000217825659 DG In-Stock Unstable FAAH 26 41 COc1ccc(CCCNC(=O)COc2ccccc2C)cc1 ZINC000217825659 DG In-Stock Unstable ABCB1 20 40 COc1ccc(CCCNC(=O)COc2ccccc2C)cc1 ZINC000217825659 DG In-Stock Unstable CA9 18 44 COc1ccc(CCCNC(=O)COc2ccccc2C)cc1 ZINC000217825659 DG In-Stock Unstable CRTM 46 43 COc1ccc(CCC(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1OC ZINC000217825686 GG For-Sale Unstable DRD2 38 41 COc1ccc(CCC(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1OC ZINC000217825686 GG For-Sale Unstable ACKR3 65 35 CCCN(Cc1ccc(F)c(/C=C\C(=O)O)c1)C1CC1 ZINC000217825688 CG For-Sale Unstable HTR1A 0 41 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)CCCCCCN ZINC000217825724 CG For-Sale Unstable TRPM8 19 66 C[C@H](O)[C@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)O ZINC000217825741 CC For-Sale Unstable MME 42 46 C[C@H](O)[C@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)O ZINC000217825741 CC For-Sale Unstable ANPEP 50 35 C[C@H](O)[C@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)O ZINC000217825741 CC For-Sale Unstable PGA 49 38 C[C@H](O)[C@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)O ZINC000217825741 CC For-Sale Unstable POL 0 40 COc1ccc(OC[C@@H](C)NC(=O)COc2ccccc2C)cc1 ZINC000217825774 EF In-Stock Unstable ADRB2 15 40 COc1ccc(OC[C@@H](C)NC(=O)COc2ccccc2C)cc1 ZINC000217825774 EF In-Stock Unstable SDH1 0 41 COc1ccc(OC[C@@H](C)NC(=O)COc2ccccc2C)cc1 ZINC000217825774 EF In-Stock Unstable CAPN2 25 40 Cc1ccnc2ccc(C(=O)NC[C@@H]3CCCN3c3ccccc3)cc12 ZINC000217825807 EH For-Sale Unstable MAPK14 19 40 Cc1ccnc2ccc(C(=O)NC[C@@H]3CCCN3c3ccccc3)cc12 ZINC000217825807 EH For-Sale Unstable PREP 23 42 Cc1ccnc2ccc(C(=O)NC[C@@H]3CCCN3c3ccccc3)cc12 ZINC000217825807 EH For-Sale Unstable ACKR3 52 33 CCCCCN(C)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217825810 CG For-Sale Unstable ACHE 0 43 CCCCCN(C)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217825810 CG For-Sale Unstable AKR1C3 29 44 O=c1cc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)oc(CN2CCN(c3ccc(Cl)cc3)CC2)c1O ZINC000217825818 KG In-Stock Unstable CHRNA4 28 48 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)CCCCCCN ZINC000217825821 CG For-Sale Unstable TRPM8 19 66 CC(C)(C)OC(=O)NCCNCc1ccc(O)c(F)c1 ZINC000217825822 CE On-Demand Unstable TRPV1 18 50 CC(C)(C)OC(=O)NCCNCc1ccc(O)c(F)c1 ZINC000217825822 CE On-Demand Unstable LEF 63 37 COc1ccc(OC[C@H](C)NC(=O)COc2ccccc2C)cc1 ZINC000217825848 EF In-Stock Unstable ADRB2 15 40 COc1ccc(OC[C@H](C)NC(=O)COc2ccccc2C)cc1 ZINC000217825848 EF In-Stock Unstable SDH1 0 41 COc1ccc(OC[C@H](C)NC(=O)COc2ccccc2C)cc1 ZINC000217825848 EF In-Stock Unstable CAPN2 25 40 Cc1ccnc2ccc(C(=O)NC[C@H]3CCCN3c3ccccc3)cc12 ZINC000217825876 EH For-Sale Unstable MAPK14 19 40 Cc1ccnc2ccc(C(=O)NC[C@H]3CCCN3c3ccccc3)cc12 ZINC000217825876 EH For-Sale Unstable PREP 23 42 Cc1ccnc2ccc(C(=O)NC[C@H]3CCCN3c3ccccc3)cc12 ZINC000217825876 EH For-Sale Unstable ACKR3 52 33 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)CCCCCCN ZINC000217825885 CG For-Sale Unstable TRPM8 19 66 CN(C)CCN(C(=O)c1ccc(=O)[nH]n1)C1CCCC1 ZINC000217825909 CC On-Demand Unstable ACE 41 34 CCCCCN(C)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217825918 CG For-Sale Unstable THRA 43 41 CCCCCN(C)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217825918 CG For-Sale Unstable ACHE 0 42 CCCCCN(C)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217825918 CG For-Sale Unstable PTGER2 29 42 CCCCCN(C)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217825918 CG For-Sale Unstable PTGER4 0 42 CCCCCN(C)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217825918 CG For-Sale Unstable THRB 24 41 C[C@@H](O)[C@@H](NC(=O)[C@@H](N)CCS(C)(=O)=O)C(=O)O ZINC000217825938 CA For-Sale Unstable ENPEP 74 42 C[C@@H](O)[C@@H](NC(=O)[C@@H](N)CCS(C)(=O)=O)C(=O)O ZINC000217825938 CA For-Sale Unstable DLG4 42 33 O=C(N/C=C/c1ccccc1Cl)N1CCN(c2ccccc2F)CC1 ZINC000217825960 FH For-Sale Unstable KCNQ2 42 36 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)[C@@H](C)N ZINC000217825963 BD On-Demand Unstable TRPM8 22 56 Cc1ccccc1OCC(=O)Nc1ccccc1C(=O)c1ccccc1 ZINC000217825972 EI In-Stock Unstable CETP 0 43 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)c3cccn(C)c3=O)C2)n1 ZINC000217825974 GF In-Stock Unstable Q8MHZ5_SHEEP 49 33 C[C@H](O)[C@@H](NC(=O)[C@@H](N)CCS(C)(=O)=O)C(=O)O ZINC000217826012 CA For-Sale Unstable ENPEP 74 42 C[C@H](O)[C@@H](NC(=O)[C@@H](N)CCS(C)(=O)=O)C(=O)O ZINC000217826012 CA For-Sale Unstable DLG4 42 33 CN(C)CCN(C(=O)c1cc(Cl)ccc1I)C1CCCC1 ZINC000217826021 HH On-Demand Unstable ACE 61 51 CN(C)CCN(C(=O)c1cc(Cl)ccc1I)C1CCCC1 ZINC000217826021 HH On-Demand Unstable C5AR1 23 40 CN(Cc1ccsc1)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217826032 CG For-Sale Unstable PTGER2 24 42 CN(Cc1ccsc1)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217826032 CG For-Sale Unstable HSD17B2 26 42 CN(Cc1ccsc1)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217826032 CG For-Sale Unstable HCAR3 23 40 CN(Cc1ccsc1)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217826032 CG For-Sale Unstable AKR1C3 32 40 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)c3cccn(C)c3=O)C2)n1 ZINC000217826042 GF In-Stock Unstable Q8MHZ5_SHEEP 49 33 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)[C@@H](C)N ZINC000217826043 BD On-Demand Unstable TRPM8 22 56 Cc1ccnc(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217826058 CH For-Sale Unstable TYK2 65 39 Cc1ccccc1OCC(=O)NCCCc1cccc(OC(C)C)c1 ZINC000217826091 EH In-Stock Unstable HRH2 27 40 Cc1ccccc1OCC(=O)NCCCc1cccc(OC(C)C)c1 ZINC000217826091 EH In-Stock Unstable FDFT1 24 50 Cc1ccccc1OCC(=O)NCCCc1cccc(OC(C)C)c1 ZINC000217826091 EH In-Stock Unstable CYSP_TRYCR 0 45 Cc1ccccc1OCC(=O)NCCCc1cccc(OC(C)C)c1 ZINC000217826091 EH In-Stock Unstable MTNR1A 40 45 Cc1ccccc1OCC(=O)NCCCc1cccc(OC(C)C)c1 ZINC000217826091 EH In-Stock Unstable MTNR1B 43 40 Cc1ccccc1OCC(=O)NCCCc1cccc(OC(C)C)c1 ZINC000217826091 EH In-Stock Unstable AMP1_PLAFQ 24 43 Cc1ccccc1OCC(=O)NCCCc1cccc(OC(C)C)c1 ZINC000217826091 EH In-Stock Unstable FFAR1 15 41 Cc1ccccc1OCC(=O)NCCCc1cccc(OC(C)C)c1 ZINC000217826091 EH In-Stock Unstable CRTM 79 50 Cc1ccccc1OCC(=O)NCCCc1cccc(OC(C)C)c1 ZINC000217826091 EH In-Stock Unstable PDS 41 38 C[C@H](O)[C@H](NC(=O)[C@@H](N)CCS(C)(=O)=O)C(=O)O ZINC000217826095 CA For-Sale Unstable ENPEP 74 42 C[C@H](O)[C@H](NC(=O)[C@@H](N)CCS(C)(=O)=O)C(=O)O ZINC000217826095 CA For-Sale Unstable DLG4 42 33 CNC(=O)[C@@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000217826120 BD On-Demand Unstable SLC6A1 92 39 CNC(=O)[C@@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000217826120 BD On-Demand Unstable VACHT_TETCF 0 42 CNC(=O)[C@@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000217826120 BD On-Demand Unstable HRH3 22 40 CNC(=O)[C@@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000217826120 BD On-Demand Unstable HSD11B1 18 41 CNC(=O)[C@@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000217826120 BD On-Demand Unstable NPY2R 18 46 CNC(=O)[C@@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000217826120 BD On-Demand Unstable PREP 46 50 CNC(=O)[C@@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000217826120 BD On-Demand Unstable EPHX2 21 53 CNC(=O)[C@@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000217826120 BD On-Demand Unstable MMP1 15 40 CNC(=O)[C@@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000217826120 BD On-Demand Unstable SMO 41 40 CNC(=O)[C@@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000217826120 BD On-Demand Unstable RHOA 0 55 CNC(=O)[C@@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000217826120 BD On-Demand Unstable L3MBTL1 0 43 CNC(=O)[C@@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000217826120 BD On-Demand Unstable L3MBTL3 79 43 CNC(=O)[C@@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000217826120 BD On-Demand Unstable MBTD1 0 42 CNC(=O)[C@@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000217826120 BD On-Demand Unstable MAP3K12 39 44 C=CCN(C(=O)c1ccc(=O)[nH]n1)C1CCCC1 ZINC000217826122 BD For-Sale Unstable ACE 40 34 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)[C@@H](C)N ZINC000217826128 BD For-Sale Unstable TRPM8 22 56 COc1cccc2cc(C(=O)N3CCC[C@@H](Cc4nc(-c5ccccc5C)no4)C3)oc12 ZINC000217826155 IJ In-Stock Unstable HRH3 16 41 Cc1cn2c(CN(C)C(=O)c3ccc(S(=O)(=O)NC4CC4)cc3)c(C)nc2s1 ZINC000217826178 HF On-Demand Unstable CCR8 41 31 CCC[C@@H](N)C(=O)N1C[C@H](C)C[C@@H](C)C1 ZINC000217826203 BD For-Sale Unstable DPP7 60 38 CC(C)N(C)CCCNCc1ccc(Br)c(F)c1 ZINC000217826205 DG On-Demand Unstable LEF 63 35 Cc1ccccc1OCC(=O)NCCCc1ccc(OC(C)C)cc1 ZINC000217826209 EH In-Stock Unstable CYSP_TRYCR 0 47 Cc1ccccc1OCC(=O)NCCCc1ccc(OC(C)C)cc1 ZINC000217826209 EH In-Stock Unstable MTNR1B 25 41 Cc1ccccc1OCC(=O)NCCCc1ccc(OC(C)C)cc1 ZINC000217826209 EH In-Stock Unstable CRTM 44 41 COc1cccc2cc(C(=O)N3CCC[C@H](Cc4nc(-c5ccccc5C)no4)C3)oc12 ZINC000217826220 IJ In-Stock Unstable HRH3 16 41 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)[C@@H](C)N ZINC000217826227 BD For-Sale Unstable TRPM8 22 56 CCC[C@H](N)C(=O)N1C[C@H](C)C[C@@H](C)C1 ZINC000217826268 BD On-Demand Unstable DPP7 60 38 CCC[C@H](N)C(=O)N1C[C@H](C)C[C@@H](C)C1 ZINC000217826268 BD On-Demand Unstable DPP8 18 40 COC[C@H](O)CNC(c1ccccc1)(c1ccccc1)c1ccc(OC)cc1 ZINC000217826314 GH For-Sale Unstable ADRB2 32 43 COC[C@H](O)CNC(c1ccccc1)(c1ccccc1)c1ccc(OC)cc1 ZINC000217826314 GH For-Sale Unstable ADRB3 26 41 COC[C@H](O)CNC(c1ccccc1)(c1ccccc1)c1ccc(OC)cc1 ZINC000217826314 GH For-Sale Unstable CASR 38 45 COC[C@H](O)CNC(c1ccccc1)(c1ccccc1)c1ccc(OC)cc1 ZINC000217826314 GH For-Sale Unstable CYP2D6 26 43 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)[C@@H](N)CCS(C)(=O)=O ZINC000217826328 DD For-Sale Unstable TRPM8 16 45 Cc1cc(C)n(CCC(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)n1 ZINC000217826334 ED In-Stock Unstable CHRNA4 30 52 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)c3ccc(=O)n(C)n3)C2)n1 ZINC000217826340 GE In-Stock Unstable HRH3 15 40 COc1ccc(CN(C)[C@@H](C)C2CC2)cc1/C=C\C(=O)O ZINC000217826400 CG For-Sale Unstable PTGER2 23 40 COc1ccc(CN(C)[C@@H](C)C2CC2)cc1/C=C\C(=O)O ZINC000217826400 CG For-Sale Unstable PTGER4 0 40 Cc1cn2c(CN(C)C(=O)c3ccc(S(=O)(=O)NC(C)C)cc3)c(C)nc2s1 ZINC000217826404 HF On-Demand Unstable LIMK2 45 41 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)c3ccc(=O)n(C)n3)C2)n1 ZINC000217826435 GE In-Stock Unstable HRH3 15 40 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)[C@@H](N)CCS(C)(=O)=O ZINC000217826439 DD For-Sale Unstable TRPM8 16 45 COc1ccc(CN(C)[C@H](C)C2CC2)cc1/C=C\C(=O)O ZINC000217826460 CG For-Sale Unstable PTGER2 23 40 COc1ccc(CN(C)[C@H](C)C2CC2)cc1/C=C\C(=O)O ZINC000217826460 CG For-Sale Unstable PTGER4 15 40 O=C1CNC(=O)N1C[C@@H]1CCCCO1 ZINC000217826465 AC On-Demand Unstable PDE8B 51 35 Cc1cn2c(CN(C)C(=O)c3ccc(S(=O)(=O)NC(C)(C)C)cc3)c(C)nc2s1 ZINC000217826490 IG On-Demand Unstable LIMK2 43 39 O=C(NCC1(O)CCC1)c1ccc(Br)c(Cl)c1 ZINC000217826491 DF On-Demand Unstable P2RX7 0 45 CCOc1ccc(CCCNC(=O)COc2ccccc2C)cc1 ZINC000217826517 EH In-Stock Unstable CYSP_TRYCR 0 48 CCOc1ccc(CCCNC(=O)COc2ccccc2C)cc1 ZINC000217826517 EH In-Stock Unstable SCN2A 26 47 CCOc1ccc(CCCNC(=O)COc2ccccc2C)cc1 ZINC000217826517 EH In-Stock Unstable MTNR1A 44 41 CCOc1ccc(CCCNC(=O)COc2ccccc2C)cc1 ZINC000217826517 EH In-Stock Unstable MTNR1B 34 43 CCOc1ccc(CCCNC(=O)COc2ccccc2C)cc1 ZINC000217826517 EH In-Stock Unstable FAAH 17 41 CCOc1ccc(CCCNC(=O)COc2ccccc2C)cc1 ZINC000217826517 EH In-Stock Unstable CRTM 45 43 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)[C@@H](N)CCS(C)(=O)=O ZINC000217826529 DD For-Sale Unstable TRPM8 16 45 O=C1CNC(=O)N1C[C@H]1CCCCO1 ZINC000217826544 AC On-Demand Unstable PDE8B 51 35 CC(=O)N1CCC[C@@H](Cc2nc(-c3ccccc3C)no2)C1 ZINC000217826556 CF In-Stock Unstable HRH3 19 43 CC(=O)N1CCC[C@@H](Cc2nc(-c3ccccc3C)no2)C1 ZINC000217826556 CF In-Stock Unstable Q8MHZ5_SHEEP 42 33 CCCOc1ccccc1CCCNC(=O)COc1ccccc1C ZINC000217826602 EH In-Stock Unstable CYSP_TRYCR 0 48 CCCOc1ccccc1CCCNC(=O)COc1ccccc1C ZINC000217826602 EH In-Stock Unstable MTNR1A 43 42 CCCOc1ccccc1CCCNC(=O)COc1ccccc1C ZINC000217826602 EH In-Stock Unstable MTNR1B 48 43 CC[C@@H](C)NS(=O)(=O)c1ccc(C(=O)N(C)Cc2c(C)nc3sc(C)cn23)cc1 ZINC000217826604 IG On-Demand Unstable LIMK2 29 40 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)[C@@H](N)CCS(C)(=O)=O ZINC000217826624 DD For-Sale Unstable TRPM8 16 45 CC(=O)N1CCC[C@H](Cc2nc(-c3ccccc3C)no2)C1 ZINC000217826631 CF In-Stock Unstable HRH3 19 43 CC(=O)N1CCC[C@H](Cc2nc(-c3ccccc3C)no2)C1 ZINC000217826631 CF In-Stock Unstable Q8MHZ5_SHEEP 42 33 COC(=O)C[C@H](c1ccc(OC)cc1)c1c(O)c2ccccc2oc1=O ZINC000217826643 FG In-Stock Unstable MAOB 20 40 COC(=O)C[C@H](c1ccc(OC)cc1)c1c(O)c2ccccc2oc1=O ZINC000217826643 FG In-Stock Unstable CYP2C9 17 41 COC(=O)C[C@H](c1ccc(OC)cc1)c1c(O)c2ccccc2oc1=O ZINC000217826643 FG In-Stock Unstable NQO1 73 69 COC(=O)C[C@H](c1ccc(OC)cc1)c1c(O)c2ccccc2oc1=O ZINC000217826643 FG In-Stock Unstable GPR35 21 41 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1ccc(Cl)c(N)c1 ZINC000217826699 DI For-Sale Unstable TRPM8 21 74 Cc1ccccc1OCC(=O)N[C@H](C)COc1ccccc1C ZINC000217826702 DG In-Stock Unstable ADRB2 22 45 Cc1ccccc1OCC(=O)N[C@H](C)COc1ccccc1C ZINC000217826702 DG In-Stock Unstable SDH1 0 43 Cc1ccccc1OCC(=O)N[C@H](C)COc1ccccc1C ZINC000217826702 DG In-Stock Unstable CETP 0 41 Cc1ccccc1OCC(=O)N[C@H](C)COc1ccccc1C ZINC000217826702 DG In-Stock Unstable CAPN2 26 40 CC[C@H](C)NS(=O)(=O)c1ccc(C(=O)N(C)Cc2c(C)nc3sc(C)cn23)cc1 ZINC000217826703 IG On-Demand Unstable LIMK2 29 40 CCOCC(=O)N1CCC[C@H](Cc2nc(-c3ccccc3C)no2)C1 ZINC000217826720 EF In-Stock Unstable HRH3 15 40 CCOCC(=O)N1CCC[C@H](Cc2nc(-c3ccccc3C)no2)C1 ZINC000217826720 EF In-Stock Unstable Q8MHZ5_SHEEP 40 31 CCOC(=O)[C@H](Oc1ccc(F)c(Cl)c1)c1ccccc1 ZINC000217826734 DI On-Demand Unstable PPARG 17 42 CCOC(=O)[C@H](Oc1ccc(F)c(Cl)c1)c1ccccc1 ZINC000217826734 DI On-Demand Unstable PPARA 21 42 COC(=O)C[C@@H](c1ccc(OC)cc1)c1c(O)c2ccccc2oc1=O ZINC000217826743 FG In-Stock Unstable MAOB 20 40 COC(=O)C[C@@H](c1ccc(OC)cc1)c1c(O)c2ccccc2oc1=O ZINC000217826743 FG In-Stock Unstable CYP2C9 17 41 COC(=O)C[C@@H](c1ccc(OC)cc1)c1c(O)c2ccccc2oc1=O ZINC000217826743 FG In-Stock Unstable NQO1 73 69 COC(=O)C[C@@H](c1ccc(OC)cc1)c1c(O)c2ccccc2oc1=O ZINC000217826743 FG In-Stock Unstable GPR35 21 41 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1ccc(Cl)c(N)c1 ZINC000217826757 DI For-Sale Unstable TRPM8 21 74 CCOCC(=O)N1CCC[C@@H](Cc2nc(-c3ccccc3C)no2)C1 ZINC000217826783 EF In-Stock Unstable HRH3 15 40 CCOCC(=O)N1CCC[C@@H](Cc2nc(-c3ccccc3C)no2)C1 ZINC000217826783 EF In-Stock Unstable Q8MHZ5_SHEEP 40 31 Cc1cn2c(CN(C)C(=O)Cn3nnc(-c4ccc(Cl)cc4)n3)c(C)nc2s1 ZINC000217826798 HF On-Demand Unstable SCARB1 34 41 Cc1ccc(OC[C@@H](C)NC(=O)COc2ccccc2C)cc1 ZINC000217826807 DG In-Stock Unstable SDH1 0 42 Cc1ccc(OC[C@@H](C)NC(=O)COc2ccccc2C)cc1 ZINC000217826807 DG In-Stock Unstable CETP 0 42 Cc1ccc(OC[C@@H](C)NC(=O)COc2ccccc2C)cc1 ZINC000217826807 DG In-Stock Unstable CAPN2 22 40 Cc1nc2sccn2c1CN[C@@H]1CCN(C)C1=O ZINC000217826821 CD For-Sale Unstable HA 0 42 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)c1ccc(Cl)c(N)c1 ZINC000217826833 DI For-Sale Unstable TRPM8 21 74 CC[C@@H](C)c1ccccc1NC(=O)N/C=C/c1ccccc1Cl ZINC000217826842 EK For-Sale Unstable CXCL8 42 37 O=C(CCCCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)Nc1cccnc1 ZINC000217826868 II In-Stock Unstable HDAC3 28 50 O=C(CCCCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)Nc1cccnc1 ZINC000217826868 II In-Stock Unstable HDAC6 23 50 Cc1ccc(OC[C@H](C)NC(=O)COc2ccccc2C)cc1 ZINC000217826886 DG In-Stock Unstable SDH1 0 42 Cc1ccc(OC[C@H](C)NC(=O)COc2ccccc2C)cc1 ZINC000217826886 DG In-Stock Unstable CETP 0 42 Cc1ccc(OC[C@H](C)NC(=O)COc2ccccc2C)cc1 ZINC000217826886 DG In-Stock Unstable CAPN2 22 40 Cc1nc2sccn2c1CN[C@H]1CCN(C)C1=O ZINC000217826887 CD For-Sale Unstable HA 0 42 CCOC(=O)CCC(=O)N1CCC[C@H](Cc2nc(-c3ccccc3C)no2)C1 ZINC000217826900 GG In-Stock Unstable HRH3 15 40 CCOC(=O)CCC(=O)N1CCC[C@H](Cc2nc(-c3ccccc3C)no2)C1 ZINC000217826900 GG In-Stock Unstable Q8MHZ5_SHEEP 40 30 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)c1ccc(Cl)c(N)c1 ZINC000217826921 DI For-Sale Unstable TRPM8 21 74 CC[C@H](C)c1ccccc1NC(=O)N/C=C/c1ccccc1Cl ZINC000217826927 EK For-Sale Unstable CXCL8 42 37 COc1ccc(/C=C\C(=O)O)cc1CN1CCOC1=O ZINC000217826960 CD For-Sale Unstable PTGER2 0 42 O=C(CCCCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)Nc1cccnc1 ZINC000217826961 II In-Stock Unstable HDAC3 28 50 O=C(CCCCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)Nc1cccnc1 ZINC000217826961 II In-Stock Unstable HDAC6 23 50 CCOC(=O)CCC(=O)N1CCC[C@@H](Cc2nc(-c3ccccc3C)no2)C1 ZINC000217826976 GG In-Stock Unstable HRH3 15 40 CCOC(=O)CCC(=O)N1CCC[C@@H](Cc2nc(-c3ccccc3C)no2)C1 ZINC000217826976 GG In-Stock Unstable Q8MHZ5_SHEEP 40 30 CSC[C@@](C)(O)CNC(=O)c1cc(C)cc(Cl)c1 ZINC000217826993 CE On-Demand Unstable CACNA1I 40 36 CN1CCN(C(=O)c2ccc(Br)cc2C(F)(F)F)CC1 ZINC000217826994 FF On-Demand Unstable HRH4 29 40 CC[C@@H](C)[C@@H](N)C(=O)N[C@@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217827023 CF For-Sale Unstable TRPM8 18 48 O=C(O)/C=C\c1ccccc1CN1C(=O)CCCC1=O ZINC000217827048 CD For-Sale Unstable PTGER2 44 49 O=C(O)/C=C\c1ccccc1CN1C(=O)CCCC1=O ZINC000217827048 CD For-Sale Unstable PTGER4 23 49 O=C(O)/C=C\c1ccccc1CN1C(=O)CCCC1=O ZINC000217827048 CD For-Sale Unstable PTGER3 25 49 CSC[C@](C)(O)CNC(=O)c1cc(C)cc(Cl)c1 ZINC000217827070 CE On-Demand Unstable CACNA1I 40 36 COc1cccc(C(=O)N2CCC[C@@H](Cc3nc(-c4ccccc4C)no3)C2)c1 ZINC000217827079 GI In-Stock Unstable DRD4 45 35 COc1cccc(C(=O)N2CCC[C@@H](Cc3nc(-c4ccccc4C)no3)C2)c1 ZINC000217827079 GI In-Stock Unstable HRH3 22 47 COc1cccc(C(=O)N2CCC[C@@H](Cc3nc(-c4ccccc4C)no3)C2)c1 ZINC000217827079 GI In-Stock Unstable HSD11B1 19 42 COc1cccc(C(=O)N2CCC[C@@H](Cc3nc(-c4ccccc4C)no3)C2)c1 ZINC000217827079 GI In-Stock Unstable Q8MHZ5_SHEEP 49 32 COc1cccc(C(=O)N2CCC[C@@H](Cc3nc(-c4ccccc4C)no3)C2)c1 ZINC000217827079 GI In-Stock Unstable MAP3K12 31 41 CC[C@H](C)[C@@H](N)C(=O)N[C@@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217827092 CF For-Sale Unstable TRPM8 18 48 CCC[C@@H](N)C(=O)N[C@@H]1CCC[C@@H](C)C1 ZINC000217827126 BD For-Sale Unstable DPP7 0 40 CCC[C@@H](N)C(=O)N[C@@H]1CCC[C@@H](C)C1 ZINC000217827126 BD For-Sale Unstable DPP8 0 40 CCC[C@@H](N)C(=O)N[C@@H]1CCC[C@@H](C)C1 ZINC000217827126 BD For-Sale Unstable DPP9 0 40 O=S(=O)(Cl)Cc1cccc(OC2CC2)c1 ZINC000217827159 BE In-Stock Unstable PRSS2 45 33 O=C(N/C=C/c1ccccc1Cl)NC1CCN(Cc2ccccc2)CC1 ZINC000217827161 FI For-Sale Unstable CHRM2 22 42 O=C(N/C=C/c1ccccc1Cl)NC1CCN(Cc2ccccc2)CC1 ZINC000217827161 FI For-Sale Unstable CHRM1 15 47 O=C(N/C=C/c1ccccc1Cl)NC1CCN(Cc2ccccc2)CC1 ZINC000217827161 FI For-Sale Unstable DRD2 25 59 O=C(N/C=C/c1ccccc1Cl)NC1CCN(Cc2ccccc2)CC1 ZINC000217827161 FI For-Sale Unstable DRD4 55 60 O=C(N/C=C/c1ccccc1Cl)NC1CCN(Cc2ccccc2)CC1 ZINC000217827161 FI For-Sale Unstable ACHE 42 48 O=C(N/C=C/c1ccccc1Cl)NC1CCN(Cc2ccccc2)CC1 ZINC000217827161 FI For-Sale Unstable HRH2 19 41 O=C(N/C=C/c1ccccc1Cl)NC1CCN(Cc2ccccc2)CC1 ZINC000217827161 FI For-Sale Unstable DRD3 21 59 O=C(N/C=C/c1ccccc1Cl)NC1CCN(Cc2ccccc2)CC1 ZINC000217827161 FI For-Sale Unstable KCNH2 15 42 O=C(N/C=C/c1ccccc1Cl)NC1CCN(Cc2ccccc2)CC1 ZINC000217827161 FI For-Sale Unstable CHRM3 25 47 O=C(N/C=C/c1ccccc1Cl)NC1CCN(Cc2ccccc2)CC1 ZINC000217827161 FI For-Sale Unstable LTA4H 16 40 O=C(N/C=C/c1ccccc1Cl)NC1CCN(Cc2ccccc2)CC1 ZINC000217827161 FI For-Sale Unstable SIGMAR1 60 60 O=C(N/C=C/c1ccccc1Cl)NC1CCN(Cc2ccccc2)CC1 ZINC000217827161 FI For-Sale Unstable SSTR5 47 40 O=C(N/C=C/c1ccccc1Cl)NC1CCN(Cc2ccccc2)CC1 ZINC000217827161 FI For-Sale Unstable CCR3 45 49 O=C(N/C=C/c1ccccc1Cl)NC1CCN(Cc2ccccc2)CC1 ZINC000217827161 FI For-Sale Unstable SLC6A5 16 43 O=C(N/C=C/c1ccccc1Cl)NC1CCN(Cc2ccccc2)CC1 ZINC000217827161 FI For-Sale Unstable EPHX2 21 53 O=C(N/C=C/c1ccccc1Cl)NC1CCN(Cc2ccccc2)CC1 ZINC000217827161 FI For-Sale Unstable MCHR1 55 52 O=C(N/C=C/c1ccccc1Cl)NC1CCN(Cc2ccccc2)CC1 ZINC000217827161 FI For-Sale Unstable CACNA1G 28 43 O=C(N/C=C/c1ccccc1Cl)NC1CCN(Cc2ccccc2)CC1 ZINC000217827161 FI For-Sale Unstable CCR8 15 45 O=C(N/C=C/c1ccccc1Cl)NC1CCN(Cc2ccccc2)CC1 ZINC000217827161 FI For-Sale Unstable ADIPOR1 0 48 O=C(N/C=C/c1ccccc1Cl)NC1CCN(Cc2ccccc2)CC1 ZINC000217827161 FI For-Sale Unstable ADIPOR2 0 48 CC[C@@H](C)[C@H](N)C(=O)N[C@@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217827174 CF For-Sale Unstable TRPM8 18 48 CCC[C@H](N)C(=O)N[C@@H]1CCC[C@@H](C)C1 ZINC000217827186 BD On-Demand Unstable DPP7 0 40 CCC[C@H](N)C(=O)N[C@@H]1CCC[C@@H](C)C1 ZINC000217827186 BD On-Demand Unstable DPP8 0 40 CCC[C@H](N)C(=O)N[C@@H]1CCC[C@@H](C)C1 ZINC000217827186 BD On-Demand Unstable DPP9 0 40 COc1cccc(C(=O)N2CCC[C@H](Cc3nc(-c4ccccc4C)no3)C2)c1 ZINC000217827189 GI In-Stock Unstable DRD4 45 35 COc1cccc(C(=O)N2CCC[C@H](Cc3nc(-c4ccccc4C)no3)C2)c1 ZINC000217827189 GI In-Stock Unstable HRH3 22 47 COc1cccc(C(=O)N2CCC[C@H](Cc3nc(-c4ccccc4C)no3)C2)c1 ZINC000217827189 GI In-Stock Unstable HSD11B1 19 42 COc1cccc(C(=O)N2CCC[C@H](Cc3nc(-c4ccccc4C)no3)C2)c1 ZINC000217827189 GI In-Stock Unstable CCR3 15 41 COc1cccc(C(=O)N2CCC[C@H](Cc3nc(-c4ccccc4C)no3)C2)c1 ZINC000217827189 GI In-Stock Unstable Q8MHZ5_SHEEP 49 32 COc1cccc(C(=O)N2CCC[C@H](Cc3nc(-c4ccccc4C)no3)C2)c1 ZINC000217827189 GI In-Stock Unstable MAP3K12 31 41 CCCn1c(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc2c(=O)n3ccccc3nc21 ZINC000217827213 IG For-Sale Unstable POLR1A 70 34 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)NCc3ccccn3)[C@H]21 ZINC000217827221 JF In-Stock Unstable HTR7 18 43 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)NCc3ccccn3)[C@H]21 ZINC000217827221 JF In-Stock Unstable SCN9A 0 41 O=C(NCC1(c2ccccc2)CCC1)c1cc(N2CCCC2)ccn1 ZINC000217827222 EH On-Demand Unstable KCNA3 48 41 O=C(NCC1(c2ccccc2)CCC1)c1cc(N2CCCC2)ccn1 ZINC000217827222 EH On-Demand Unstable ACAT 0 45 O=C(NCC1(c2ccccc2)CCC1)c1cc(N2CCCC2)ccn1 ZINC000217827222 EH On-Demand Unstable HCN1 65 33 O=C(NCC1(c2ccccc2)CCC1)c1cc(N2CCCC2)ccn1 ZINC000217827222 EH On-Demand Unstable HCN4 48 31 CC[C@@H](C)c1ccc(OCc2ccccc2Br)cc1 ZINC000217827258 DK For-Sale Unstable FFAR1 15 49 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)CCCN ZINC000217827265 BE On-Demand Unstable TRPM8 20 62 CCC[C@@H](N)C(=O)N[C@H]1CCC[C@@H](C)C1 ZINC000217827270 BD For-Sale Unstable DPP7 0 40 CCC[C@@H](N)C(=O)N[C@H]1CCC[C@@H](C)C1 ZINC000217827270 BD For-Sale Unstable DPP8 0 40 CCC[C@@H](N)C(=O)N[C@H]1CCC[C@@H](C)C1 ZINC000217827270 BD For-Sale Unstable DPP9 0 40 CCCn1c(C(=O)NC[C@H]2CCCN2c2ccccc2)cc2c(=O)n3ccccc3nc21 ZINC000217827279 IG For-Sale Unstable POLR1A 70 34 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)NCc3ccccn3)[C@@H]21 ZINC000217827295 JF In-Stock Unstable HTR7 18 43 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)NCc3ccccn3)[C@@H]21 ZINC000217827295 JF In-Stock Unstable SCN9A 0 41 Cc1ccc2c(c1)[C@@H](NC(=O)COc1ccccc1C)CC(C)(C)O2 ZINC000217827301 EI In-Stock Unstable CETP 0 40 O=C(NCC1(c2ccccc2)CCC1)c1nn(-c2ccccc2)cc1O ZINC000217827308 EG On-Demand Unstable KCNA3 41 40 O=C(NCC1(c2ccccc2)CCC1)c1nn(-c2ccccc2)cc1O ZINC000217827308 EG On-Demand Unstable ACAT 0 47 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)c3ccccc3F)C2)n1 ZINC000217827326 GI In-Stock Unstable HRH3 19 46 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)c3ccccc3F)C2)n1 ZINC000217827326 GI In-Stock Unstable Q8MHZ5_SHEEP 41 31 Cc1nn(Cc2ccc(F)cc2/C=C\C(=O)O)c(C)c1C ZINC000217827328 CG For-Sale Unstable P2RX7 29 42 CC[C@H](C)c1ccc(OCc2ccccc2Br)cc1 ZINC000217827337 DK For-Sale Unstable FFAR1 15 49 CCC[C@H](N)C(=O)N[C@H]1CCC[C@@H](C)C1 ZINC000217827341 BD On-Demand Unstable DPP7 0 40 CCC[C@H](N)C(=O)N[C@H]1CCC[C@@H](C)C1 ZINC000217827341 BD On-Demand Unstable DPP8 0 40 CCC[C@H](N)C(=O)N[C@H]1CCC[C@@H](C)C1 ZINC000217827341 BD On-Demand Unstable DPP9 0 40 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)CCCN ZINC000217827345 BE On-Demand Unstable TRPM8 20 62 Cc1ccc2c(c1)[C@H](NC(=O)COc1ccccc1C)CC(C)(C)O2 ZINC000217827366 EI In-Stock Unstable CETP 0 40 COCCn1c(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc2c(=O)n3ccccc3nc21 ZINC000217827394 IF For-Sale Unstable POLR1A 69 33 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)Nc3nccs3)[C@H]21 ZINC000217827403 JG In-Stock Unstable MAP1 64 38 NS(=O)(=O)c1ccc(CN[C@@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217827421 CD For-Sale Unstable CA2 51 42 NS(=O)(=O)c1ccc(CN[C@@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217827421 CD For-Sale Unstable CA6 16 40 NS(=O)(=O)c1ccc(CN[C@@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217827421 CD For-Sale Unstable CA1 48 42 NS(=O)(=O)c1ccc(CN[C@@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217827421 CD For-Sale Unstable CA7 32 40 NS(=O)(=O)c1ccc(CN[C@@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217827421 CD For-Sale Unstable CA13 16 40 NS(=O)(=O)c1ccc(CN[C@@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217827421 CD For-Sale Unstable CA5B 26 40 NS(=O)(=O)c1ccc(CN[C@@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217827421 CD For-Sale Unstable CA4 30 40 NS(=O)(=O)c1ccc(CN[C@@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217827421 CD For-Sale Unstable CA12 37 44 NS(=O)(=O)c1ccc(CN[C@@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217827421 CD For-Sale Unstable CA9 44 44 NS(=O)(=O)c1ccc(CN[C@@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217827421 CD For-Sale Unstable CAH_METTE 24 40 NS(=O)(=O)c1ccc(CN[C@@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217827421 CD For-Sale Unstable CYNT 27 40 NS(=O)(=O)c1ccc(CN[C@@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217827421 CD For-Sale Unstable NCE103 16 40 NS(=O)(=O)c1ccc(CN[C@@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217827421 CD For-Sale Unstable A6YCJ1_9METZ 22 40 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)c3ccccc3F)C2)n1 ZINC000217827432 GI In-Stock Unstable HRH3 19 46 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)c3ccccc3F)C2)n1 ZINC000217827432 GI In-Stock Unstable Q8MHZ5_SHEEP 41 31 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)CCCN ZINC000217827444 BE For-Sale Unstable TRPM8 19 62 COCCn1c(C(=O)NC[C@H]2CCCN2c2ccccc2)cc2c(=O)n3ccccc3nc21 ZINC000217827456 IF For-Sale Unstable POLR1A 69 33 O=C(N/C=C/c1ccccc1Cl)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217827457 GH For-Sale Unstable DRD4 30 47 O=C(N/C=C/c1ccccc1Cl)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217827457 GH For-Sale Unstable SIGMAR1 23 52 O=C(N/C=C/c1ccccc1Cl)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217827457 GH For-Sale Unstable SSTR3 67 32 O=C(N/C=C/c1ccccc1Cl)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217827457 GH For-Sale Unstable FAAH 22 43 O=C(N/C=C/c1ccccc1Cl)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217827457 GH For-Sale Unstable MCHR1 30 50 Cc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)COc1ccccc1C ZINC000217827472 EI In-Stock Unstable CETP 0 41 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)Nc3nccs3)[C@@H]21 ZINC000217827481 JG In-Stock Unstable MAP1 64 38 NS(=O)(=O)c1ccc(CN[C@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217827509 CD For-Sale Unstable CA2 51 42 NS(=O)(=O)c1ccc(CN[C@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217827509 CD For-Sale Unstable CA6 16 40 NS(=O)(=O)c1ccc(CN[C@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217827509 CD For-Sale Unstable CA1 48 42 NS(=O)(=O)c1ccc(CN[C@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217827509 CD For-Sale Unstable CA7 32 40 NS(=O)(=O)c1ccc(CN[C@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217827509 CD For-Sale Unstable CA13 16 40 NS(=O)(=O)c1ccc(CN[C@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217827509 CD For-Sale Unstable CA5B 26 40 NS(=O)(=O)c1ccc(CN[C@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217827509 CD For-Sale Unstable CA4 30 40 NS(=O)(=O)c1ccc(CN[C@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217827509 CD For-Sale Unstable CA12 37 44 NS(=O)(=O)c1ccc(CN[C@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217827509 CD For-Sale Unstable CA9 44 44 NS(=O)(=O)c1ccc(CN[C@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217827509 CD For-Sale Unstable CAH_METTE 24 40 NS(=O)(=O)c1ccc(CN[C@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217827509 CD For-Sale Unstable CYNT 27 40 NS(=O)(=O)c1ccc(CN[C@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217827509 CD For-Sale Unstable NCE103 16 40 NS(=O)(=O)c1ccc(CN[C@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217827509 CD For-Sale Unstable A6YCJ1_9METZ 22 40 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)CCCN ZINC000217827510 BE For-Sale Unstable TRPM8 19 62 C[C@@H]1CC(=O)N(Cc2ccccc2/C=C\C(=O)O)C1=O ZINC000217827511 CD For-Sale Unstable PTGER2 39 44 C[C@@H]1CC(=O)N(Cc2ccccc2/C=C\C(=O)O)C1=O ZINC000217827511 CD For-Sale Unstable PTGER4 0 44 C[C@@H]1CC(=O)N(Cc2ccccc2/C=C\C(=O)O)C1=O ZINC000217827511 CD For-Sale Unstable PTGER3 26 48 Cc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)COc1ccccc1C ZINC000217827526 EI In-Stock Unstable CETP 0 41 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)c3cccc(Cl)c3)C2)n1 ZINC000217827551 GJ In-Stock Unstable HRH3 18 45 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)c3cccc(Cl)c3)C2)n1 ZINC000217827551 GJ In-Stock Unstable HSD11B1 15 54 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)c3cccc(Cl)c3)C2)n1 ZINC000217827551 GJ In-Stock Unstable GRM5 27 41 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)c3cccc(Cl)c3)C2)n1 ZINC000217827551 GJ In-Stock Unstable Q8MHZ5_SHEEP 54 37 CCOC(=O)N1CCN(C(=O)N/C=C/c2ccccc2Cl)CC1 ZINC000217827561 EF For-Sale Unstable P2RY12 41 38 CCCCn1c(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc2c(=O)n3ccccc3nc21 ZINC000217827564 IH For-Sale Unstable POLR1A 64 33 NS(=O)(=O)c1ccc(CN[C@@H]2C[C@H]3CC=C[C@H]32)cc1 ZINC000217827569 CD For-Sale Unstable CA2 51 42 NS(=O)(=O)c1ccc(CN[C@@H]2C[C@H]3CC=C[C@H]32)cc1 ZINC000217827569 CD For-Sale Unstable CA6 16 40 NS(=O)(=O)c1ccc(CN[C@@H]2C[C@H]3CC=C[C@H]32)cc1 ZINC000217827569 CD For-Sale Unstable CA1 48 42 NS(=O)(=O)c1ccc(CN[C@@H]2C[C@H]3CC=C[C@H]32)cc1 ZINC000217827569 CD For-Sale Unstable CA7 32 40 NS(=O)(=O)c1ccc(CN[C@@H]2C[C@H]3CC=C[C@H]32)cc1 ZINC000217827569 CD For-Sale Unstable CA13 16 40 NS(=O)(=O)c1ccc(CN[C@@H]2C[C@H]3CC=C[C@H]32)cc1 ZINC000217827569 CD For-Sale Unstable CA5B 26 40 NS(=O)(=O)c1ccc(CN[C@@H]2C[C@H]3CC=C[C@H]32)cc1 ZINC000217827569 CD For-Sale Unstable CA4 30 40 NS(=O)(=O)c1ccc(CN[C@@H]2C[C@H]3CC=C[C@H]32)cc1 ZINC000217827569 CD For-Sale Unstable CA12 37 44 NS(=O)(=O)c1ccc(CN[C@@H]2C[C@H]3CC=C[C@H]32)cc1 ZINC000217827569 CD For-Sale Unstable CA9 44 44 NS(=O)(=O)c1ccc(CN[C@@H]2C[C@H]3CC=C[C@H]32)cc1 ZINC000217827569 CD For-Sale Unstable CAH_METTE 24 40 NS(=O)(=O)c1ccc(CN[C@@H]2C[C@H]3CC=C[C@H]32)cc1 ZINC000217827569 CD For-Sale Unstable CYNT 27 40 NS(=O)(=O)c1ccc(CN[C@@H]2C[C@H]3CC=C[C@H]32)cc1 ZINC000217827569 CD For-Sale Unstable NCE103 16 40 NS(=O)(=O)c1ccc(CN[C@@H]2C[C@H]3CC=C[C@H]32)cc1 ZINC000217827569 CD For-Sale Unstable A6YCJ1_9METZ 22 40 C[C@H]1CC(=O)N(Cc2ccccc2/C=C\C(=O)O)C1=O ZINC000217827580 CD For-Sale Unstable PTGER2 39 44 C[C@H]1CC(=O)N(Cc2ccccc2/C=C\C(=O)O)C1=O ZINC000217827580 CD For-Sale Unstable PTGER4 0 44 C[C@H]1CC(=O)N(Cc2ccccc2/C=C\C(=O)O)C1=O ZINC000217827580 CD For-Sale Unstable PTGER3 26 48 CC(C)C[C@@H](N)C(=O)N[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217827581 CF For-Sale Unstable TRPM8 18 49 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)c3cccc(Cl)c3)C2)n1 ZINC000217827585 GJ In-Stock Unstable HRH3 17 45 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)c3cccc(Cl)c3)C2)n1 ZINC000217827585 GJ In-Stock Unstable HSD11B1 15 54 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)c3cccc(Cl)c3)C2)n1 ZINC000217827585 GJ In-Stock Unstable GRM5 27 41 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)c3cccc(Cl)c3)C2)n1 ZINC000217827585 GJ In-Stock Unstable Q8MHZ5_SHEEP 54 37 CCCCn1c(C(=O)NC[C@H]2CCCN2c2ccccc2)cc2c(=O)n3ccccc3nc21 ZINC000217827617 IH For-Sale Unstable POLR1A 64 33 NS(=O)(=O)c1ccc(CN[C@H]2C[C@H]3CC=C[C@@H]23)cc1 ZINC000217827627 CD For-Sale Unstable CA2 51 42 NS(=O)(=O)c1ccc(CN[C@H]2C[C@H]3CC=C[C@@H]23)cc1 ZINC000217827627 CD For-Sale Unstable CA6 16 40 NS(=O)(=O)c1ccc(CN[C@H]2C[C@H]3CC=C[C@@H]23)cc1 ZINC000217827627 CD For-Sale Unstable CA1 48 42 NS(=O)(=O)c1ccc(CN[C@H]2C[C@H]3CC=C[C@@H]23)cc1 ZINC000217827627 CD For-Sale Unstable CA7 32 40 NS(=O)(=O)c1ccc(CN[C@H]2C[C@H]3CC=C[C@@H]23)cc1 ZINC000217827627 CD For-Sale Unstable CA13 16 40 NS(=O)(=O)c1ccc(CN[C@H]2C[C@H]3CC=C[C@@H]23)cc1 ZINC000217827627 CD For-Sale Unstable CA5B 26 40 NS(=O)(=O)c1ccc(CN[C@H]2C[C@H]3CC=C[C@@H]23)cc1 ZINC000217827627 CD For-Sale Unstable CA4 30 40 NS(=O)(=O)c1ccc(CN[C@H]2C[C@H]3CC=C[C@@H]23)cc1 ZINC000217827627 CD For-Sale Unstable CA12 37 44 NS(=O)(=O)c1ccc(CN[C@H]2C[C@H]3CC=C[C@@H]23)cc1 ZINC000217827627 CD For-Sale Unstable CA9 44 44 NS(=O)(=O)c1ccc(CN[C@H]2C[C@H]3CC=C[C@@H]23)cc1 ZINC000217827627 CD For-Sale Unstable CAH_METTE 24 40 NS(=O)(=O)c1ccc(CN[C@H]2C[C@H]3CC=C[C@@H]23)cc1 ZINC000217827627 CD For-Sale Unstable CYNT 27 40 NS(=O)(=O)c1ccc(CN[C@H]2C[C@H]3CC=C[C@@H]23)cc1 ZINC000217827627 CD For-Sale Unstable NCE103 16 40 NS(=O)(=O)c1ccc(CN[C@H]2C[C@H]3CC=C[C@@H]23)cc1 ZINC000217827627 CD For-Sale Unstable A6YCJ1_9METZ 22 40 CCOC(=O)[C@@H](C)NC(=O)c1ccc(OC)cc1F ZINC000217827659 CD On-Demand Unstable MTNR1A 40 41 CCOC(=O)[C@@H](C)NC(=O)c1ccc(OC)cc1F ZINC000217827659 CD On-Demand Unstable MTNR1B 36 41 CCOC(=O)[C@@H](C)NC(=O)c1ccc(OC)cc1F ZINC000217827659 CD On-Demand Unstable AKR1C2 43 37 CCOC(=O)[C@@H](C)NC(=O)c1ccc(OC)cc1F ZINC000217827659 CD On-Demand Unstable GPR35 20 41 O=C(O)/C=C\c1cccc(COCc2ccccc2)c1 ZINC000217827673 CH For-Sale Unstable NA 0 42 O=C(O)/C=C\c1cccc(COCc2ccccc2)c1 ZINC000217827673 CH For-Sale Unstable PTGER2 26 54 O=C(O)/C=C\c1cccc(COCc2ccccc2)c1 ZINC000217827673 CH For-Sale Unstable PTGER4 27 48 O=C(O)/C=C\c1cccc(COCc2ccccc2)c1 ZINC000217827673 CH For-Sale Unstable PTGER3 24 48 O=C(O)/C=C\c1cccc(COCc2ccccc2)c1 ZINC000217827673 CH For-Sale Unstable F3 24 43 O=C(O)/C=C\c1cccc(COCc2ccccc2)c1 ZINC000217827673 CH For-Sale Unstable MMP2 0 47 O=C(O)/C=C\c1cccc(COCc2ccccc2)c1 ZINC000217827673 CH For-Sale Unstable HDAC1 15 41 O=C(O)/C=C\c1cccc(COCc2ccccc2)c1 ZINC000217827673 CH For-Sale Unstable MMP9 0 47 O=C(O)/C=C\c1cccc(COCc2ccccc2)c1 ZINC000217827673 CH For-Sale Unstable PTGDR 0 43 O=C(O)/C=C\c1cccc(COCc2ccccc2)c1 ZINC000217827673 CH For-Sale Unstable MMP1 0 45 O=C(O)/C=C\c1cccc(COCc2ccccc2)c1 ZINC000217827673 CH For-Sale Unstable HCAR2 0 45 O=C(O)/C=C\c1cccc(COCc2ccccc2)c1 ZINC000217827673 CH For-Sale Unstable AKR1C3 37 51 O=C(O)/C=C\c1cccc(COCc2ccccc2)c1 ZINC000217827673 CH For-Sale Unstable AKR1B10 24 44 CC(C)C[C@H](N)C(=O)N[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217827684 CF For-Sale Unstable TRPM8 18 49 CCCCCN(C(C)C)[C@H](c1cccc(Cl)c1)[C@@H](N)CC ZINC000217827685 DK For-Sale Unstable OPRL1 0 41 O=C(CCc1ccc([N+](=O)[O-])cc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217827707 FG For-Sale Unstable LUXR 17 44 CCOC(=O)[C@H](C)NC(=O)c1ccc(OC)cc1F ZINC000217827730 CD On-Demand Unstable MTNR1A 40 41 CCOC(=O)[C@H](C)NC(=O)c1ccc(OC)cc1F ZINC000217827730 CD On-Demand Unstable MTNR1B 36 41 CCOC(=O)[C@H](C)NC(=O)c1ccc(OC)cc1F ZINC000217827730 CD On-Demand Unstable AKR1C2 43 37 CCOC(=O)[C@H](C)NC(=O)c1ccc(OC)cc1F ZINC000217827730 CD On-Demand Unstable GPR35 20 41 CCCCCN(C(C)C)[C@@H](c1cccc(Cl)c1)[C@@H](N)CC ZINC000217827760 DK For-Sale Unstable OPRL1 0 41 O=C(CCc1ccc([N+](=O)[O-])cc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217827783 FG For-Sale Unstable LUXR 17 44 O=C(O)/C=C\c1cc(F)ccc1COCc1ccccc1 ZINC000217827785 CH For-Sale Unstable PTGER2 22 49 O=C(O)/C=C\c1cc(F)ccc1COCc1ccccc1 ZINC000217827785 CH For-Sale Unstable PTGER4 29 49 O=C(O)/C=C\c1cc(F)ccc1COCc1ccccc1 ZINC000217827785 CH For-Sale Unstable PTGER3 24 49 O=C(O)/C=C\c1cc(F)ccc1COCc1ccccc1 ZINC000217827785 CH For-Sale Unstable PTGDR 0 46 O=C(O)/C=C\c1cc(F)ccc1COCc1ccccc1 ZINC000217827785 CH For-Sale Unstable HCAR2 0 46 O=C(O)/C=C\c1cc(F)ccc1COCc1ccccc1 ZINC000217827785 CH For-Sale Unstable AKR1C3 30 43 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(C(F)(F)F)cc1 ZINC000217827796 EK For-Sale Anodyne TRPV1 19 43 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(C(F)(F)F)cc1 ZINC000217827796 EK For-Sale Anodyne EPHX2 28 41 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(C(F)(F)F)cc1 ZINC000217827796 EK For-Sale Anodyne FPR2 28 41 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(C(F)(F)F)cc1 ZINC000217827796 EK For-Sale Anodyne PTPA 0 40 CNCC(=O)N[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217827800 BD For-Sale Unstable TRPM8 0 53 COc1ccc2occ(-c3c4cn[nH]c4nc4c3oc3cc(O)ccc34)c(=O)c2c1 ZINC000217827813 GI In-Stock Unstable ALDH2 68 34 Cn1c(=O)n(CCC(=O)Nc2ccc([N+](=O)[O-])cc2C(=O)c2ccccc2)c2ccccc21 ZINC000217827859 IH On-Demand Unstable F2RL3 50 37 O=C(O)/C=C\c1cc(COCc2ccccc2)ccc1F ZINC000217827864 CH For-Sale Unstable PTGER2 17 50 O=C(O)/C=C\c1cc(COCc2ccccc2)ccc1F ZINC000217827864 CH For-Sale Unstable PTGER4 25 46 O=C(O)/C=C\c1cc(COCc2ccccc2)ccc1F ZINC000217827864 CH For-Sale Unstable PTGER3 26 46 O=C(O)/C=C\c1cc(COCc2ccccc2)ccc1F ZINC000217827864 CH For-Sale Unstable PTGDR 0 47 O=C(O)/C=C\c1cc(COCc2ccccc2)ccc1F ZINC000217827864 CH For-Sale Unstable HCAR2 0 44 O=C(O)/C=C\c1cc(COCc2ccccc2)ccc1F ZINC000217827864 CH For-Sale Unstable AKR1C3 30 42 COc1ccc(Cl)cc1C(=O)N1CCC[C@@H](Cc2nc(-c3ccccc3C)no2)C1 ZINC000217827880 IJ In-Stock Unstable HRH3 18 43 COc1ccc(Cl)cc1C(=O)N1CCC[C@@H](Cc2nc(-c3ccccc3C)no2)C1 ZINC000217827880 IJ In-Stock Unstable HSD11B1 16 46 COc1ccc(Cl)cc1C(=O)N1CCC[C@@H](Cc2nc(-c3ccccc3C)no2)C1 ZINC000217827880 IJ In-Stock Unstable RBP4 25 40 COc1ccc(Cl)cc1C(=O)N1CCC[C@@H](Cc2nc(-c3ccccc3C)no2)C1 ZINC000217827880 IJ In-Stock Unstable Q8MHZ5_SHEEP 52 35 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(F)cc1F ZINC000217827886 DI For-Sale Anodyne SOAT1 38 44 CC(=O)Nc1ccc(CC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217827893 FF For-Sale Unstable LTA4H 20 40 CNCC(=O)N[C@H]1C[C@H](C)CC[C@@H]1C(C)C ZINC000217827927 BD For-Sale Unstable TRPM8 0 53 CC(=O)Nc1ccc(CC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217827951 FF For-Sale Unstable LTA4H 20 40 COc1ccc(COCC(F)(F)F)cc1/C=C\C(=O)O ZINC000217827954 CF For-Sale Unstable PTGER2 42 46 COc1ccc(COCC(F)(F)F)cc1/C=C\C(=O)O ZINC000217827954 CF For-Sale Unstable PTGER4 24 46 COc1ccc(COCC(F)(F)F)cc1/C=C\C(=O)O ZINC000217827954 CF For-Sale Unstable PTGER3 19 46 COc1ccc(COCC(F)(F)F)cc1/C=C\C(=O)O ZINC000217827954 CF For-Sale Unstable AKR1B10 32 40 COc1ccc(Cl)cc1C(=O)N1CCC[C@H](Cc2nc(-c3ccccc3C)no2)C1 ZINC000217827967 IJ In-Stock Unstable HRH3 18 43 COc1ccc(Cl)cc1C(=O)N1CCC[C@H](Cc2nc(-c3ccccc3C)no2)C1 ZINC000217827967 IJ In-Stock Unstable HSD11B1 16 46 COc1ccc(Cl)cc1C(=O)N1CCC[C@H](Cc2nc(-c3ccccc3C)no2)C1 ZINC000217827967 IJ In-Stock Unstable RBP4 25 40 COc1ccc(Cl)cc1C(=O)N1CCC[C@H](Cc2nc(-c3ccccc3C)no2)C1 ZINC000217827967 IJ In-Stock Unstable Q8MHZ5_SHEEP 52 35 Cc1cc(C(=O)N[C@H]2C[C@H](C)CC[C@H]2C(C)C)ccc1N ZINC000217827992 CH For-Sale Unstable TRPM8 21 68 CCc1nc2ccc(C(=O)NC[C@@H]3CCCN3c3ccccc3)cc2s1 ZINC000217828054 FI For-Sale Unstable LCK 27 43 O=C(CN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCc1ccc2c(c1)OCO2 ZINC000217828059 IF In-Stock Unstable SCN9A 0 40 O=C(CN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCc1ccc2c(c1)OCO2 ZINC000217828059 IF In-Stock Unstable NOS2 86 35 O=C(O)/C=C\c1cc(F)ccc1CN1CCC(O)CC1 ZINC000217828060 CD For-Sale Unstable SIGMAR1 24 43 O=C(O)/C=C\c1cc(F)ccc1CN1CCC(O)CC1 ZINC000217828060 CD For-Sale Unstable CCR3 25 41 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)c3cccc(C(F)(F)F)c3)C2)n1 ZINC000217828067 IK In-Stock Unstable HRH3 16 47 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)c3cccc(C(F)(F)F)c3)C2)n1 ZINC000217828067 IK In-Stock Unstable CCR2 58 39 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)c3cccc(C(F)(F)F)c3)C2)n1 ZINC000217828067 IK In-Stock Unstable Q8MHZ5_SHEEP 41 31 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)c3cccc(C(F)(F)F)c3)C2)n1 ZINC000217828067 IK In-Stock Unstable MAP3K12 34 43 Cc1cc(C(=O)N[C@H]2C[C@@H](C)CC[C@H]2C(C)C)ccc1N ZINC000217828083 CH For-Sale Unstable TRPM8 21 68 C[C@@H](c1ccc(Cl)cc1)N(C)[C@H](C)C(N)=O ZINC000217828086 BE On-Demand Unstable CHRNA4 0 42 C[C@@H](c1ccc(Cl)cc1)N(C)[C@H](C)C(N)=O ZINC000217828086 BE On-Demand Unstable UTS2 49 37 O=C(CN1CCC[C@@H](O)C1)NCc1cc2cc(F)ccc2[nH]1 ZINC000217828117 DD In-Stock Unstable PYGL 24 41 O=C(CN1CCC[C@@H](O)C1)NCc1cc2cc(F)ccc2[nH]1 ZINC000217828117 DD In-Stock Unstable PLD2 40 38 CCc1nc2ccc(C(=O)NC[C@H]3CCCN3c3ccccc3)cc2s1 ZINC000217828133 FI For-Sale Unstable LCK 27 43 O=C(CN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCc1ccc2c(c1)OCO2 ZINC000217828137 IF In-Stock Unstable SCN9A 0 40 O=C(CN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCc1ccc2c(c1)OCO2 ZINC000217828137 IF In-Stock Unstable NOS2 86 35 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)c3cccc(C(F)(F)F)c3)C2)n1 ZINC000217828138 IK In-Stock Unstable HRH3 16 47 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)c3cccc(C(F)(F)F)c3)C2)n1 ZINC000217828138 IK In-Stock Unstable CCR2 58 39 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)c3cccc(C(F)(F)F)c3)C2)n1 ZINC000217828138 IK In-Stock Unstable Q8MHZ5_SHEEP 41 31 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)c3cccc(C(F)(F)F)c3)C2)n1 ZINC000217828138 IK In-Stock Unstable MAP3K12 34 43 C[C@@H](c1ccccc1Cl)N(C)[C@H](C)C(N)=O ZINC000217828168 BE On-Demand Unstable CXCL8 34 45 O=C(O)/C=C\c1cc(CN2CCC(O)CC2)ccc1F ZINC000217828191 CD For-Sale Unstable SIGMAR1 37 47 O=C(O)/C=C\c1cc(CN2CCC(O)CC2)ccc1F ZINC000217828191 CD For-Sale Unstable CCR1 0 41 O=C(O)/C=C\c1cc(CN2CCC(O)CC2)ccc1F ZINC000217828191 CD For-Sale Unstable CCR3 31 42 O=C(O)/C=C\c1cc(CN2CCC(O)CC2)ccc1F ZINC000217828191 CD For-Sale Unstable MCHR1 38 42 O=C(CN1CCC[C@H](O)C1)NCc1cc2cc(F)ccc2[nH]1 ZINC000217828192 DD In-Stock Unstable PYGL 24 41 O=C(CN1CCC[C@H](O)C1)NCc1cc2cc(F)ccc2[nH]1 ZINC000217828192 DD In-Stock Unstable PLD2 40 38 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)[C@@H]1CSCN1 ZINC000217828197 CE For-Sale Unstable TRPM8 19 47 CC[C@@H](NC(=O)COc1ccccc1C)c1ccc(C)cc1C ZINC000217828201 DI In-Stock Unstable CETP 0 43 CC[C@@H](NC(=O)COc1ccccc1C)c1ccc(C)cc1C ZINC000217828201 DI In-Stock Unstable CTSA 47 33 CNC(=O)[C@@H]1CCCN1[C@@H](C)c1ccc(OC)cc1O ZINC000217828220 CD For-Sale Unstable MMP13 18 40 CNC(=O)[C@@H]1CCCN1[C@@H](C)c1ccc(OC)cc1O ZINC000217828220 CD For-Sale Unstable MMP3 24 40 CNC(=O)[C@@H]1CCCN1[C@@H](C)c1ccc(OC)cc1O ZINC000217828220 CD For-Sale Unstable MMP1 21 40 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)/C=C\c3ccc4c(c3)OCO4)C2)n1 ZINC000217828245 II In-Stock Unstable SSTR3 48 31 CC(=O)Nc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217828254 EG For-Sale Unstable DRD2 25 40 CC(=O)Nc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217828254 EG For-Sale Unstable AVPR2 43 40 CC(=O)Nc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217828254 EG For-Sale Unstable NPY2R 19 43 CC(=O)Nc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217828254 EG For-Sale Unstable PRNP 51 39 CC(=O)Nc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217828254 EG For-Sale Unstable EPHX2 15 42 CC(=O)Nc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217828254 EG For-Sale Unstable NOD2 41 34 CC(=O)Nc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217828254 EG For-Sale Unstable ACKR3 48 33 C[C@@H](c1cccc(Cl)c1)N(C)[C@H](C)C(N)=O ZINC000217828270 BE On-Demand Unstable ADRB1 18 40 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)[C@@H]1CSCN1 ZINC000217828277 CE For-Sale Unstable TRPM8 19 47 CC[C@H](NC(=O)COc1ccccc1C)c1ccc(C)cc1C ZINC000217828296 DI In-Stock Unstable CETP 0 43 CC[C@H](NC(=O)COc1ccccc1C)c1ccc(C)cc1C ZINC000217828296 DI In-Stock Unstable CTSA 47 33 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)/C=C\c3ccc4c(c3)OCO4)C2)n1 ZINC000217828305 II In-Stock Unstable SSTR3 48 31 CN1CCCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217828314 CD For-Sale Unstable ACHE 19 41 CN1CCCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217828314 CD For-Sale Unstable SIGMAR1 46 45 CN1CCCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217828314 CD For-Sale Unstable HDAC1 18 42 CN1CCCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217828314 CD For-Sale Unstable AKR1C3 31 40 CNC(=O)[C@@H]1CCCN1[C@@H](C)c1ccc(C)cc1O ZINC000217828317 CD For-Sale Unstable XPNPEP1 0 41 CNC(=O)[C@@H]1CCCN1[C@@H](C)c1ccc(C)cc1O ZINC000217828317 CD For-Sale Unstable XPNPEP2 0 41 CCC[C@@H](N)C(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217828321 BE For-Sale Unstable ACE 21 43 CCC[C@@H](N)C(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217828321 BE For-Sale Unstable DPP4 28 53 CCC[C@@H](N)C(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217828321 BE For-Sale Unstable DPP7 67 63 CCC[C@@H](N)C(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217828321 BE For-Sale Unstable TPP2 51 48 CCC[C@@H](N)C(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217828321 BE For-Sale Unstable DPP8 33 53 CCC[C@@H](N)C(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217828321 BE For-Sale Unstable DPP9 23 53 CCC[C@@H](N)C(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217828321 BE For-Sale Unstable FAP 0 53 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)[C@@H]1CSCN1 ZINC000217828347 CE For-Sale Unstable TRPM8 19 47 CC(=O)Nc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217828349 EG For-Sale Unstable DRD2 25 40 CC(=O)Nc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217828349 EG For-Sale Unstable AVPR2 43 40 CC(=O)Nc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217828349 EG For-Sale Unstable NPY2R 19 43 CC(=O)Nc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217828349 EG For-Sale Unstable PRNP 51 39 CC(=O)Nc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217828349 EG For-Sale Unstable EPHX2 15 42 CC(=O)Nc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217828349 EG For-Sale Unstable NOD2 41 34 CC(=O)Nc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217828349 EG For-Sale Unstable ACKR3 48 33 CN1CCN(C(=O)C[C@H](c2ccc3c(c2)OCO3)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)CC1 ZINC000217828352 KH In-Stock Unstable RORC 0 46 CCC[C@H](N)C(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217828393 BE On-Demand Unstable DPP4 22 49 CCC[C@H](N)C(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217828393 BE On-Demand Unstable DPP7 56 53 CCC[C@H](N)C(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217828393 BE On-Demand Unstable TPP2 57 48 CCC[C@H](N)C(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217828393 BE On-Demand Unstable DPP8 35 53 CCC[C@H](N)C(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217828393 BE On-Demand Unstable FAP 0 53 O=C(N/C=C/c1ccccc1Cl)N1CCN(c2ccccn2)CC1 ZINC000217828412 EG For-Sale Unstable DRD4 27 41 O=C(N/C=C/c1ccccc1Cl)N1CCN(c2ccccn2)CC1 ZINC000217828412 EG For-Sale Unstable EBP 21 41 O=C(N/C=C/c1ccccc1Cl)N1CCN(c2ccccn2)CC1 ZINC000217828412 EG For-Sale Unstable SLC6A7 0 45 CC[C@@H](NC(=O)COc1ccccc1C)c1ccc(OC)c(OC)c1 ZINC000217828416 EH In-Stock Unstable ENPP1 49 35 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)[C@@H]1CSCN1 ZINC000217828417 CE For-Sale Unstable TRPM8 19 47 CN1CCN(C(=O)C[C@@H](c2ccc3c(c2)OCO3)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)CC1 ZINC000217828434 KH In-Stock Unstable RORC 43 46 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)COc3ccccc3F)C2)n1 ZINC000217828435 HI In-Stock Unstable HRH3 21 44 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)COc3ccccc3F)C2)n1 ZINC000217828435 HI In-Stock Unstable COLA 44 37 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)COc3ccccc3F)C2)n1 ZINC000217828435 HI In-Stock Unstable CPT1A 42 37 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)COc3ccccc3F)C2)n1 ZINC000217828435 HI In-Stock Unstable Q8MHZ5_SHEEP 46 32 COCCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217828448 FG For-Sale Unstable DRD2 31 45 COCCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217828448 FG For-Sale Unstable DRD3 24 40 COCCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217828448 FG For-Sale Unstable GRIN2B 20 47 COCCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217828448 FG For-Sale Unstable LTA4H 38 42 COCCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217828448 FG For-Sale Unstable HCRTR1 17 42 COCCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217828448 FG For-Sale Unstable CYSLTR2 44 36 COCCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217828448 FG For-Sale Unstable COLA 43 34 COCCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217828448 FG For-Sale Unstable CPT1A 45 34 COCCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217828448 FG For-Sale Unstable ITGA4 43 33 COCCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217828448 FG For-Sale Unstable CHRNA10 51 41 COCCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217828448 FG For-Sale Unstable HCRTR2 15 42 COCCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217828448 FG For-Sale Unstable CACNA1I 40 31 COCCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217828448 FG For-Sale Unstable ACKR3 65 35 CNC(=O)[C@@H]1CCCN1[C@@H](C)c1ccc(O)cc1 ZINC000217828463 BD For-Sale Unstable XIAP 43 35 CCC[C@@H](N)C(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217828465 BE For-Sale Unstable ACE 21 43 CCC[C@@H](N)C(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217828465 BE For-Sale Unstable DPP4 28 53 CCC[C@@H](N)C(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217828465 BE For-Sale Unstable DPP7 67 63 CCC[C@@H](N)C(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217828465 BE For-Sale Unstable TPP2 51 48 CCC[C@@H](N)C(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217828465 BE For-Sale Unstable DPP8 33 53 CCC[C@@H](N)C(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217828465 BE For-Sale Unstable DPP9 23 53 CCC[C@@H](N)C(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217828465 BE For-Sale Unstable FAP 0 53 Cc1nn(Cc2ccccc2)c2sc(C(=O)N3CCN(Cc4cccnc4)CC3)cc12 ZINC000217828497 IH On-Demand Unstable FAAH 21 40 CC[C@H](NC(=O)COc1ccccc1C)c1ccc(OC)c(OC)c1 ZINC000217828500 EH In-Stock Unstable ENPP1 49 35 COCCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217828511 FG For-Sale Unstable DRD2 31 45 COCCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217828511 FG For-Sale Unstable DRD3 24 40 COCCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217828511 FG For-Sale Unstable GRIN2B 20 47 COCCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217828511 FG For-Sale Unstable LTA4H 38 42 COCCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217828511 FG For-Sale Unstable HCRTR1 17 42 COCCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217828511 FG For-Sale Unstable CYSLTR2 44 36 COCCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217828511 FG For-Sale Unstable COLA 43 34 COCCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217828511 FG For-Sale Unstable CPT1A 45 34 COCCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217828511 FG For-Sale Unstable ITGA4 43 33 COCCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217828511 FG For-Sale Unstable CHRNA10 51 41 COCCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217828511 FG For-Sale Unstable HCRTR2 15 42 COCCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217828511 FG For-Sale Unstable CACNA1I 40 31 COCCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217828511 FG For-Sale Unstable ACKR3 65 35 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)COc3ccccc3F)C2)n1 ZINC000217828513 HI In-Stock Unstable HRH3 21 44 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)COc3ccccc3F)C2)n1 ZINC000217828513 HI In-Stock Unstable COLA 44 37 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)COc3ccccc3F)C2)n1 ZINC000217828513 HI In-Stock Unstable CPT1A 42 37 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)COc3ccccc3F)C2)n1 ZINC000217828513 HI In-Stock Unstable Q8MHZ5_SHEEP 46 32 CCC[C@@H](N)C(=O)N[C@@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217828530 CF For-Sale Unstable TRPM8 18 49 CN1CCCN(Cc2ccc(F)c(/C=C\C(=O)O)c2)CC1 ZINC000217828558 CE For-Sale Unstable CCR1 17 42 CCC[C@H](N)C(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217828566 BE On-Demand Unstable DPP4 22 49 CCC[C@H](N)C(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217828566 BE On-Demand Unstable DPP7 56 53 CCC[C@H](N)C(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217828566 BE On-Demand Unstable TPP2 57 48 CCC[C@H](N)C(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217828566 BE On-Demand Unstable DPP8 35 53 CCC[C@H](N)C(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217828566 BE On-Demand Unstable FAP 0 53 Cc1ccc(-c2csc(NC(=O)CCn3c(=O)n(C)c4ccccc43)n2)cc1[N+](=O)[O-] ZINC000217828605 IH On-Demand Unstable HDAC9 16 45 Cc1ccc(-c2csc(NC(=O)CCn3c(=O)n(C)c4ccccc43)n2)cc1[N+](=O)[O-] ZINC000217828605 IH On-Demand Unstable TRPA1 21 41 CCC[C@H](N)C(=O)N[C@@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217828613 CF For-Sale Unstable TRPM8 20 50 CC[C@@H](C)c1ccc(OCc2cccc(Br)c2)cc1 ZINC000217828614 DK For-Sale Unstable MAOB 46 50 CC[C@@H](C)c1ccc(OCc2cccc(Br)c2)cc1 ZINC000217828614 DK For-Sale Unstable ADAMTS4 22 50 CC[C@@H](C)c1ccc(OCc2cccc(Br)c2)cc1 ZINC000217828614 DK For-Sale Unstable FFAR1 38 51 OCc1cc2n(n1)CCN(CCc1c[nH]c3ccccc13)C2 ZINC000217828623 CD In-Stock Unstable HTR1D 81 41 OCc1cc2n(n1)CCN(CCc1c[nH]c3ccccc13)C2 ZINC000217828623 CD In-Stock Unstable HTR1B 79 41 OCc1cc2n(n1)CCN(CCc1c[nH]c3ccccc13)C2 ZINC000217828623 CD In-Stock Unstable MPO 16 40 COc1ccc(CCN2C(=O)N[C@@H](CCC(=O)NCCc3ccc(O)cc3)C2=O)cc1OC ZINC000217828627 JE In-Stock Unstable IAP 0 41 COc1ccc(CCN2C(=O)N[C@@H](CCC(=O)NCCc3ccc(O)cc3)C2=O)cc1OC ZINC000217828627 JE In-Stock Unstable CAN2 0 48 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)Cc3cccs3)C2)n1 ZINC000217828628 GI In-Stock Unstable ETHR 37 49 O=C(CCCCCN1C(=O)c2ccccc2C1=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217828630 HH For-Sale Unstable HTR1A 21 47 O=C(CCCCCN1C(=O)c2ccccc2C1=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217828630 HH For-Sale Unstable HTR7 40 39 O=C(CCCCCN1C(=O)c2ccccc2C1=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217828630 HH For-Sale Unstable HDAC10 17 43 O=C(CCCCCN1C(=O)c2ccccc2C1=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217828630 HH For-Sale Unstable HDAC3 16 43 CC[C@@H]1CCCCN1Cc1ccccc1/C=C\C(=O)O ZINC000217828664 CH For-Sale Unstable PTGER2 38 42 CC[C@@H]1CCCCN1Cc1ccccc1/C=C\C(=O)O ZINC000217828664 CH For-Sale Unstable PTGER4 0 42 CC[C@@H]1CCCCN1Cc1ccccc1/C=C\C(=O)O ZINC000217828664 CH For-Sale Unstable PTGER3 15 42 CC[C@@H]1CCCCN1Cc1ccccc1/C=C\C(=O)O ZINC000217828664 CH For-Sale Unstable PTGDR 0 41 CC[C@H](C)c1ccc(OCc2cccc(Br)c2)cc1 ZINC000217828677 DK For-Sale Unstable MAOB 46 50 CC[C@H](C)c1ccc(OCc2cccc(Br)c2)cc1 ZINC000217828677 DK For-Sale Unstable ADAMTS4 22 50 CC[C@H](C)c1ccc(OCc2cccc(Br)c2)cc1 ZINC000217828677 DK For-Sale Unstable FFAR1 38 51 CCC[C@@H](N)C(=O)N[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217828682 CF For-Sale Unstable TRPM8 18 49 CNC(=O)[C@@H]1CCCN1[C@@H](C)Cc1ccc(O)cc1 ZINC000217828686 CD For-Sale Unstable F2 25 40 CNC(=O)[C@@H]1CCCN1[C@@H](C)Cc1ccc(O)cc1 ZINC000217828686 CD For-Sale Unstable ACE 44 42 CNC(=O)[C@@H]1CCCN1[C@@H](C)Cc1ccc(O)cc1 ZINC000217828686 CD For-Sale Unstable OPRM1 43 46 CNC(=O)[C@@H]1CCCN1[C@@H](C)Cc1ccc(O)cc1 ZINC000217828686 CD For-Sale Unstable OPRD1 23 45 CNC(=O)[C@@H]1CCCN1[C@@H](C)Cc1ccc(O)cc1 ZINC000217828686 CD For-Sale Unstable OPRK1 0 40 CNC(=O)[C@@H]1CCCN1[C@@H](C)Cc1ccc(O)cc1 ZINC000217828686 CD For-Sale Unstable NTSR1 101 35 CNC(=O)[C@@H]1CCCN1[C@@H](C)Cc1ccc(O)cc1 ZINC000217828686 CD For-Sale Unstable NTSR2 73 33 CNC(=O)[C@@H]1CCCN1[C@@H](C)Cc1ccc(O)cc1 ZINC000217828686 CD For-Sale Unstable HLA-A 50 36 CNC(=O)[C@@H]1CCCN1[C@@H](C)Cc1ccc(O)cc1 ZINC000217828686 CD For-Sale Unstable LGMN 68 35 CNC(=O)[C@@H]1CCCN1[C@@H](C)Cc1ccc(O)cc1 ZINC000217828686 CD For-Sale Unstable SORT1 49 33 CNC(=O)[C@@H]1CCCN1[C@@H](C)Cc1ccc(O)cc1 ZINC000217828686 CD For-Sale Unstable YARS 50 32 CNC(=O)[C@@H]1CCCN1[C@@H](C)Cc1ccc(O)cc1 ZINC000217828686 CD For-Sale Unstable MARS 48 35 CNC(=O)[C@@H]1CCCN1[C@@H](C)Cc1ccc(O)cc1 ZINC000217828686 CD For-Sale Unstable XIAP 48 45 CNC(=O)[C@@H]1CCCN1[C@@H](C)Cc1ccc(O)cc1 ZINC000217828686 CD For-Sale Unstable BRCA1 52 33 O=C(CCCCCN1C(=O)c2ccccc2C1=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217828696 HH For-Sale Unstable HTR1A 21 47 O=C(CCCCCN1C(=O)c2ccccc2C1=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217828696 HH For-Sale Unstable HTR7 40 39 O=C(CCCCCN1C(=O)c2ccccc2C1=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217828696 HH For-Sale Unstable HDAC10 17 43 O=C(CCCCCN1C(=O)c2ccccc2C1=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217828696 HH For-Sale Unstable HDAC3 16 43 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)Cc3cccs3)C2)n1 ZINC000217828709 GI In-Stock Unstable ETHR 37 49 CC[C@H]1CCCCN1Cc1ccccc1/C=C\C(=O)O ZINC000217828719 CH For-Sale Unstable PTGER2 38 42 CC[C@H]1CCCCN1Cc1ccccc1/C=C\C(=O)O ZINC000217828719 CH For-Sale Unstable PTGER4 0 42 CC[C@H]1CCCCN1Cc1ccccc1/C=C\C(=O)O ZINC000217828719 CH For-Sale Unstable PTGER3 15 42 CC[C@H]1CCCCN1Cc1ccccc1/C=C\C(=O)O ZINC000217828719 CH For-Sale Unstable PTGDR 0 41 CCCN(CC)CCNC(=O)[C@@H]1CCC[C@@H]1C(=O)O ZINC000217828722 CD For-Sale Unstable ACE 0 44 CCC[C@@H](N)CN1C[C@H](C)O[C@@H](C)C1 ZINC000217828723 BD For-Sale Unstable ZM.86993 0 47 CCC[C@@H](N)CN1C[C@H](C)O[C@@H](C)C1 ZINC000217828723 BD For-Sale Unstable Q2TU57_MAIZE 23 47 C[C@@H](c1ccc(Cl)cc1)N(C)C[C@@H](N)C(=O)O ZINC000217828750 CD For-Sale Unstable CACNA2D1 26 44 C[C@@H](c1ccc(Cl)cc1)N(C)C[C@@H](N)C(=O)O ZINC000217828750 CD For-Sale Unstable CHRNA4 0 42 C[C@@H](c1ccc(Cl)cc1)N(C)C[C@@H](N)C(=O)O ZINC000217828750 CD For-Sale Unstable GRIK3 38 40 C[C@@H](c1ccc(Cl)cc1)N(C)C[C@@H](N)C(=O)O ZINC000217828750 CD For-Sale Unstable GRIK1 42 40 C[C@@H](c1ccc(Cl)cc1)N(C)C[C@@H](N)C(=O)O ZINC000217828750 CD For-Sale Unstable KIF11 0 40 C[C@@H](c1ccc(Cl)cc1)N(C)C[C@@H](N)C(=O)O ZINC000217828750 CD For-Sale Unstable UTS2 46 37 Cc1nn(-c2ccc(Cl)cc2)c2sc(C(=O)N3CCN(Cc4cccnc4)CC3)cc12 ZINC000217828751 JI On-Demand Unstable FAAH 21 42 CCC[C@H](N)C(=O)N[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217828774 CF For-Sale Unstable TRPM8 18 49 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)c3ccco3)C2)n1 ZINC000217828793 FH In-Stock Unstable HRH3 21 43 CCCN(CC)CCNC(=O)[C@H]1CCC[C@@H]1C(=O)O ZINC000217828797 CD For-Sale Unstable ACE 0 44 COc1ccc(-c2noc(CNC(=O)COc3ccccc3C)n2)c(OC)c1 ZINC000217828814 GF In-Stock Unstable MTNR1A 63 38 COc1ccc(-c2noc(CNC(=O)COc3ccccc3C)n2)c(OC)c1 ZINC000217828814 GF In-Stock Unstable MTNR1B 54 38 CCC[C@H](N)CN1C[C@H](C)O[C@@H](C)C1 ZINC000217828825 BD For-Sale Unstable ZM.86993 0 47 CCC[C@H](N)CN1C[C@H](C)O[C@@H](C)C1 ZINC000217828825 BD For-Sale Unstable Q2TU57_MAIZE 23 47 C[C@H](c1ccc(Cl)cc1)N(C)C[C@@H](N)C(=O)O ZINC000217828834 CD For-Sale Unstable CACNA2D1 26 44 C[C@H](c1ccc(Cl)cc1)N(C)C[C@@H](N)C(=O)O ZINC000217828834 CD For-Sale Unstable CHRNA4 0 42 C[C@H](c1ccc(Cl)cc1)N(C)C[C@@H](N)C(=O)O ZINC000217828834 CD For-Sale Unstable GRIK3 38 40 C[C@H](c1ccc(Cl)cc1)N(C)C[C@@H](N)C(=O)O ZINC000217828834 CD For-Sale Unstable GRIK1 42 40 C[C@H](c1ccc(Cl)cc1)N(C)C[C@@H](N)C(=O)O ZINC000217828834 CD For-Sale Unstable KIF11 0 40 C[C@H](c1ccc(Cl)cc1)N(C)C[C@@H](N)C(=O)O ZINC000217828834 CD For-Sale Unstable UTS2 46 37 COC(=O)CNC(=O)N/C=C/c1ccccc1Cl ZINC000217828842 CD For-Sale Unstable TLR4 16 45 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)Nc3cccc(O)c3)[C@H]21 ZINC000217828854 JG In-Stock Unstable TSHR 50 33 Cc1cc(N[C@@H]2CCc3ccccc32)ncn1 ZINC000217828863 BF On-Demand Unstable KCNN3 22 44 C/C=C/C=C\C(=O)N[C@@H](C)C(=O)OCC ZINC000217828865 BD On-Demand Unstable METAP2 24 42 C[C@@H]1Cc2ccccc2N1S(=O)(=O)c1cccc(C(=O)N2CCN(Cc3cccnc3)CC2)c1 ZINC000217828871 JG On-Demand Unstable DRD4 30 42 C[C@@H]1Cc2ccccc2N1S(=O)(=O)c1cccc(C(=O)N2CCN(Cc3cccnc3)CC2)c1 ZINC000217828871 JG On-Demand Unstable AKR1C3 30 42 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)c3ccco3)C2)n1 ZINC000217828878 FH In-Stock Unstable HRH3 21 43 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)[C@@H]1C[C@@H](O)CN1 ZINC000217828896 CD For-Sale Unstable TRPM8 17 47 CNC(=O)[C@@H]1CCCN1[C@@H](C)CCc1ccc(O)cc1 ZINC000217828914 CD For-Sale Unstable F2 15 40 CNC(=O)[C@@H]1CCCN1[C@@H](C)CCc1ccc(O)cc1 ZINC000217828914 CD For-Sale Unstable ACE 42 50 CNC(=O)[C@@H]1CCCN1[C@@H](C)CCc1ccc(O)cc1 ZINC000217828914 CD For-Sale Unstable FKBP1A 20 40 CNC(=O)[C@@H]1CCCN1[C@@H](C)CCc1ccc(O)cc1 ZINC000217828914 CD For-Sale Unstable OPRM1 32 42 CNC(=O)[C@@H]1CCCN1[C@@H](C)CCc1ccc(O)cc1 ZINC000217828914 CD For-Sale Unstable MME 15 40 CNC(=O)[C@@H]1CCCN1[C@@H](C)CCc1ccc(O)cc1 ZINC000217828914 CD For-Sale Unstable XPNPEP1 0 48 CNC(=O)[C@@H]1CCCN1[C@@H](C)CCc1ccc(O)cc1 ZINC000217828914 CD For-Sale Unstable NTSR1 98 35 CNC(=O)[C@@H]1CCCN1[C@@H](C)CCc1ccc(O)cc1 ZINC000217828914 CD For-Sale Unstable NTSR2 85 33 CNC(=O)[C@@H]1CCCN1[C@@H](C)CCc1ccc(O)cc1 ZINC000217828914 CD For-Sale Unstable HLA-A 47 34 CNC(=O)[C@@H]1CCCN1[C@@H](C)CCc1ccc(O)cc1 ZINC000217828914 CD For-Sale Unstable LGMN 65 34 CNC(=O)[C@@H]1CCCN1[C@@H](C)CCc1ccc(O)cc1 ZINC000217828914 CD For-Sale Unstable SORT1 48 33 CNC(=O)[C@@H]1CCCN1[C@@H](C)CCc1ccc(O)cc1 ZINC000217828914 CD For-Sale Unstable XPNPEP2 0 48 CNC(=O)[C@@H]1CCCN1[C@@H](C)CCc1ccc(O)cc1 ZINC000217828914 CD For-Sale Unstable XIAP 54 41 CNC(=O)[C@@H]1CCCN1[C@@H](C)CCc1ccc(O)cc1 ZINC000217828914 CD For-Sale Unstable BIRC2 67 44 C[C@@H](c1ccccc1Cl)N(C)C[C@@H](N)C(=O)O ZINC000217828919 CD For-Sale Unstable CACNA2D1 25 40 C[C@@H](c1ccccc1Cl)N(C)C[C@@H](N)C(=O)O ZINC000217828919 CD For-Sale Unstable CXCL8 44 40 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)Nc3cccc(O)c3)[C@@H]21 ZINC000217828924 JG In-Stock Unstable TSHR 50 33 COC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217828946 EH For-Sale Unstable PPIA 18 43 COC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217828946 EH For-Sale Unstable IMDH_CRYPV 42 34 COC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217828946 EH For-Sale Unstable KCNK3 93 40 COC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217828946 EH For-Sale Unstable KCNK9 58 34 C[C@H]1Cc2ccccc2N1S(=O)(=O)c1cccc(C(=O)N2CCN(Cc3cccnc3)CC2)c1 ZINC000217828952 JG On-Demand Unstable DRD4 30 42 C[C@H]1Cc2ccccc2N1S(=O)(=O)c1cccc(C(=O)N2CCN(Cc3cccnc3)CC2)c1 ZINC000217828952 JG On-Demand Unstable AKR1C3 30 42 C[C@@H](Cn1cncn1)NC(=O)C(=O)c1ccco1 ZINC000217828955 BC In-Stock Unstable HIS3 87 43 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)[C@@H]1C[C@@H](O)CN1 ZINC000217828970 CD For-Sale Unstable TRPM8 17 47 COc1cccc(C(=O)NCC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217828993 FE For-Sale Unstable DRD4 57 43 COc1cccc(C(=O)NCC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217828993 FE For-Sale Unstable DRD3 24 52 COc1cccc(C(=O)NCC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217828993 FE For-Sale Unstable CCR3 15 44 COc1cccc(C(=O)NCC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217828993 FE For-Sale Unstable PREP 21 42 COc1cccc(C(=O)NCC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217828993 FE For-Sale Unstable MTNR1B 36 43 COc1cccc(C(=O)NCC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217828993 FE For-Sale Unstable CCR2 53 47 COc1cccc(C(=O)NCC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217828993 FE For-Sale Unstable CHRNA10 41 41 COc1cccc(C(=O)NCC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217828993 FE For-Sale Unstable MCHR1 20 45 COc1cccc(C(=O)NCC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217828993 FE For-Sale Unstable ACKR3 68 37 C[C@H](c1ccccc1Cl)N(C)C[C@@H](N)C(=O)O ZINC000217829005 CD For-Sale Unstable CACNA2D1 25 40 C[C@H](c1ccccc1Cl)N(C)C[C@@H](N)C(=O)O ZINC000217829005 CD For-Sale Unstable CXCL8 44 40 CNC(=O)[C@@H]1CCCN1[C@@H](C)c1ccccc1O ZINC000217829021 BD For-Sale Unstable XPNPEP1 0 43 CNC(=O)[C@@H]1CCCN1[C@@H](C)c1ccccc1O ZINC000217829021 BD For-Sale Unstable XPNPEP2 0 43 CNC(=O)[C@@H]1CCCN1[C@@H](C)c1ccccc1O ZINC000217829021 BD For-Sale Unstable XIAP 43 37 COc1ccc([C@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c(OC)c1 ZINC000217829028 KH In-Stock Unstable PRKDC 24 40 COc1ccc([C@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c(OC)c1 ZINC000217829028 KH In-Stock Unstable CYP1B1 45 36 COc1ccc([C@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c(OC)c1 ZINC000217829028 KH In-Stock Unstable RORC 0 43 C[C@H](Cn1cncn1)NC(=O)C(=O)c1ccco1 ZINC000217829034 BC In-Stock Unstable HIS3 87 43 CCOC(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2Cl)cc1 ZINC000217829047 FH For-Sale Unstable P2RY12 21 40 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)[C@@H]1C[C@@H](O)CN1 ZINC000217829051 CD For-Sale Unstable TRPM8 17 47 COc1cccc(C(=O)NCC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217829074 FE For-Sale Unstable DRD4 57 43 COc1cccc(C(=O)NCC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217829074 FE For-Sale Unstable DRD3 24 52 COc1cccc(C(=O)NCC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217829074 FE For-Sale Unstable CCR3 15 44 COc1cccc(C(=O)NCC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217829074 FE For-Sale Unstable PREP 21 42 COc1cccc(C(=O)NCC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217829074 FE For-Sale Unstable MTNR1B 36 43 COc1cccc(C(=O)NCC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217829074 FE For-Sale Unstable CCR2 53 47 COc1cccc(C(=O)NCC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217829074 FE For-Sale Unstable CHRNA10 41 41 COc1cccc(C(=O)NCC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217829074 FE For-Sale Unstable MCHR1 20 45 COc1cccc(C(=O)NCC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217829074 FE For-Sale Unstable ACKR3 68 37 C[C@@H](c1cccc(Cl)c1)N(C)C[C@@H](N)C(=O)O ZINC000217829099 CD For-Sale Unstable CACNA2D1 26 54 C[C@@H](c1cccc(Cl)c1)N(C)C[C@@H](N)C(=O)O ZINC000217829099 CD For-Sale Unstable GRIK1 23 42 C[C@@H](c1cccc(Cl)c1)N(C)C[C@@H](N)C(=O)O ZINC000217829099 CD For-Sale Unstable AOC3 23 45 C[C@@H](c1cccc(Cl)c1)N(C)C[C@@H](N)C(=O)O ZINC000217829099 CD For-Sale Unstable KIF11 32 47 COc1ccc([C@@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c(OC)c1 ZINC000217829107 KH In-Stock Unstable PRKDC 24 40 COc1ccc([C@@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c(OC)c1 ZINC000217829107 KH In-Stock Unstable CYP1B1 45 36 COc1ccc([C@@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c(OC)c1 ZINC000217829107 KH In-Stock Unstable RORC 52 43 O=S(=O)(Cl)Cc1ccccc1OC1CC1 ZINC000217829114 BE For-Sale Unstable SLC5A4 53 33 COC(=O)c1ccccc1C(=O)N1CCC[C@@H](Cc2nc(-c3ccccc3C)no2)C1 ZINC000217829144 HH In-Stock Unstable HRH3 17 44 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)[C@@H]1C[C@@H](O)CN1 ZINC000217829157 CD For-Sale Unstable TRPM8 17 47 C[C@@H](NS(=O)(=O)c1cccc(C(=O)N(C)C2CCCCCC2)c1)c1ccccc1 ZINC000217829164 HJ On-Demand Unstable F2 22 44 Cc1ccccc1OCC(=O)NCCCc1ccc(C(C)C)cc1 ZINC000217829175 EI In-Stock Unstable CYSP_TRYCR 0 48 Cc1ccccc1OCC(=O)NCCCc1ccc(C(C)C)cc1 ZINC000217829175 EI In-Stock Unstable CRTM 43 43 Cc1ccccc1OCC(=O)NCCCc1ccc(C(C)C)cc1 ZINC000217829175 EI In-Stock Unstable ACAT 0 41 CN1CCC(C(=O)NC[C@@H]2CCCN2c2ccccc2)CC1 ZINC000217829178 DE For-Sale Unstable SLC6A1 45 33 C[C@H](c1cccc(Cl)c1)N(C)C[C@@H](N)C(=O)O ZINC000217829202 CD For-Sale Unstable CACNA2D1 26 54 C[C@H](c1cccc(Cl)c1)N(C)C[C@@H](N)C(=O)O ZINC000217829202 CD For-Sale Unstable GRIK1 23 42 C[C@H](c1cccc(Cl)c1)N(C)C[C@@H](N)C(=O)O ZINC000217829202 CD For-Sale Unstable AOC3 23 45 C[C@H](c1cccc(Cl)c1)N(C)C[C@@H](N)C(=O)O ZINC000217829202 CD For-Sale Unstable KIF11 32 47 COC(=O)c1ccccc1C(=O)N1CCC[C@H](Cc2nc(-c3ccccc3C)no2)C1 ZINC000217829214 HH In-Stock Unstable HRH3 17 44 CNC(=O)[C@@H]1CCCN1[C@@H](C)c1cc(C)ccc1O ZINC000217829219 CD For-Sale Unstable XPNPEP1 0 41 CNC(=O)[C@@H]1CCCN1[C@@H](C)c1cc(C)ccc1O ZINC000217829219 CD For-Sale Unstable XPNPEP2 0 41 C[C@H](NS(=O)(=O)c1cccc(C(=O)N(C)C2CCCCCC2)c1)c1ccccc1 ZINC000217829230 HJ On-Demand Unstable F2 22 44 O=S(=O)(Cl)CCc1cccc2c1CCO2 ZINC000217829233 BD For-Sale Unstable MTNR1B 15 41 CN1CCC(C(=O)NC[C@H]2CCCN2c2ccccc2)CC1 ZINC000217829254 DE For-Sale Unstable SLC6A1 45 33 Cc1ccc(CN(C)Cc2ccccc2/C=C\C(=O)O)o1 ZINC000217829264 CG For-Sale Unstable PTGER2 43 44 Cc1ccc(CN(C)Cc2ccccc2/C=C\C(=O)O)o1 ZINC000217829264 CG For-Sale Unstable PTGER4 22 44 Cc1ccc(CN(C)Cc2ccccc2/C=C\C(=O)O)o1 ZINC000217829264 CG For-Sale Unstable PTGER3 17 44 C[C@@H](c1ccccc1F)N(C)C[C@@H](N)C(=O)O ZINC000217829277 BD For-Sale Unstable CACNA2D1 32 51 Cc1ccccc1OCC(=O)NCCCN1CCCc2ccccc21 ZINC000217829288 EG In-Stock Unstable DRD2 27 41 Cc1ccccc1OCC(=O)NCCCN1CCCc2ccccc21 ZINC000217829288 EG In-Stock Unstable ADRA1D 25 42 Cc1ccccc1OCC(=O)NCCCN1CCCc2ccccc21 ZINC000217829288 EG In-Stock Unstable DRD3 40 41 Cc1ccccc1OCC(=O)NCCCN1CCCc2ccccc21 ZINC000217829288 EG In-Stock Unstable MTNR1C 0 42 O=C(NCC(=O)N1CCN(Cc2cccnc2)CC1)c1ccc(Br)cc1 ZINC000217829332 HD On-Demand Unstable PTAFR 35 57 O=C(NCC(=O)N1CCN(Cc2cccnc2)CC1)c1ccc(Br)cc1 ZINC000217829332 HD On-Demand Unstable CHRNA7 41 48 O=C(NCC(=O)N1CCN(Cc2cccnc2)CC1)c1ccc(Br)cc1 ZINC000217829332 HD On-Demand Unstable C3AR1 41 38 O=C(NCC(=O)N1CCN(Cc2cccnc2)CC1)c1ccc(Br)cc1 ZINC000217829332 HD On-Demand Unstable ACHP_LYMST 22 48 O=C(NCC(=O)N1CCN(Cc2cccnc2)CC1)c1ccc(Br)cc1 ZINC000217829332 HD On-Demand Unstable NAMPT 54 39 C[C@H](c1ccccc1F)N(C)C[C@@H](N)C(=O)O ZINC000217829351 BD For-Sale Unstable CACNA2D1 32 51 Cc1ccccc1CNC(=O)N/C=C/c1ccccc1Cl ZINC000217829371 DI For-Sale Unstable CXCL8 43 35 Cc1ccccc1CNC(=O)N/C=C/c1ccccc1Cl ZINC000217829371 DI For-Sale Unstable P2RX7 31 42 Cc1ccccc1CNC(=O)N/C=C/c1ccccc1Cl ZINC000217829371 DI For-Sale Unstable SCN10A 15 40 CC(C)Oc1cccc(CNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217829404 EH In-Stock Unstable MAOB 24 42 CC(C)Oc1cccc(CNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217829404 EH In-Stock Unstable ANPEP 18 40 CC(C)Oc1cccc(CNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217829404 EH In-Stock Unstable FDFT1 0 45 CC(C)Oc1cccc(CNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217829404 EH In-Stock Unstable GUAB 0 40 CC(C)Oc1cccc(CNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217829404 EH In-Stock Unstable FAAH 20 45 CC(C)Oc1cccc(CNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217829404 EH In-Stock Unstable AMP1_PLAFQ 30 42 CC(C)Oc1cccc(CNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217829404 EH In-Stock Unstable CRTM 48 45 CC(C)Oc1cccc(CNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217829404 EH In-Stock Unstable PDS 85 42 COC(=O)C[C@H](c1cc(Cl)c2c(c1)OCO2)c1c(O)c2ccccc2oc1=O ZINC000217829411 HH In-Stock Unstable NQO1 47 44 O=C(N[C@@H]1CN2CCC1CC2)c1ccc(=O)[nH]n1 ZINC000217829433 BB For-Sale Unstable HTR3A 24 52 O=C(N[C@@H]1CN2CCC1CC2)c1ccc(=O)[nH]n1 ZINC000217829433 BB For-Sale Unstable HTR4 15 47 O=C(N[C@@H]1CN2CCC1CC2)c1ccc(=O)[nH]n1 ZINC000217829433 BB For-Sale Unstable CHRNA7 25 57 CNC(=O)[C@@H]1CCCN1[C@@H](C)c1cc(Cl)ccc1O ZINC000217829443 CE For-Sale Unstable F2 17 42 Cc1ccc(CN(C)Cc2cccc(/C=C\C(=O)O)c2)o1 ZINC000217829482 CG For-Sale Unstable PTGER2 0 40 COC(=O)C[C@@H](c1cc(Cl)c2c(c1)OCO2)c1c(O)c2ccccc2oc1=O ZINC000217829492 HH In-Stock Unstable NQO1 47 44 O=C(N[C@H]1CN2CCC1CC2)c1ccc(=O)[nH]n1 ZINC000217829511 BB For-Sale Unstable HTR3A 24 52 O=C(N[C@H]1CN2CCC1CC2)c1ccc(=O)[nH]n1 ZINC000217829511 BB For-Sale Unstable HTR4 15 47 O=C(N[C@H]1CN2CCC1CC2)c1ccc(=O)[nH]n1 ZINC000217829511 BB For-Sale Unstable CHRNA7 25 57 COc1cc(CNC(=O)COc2ccc(Cl)cc2)ccc1OC(C)C ZINC000217829515 FH In-Stock Unstable TRPV1 27 43 COc1cc(CNC(=O)COc2ccc(Cl)cc2)ccc1OC(C)C ZINC000217829515 FH In-Stock Unstable PDE6A 44 35 COc1cc(CNC(=O)COc2ccc(Cl)cc2)ccc1OC(C)C ZINC000217829515 FH In-Stock Unstable MT-ND1 25 43 COc1cc(CNC(=O)COc2ccc(Cl)cc2)ccc1OC(C)C ZINC000217829515 FH In-Stock Unstable U38 0 44 COc1cc(CNC(=O)COc2ccc(Cl)cc2)ccc1OC(C)C ZINC000217829515 FH In-Stock Unstable DRTS_TRYCR 46 32 COc1cc(CNC(=O)COc2ccc(Cl)cc2)ccc1OC(C)C ZINC000217829515 FH In-Stock Unstable CAN2 0 40 CNC(=O)[C@@H]1CCCN1[C@@H](C)c1cccc(O)c1 ZINC000217829547 BD For-Sale Unstable XPNPEP1 0 41 CNC(=O)[C@@H]1CCCN1[C@@H](C)c1cccc(O)c1 ZINC000217829547 BD For-Sale Unstable XPNPEP2 0 41 O=C(NC[C@H]1CCCN1c1ccccc1)c1n[nH]c2cc(F)ccc12 ZINC000217829567 EG For-Sale Unstable HCRTR1 26 42 O=C(NC[C@H]1CCCN1c1ccccc1)c1n[nH]c2cc(F)ccc12 ZINC000217829567 EG For-Sale Unstable MC1R 20 41 O=C(NC[C@H]1CCCN1c1ccccc1)c1n[nH]c2cc(F)ccc12 ZINC000217829567 EG For-Sale Unstable HCRTR2 17 42 O=C(NC[C@H]1CCCN1c1ccccc1)c1n[nH]c2cc(F)ccc12 ZINC000217829567 EG For-Sale Unstable ACKR3 44 33 Cc1cccc(CNC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217829583 DI For-Sale Unstable ANPEP 17 46 CC(=O)c1cn(CCNC(=O)C[C@@H]2NC(=O)c3ccccc3NC2=O)c2ccccc12 ZINC000217829586 HE In-Stock Unstable CNR1 15 40 CC(=O)c1cn(CCNC(=O)C[C@@H]2NC(=O)c3ccccc3NC2=O)c2ccccc12 ZINC000217829586 HE In-Stock Unstable CNR2 23 40 O=C(COc1ccc(Cl)cc1)NCCCc1ccccc1Cl ZINC000217829616 EI In-Stock Unstable MTNR1A 40 40 O=C(COc1ccc(Cl)cc1)NCCCc1ccccc1Cl ZINC000217829616 EI In-Stock Unstable MTNR1B 46 36 O=C(COc1ccc(Cl)cc1)NCCCc1ccccc1Cl ZINC000217829616 EI In-Stock Unstable FFAR4 32 41 O=C(COc1ccc(Cl)cc1)NCCCc1ccccc1Cl ZINC000217829616 EI In-Stock Unstable CRTM 45 46 O=C(NC[C@@H]1CCCN1c1ccccc1)c1n[nH]c2cc(F)ccc12 ZINC000217829653 EG For-Sale Unstable HCRTR1 26 42 O=C(NC[C@@H]1CCCN1c1ccccc1)c1n[nH]c2cc(F)ccc12 ZINC000217829653 EG For-Sale Unstable MC1R 20 41 O=C(NC[C@@H]1CCCN1c1ccccc1)c1n[nH]c2cc(F)ccc12 ZINC000217829653 EG For-Sale Unstable HCRTR2 17 42 O=C(NC[C@@H]1CCCN1c1ccccc1)c1n[nH]c2cc(F)ccc12 ZINC000217829653 EG For-Sale Unstable ACKR3 44 33 CC(C)C[C@@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217829666 CD For-Sale Unstable CTSC 24 41 CC(C)C[C@@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217829666 CD For-Sale Unstable MAN1B1 52 33 COc1cccc(CNC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217829683 DH For-Sale Unstable DRD4 46 39 COc1cccc(CNC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217829683 DH For-Sale Unstable ROCK1 36 43 COc1cccc(CNC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217829683 DH For-Sale Unstable MTNR1A 47 46 COc1cccc(CNC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217829683 DH For-Sale Unstable MTNR1B 47 46 COc1cccc(CNC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217829683 DH For-Sale Unstable ROCK2 45 48 COc1cccc(CNC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217829683 DH For-Sale Unstable PDS 67 40 COc1ccc(S(=O)(=O)CC2(CN)CC2)cc1 ZINC000217829720 CD For-Sale Unstable MMP13 29 46 O=C(COc1ccc(Cl)cc1)NCCCc1ccc(Cl)cc1 ZINC000217829723 EI In-Stock Unstable SCNN1A 70 43 O=C(COc1ccc(Cl)cc1)NCCCc1ccc(Cl)cc1 ZINC000217829723 EI In-Stock Unstable AVPR1A 0 42 O=C(COc1ccc(Cl)cc1)NCCCc1ccc(Cl)cc1 ZINC000217829723 EI In-Stock Unstable FFAR1 23 40 O=C(COc1ccc(Cl)cc1)NCCCc1ccc(Cl)cc1 ZINC000217829723 EI In-Stock Unstable FFAR4 26 40 O=C(COc1ccc(Cl)cc1)NCCCc1ccc(Cl)cc1 ZINC000217829723 EI In-Stock Unstable CRTM 50 53 O=C(COc1ccc(Cl)cc1)NCCCc1ccc(Cl)cc1 ZINC000217829723 EI In-Stock Unstable TRAR 28 44 CC(C)C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217829740 CD For-Sale Unstable CTSC 24 41 CC(C)C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217829740 CD For-Sale Unstable MAN1B1 52 33 COC(=O)CCCCCn1c(SCc2ccc3ccccc3n2)nc2ccccc2c1=O ZINC000217829747 IJ On-Demand Unstable PTGDR2 16 40 O=C(CC12CC3CC(CC(C3)C1)C2)NC[C@H]1CCCN1c1ccccc1 ZINC000217829751 FI For-Sale Unstable BOTA 27 41 CC(C)C[C@@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217829811 CD For-Sale Unstable CTSC 24 41 CC(C)C[C@@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217829811 CD For-Sale Unstable MAN1B1 52 33 O=C(COc1ccc(Cl)cc1)NCCCc1ccc(F)cc1 ZINC000217829819 DH In-Stock Unstable SCNN1A 46 39 O=C(COc1ccc(Cl)cc1)NCCCc1ccc(F)cc1 ZINC000217829819 DH In-Stock Unstable LEF 47 35 O=C(COc1ccc(Cl)cc1)NCCCc1ccc(F)cc1 ZINC000217829819 DH In-Stock Unstable CRTM 46 48 O=C(COc1ccc(Cl)cc1)NCCCc1ccc(F)cc1 ZINC000217829819 DH In-Stock Unstable TRAR 21 40 O=C(CC12CC3CC(CC(C3)C1)C2)NC[C@@H]1CCCN1c1ccccc1 ZINC000217829823 FI For-Sale Unstable BOTA 27 41 COc1cccc(S(=O)(=O)CC2(CN)CC2)c1 ZINC000217829824 CD For-Sale Unstable MTNR1B 20 40 COc1cc2c(cc1OC)CN(C(=O)Cn1ccc3c(NS(C)(=O)=O)cccc31)CC2 ZINC000217829857 IF In-Stock Unstable ABCB1B 54 35 COc1cc2c(cc1OC)CN(C(=O)Cn1ccc3c(NS(C)(=O)=O)cccc31)CC2 ZINC000217829857 IF In-Stock Unstable ABCB1 17 43 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)CN3C(=O)CCC3=O)C2)n1 ZINC000217829866 GD In-Stock Unstable Q8MHZ5_SHEEP 42 33 CC(C)C[C@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217829886 CD For-Sale Unstable CTSC 24 41 CC(C)C[C@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217829886 CD For-Sale Unstable MAN1B1 52 33 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(-c2cccs2)cc1 ZINC000217829898 FJ For-Sale Unstable HCRTR1 26 43 CN1C(=O)C[C@H](CNC(=O)c2ccc(N3CCCC3)cc2)c2ccccc21 ZINC000217829911 FG In-Stock Unstable DRD2 25 40 CN1C(=O)C[C@H](CNC(=O)c2ccc(N3CCCC3)cc2)c2ccccc21 ZINC000217829911 FG In-Stock Unstable DRD4 43 33 CN1C(=O)C[C@H](CNC(=O)c2ccc(N3CCCC3)cc2)c2ccccc21 ZINC000217829911 FG In-Stock Unstable KCNQ2 66 34 CN1C(=O)C[C@H](CNC(=O)c2ccc(N3CCCC3)cc2)c2ccccc21 ZINC000217829911 FG In-Stock Unstable PRNP 46 37 COc1ccccc1CCCNC(=O)COc1ccc(Cl)cc1 ZINC000217829917 EG In-Stock Unstable DRD2 15 41 COc1ccccc1CCCNC(=O)COc1ccc(Cl)cc1 ZINC000217829917 EG In-Stock Unstable DRD3 24 41 COc1ccccc1CCCNC(=O)COc1ccc(Cl)cc1 ZINC000217829917 EG In-Stock Unstable TSPO 35 40 COc1ccccc1CCCNC(=O)COc1ccc(Cl)cc1 ZINC000217829917 EG In-Stock Unstable MTNR1A 69 44 COc1ccccc1CCCNC(=O)COc1ccc(Cl)cc1 ZINC000217829917 EG In-Stock Unstable MTNR1B 57 48 COc1ccccc1CCCNC(=O)COc1ccc(Cl)cc1 ZINC000217829917 EG In-Stock Unstable CRTM 37 43 COc1ccccc1CCCNC(=O)COc1ccc(Cl)cc1 ZINC000217829917 EG In-Stock Unstable MBTPS1 40 38 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)CN3C(=O)CCC3=O)C2)n1 ZINC000217829939 GD In-Stock Unstable Q8MHZ5_SHEEP 42 33 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(-c2cccs2)cc1 ZINC000217829962 FJ For-Sale Unstable HCRTR1 26 43 CN1C(=O)C[C@@H](CNC(=O)c2ccc(N3CCCC3)cc2)c2ccccc21 ZINC000217830014 FG In-Stock Unstable DRD2 25 40 CN1C(=O)C[C@@H](CNC(=O)c2ccc(N3CCCC3)cc2)c2ccccc21 ZINC000217830014 FG In-Stock Unstable DRD4 43 33 CN1C(=O)C[C@@H](CNC(=O)c2ccc(N3CCCC3)cc2)c2ccccc21 ZINC000217830014 FG In-Stock Unstable KCNQ2 66 34 CN1C(=O)C[C@@H](CNC(=O)c2ccc(N3CCCC3)cc2)c2ccccc21 ZINC000217830014 FG In-Stock Unstable PRNP 46 37 COc1cccc(CCCNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217830033 EG In-Stock Unstable DRD4 46 40 COc1cccc(CCCNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217830033 EG In-Stock Unstable PTGS1 0 41 COc1cccc(CCCNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217830033 EG In-Stock Unstable HRH2 30 40 COc1cccc(CCCNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217830033 EG In-Stock Unstable MAOB 22 40 COc1cccc(CCCNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217830033 EG In-Stock Unstable PTGS2 33 43 COc1cccc(CCCNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217830033 EG In-Stock Unstable PTAFR 22 42 COc1cccc(CCCNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217830033 EG In-Stock Unstable FDFT1 22 63 COc1cccc(CCCNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217830033 EG In-Stock Unstable MTNR1A 97 55 COc1cccc(CCCNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217830033 EG In-Stock Unstable MTNR1B 80 68 COc1cccc(CCCNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217830033 EG In-Stock Unstable ROCK2 41 38 COc1cccc(CCCNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217830033 EG In-Stock Unstable AMP1_PLAFQ 20 40 COc1cccc(CCCNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217830033 EG In-Stock Unstable MCHR1 16 40 COc1cccc(CCCNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217830033 EG In-Stock Unstable TAAR1 26 43 COc1cccc(CCCNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217830033 EG In-Stock Unstable AKR1C3 22 41 COc1cccc(CCCNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217830033 EG In-Stock Unstable NCE103 20 54 COc1cccc(CCCNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217830033 EG In-Stock Unstable CRTM 84 63 COc1cccc(CCCNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217830033 EG In-Stock Unstable CRTH2 0 43 COc1cccc(CCCNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217830033 EG In-Stock Unstable CAN2 0 54 COc1cccc(CCCNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217830033 EG In-Stock Unstable PDS 60 38 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)Cn3c(=O)oc4ccccc43)C2)n1 ZINC000217830035 IG In-Stock Unstable Q8MHZ5_SHEEP 41 32 Cc1cc(NC(=O)C2CCN(c3nc4ccccc4o3)CC2)n(-c2ccc(F)cc2)n1 ZINC000217830041 HI On-Demand Unstable PTGES 32 40 COCCC(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217830075 CD For-Sale Unstable ACKR3 52 34 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)Cn3c(=O)oc4ccccc43)C2)n1 ZINC000217830109 IG In-Stock Unstable Q8MHZ5_SHEEP 41 32 O=C(O)/C=C\c1cc(CN2CCCCCC2=O)ccc1F ZINC000217830121 CF For-Sale Unstable PTGER3 20 52 Cc1ccccc1CCNC(=O)N/C=C/c1ccccc1Cl ZINC000217830144 DI For-Sale Unstable CXCL8 42 34 COc1ccc(CCCNC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217830146 EG In-Stock Unstable PTGS2 27 42 COc1ccc(CCCNC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217830146 EG In-Stock Unstable SCNN1A 73 44 COc1ccc(CCCNC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217830146 EG In-Stock Unstable BMP1 23 40 COc1ccc(CCCNC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217830146 EG In-Stock Unstable KCNA5 0 41 COc1ccc(CCCNC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217830146 EG In-Stock Unstable SCN2A 16 42 COc1ccc(CCCNC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217830146 EG In-Stock Unstable MTNR1A 69 42 COc1ccc(CCCNC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217830146 EG In-Stock Unstable MTNR1B 41 45 COc1ccc(CCCNC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217830146 EG In-Stock Unstable CA9 20 46 COc1ccc(CCCNC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217830146 EG In-Stock Unstable U38 0 43 COc1ccc(CCCNC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217830146 EG In-Stock Unstable NCE103 22 40 COc1ccc(CCCNC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217830146 EG In-Stock Unstable CRTM 46 48 COc1ccc(CCCNC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217830146 EG In-Stock Unstable PROKR1 57 40 COc1ccc(CCCNC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217830146 EG In-Stock Unstable TRAR 16 40 COc1ccc(CCCNC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217830146 EG In-Stock Unstable CAN2 0 40 COCCC(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217830147 CD For-Sale Unstable ACKR3 52 34 Cc1[nH]c2ccccc2c1CCNC(=O)COCC(F)(F)C(F)F ZINC000217830202 EG In-Stock Unstable MTNR1B 16 43 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)CCSc3ccccc3)C2)n1 ZINC000217830203 HK In-Stock Unstable Q8MHZ5_SHEEP 50 33 CC1(C)NC(=O)N(Cc2ccccc2/C=C\C(=O)O)C1=O ZINC000217830228 CD For-Sale Unstable PTGER2 44 45 CC1(C)NC(=O)N(Cc2ccccc2/C=C\C(=O)O)C1=O ZINC000217830228 CD For-Sale Unstable PTGER4 22 45 CC1(C)NC(=O)N(Cc2ccccc2/C=C\C(=O)O)C1=O ZINC000217830228 CD For-Sale Unstable PTGER3 22 46 COc1ccccc1CCNC(=O)N/C=C/c1ccccc1Cl ZINC000217830244 EH For-Sale Unstable MTNR1A 30 42 COc1ccccc1CCNC(=O)N/C=C/c1ccccc1Cl ZINC000217830244 EH For-Sale Unstable MTNR1B 21 42 COc1ccc(OC[C@@H](C)NC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217830251 EG In-Stock Unstable PTGS2 26 44 COc1ccc(OC[C@@H](C)NC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217830251 EG In-Stock Unstable SDH1 0 41 COc1ccc(OC[C@@H](C)NC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217830251 EG In-Stock Unstable DXR 19 40 COc1ccc(OC[C@@H](C)NC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217830251 EG In-Stock Unstable TRAR 16 41 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)CCSc3ccccc3)C2)n1 ZINC000217830285 HK In-Stock Unstable Q8MHZ5_SHEEP 50 33 CCOC(=O)[C@H](C)NC(=O)[C@@H]1CCC[C@@H](C(F)(F)F)C1 ZINC000217830313 CE On-Demand Unstable METAP2 22 42 COc1ccc(OC[C@H](C)NC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217830333 EG In-Stock Unstable PTGS2 26 44 COc1ccc(OC[C@H](C)NC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217830333 EG In-Stock Unstable SDH1 0 41 COc1ccc(OC[C@H](C)NC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217830333 EG In-Stock Unstable DXR 19 40 COc1ccc(OC[C@H](C)NC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217830333 EG In-Stock Unstable TRAR 16 41 CC(C)c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2)cc1 ZINC000217830348 CD In-Stock Unstable SDH1 0 42 Nc1cnc(-c2ccc(-c3ccccc3O[C@H]3CCCNC3)cc2F)cn1 ZINC000217830375 FH Annotated Unstable PIM3 16 43 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)c3ccc(C#N)cc3)C2)n1 ZINC000217830391 GI In-Stock Unstable HRH3 15 44 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)c3ccc(C#N)cc3)C2)n1 ZINC000217830391 GI In-Stock Unstable MAP3K12 31 41 COc1ccc(CN2CCOC2=O)cc1/C=C\C(=O)O ZINC000217830401 CD For-Sale Unstable PTGER2 37 42 COc1ccc(CN2CCOC2=O)cc1/C=C\C(=O)O ZINC000217830401 CD For-Sale Unstable PTGER4 23 42 COc1ccc(CN2CCOC2=O)cc1/C=C\C(=O)O ZINC000217830401 CD For-Sale Unstable PTGER3 19 42 CC(C)c1ccc([C@@H](C)NC(=O)[C@H]2C[C@@H](O)CN2)cc1 ZINC000217830418 CD On-Demand Unstable SDH1 0 42 CC(C)Oc1cccc(CCCNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217830461 FI In-Stock Unstable ADRB1 15 41 CC(C)Oc1cccc(CCCNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217830461 FI In-Stock Unstable FDFT1 24 61 CC(C)Oc1cccc(CCCNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217830461 FI In-Stock Unstable MTNR1A 41 44 CC(C)Oc1cccc(CCCNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217830461 FI In-Stock Unstable MTNR1B 41 38 CC(C)Oc1cccc(CCCNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217830461 FI In-Stock Unstable FAAH 19 40 CC(C)Oc1cccc(CCCNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217830461 FI In-Stock Unstable AMP1_PLAFQ 30 41 CC(C)Oc1cccc(CCCNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217830461 FI In-Stock Unstable NCE103 16 42 CC(C)Oc1cccc(CCCNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217830461 FI In-Stock Unstable CRTM 82 61 CC(C)Oc1cccc(CCCNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217830461 FI In-Stock Unstable CAN2 0 42 CC(C)Oc1cccc(CCCNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217830461 FI In-Stock Unstable PDS 69 39 CC(C)Oc1cccc(CCCNC(=O)COc2ccc(Cl)cc2)c1 ZINC000217830461 FI In-Stock Unstable LMGT2 0 41 Cn1nc(-c2ccccc2)cc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217830468 FG For-Sale Unstable P2RY12 54 33 Cn1nc(-c2ccccc2)cc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217830468 FG For-Sale Unstable HCRTR1 39 43 Cn1nc(-c2ccccc2)cc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217830468 FG For-Sale Unstable HCRTR2 32 43 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)c3ccc(C#N)cc3)C2)n1 ZINC000217830471 GI In-Stock Unstable HRH3 15 44 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)c3ccc(C#N)cc3)C2)n1 ZINC000217830471 GI In-Stock Unstable MAP3K12 31 41 CCOC(=O)[C@H](C)NC(=O)[C@H]1CCC[C@@H](C(F)(F)F)C1 ZINC000217830477 CE On-Demand Unstable METAP2 22 42 CC(C)c1ccc([C@H](C)NC(=O)[C@H]2C[C@@H](O)CN2)cc1 ZINC000217830505 CD In-Stock Unstable SDH1 0 42 Cn1nc(-c2ccccc2)cc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217830555 FG For-Sale Unstable P2RY12 54 33 Cn1nc(-c2ccccc2)cc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217830555 FG For-Sale Unstable HCRTR1 39 43 Cn1nc(-c2ccccc2)cc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217830555 FG For-Sale Unstable HCRTR2 32 43 CC(C)Oc1ccc(CCCNC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217830561 FI In-Stock Unstable CRTM 44 46 O=C(O)/C=C\c1cccc(OCCN2CCCS2(=O)=O)c1 ZINC000217830577 DD For-Sale Unstable CYSLTR2 16 40 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)c3ccc(Cl)s3)C2)n1 ZINC000217830580 HJ In-Stock Unstable F10 0 43 CCOC(=O)[C@@H](C)NC(=O)c1ccc2c(c1)CC(=O)N2 ZINC000217830612 CC For-Sale Unstable HDAC9 21 40 Cn1nccc1CCNC(=O)[C@@H]1C[C@H]1c1ccccc1 ZINC000217830619 CD In-Stock Unstable NAMPT 21 42 O=C(COc1ccc(Cl)cc1)Nc1ccc(OC2CCCC2)cc1 ZINC000217830646 EJ In-Stock Unstable ADORA2B 44 45 O=C(COc1ccc(Cl)cc1)Nc1ccc(OC2CCCC2)cc1 ZINC000217830646 EJ In-Stock Unstable CETP 0 48 O=C(COc1ccc(Cl)cc1)Nc1ccc(OC2CCCC2)cc1 ZINC000217830646 EJ In-Stock Unstable EPHX2 33 51 O=C(COc1ccc(Cl)cc1)Nc1ccc(OC2CCCC2)cc1 ZINC000217830646 EJ In-Stock Unstable MCHR1 20 48 O=C(COc1ccc(Cl)cc1)Nc1ccc(OC2CCCC2)cc1 ZINC000217830646 EJ In-Stock Unstable TRAR 31 47 CCCN(CC)CCNC(=O)c1cccnc1F ZINC000217830647 CD On-Demand Unstable POLR1A 29 41 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)c3ccc(Cl)s3)C2)n1 ZINC000217830648 HJ In-Stock Unstable F10 0 43 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc(Cl)c2F)CC(=O)O4)cc1O ZINC000217830653 JK In-Stock Unstable CYP1B1 67 39 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc(Cl)c2F)CC(=O)O4)cc1O ZINC000217830653 JK In-Stock Unstable CYP1A1 44 44 COc1cc(C(=O)NC[C@@H]2CCC[C@@H](O)C2)ccc1F ZINC000217830654 CE On-Demand Unstable CACNA1I 55 36 COc1cc(C(=O)NC[C@@H]2CCC[C@@H](O)C2)ccc1F ZINC000217830654 CE On-Demand Unstable HSPB1 0 41 COc1cc(C(=O)NC[C@@H]2CCC[C@@H](O)C2)ccc1F ZINC000217830654 CE On-Demand Unstable ACKR3 57 33 CCCCN([C@@H](C)CC)[C@H](c1cccc(Cl)c1)[C@@H](C)N ZINC000217830684 CJ For-Sale Unstable OPRL1 0 43 O=C(O)/C=C\c1ccc(OCCN2CCCS2(=O)=O)cc1 ZINC000217830688 DD For-Sale Unstable PSMB2 46 38 CCOC(=O)[C@H](C)NC(=O)c1ccc2c(c1)CC(=O)N2 ZINC000217830696 CC For-Sale Unstable HDAC9 21 40 C[C@@H](c1ccccc1F)N(C)[C@@H](C)[C@@H](O)c1ccccc1 ZINC000217830723 CH For-Sale Unstable NPY5R 21 40 C[C@@H](c1ccccc1F)N(C)[C@@H](C)[C@@H](O)c1ccccc1 ZINC000217830723 CH For-Sale Unstable AOC3 20 53 COc1cc(C(=O)NC[C@H]2CCC[C@@H](O)C2)ccc1F ZINC000217830726 CE On-Demand Unstable CACNA1I 55 36 COc1cc(C(=O)NC[C@H]2CCC[C@@H](O)C2)ccc1F ZINC000217830726 CE On-Demand Unstable HSPB1 0 41 COc1cc(C(=O)NC[C@H]2CCC[C@@H](O)C2)ccc1F ZINC000217830726 CE On-Demand Unstable ACKR3 57 33 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc(Cl)c2F)CC(=O)O4)cc1O ZINC000217830732 JK In-Stock Unstable CYP1B1 67 39 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc(Cl)c2F)CC(=O)O4)cc1O ZINC000217830732 JK In-Stock Unstable CYP1A1 44 44 COc1cccc(CCNC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217830746 EH For-Sale Unstable DRD4 48 40 COc1cccc(CCNC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217830746 EH For-Sale Unstable HRH2 26 40 COc1cccc(CCNC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217830746 EH For-Sale Unstable MTNR1A 88 51 COc1cccc(CCNC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217830746 EH For-Sale Unstable MTNR1B 80 51 COc1cccc(CCNC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217830746 EH For-Sale Unstable CRTM 61 38 COc1cccc(CCNC(=O)N/C=C/c2ccccc2Cl)c1 ZINC000217830746 EH For-Sale Unstable CAN2 0 53 CC1(C)C[C@@H](NC(=O)COc2ccc(Cl)cc2)c2ccccc2O1 ZINC000217830748 EI In-Stock Unstable TRAR 35 52 CC1(C)C[C@@H](NC(=O)COc2ccc(Cl)cc2)c2ccccc2O1 ZINC000217830748 EI In-Stock Unstable LUXN 0 42 CC1(C)C[C@@H](NC(=O)COc2ccc(Cl)cc2)c2ccccc2O1 ZINC000217830748 EI In-Stock Unstable CVIR 0 40 CCCCN([C@H](C)CC)[C@H](c1cccc(Cl)c1)[C@@H](C)N ZINC000217830761 CJ For-Sale Unstable OPRL1 0 43 CC(C)=C=CC[C@H](N)C(=O)O ZINC000217830790 AC For-Sale Unstable GRIK3 46 40 CC(C)=C=CC[C@H](N)C(=O)O ZINC000217830790 AC For-Sale Unstable GRIK2 44 35 CC(C)=C=CC[C@H](N)C(=O)O ZINC000217830790 AC For-Sale Unstable GRIK1 67 46 C[C@@H]([C@@H](O)c1ccccc1)N(C)[C@H](C)c1ccccc1F ZINC000217830806 CH For-Sale Unstable NPY5R 21 40 C[C@@H]([C@@H](O)c1ccccc1)N(C)[C@H](C)c1ccccc1F ZINC000217830806 CH For-Sale Unstable AOC3 20 53 CC1(C)C[C@H](NC(=O)COc2ccc(Cl)cc2)c2ccccc2O1 ZINC000217830809 EI In-Stock Unstable TRAR 35 52 CC1(C)C[C@H](NC(=O)COc2ccc(Cl)cc2)c2ccccc2O1 ZINC000217830809 EI In-Stock Unstable LUXN 0 42 CC1(C)C[C@H](NC(=O)COc2ccc(Cl)cc2)c2ccccc2O1 ZINC000217830809 EI In-Stock Unstable CVIR 0 40 COc1cc(C(=O)NC[C@@H]2CCC[C@H](O)C2)ccc1F ZINC000217830825 CE On-Demand Unstable CACNA1I 55 36 COc1cc(C(=O)NC[C@@H]2CCC[C@H](O)C2)ccc1F ZINC000217830825 CE On-Demand Unstable HSPB1 0 41 COc1cc(C(=O)NC[C@@H]2CCC[C@H](O)C2)ccc1F ZINC000217830825 CE On-Demand Unstable ACKR3 57 33 CC[C@@H](C)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)O ZINC000217830834 CD For-Sale Unstable ACE 19 41 CC[C@@H](C)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)O ZINC000217830834 CD For-Sale Unstable MME 50 45 CC[C@@H](C)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)O ZINC000217830834 CD For-Sale Unstable ANPEP 47 33 CC[C@@H](C)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)O ZINC000217830834 CD For-Sale Unstable HLA-A 40 44 CC[C@@H](C)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)O ZINC000217830834 CD For-Sale Unstable ENPEP 67 39 CC[C@@H](C)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)O ZINC000217830834 CD For-Sale Unstable ACE2 55 38 O=C(CC[C@@H]1NC(=O)c2ccccc2NC1=O)N[C@H](Cc1ccccc1)c1nc2ccccc2[nH]1 ZINC000217830850 JG In-Stock Unstable F11 47 36 O=C(CC[C@@H]1NC(=O)c2ccccc2NC1=O)N[C@H](Cc1ccccc1)c1nc2ccccc2[nH]1 ZINC000217830850 JG In-Stock Unstable PTPN1 36 49 CC(C)=C=CC[C@@H](N)C(=O)O ZINC000217830877 AC For-Sale Unstable GRIK3 46 40 CC(C)=C=CC[C@@H](N)C(=O)O ZINC000217830877 AC For-Sale Unstable GRIK2 44 35 CC(C)=C=CC[C@@H](N)C(=O)O ZINC000217830877 AC For-Sale Unstable GRIK1 67 46 CS(=O)(=O)CC(=O)Nc1cccnc1Cl ZINC000217830889 BC On-Demand Unstable G2YM83_BOTF4 78 39 COc1cc(C(=O)NC[C@H]2CCC[C@H](O)C2)ccc1F ZINC000217830902 CE On-Demand Unstable CACNA1I 55 36 COc1cc(C(=O)NC[C@H]2CCC[C@H](O)C2)ccc1F ZINC000217830902 CE On-Demand Unstable HSPB1 0 41 COc1cc(C(=O)NC[C@H]2CCC[C@H](O)C2)ccc1F ZINC000217830902 CE On-Demand Unstable ACKR3 57 33 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)c3cn(C)nn3)C2)n1 ZINC000217830915 FE In-Stock Unstable HRH3 17 41 CCOc1ccc(CCCNC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217830916 EH In-Stock Unstable SCNN1A 47 39 CCOc1ccc(CCCNC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217830916 EH In-Stock Unstable SCN2A 31 46 CCOc1ccc(CCCNC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217830916 EH In-Stock Unstable PLA2G4B 65 35 CCOc1ccc(CCCNC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217830916 EH In-Stock Unstable CRTM 47 48 CCOc1ccc(CCCNC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217830916 EH In-Stock Unstable TRAR 16 40 CC[C@H](C)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)O ZINC000217830918 CD On-Demand Unstable MME 36 41 CC[C@H](C)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)O ZINC000217830918 CD On-Demand Unstable ANPEP 47 33 CC[C@H](C)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)O ZINC000217830918 CD On-Demand Unstable HLA-A 34 42 CC[C@H](C)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)O ZINC000217830918 CD On-Demand Unstable ENPEP 67 39 CC[C@H](C)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)O ZINC000217830918 CD On-Demand Unstable ACE2 55 38 CC[C@H](C)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)O ZINC000217830918 CD On-Demand Unstable POL 0 42 O=C(CC[C@@H]1NC(=O)c2ccccc2NC1=O)N[C@@H](Cc1ccccc1)c1nc2ccccc2[nH]1 ZINC000217830948 JG In-Stock Unstable F11 47 36 O=C(CC[C@@H]1NC(=O)c2ccccc2NC1=O)N[C@@H](Cc1ccccc1)c1nc2ccccc2[nH]1 ZINC000217830948 JG In-Stock Unstable PTPN1 36 49 COc1ccc(-c2noc(CCC(=O)Nc3cc(C)nn3-c3ccc(F)cc3)n2)cc1 ZINC000217830992 HH On-Demand Unstable HCAR2 23 41 COc1ccc(-c2noc(CCC(=O)Nc3cc(C)nn3-c3ccc(F)cc3)n2)cc1 ZINC000217830992 HH On-Demand Unstable TNKS2 15 47 O=C(c1ccc(SCCO)cc1)N1CCc2c(Cl)cccc2C1 ZINC000217830997 EH In-Stock Unstable FABI 48 35 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)c3cn(C)nn3)C2)n1 ZINC000217831002 FE In-Stock Unstable HRH3 17 41 Cc1cc(Cl)cc(C(=O)NC[C@@H]2CCC[C@@H](O)C2)c1 ZINC000217831011 CF On-Demand Unstable CACNA1I 68 50 CCCOc1ccccc1CCCNC(=O)COc1ccc(Cl)cc1 ZINC000217831014 FI In-Stock Unstable MTNR1A 48 43 CCCOc1ccccc1CCCNC(=O)COc1ccc(Cl)cc1 ZINC000217831014 FI In-Stock Unstable MTNR1B 52 43 CCCOc1ccccc1CCCNC(=O)COc1ccc(Cl)cc1 ZINC000217831014 FI In-Stock Unstable PLA2G4B 70 33 CCCOc1ccccc1CCCNC(=O)COc1ccc(Cl)cc1 ZINC000217831014 FI In-Stock Unstable CRTM 35 41 CCCCN([C@H](C)CC)[C@@H]1CCCc2cc(O)ccc21 ZINC000217831017 CJ For-Sale Unstable HSD17B1 40 34 COc1cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc(OC)c1OC ZINC000217831031 FG For-Sale Unstable HTR1A 27 47 COc1cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc(OC)c1OC ZINC000217831031 FG For-Sale Unstable DRD2 58 53 COc1cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc(OC)c1OC ZINC000217831031 FG For-Sale Unstable ACHE 15 42 COc1cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc(OC)c1OC ZINC000217831031 FG For-Sale Unstable DRD3 49 49 COc1cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc(OC)c1OC ZINC000217831031 FG For-Sale Unstable SIGMAR1 15 49 COc1cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc(OC)c1OC ZINC000217831031 FG For-Sale Unstable CHRNA10 44 36 COc1cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc(OC)c1OC ZINC000217831031 FG For-Sale Unstable MCHR1 17 46 COc1cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc(OC)c1OC ZINC000217831031 FG For-Sale Unstable CACNA1I 62 34 COc1cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc(OC)c1OC ZINC000217831031 FG For-Sale Unstable ALK 16 40 COc1cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc(OC)c1OC ZINC000217831031 FG For-Sale Unstable SMO 22 40 COc1cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc(OC)c1OC ZINC000217831031 FG For-Sale Unstable ACKR3 93 50 CC[C@@H](C)[C@@H](NC(=O)[C@@H](N)CCS(C)(=O)=O)C(=O)O ZINC000217831090 CB For-Sale Unstable HLA-A 50 42 CC[C@@H](C)[C@@H](NC(=O)[C@@H](N)CCS(C)(=O)=O)C(=O)O ZINC000217831090 CB For-Sale Unstable ENPEP 99 59 Cc1ccccc1OC[C@H](C)NC(=O)COc1ccc(Cl)cc1 ZINC000217831094 EH In-Stock Unstable SDH1 0 41 Cc1ccccc1OC[C@H](C)NC(=O)COc1ccc(Cl)cc1 ZINC000217831094 EH In-Stock Unstable CETP 0 40 Cc1cc(Cl)cc(C(=O)NC[C@H]2CCC[C@@H](O)C2)c1 ZINC000217831111 CF On-Demand Unstable CACNA1I 68 50 COc1cc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc(OC)c1OC ZINC000217831113 FG For-Sale Unstable HTR1A 27 47 COc1cc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc(OC)c1OC ZINC000217831113 FG For-Sale Unstable DRD2 58 53 COc1cc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc(OC)c1OC ZINC000217831113 FG For-Sale Unstable ACHE 15 42 COc1cc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc(OC)c1OC ZINC000217831113 FG For-Sale Unstable DRD3 49 49 COc1cc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc(OC)c1OC ZINC000217831113 FG For-Sale Unstable SIGMAR1 15 49 COc1cc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc(OC)c1OC ZINC000217831113 FG For-Sale Unstable CHRNA10 44 36 COc1cc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc(OC)c1OC ZINC000217831113 FG For-Sale Unstable MCHR1 17 46 COc1cc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc(OC)c1OC ZINC000217831113 FG For-Sale Unstable CACNA1I 62 34 COc1cc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc(OC)c1OC ZINC000217831113 FG For-Sale Unstable ALK 16 40 COc1cc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc(OC)c1OC ZINC000217831113 FG For-Sale Unstable SMO 22 40 COc1cc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc(OC)c1OC ZINC000217831113 FG For-Sale Unstable ACKR3 93 50 CC(C)(C)OC(=O)N1CCC(CC2(O)CC2)CC1 ZINC000217831122 CF For-Sale Unstable GPR119 46 44 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)c3cc(C4CC4)on3)C2)n1 ZINC000217831136 GI In-Stock Unstable Q8MHZ5_SHEEP 40 31 CCCCN([C@H](C)CC)[C@@H]1CCc2c(O)cccc21 ZINC000217831140 CI For-Sale Unstable HTR1A 0 47 CC[C@H](C)[C@@H](NC(=O)[C@@H](N)CCS(C)(=O)=O)C(=O)O ZINC000217831168 CB For-Sale Unstable HLA-A 50 42 CC[C@H](C)[C@@H](NC(=O)[C@@H](N)CCS(C)(=O)=O)C(=O)O ZINC000217831168 CB For-Sale Unstable ENPEP 99 59 Cc1cc(NC(=O)c2ccc(S(=O)(=O)NC(C)(C)C)cc2)n(-c2ccc(F)cc2)n1 ZINC000217831175 IH On-Demand Unstable MAPK14 0 40 Cc1cc(NC(=O)c2ccc(S(=O)(=O)NC(C)(C)C)cc2)n(-c2ccc(F)cc2)n1 ZINC000217831175 IH On-Demand Unstable FPR1 15 42 Cc1cc(Cl)cc(C(=O)NC[C@@H]2CCC[C@H](O)C2)c1 ZINC000217831178 CF On-Demand Unstable CACNA1I 68 50 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)c3cc(C4CC4)on3)C2)n1 ZINC000217831190 GI In-Stock Unstable Q8MHZ5_SHEEP 40 31 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccccc1Cl ZINC000217831207 DH For-Sale Unstable DRD2 36 42 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccccc1Cl ZINC000217831207 DH For-Sale Unstable SLC6A1 60 37 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccccc1Cl ZINC000217831207 DH For-Sale Unstable DRD3 22 43 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccccc1Cl ZINC000217831207 DH For-Sale Unstable HCRTR1 35 47 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccccc1Cl ZINC000217831207 DH For-Sale Unstable P2RX7 17 45 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccccc1Cl ZINC000217831207 DH For-Sale Unstable PREP 28 40 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccccc1Cl ZINC000217831207 DH For-Sale Unstable HCRTR2 28 47 Cc1ccc(OC[C@@H](C)NC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217831210 EH In-Stock Unstable SDH1 0 41 Cc1ccc(OC[C@@H](C)NC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217831210 EH In-Stock Unstable TRAR 16 41 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1Cl ZINC000217831276 DH For-Sale Unstable DRD2 36 42 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1Cl ZINC000217831276 DH For-Sale Unstable SLC6A1 60 37 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1Cl ZINC000217831276 DH For-Sale Unstable DRD3 22 43 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1Cl ZINC000217831276 DH For-Sale Unstable HCRTR1 35 47 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1Cl ZINC000217831276 DH For-Sale Unstable P2RX7 17 45 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1Cl ZINC000217831276 DH For-Sale Unstable PREP 28 40 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1Cl ZINC000217831276 DH For-Sale Unstable HCRTR2 28 47 Cc1cc(Cl)cc(C(=O)NC[C@H]2CCC[C@H](O)C2)c1 ZINC000217831278 CF On-Demand Unstable CACNA1I 68 50 Cc1ccc(OC[C@H](C)NC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217831284 EH In-Stock Unstable SDH1 0 41 Cc1ccc(OC[C@H](C)NC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217831284 EH In-Stock Unstable TRAR 16 41 CC[C@@H](C)NS(=O)(=O)c1ccc(C(=O)Nc2cc(C)nn2-c2ccc(F)cc2)cc1 ZINC000217831318 IH On-Demand Unstable FPR1 19 40 O=C(N/C=C/c1ccccc1Cl)NCCc1ccc(Cl)cc1 ZINC000217831321 EJ For-Sale Unstable NCE103 22 40 O=C(N/C=C/c1ccccc1Cl)NCCc1ccc(Cl)cc1 ZINC000217831321 EJ For-Sale Unstable CAN2 0 40 CC(C)[C@@H]1CN(c2nc3ccccc3nc2C(F)(F)F)CCN1 ZINC000217831359 DG For-Sale Unstable PRKCQ 45 35 CC1CCN(c2ccc([C@@H](C)NC(=O)COc3ccc(Cl)cc3)cc2)CC1 ZINC000217831375 GJ In-Stock Unstable PRCP 22 45 CC1CCN(c2ccc([C@@H](C)NC(=O)COc3ccc(Cl)cc3)cc2)CC1 ZINC000217831375 GJ In-Stock Unstable ACACB 24 41 CC1CCN(c2ccc([C@@H](C)NC(=O)COc3ccc(Cl)cc3)cc2)CC1 ZINC000217831375 GJ In-Stock Unstable EBP 20 46 CC1CCN(c2ccc([C@@H](C)NC(=O)COc3ccc(Cl)cc3)cc2)CC1 ZINC000217831375 GJ In-Stock Unstable TRAR 26 40 COc1ccc(/C=C\C(=O)O)cc1COCc1ccco1 ZINC000217831386 CG For-Sale Unstable PTGER2 24 42 COc1ccc(/C=C\C(=O)O)cc1COCc1ccco1 ZINC000217831386 CG For-Sale Unstable AKR1C3 23 41 CC[C@H](C)NS(=O)(=O)c1ccc(C(=O)Nc2cc(C)nn2-c2ccc(F)cc2)cc1 ZINC000217831389 IH On-Demand Unstable FPR1 19 40 CC(C)[C@H]1CN(c2nc3ccccc3nc2C(F)(F)F)CCN1 ZINC000217831410 DG For-Sale Unstable PRKCQ 45 35 CC1CCN(c2ccc([C@H](C)NC(=O)COc3ccc(Cl)cc3)cc2)CC1 ZINC000217831425 GJ In-Stock Unstable PRCP 22 45 CC1CCN(c2ccc([C@H](C)NC(=O)COc3ccc(Cl)cc3)cc2)CC1 ZINC000217831425 GJ In-Stock Unstable ACACB 24 41 CC1CCN(c2ccc([C@H](C)NC(=O)COc3ccc(Cl)cc3)cc2)CC1 ZINC000217831425 GJ In-Stock Unstable EBP 20 46 CC1CCN(c2ccc([C@H](C)NC(=O)COc3ccc(Cl)cc3)cc2)CC1 ZINC000217831425 GJ In-Stock Unstable TRAR 26 40 COc1ccc(COCc2ccco2)cc1/C=C\C(=O)O ZINC000217831432 CG For-Sale Unstable PTGER2 41 45 COc1ccc(COCc2ccco2)cc1/C=C\C(=O)O ZINC000217831432 CG For-Sale Unstable PTGER4 0 45 COc1ccc(COCc2ccco2)cc1/C=C\C(=O)O ZINC000217831432 CG For-Sale Unstable PTGER3 19 45 CN1CC[C@@H](NC(=O)c2ccc(Cl)o2)C1 ZINC000217831464 BD For-Sale Unstable UTS2R 25 41 CN1CC[C@@H](NC(=O)c2ccc(Cl)o2)C1 ZINC000217831464 BD For-Sale Unstable SLC6A5 30 44 CN1CC[C@@H](NC(=O)c2ccc(Cl)o2)C1 ZINC000217831464 BD For-Sale Unstable CSF1R 0 43 O=S(=O)(Cl)c1cccc(OC2CCC2)c1 ZINC000217831468 BF For-Sale Unstable DUT 17 41 CC[C@@H](C)[C@@H](NC(=O)[C@@](C)(N)C1CC1)C(=O)O ZINC000217831501 BC For-Sale Unstable ENPEP 66 38 O=C(Cc1ccc(O)c(F)c1)NCCc1ccncc1 ZINC000217831502 CD In-Stock Unstable CA5B 22 59 O=C(Cc1ccc(O)c(F)c1)NCCc1ccncc1 ZINC000217831502 CD In-Stock Unstable CA5A 19 59 O=C(Cc1ccc(O)c(F)c1)NCCc1ccncc1 ZINC000217831502 CD In-Stock Unstable NCE103 36 53 O=C(Cc1ccc(O)c(F)c1)NCCc1ccncc1 ZINC000217831502 CD In-Stock Unstable P96878_MYCTU 22 53 O=C(Cc1ccc(O)c(F)c1)NCCc1ccncc1 ZINC000217831502 CD In-Stock Unstable CAN2 0 53 O=C(O)/C=C\c1ccc(COCc2ccco2)c(F)c1 ZINC000217831512 CG For-Sale Unstable AKR1C3 29 41 CN1CC[C@H](NC(=O)c2ccc(Cl)o2)C1 ZINC000217831514 BD For-Sale Unstable UTS2R 25 41 CN1CC[C@H](NC(=O)c2ccc(Cl)o2)C1 ZINC000217831514 BD For-Sale Unstable SLC6A5 30 44 CN1CC[C@H](NC(=O)c2ccc(Cl)o2)C1 ZINC000217831514 BD For-Sale Unstable CSF1R 0 43 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)COc3ccc(Cl)cc3)cc2)C1 ZINC000217831553 GJ In-Stock Unstable EBP 18 40 NS(=O)(=O)c1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217831558 FD For-Sale Unstable CA2 85 57 NS(=O)(=O)c1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217831558 FD For-Sale Unstable DRD2 19 46 NS(=O)(=O)c1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217831558 FD For-Sale Unstable CA1 61 48 NS(=O)(=O)c1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217831558 FD For-Sale Unstable CA7 46 46 NS(=O)(=O)c1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217831558 FD For-Sale Unstable CA13 17 40 NS(=O)(=O)c1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217831558 FD For-Sale Unstable CA5B 45 40 NS(=O)(=O)c1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217831558 FD For-Sale Unstable CA4 53 48 NS(=O)(=O)c1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217831558 FD For-Sale Unstable CA5A 47 40 NS(=O)(=O)c1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217831558 FD For-Sale Unstable CA14 37 44 NS(=O)(=O)c1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217831558 FD For-Sale Unstable CA12 43 46 NS(=O)(=O)c1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217831558 FD For-Sale Unstable CA9 50 46 NS(=O)(=O)c1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217831558 FD For-Sale Unstable CYNT 20 40 NS(=O)(=O)c1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217831558 FD For-Sale Unstable P96878_MYCTU 49 38 CC[C@H](C)[C@@H](NC(=O)[C@@](C)(N)C1CC1)C(=O)O ZINC000217831582 BC For-Sale Unstable ENPEP 66 38 NS(=O)(=O)c1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217831605 FD For-Sale Unstable CA2 85 57 NS(=O)(=O)c1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217831605 FD For-Sale Unstable DRD2 19 46 NS(=O)(=O)c1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217831605 FD For-Sale Unstable CA1 61 48 NS(=O)(=O)c1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217831605 FD For-Sale Unstable CA7 46 46 NS(=O)(=O)c1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217831605 FD For-Sale Unstable CA13 17 40 NS(=O)(=O)c1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217831605 FD For-Sale Unstable CA5B 45 40 NS(=O)(=O)c1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217831605 FD For-Sale Unstable CA4 53 48 NS(=O)(=O)c1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217831605 FD For-Sale Unstable CA5A 47 40 NS(=O)(=O)c1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217831605 FD For-Sale Unstable CA14 37 44 NS(=O)(=O)c1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217831605 FD For-Sale Unstable CA12 43 46 NS(=O)(=O)c1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217831605 FD For-Sale Unstable CA9 50 46 NS(=O)(=O)c1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217831605 FD For-Sale Unstable CYNT 20 40 NS(=O)(=O)c1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217831605 FD For-Sale Unstable P96878_MYCTU 49 38 C[C@H](NC(=O)COc1ccc(Cl)cc1)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217831608 GJ In-Stock Unstable EBP 18 40 O=C(O)/C=C\c1cccc(OCCN2CCSCC2)c1 ZINC000217831619 CE For-Sale Unstable LTA4H 39 44 O=C(O)/C=C\c1cccc(OCCN2CCSCC2)c1 ZINC000217831619 CE For-Sale Unstable EPHX2 19 42 O=C(O)/C=C\c1cccc(OCCN2CCSCC2)c1 ZINC000217831619 CE For-Sale Unstable PSMB2 48 40 O=C(O)/C=C\c1cccc(OCCN2CCSCC2)c1 ZINC000217831619 CE For-Sale Unstable PSMB1 41 40 Cc1ccc(NC(=O)N/C=C/c2ccccc2Cl)nc1 ZINC000217831679 CH For-Sale Unstable GCK 15 40 Cc1ccc(NC(=O)N/C=C/c2ccccc2Cl)nc1 ZINC000217831679 CH For-Sale Unstable LUCI_LUCLA 40 39 CN(Cc1nc2ccc(F)cc2[nH]1)C(=O)Cn1ccc(=O)[nH]c1=O ZINC000217831681 EC In-Stock Unstable PLA2G7 40 37 CC[C@H](C)[C@@H](NC(=O)CN[C@H](C)CC)C(=O)O ZINC000217831700 BC For-Sale Unstable HLA-A 38 45 CC[C@H](C)[C@@H](NC(=O)CN[C@H](C)CC)C(=O)O ZINC000217831700 BC For-Sale Unstable ENPEP 58 39 O=C(O)/C=C\c1ccc(OCCN2CCSCC2)cc1 ZINC000217831719 CE On-Demand Unstable ESR1 56 40 O=C(O)/C=C\c1ccc(OCCN2CCSCC2)cc1 ZINC000217831719 CE On-Demand Unstable ESR2 38 40 O=C(O)/C=C\c1ccc(OCCN2CCSCC2)cc1 ZINC000217831719 CE On-Demand Unstable LTA4H 57 42 O=C(O)/C=C\c1ccc(OCCN2CCSCC2)cc1 ZINC000217831719 CE On-Demand Unstable HRH3 34 52 O=C(O)/C=C\c1ccc(OCCN2CCSCC2)cc1 ZINC000217831719 CE On-Demand Unstable PSMB2 56 43 O=C(O)/C=C\c1ccc(OCCN2CCSCC2)cc1 ZINC000217831719 CE On-Demand Unstable PSMB1 49 44 Cc1ccc([C@@H](C)N2CC[C@@H](c3ccccc3)C2)c(O)c1 ZINC000217831731 CI For-Sale Unstable CCR5 17 41 CC(C)[C@@H]1CN(c2cnc3cc(F)ccc3n2)CCN1 ZINC000217831733 CE For-Sale Unstable PRKCQ 22 42 OC1=NN=C(c2cccnc2)[C@@H]2C[C@@H]12 ZINC000217831756 AD In-Stock Unstable CYP2A6 42 38 Cc1ccc2c(c1)[C@@H](NC(=O)COc1ccc(Cl)cc1)CC(C)(C)O2 ZINC000217831758 FI In-Stock Unstable TRAR 33 48 O=C(CCn1cnc2ccccc2c1=O)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217831759 FE In-Stock Unstable HTR7 16 42 O=C(N[C@@H]1CCN(Cc2ccccc2)C1)[C@@H]1C[C@@H](O)CN1 ZINC000217831761 CC On-Demand Unstable DRD4 34 49 O=C(N[C@@H]1CCN(Cc2ccccc2)C1)[C@@H]1C[C@@H](O)CN1 ZINC000217831761 CC On-Demand Unstable DRD3 24 47 O=C(N[C@@H]1CCN(Cc2ccccc2)C1)[C@@H]1C[C@@H](O)CN1 ZINC000217831761 CC On-Demand Unstable SIGMAR1 46 51 O=C(N[C@@H]1CCN(Cc2ccccc2)C1)[C@@H]1C[C@@H](O)CN1 ZINC000217831761 CC On-Demand Unstable CCR3 30 48 O=C(N[C@@H]1CCN(Cc2ccccc2)C1)[C@@H]1C[C@@H](O)CN1 ZINC000217831761 CC On-Demand Unstable MCHR1 27 52 O=C(N[C@@H]1CCN(Cc2ccccc2)C1)[C@@H]1C[C@@H](O)CN1 ZINC000217831761 CC On-Demand Unstable BIRC2 30 41 O=C(N[C@@H]1CCN(Cc2ccccc2)C1)[C@@H]1C[C@@H](O)CN1 ZINC000217831761 CC On-Demand Unstable ADIPOR1 0 41 O=C(N[C@@H]1CCN(Cc2ccccc2)C1)[C@@H]1C[C@@H](O)CN1 ZINC000217831761 CC On-Demand Unstable ADIPOR2 0 41 O=S(=O)(Cl)c1cccc(OCC2CC2)c1 ZINC000217831764 BE For-Sale Unstable CHRNA10 49 35 O=C(NC[C@H]1CCCN1c1ccccc1)c1cc2ccccc2[nH]1 ZINC000217831766 DH For-Sale Unstable DRD3 18 44 O=C(NC[C@H]1CCCN1c1ccccc1)c1cc2ccccc2[nH]1 ZINC000217831766 DH For-Sale Unstable CCKAR 31 48 O=C(NC[C@H]1CCCN1c1ccccc1)c1cc2ccccc2[nH]1 ZINC000217831766 DH For-Sale Unstable CYP51A1 24 46 O=C(NC[C@H]1CCCN1c1ccccc1)c1cc2ccccc2[nH]1 ZINC000217831766 DH For-Sale Unstable PYGL 89 42 O=C(NC[C@H]1CCCN1c1ccccc1)c1cc2ccccc2[nH]1 ZINC000217831766 DH For-Sale Unstable PLD1 50 45 O=C(NC[C@H]1CCCN1c1ccccc1)c1cc2ccccc2[nH]1 ZINC000217831766 DH For-Sale Unstable PYGM 34 42 O=C(NC[C@H]1CCCN1c1ccccc1)c1cc2ccccc2[nH]1 ZINC000217831766 DH For-Sale Unstable PLD2 40 46 O=C(NC[C@H]1CCCN1c1ccccc1)c1cc2ccccc2[nH]1 ZINC000217831766 DH For-Sale Unstable AKR1C3 28 47 O=C(N[C@@H]1CCN(Cc2ccccc2)C1)[C@H]1C[C@H](O)CN1 ZINC000217831811 CC On-Demand Unstable DRD4 34 49 O=C(N[C@@H]1CCN(Cc2ccccc2)C1)[C@H]1C[C@H](O)CN1 ZINC000217831811 CC On-Demand Unstable DRD3 24 47 O=C(N[C@@H]1CCN(Cc2ccccc2)C1)[C@H]1C[C@H](O)CN1 ZINC000217831811 CC On-Demand Unstable SIGMAR1 46 51 O=C(N[C@@H]1CCN(Cc2ccccc2)C1)[C@H]1C[C@H](O)CN1 ZINC000217831811 CC On-Demand Unstable CCR3 30 48 O=C(N[C@@H]1CCN(Cc2ccccc2)C1)[C@H]1C[C@H](O)CN1 ZINC000217831811 CC On-Demand Unstable MCHR1 27 52 O=C(N[C@@H]1CCN(Cc2ccccc2)C1)[C@H]1C[C@H](O)CN1 ZINC000217831811 CC On-Demand Unstable BIRC2 30 41 O=C(N[C@@H]1CCN(Cc2ccccc2)C1)[C@H]1C[C@H](O)CN1 ZINC000217831811 CC On-Demand Unstable ADIPOR1 0 41 O=C(N[C@@H]1CCN(Cc2ccccc2)C1)[C@H]1C[C@H](O)CN1 ZINC000217831811 CC On-Demand Unstable ADIPOR2 0 41 OC1=NN=C(c2cccnc2)[C@H]2C[C@@H]12 ZINC000217831820 AD In-Stock Unstable CYP2A6 42 38 Cc1ccc([C@H](C)N2CC[C@@H](c3ccccc3)C2)c(O)c1 ZINC000217831835 CI For-Sale Unstable CCR5 17 41 Cc1ccc2c(c1)[C@H](NC(=O)COc1ccc(Cl)cc1)CC(C)(C)O2 ZINC000217831836 FI In-Stock Unstable TRAR 33 48 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cc2ccccc2[nH]1 ZINC000217831847 DH For-Sale Unstable DRD3 18 44 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cc2ccccc2[nH]1 ZINC000217831847 DH For-Sale Unstable CCKAR 31 48 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cc2ccccc2[nH]1 ZINC000217831847 DH For-Sale Unstable CYP51A1 24 46 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cc2ccccc2[nH]1 ZINC000217831847 DH For-Sale Unstable PYGL 89 42 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cc2ccccc2[nH]1 ZINC000217831847 DH For-Sale Unstable PLD1 50 45 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cc2ccccc2[nH]1 ZINC000217831847 DH For-Sale Unstable PYGM 34 42 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cc2ccccc2[nH]1 ZINC000217831847 DH For-Sale Unstable PLD2 40 46 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cc2ccccc2[nH]1 ZINC000217831847 DH For-Sale Unstable AKR1C3 28 47 CC[C@@H](C)[C@@H](CO)NC(=O)CCCc1c[nH]c2ccccc12 ZINC000217831870 DG In-Stock Unstable ACE 15 43 CC[C@@H](C)[C@@H](CO)NC(=O)CCCc1c[nH]c2ccccc12 ZINC000217831870 DG In-Stock Unstable GNRHR 0 41 CC[C@@H](C)[C@@H](CO)NC(=O)CCCc1c[nH]c2ccccc12 ZINC000217831870 DG In-Stock Unstable MME 20 40 CC[C@@H](C)[C@@H](CO)NC(=O)CCCc1c[nH]c2ccccc12 ZINC000217831870 DG In-Stock Unstable EDNRB 24 41 CC[C@@H](C)[C@@H](CO)NC(=O)CCCc1c[nH]c2ccccc12 ZINC000217831870 DG In-Stock Unstable EDNRA 45 41 CC[C@@H](C)[C@@H](CO)NC(=O)CCCc1c[nH]c2ccccc12 ZINC000217831870 DG In-Stock Unstable TACR1 48 44 CC[C@@H](C)[C@@H](CO)NC(=O)CCCc1c[nH]c2ccccc12 ZINC000217831870 DG In-Stock Unstable BMP1 26 42 CC[C@@H](C)[C@@H](CO)NC(=O)CCCc1c[nH]c2ccccc12 ZINC000217831870 DG In-Stock Unstable CTSB 16 47 CC[C@@H](C)[C@@H](CO)NC(=O)CCCc1c[nH]c2ccccc12 ZINC000217831870 DG In-Stock Unstable CCKAR 80 41 CC[C@@H](C)[C@@H](CO)NC(=O)CCCc1c[nH]c2ccccc12 ZINC000217831870 DG In-Stock Unstable CTSL 34 47 CC[C@@H](C)[C@@H](CO)NC(=O)CCCc1c[nH]c2ccccc12 ZINC000217831870 DG In-Stock Unstable MPO 55 44 CC[C@@H](C)[C@@H](CO)NC(=O)CCCc1c[nH]c2ccccc12 ZINC000217831870 DG In-Stock Unstable BRS3 23 41 CC[C@@H](C)[C@@H](CO)NC(=O)CCCc1c[nH]c2ccccc12 ZINC000217831870 DG In-Stock Unstable NMBR 43 33 CC[C@@H](C)[C@@H](CO)NC(=O)CCCc1c[nH]c2ccccc12 ZINC000217831870 DG In-Stock Unstable MC5R 55 34 CC[C@@H](C)[C@@H](CO)NC(=O)CCCc1c[nH]c2ccccc12 ZINC000217831870 DG In-Stock Unstable MMP2 22 40 CC[C@@H](C)[C@@H](CO)NC(=O)CCCc1c[nH]c2ccccc12 ZINC000217831870 DG In-Stock Unstable MMP8 32 40 CC[C@@H](C)[C@@H](CO)NC(=O)CCCc1c[nH]c2ccccc12 ZINC000217831870 DG In-Stock Unstable MMP14 80 42 CC[C@@H](C)[C@@H](CO)NC(=O)CCCc1c[nH]c2ccccc12 ZINC000217831870 DG In-Stock Unstable GRPR 56 32 CC[C@@H](C)[C@@H](CO)NC(=O)CCCc1c[nH]c2ccccc12 ZINC000217831870 DG In-Stock Unstable ECE1 50 43 CC[C@@H](C)[C@@H](CO)NC(=O)CCCc1c[nH]c2ccccc12 ZINC000217831870 DG In-Stock Unstable HDAC3 15 40 CC[C@@H](C)[C@@H](CO)NC(=O)CCCc1c[nH]c2ccccc12 ZINC000217831870 DG In-Stock Unstable MMP11 59 35 CC[C@@H](C)[C@@H](CO)NC(=O)CCCc1c[nH]c2ccccc12 ZINC000217831870 DG In-Stock Unstable CCKBR 67 38 CC[C@@H](C)[C@@H](CO)NC(=O)CCCc1c[nH]c2ccccc12 ZINC000217831870 DG In-Stock Unstable GHSR 74 40 CC[C@@H](C)[C@@H](CO)NC(=O)CCCc1c[nH]c2ccccc12 ZINC000217831870 DG In-Stock Unstable MMP9 19 42 CC[C@@H](C)[C@@H](CO)NC(=O)CCCc1c[nH]c2ccccc12 ZINC000217831870 DG In-Stock Unstable MC1R 54 39 CC[C@@H](C)[C@@H](CO)NC(=O)CCCc1c[nH]c2ccccc12 ZINC000217831870 DG In-Stock Unstable MMP7 0 40 CC[C@@H](C)[C@@H](CO)NC(=O)CCCc1c[nH]c2ccccc12 ZINC000217831870 DG In-Stock Unstable MMP1 21 40 CC[C@@H](C)[C@@H](CO)NC(=O)CCCc1c[nH]c2ccccc12 ZINC000217831870 DG In-Stock Unstable NPR 29 40 CC[C@@H](C)[C@@H](CO)NC(=O)CCCc1c[nH]c2ccccc12 ZINC000217831870 DG In-Stock Unstable KISS1R 50 32 OC1=NN=C(c2cccnc2)[C@@H]2C[C@H]12 ZINC000217831893 AD In-Stock Unstable CYP2A6 42 38 O=C(N[C@@H]1CCN(Cc2ccccc2)C1)[C@H]1C[C@@H](O)CN1 ZINC000217831898 CC On-Demand Unstable DRD4 34 49 O=C(N[C@@H]1CCN(Cc2ccccc2)C1)[C@H]1C[C@@H](O)CN1 ZINC000217831898 CC On-Demand Unstable DRD3 24 47 O=C(N[C@@H]1CCN(Cc2ccccc2)C1)[C@H]1C[C@@H](O)CN1 ZINC000217831898 CC On-Demand Unstable SIGMAR1 46 51 O=C(N[C@@H]1CCN(Cc2ccccc2)C1)[C@H]1C[C@@H](O)CN1 ZINC000217831898 CC On-Demand Unstable CCR3 30 48 O=C(N[C@@H]1CCN(Cc2ccccc2)C1)[C@H]1C[C@@H](O)CN1 ZINC000217831898 CC On-Demand Unstable MCHR1 27 52 O=C(N[C@@H]1CCN(Cc2ccccc2)C1)[C@H]1C[C@@H](O)CN1 ZINC000217831898 CC On-Demand Unstable BIRC2 30 41 O=C(N[C@@H]1CCN(Cc2ccccc2)C1)[C@H]1C[C@@H](O)CN1 ZINC000217831898 CC On-Demand Unstable ADIPOR1 0 41 O=C(N[C@@H]1CCN(Cc2ccccc2)C1)[C@H]1C[C@@H](O)CN1 ZINC000217831898 CC On-Demand Unstable ADIPOR2 0 41 Oc1cccc2c1CC[C@@H]2N1CC[C@@H](c2ccccc2)C1 ZINC000217831941 CH For-Sale Unstable SLC6A1 0 48 Oc1cccc2c1CC[C@@H]2N1CC[C@@H](c2ccccc2)C1 ZINC000217831941 CH For-Sale Unstable SLC18A3 63 41 COc1ccc(OC2CCN(C(=O)c3n[nH]c(N)c3Cl)CC2)cc1 ZINC000217831950 FE In-Stock Unstable HRH1 35 41 COc1ccc(OC2CCN(C(=O)c3n[nH]c(N)c3Cl)CC2)cc1 ZINC000217831950 FE In-Stock Unstable PRSS2 57 33 COc1ccc(OC2CCN(C(=O)c3n[nH]c(N)c3Cl)CC2)cc1 ZINC000217831950 FE In-Stock Unstable HRH3 25 42 COc1ccc(OC2CCN(C(=O)c3n[nH]c(N)c3Cl)CC2)cc1 ZINC000217831950 FE In-Stock Unstable CCR3 28 41 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc2nc[nH]c2c1 ZINC000217831964 DF For-Sale Unstable PLD2 48 35 OC1=NN=C(c2cccnc2)[C@H]2C[C@H]12 ZINC000217831965 AD In-Stock Unstable CYP2A6 42 38 Cc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)COc1ccc(Cl)cc1 ZINC000217831972 FI In-Stock Unstable TRAR 33 48 O=C(N/C=C/c1ccccc1Cl)Nc1ccc(Cl)cn1 ZINC000217832008 DI For-Sale Anodyne LUCI_LUCLA 33 44 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc2nc[nH]c2c1 ZINC000217832013 DF For-Sale Unstable PLD2 48 35 C[C@@H](c1ccc(O)cc1)N1CC[C@@H](c2ccccc2)C1 ZINC000217832020 CH For-Sale Unstable SLC18A3 43 40 C[C@@H](c1ccc(O)cc1)N1CC[C@@H](c2ccccc2)C1 ZINC000217832020 CH For-Sale Unstable GRIN2C 18 45 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)c3ccccc3OC(F)(F)F)C2)n1 ZINC000217832059 IK In-Stock Unstable HRH3 15 42 Cc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)COc1ccc(Cl)cc1 ZINC000217832075 FI In-Stock Unstable TRAR 33 48 O=C(c1ccccc1Cl)N1C[C@H]2CNC[C@@H](C2)C1 ZINC000217832097 CE For-Sale Unstable P2RX7 23 41 O=C(c1ccccc1Cl)N1C[C@H]2CNC[C@@H](C2)C1 ZINC000217832097 CE For-Sale Unstable CHRNA7 34 56 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)c3ccccc3OC(F)(F)F)C2)n1 ZINC000217832098 IK In-Stock Unstable HRH3 15 42 C[C@H](c1ccc(O)cc1)N1CC[C@@H](c2ccccc2)C1 ZINC000217832113 CH For-Sale Unstable SLC18A3 43 40 C[C@H](c1ccc(O)cc1)N1CC[C@@H](c2ccccc2)C1 ZINC000217832113 CH For-Sale Unstable GRIN2C 18 45 O=C(N/C=C/c1ccccc1Cl)Nc1cc(Cl)ccn1 ZINC000217832128 DI For-Sale Anodyne JAK1 0 41 O=C(N/C=C/c1ccccc1Cl)Nc1cc(Cl)ccn1 ZINC000217832128 DI For-Sale Anodyne TYK2 66 39 CC[C@@H](CCO)N[C@@H]1CCCCNC1=O ZINC000217832173 BC For-Sale Unstable MMP1 0 42 O=C(c1cccc(N2CCOCC2)c1)N1CCC[C@@H]1c1ccc(F)cc1 ZINC000217832174 FH In-Stock Unstable KCNA5 19 43 O=C(c1cccc(N2CCOCC2)c1)N1CCC[C@@H]1c1ccc(F)cc1 ZINC000217832174 FH In-Stock Unstable PREP 20 40 O=C(c1cccc(N2CCOCC2)c1)N1CCC[C@@H]1c1ccc(F)cc1 ZINC000217832174 FH In-Stock Unstable GRM5 0 46 O=C(c1cccc(N2CCOCC2)c1)N1CCC[C@@H]1c1ccc(F)cc1 ZINC000217832174 FH In-Stock Unstable AKR1C3 0 43 CN1CC[C@@H](NC(=O)c2ccc3c(c2)CC(=O)N3)C1 ZINC000217832177 CC For-Sale Unstable HTR1F 48 36 CN1CC[C@@H](NC(=O)c2ccc3c(c2)CC(=O)N3)C1 ZINC000217832177 CC For-Sale Unstable MAPK14 28 43 CN1CC[C@@H](NC(=O)c2ccc3c(c2)CC(=O)N3)C1 ZINC000217832177 CC For-Sale Unstable UTS2R 22 43 CN1CC[C@@H](NC(=O)c2ccc3c(c2)CC(=O)N3)C1 ZINC000217832177 CC For-Sale Unstable SLC6A5 31 41 CN1CC[C@@H](NC(=O)c2ccc3c(c2)CC(=O)N3)C1 ZINC000217832177 CC For-Sale Unstable HDAC9 22 40 COc1ccc2c(c1)[C@@H](NC(=O)COc1ccc(Cl)cc1)CC(C)(C)O2 ZINC000217832178 GI In-Stock Unstable TRAR 33 48 C[C@@H](c1ccc(F)cc1O)N1CC[C@@H](c2ccccc2)C1 ZINC000217832215 CI For-Sale Unstable CCR5 101 36 C[C@@H](c1ccc(F)cc1O)N1CC[C@@H](c2ccccc2)C1 ZINC000217832215 CI For-Sale Unstable SLC18A3 36 40 O=C(N/C=C/c1ccccc1Cl)Nc1cc(Br)ccn1 ZINC000217832232 FI For-Sale Anodyne TYK2 72 37 O=C(c1cccc(N2CCOCC2)c1)N1CCC[C@H]1c1ccc(F)cc1 ZINC000217832248 FH In-Stock Unstable KCNA5 19 43 O=C(c1cccc(N2CCOCC2)c1)N1CCC[C@H]1c1ccc(F)cc1 ZINC000217832248 FH In-Stock Unstable PREP 20 40 O=C(c1cccc(N2CCOCC2)c1)N1CCC[C@H]1c1ccc(F)cc1 ZINC000217832248 FH In-Stock Unstable GRM5 0 46 O=C(c1cccc(N2CCOCC2)c1)N1CCC[C@H]1c1ccc(F)cc1 ZINC000217832248 FH In-Stock Unstable AKR1C3 0 43 CC[C@H](CCO)N[C@@H]1CCCCNC1=O ZINC000217832249 BC For-Sale Unstable MMP1 0 42 O=C(c1cccc(Cl)c1)N1C[C@H]2CNC[C@@H](C2)C1 ZINC000217832262 CE For-Sale Unstable CHRNA7 25 54 O=C(c1cccc(Cl)c1)N1C[C@H]2CNC[C@@H](C2)C1 ZINC000217832262 CE For-Sale Unstable CCKBR 16 40 COc1ccc2c(c1)[C@H](NC(=O)COc1ccc(Cl)cc1)CC(C)(C)O2 ZINC000217832263 GI In-Stock Unstable TRAR 33 48 CN1CC[C@H](NC(=O)c2ccc3c(c2)CC(=O)N3)C1 ZINC000217832274 CC For-Sale Unstable HTR1F 48 36 CN1CC[C@H](NC(=O)c2ccc3c(c2)CC(=O)N3)C1 ZINC000217832274 CC For-Sale Unstable MAPK14 28 43 CN1CC[C@H](NC(=O)c2ccc3c(c2)CC(=O)N3)C1 ZINC000217832274 CC For-Sale Unstable UTS2R 22 43 CN1CC[C@H](NC(=O)c2ccc3c(c2)CC(=O)N3)C1 ZINC000217832274 CC For-Sale Unstable SLC6A5 31 41 CN1CC[C@H](NC(=O)c2ccc3c(c2)CC(=O)N3)C1 ZINC000217832274 CC For-Sale Unstable HDAC9 22 40 C[C@H](c1ccc(F)cc1O)N1CC[C@@H](c2ccccc2)C1 ZINC000217832302 CI For-Sale Unstable CCR5 101 36 C[C@H](c1ccc(F)cc1O)N1CC[C@@H](c2ccccc2)C1 ZINC000217832302 CI For-Sale Unstable SLC18A3 36 40 O=C(/C=C/c1ccc(Cl)cc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217832327 EI For-Sale Unstable MMP2 15 44 O=C(/C=C/c1ccc(Cl)cc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217832327 EI For-Sale Unstable CCR2 16 44 CC[C@@H](CCO)N[C@H]1CCCCNC1=O ZINC000217832335 BC For-Sale Unstable MMP1 0 42 O=C(N/C=C/c1ccccc1Cl)NCCCc1ccccc1 ZINC000217832340 DI For-Sale Unstable MTNR1A 15 41 O=C(N/C=C/c1ccccc1Cl)NCCCc1ccccc1 ZINC000217832340 DI For-Sale Unstable MTNR1B 28 41 O=C(N/C=C/c1ccccc1Cl)NCCCc1ccccc1 ZINC000217832340 DI For-Sale Unstable SCN5A 0 45 O=C(N/C=C/c1ccccc1Cl)NCCCc1ccccc1 ZINC000217832340 DI For-Sale Unstable AMP1_PLAFQ 27 42 O=C(N/C=C/c1ccccc1Cl)NCCCc1ccccc1 ZINC000217832340 DI For-Sale Unstable CRTM 43 38 C[C@@H](O)C1CCN(CCCOc2cccc(C#N)c2)CC1 ZINC000217832369 CE On-Demand Unstable HRH2 23 44 C[C@@H](O)C1CCN(CCCOc2cccc(C#N)c2)CC1 ZINC000217832369 CE On-Demand Unstable SLC6A4 22 46 C[C@@H](O)C1CCN(CCCOc2cccc(C#N)c2)CC1 ZINC000217832369 CE On-Demand Unstable HRH3 78 47 C[C@@H](O)C1CCN(CCCOc2cccc(C#N)c2)CC1 ZINC000217832369 CE On-Demand Unstable CHRNA10 57 52 C[C@@H](O)C1CCN(CCCOc2cccc(C#N)c2)CC1 ZINC000217832369 CE On-Demand Unstable MEN1 64 46 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)COc1ccc(Cl)cc1 ZINC000217832386 GI In-Stock Unstable TRAR 33 48 CC[C@H](CCO)N[C@H]1CCCCNC1=O ZINC000217832391 BC For-Sale Unstable MMP1 0 42 C[C@@H](Cc1ccc(O)cc1)N1CC[C@@H](c2ccccc2)C1 ZINC000217832394 CH For-Sale Unstable CCR5 23 40 C[C@@H](Cc1ccc(O)cc1)N1CC[C@@H](c2ccccc2)C1 ZINC000217832394 CH For-Sale Unstable SLC18A3 45 43 C[C@@H](Cc1ccc(O)cc1)N1CC[C@@H](c2ccccc2)C1 ZINC000217832394 CH For-Sale Unstable GRIN2C 17 43 O=C(/C=C/c1ccc(Cl)cc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217832403 EI For-Sale Unstable MMP2 15 44 O=C(/C=C/c1ccc(Cl)cc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217832403 EI For-Sale Unstable CCR2 16 44 O=C(c1ccc(Cl)cc1)N1C[C@H]2CNC[C@@H](C2)C1 ZINC000217832408 CE For-Sale Unstable CHRNA7 35 66 O=C(c1ccc(Cl)cc1)N1C[C@H]2CNC[C@@H](C2)C1 ZINC000217832408 CE For-Sale Unstable L3MBTL3 47 38 O=C(N/C=C/c1ccccc1Cl)NCCCCc1ccccc1 ZINC000217832432 EJ For-Sale Unstable SCNN1A 53 40 O=C(N/C=C/c1ccccc1Cl)NCCCCc1ccccc1 ZINC000217832432 EJ For-Sale Unstable MTNR1A 16 40 O=C(N/C=C/c1ccccc1Cl)NCCCCc1ccccc1 ZINC000217832432 EJ For-Sale Unstable MTNR1B 26 40 O=C(N/C=C/c1ccccc1Cl)NCCCCc1ccccc1 ZINC000217832432 EJ For-Sale Unstable FAAH 30 41 O=C(N/C=C/c1ccccc1Cl)NCCCCc1ccccc1 ZINC000217832432 EJ For-Sale Unstable AMP1_PLAFQ 22 44 O=C(N/C=C/c1ccccc1Cl)NCCCCc1ccccc1 ZINC000217832432 EJ For-Sale Unstable CRTM 40 35 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)COc1ccc(Cl)cc1 ZINC000217832450 GI In-Stock Unstable TRAR 33 48 C[C@H](O)C1CCN(CCCOc2cccc(C#N)c2)CC1 ZINC000217832455 CE On-Demand Unstable HRH2 23 44 C[C@H](O)C1CCN(CCCOc2cccc(C#N)c2)CC1 ZINC000217832455 CE On-Demand Unstable SLC6A4 22 46 C[C@H](O)C1CCN(CCCOc2cccc(C#N)c2)CC1 ZINC000217832455 CE On-Demand Unstable HRH3 78 47 C[C@H](O)C1CCN(CCCOc2cccc(C#N)c2)CC1 ZINC000217832455 CE On-Demand Unstable CHRNA10 57 52 C[C@H](O)C1CCN(CCCOc2cccc(C#N)c2)CC1 ZINC000217832455 CE On-Demand Unstable MEN1 64 46 C[C@H](Cc1ccc(O)cc1)N1CC[C@@H](c2ccccc2)C1 ZINC000217832457 CH For-Sale Unstable CCR5 23 40 C[C@H](Cc1ccc(O)cc1)N1CC[C@@H](c2ccccc2)C1 ZINC000217832457 CH For-Sale Unstable SLC18A3 45 43 C[C@H](Cc1ccc(O)cc1)N1CC[C@@H](c2ccccc2)C1 ZINC000217832457 CH For-Sale Unstable GRIN2C 17 43 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc2[nH]ccc2c1 ZINC000217832493 DH In-Stock Unstable HCRTR1 16 40 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc2[nH]ccc2c1 ZINC000217832493 DH In-Stock Unstable PLD1 45 36 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc2[nH]ccc2c1 ZINC000217832493 DH In-Stock Unstable PLD2 49 36 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc2[nH]ccc2c1 ZINC000217832493 DH In-Stock Unstable HCRTR2 15 40 CC[C@@H](c1ccccc1O)N1CC[C@@H](c2ccccc2)C1 ZINC000217832542 CI For-Sale Unstable VACHT_TETCF 0 40 CC[C@@H](c1ccccc1O)N1CC[C@@H](c2ccccc2)C1 ZINC000217832542 CI For-Sale Unstable CCR5 29 44 CC[C@@H](c1ccccc1O)N1CC[C@@H](c2ccccc2)C1 ZINC000217832542 CI For-Sale Unstable SLC18A3 53 50 COc1ccc(C(=O)N[C@@H](C)c2ccc(C)s2)c(F)c1 ZINC000217832543 CH On-Demand Unstable GPR35 26 41 CN(CC(=O)N(C)C)Cc1ccccc1/C=C\C(=O)O ZINC000217832546 CD For-Sale Unstable PTGER2 17 40 CN(CC(=O)N(C)C)Cc1ccccc1/C=C\C(=O)O ZINC000217832546 CD For-Sale Unstable PTGER4 20 40 CN(CC(=O)N(C)C)Cc1ccccc1/C=C\C(=O)O ZINC000217832546 CD For-Sale Unstable PTGER3 19 49 C[C@@H](O)C1CCN(C[C@@H](O)c2ccc(C#N)cc2)CC1 ZINC000217832565 CD On-Demand Unstable O19067_PIG 0 40 CC[C@@H](NC(=O)COc1ccc(Cl)cc1)c1ccc(C)c(C)c1 ZINC000217832566 EJ In-Stock Unstable UTS2 43 34 CC[C@@H](NC(=O)COc1ccc(Cl)cc1)c1ccc(C)c(C)c1 ZINC000217832566 EJ In-Stock Unstable PDS 45 36 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc2[nH]ccc2c1 ZINC000217832574 DH In-Stock Unstable HCRTR1 16 40 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc2[nH]ccc2c1 ZINC000217832574 DH In-Stock Unstable PLD1 45 36 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc2[nH]ccc2c1 ZINC000217832574 DH In-Stock Unstable PLD2 49 36 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc2[nH]ccc2c1 ZINC000217832574 DH In-Stock Unstable HCRTR2 15 40 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)Nc3ccccc3F)C2)n1 ZINC000217832604 GJ In-Stock Unstable HRH3 20 44 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)Nc3ccccc3F)C2)n1 ZINC000217832604 GJ In-Stock Unstable Q8MHZ5_SHEEP 49 32 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)Nc3ccccc3F)C2)n1 ZINC000217832604 GJ In-Stock Unstable SMO 37 40 CC[C@H](c1ccccc1O)N1CC[C@@H](c2ccccc2)C1 ZINC000217832614 CI For-Sale Unstable VACHT_TETCF 0 40 CC[C@H](c1ccccc1O)N1CC[C@@H](c2ccccc2)C1 ZINC000217832614 CI For-Sale Unstable CCR5 29 44 CC[C@H](c1ccccc1O)N1CC[C@@H](c2ccccc2)C1 ZINC000217832614 CI For-Sale Unstable SLC18A3 53 50 CC[C@H](NC(=O)COc1ccc(Cl)cc1)c1ccc(C)c(C)c1 ZINC000217832624 EJ In-Stock Unstable UTS2 43 34 CC[C@H](NC(=O)COc1ccc(Cl)cc1)c1ccc(C)c(C)c1 ZINC000217832624 EJ In-Stock Unstable PDS 45 36 C[C@H](O)C1CCN(C[C@@H](O)c2ccc(C#N)cc2)CC1 ZINC000217832628 CD On-Demand Unstable O19067_PIG 0 40 CCCN(CC)CCNC(=O)CCCCC(=O)O ZINC000217832650 CD For-Sale Unstable FABP2 0 41 CCCN(CC)CCNC(=O)CCCCC(=O)O ZINC000217832650 CD For-Sale Unstable FABP4 16 41 CCCN(CC)CCNC(=O)CCCCC(=O)O ZINC000217832650 CD For-Sale Unstable DNM1 0 53 CCCN(CC)CCNC(=O)CCCCC(=O)O ZINC000217832650 CD For-Sale Unstable EPHX2 0 52 CCCN(CC)CCNC(=O)CCCCC(=O)O ZINC000217832650 CD For-Sale Unstable FABP5 15 41 CCCN(CC)CCNC(=O)CCCCC(=O)O ZINC000217832650 CD For-Sale Unstable SLC22A20 0 42 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc2cc[nH]c2c1 ZINC000217832667 DH For-Sale Unstable GRIN2B 22 41 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc2cc[nH]c2c1 ZINC000217832667 DH For-Sale Unstable PLD1 46 38 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc2cc[nH]c2c1 ZINC000217832667 DH For-Sale Unstable PLD2 51 38 CN1CCO[C@@H]([C@@H](O)Cc2ccc(Cl)c(Cl)c2)C1 ZINC000217832693 CE For-Sale Unstable SIGMAR1 17 44 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)Nc3ccccc3F)C2)n1 ZINC000217832697 GJ In-Stock Unstable HRH3 20 44 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)Nc3ccccc3F)C2)n1 ZINC000217832697 GJ In-Stock Unstable Q8MHZ5_SHEEP 49 32 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)Nc3ccccc3F)C2)n1 ZINC000217832697 GJ In-Stock Unstable SMO 37 40 C[C@H]1CCCCN1CCCN[C@H](C)c1ccc(Br)cc1Br ZINC000217832700 HK For-Sale Unstable HRH3 42 36 C[C@@H](O)C1CCN(C[C@H](O)c2ccc(C#N)cc2)CC1 ZINC000217832720 CD On-Demand Unstable O19067_PIG 0 40 CCCCN([C@@H](C)CC)[C@H](c1cccc(Cl)c1)[C@@H](N)CC ZINC000217832730 DK For-Sale Unstable OPRL1 0 42 C[C@@H](c1cc(Br)ccc1O)N1CC[C@@H](c2ccccc2)C1 ZINC000217832732 EJ For-Sale Unstable VACHT_TETCF 0 41 C[C@@H](c1cc(Br)ccc1O)N1CC[C@@H](c2ccccc2)C1 ZINC000217832732 EJ For-Sale Unstable CCR5 15 40 C[C@@H](c1cc(Br)ccc1O)N1CC[C@@H](c2ccccc2)C1 ZINC000217832732 EJ For-Sale Unstable SLC18A3 29 43 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc2cc[nH]c2c1 ZINC000217832738 DH For-Sale Unstable GRIN2B 22 41 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc2cc[nH]c2c1 ZINC000217832738 DH For-Sale Unstable PLD1 46 38 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc2cc[nH]c2c1 ZINC000217832738 DH For-Sale Unstable PLD2 51 38 CN1CCO[C@H]([C@@H](O)Cc2ccc(Cl)c(Cl)c2)C1 ZINC000217832770 CE For-Sale Unstable SIGMAR1 17 44 CN(Cc1ccco1)Cc1ccccc1/C=C\C(=O)O ZINC000217832782 CG For-Sale Unstable PTGER2 42 45 CN(Cc1ccco1)Cc1ccccc1/C=C\C(=O)O ZINC000217832782 CG For-Sale Unstable PTGER4 0 45 CN(Cc1ccco1)Cc1ccccc1/C=C\C(=O)O ZINC000217832782 CG For-Sale Unstable PTGER3 16 46 C[C@H](c1cc(Br)ccc1O)N1CC[C@@H](c2ccccc2)C1 ZINC000217832797 EJ For-Sale Unstable VACHT_TETCF 0 41 C[C@H](c1cc(Br)ccc1O)N1CC[C@@H](c2ccccc2)C1 ZINC000217832797 EJ For-Sale Unstable CCR5 15 40 C[C@H](c1cc(Br)ccc1O)N1CC[C@@H](c2ccccc2)C1 ZINC000217832797 EJ For-Sale Unstable SLC18A3 29 43 C[C@H](O)C1CCN(C[C@H](O)c2ccc(C#N)cc2)CC1 ZINC000217832802 CD On-Demand Unstable O19067_PIG 0 40 CCCCN([C@H](C)CC)[C@H](c1cccc(Cl)c1)[C@@H](N)CC ZINC000217832814 DK For-Sale Unstable OPRL1 0 42 C[C@H]1CCCCN1CCCN[C@H](C)c1ccc(I)cc1 ZINC000217832839 GI For-Sale Unstable HRH3 50 38 O=C(C[C@@H]1NC(=O)N(CCc2cccc(F)c2)C1=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217832846 JD In-Stock Unstable CHRNA4 29 48 O=C(CCCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217832857 DH For-Sale Unstable FKBP1A 35 42 O=C(CCCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217832857 DH For-Sale Unstable SLC18A2 46 39 O=C(CCCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217832857 DH For-Sale Unstable PREP 76 45 O=C(CCCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217832857 DH For-Sale Unstable MTNR1A 20 41 O=C(CCCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217832857 DH For-Sale Unstable MTNR1B 18 41 O=C(N/C=C/c1ccccc1Cl)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217832871 HG For-Sale Unstable TGM2 71 41 O=C(N/C=C/c1ccccc1Cl)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217832871 HG For-Sale Unstable F13A1 89 41 O=C(N/C=C/c1ccccc1Cl)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217832871 HG For-Sale Unstable AKR1C3 47 41 C[C@@H](c1ccccc1O)N1CC[C@@H](c2ccccc2)C1 ZINC000217832904 CH For-Sale Unstable VACHT_TETCF 0 41 C[C@@H](c1ccccc1O)N1CC[C@@H](c2ccccc2)C1 ZINC000217832904 CH For-Sale Unstable CCR5 17 46 C[C@@H](c1ccccc1O)N1CC[C@@H](c2ccccc2)C1 ZINC000217832904 CH For-Sale Unstable SLC18A3 49 43 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable PLG 19 41 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable KLKB1 15 41 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable ACE 74 54 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable SSTR2 53 38 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable OPRM1 78 52 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable OPRD1 96 52 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable OPRK1 22 45 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable MME 164 54 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable LTA4H 23 44 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable ANPEP 104 44 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable EDNRA 18 42 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable TACR1 35 53 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable CTSD 42 48 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable PGC 70 48 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable CTRA_BOVIN 26 42 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable FCER2 104 41 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable CASP3 16 43 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable BMP1 70 38 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable TACR2 48 48 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable RNPEP 36 44 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable KLK3 89 38 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable CTSB 112 55 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable SRC 18 43 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable PAPA1_CARPA 110 53 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable CYSP_TRYCR 90 48 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable CCKAR 68 41 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable CTSK 44 52 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable CTSL 85 53 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable CPA1 44 45 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable CACNA1B 53 50 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable CCR3 32 57 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable PGA 64 48 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable F2R 51 50 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable NPFFR2 74 39 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable TIMP3 83 41 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable HLA-A 54 49 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable CTRB1 42 52 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable SCN9A 23 41 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable TACR3 34 48 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable MC3R 52 33 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable MC5R 45 33 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable CAPNS1 82 45 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable MMP2 34 46 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable MMP3 56 45 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable MMP8 37 45 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable GRIA1 51 38 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable MMP14 43 35 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable ECE1 31 40 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable HLA-DRB1 106 56 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable REN 121 54 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable REN1 53 49 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable LNPEP 22 44 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable FURIN 57 37 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable CCKBR 38 47 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable CTSS 40 53 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable GHSR 29 48 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable CAPN1 136 52 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable MMP9 37 49 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable CASP1 33 41 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable CTRC 21 41 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable CAPN2 152 49 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable CTSE 41 39 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable ACE2 94 45 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable MC1R 83 36 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable BACE1 20 41 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable LAP3 55 44 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable PROTEASE 15 41 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable MMP7 33 41 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable MMP1 58 49 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable FPR1 108 59 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable CTRB_BOVIN 61 43 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable NPR 90 45 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable AMP1_PLAFQ 48 44 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable XIAP 36 47 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable PSMB5 79 42 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable BLA1_STEMA 78 38 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable KISS1R 64 33 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable POLG_WNV 46 31 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable QRFPR 57 38 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable PSMB8 76 37 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable BRCA1 43 30 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable NPFFR1 79 39 C[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217832913 FC For-Sale Unstable METAP2 22 46 O=C(CCCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217832935 DH For-Sale Unstable FKBP1A 35 42 O=C(CCCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217832935 DH For-Sale Unstable SLC18A2 46 39 O=C(CCCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217832935 DH For-Sale Unstable PREP 76 45 O=C(CCCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217832935 DH For-Sale Unstable MTNR1A 20 41 O=C(CCCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217832935 DH For-Sale Unstable MTNR1B 18 41 CC[C@@H](NC(=O)COc1ccc(Cl)cc1)c1ccc(OC)c(OC)c1 ZINC000217832955 FI In-Stock Unstable PTGER3 16 40 CC[C@@H](NC(=O)COc1ccc(Cl)cc1)c1ccc(OC)c(OC)c1 ZINC000217832955 FI In-Stock Unstable ENPP1 49 35 CC[C@@H](NC(=O)COc1ccc(Cl)cc1)c1ccc(OC)c(OC)c1 ZINC000217832955 FI In-Stock Unstable UTS2 43 38 CC[C@@H](NC(=O)COc1ccc(Cl)cc1)c1ccc(OC)c(OC)c1 ZINC000217832955 FI In-Stock Unstable PDS 45 35 CC(C)[C@H](NCCCN1CCCC[C@@H]1C)c1cccs1 ZINC000217832962 CI For-Sale Unstable HRH3 41 42 Cc1ccc(S(=O)(=O)N2CCN(C(=O)N/C=C/c3ccccc3Cl)CC2)cc1 ZINC000217832975 HG For-Sale Unstable EPHX2 17 41 Cc1ccc(S(=O)(=O)N2CCN(C(=O)N/C=C/c3ccccc3Cl)CC2)cc1 ZINC000217832975 HG For-Sale Unstable TGM2 69 41 Cc1ccc(S(=O)(=O)N2CCN(C(=O)N/C=C/c3ccccc3Cl)CC2)cc1 ZINC000217832975 HG For-Sale Unstable F13A1 88 41 C[C@H](c1ccccc1O)N1CC[C@@H](c2ccccc2)C1 ZINC000217832979 CH For-Sale Unstable VACHT_TETCF 0 41 C[C@H](c1ccccc1O)N1CC[C@@H](c2ccccc2)C1 ZINC000217832979 CH For-Sale Unstable CCR5 17 46 C[C@H](c1ccccc1O)N1CC[C@@H](c2ccccc2)C1 ZINC000217832979 CH For-Sale Unstable SLC18A3 49 43 CC[C@H](NC(=O)COc1ccc(Cl)cc1)c1ccc(OC)c(OC)c1 ZINC000217833032 FI In-Stock Unstable PTGER3 16 40 CC[C@H](NC(=O)COc1ccc(Cl)cc1)c1ccc(OC)c(OC)c1 ZINC000217833032 FI In-Stock Unstable ENPP1 49 35 CC[C@H](NC(=O)COc1ccc(Cl)cc1)c1ccc(OC)c(OC)c1 ZINC000217833032 FI In-Stock Unstable UTS2 43 38 CC[C@H](NC(=O)COc1ccc(Cl)cc1)c1ccc(OC)c(OC)c1 ZINC000217833032 FI In-Stock Unstable PDS 45 35 Oc1ccc2c(oc3c(-c4ccc5c(c4)OCO5)c4cn[nH]c4nc32)c1O ZINC000217833065 FH In-Stock Unstable CLK4 46 35 COc1ccc(OCC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217833074 EF For-Sale Unstable COLA 95 41 COc1ccc(OCC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217833074 EF For-Sale Unstable CPT1A 87 41 COc1ccc(OCC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217833074 EF For-Sale Unstable MTNR1B 44 32 COc1ccc(OCC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217833074 EF For-Sale Unstable MCHR1 19 41 COc1ccc(OCC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217833074 EF For-Sale Unstable ACKR3 51 33 C[C@@H](c1cc(F)ccc1O)N1CC[C@@H](c2ccccc2)C1 ZINC000217833094 CI For-Sale Unstable CCR5 87 35 C[C@@H](c1cc(F)ccc1O)N1CC[C@@H](c2ccccc2)C1 ZINC000217833094 CI For-Sale Unstable SLC18A3 37 40 COc1ccc(OCC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217833116 EF For-Sale Unstable COLA 95 41 COc1ccc(OCC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217833116 EF For-Sale Unstable CPT1A 87 41 COc1ccc(OCC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217833116 EF For-Sale Unstable MTNR1B 44 32 COc1ccc(OCC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217833116 EF For-Sale Unstable MCHR1 19 41 COc1ccc(OCC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217833116 EF For-Sale Unstable ACKR3 51 33 C[C@@H]1CN(C)CCN1CCCOc1cccc(C#N)c1 ZINC000217833121 CD On-Demand Unstable HRH3 38 51 C[C@@H]1CN(C)CCN1CCCOc1cccc(C#N)c1 ZINC000217833121 CD On-Demand Unstable MEN1 42 35 CC[C@@H](NC(=O)COc1ccc(Cl)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217833128 GG In-Stock Unstable PTGS2 20 42 CC[C@@H](NC(=O)COc1ccc(Cl)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217833128 GG In-Stock Unstable UTS2 42 35 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)Nc3ccc(C(F)(F)F)cc3)C2)n1 ZINC000217833151 IK In-Stock Unstable TRPV1 18 49 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)Nc3ccc(C(F)(F)F)cc3)C2)n1 ZINC000217833151 IK In-Stock Unstable HRH3 18 41 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)Nc3ccc(C(F)(F)F)cc3)C2)n1 ZINC000217833151 IK In-Stock Unstable EPHX2 40 47 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)Nc3ccc(C(F)(F)F)cc3)C2)n1 ZINC000217833151 IK In-Stock Unstable P2RY14 40 37 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)Nc3ccc(C(F)(F)F)cc3)C2)n1 ZINC000217833151 IK In-Stock Unstable TRPM8 44 39 C[C@H](c1cc(F)ccc1O)N1CC[C@@H](c2ccccc2)C1 ZINC000217833181 CI For-Sale Unstable CCR5 87 35 C[C@H](c1cc(F)ccc1O)N1CC[C@@H](c2ccccc2)C1 ZINC000217833181 CI For-Sale Unstable SLC18A3 37 40 C[C@H]1CN(C)CCN1CCCOc1cccc(C#N)c1 ZINC000217833202 CD On-Demand Unstable HRH3 38 51 C[C@H]1CN(C)CCN1CCCOc1cccc(C#N)c1 ZINC000217833202 CD On-Demand Unstable MEN1 42 35 CC[C@H](NC(=O)COc1ccc(Cl)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217833224 GG In-Stock Unstable PTGS2 15 42 CC[C@H](NC(=O)COc1ccc(Cl)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217833224 GG In-Stock Unstable UTS2 42 35 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)Nc3ccc(C(F)(F)F)cc3)C2)n1 ZINC000217833227 IK In-Stock Unstable TRPV1 18 49 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)Nc3ccc(C(F)(F)F)cc3)C2)n1 ZINC000217833227 IK In-Stock Unstable HRH3 18 41 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)Nc3ccc(C(F)(F)F)cc3)C2)n1 ZINC000217833227 IK In-Stock Unstable EPHX2 40 47 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)Nc3ccc(C(F)(F)F)cc3)C2)n1 ZINC000217833227 IK In-Stock Unstable P2RY14 40 37 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)Nc3ccc(C(F)(F)F)cc3)C2)n1 ZINC000217833227 IK In-Stock Unstable TRPM8 44 39 Cc1ccc(O)c([C@@H](C)N2CC[C@@H](c3ccccc3)C2)c1 ZINC000217833248 CI For-Sale Unstable CCR5 17 41 COCCNC(=O)CCNC(=O)c1ccc(=O)[nH]n1 ZINC000217833269 CA For-Sale Unstable ALPL 20 41 C[C@H]1CCCCN1CCCN[C@H](C)c1ccc(F)cc1Cl ZINC000217833281 DI For-Sale Unstable HRH3 47 39 COc1cn(CC(=O)N2CCc3c([nH]c4ccccc34)C2)c(C)cc1=O ZINC000217833310 FE In-Stock Unstable DRD5 21 41 COc1cn(CC(=O)N2CCc3c([nH]c4ccccc34)C2)c(C)cc1=O ZINC000217833310 FE In-Stock Unstable CYP1B1 15 41 Cc1ccc(O)c([C@H](C)N2CC[C@@H](c3ccccc3)C2)c1 ZINC000217833317 CI For-Sale Unstable CCR5 17 41 Cc1ccccc1NC(=O)N1CCC[C@@H](Cc2nc(-c3ccccc3C)no2)C1 ZINC000217833330 GJ In-Stock Unstable HRH3 18 41 Cc1ccccc1NC(=O)N1CCC[C@@H](Cc2nc(-c3ccccc3C)no2)C1 ZINC000217833330 GJ In-Stock Unstable Q8MHZ5_SHEEP 42 32 Cc1ccccc1NC(=O)N1CCC[C@@H](Cc2nc(-c3ccccc3C)no2)C1 ZINC000217833330 GJ In-Stock Unstable SMO 47 46 O=C(O)/C=C\c1ccccc1CN1CCCCCCC1=O ZINC000217833367 CG For-Sale Unstable PTGER2 44 50 O=C(O)/C=C\c1ccccc1CN1CCCCCCC1=O ZINC000217833367 CG For-Sale Unstable PTGER4 23 48 O=C(O)/C=C\c1ccccc1CN1CCCCCCC1=O ZINC000217833367 CG For-Sale Unstable PTGER3 19 50 COc1ccc(-c2noc(CNC(=O)COc3ccc(Cl)cc3)n2)c(OC)c1 ZINC000217833378 HG In-Stock Unstable MTNR1A 46 38 Oc1ccc2c(c1)OC[C@@H]2N1CC[C@@H](c2ccccc2)C1 ZINC000217833390 CG For-Sale Unstable SLC18A3 46 38 C[C@H]1CCCCN1CCCN[C@H](C)c1ccc(F)c(Br)c1 ZINC000217833405 FJ For-Sale Unstable HRH3 40 39 Cc1ccccc1NC(=O)N1CCC[C@H](Cc2nc(-c3ccccc3C)no2)C1 ZINC000217833425 GJ In-Stock Unstable HRH3 18 41 Cc1ccccc1NC(=O)N1CCC[C@H](Cc2nc(-c3ccccc3C)no2)C1 ZINC000217833425 GJ In-Stock Unstable Q8MHZ5_SHEEP 42 32 Cc1ccccc1NC(=O)N1CCC[C@H](Cc2nc(-c3ccccc3C)no2)C1 ZINC000217833425 GJ In-Stock Unstable SMO 47 46 CC(C)(C)OC(=O)NCCNC(=O)N/C=C/c1ccccc1Cl ZINC000217833473 EG For-Sale Unstable ECR 42 33 O=C(NC[C@H]1CCCN1c1ccccc1)c1cc(Br)ccc1Cl ZINC000217833474 GJ For-Sale Unstable DRD2 35 49 O=C(NC[C@H]1CCCN1c1ccccc1)c1cc(Br)ccc1Cl ZINC000217833474 GJ For-Sale Unstable DRD3 15 47 O=C(NC[C@H]1CCCN1c1ccccc1)c1cc(Br)ccc1Cl ZINC000217833474 GJ For-Sale Unstable CCR3 15 41 CC[C@@H](c1ccc(O)cc1)N1CC[C@@H](c2ccccc2)C1 ZINC000217833501 CI For-Sale Unstable VACHT_TETCF 0 44 CC[C@@H](c1ccc(O)cc1)N1CC[C@@H](c2ccccc2)C1 ZINC000217833501 CI For-Sale Unstable CCR5 16 40 CC[C@@H](c1ccc(O)cc1)N1CC[C@@H](c2ccccc2)C1 ZINC000217833501 CI For-Sale Unstable SLC18A3 45 46 CC[C@@H](c1ccc(O)cc1)N1CC[C@@H](c2ccccc2)C1 ZINC000217833501 CI For-Sale Unstable GRIN2C 17 43 O=C(COc1ccc(Cl)cc1)NCc1nc(-c2cccc(Br)c2)no1 ZINC000217833505 HH In-Stock Unstable TPSAB1 40 33 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)NCc3ccc(F)cc3)C2)n1 ZINC000217833511 HI In-Stock Unstable HRH3 20 41 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)NCc3ccc(F)cc3)C2)n1 ZINC000217833511 HI In-Stock Unstable CCR3 120 39 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)NCc3ccc(F)cc3)C2)n1 ZINC000217833511 HI In-Stock Unstable NPSR1 25 41 CC(C)[C@H](NCCCN1CCCC[C@@H]1C)c1ccccc1 ZINC000217833514 CI For-Sale Unstable HRH3 51 39 CC(C)(C)OC(=O)Nc1ccc(C=O)c(Cl)c1 ZINC000217833548 CG For-Sale Unstable AGPAT2 41 38 CC(C)(C)OC(=O)Nc1ccc(C=O)c(Cl)c1 ZINC000217833548 CG For-Sale Unstable F13A1 21 40 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cc(Br)ccc1Cl ZINC000217833564 GJ For-Sale Unstable DRD2 35 49 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cc(Br)ccc1Cl ZINC000217833564 GJ For-Sale Unstable DRD3 15 47 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cc(Br)ccc1Cl ZINC000217833564 GJ For-Sale Unstable CCR3 15 41 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)NCc3ccc(F)cc3)C2)n1 ZINC000217833565 HI In-Stock Unstable HRH3 20 41 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)NCc3ccc(F)cc3)C2)n1 ZINC000217833565 HI In-Stock Unstable CCR3 120 39 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)NCc3ccc(F)cc3)C2)n1 ZINC000217833565 HI In-Stock Unstable NPSR1 25 41 CC(C)c1nccn1Cc1ccccc1/C=C\C(=O)O ZINC000217833566 CG For-Sale Unstable PTGER2 47 43 CC(C)c1nccn1Cc1ccccc1/C=C\C(=O)O ZINC000217833566 CG For-Sale Unstable PTGER4 24 43 CC(C)c1nccn1Cc1ccccc1/C=C\C(=O)O ZINC000217833566 CG For-Sale Unstable PTGER3 23 43 CC[C@H](c1ccc(O)cc1)N1CC[C@@H](c2ccccc2)C1 ZINC000217833571 CI For-Sale Unstable VACHT_TETCF 0 44 CC[C@H](c1ccc(O)cc1)N1CC[C@@H](c2ccccc2)C1 ZINC000217833571 CI For-Sale Unstable CCR5 16 40 CC[C@H](c1ccc(O)cc1)N1CC[C@@H](c2ccccc2)C1 ZINC000217833571 CI For-Sale Unstable SLC18A3 45 46 CC[C@H](c1ccc(O)cc1)N1CC[C@@H](c2ccccc2)C1 ZINC000217833571 CI For-Sale Unstable GRIN2C 17 43 CC(C)(C)OC(=O)N1CCN(C(=O)N/C=C/c2ccccc2Cl)CC1 ZINC000217833586 FH For-Sale Unstable F13A1 16 42 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCc1ccccn1 ZINC000217833593 GD In-Stock Unstable MC4R 30 41 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCc1ccccn1 ZINC000217833593 GD In-Stock Unstable CCKAR 15 40 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCc1ccccn1 ZINC000217833593 GD In-Stock Unstable MMP8 18 44 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCc1ccccn1 ZINC000217833593 GD In-Stock Unstable GHSR 32 41 Nc1ccc(C(=O)N2CCC(c3ccncc3)CC2)cn1 ZINC000217833597 CE In-Stock Unstable SLC9A1 30 42 Nc1ccc(C(=O)N2CCC(c3ccncc3)CC2)cn1 ZINC000217833597 CE In-Stock Unstable PTR1 46 37 Nc1ccc(C(=O)N2CCC(c3ccncc3)CC2)cn1 ZINC000217833597 CE In-Stock Unstable L3MBTL1 0 44 Nc1ccc(C(=O)N2CCC(c3ccncc3)CC2)cn1 ZINC000217833597 CE In-Stock Unstable L3MBTL3 59 38 Nc1ccc(C(=O)N2CCC(c3ccncc3)CC2)cn1 ZINC000217833597 CE In-Stock Unstable SLC6A7 0 44 C[C@@H](c1cc(Cl)ccc1O)N1CC[C@@H](c2ccccc2)C1 ZINC000217833652 DJ For-Sale Unstable PRCP 16 40 C[C@@H](c1cc(Cl)ccc1O)N1CC[C@@H](c2ccccc2)C1 ZINC000217833652 DJ For-Sale Unstable CCR1 41 39 C[C@@H](c1cc(Cl)ccc1O)N1CC[C@@H](c2ccccc2)C1 ZINC000217833652 DJ For-Sale Unstable CCR5 18 40 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable ACE 25 54 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable TYR 15 43 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable SSTR2 97 59 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable OPRM1 25 54 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable OPRD1 21 54 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable GHRHR 30 41 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable MME 42 52 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable EDNRB 55 40 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable EDNRA 50 63 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable TACR1 42 57 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable PGC 42 36 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable MC4R 59 47 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable CTSB 26 51 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable PAPA1_CARPA 47 43 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable CCKAR 155 56 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable CTSL 38 51 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable PGA 27 55 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable BRS3 33 56 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable TIMP3 15 53 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable C3AR1 21 47 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable NMBR 70 54 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable MC3R 80 44 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable MC5R 78 43 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable CAPNS1 47 32 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable MMP2 34 52 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable MMP8 49 49 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable GRIA1 23 40 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable MMP14 28 49 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable GRPR 116 47 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable ECE1 74 52 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable HLA-DRB1 80 41 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable REN 63 52 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable REN1 37 55 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable LNPEP 27 40 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable SSTR3 27 51 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable MMP11 103 44 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable FURIN 15 44 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable CCKBR 120 60 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable GHSR 79 55 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable CAPN1 38 51 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable MMP9 33 53 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable CAPN2 42 43 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable MC1R 113 47 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable ADAM9 48 49 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable CTSC 15 49 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable ST14 15 45 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable MMP7 20 48 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable MMP1 30 52 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable FPR1 63 62 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable NPR 40 52 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable ADAM12 16 49 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable KISS1R 91 43 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable ERAP2 48 45 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable PSMB8 29 42 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable TMPRSS6 18 45 C[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)OC(C)(C)C ZINC000217833675 HD For-Sale Unstable HPN 22 43 CCCCOc1ccc(NC(=O)N2CCC[C@H](Cc3nc(-c4ccccc4C)no3)C2)cc1 ZINC000217833678 IK In-Stock Unstable HRH3 36 47 CCCCOc1ccc(NC(=O)N2CCC[C@H](Cc3nc(-c4ccccc4C)no3)C2)cc1 ZINC000217833678 IK In-Stock Unstable EPHX2 17 41 CCCCOc1ccc(NC(=O)N2CCC[C@H](Cc3nc(-c4ccccc4C)no3)C2)cc1 ZINC000217833678 IK In-Stock Unstable P2RY14 40 38 CC(C)(C)OC(=O)N1CCC(NC(=O)N/C=C/c2ccccc2Cl)CC1 ZINC000217833713 GI For-Sale Unstable EPHX2 42 46 CC(C)(C)OC(=O)N1CCC(NC(=O)N/C=C/c2ccccc2Cl)CC1 ZINC000217833713 GI For-Sale Unstable CCR8 21 42 CC(C)(C)OC(=O)N1CCC(NC(=O)N/C=C/c2ccccc2Cl)CC1 ZINC000217833713 GI For-Sale Unstable GPR119 35 41 CC(C)(C)OC(=O)N1CCC(NC(=O)N/C=C/c2ccccc2Cl)CC1 ZINC000217833713 GI For-Sale Unstable SFRP1 35 40 Cc1cc(=O)c(O)c([C@@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccc(Cl)cc2)o1 ZINC000217833723 JJ In-Stock Unstable SSTR4 44 34 C[C@H](c1cc(Cl)ccc1O)N1CC[C@@H](c2ccccc2)C1 ZINC000217833753 DJ For-Sale Unstable PRCP 16 40 C[C@H](c1cc(Cl)ccc1O)N1CC[C@@H](c2ccccc2)C1 ZINC000217833753 DJ For-Sale Unstable CCR1 41 39 C[C@H](c1cc(Cl)ccc1O)N1CC[C@@H](c2ccccc2)C1 ZINC000217833753 DJ For-Sale Unstable CCR5 18 40 COc1ccc(CN2CCCS2(=O)=O)cc1/C=C\C(=O)O ZINC000217833755 DD For-Sale Unstable PTGER2 23 40 COc1ccc(CN2CCCS2(=O)=O)cc1/C=C\C(=O)O ZINC000217833755 DD For-Sale Unstable PTGER4 0 40 Cc1cc(=O)c(O)c([C@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccc(Cl)cc2)o1 ZINC000217833783 JJ In-Stock Unstable SSTR4 44 34 CCCCOc1ccc(NC(=O)N2CCC[C@@H](Cc3nc(-c4ccccc4C)no3)C2)cc1 ZINC000217833792 IK In-Stock Unstable HRH3 36 47 CCCCOc1ccc(NC(=O)N2CCC[C@@H](Cc3nc(-c4ccccc4C)no3)C2)cc1 ZINC000217833792 IK In-Stock Unstable EPHX2 17 41 CCCCOc1ccc(NC(=O)N2CCC[C@@H](Cc3nc(-c4ccccc4C)no3)C2)cc1 ZINC000217833792 IK In-Stock Unstable P2RY14 40 38 CC(C)c1ccc(CCCNC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217833821 EJ In-Stock Unstable ADRB1 16 41 CC(C)c1ccc(CCCNC(=O)COc2ccc(Cl)cc2)cc1 ZINC000217833821 EJ In-Stock Unstable CRTM 45 47 CCc1c(C)nn(Cc2ccccc2/C=C\C(=O)O)c1C ZINC000217833826 CG For-Sale Unstable PTGER2 42 44 CCc1c(C)nn(Cc2ccccc2/C=C\C(=O)O)c1C ZINC000217833826 CG For-Sale Unstable PTGER4 0 44 CCc1c(C)nn(Cc2ccccc2/C=C\C(=O)O)c1C ZINC000217833826 CG For-Sale Unstable PTGER3 17 44 C[C@@H](c1cccc(O)c1)N1CC[C@@H](c2ccccc2)C1 ZINC000217833839 CH For-Sale Unstable OPRM1 22 53 C[C@@H](c1cccc(O)c1)N1CC[C@@H](c2ccccc2)C1 ZINC000217833839 CH For-Sale Unstable OPRD1 23 53 C[C@@H](c1cccc(O)c1)N1CC[C@@H](c2ccccc2)C1 ZINC000217833839 CH For-Sale Unstable OPRK1 23 43 C[C@@H]1CCc2[nH]c3ccc(C(=O)Nc4ccc(Sc5nncn5C)cc4)cc3c2C1 ZINC000217833848 HJ On-Demand Unstable HTR1F 22 45 C[C@@H]1CCc2[nH]c3ccc(C(=O)Nc4ccc(Sc5nncn5C)cc4)cc3c2C1 ZINC000217833848 HJ On-Demand Unstable MAPKAPK2 22 40 COc1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1OC ZINC000217833850 GI For-Sale Unstable IMPDH2 0 42 COc1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1OC ZINC000217833850 GI For-Sale Unstable ENPP1 71 37 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217833855 FJ For-Sale Unstable GRIN2B 19 45 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217833855 FJ For-Sale Unstable LTA4H 50 43 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217833855 FJ For-Sale Unstable HCRTR1 18 47 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217833855 FJ For-Sale Unstable MMP13 18 44 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217833855 FJ For-Sale Unstable PREP 28 44 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217833855 FJ For-Sale Unstable CHRNA10 50 38 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217833855 FJ For-Sale Unstable PLAU 19 42 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217833855 FJ For-Sale Unstable ST14 21 42 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217833855 FJ For-Sale Unstable ACKR3 57 33 C[C@H]1CCCCN1CCCN[C@H](C)c1cccc(C#N)c1 ZINC000217833898 CG On-Demand Unstable HRH3 42 44 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)NCc3ccc4c(c3)OCO4)C2)n1 ZINC000217833902 IH In-Stock Unstable NOS2 100 40 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)NCc3ccc4c(c3)OCO4)C2)n1 ZINC000217833902 IH In-Stock Unstable SSTR3 107 35 Cc1c[nH]c(C(=O)N2CCC[C@@H]2c2ccccn2)n1 ZINC000217833904 CE In-Stock Unstable COLA 76 38 Cc1c[nH]c(C(=O)N2CCC[C@@H]2c2ccccn2)n1 ZINC000217833904 CE In-Stock Unstable CPT1A 72 38 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1cccnc1N(C)C ZINC000217833909 CI For-Sale Unstable TRPM8 15 40 C[C@H](c1cccc(O)c1)N1CC[C@@H](c2ccccc2)C1 ZINC000217833921 CH For-Sale Unstable OPRM1 22 53 C[C@H](c1cccc(O)c1)N1CC[C@@H](c2ccccc2)C1 ZINC000217833921 CH For-Sale Unstable OPRD1 23 53 C[C@H](c1cccc(O)c1)N1CC[C@@H](c2ccccc2)C1 ZINC000217833921 CH For-Sale Unstable OPRK1 23 43 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217833933 FJ For-Sale Unstable GRIN2B 19 45 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217833933 FJ For-Sale Unstable LTA4H 50 43 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217833933 FJ For-Sale Unstable HCRTR1 18 47 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217833933 FJ For-Sale Unstable MMP13 18 44 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217833933 FJ For-Sale Unstable PREP 28 44 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217833933 FJ For-Sale Unstable CHRNA10 50 38 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217833933 FJ For-Sale Unstable PLAU 19 42 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217833933 FJ For-Sale Unstable ST14 21 42 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217833933 FJ For-Sale Unstable ACKR3 57 33 C[C@H]1CCc2[nH]c3ccc(C(=O)Nc4ccc(Sc5nncn5C)cc4)cc3c2C1 ZINC000217833941 HJ On-Demand Unstable HTR1F 22 45 C[C@H]1CCc2[nH]c3ccc(C(=O)Nc4ccc(Sc5nncn5C)cc4)cc3c2C1 ZINC000217833941 HJ On-Demand Unstable MAPKAPK2 22 40 O=C(N/C=C/c1ccccc1Br)NCCCN1CCCC1=O ZINC000217833950 FF For-Sale Unstable TYRO3 24 40 O=C(COc1ccc(Cl)cc1)NCCCN1CCCc2ccccc21 ZINC000217833956 FH In-Stock Unstable PLA2G4A 62 34 O=C(COc1ccc(Cl)cc1)NCCCN1CCCc2ccccc21 ZINC000217833956 FH In-Stock Unstable ADAMTS5 17 45 CN1CCO[C@@H]([C@@H](O)c2ccc(-c3ccccc3)cc2)C1 ZINC000217833977 CF For-Sale Unstable FDFT1 0 50 CN1CCO[C@@H]([C@@H](O)c2ccc(-c3ccccc3)cc2)C1 ZINC000217833977 CF For-Sale Unstable HSD17B2 28 42 Cc1c[nH]c(C(=O)N2CCC[C@H]2c2ccccn2)n1 ZINC000217833987 CE In-Stock Unstable COLA 76 38 Cc1c[nH]c(C(=O)N2CCC[C@H]2c2ccccn2)n1 ZINC000217833987 CE In-Stock Unstable CPT1A 72 38 NC1C[C@@H]2CC[C@H](C1)N2CCc1cccc(Cl)c1 ZINC000217833992 CF For-Sale Unstable SLC6A3 15 40 NC1C[C@@H]2CC[C@H](C1)N2CCc1cccc(Cl)c1 ZINC000217833992 CF For-Sale Unstable KCNH2 22 42 NC1C[C@@H]2CC[C@H](C1)N2CCc1cccc(Cl)c1 ZINC000217833992 CF For-Sale Unstable CACNA1D 53 50 NC1C[C@@H]2CC[C@H](C1)N2CCc1cccc(Cl)c1 ZINC000217833992 CF For-Sale Unstable ACHP_LYMST 19 43 NC1C[C@@H]2CC[C@H](C1)N2CCc1cccc(Cl)c1 ZINC000217833992 CF For-Sale Unstable Q8WSF8_APLCA 19 43 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)NCc3ccc4c(c3)OCO4)C2)n1 ZINC000217833993 IH In-Stock Unstable NOS2 100 40 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)NCc3ccc4c(c3)OCO4)C2)n1 ZINC000217833993 IH In-Stock Unstable SSTR3 107 35 CCc1c(C)nn(Cc2cccc(/C=C\C(=O)O)c2)c1C ZINC000217834000 CG For-Sale Unstable HDAC8 37 42 CCc1c(C)nn(Cc2cccc(/C=C\C(=O)O)c2)c1C ZINC000217834000 CG For-Sale Unstable HDAC6 23 42 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1cccnc1N(C)C ZINC000217834003 CI For-Sale Unstable TRPM8 15 40 CCCCCCOc1ccsc1Br ZINC000217834041 CI For-Sale Unstable PLA2G4B 51 33 CCCCCCOc1ccsc1Br ZINC000217834041 CI For-Sale Unstable S1PR2 40 35 CN1CCO[C@H]([C@@H](O)c2ccc(-c3ccccc3)cc2)C1 ZINC000217834048 CF For-Sale Unstable FDFT1 0 50 CN1CCO[C@H]([C@@H](O)c2ccc(-c3ccccc3)cc2)C1 ZINC000217834048 CF For-Sale Unstable HSD17B2 28 42 CCOc1ccc2ccccc2c1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217834050 FJ For-Sale Unstable DRD2 31 41 CCOc1ccc2ccccc2c1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217834050 FJ For-Sale Unstable HCN1 51 34 CCOc1ccc2ccccc2c1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217834050 FJ For-Sale Unstable HCN4 44 34 CCOc1ccc2ccccc2c1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217834050 FJ For-Sale Unstable ACKR3 50 33 O=C(N/C=C/c1ccccc1Br)Nc1ccc(Br)cc1 ZINC000217834067 GK For-Sale Anodyne MTCA1 23 44 O=C(N/C=C/c1ccccc1Br)Nc1ccc(Br)cc1 ZINC000217834067 GK For-Sale Anodyne P96878_MYCTU 24 44 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1cccnc1N(C)C ZINC000217834093 CI For-Sale Unstable TRPM8 15 40 CC(C)Oc1cccc(CNC(=O)COc2ccc(Cl)cc2Cl)c1 ZINC000217834098 FI In-Stock Unstable PPARG 15 41 CC(C)Oc1cccc(CNC(=O)COc2ccc(Cl)cc2Cl)c1 ZINC000217834098 FI In-Stock Unstable PPARD 24 41 CC(C)Oc1cccc(CNC(=O)COc2ccc(Cl)cc2Cl)c1 ZINC000217834098 FI In-Stock Unstable CRTM 40 38 CC(C)Oc1cccc(CNC(=O)COc2ccc(Cl)cc2Cl)c1 ZINC000217834098 FI In-Stock Unstable PDS 82 41 COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OCc1nccn1C ZINC000217834107 KI In-Stock Unstable ALOX5 0 40 COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OCc1nccn1C ZINC000217834107 KI In-Stock Unstable CYP1B1 41 38 COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OCc1nccn1C ZINC000217834107 KI In-Stock Unstable CYP1A1 41 38 CCN1CCN(C(=O)N2CCC[C@H](Cc3nc(-c4ccccc4C)no3)C2)C(=O)C1=O ZINC000217834115 IE In-Stock Unstable Q8MHZ5_SHEEP 42 33 CCOc1ccc2ccccc2c1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217834146 FJ For-Sale Unstable DRD2 31 41 CCOc1ccc2ccccc2c1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217834146 FJ For-Sale Unstable HCN1 51 34 CCOc1ccc2ccccc2c1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217834146 FJ For-Sale Unstable HCN4 44 34 CCOc1ccc2ccccc2c1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217834146 FJ For-Sale Unstable ACKR3 50 33 CCN1CCN(C(=O)N2CCC[C@@H](Cc3nc(-c4ccccc4C)no3)C2)C(=O)C1=O ZINC000217834161 IE In-Stock Unstable Q8MHZ5_SHEEP 42 33 COc1cc(CN2CCC[C@@H](C)[C@@H]2C)cc(Cl)c1O ZINC000217834186 CH For-Sale Unstable DRD2 40 42 COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OCc1nccn1C ZINC000217834189 KI In-Stock Unstable ALOX5 0 40 COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OCc1nccn1C ZINC000217834189 KI In-Stock Unstable CYP1B1 41 38 COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OCc1nccn1C ZINC000217834189 KI In-Stock Unstable CYP1A1 41 38 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1cccnc1N(C)C ZINC000217834208 CI For-Sale Unstable TRPM8 15 40 O=C(N/C=C/c1ccccc1Br)Nc1cccc(C(=O)O)c1 ZINC000217834230 FH For-Sale Anodyne PARP14 0 40 O=C(N/C=C/c1ccccc1Br)Nc1cccc(C(=O)O)c1 ZINC000217834230 FH For-Sale Anodyne PARP10 0 40 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccccc1Oc1ccccc1 ZINC000217834236 FJ For-Sale Unstable DRD2 34 41 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccccc1Oc1ccccc1 ZINC000217834236 FJ For-Sale Unstable HCRTR1 33 43 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccccc1Oc1ccccc1 ZINC000217834236 FJ For-Sale Unstable KCNA3 40 34 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccccc1Oc1ccccc1 ZINC000217834236 FJ For-Sale Unstable HCRTR2 16 43 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccccc1Oc1ccccc1 ZINC000217834236 FJ For-Sale Unstable HCN1 76 35 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccccc1Oc1ccccc1 ZINC000217834236 FJ For-Sale Unstable HCN4 54 35 CCOc1ccc(CNC(=O)COc2ccc(Cl)cc2Cl)cc1OCC ZINC000217834243 GI In-Stock Unstable GSTA1 0 41 CCOc1ccc(CNC(=O)COc2ccc(Cl)cc2Cl)cc1OCC ZINC000217834243 GI In-Stock Unstable PDE6A 48 38 CCOc1ccc(CNC(=O)COc2ccc(Cl)cc2Cl)cc1OCC ZINC000217834243 GI In-Stock Unstable AGPAT2 30 41 CCOc1ccc(CNC(=O)COc2ccc(Cl)cc2Cl)cc1OCC ZINC000217834243 GI In-Stock Unstable PTGDR2 32 41 CCOc1ccc(CNC(=O)COc2ccc(Cl)cc2Cl)cc1OCC ZINC000217834243 GI In-Stock Unstable ENR 0 42 Cc1ccccc1-c1noc(C[C@@H]2CCCN(C(=O)N3CCNC3=O)C2)n1 ZINC000217834270 FE In-Stock Unstable Q8MHZ5_SHEEP 53 31 COc1ccc(CC[C@H](O)[C@@H]2CN(C)CCO2)cc1 ZINC000217834275 CD For-Sale Unstable SLC18A2 21 40 COc1cc(CN2CCC[C@H](C)[C@@H]2C)cc(Cl)c1O ZINC000217834281 CH For-Sale Unstable DRD2 40 42 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1Oc1ccccc1 ZINC000217834305 FJ For-Sale Unstable DRD2 34 41 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1Oc1ccccc1 ZINC000217834305 FJ For-Sale Unstable HCRTR1 33 43 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1Oc1ccccc1 ZINC000217834305 FJ For-Sale Unstable KCNA3 40 34 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1Oc1ccccc1 ZINC000217834305 FJ For-Sale Unstable HCRTR2 16 43 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1Oc1ccccc1 ZINC000217834305 FJ For-Sale Unstable HCN1 76 35 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1Oc1ccccc1 ZINC000217834305 FJ For-Sale Unstable HCN4 54 35 COc1cc(CNC(=O)COc2ccc(Cl)cc2Cl)ccc1OC(C)C ZINC000217834333 GI In-Stock Unstable PDE5A 44 41 COc1cc(CNC(=O)COc2ccc(Cl)cc2Cl)ccc1OC(C)C ZINC000217834333 GI In-Stock Unstable TRPV1 27 42 COc1cc(CNC(=O)COc2ccc(Cl)cc2Cl)ccc1OC(C)C ZINC000217834333 GI In-Stock Unstable CPT1A 44 31 COc1cc(CNC(=O)COc2ccc(Cl)cc2Cl)ccc1OC(C)C ZINC000217834333 GI In-Stock Unstable PDE6A 49 38 COc1cc(CNC(=O)COc2ccc(Cl)cc2Cl)ccc1OC(C)C ZINC000217834333 GI In-Stock Unstable TTR 0 44 COc1cc(CNC(=O)COc2ccc(Cl)cc2Cl)ccc1OC(C)C ZINC000217834333 GI In-Stock Unstable DRTS_TRYCR 46 33 COc1cc(CNC(=O)COc2ccc(Cl)cc2Cl)ccc1OC(C)C ZINC000217834333 GI In-Stock Unstable CAN2 0 42 O=C(N/C=C/c1ccccc1Br)Nc1ccccc1[N+](=O)[O-] ZINC000217834341 FI For-Sale Bother COLA 59 31 Cc1ccccc1-c1noc(C[C@H]2CCCN(C(=O)N3CCNC3=O)C2)n1 ZINC000217834353 FE In-Stock Unstable Q8MHZ5_SHEEP 53 31 COc1ccc(CC[C@H](O)[C@H]2CN(C)CCO2)cc1 ZINC000217834355 CD For-Sale Unstable SLC18A2 21 40 COCc1cccc(/C=C\C(=O)O)c1 ZINC000217834367 AD For-Sale Unstable MAOB 17 40 COCc1cccc(/C=C\C(=O)O)c1 ZINC000217834367 AD For-Sale Unstable PTGER2 24 51 COCc1cccc(/C=C\C(=O)O)c1 ZINC000217834367 AD For-Sale Unstable PTGER4 22 43 COCc1cccc(/C=C\C(=O)O)c1 ZINC000217834367 AD For-Sale Unstable CA7 0 49 COCc1cccc(/C=C\C(=O)O)c1 ZINC000217834367 AD For-Sale Unstable PTGER3 22 42 COCc1cccc(/C=C\C(=O)O)c1 ZINC000217834367 AD For-Sale Unstable LTB4R 25 52 COCc1cccc(/C=C\C(=O)O)c1 ZINC000217834367 AD For-Sale Unstable KCNA3 0 40 COCc1cccc(/C=C\C(=O)O)c1 ZINC000217834367 AD For-Sale Unstable CA14 0 49 COCc1cccc(/C=C\C(=O)O)c1 ZINC000217834367 AD For-Sale Unstable MMP2 0 45 COCc1cccc(/C=C\C(=O)O)c1 ZINC000217834367 AD For-Sale Unstable SLC1A6 48 31 COCc1cccc(/C=C\C(=O)O)c1 ZINC000217834367 AD For-Sale Unstable NR1H4 50 36 COCc1cccc(/C=C\C(=O)O)c1 ZINC000217834367 AD For-Sale Unstable SLC1A7 48 31 COCc1cccc(/C=C\C(=O)O)c1 ZINC000217834367 AD For-Sale Unstable MMP1 0 45 COCc1cccc(/C=C\C(=O)O)c1 ZINC000217834367 AD For-Sale Unstable 17HSDCL 0 48 COCc1cccc(/C=C\C(=O)O)c1 ZINC000217834367 AD For-Sale Unstable FFAR1 25 44 COCc1cccc(/C=C\C(=O)O)c1 ZINC000217834367 AD For-Sale Unstable AKR1C3 43 48 COCc1cccc(/C=C\C(=O)O)c1 ZINC000217834367 AD For-Sale Unstable AKR1B10 36 41 COCc1cccc(/C=C\C(=O)O)c1 ZINC000217834367 AD For-Sale Unstable GPR183 42 39 O=C(CCCCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217834405 EI For-Sale Unstable ACE 30 40 O=C(CCCCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217834405 EI For-Sale Unstable FKBP1A 37 43 O=C(CCCCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217834405 EI For-Sale Unstable SLC18A2 45 38 O=C(CCCCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217834405 EI For-Sale Unstable PREP 71 42 O=C(CCCCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217834405 EI For-Sale Unstable MTNR1A 23 43 O=C(CCCCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217834405 EI For-Sale Unstable MTNR1B 21 43 O=C(CCCCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217834405 EI For-Sale Unstable FAAH 60 38 O=C(CCCCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217834405 EI For-Sale Unstable CES1 60 37 O=C(CCCCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217834405 EI For-Sale Unstable CES1D 52 30 N#Cc1cccc(OCCCN2CCCS(=O)(=O)CC2)c1 ZINC000217834434 DD On-Demand Unstable KCNH2 0 42 N#Cc1cccc(OCCCN2CCCS(=O)(=O)CC2)c1 ZINC000217834434 DD On-Demand Unstable HRH3 76 41 O=C(COc1ccc(Cl)cc1Cl)NCCCc1ccccc1Cl ZINC000217834438 FJ In-Stock Unstable POLG_WNV 46 33 O=C(COc1ccc(Cl)cc1Cl)NCCCc1ccccc1Cl ZINC000217834438 FJ In-Stock Unstable CRTM 41 39 O=C(N/C=C/c1ccccc1Br)Nc1cccc(O)c1 ZINC000217834439 EH For-Sale Anodyne KCNK3 66 33 CCS(=O)(=O)N1CCC[C@H](Cc2nc(-c3ccccc3C)no2)C1 ZINC000217834451 EF In-Stock Unstable Q8MHZ5_SHEEP 43 33 O=C(CCCCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217834464 EI For-Sale Unstable ACE 30 40 O=C(CCCCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217834464 EI For-Sale Unstable FKBP1A 37 43 O=C(CCCCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217834464 EI For-Sale Unstable SLC18A2 45 38 O=C(CCCCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217834464 EI For-Sale Unstable PREP 71 42 O=C(CCCCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217834464 EI For-Sale Unstable MTNR1A 23 43 O=C(CCCCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217834464 EI For-Sale Unstable MTNR1B 21 43 O=C(CCCCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217834464 EI For-Sale Unstable FAAH 60 38 O=C(CCCCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217834464 EI For-Sale Unstable CES1 60 37 O=C(CCCCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217834464 EI For-Sale Unstable CES1D 52 30 O=C(c1cccnc1)N1CCN(C/C=C\c2ccc(F)cc2)CC1 ZINC000217834480 EF On-Demand Unstable TBXAS1 31 41 COc1ccc(CN2CCCCC2)cc1/C=C\C(=O)O ZINC000217834492 CF For-Sale Unstable ACHE 25 56 COc1ccc(CN2CCCCC2)cc1/C=C\C(=O)O ZINC000217834492 CF For-Sale Unstable HRH2 26 41 COc1ccc(CN2CCCCC2)cc1/C=C\C(=O)O ZINC000217834492 CF For-Sale Unstable PTGER2 39 43 COc1ccc(CN2CCCCC2)cc1/C=C\C(=O)O ZINC000217834492 CF For-Sale Unstable PTGER4 22 43 COc1ccc(CN2CCCCC2)cc1/C=C\C(=O)O ZINC000217834492 CF For-Sale Unstable HRH3 21 41 COc1ccc(CN2CCCCC2)cc1/C=C\C(=O)O ZINC000217834492 CF For-Sale Unstable SIGMAR1 17 40 COc1ccc(CN2CCCCC2)cc1/C=C\C(=O)O ZINC000217834492 CF For-Sale Unstable PTGER3 18 43 COc1ccc(CN2CCCCC2)cc1/C=C\C(=O)O ZINC000217834492 CF For-Sale Unstable MCHR1 17 40 COc1ccc(NC(=O)CN2C(=O)c3ccccc3N3C(=O)c4c(ccc(OC)c4OC)[C@H]23)cn1 ZINC000217834497 JF In-Stock Unstable TSHR 42 32 CN[C@H](CCN(C)[C@@H](C)c1ccc(Cl)cc1)C(C)(C)C ZINC000217834500 CI For-Sale Unstable UTS2 41 33 CCS(=O)(=O)N1CCC[C@@H](Cc2nc(-c3ccccc3C)no2)C1 ZINC000217834542 EF In-Stock Unstable Q8MHZ5_SHEEP 43 33 O=C(O)[C@H]1CN(Cc2ccco2)CCN(C2CCCCC2)C1 ZINC000217834566 DE In-Stock Unstable SLC6A1 93 37 O=C(O)[C@H]1CN(Cc2ccco2)CCN(C2CCCCC2)C1 ZINC000217834566 DE In-Stock Unstable SIGMAR1 15 40 O=C(COc1ccc(Cl)cc1Cl)NCCCc1ccc(Cl)cc1 ZINC000217834574 FJ In-Stock Unstable SCNN1A 54 33 O=C(COc1ccc(Cl)cc1Cl)NCCCc1ccc(Cl)cc1 ZINC000217834574 FJ In-Stock Unstable TTR 0 41 O=C(COc1ccc(Cl)cc1Cl)NCCCc1ccc(Cl)cc1 ZINC000217834574 FJ In-Stock Unstable ALPL 43 38 O=C(COc1ccc(Cl)cc1Cl)NCCCc1ccc(Cl)cc1 ZINC000217834574 FJ In-Stock Unstable CRTM 45 46 COc1ccc(NC(=O)CN2C(=O)c3ccccc3N3C(=O)c4c(ccc(OC)c4OC)[C@@H]23)cn1 ZINC000217834577 JF In-Stock Unstable TSHR 42 32 COc1ccc(/C=C/C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217834583 FH For-Sale Unstable DRD2 38 40 COc1ccc(/C=C/C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217834583 FH For-Sale Unstable DRD3 21 41 COc1ccc(/C=C/C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217834583 FH For-Sale Unstable CYP1B1 17 41 COc1ccc(/C=C/C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217834583 FH For-Sale Unstable HDAC8 43 37 COc1ccc(/C=C/C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217834583 FH For-Sale Unstable CYP1A1 19 41 COc1ccc(/C=C/C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217834583 FH For-Sale Unstable HDAC1 30 41 COc1ccc(/C=C/C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217834583 FH For-Sale Unstable ACKR3 77 44 COc1ccc(/C=C\C(=O)O)cc1CN1CCSCC1 ZINC000217834593 CE For-Sale Unstable AKR1C3 37 40 O=C(O)COc1cc(O)ccc1Br ZINC000217834613 BD For-Sale Unstable PTGDR2 30 46 COc1ccc(/C=C/C(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217834664 FH For-Sale Unstable DRD2 38 40 COc1ccc(/C=C/C(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217834664 FH For-Sale Unstable DRD3 21 41 COc1ccc(/C=C/C(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217834664 FH For-Sale Unstable CYP1B1 17 41 COc1ccc(/C=C/C(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217834664 FH For-Sale Unstable HDAC8 43 37 COc1ccc(/C=C/C(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217834664 FH For-Sale Unstable CYP1A1 19 41 COc1ccc(/C=C/C(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217834664 FH For-Sale Unstable HDAC1 30 41 COc1ccc(/C=C/C(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217834664 FH For-Sale Unstable ACKR3 77 44 O=C(COc1ccc(Cl)cc1Cl)NCCCc1ccc(F)cc1 ZINC000217834678 FI In-Stock Unstable SCNN1A 40 32 O=C(COc1ccc(Cl)cc1Cl)NCCCc1ccc(F)cc1 ZINC000217834678 FI In-Stock Unstable CCR1 20 40 O=C(COc1ccc(Cl)cc1Cl)NCCCc1ccc(F)cc1 ZINC000217834678 FI In-Stock Unstable ALPL 61 40 O=C(COc1ccc(Cl)cc1Cl)NCCCc1ccc(F)cc1 ZINC000217834678 FI In-Stock Unstable LEF 44 34 O=C(COc1ccc(Cl)cc1Cl)NCCCc1ccc(F)cc1 ZINC000217834678 FI In-Stock Unstable CRTM 37 40 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)cc1 ZINC000217834683 JI In-Stock Unstable AKR1B1 22 49 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)cc1 ZINC000217834683 JI In-Stock Unstable CYP1B1 62 45 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)cc1 ZINC000217834683 JI In-Stock Unstable CYP1A1 46 49 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)cc1 ZINC000217834683 JI In-Stock Unstable CYP1A2 35 45 COc1ccc(CN2CCSCC2)cc1/C=C\C(=O)O ZINC000217834711 CE For-Sale Unstable PTGER2 30 42 COc1ccc(CN2CCSCC2)cc1/C=C\C(=O)O ZINC000217834711 CE For-Sale Unstable PTGER4 19 42 COc1ccc(CN2CCSCC2)cc1/C=C\C(=O)O ZINC000217834711 CE For-Sale Unstable PTGER3 15 42 O=C(O)COc1ccc(Br)cc1O ZINC000217834728 BD For-Sale Unstable PPARD 38 47 O=C(O)COc1ccc(Br)cc1O ZINC000217834728 BD For-Sale Unstable PTGDR2 48 62 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)cc1 ZINC000217834758 JI In-Stock Unstable AKR1B1 22 49 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)cc1 ZINC000217834758 JI In-Stock Unstable CYP1B1 62 45 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)cc1 ZINC000217834758 JI In-Stock Unstable CYP1A1 46 49 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)cc1 ZINC000217834758 JI In-Stock Unstable CYP1A2 35 45 COc1ccccc1CCCNC(=O)COc1ccc(Cl)cc1Cl ZINC000217834775 FI In-Stock Unstable CYSP_TRYCR 0 41 COc1ccccc1CCCNC(=O)COc1ccc(Cl)cc1Cl ZINC000217834775 FI In-Stock Unstable CPT1A 45 32 COc1ccccc1CCCNC(=O)COc1ccc(Cl)cc1Cl ZINC000217834775 FI In-Stock Unstable MTNR1A 43 42 COc1ccccc1CCCNC(=O)COc1ccc(Cl)cc1Cl ZINC000217834775 FI In-Stock Unstable MTNR1B 45 45 COc1ccccc1CCCNC(=O)COc1ccc(Cl)cc1Cl ZINC000217834775 FI In-Stock Unstable TTR 0 44 COc1ccccc1CCCNC(=O)COc1ccc(Cl)cc1Cl ZINC000217834775 FI In-Stock Unstable PTGDR2 43 37 COc1ccccc1CCCNC(=O)COc1ccc(Cl)cc1Cl ZINC000217834775 FI In-Stock Unstable NCE103 15 41 COc1ccccc1CCCNC(=O)COc1ccc(Cl)cc1Cl ZINC000217834775 FI In-Stock Unstable CAN2 0 41 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc2n[nH]nc2c1 ZINC000217834776 DE For-Sale Unstable HCRTR1 15 44 Nc1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217834811 EH For-Sale Unstable P96878_MYCTU 40 37 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc2n[nH]nc2c1 ZINC000217834867 DE For-Sale Unstable HCRTR1 15 44 COc1cc(CN2CCC[C@@H](C)[C@@H]2C)ccc1O ZINC000217834869 BG For-Sale Unstable DRD2 40 39 COc1cc(CN2CCC[C@@H](C)[C@@H]2C)ccc1O ZINC000217834869 BG For-Sale Unstable SHBG 19 45 COc1cc(CN2CCC[C@@H](C)[C@@H]2C)ccc1O ZINC000217834869 BG For-Sale Unstable CAN2 0 43 COc1cccc(CCCNC(=O)COc2ccc(Cl)cc2Cl)c1 ZINC000217834904 FI In-Stock Unstable DRD4 44 36 COc1cccc(CCCNC(=O)COc2ccc(Cl)cc2Cl)c1 ZINC000217834904 FI In-Stock Unstable FDFT1 0 53 COc1cccc(CCCNC(=O)COc2ccc(Cl)cc2Cl)c1 ZINC000217834904 FI In-Stock Unstable S1PR4 40 38 COc1cccc(CCCNC(=O)COc2ccc(Cl)cc2Cl)c1 ZINC000217834904 FI In-Stock Unstable MTNR1A 61 54 COc1cccc(CCCNC(=O)COc2ccc(Cl)cc2Cl)c1 ZINC000217834904 FI In-Stock Unstable MTNR1B 51 63 COc1cccc(CCCNC(=O)COc2ccc(Cl)cc2Cl)c1 ZINC000217834904 FI In-Stock Unstable ABCB1 0 40 COc1cccc(CCCNC(=O)COc2ccc(Cl)cc2Cl)c1 ZINC000217834904 FI In-Stock Unstable TTR 0 40 COc1cccc(CCCNC(=O)COc2ccc(Cl)cc2Cl)c1 ZINC000217834904 FI In-Stock Unstable NCE103 15 53 COc1cccc(CCCNC(=O)COc2ccc(Cl)cc2Cl)c1 ZINC000217834904 FI In-Stock Unstable CRTM 78 53 COc1cccc(CCCNC(=O)COc2ccc(Cl)cc2Cl)c1 ZINC000217834904 FI In-Stock Unstable CAN2 0 53 COc1cccc(CCCNC(=O)COc2ccc(Cl)cc2Cl)c1 ZINC000217834904 FI In-Stock Unstable PDS 41 36 COc1cc(CN2CCC[C@H](C)[C@@H]2C)ccc1O ZINC000217834964 BG For-Sale Unstable DRD2 40 39 COc1cc(CN2CCC[C@H](C)[C@@H]2C)ccc1O ZINC000217834964 BG For-Sale Unstable SHBG 19 45 COc1cc(CN2CCC[C@H](C)[C@@H]2C)ccc1O ZINC000217834964 BG For-Sale Unstable CAN2 0 43 COc1cc(C(=O)O)c(O)cc1Br ZINC000217835003 BD For-Sale Unstable APP 40 37 COc1cc(C(=O)O)c(O)cc1Br ZINC000217835003 BD For-Sale Unstable CA14 15 44 COc1cc(C(=O)O)c(O)cc1Br ZINC000217835003 BD For-Sale Unstable AKR1C1 24 40 COc1ccc(CCCNC(=O)COc2ccc(Cl)cc2Cl)cc1 ZINC000217835006 FI In-Stock Unstable SCNN1A 72 42 COc1ccc(CCCNC(=O)COc2ccc(Cl)cc2Cl)cc1 ZINC000217835006 FI In-Stock Unstable MTNR1A 52 44 COc1ccc(CCCNC(=O)COc2ccc(Cl)cc2Cl)cc1 ZINC000217835006 FI In-Stock Unstable MTNR1B 35 43 COc1ccc(CCCNC(=O)COc2ccc(Cl)cc2Cl)cc1 ZINC000217835006 FI In-Stock Unstable PDE6A 41 32 COc1ccc(CCCNC(=O)COc2ccc(Cl)cc2Cl)cc1 ZINC000217835006 FI In-Stock Unstable TTR 0 43 COc1ccc(CCCNC(=O)COc2ccc(Cl)cc2Cl)cc1 ZINC000217835006 FI In-Stock Unstable ALPL 40 35 COc1ccc(CCCNC(=O)COc2ccc(Cl)cc2Cl)cc1 ZINC000217835006 FI In-Stock Unstable CA9 16 41 COc1ccc(CCCNC(=O)COc2ccc(Cl)cc2Cl)cc1 ZINC000217835006 FI In-Stock Unstable MCHR2 21 41 COc1ccc(CCCNC(=O)COc2ccc(Cl)cc2Cl)cc1 ZINC000217835006 FI In-Stock Unstable NCE103 18 42 COc1ccc(CCCNC(=O)COc2ccc(Cl)cc2Cl)cc1 ZINC000217835006 FI In-Stock Unstable CRTM 44 44 COc1ccc(CCCNC(=O)COc2ccc(Cl)cc2Cl)cc1 ZINC000217835006 FI In-Stock Unstable CAN2 0 42 Cc1noc(C)c1CC(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217835010 DF For-Sale Unstable P2RX7 26 51 CN(CCOc1cccc(/C=C\C(=O)O)c1)C1CCCC1 ZINC000217835012 CG For-Sale Unstable PPARG 21 42 COc1ccc(C)cc1S(=O)(=O)N1CCC[C@H](Cc2nc(-c3ccccc3C)no2)C1 ZINC000217835013 II In-Stock Unstable Q8MHZ5_SHEEP 41 31 COc1ccc(C)cc1S(=O)(=O)N1CCC[C@@H](Cc2nc(-c3ccccc3C)no2)C1 ZINC000217835052 II In-Stock Unstable Q8MHZ5_SHEEP 41 31 COc1ccc2cc(CNC(=O)c3cc(N4CCCC4)ccn3)ccc2c1 ZINC000217835060 FH On-Demand Unstable DRD4 43 34 COc1ccc2cc(CNC(=O)c3cc(N4CCCC4)ccn3)ccc2c1 ZINC000217835060 FH On-Demand Unstable DRD3 15 42 COc1ccc2cc(CNC(=O)c3cc(N4CCCC4)ccn3)ccc2c1 ZINC000217835060 FH On-Demand Unstable MMP13 40 47 COc1ccc2cc(CNC(=O)c3cc(N4CCCC4)ccn3)ccc2c1 ZINC000217835060 FH On-Demand Unstable ALK 16 41 Cc1noc(C)c1CC(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217835085 DF For-Sale Unstable P2RX7 26 51 COc1ccc(OC[C@@H](C)NC(=O)COc2ccc(Cl)cc2Cl)cc1 ZINC000217835098 GH In-Stock Unstable S1PR4 29 42 O=C(N/C=C/c1ccccc1Br)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217835101 GG For-Sale Anodyne CA2 20 43 O=C(N/C=C/c1ccccc1Br)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217835101 GG For-Sale Anodyne CA1 25 40 O=C(N/C=C/c1ccccc1Br)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217835101 GG For-Sale Anodyne CA12 28 43 O=C(N/C=C/c1ccccc1Br)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217835101 GG For-Sale Anodyne CA9 26 40 O=C(N/C=C/c1ccccc1Br)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217835101 GG For-Sale Anodyne MTCA1 46 43 O=C(N/C=C/c1ccccc1Br)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217835101 GG For-Sale Anodyne P96878_MYCTU 58 43 COc1ccc2cc(CNC(=O)c3nn(-c4ccccc4)cc3O)ccc2c1 ZINC000217835158 FH On-Demand Unstable ROCK1 21 42 COc1ccc2cc(CNC(=O)c3nn(-c4ccccc4)cc3O)ccc2c1 ZINC000217835158 FH On-Demand Unstable SCD1 18 42 COc1ccc2cc(CNC(=O)c3nn(-c4ccccc4)cc3O)ccc2c1 ZINC000217835158 FH On-Demand Unstable CARM1 43 33 CN(CCOc1ccc(/C=C\C(=O)O)cc1)C1CCCC1 ZINC000217835160 CG On-Demand Unstable LSS 23 43 Cc1ccccc1-c1noc(C[C@@H]2CCCN(S(=O)(=O)/C=C/c3ccccc3)C2)n1 ZINC000217835173 HI In-Stock Unstable Q8MHZ5_SHEEP 42 33 COc1ccc(OC[C@H](C)NC(=O)COc2ccc(Cl)cc2Cl)cc1 ZINC000217835186 GH In-Stock Unstable S1PR4 29 42 O=C(N/C=C/c1ccccc1Br)Nc1cccc(S(=O)(=O)O)c1 ZINC000217835202 GG For-Sale Anodyne CA4 16 40 COc1ccc(CCNc2nc(C)cc(N[C@H](C)c3ccccc3)n2)cc1 ZINC000217835231 FJ For-Sale Unstable HTR7 25 58 COc1ccc(CCNc2nc(C)cc(N[C@H](C)c3ccccc3)n2)cc1 ZINC000217835231 FJ For-Sale Unstable PLK1 19 45 COc1ccc(CCNc2nc(C)cc(N[C@H](C)c3ccccc3)n2)cc1 ZINC000217835231 FJ For-Sale Unstable PTGDR 26 41 Cc1ccccc1-c1noc(C[C@H]2CCCN(S(=O)(=O)/C=C/c3ccccc3)C2)n1 ZINC000217835238 HI In-Stock Unstable Q8MHZ5_SHEEP 42 33 CC(C)Oc1cccc(CCCNC(=O)COc2ccc(Cl)cc2Cl)c1 ZINC000217835280 GJ In-Stock Unstable FDFT1 0 52 CC(C)Oc1cccc(CCCNC(=O)COc2ccc(Cl)cc2Cl)c1 ZINC000217835280 GJ In-Stock Unstable MTNR1A 22 49 CC(C)Oc1cccc(CCCNC(=O)COc2ccc(Cl)cc2Cl)c1 ZINC000217835280 GJ In-Stock Unstable MTNR1B 24 49 CC(C)Oc1cccc(CCCNC(=O)COc2ccc(Cl)cc2Cl)c1 ZINC000217835280 GJ In-Stock Unstable CRTM 76 52 CC(C)Oc1cccc(CCCNC(=O)COc2ccc(Cl)cc2Cl)c1 ZINC000217835280 GJ In-Stock Unstable CAN2 0 42 CC(C)Oc1cccc(CCCNC(=O)COc2ccc(Cl)cc2Cl)c1 ZINC000217835280 GJ In-Stock Unstable PDS 62 36 CC(=O)c1cccc(S(=O)(=O)N2CCC[C@@H](Cc3nc(-c4ccccc4C)no3)C2)c1 ZINC000217835360 IH In-Stock Unstable AKR1C3 45 36 CC(=O)c1cccc(S(=O)(=O)N2CCC[C@@H](Cc3nc(-c4ccccc4C)no3)C2)c1 ZINC000217835360 IH In-Stock Unstable Q8MHZ5_SHEEP 41 31 CN(CC(=O)N(C)C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217835364 CD For-Sale Unstable PTGER2 23 41 CN(CC(=O)N(C)C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217835364 CD For-Sale Unstable NR1H4 49 38 CN(CC(=O)N(C)C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217835364 CD For-Sale Unstable AKR1C3 32 42 CC(C)Oc1ccc(CCCNC(=O)COc2ccc(Cl)cc2Cl)cc1 ZINC000217835385 GJ In-Stock Unstable CRTM 42 42 CCCCCCC(=O)CCCCCC/C=C/C=C/C(=O)NCC(C)C ZINC000217835389 EK Annotated Unstable CNR1 28 86 CCCCCCC(=O)CCCCCC/C=C/C=C/C(=O)NCC(C)C ZINC000217835389 EK Annotated Unstable OPRM1 0 86 CCCCCCC(=O)CCCCCC/C=C/C=C/C(=O)NCC(C)C ZINC000217835389 EK Annotated Unstable PPARA 0 61 CCCCCCC(=O)CCCCCC/C=C/C=C/C(=O)NCC(C)C ZINC000217835389 EK Annotated Unstable FABP4 16 43 CCCCCCC(=O)CCCCCC/C=C/C=C/C(=O)NCC(C)C ZINC000217835389 EK Annotated Unstable FAAH 33 50 CCCCCCC(=O)CCCCCC/C=C/C=C/C(=O)NCC(C)C ZINC000217835389 EK Annotated Unstable EPHX2 0 42 CCCCCCC(=O)CCCCCC/C=C/C=C/C(=O)NCC(C)C ZINC000217835389 EK Annotated Unstable FABP3 34 43 CCCCCCC(=O)CCCCCC/C=C/C=C/C(=O)NCC(C)C ZINC000217835389 EK Annotated Unstable CQSS 53 35 COc1ccc(CN2CCC[C@@H](C)[C@@H]2C)cc1O ZINC000217835413 BG On-Demand Unstable DRD2 42 39 Cn1cc(CNC(=O)c2ccc(Cl)o2)cn1 ZINC000217835420 BD On-Demand Unstable NAMPT 43 36 CC(=O)c1cccc(S(=O)(=O)N2CCC[C@H](Cc3nc(-c4ccccc4C)no3)C2)c1 ZINC000217835425 IH In-Stock Unstable AKR1C3 45 36 CC(=O)c1cccc(S(=O)(=O)N2CCC[C@H](Cc3nc(-c4ccccc4C)no3)C2)c1 ZINC000217835425 IH In-Stock Unstable Q8MHZ5_SHEEP 41 31 Cc1cn(-c2ccccc2)nc1OCC(=O)O ZINC000217835460 BD In-Stock Unstable FABP4 45 36 Cc1cn(-c2ccccc2)nc1OCC(=O)O ZINC000217835460 BD In-Stock Unstable PTGDR2 17 48 O=C(NCc1ccc(COCC(F)(F)F)cc1)c1cc(N2CCOCC2)ccn1 ZINC000217835467 HF On-Demand Unstable SCN10A 15 40 O=C(NCc1ccc(COCC(F)(F)F)cc1)c1cc(N2CCOCC2)ccn1 ZINC000217835467 HF On-Demand Unstable EPHB4 42 32 COc1ccc(CN2CCC[C@H](C)[C@@H]2C)cc1O ZINC000217835474 BG On-Demand Unstable DRD2 42 39 O=C(COc1ccc(Cl)cc1Cl)Nc1ccc(OC2CCCC2)cc1 ZINC000217835478 GK In-Stock Unstable CETP 32 43 O=C(COc1ccc(Cl)cc1Cl)Nc1ccc(OC2CCCC2)cc1 ZINC000217835478 GK In-Stock Unstable EPHX2 25 43 O=C(COc1ccc(Cl)cc1Cl)Nc1ccc(OC2CCCC2)cc1 ZINC000217835478 GK In-Stock Unstable MCHR1 17 40 O=C(COc1ccc(Cl)cc1Cl)Nc1ccc(OC2CCCC2)cc1 ZINC000217835478 GK In-Stock Unstable MCHR2 43 49 CC(C)c1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217835544 FK For-Sale Unstable P96878_MYCTU 16 46 COc1ccc(O)c(CN2CCC[C@@H](C)[C@@H]2C)c1 ZINC000217835552 BG On-Demand Unstable SIGMAR1 19 43 COc1ccc(O)c(CN2CCC[C@@H](C)[C@@H]2C)c1 ZINC000217835552 BG On-Demand Unstable EBP 39 40 N#Cc1ccc([C@@H](O)CN2CC[C@@H](CO)C2)cc1 ZINC000217835575 BC On-Demand Unstable O19067_PIG 0 42 Cc1ccccc1-c1noc(C[C@@H]2CCCN(S(=O)(=O)c3c(F)cccc3F)C2)n1 ZINC000217835584 IH In-Stock Unstable Q8MHZ5_SHEEP 41 31 CC1(C)C[C@@H](NC(=O)COc2ccc(Cl)cc2Cl)c2ccccc2O1 ZINC000217835589 GJ In-Stock Unstable CNR1 15 42 CC1(C)C[C@@H](NC(=O)COc2ccc(Cl)cc2Cl)c2ccccc2O1 ZINC000217835589 GJ In-Stock Unstable PTGDR2 15 41 O=C(NCc1ccc(COCC(F)(F)F)cc1)c1nn(-c2ccccc2)cc1O ZINC000217835605 HH On-Demand Unstable CARM1 48 35 Cn1cc(CNC(=O)c2ccc3c(c2)CC(=O)N3)cn1 ZINC000217835616 CC For-Sale Unstable HDAC9 27 47 COc1ccc(O)c(CN2CCC[C@H](C)[C@@H]2C)c1 ZINC000217835636 BG On-Demand Unstable SIGMAR1 19 43 COc1ccc(O)c(CN2CCC[C@H](C)[C@@H]2C)c1 ZINC000217835636 BG On-Demand Unstable EBP 39 40 N#Cc1ccc([C@H](O)CN2CC[C@@H](CO)C2)cc1 ZINC000217835641 BC On-Demand Unstable O19067_PIG 0 42 C[C@@H](c1ccccc1Cl)N(C)CC[C@@H](N)c1ccccc1 ZINC000217835644 DI For-Sale Unstable AOC3 19 41 CC1(C)C[C@H](NC(=O)COc2ccc(Cl)cc2Cl)c2ccccc2O1 ZINC000217835661 GJ In-Stock Unstable CNR1 15 42 CC1(C)C[C@H](NC(=O)COc2ccc(Cl)cc2Cl)c2ccccc2O1 ZINC000217835661 GJ In-Stock Unstable PTGDR2 15 41 O=C(O)[C@@H]1C[C@@H]2CCCC[C@@H]2N1C(=O)CNC1CC1 ZINC000217835676 CC On-Demand Unstable ACE 17 61 Cc1ccccc1-c1noc(C[C@H]2CCCN(S(=O)(=O)c3c(F)cccc3F)C2)n1 ZINC000217835678 IH In-Stock Unstable Q8MHZ5_SHEEP 41 31 C[C@@H]1C(=O)NC(=O)CN1C(=O)/C=C\c1ccc(Cl)cc1Cl ZINC000217835688 ED For-Sale Unstable BOTA 20 43 O=C(CN1CCOC1=O)N1CC(c2nc3ccccc3[nH]2)C1 ZINC000217835701 DC In-Stock Unstable SMO 0 42 C[C@H](c1ccccc1Cl)N(C)CC[C@@H](N)c1ccccc1 ZINC000217835727 DI For-Sale Unstable AOC3 19 41 O=C(CCCN1C(=O)c2ccccc2C1=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217835734 GF For-Sale Unstable HTR1A 18 46 O=C(CCCN1C(=O)c2ccccc2C1=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217835734 GF For-Sale Unstable SLC6A1 42 33 Cc1ccc(C2=NO[C@H](C#N)C2)cc1 ZINC000217835737 AE In-Stock Unstable LUCI_PHOPY 42 40 O=C(O)[C@@H]1C[C@H]2CCCC[C@@H]2N1C(=O)CNC1CC1 ZINC000217835771 CC On-Demand Unstable ACE 17 61 C[C@H]1C(=O)NC(=O)CN1C(=O)/C=C\c1ccc(Cl)cc1Cl ZINC000217835774 ED For-Sale Unstable BOTA 20 43 COc1ccc(S(=O)(=O)N2CCC[C@@H](Cc3nc(-c4ccccc4C)no3)C2)cc1F ZINC000217835782 IH In-Stock Unstable Q8MHZ5_SHEEP 40 31 CC(C)[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(CCc2ccccc2)C1=O ZINC000217835783 EC In-Stock Unstable DEF 0 41 CC(C)[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(CCc2ccccc2)C1=O ZINC000217835783 EC In-Stock Unstable GALR1 44 32 CCOc1ccc(CCCNC(=O)COc2ccc(Cl)cc2Cl)cc1 ZINC000217835806 GJ In-Stock Unstable SCN2A 23 43 CCOc1ccc(CCCNC(=O)COc2ccc(Cl)cc2Cl)cc1 ZINC000217835806 GJ In-Stock Unstable AGPAT2 24 41 CCOc1ccc(CCCNC(=O)COc2ccc(Cl)cc2Cl)cc1 ZINC000217835806 GJ In-Stock Unstable CRTM 49 43 Cc1ccccc1NC(=O)N/C=C/c1ccccc1Br ZINC000217835809 EJ For-Sale Unstable DDX3X 0 41 CCN(C[C@H]1CCCO1)C(=O)c1ccc(Cl)o1 ZINC000217835814 CF On-Demand Unstable OXTR 31 50 CCN(C[C@H]1CCCO1)C(=O)c1ccc(Cl)o1 ZINC000217835814 CF On-Demand Unstable AVPR1A 20 44 Cc1ccc(C2=NO[C@@H](C#N)C2)cc1 ZINC000217835822 AE In-Stock Unstable LUCI_PHOPY 42 40 O=C(CCCN1C(=O)c2ccccc2C1=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217835842 GF For-Sale Unstable HTR1A 18 46 O=C(CCCN1C(=O)c2ccccc2C1=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217835842 GF For-Sale Unstable SLC6A1 42 33 COc1ccc(S(=O)(=O)N2CCC[C@H](Cc3nc(-c4ccccc4C)no3)C2)cc1F ZINC000217835850 IH In-Stock Unstable Q8MHZ5_SHEEP 40 31 CCCOc1ccccc1CCCNC(=O)COc1ccc(Cl)cc1Cl ZINC000217835875 GJ In-Stock Unstable PTGER1 30 40 CCCOc1ccccc1CCCNC(=O)COc1ccc(Cl)cc1Cl ZINC000217835875 GJ In-Stock Unstable S1PR4 27 40 CCCOc1ccccc1CCCNC(=O)COc1ccc(Cl)cc1Cl ZINC000217835875 GJ In-Stock Unstable MTNR1A 40 48 CCCOc1ccccc1CCCNC(=O)COc1ccc(Cl)cc1Cl ZINC000217835875 GJ In-Stock Unstable MTNR1B 41 41 CCCOc1ccccc1CCCNC(=O)COc1ccc(Cl)cc1Cl ZINC000217835875 GJ In-Stock Unstable PTGDR2 35 49 COc1ccc(/C=C\C(=O)O)cc1CN(C)[C@H](C)C(C)C ZINC000217835877 CG For-Sale Unstable PTGER2 20 43 COc1ccc(/C=C\C(=O)O)cc1CN(C)[C@H](C)C(C)C ZINC000217835877 CG For-Sale Unstable APP 20 42 COc1ccc(/C=C\C(=O)O)cc1CN(C)[C@H](C)C(C)C ZINC000217835877 CG For-Sale Unstable TUBB1 48 40 COc1ccc(/C=C\C(=O)O)cc1CN(C)[C@H](C)C(C)C ZINC000217835877 CG For-Sale Unstable AKR1C3 41 43 O=C(N/C=C/c1ccccc1Br)Nc1ccc(Cl)c(Cl)c1 ZINC000217835898 GK For-Sale Anodyne BLM 0 40 O=C(N/C=C/c1ccccc1Br)Nc1ccc(Cl)c(Cl)c1 ZINC000217835898 GK For-Sale Anodyne P95276_MYCTO 0 48 O=C(N/C=C/c1ccccc1Br)Nc1ccc(Cl)c(Cl)c1 ZINC000217835898 GK For-Sale Anodyne WRN 0 40 O=C(N/C=C/c1ccccc1Br)Nc1ccc(Cl)c(Cl)c1 ZINC000217835898 GK For-Sale Anodyne PPX1 0 40 COc1cccc(C2=NO[C@H](C#N)C2)c1 ZINC000217835955 BD In-Stock Unstable LUCI_PHOPY 48 57 COc1ccc(/C=C\C(=O)O)cc1CN(C)[C@@H](C)C(C)C ZINC000217835975 CG For-Sale Unstable PTGER2 0 43 COc1ccc(/C=C\C(=O)O)cc1CN(C)[C@@H](C)C(C)C ZINC000217835975 CG For-Sale Unstable APP 20 42 COc1ccc(/C=C\C(=O)O)cc1CN(C)[C@@H](C)C(C)C ZINC000217835975 CG For-Sale Unstable TUBB1 48 40 COc1ccc(/C=C\C(=O)O)cc1CN(C)[C@@H](C)C(C)C ZINC000217835975 CG For-Sale Unstable AKR1C3 31 40 Cc1noc(C)c1COc1ccc(CC(=O)N2CCC(c3c[nH]c4ccccc34)CC2)cc1 ZINC000217835991 IK On-Demand Unstable ADAM17 47 34 Cc1noc(C)c1COc1ccc(CC(=O)N2CCC(c3c[nH]c4ccccc34)CC2)cc1 ZINC000217835991 IK On-Demand Unstable CCR2 106 46 Cc1ccccc1OC[C@@H](C)NC(=O)COc1ccc(Cl)cc1Cl ZINC000217835997 FI In-Stock Unstable SDH1 0 40 Cc1ccccc1OC[C@@H](C)NC(=O)COc1ccc(Cl)cc1Cl ZINC000217835997 FI In-Stock Unstable CETP 0 44 Cc1ccccc1OC[C@@H](C)NC(=O)COc1ccc(Cl)cc1Cl ZINC000217835997 FI In-Stock Unstable MCHR2 22 42 Cc1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1Cl ZINC000217836003 FK For-Sale Unstable LPL 42 32 COc1cccc(C2=NO[C@@H](C#N)C2)c1 ZINC000217836015 BD In-Stock Unstable LUCI_PHOPY 48 57 Cc1ccccc1OC[C@H](C)NC(=O)COc1ccc(Cl)cc1Cl ZINC000217836065 FI In-Stock Unstable SDH1 0 40 Cc1ccccc1OC[C@H](C)NC(=O)COc1ccc(Cl)cc1Cl ZINC000217836065 FI In-Stock Unstable CETP 0 44 Cc1ccccc1OC[C@H](C)NC(=O)COc1ccc(Cl)cc1Cl ZINC000217836065 FI In-Stock Unstable MCHR2 22 42 COc1ccc(CN(C)[C@H](C)C(C)C)cc1/C=C\C(=O)O ZINC000217836086 CG For-Sale Unstable PTGER2 34 47 COc1ccc(CN(C)[C@H](C)C(C)C)cc1/C=C\C(=O)O ZINC000217836086 CG For-Sale Unstable PTGER4 20 47 COc1ccc(CN(C)[C@H](C)C(C)C)cc1/C=C\C(=O)O ZINC000217836086 CG For-Sale Unstable PTGER3 18 42 O=C(O)[C@@H]1C[C@@H]2CCCC[C@@H]2N1C(=O)CNCC1CC1 ZINC000217836087 CD On-Demand Unstable ACE 17 60 Cc1cccc(C(C)C)c1NC(=O)N/C=C/c1ccccc1Br ZINC000217836099 FK For-Sale Unstable SOAT1 48 39 Cc1cccc(C(C)C)c1NC(=O)N/C=C/c1ccccc1Br ZINC000217836099 FK For-Sale Unstable ACAT 0 45 C[C@@H]1C(=O)NC(=O)CN1C(=O)/C=C\c1ccc(O)cc1 ZINC000217836120 CC For-Sale Unstable F3 18 40 N#Cc1cccc(OCCCN2CC[C@@H](CCO)C2)c1 ZINC000217836129 CE On-Demand Unstable HRH3 45 48 N#Cc1cccc(OCCCN2CC[C@@H](CCO)C2)c1 ZINC000217836129 CE On-Demand Unstable NPY1R 41 34 N#Cc1cccc(OCCCN2CC[C@@H](CCO)C2)c1 ZINC000217836129 CE On-Demand Unstable CHRNA10 45 48 N#Cc1cccc(OCCCN2CC[C@@H](CCO)C2)c1 ZINC000217836129 CE On-Demand Unstable MEN1 61 43 N#C[C@@H]1CC(c2ccc3c(c2)OCO3)=NO1 ZINC000217836135 BD In-Stock Unstable DYRK1A 41 33 N#C[C@@H]1CC(c2ccc3c(c2)OCO3)=NO1 ZINC000217836135 BD In-Stock Unstable CLK2 41 33 N#C[C@@H]1CC(c2ccc3c(c2)OCO3)=NO1 ZINC000217836135 BD In-Stock Unstable CLK4 68 33 O=C(NC[C@H]1CCCN1c1ccccc1)C1CCCC1 ZINC000217836137 CF For-Sale Unstable SLC6A1 58 34 O=C(NC[C@H]1CCCN1c1ccccc1)C1CCCC1 ZINC000217836137 CF For-Sale Unstable HCRTR1 15 41 O=C(O)[C@@H]1C[C@H]2CCCC[C@@H]2N1C(=O)CNCC1CC1 ZINC000217836154 CD On-Demand Unstable ACE 17 60 COc1ccc(CN(C)[C@@H](C)C(C)C)cc1/C=C\C(=O)O ZINC000217836163 CG For-Sale Unstable PTGER2 34 47 COc1ccc(CN(C)[C@@H](C)C(C)C)cc1/C=C\C(=O)O ZINC000217836163 CG For-Sale Unstable PTGER4 0 47 COc1ccc(CN(C)[C@@H](C)C(C)C)cc1/C=C\C(=O)O ZINC000217836163 CG For-Sale Unstable PTGER3 16 47 Cc1ccc(OC[C@@H](C)NC(=O)COc2ccc(Cl)cc2Cl)cc1 ZINC000217836181 FI In-Stock Unstable S1PR4 23 40 N#C[C@H]1CC(c2ccc3c(c2)OCO3)=NO1 ZINC000217836192 BD In-Stock Unstable DYRK1A 41 33 N#C[C@H]1CC(c2ccc3c(c2)OCO3)=NO1 ZINC000217836192 BD In-Stock Unstable CLK2 41 33 N#C[C@H]1CC(c2ccc3c(c2)OCO3)=NO1 ZINC000217836192 BD In-Stock Unstable CLK4 68 33 C[C@H]1C(=O)NC(=O)CN1C(=O)/C=C\c1ccc(O)cc1 ZINC000217836200 CC For-Sale Unstable F3 18 40 O=C(NC[C@@H]1CCCN1c1ccccc1)C1CCCC1 ZINC000217836206 CF For-Sale Unstable SLC6A1 58 34 O=C(NC[C@@H]1CCCN1c1ccccc1)C1CCCC1 ZINC000217836206 CF For-Sale Unstable HCRTR1 15 41 N#Cc1cccc(OCCCN2CC[C@H](CCO)C2)c1 ZINC000217836222 CE On-Demand Unstable HRH3 45 48 N#Cc1cccc(OCCCN2CC[C@H](CCO)C2)c1 ZINC000217836222 CE On-Demand Unstable NPY1R 41 34 N#Cc1cccc(OCCCN2CC[C@H](CCO)C2)c1 ZINC000217836222 CE On-Demand Unstable CHRNA10 45 48 N#Cc1cccc(OCCCN2CC[C@H](CCO)C2)c1 ZINC000217836222 CE On-Demand Unstable MEN1 61 43 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)NCC2(c3ccccc3)CC2)[C@@H](C)O)cc1 ZINC000217836252 HD On-Demand Unstable MMP13 40 47 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)NCC2(c3ccccc3)CC2)[C@@H](C)O)cc1 ZINC000217836252 HD On-Demand Unstable KCNA3 46 37 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)NCC2(c3ccccc3)CC2)[C@@H](C)O)cc1 ZINC000217836252 HD On-Demand Unstable CAPNS1 24 42 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)NCC2(c3ccccc3)CC2)[C@@H](C)O)cc1 ZINC000217836252 HD On-Demand Unstable MMP2 36 47 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)NCC2(c3ccccc3)CC2)[C@@H](C)O)cc1 ZINC000217836252 HD On-Demand Unstable MMP3 16 47 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)NCC2(c3ccccc3)CC2)[C@@H](C)O)cc1 ZINC000217836252 HD On-Demand Unstable MMP8 15 43 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)NCC2(c3ccccc3)CC2)[C@@H](C)O)cc1 ZINC000217836252 HD On-Demand Unstable CAPN1 16 48 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)NCC2(c3ccccc3)CC2)[C@@H](C)O)cc1 ZINC000217836252 HD On-Demand Unstable MMP9 22 41 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)NCC2(c3ccccc3)CC2)[C@@H](C)O)cc1 ZINC000217836252 HD On-Demand Unstable MMP12 46 43 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)NCC2(c3ccccc3)CC2)[C@@H](C)O)cc1 ZINC000217836252 HD On-Demand Unstable MMP7 19 43 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)NCC2(c3ccccc3)CC2)[C@@H](C)O)cc1 ZINC000217836252 HD On-Demand Unstable ADAMTS4 66 39 CC[C@@H](C)c1ccc(OCc2cccc(C)c2)cc1 ZINC000217836255 CK For-Sale Unstable MAOB 46 48 CC[C@@H](C)c1ccc(OCc2cccc(C)c2)cc1 ZINC000217836255 CK For-Sale Unstable FFAR1 49 57 Cc1ccc(OC[C@H](C)NC(=O)COc2ccc(Cl)cc2Cl)cc1 ZINC000217836261 FI In-Stock Unstable S1PR4 23 40 CCn1cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c(=O)c2ccc(C)nc21 ZINC000217836301 GG For-Sale Unstable CNR2 24 54 CC[C@H](C)c1ccc(OCc2cccc(C)c2)cc1 ZINC000217836337 CK For-Sale Unstable MAOB 46 48 CC[C@H](C)c1ccc(OCc2cccc(C)c2)cc1 ZINC000217836337 CK For-Sale Unstable FFAR1 49 57 Cc1ccc(S(=O)(=O)N[C@H](C(=O)NCC2(c3ccccc3)CC2)[C@@H](C)O)cc1 ZINC000217836344 HD On-Demand Unstable MMP13 40 47 Cc1ccc(S(=O)(=O)N[C@H](C(=O)NCC2(c3ccccc3)CC2)[C@@H](C)O)cc1 ZINC000217836344 HD On-Demand Unstable KCNA3 46 37 Cc1ccc(S(=O)(=O)N[C@H](C(=O)NCC2(c3ccccc3)CC2)[C@@H](C)O)cc1 ZINC000217836344 HD On-Demand Unstable CAPNS1 24 42 Cc1ccc(S(=O)(=O)N[C@H](C(=O)NCC2(c3ccccc3)CC2)[C@@H](C)O)cc1 ZINC000217836344 HD On-Demand Unstable MMP2 36 47 Cc1ccc(S(=O)(=O)N[C@H](C(=O)NCC2(c3ccccc3)CC2)[C@@H](C)O)cc1 ZINC000217836344 HD On-Demand Unstable MMP3 16 47 Cc1ccc(S(=O)(=O)N[C@H](C(=O)NCC2(c3ccccc3)CC2)[C@@H](C)O)cc1 ZINC000217836344 HD On-Demand Unstable MMP8 15 43 Cc1ccc(S(=O)(=O)N[C@H](C(=O)NCC2(c3ccccc3)CC2)[C@@H](C)O)cc1 ZINC000217836344 HD On-Demand Unstable CAPN1 16 48 Cc1ccc(S(=O)(=O)N[C@H](C(=O)NCC2(c3ccccc3)CC2)[C@@H](C)O)cc1 ZINC000217836344 HD On-Demand Unstable MMP9 22 41 Cc1ccc(S(=O)(=O)N[C@H](C(=O)NCC2(c3ccccc3)CC2)[C@@H](C)O)cc1 ZINC000217836344 HD On-Demand Unstable MMP12 46 43 Cc1ccc(S(=O)(=O)N[C@H](C(=O)NCC2(c3ccccc3)CC2)[C@@H](C)O)cc1 ZINC000217836344 HD On-Demand Unstable MMP7 19 43 Cc1ccc(S(=O)(=O)N[C@H](C(=O)NCC2(c3ccccc3)CC2)[C@@H](C)O)cc1 ZINC000217836344 HD On-Demand Unstable ADAMTS4 66 39 NC(=O)C[C@H](N)C(=O)N1[C@@H](C(=O)O)C[C@H]2CCCC[C@H]21 ZINC000217836350 CB For-Sale Unstable ACE 20 59 CC1CCN(c2ccc([C@@H](C)NC(=O)COc3ccc(Cl)cc3Cl)cc2)CC1 ZINC000217836353 HK In-Stock Unstable PRCP 22 40 Cc1csc(NCCNC(=O)OC(C)(C)C)n1 ZINC000217836361 CE On-Demand Unstable PAPA1_CARPA 42 36 CCn1cc(C(=O)NC[C@H]2CCCN2c2ccccc2)c(=O)c2ccc(C)nc21 ZINC000217836396 GG For-Sale Unstable CNR2 24 54 Cc1c(Cl)cccc1NC(=O)N/C=C/c1ccccc1Br ZINC000217836397 FK For-Sale Unstable CXCL8 41 33 CC1CCN(c2ccc([C@H](C)NC(=O)COc3ccc(Cl)cc3Cl)cc2)CC1 ZINC000217836421 HK In-Stock Unstable PRCP 22 40 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)NCC2(c3ccccc3)CC2)[C@H](C)O)cc1 ZINC000217836438 HD On-Demand Unstable MMP13 40 47 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)NCC2(c3ccccc3)CC2)[C@H](C)O)cc1 ZINC000217836438 HD On-Demand Unstable KCNA3 46 37 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)NCC2(c3ccccc3)CC2)[C@H](C)O)cc1 ZINC000217836438 HD On-Demand Unstable CAPNS1 24 42 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)NCC2(c3ccccc3)CC2)[C@H](C)O)cc1 ZINC000217836438 HD On-Demand Unstable MMP2 36 47 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)NCC2(c3ccccc3)CC2)[C@H](C)O)cc1 ZINC000217836438 HD On-Demand Unstable MMP3 16 47 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)NCC2(c3ccccc3)CC2)[C@H](C)O)cc1 ZINC000217836438 HD On-Demand Unstable MMP8 15 43 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)NCC2(c3ccccc3)CC2)[C@H](C)O)cc1 ZINC000217836438 HD On-Demand Unstable CAPN1 16 48 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)NCC2(c3ccccc3)CC2)[C@H](C)O)cc1 ZINC000217836438 HD On-Demand Unstable MMP9 22 41 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)NCC2(c3ccccc3)CC2)[C@H](C)O)cc1 ZINC000217836438 HD On-Demand Unstable MMP12 46 43 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)NCC2(c3ccccc3)CC2)[C@H](C)O)cc1 ZINC000217836438 HD On-Demand Unstable MMP7 19 43 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)NCC2(c3ccccc3)CC2)[C@H](C)O)cc1 ZINC000217836438 HD On-Demand Unstable ADAMTS4 66 39 NC(=O)C[C@H](N)C(=O)N1[C@H]2CCCC[C@@H]2C[C@@H]1C(=O)O ZINC000217836442 CB For-Sale Unstable ACE 20 59 N#C[C@@H]1CC(c2ccccc2Cl)=NO1 ZINC000217836478 BE In-Stock Unstable LUCI_PHOPY 37 53 Cc1cccc(COc2cccc(C)c2C)c1 ZINC000217836481 BI For-Sale Unstable MAOB 19 45 Cc1cccc(COc2cccc(C)c2C)c1 ZINC000217836481 BI For-Sale Unstable FFAR1 29 41 CCOC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217836485 GI For-Sale Unstable CA1 18 43 CCOC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217836485 GI For-Sale Unstable ACR 63 36 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc2noc(-c3ccccc3)c2c1 ZINC000217836487 GJ For-Sale Unstable HCRTR1 19 41 Cc1cc(CC(=O)O)cc(Br)c1F ZINC000217836491 BF For-Sale Unstable THRA 41 45 Cc1ccc(S(=O)(=O)N[C@H](C(=O)NCC2(c3ccccc3)CC2)[C@H](C)O)cc1 ZINC000217836527 HD On-Demand Unstable MMP13 40 47 Cc1ccc(S(=O)(=O)N[C@H](C(=O)NCC2(c3ccccc3)CC2)[C@H](C)O)cc1 ZINC000217836527 HD On-Demand Unstable KCNA3 46 37 Cc1ccc(S(=O)(=O)N[C@H](C(=O)NCC2(c3ccccc3)CC2)[C@H](C)O)cc1 ZINC000217836527 HD On-Demand Unstable CAPNS1 24 42 Cc1ccc(S(=O)(=O)N[C@H](C(=O)NCC2(c3ccccc3)CC2)[C@H](C)O)cc1 ZINC000217836527 HD On-Demand Unstable MMP2 36 47 Cc1ccc(S(=O)(=O)N[C@H](C(=O)NCC2(c3ccccc3)CC2)[C@H](C)O)cc1 ZINC000217836527 HD On-Demand Unstable MMP3 16 47 Cc1ccc(S(=O)(=O)N[C@H](C(=O)NCC2(c3ccccc3)CC2)[C@H](C)O)cc1 ZINC000217836527 HD On-Demand Unstable MMP8 15 43 Cc1ccc(S(=O)(=O)N[C@H](C(=O)NCC2(c3ccccc3)CC2)[C@H](C)O)cc1 ZINC000217836527 HD On-Demand Unstable CAPN1 16 48 Cc1ccc(S(=O)(=O)N[C@H](C(=O)NCC2(c3ccccc3)CC2)[C@H](C)O)cc1 ZINC000217836527 HD On-Demand Unstable MMP9 22 41 Cc1ccc(S(=O)(=O)N[C@H](C(=O)NCC2(c3ccccc3)CC2)[C@H](C)O)cc1 ZINC000217836527 HD On-Demand Unstable MMP12 46 43 Cc1ccc(S(=O)(=O)N[C@H](C(=O)NCC2(c3ccccc3)CC2)[C@H](C)O)cc1 ZINC000217836527 HD On-Demand Unstable MMP7 19 43 Cc1ccc(S(=O)(=O)N[C@H](C(=O)NCC2(c3ccccc3)CC2)[C@H](C)O)cc1 ZINC000217836527 HD On-Demand Unstable ADAMTS4 66 39 Cc1cc(C)n(Cc2ccccc2/C=C\C(=O)O)c(=O)n1 ZINC000217836550 CE For-Sale Unstable PTGER3 22 45 N#C[C@H]1CC(c2ccccc2Cl)=NO1 ZINC000217836556 BE In-Stock Unstable LUCI_PHOPY 37 53 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc2noc(-c3ccccc3)c2c1 ZINC000217836568 GJ For-Sale Unstable HCRTR1 19 41 O=C(O)[C@@H]1C[C@@H]2CCCC[C@@H]2N1C(=O)CNC1CCCC1 ZINC000217836615 CD For-Sale Unstable ACE 20 61 O=C(O)[C@@H]1C[C@@H]2CCCC[C@@H]2N1C(=O)CNC1CCCC1 ZINC000217836615 CD For-Sale Unstable DPP7 17 40 Cc1cc(C)n(Cc2ccc(/C=C\C(=O)O)cc2)c(=O)n1 ZINC000217836625 CE For-Sale Unstable HDAC6 23 44 COc1ccc(CN2C(=O)N[C@@H](CCC(=O)NCCc3ccc(O)cc3)C2=O)cc1 ZINC000217836637 HD In-Stock Unstable PROKR1 60 37 CC(C)c1ccccc1NC(=O)N/C=C/c1ccccc1Br ZINC000217836641 FK For-Sale Unstable ACAT 0 40 O=C(NCC1(c2ccccc2)CC1)c1nn(-c2ccccc2)cc1O ZINC000217836647 EG On-Demand Unstable ACAT 0 43 O=C(O)[C@@H]1C[C@H]2CCCC[C@@H]2N1C(=O)CNC1CCCC1 ZINC000217836691 CD For-Sale Unstable ACE 20 61 O=C(O)[C@@H]1C[C@H]2CCCC[C@@H]2N1C(=O)CNC1CCCC1 ZINC000217836691 CD For-Sale Unstable DPP7 17 40 N#C[C@@H]1CC(c2ccccc2F)=NO1 ZINC000217836704 AD In-Stock Unstable LUCI_PHOPY 46 53 COC(=O)c1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217836707 EF For-Sale Unstable DRD2 42 45 COC(=O)c1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217836707 EF For-Sale Unstable DRD3 19 46 COC(=O)c1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217836707 EF For-Sale Unstable HCRTR1 31 43 COC(=O)c1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217836707 EF For-Sale Unstable HCRTR2 28 43 COC(=O)c1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217836707 EF For-Sale Unstable HCN1 56 34 COC(=O)c1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217836707 EF For-Sale Unstable HCN4 51 33 COC(=O)c1ccccc1C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217836707 EF For-Sale Unstable ACKR3 50 33 O=C(O)Cc1ccc(CF)c(Br)c1 ZINC000217836708 BF For-Sale Unstable THRA 39 40 O=C(O)Cc1ccc(CF)c(Br)c1 ZINC000217836708 BF For-Sale Unstable THRB 31 40 COC(=O)c1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217836762 EF For-Sale Unstable DRD2 42 45 COC(=O)c1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217836762 EF For-Sale Unstable DRD3 19 46 COC(=O)c1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217836762 EF For-Sale Unstable HCRTR1 31 43 COC(=O)c1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217836762 EF For-Sale Unstable HCRTR2 28 43 COC(=O)c1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217836762 EF For-Sale Unstable HCN1 56 34 COC(=O)c1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217836762 EF For-Sale Unstable HCN4 51 33 COC(=O)c1ccccc1C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217836762 EF For-Sale Unstable ACKR3 50 33 N#C[C@H]1CC(c2ccccc2F)=NO1 ZINC000217836767 AD In-Stock Unstable LUCI_PHOPY 46 53 N[C@@H](CCCS)CC(=O)O ZINC000217836800 AC For-Sale Unstable ANPEP 0 52 N[C@@H](CCCS)CC(=O)O ZINC000217836800 AC For-Sale Unstable ENPEP 52 52 N[C@@H](CCCS)CC(=O)O ZINC000217836800 AC For-Sale Unstable GSTK1 48 36 C/C(=C/c1ccccc1)CN1CCN(C(=O)c2cccnc2)CC1 ZINC000217836821 DF On-Demand Unstable ADRA2A 28 43 C/C(=C/c1ccccc1)CN1CCN(C(=O)c2cccnc2)CC1 ZINC000217836821 DF On-Demand Unstable ADRA2C 63 39 C/C(=C/c1ccccc1)CN1CCN(C(=O)c2cccnc2)CC1 ZINC000217836821 DF On-Demand Unstable SMO 15 40 N[C@H](CCCS)CC(=O)O ZINC000217836870 AC For-Sale Unstable ANPEP 0 52 N[C@H](CCCS)CC(=O)O ZINC000217836870 AC For-Sale Unstable ENPEP 52 52 N[C@H](CCCS)CC(=O)O ZINC000217836870 AC For-Sale Unstable GSTK1 48 36 O=C(c1csc(-c2ccccc2)n1)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217836886 IH In-Stock Unstable COLA 40 39 O=C(NC[C@H]1CCCN1c1ccccc1)c1cccc(F)c1 ZINC000217836889 CG For-Sale Unstable SLC6A1 44 37 O=C(NC[C@H]1CCCN1c1ccccc1)c1cccc(F)c1 ZINC000217836889 CG For-Sale Unstable HCRTR1 32 45 O=C(NC[C@H]1CCCN1c1ccccc1)c1cccc(F)c1 ZINC000217836889 CG For-Sale Unstable CCR3 24 41 O=C(NC[C@H]1CCCN1c1ccccc1)c1cccc(F)c1 ZINC000217836889 CG For-Sale Unstable PREP 24 41 O=C(NC[C@H]1CCCN1c1ccccc1)c1cccc(F)c1 ZINC000217836889 CG For-Sale Unstable CCR2 28 41 O=C(NC[C@H]1CCCN1c1ccccc1)c1cccc(F)c1 ZINC000217836889 CG For-Sale Unstable PLD2 41 36 O=C(NC[C@H]1CCCN1c1ccccc1)c1cccc(F)c1 ZINC000217836889 CG For-Sale Unstable HCRTR2 23 45 O=C(NC[C@H]1CCCN1c1ccccc1)c1cccc(F)c1 ZINC000217836889 CG For-Sale Unstable ACKR3 68 36 O=C(NC[C@H]1CCCN1c1ccccc1)c1cccc(F)c1 ZINC000217836889 CG For-Sale Unstable KCNK3 15 42 CC(C)c1nccn1Cc1cccc(/C=C\C(=O)O)c1 ZINC000217836923 CG For-Sale Unstable AKR1C3 30 41 O=C(c1csc(-c2ccccc2)n1)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217836967 IH In-Stock Unstable COLA 40 39 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cccc(F)c1 ZINC000217836978 CG For-Sale Unstable SLC6A1 44 37 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cccc(F)c1 ZINC000217836978 CG For-Sale Unstable HCRTR1 32 45 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cccc(F)c1 ZINC000217836978 CG For-Sale Unstable CCR3 24 41 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cccc(F)c1 ZINC000217836978 CG For-Sale Unstable PREP 24 41 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cccc(F)c1 ZINC000217836978 CG For-Sale Unstable CCR2 28 41 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cccc(F)c1 ZINC000217836978 CG For-Sale Unstable PLD2 41 36 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cccc(F)c1 ZINC000217836978 CG For-Sale Unstable HCRTR2 23 45 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cccc(F)c1 ZINC000217836978 CG For-Sale Unstable ACKR3 68 36 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cccc(F)c1 ZINC000217836978 CG For-Sale Unstable KCNK3 15 42 COc1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1Cl ZINC000217836996 GJ For-Sale Unstable HTR2A 22 40 COc1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1Cl ZINC000217836996 GJ For-Sale Unstable GRM4 19 49 COc1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1Cl ZINC000217836996 GJ For-Sale Unstable IMPDH2 0 42 COc1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1Cl ZINC000217836996 GJ For-Sale Unstable CYSP_PLAFA 41 34 CN1CCO[C@@H]([C@@H](O)CCCc2ccccc2)C1 ZINC000217837023 BD For-Sale Unstable SLC18A2 34 41 CN1CCO[C@@H]([C@@H](O)CCCc2ccccc2)C1 ZINC000217837023 BD For-Sale Unstable SIGMAR1 29 40 N[C@@H]1CCCN(S(=O)(=O)N2CCc3ccccc3C2)C1 ZINC000217837043 CC On-Demand Unstable AKR1C3 46 41 O=C(Nc1nc2c(s1)CN(Cc1ccccc1)CC2)c1nn(-c2ccccc2)cc1O ZINC000217837061 IH On-Demand Unstable SLC27A1 28 42 CN1C[C@@]2(C)CN(C(=S)NC(=O)c3ccccc3)C[C@@](C)(C1)[C@H]2O ZINC000217837071 ED In-Stock Unstable EPHX1 0 40 COc1cc(CN2CCC[C@@H](C)[C@@H]2C)cc(Br)c1O ZINC000217837081 EH For-Sale Unstable DRD2 30 40 CN1CC[C@@H](NCc2ccc(O)c(Cl)c2)C1=O ZINC000217837085 CD For-Sale Unstable DRD1 20 41 CN1CC[C@@H](NCc2ccc(O)c(Cl)c2)C1=O ZINC000217837085 CD For-Sale Unstable DRD5 23 41 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1c[nH]nn1 ZINC000217837092 CD For-Sale Unstable TRPM8 21 58 CN1CCO[C@H]([C@@H](O)CCCc2ccccc2)C1 ZINC000217837106 BD For-Sale Unstable SLC18A2 34 41 CN1CCO[C@H]([C@@H](O)CCCc2ccccc2)C1 ZINC000217837106 BD For-Sale Unstable SIGMAR1 29 40 O=C(N/C=C/c1ccccc1Br)Nc1cccc(C(F)(F)F)c1 ZINC000217837121 GK For-Sale Anodyne KDR 15 40 O=C(N/C=C/c1ccccc1Br)Nc1cccc(C(F)(F)F)c1 ZINC000217837121 GK For-Sale Anodyne RIPK1 42 39 O=C(N/C=C/c1ccccc1Br)Nc1cccc(C(F)(F)F)c1 ZINC000217837121 GK For-Sale Anodyne TRPM4 0 41 O=C(N/C=C/c1ccccc1Br)Nc1cccc(C(F)(F)F)c1 ZINC000217837121 GK For-Sale Anodyne KCNK3 44 47 Cc1ccc(/C=C\C(=O)N2CC(=O)NC(=O)[C@@H]2C)cc1 ZINC000217837150 CC For-Sale Unstable GPR183 0 41 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1c[nH]nn1 ZINC000217837160 CD For-Sale Unstable TRPM8 21 58 CN1CC[C@H](NCc2ccc(O)c(Cl)c2)C1=O ZINC000217837166 CD For-Sale Unstable DRD1 20 41 CN1CC[C@H](NCc2ccc(O)c(Cl)c2)C1=O ZINC000217837166 CD For-Sale Unstable DRD5 23 41 COc1cc(CN2CCC[C@H](C)[C@@H]2C)cc(Br)c1O ZINC000217837177 EH For-Sale Unstable DRD2 30 40 CSCC[C@H](N)C(=O)N1[C@H](C(=O)O)C[C@@H]2CCCC[C@H]21 ZINC000217837180 DD For-Sale Unstable ACE 23 57 COc1ccc(O)c(C(=O)Nc2nc3c(s2)CN(Cc2ccccc2)CC3)c1 ZINC000217837191 GH On-Demand Unstable GABRA1 23 43 COc1ccc(O)c(C(=O)Nc2nc3c(s2)CN(Cc2ccccc2)CC3)c1 ZINC000217837191 GH On-Demand Unstable DRD3 25 41 COc1ccc(O)c(C(=O)Nc2nc3c(s2)CN(Cc2ccccc2)CC3)c1 ZINC000217837191 GH On-Demand Unstable F10 16 44 COc1ccc(O)c(C(=O)Nc2nc3c(s2)CN(Cc2ccccc2)CC3)c1 ZINC000217837191 GH On-Demand Unstable SIGMAR1 17 40 COc1ccc(O)c(C(=O)Nc2nc3c(s2)CN(Cc2ccccc2)CC3)c1 ZINC000217837191 GH On-Demand Unstable PDK1 40 39 COc1ccc(O)c(C(=O)Nc2nc3c(s2)CN(Cc2ccccc2)CC3)c1 ZINC000217837191 GH On-Demand Unstable GABRA2 26 43 COc1ccc(O)c(C(=O)Nc2nc3c(s2)CN(Cc2ccccc2)CC3)c1 ZINC000217837191 GH On-Demand Unstable NOD1 29 45 COc1ccc(O)c(C(=O)Nc2nc3c(s2)CN(Cc2ccccc2)CC3)c1 ZINC000217837191 GH On-Demand Unstable NOD2 46 45 Cc1ccc(/C=C\C(=O)N2CC(=O)NC(=O)[C@H]2C)cc1 ZINC000217837235 CC For-Sale Unstable GPR183 0 41 O=C(c1cc2ccccc2[nH]1)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217837242 GG In-Stock Unstable AKR1C3 18 43 O=C(O)/C=C\c1ccccc1CN1C(=O)COCC1=O ZINC000217837260 CC For-Sale Unstable PTGER2 40 48 O=C(O)/C=C\c1ccccc1CN1C(=O)COCC1=O ZINC000217837260 CC For-Sale Unstable PTGER4 0 48 O=C(O)/C=C\c1ccccc1CN1C(=O)COCC1=O ZINC000217837260 CC For-Sale Unstable PTGER3 22 48 CSCC[C@H](N)C(=O)N1[C@H](C(=O)O)C[C@H]2CCCC[C@H]21 ZINC000217837262 DD For-Sale Unstable ACE 23 57 C[C@@H](c1cccc(Cl)c1)N(C)CC[C@@H](N)c1ccccc1 ZINC000217837307 DI For-Sale Unstable OPRL1 0 44 C[C@@H](c1cccc(Cl)c1)N(C)CC[C@@H](N)c1ccccc1 ZINC000217837307 DI For-Sale Unstable AOC3 16 43 O=C(c1cc2ccccc2[nH]1)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217837327 GG In-Stock Unstable AKR1C3 18 43 C[C@H](c1cccc(Cl)c1)N(C)CC[C@@H](N)c1ccccc1 ZINC000217837361 DI For-Sale Unstable OPRL1 0 44 C[C@H](c1cccc(Cl)c1)N(C)CC[C@@H](N)c1ccccc1 ZINC000217837361 DI For-Sale Unstable AOC3 16 43 COCCn1cc(CC(=O)Nc2ccc3c(ccn3C)c2)c2ccccc21 ZINC000217837399 FH In-Stock Unstable CNR1 0 43 COCCn1cc(CC(=O)Nc2ccc3c(ccn3C)c2)c2ccccc21 ZINC000217837399 FH In-Stock Unstable CYSLTR1 0 41 COCCn1cc(CC(=O)Nc2ccc3c(ccn3C)c2)c2ccccc21 ZINC000217837399 FH In-Stock Unstable CNR2 17 57 COCCn1cc(CC(=O)Nc2ccc3c(ccn3C)c2)c2ccccc21 ZINC000217837399 FH In-Stock Unstable RORC 38 42 CN(Cc1ccccc1)S(=O)(=O)N1CCC[C@@H](N)C1 ZINC000217837425 CC For-Sale Unstable DPP4 21 41 CS(=O)(=O)CC(=O)Nc1ccc(I)cc1Cl ZINC000217837446 FD On-Demand Unstable CA1 25 46 CS(=O)(=O)CC(=O)Nc1ccc(I)cc1Cl ZINC000217837446 FD On-Demand Unstable CA4 29 46 CCCCOc1ccc(CN[C@@H]2CCN(C)C2=O)cc1 ZINC000217837494 CE For-Sale Unstable LTA4H 40 40 CCCCOc1ccc(CN[C@@H]2CCN(C)C2=O)cc1 ZINC000217837494 CE For-Sale Unstable HRH3 73 51 CCCCOc1ccc(CN[C@@H]2CCN(C)C2=O)cc1 ZINC000217837494 CE For-Sale Unstable PLA2G4B 65 34 CC[C@@H](NC(=O)COc1ccc(Cl)cc1Cl)c1ccc(C)c(C)c1 ZINC000217837500 FK In-Stock Unstable MCHR2 22 42 N#C[C@@H]1CC(c2cccc(Cl)c2Cl)=NO1 ZINC000217837502 BG In-Stock Unstable LUCI_PHOPY 32 42 O=C(O)/C=C\c1ccccc1COc1ccc(F)cc1F ZINC000217837506 CH For-Sale Unstable PTGER2 25 52 O=C(O)/C=C\c1ccccc1COc1ccc(F)cc1F ZINC000217837506 CH For-Sale Unstable PTGER1 39 41 O=C(O)/C=C\c1ccccc1COc1ccc(F)cc1F ZINC000217837506 CH For-Sale Unstable PTGER4 41 52 O=C(O)/C=C\c1ccccc1COc1ccc(F)cc1F ZINC000217837506 CH For-Sale Unstable FABP4 17 40 O=C(O)/C=C\c1ccccc1COc1ccc(F)cc1F ZINC000217837506 CH For-Sale Unstable PTGER3 35 52 O=C(O)/C=C\c1ccccc1COc1ccc(F)cc1F ZINC000217837506 CH For-Sale Unstable PTGDR 0 46 O=C(O)/C=C\c1ccccc1COc1ccc(F)cc1F ZINC000217837506 CH For-Sale Unstable AKR1C3 32 48 COc1ccc(Cl)cc1NC(=O)N/C=C/c1ccccc1Br ZINC000217837556 GJ For-Sale Unstable RBP4 24 44 COc1ccc(Cl)cc1NC(=O)N/C=C/c1ccccc1Br ZINC000217837556 GJ For-Sale Unstable CYSP_PLAFA 44 37 O=C(CNC(=O)c1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217837564 EE For-Sale Unstable CA2 17 42 O=C(CNC(=O)c1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217837564 EE For-Sale Unstable PREP 26 51 O=C(CNC(=O)c1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217837564 EE For-Sale Unstable CCR2 33 48 CC[C@@H](C)[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(Cc2ccccc2)C1=O ZINC000217837573 ED In-Stock Unstable GALR1 49 36 CC[C@H](NC(=O)COc1ccc(Cl)cc1Cl)c1ccc(C)c(C)c1 ZINC000217837580 FK In-Stock Unstable MCHR2 22 42 CCCCOc1ccc(CN[C@H]2CCN(C)C2=O)cc1 ZINC000217837592 CE For-Sale Unstable LTA4H 40 40 CCCCOc1ccc(CN[C@H]2CCN(C)C2=O)cc1 ZINC000217837592 CE For-Sale Unstable HRH3 73 51 CCCCOc1ccc(CN[C@H]2CCN(C)C2=O)cc1 ZINC000217837592 CE For-Sale Unstable PLA2G4B 65 34 N#C[C@H]1CC(c2cccc(Cl)c2Cl)=NO1 ZINC000217837594 BG In-Stock Unstable LUCI_PHOPY 32 42 O=C(O)[C@H]1CN(C(=O)[C@@H]2C[C@@H](O)CN2)c2ccccc2O1 ZINC000217837603 CB For-Sale Unstable DPP8 15 40 O=C(O)/C=C\c1ccc(COc2ccc(F)cc2F)cc1 ZINC000217837604 CH For-Sale Unstable PTGER2 16 48 O=C(O)/C=C\c1ccc(COc2ccc(F)cc2F)cc1 ZINC000217837604 CH For-Sale Unstable PTGER1 45 39 O=C(O)/C=C\c1ccc(COc2ccc(F)cc2F)cc1 ZINC000217837604 CH For-Sale Unstable PTGER4 32 43 O=C(O)/C=C\c1ccc(COc2ccc(F)cc2F)cc1 ZINC000217837604 CH For-Sale Unstable AKR1C3 41 58 O=C(O)/C=C\c1ccc(COc2ccc(F)cc2F)cc1 ZINC000217837604 CH For-Sale Unstable AKR1B10 16 41 O=C(CNC(=O)c1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217837643 EE For-Sale Unstable CA2 17 42 O=C(CNC(=O)c1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217837643 EE For-Sale Unstable PREP 26 51 O=C(CNC(=O)c1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217837643 EE For-Sale Unstable CCR2 33 48 CCCCc1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217837647 FK For-Sale Unstable P96878_MYCTU 17 51 CC[C@@H]1CN(c2cnc3ccccc3n2)CCN1 ZINC000217837651 BD For-Sale Unstable PRKCD 15 50 CC[C@@H]1CN(c2cnc3ccccc3n2)CCN1 ZINC000217837651 BD For-Sale Unstable PRKCQ 31 50 CC[C@@H](NC(=O)COc1ccc(Cl)cc1Cl)c1ccc(C)cc1C ZINC000217837686 FK In-Stock Unstable S1PR4 24 41 O=C(O)[C@H]1CN(C(=O)[C@H]2C[C@@H](O)CN2)c2ccccc2O1 ZINC000217837695 CB For-Sale Unstable DPP8 15 40 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2F)c1 ZINC000217837702 CH For-Sale Unstable EGFR 15 41 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2F)c1 ZINC000217837702 CH For-Sale Unstable MAOB 16 44 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2F)c1 ZINC000217837702 CH For-Sale Unstable PTGER2 23 47 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2F)c1 ZINC000217837702 CH For-Sale Unstable PPIA 25 42 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2F)c1 ZINC000217837702 CH For-Sale Unstable ERBB2 24 41 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2F)c1 ZINC000217837702 CH For-Sale Unstable PTGER1 63 39 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2F)c1 ZINC000217837702 CH For-Sale Unstable PTGER4 31 44 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2F)c1 ZINC000217837702 CH For-Sale Unstable LTB4R 22 43 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2F)c1 ZINC000217837702 CH For-Sale Unstable HCAR2 0 49 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2F)c1 ZINC000217837702 CH For-Sale Unstable AKR1C3 44 62 CC[C@H]1CN(c2cnc3ccccc3n2)CCN1 ZINC000217837723 BD For-Sale Unstable PRKCD 15 50 CC[C@H]1CN(c2cnc3ccccc3n2)CCN1 ZINC000217837723 BD For-Sale Unstable PRKCQ 31 50 O=C(O)C[C@@H](F)c1ccccc1Br ZINC000217837743 BF For-Sale Unstable CPA1 28 42 COc1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217837747 EI For-Sale Unstable CA1 45 36 COc1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217837747 EI For-Sale Unstable MTNR1B 18 45 COc1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217837747 EI For-Sale Unstable CA12 24 43 Cc1cc(C)cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217837752 DH For-Sale Unstable HCRTR1 24 43 Cc1cc(C)cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217837752 DH For-Sale Unstable PREP 22 42 Cc1cc(C)cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217837752 DH For-Sale Unstable HCRTR2 18 43 Cc1cc(C)cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217837752 DH For-Sale Unstable CACNA1I 64 39 Cc1cc(C)cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217837752 DH For-Sale Unstable ACKR3 53 35 CC[C@H](NC(=O)COc1ccc(Cl)cc1Cl)c1ccc(C)cc1C ZINC000217837767 FK In-Stock Unstable S1PR4 24 41 COc1cccc(C(=O)Nc2ccc3nc(N4CCCC4)sc3c2)c1O ZINC000217837785 FH On-Demand Unstable CSNK1D 22 40 COc1cccc(C(=O)Nc2ccc3nc(N4CCCC4)sc3c2)c1O ZINC000217837785 FH On-Demand Unstable ENPP1 51 33 COc1cccc(C(=O)Nc2ccc3nc(N4CCCC4)sc3c2)c1O ZINC000217837785 FH On-Demand Unstable KCNK3 56 43 COc1cccc(C(=O)Nc2ccc3nc(N4CCCC4)sc3c2)c1O ZINC000217837785 FH On-Demand Unstable KCNK9 56 43 CC[C@@H](C)c1ccc(OCc2cc(C)cc(C)c2)cc1 ZINC000217837796 CK For-Sale Unstable SCN2A 23 40 CC[C@@H](C)c1ccc(OCc2cc(C)cc(C)c2)cc1 ZINC000217837796 CK For-Sale Unstable FFAR1 18 42 C[C@@H]1C(=O)Nc2ccc(S(=O)(=O)N3CCC[C@@H](N)C3)cc21 ZINC000217837800 DC For-Sale Unstable CASP3 16 43 O=C(O)/C=C\c1ccccc1CN1CCCC[C@@H]1CCO ZINC000217837802 CF For-Sale Unstable SLC6A1 51 40 O=C(O)/C=C\c1ccccc1CN1CCCC[C@@H]1CCO ZINC000217837802 CF For-Sale Unstable PTGER2 28 42 O=C(O)C[C@H](F)c1ccccc1Br ZINC000217837819 BF For-Sale Unstable CPA1 28 42 Cc1cc(C)cc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217837824 DH For-Sale Unstable HCRTR1 24 43 Cc1cc(C)cc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217837824 DH For-Sale Unstable PREP 22 42 Cc1cc(C)cc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217837824 DH For-Sale Unstable HCRTR2 18 43 Cc1cc(C)cc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217837824 DH For-Sale Unstable CACNA1I 64 39 Cc1cc(C)cc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217837824 DH For-Sale Unstable ACKR3 53 35 C[C@H]1C(=O)Nc2ccc(S(=O)(=O)N3CCC[C@@H](N)C3)cc21 ZINC000217837847 DC For-Sale Unstable CASP3 16 43 O=C(CN1CCCCCC1)N1CCC(n2cnnc2)CC1 ZINC000217837857 CD In-Stock Unstable L3MBTL3 50 36 CC[C@H](C)c1ccc(OCc2cc(C)cc(C)c2)cc1 ZINC000217837864 CK For-Sale Unstable SCN2A 23 40 CC[C@H](C)c1ccc(OCc2cc(C)cc(C)c2)cc1 ZINC000217837864 CK For-Sale Unstable FFAR1 18 42 CC[C@@H](NC(=O)COc1ccc(Cl)cc1Cl)c1ccc(OC)c(OC)c1 ZINC000217837879 GJ In-Stock Unstable S1PR4 27 40 CC[C@@H](NC(=O)COc1ccc(Cl)cc1Cl)c1ccc(OC)c(OC)c1 ZINC000217837879 GJ In-Stock Unstable TTR 0 44 CC[C@@H](NC(=O)COc1ccc(Cl)cc1Cl)c1ccc(OC)c(OC)c1 ZINC000217837879 GJ In-Stock Unstable ENPP1 52 34 N#C[C@@H]1CC(c2cccc(F)c2)=NO1 ZINC000217837890 AD In-Stock Unstable LUCI_PHOPY 53 54 COc1ccc(CN2CCC[C@@H](C)[C@@H]2C)c(O)c1 ZINC000217837905 BG For-Sale Unstable SIGMAR1 21 45 CCCN(CC)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217837918 CF For-Sale Unstable SQLE 47 35 CCCN(CC)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217837918 CF For-Sale Unstable AKR1C3 35 40 O=C(Nc1ccc2nc(N3CCCC3)sc2c1)C1(c2ccccc2)CC1 ZINC000217837936 FJ On-Demand Unstable NMT1 32 41 O=C(Nc1ccc2nc(N3CCCC3)sc2c1)C1(c2ccccc2)CC1 ZINC000217837936 FJ On-Demand Unstable MLYCD 27 41 CC(C)[C@@H]1CN(c2cnc3cccc(C(F)(F)F)c3n2)CCN1 ZINC000217837950 DG For-Sale Unstable PRKCQ 25 45 CC[C@H](NC(=O)COc1ccc(Cl)cc1Cl)c1ccc(OC)c(OC)c1 ZINC000217837983 GJ In-Stock Unstable S1PR4 27 40 CC[C@H](NC(=O)COc1ccc(Cl)cc1Cl)c1ccc(OC)c(OC)c1 ZINC000217837983 GJ In-Stock Unstable TTR 0 44 CC[C@H](NC(=O)COc1ccc(Cl)cc1Cl)c1ccc(OC)c(OC)c1 ZINC000217837983 GJ In-Stock Unstable ENPP1 52 34 N#C[C@H]1CC(c2cccc(F)c2)=NO1 ZINC000217837986 AD In-Stock Unstable LUCI_PHOPY 53 54 COc1ccc(CN2CCC[C@H](C)[C@@H]2C)c(O)c1 ZINC000217837999 BG For-Sale Unstable SIGMAR1 21 45 CCCN(CC)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217838010 CF On-Demand Unstable ERG2 18 45 CCCN(CC)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217838010 CF On-Demand Unstable PLA2G4B 67 34 CC(C)[C@H]1CN(c2cnc3cccc(C(F)(F)F)c3n2)CCN1 ZINC000217838043 DG For-Sale Unstable PRKCQ 25 45 CC[C@@H](NC(=O)COc1ccc(Cl)cc1Cl)c1ccc(S(C)(=O)=O)cc1 ZINC000217838089 HI In-Stock Unstable PTGS2 18 41 CC[C@@H](NC(=O)COc1ccc(Cl)cc1Cl)c1ccc(S(C)(=O)=O)cc1 ZINC000217838089 HI In-Stock Unstable PTGDR2 39 47 CN1CCO[C@@H]([C@@H](O)c2ccc(Cl)cc2)C1 ZINC000217838097 BD For-Sale Unstable SLC6A1 30 40 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1Cl ZINC000217838131 EI For-Sale Unstable DRD2 33 41 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1Cl ZINC000217838131 EI For-Sale Unstable CNR1 25 41 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1Cl ZINC000217838131 EI For-Sale Unstable AVPR2 23 40 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1Cl ZINC000217838131 EI For-Sale Unstable DRD3 17 42 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1Cl ZINC000217838131 EI For-Sale Unstable P2RX7 26 46 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1Cl ZINC000217838131 EI For-Sale Unstable PREP 15 44 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1Cl ZINC000217838131 EI For-Sale Unstable SLC6A9 55 40 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1Cl ZINC000217838131 EI For-Sale Unstable CACNA1I 48 34 COc1ccc(/C=C\C(=O)O)cc1CN(C)C1CCCC1 ZINC000217838133 CG For-Sale Unstable PTGER2 0 42 COc1ccc(/C=C\C(=O)O)cc1CN(C)C1CCCC1 ZINC000217838133 CG For-Sale Unstable AKR1C3 22 40 COc1ccc(Cl)cc1NS(=O)(=O)CCCCO ZINC000217838134 CD For-Sale Unstable CPT1A 47 38 CC[C@H](NC(=O)COc1ccc(Cl)cc1Cl)c1ccc(S(C)(=O)=O)cc1 ZINC000217838152 HI In-Stock Unstable PTGS2 18 41 CC[C@H](NC(=O)COc1ccc(Cl)cc1Cl)c1ccc(S(C)(=O)=O)cc1 ZINC000217838152 HI In-Stock Unstable PTGDR2 39 47 CN1CCO[C@H]([C@@H](O)c2ccc(Cl)cc2)C1 ZINC000217838163 BD For-Sale Unstable SLC6A1 30 40 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1Cl ZINC000217838207 EI For-Sale Unstable DRD2 33 41 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1Cl ZINC000217838207 EI For-Sale Unstable CNR1 25 41 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1Cl ZINC000217838207 EI For-Sale Unstable AVPR2 23 40 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1Cl ZINC000217838207 EI For-Sale Unstable DRD3 17 42 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1Cl ZINC000217838207 EI For-Sale Unstable P2RX7 26 46 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1Cl ZINC000217838207 EI For-Sale Unstable PREP 15 44 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1Cl ZINC000217838207 EI For-Sale Unstable SLC6A9 55 40 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1Cl ZINC000217838207 EI For-Sale Unstable CACNA1I 48 34 CC(C)N(Cc1ccccc1)C(=O)N/C=C/c1ccccc1Br ZINC000217838215 FK For-Sale Unstable PTGES 0 42 CC(C)CN(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217838233 CF For-Sale Unstable AKR1C3 38 41 CC[C@@H](N)[C@H](c1cccs1)N1C[C@@H](C)Cc2ccccc21 ZINC000217838275 DI For-Sale Unstable TPP2 44 32 COc1ccc(-c2noc(CNC(=O)COc3ccc(Cl)cc3Cl)n2)c(OC)c1 ZINC000217838305 IH In-Stock Unstable COLA 51 34 COc1ccc(-c2noc(CNC(=O)COc3ccc(Cl)cc3Cl)n2)c(OC)c1 ZINC000217838305 IH In-Stock Unstable CPT1A 50 34 COc1ccc(-c2noc(CNC(=O)COc3ccc(Cl)cc3Cl)n2)c(OC)c1 ZINC000217838305 IH In-Stock Unstable PPARD 18 41 COc1ccc(-c2noc(CNC(=O)COc3ccc(Cl)cc3Cl)n2)c(OC)c1 ZINC000217838305 IH In-Stock Unstable CPT1B 61 32 COc1ccc(-c2noc(CNC(=O)COc3ccc(Cl)cc3Cl)n2)c(OC)c1 ZINC000217838305 IH In-Stock Unstable PDK1 15 40 CCOC(=O)[C@H](Oc1ccccc1Br)c1ccccc1 ZINC000217838316 EI On-Demand Unstable F9 21 41 CC[C@H](N)[C@H](c1cccs1)N1C[C@@H](C)Cc2ccccc21 ZINC000217838321 DI For-Sale Unstable TPP2 44 32 O=C(Nc1ccc2nc(N3CCCC3)sc2c1)c1ccnc2ccccc12 ZINC000217838356 FJ On-Demand Unstable NR2E3 43 31 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)c(Cl)c1 ZINC000217838360 EI For-Sale Unstable DRD2 28 41 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)c(Cl)c1 ZINC000217838360 EI For-Sale Unstable OPRK1 16 44 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)c(Cl)c1 ZINC000217838360 EI For-Sale Unstable F10 16 44 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)c(Cl)c1 ZINC000217838360 EI For-Sale Unstable CCR3 29 46 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)c(Cl)c1 ZINC000217838360 EI For-Sale Unstable PLD1 26 42 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)c(Cl)c1 ZINC000217838360 EI For-Sale Unstable PLD2 32 42 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)c(Cl)c1 ZINC000217838360 EI For-Sale Unstable CACNA1I 61 48 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)c(Cl)c1 ZINC000217838360 EI For-Sale Unstable RPA1 48 39 CC[C@@H](N)[C@@H](c1cccs1)N1C[C@@H](C)Cc2ccccc21 ZINC000217838414 DI For-Sale Unstable TPP2 44 32 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)c(Cl)c1 ZINC000217838429 EI For-Sale Unstable DRD2 28 41 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)c(Cl)c1 ZINC000217838429 EI For-Sale Unstable OPRK1 16 44 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)c(Cl)c1 ZINC000217838429 EI For-Sale Unstable F10 16 44 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)c(Cl)c1 ZINC000217838429 EI For-Sale Unstable CCR3 29 46 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)c(Cl)c1 ZINC000217838429 EI For-Sale Unstable PLD1 26 42 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)c(Cl)c1 ZINC000217838429 EI For-Sale Unstable PLD2 32 42 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)c(Cl)c1 ZINC000217838429 EI For-Sale Unstable CACNA1I 61 48 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)c(Cl)c1 ZINC000217838429 EI For-Sale Unstable RPA1 48 39 O=C(COc1ccc(Cl)cc1Cl)NCc1nc(-c2ccc(Cl)cc2)no1 ZINC000217838448 HI In-Stock Unstable CNR1 16 41 O=C(COc1ccc(Cl)cc1Cl)NCc1nc(-c2ccc(Cl)cc2)no1 ZINC000217838448 HI In-Stock Unstable CETP 0 40 CC[C@@H]1CCN(C[C@@H](O)c2ccc(C#N)cc2)C1 ZINC000217838489 BE For-Sale Unstable O19067_PIG 0 41 CC[C@H](N)[C@@H](c1cccs1)N1C[C@@H](C)Cc2ccccc21 ZINC000217838494 DI For-Sale Unstable TPP2 44 32 N#C[C@@H]1CC(Cc2ccccc2)=NO1 ZINC000217838499 AD In-Stock Unstable LUCI_PHOPY 60 39 COc1cc2c(cc1OC)CN(C(=O)c1cc3ccc(Cl)cc3n1C)CC2 ZINC000217838537 GI In-Stock Unstable ABCB1B 52 33 COc1cc2c(cc1OC)CN(C(=O)c1cc3ccc(Cl)cc3n1C)CC2 ZINC000217838537 GI In-Stock Unstable ABCB1 24 51 COc1cc2c(cc1OC)CN(C(=O)c1cc3ccc(Cl)cc3n1C)CC2 ZINC000217838537 GI In-Stock Unstable QRFPR 25 46 O=C(CC1CCCCC1)NC[C@H]1CCCN1c1ccccc1 ZINC000217838556 DH For-Sale Unstable CHRM4 17 40 O=C(CC1CCCCC1)NC[C@H]1CCCN1c1ccccc1 ZINC000217838556 DH For-Sale Unstable CHRM5 17 40 O=C(CC1CCCCC1)NC[C@H]1CCCN1c1ccccc1 ZINC000217838556 DH For-Sale Unstable DPEP1 40 32 CC[C@H]1CCN(C[C@@H](O)c2ccc(C#N)cc2)C1 ZINC000217838562 BE For-Sale Unstable O19067_PIG 0 41 N#C[C@H]1CC(Cc2ccccc2)=NO1 ZINC000217838577 AD In-Stock Unstable LUCI_PHOPY 60 39 CN(CCOc1cccc(/C=C\C(=O)O)c1)CC(N)=O ZINC000217838601 CC For-Sale Unstable FDPS 23 41 O=C(CC1CCCCC1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217838625 DH For-Sale Unstable CHRM4 17 40 O=C(CC1CCCCC1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217838625 DH For-Sale Unstable CHRM5 17 40 O=C(CC1CCCCC1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217838625 DH For-Sale Unstable DPEP1 40 32 COC(=O)C[C@@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(OC)cc1OC ZINC000217838641 GG In-Stock Unstable HDAC2 21 41 Cc1cc(F)ccc1CN[C@@H]1CCN(C)C1=O ZINC000217838642 BD For-Sale Unstable P2RX7 41 43 Cc1nc2ccccc2cc1C(=O)Nc1ccc2nc(N3CCCC3)sc2c1 ZINC000217838649 GK On-Demand Unstable NR2E3 52 34 Cc1nc2ccccc2cc1C(=O)Nc1ccc2nc(N3CCCC3)sc2c1 ZINC000217838649 GK On-Demand Unstable SHH 26 40 CC(C)c1ccc(CCCNC(=O)COc2ccc(Cl)cc2Cl)cc1 ZINC000217838658 GK In-Stock Unstable ALPL 41 35 CN(CCOc1ccc(/C=C\C(=O)O)cc1)CC(N)=O ZINC000217838702 CC For-Sale Unstable FDPS 24 42 CN(CCOc1ccc(/C=C\C(=O)O)cc1)CC(N)=O ZINC000217838702 CC For-Sale Unstable LTA4H 18 43 CCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OCC ZINC000217838703 FH For-Sale Unstable DRD2 30 40 CCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OCC ZINC000217838703 FH For-Sale Unstable DRD3 20 40 CCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OCC ZINC000217838703 FH For-Sale Unstable SSTR5 45 38 CCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OCC ZINC000217838703 FH For-Sale Unstable MCHR1 15 48 CCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OCC ZINC000217838703 FH For-Sale Unstable CACNA1I 45 36 CCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OCC ZINC000217838703 FH For-Sale Unstable HCN1 46 36 CCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OCC ZINC000217838703 FH For-Sale Unstable HCN4 46 36 CCOc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OCC ZINC000217838703 FH For-Sale Unstable ACKR3 69 38 N#C[C@@H]1CC(c2ccc(N)cc2)=NO1 ZINC000217838704 AD In-Stock Unstable LUCI_PHOPY 41 40 COC(=O)C[C@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(OC)cc1OC ZINC000217838713 GG In-Stock Unstable HDAC2 21 41 Cc1cc(F)ccc1CN[C@H]1CCN(C)C1=O ZINC000217838727 BD For-Sale Unstable P2RX7 41 43 CN(CCCNC(=O)COc1ccc(Cl)cc1Cl)c1ccccc1 ZINC000217838748 FI In-Stock Unstable MCHR2 23 46 CN(CCCNC(=O)COc1ccc(Cl)cc1Cl)c1ccccc1 ZINC000217838748 FI In-Stock Unstable PTGDR2 33 41 N#C[C@H]1CC(c2ccc(N)cc2)=NO1 ZINC000217838769 AD In-Stock Unstable LUCI_PHOPY 41 40 CCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1OCC ZINC000217838779 FH For-Sale Unstable DRD2 30 40 CCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1OCC ZINC000217838779 FH For-Sale Unstable DRD3 20 40 CCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1OCC ZINC000217838779 FH For-Sale Unstable SSTR5 45 38 CCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1OCC ZINC000217838779 FH For-Sale Unstable MCHR1 15 48 CCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1OCC ZINC000217838779 FH For-Sale Unstable CACNA1I 45 36 CCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1OCC ZINC000217838779 FH For-Sale Unstable HCN1 46 36 CCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1OCC ZINC000217838779 FH For-Sale Unstable HCN4 46 36 CCOc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1OCC ZINC000217838779 FH For-Sale Unstable ACKR3 69 38 COc1cc([C@@H]2CC(=O)Oc3ccc4c(c32)OC(=C(C)C)C4=O)ccc1OC(C)C ZINC000217838845 HJ In-Stock Unstable MT-ND4 40 30 N#C[C@@H]1CC(c2ccc([N+](=O)[O-])cc2)=NO1 ZINC000217838864 BD In-Stock Unstable H9B8T9_CAPHI 24 41 N#C[C@@H]1CC(c2ccc([N+](=O)[O-])cc2)=NO1 ZINC000217838864 BD In-Stock Unstable A0A060INS8_CAPHI 0 41 O=C(COc1ccc(Cl)cc1Cl)NCCCN1CCCc2ccccc21 ZINC000217838871 GI In-Stock Unstable AVPR2 15 40 O=C(COc1ccc(Cl)cc1Cl)NCCCN1CCCc2ccccc21 ZINC000217838871 GI In-Stock Unstable GPBAR1 19 42 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1OC ZINC000217838872 FG For-Sale Unstable HTR1A 25 49 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1OC ZINC000217838872 FG For-Sale Unstable DRD2 58 52 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1OC ZINC000217838872 FG For-Sale Unstable DRD4 26 42 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1OC ZINC000217838872 FG For-Sale Unstable DRD3 44 49 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1OC ZINC000217838872 FG For-Sale Unstable KCNA3 45 38 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1OC ZINC000217838872 FG For-Sale Unstable HCN1 68 37 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1OC ZINC000217838872 FG For-Sale Unstable HCN4 51 35 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1OC ZINC000217838872 FG For-Sale Unstable ACKR3 73 39 COc1cc(C(=O)Nc2ccc(Sc3nccn3C)cc2)ccc1OCC(C)C ZINC000217838907 HJ On-Demand Unstable COLA 53 40 COc1cc(C(=O)Nc2ccc(Sc3nccn3C)cc2)ccc1OCC(C)C ZINC000217838907 HJ On-Demand Unstable CPT1A 54 40 COc1cc(C(=O)Nc2ccc(Sc3nccn3C)cc2)ccc1OCC(C)C ZINC000217838907 HJ On-Demand Unstable SYK 22 40 COc1cc(C(=O)Nc2ccc(Sc3nccn3C)cc2)ccc1OCC(C)C ZINC000217838907 HJ On-Demand Unstable MAP2K1 25 42 COc1cc(C(=O)Nc2ccc(Sc3nccn3C)cc2)ccc1OCC(C)C ZINC000217838907 HJ On-Demand Unstable PDGFRA 47 35 COc1cc(C(=O)Nc2ccc(Sc3nccn3C)cc2)ccc1OCC(C)C ZINC000217838907 HJ On-Demand Unstable ENPP1 70 35 O=C(N/C=C/c1ccccc1Br)NC1CCCCC1 ZINC000217838916 DI For-Sale Unstable EPHX2 24 48 COc1cc([C@H]2CC(=O)Oc3ccc4c(c32)OC(=C(C)C)C4=O)ccc1OC(C)C ZINC000217838930 HJ In-Stock Unstable MT-ND4 40 30 N#C[C@H]1CC(c2ccc([N+](=O)[O-])cc2)=NO1 ZINC000217838937 BD In-Stock Unstable H9B8T9_CAPHI 24 41 N#C[C@H]1CC(c2ccc([N+](=O)[O-])cc2)=NO1 ZINC000217838937 BD In-Stock Unstable A0A060INS8_CAPHI 0 41 CN1C[C@@]2(C)CN(C(=S)NC(=O)c3ccc(Cl)cc3)C[C@@](C)(C1)[C@H]2O ZINC000217838943 GD In-Stock Unstable CCR1 44 38 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1OC ZINC000217838955 FG For-Sale Unstable HTR1A 25 49 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1OC ZINC000217838955 FG For-Sale Unstable DRD2 58 52 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1OC ZINC000217838955 FG For-Sale Unstable DRD4 26 42 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1OC ZINC000217838955 FG For-Sale Unstable DRD3 44 49 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1OC ZINC000217838955 FG For-Sale Unstable KCNA3 45 38 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1OC ZINC000217838955 FG For-Sale Unstable HCN1 68 37 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1OC ZINC000217838955 FG For-Sale Unstable HCN4 51 35 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1OC ZINC000217838955 FG For-Sale Unstable ACKR3 73 39 C[C@@H]1COCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217838960 CD On-Demand Unstable HRH3 21 42 C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1ccc2c(c1)OCCO2 ZINC000217838978 CC In-Stock Unstable KCNQ2 21 40 CSc1ccc(C(=O)N2CCC[C@@](O)(CO)CC2)cc1 ZINC000217838994 CD In-Stock Unstable L3MBTL3 49 35 COc1cc(-n2cccn2)ccc1B(O)O ZINC000217839001 BB For-Sale Unstable AMP1_PLAFQ 46 35 NC(=O)CC[C@@H](NC(=O)[C@@H]1C[C@@H]2CCCC[C@@H]2N1)C(=O)O ZINC000217839037 CB For-Sale Unstable SLC5A1 20 46 COc1ccc(OCC(=O)NCc2ccc(OC(C)C)c(OC)c2)cc1 ZINC000217839038 FG In-Stock Unstable TRPV1 42 43 COc1ccc(OCC(=O)NCc2ccc(OC(C)C)c(OC)c2)cc1 ZINC000217839038 FG In-Stock Unstable MTNR1A 53 38 COc1ccc(OCC(=O)NCc2ccc(OC(C)C)c(OC)c2)cc1 ZINC000217839038 FG In-Stock Unstable MTNR1B 45 41 COc1ccc(OCC(=O)NCc2ccc(OC(C)C)c(OC)c2)cc1 ZINC000217839038 FG In-Stock Unstable PDE6A 42 32 COc1ccc(OCC(=O)NCc2ccc(OC(C)C)c(OC)c2)cc1 ZINC000217839038 FG In-Stock Unstable MT-ND1 26 45 COc1ccc(OCC(=O)NCc2ccc(OC(C)C)c(OC)c2)cc1 ZINC000217839038 FG In-Stock Unstable CA9 15 41 COc1ccc(OCC(=O)NCc2ccc(OC(C)C)c(OC)c2)cc1 ZINC000217839038 FG In-Stock Unstable ENPP1 40 30 COc1ccc(OCC(=O)NCc2ccc(OC(C)C)c(OC)c2)cc1 ZINC000217839038 FG In-Stock Unstable N1L 0 40 COc1ccc(OCC(=O)NCc2ccc(OC(C)C)c(OC)c2)cc1 ZINC000217839038 FG In-Stock Unstable DRTS_TRYCR 48 33 C[C@@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1ccc2c(c1)OCCO2 ZINC000217839042 CC On-Demand Unstable KCNQ2 21 40 CSc1ccc(C(=O)N2CCC[C@](O)(CO)CC2)cc1 ZINC000217839061 CD In-Stock Unstable L3MBTL3 49 35 C[C@H]1COCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217839064 CD On-Demand Unstable HRH3 21 42 O=C(CSc1nc2ccccc2o1)NC[C@H]1CCCN1c1ccccc1 ZINC000217839108 FH For-Sale Unstable HCRTR1 18 48 O=C(CSc1nc2ccccc2o1)NC[C@H]1CCCN1c1ccccc1 ZINC000217839108 FH For-Sale Unstable HCRTR2 17 48 CCOc1cc(Br)cc(O)c1OC ZINC000217839118 BF In-Stock Unstable TUBB1 23 50 CCOc1cc(Br)cc(O)c1OC ZINC000217839118 BF In-Stock Unstable METG 15 40 NC(=O)CC[C@H](NC(=O)[C@@H]1C[C@@H]2CCCC[C@@H]2N1)C(=O)O ZINC000217839121 CB For-Sale Unstable SLC5A1 20 46 C[C@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1ccc2c(c1)OCCO2 ZINC000217839122 CC In-Stock Unstable KCNQ2 21 40 C[C@H]1C[C@H](C)CCN1[C@@H]1CCCc2cc(O)ccc21 ZINC000217839128 CH For-Sale Unstable DRD5 15 43 C[C@H]1C[C@H](C)CCN1[C@@H]1CCCc2cc(O)ccc21 ZINC000217839128 CH For-Sale Unstable HSD17B1 56 36 COc1ccc(OCC(=O)NCCCc2ccccc2Cl)cc1 ZINC000217839154 EG In-Stock Unstable NQO2 21 40 COc1ccc(OCC(=O)NCCCc2ccccc2Cl)cc1 ZINC000217839154 EG In-Stock Unstable CYSP_TRYCR 0 40 COc1ccc(OCC(=O)NCCCc2ccccc2Cl)cc1 ZINC000217839154 EG In-Stock Unstable MMP16 0 40 COc1ccc(OCC(=O)NCCCc2ccccc2Cl)cc1 ZINC000217839154 EG In-Stock Unstable MTNR1A 97 48 COc1ccc(OCC(=O)NCCCc2ccccc2Cl)cc1 ZINC000217839154 EG In-Stock Unstable MTNR1B 75 44 COc1ccc(OCC(=O)NCCCc2ccccc2Cl)cc1 ZINC000217839154 EG In-Stock Unstable PLA2G4B 42 31 COc1ccc(OCC(=O)NCCCc2ccccc2Cl)cc1 ZINC000217839154 EG In-Stock Unstable NCE103 17 41 COc1ccc(OCC(=O)NCCCc2ccccc2Cl)cc1 ZINC000217839154 EG In-Stock Unstable FFAR4 28 40 COc1ccc(OCC(=O)NCCCc2ccccc2Cl)cc1 ZINC000217839154 EG In-Stock Unstable CRTM 42 39 COc1ccc(OCC(=O)NCCCc2ccccc2Cl)cc1 ZINC000217839154 EG In-Stock Unstable CAN2 0 41 COc1ccc(OCC(=O)NCCCc2ccccc2Cl)cc1 ZINC000217839154 EG In-Stock Unstable ISPD 0 40 Cc1cc(C)c(C(=O)Nc2ccc(Sc3nccn3C)cc2)c(C)c1 ZINC000217839167 FJ On-Demand Unstable GCK 17 42 OCCN(Cc1cccnc1)CC(F)(F)F ZINC000217839177 BD On-Demand Unstable NR1D1 46 38 O=C(CSc1nc2ccccc2o1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217839194 FH For-Sale Unstable HCRTR1 18 48 O=C(CSc1nc2ccccc2o1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217839194 FH For-Sale Unstable HCRTR2 17 48 O=C(N/C=C/c1ccccc1Br)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217839197 JK For-Sale Unstable NMUR2 0 46 O=C(N/C=C/c1ccccc1Br)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217839197 JK For-Sale Unstable NMUR1 0 46 NC(=O)CC[C@@H](NC(=O)[C@H]1C[C@@H]2CCCC[C@@H]2N1)C(=O)O ZINC000217839209 CB For-Sale Unstable SLC5A1 20 46 COc1ccc(OCC(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217839226 EG In-Stock Unstable PTGS2 27 42 COc1ccc(OCC(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217839226 EG In-Stock Unstable SCNN1A 73 44 COc1ccc(OCC(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217839226 EG In-Stock Unstable BMP1 23 40 COc1ccc(OCC(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217839226 EG In-Stock Unstable KCNA5 0 41 COc1ccc(OCC(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217839226 EG In-Stock Unstable SCN2A 16 42 COc1ccc(OCC(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217839226 EG In-Stock Unstable MTNR1A 69 42 COc1ccc(OCC(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217839226 EG In-Stock Unstable MTNR1B 41 45 COc1ccc(OCC(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217839226 EG In-Stock Unstable CA9 20 46 COc1ccc(OCC(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217839226 EG In-Stock Unstable U38 0 43 COc1ccc(OCC(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217839226 EG In-Stock Unstable NCE103 22 40 COc1ccc(OCC(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217839226 EG In-Stock Unstable CRTM 46 48 COc1ccc(OCC(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217839226 EG In-Stock Unstable PROKR1 57 40 COc1ccc(OCC(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217839226 EG In-Stock Unstable TRAR 16 40 COc1ccc(OCC(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217839226 EG In-Stock Unstable CAN2 0 40 O=C(N[C@@H]1CCCc2ccccc21)[C@@H]1C[C@@H](O)CN1 ZINC000217839250 CC In-Stock Unstable XIAP 23 42 O=C(N[C@@H]1CCCc2ccccc21)[C@@H]1C[C@@H](O)CN1 ZINC000217839250 CC In-Stock Unstable BIRC3 29 43 O=C(N[C@@H]1CCCc2ccccc21)[C@@H]1C[C@@H](O)CN1 ZINC000217839250 CC In-Stock Unstable BIRC2 44 43 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(Br)cc1 ZINC000217839295 FH For-Sale Unstable DRD2 25 42 CN(Cc1ncc[nH]1)C(=O)c1ccc(CN2CCc3ccccc3C2)cc1 ZINC000217839305 FG In-Stock Unstable ABCG2 20 41 CN(Cc1ncc[nH]1)C(=O)c1ccc(CN2CCc3ccccc3C2)cc1 ZINC000217839305 FG In-Stock Unstable NOD1 35 45 CN(Cc1ncc[nH]1)C(=O)c1ccc(CN2CCc3ccccc3C2)cc1 ZINC000217839305 FG In-Stock Unstable NOD2 54 46 O=C(N[C@@H]1CCCc2ccccc21)[C@H]1C[C@@H](O)CN1 ZINC000217839322 CC In-Stock Unstable XIAP 23 42 O=C(N[C@@H]1CCCc2ccccc21)[C@H]1C[C@@H](O)CN1 ZINC000217839322 CC In-Stock Unstable BIRC3 29 43 O=C(N[C@@H]1CCCc2ccccc21)[C@H]1C[C@@H](O)CN1 ZINC000217839322 CC In-Stock Unstable BIRC2 44 43 CC(=O)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217839359 CD In-Stock Unstable BMP1 23 46 CC(=O)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217839359 CD In-Stock Unstable PA 19 40 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Br)cc1 ZINC000217839363 FH For-Sale Unstable DRD2 25 42 CC[C@@H](N)[C@@H](N1C[C@@H](C)Cc2ccccc21)C(F)(F)F ZINC000217839365 CG For-Sale Unstable TPP2 54 34 COc1ccc(OCC(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217839373 DF In-Stock Unstable SCNN1A 36 40 COc1ccc(OCC(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217839373 DF In-Stock Unstable HDAC8 16 48 COc1ccc(OCC(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217839373 DF In-Stock Unstable S1PR3 21 40 COc1ccc(OCC(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217839373 DF In-Stock Unstable MTNR1A 78 48 COc1ccc(OCC(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217839373 DF In-Stock Unstable MTNR1B 66 48 COc1ccc(OCC(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217839373 DF In-Stock Unstable FAAH 20 44 COc1ccc(OCC(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217839373 DF In-Stock Unstable CA9 17 46 COc1ccc(OCC(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217839373 DF In-Stock Unstable FFAR1 19 46 COc1ccc(OCC(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217839373 DF In-Stock Unstable LEF 42 35 COc1ccc(OCC(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217839373 DF In-Stock Unstable CRTM 43 40 COc1ccc(OCC(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217839373 DF In-Stock Unstable PROKR1 61 40 CC(=O)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217839435 CD In-Stock Unstable BMP1 23 46 CC(=O)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217839435 CD In-Stock Unstable PA 19 40 Fc1cc(F)c(F)c(OCc2cccc(Br)c2)c1F ZINC000217839439 EJ For-Sale Unstable MAOB 22 43 CC[C@H](N)[C@@H](N1C[C@@H](C)Cc2ccccc21)C(F)(F)F ZINC000217839443 CG For-Sale Unstable TPP2 54 34 Cc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c(C)c1 ZINC000217839470 DH For-Sale Unstable DRD2 30 41 Cc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c(C)c1 ZINC000217839470 DH For-Sale Unstable AVPR2 21 42 CC1(C(=O)N[C@@H]2CCCCNC2=O)CCCC1 ZINC000217839481 BD On-Demand Unstable MMP1 18 45 COc1ccc(OCC(=O)NCCCc2ccccc2OC)cc1 ZINC000217839490 EF In-Stock Unstable DRD2 21 41 COc1ccc(OCC(=O)NCCCc2ccccc2OC)cc1 ZINC000217839490 EF In-Stock Unstable NQO2 21 41 COc1ccc(OCC(=O)NCCCc2ccccc2OC)cc1 ZINC000217839490 EF In-Stock Unstable CYSP_TRYCR 23 41 COc1ccc(OCC(=O)NCCCc2ccccc2OC)cc1 ZINC000217839490 EF In-Stock Unstable HDAC8 15 45 COc1ccc(OCC(=O)NCCCc2ccccc2OC)cc1 ZINC000217839490 EF In-Stock Unstable MTNR1A 103 48 COc1ccc(OCC(=O)NCCCc2ccccc2OC)cc1 ZINC000217839490 EF In-Stock Unstable MTNR1B 88 54 COc1ccc(OCC(=O)NCCCc2ccccc2OC)cc1 ZINC000217839490 EF In-Stock Unstable PLA2G4B 48 33 COc1ccc(OCC(=O)NCCCc2ccccc2OC)cc1 ZINC000217839490 EF In-Stock Unstable ABCB1 0 41 COc1ccc(OCC(=O)NCCCc2ccccc2OC)cc1 ZINC000217839490 EF In-Stock Unstable CA9 17 40 COc1ccc(OCC(=O)NCCCc2ccccc2OC)cc1 ZINC000217839490 EF In-Stock Unstable CRTM 41 36 COc1ccc(OCC(=O)NCCCc2ccccc2OC)cc1 ZINC000217839490 EF In-Stock Unstable MBTPS1 41 40 CCC[C@@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217839505 CD For-Sale Unstable CTSC 24 41 CCC[C@@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217839505 CD For-Sale Unstable MAN1B1 52 33 Cc1cc(C)n(Cc2cccc(/C=C\C(=O)O)c2)c(=O)n1 ZINC000217839535 CE For-Sale Unstable HDAC8 45 43 Cc1cc(C)n(Cc2cccc(/C=C\C(=O)O)c2)c(=O)n1 ZINC000217839535 CE For-Sale Unstable HDAC1 17 43 Cc1cc(C)n(Cc2cccc(/C=C\C(=O)O)c2)c(=O)n1 ZINC000217839535 CE For-Sale Unstable HDAC6 34 43 CC[C@@H](N)[C@H](N1C[C@@H](C)Cc2ccccc21)C(F)(F)F ZINC000217839537 CG For-Sale Unstable TPP2 54 34 Cc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c(C)c1 ZINC000217839554 DH For-Sale Unstable DRD2 30 41 Cc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c(C)c1 ZINC000217839554 DH For-Sale Unstable AVPR2 21 42 CCOCC(=O)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217839555 ED In-Stock Unstable BMP1 17 43 CCC[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217839579 CD For-Sale Unstable CTSC 24 41 CCC[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217839579 CD For-Sale Unstable MAN1B1 52 33 Cn1ccnc1Sc1ccc(NC(=O)c2cc3cc(F)ccc3s2)cc1 ZINC000217839585 GK On-Demand Unstable GCK 0 44 COc1ccc(CCCNC(=O)COc2ccc(OC)cc2)cc1 ZINC000217839598 EF In-Stock Unstable ADRB1 17 41 COc1ccc(CCCNC(=O)COc2ccc(OC)cc2)cc1 ZINC000217839598 EF In-Stock Unstable SCNN1A 56 43 COc1ccc(CCCNC(=O)COc2ccc(OC)cc2)cc1 ZINC000217839598 EF In-Stock Unstable ADRB3 21 49 COc1ccc(CCCNC(=O)COc2ccc(OC)cc2)cc1 ZINC000217839598 EF In-Stock Unstable BMP1 35 41 COc1ccc(CCCNC(=O)COc2ccc(OC)cc2)cc1 ZINC000217839598 EF In-Stock Unstable MMP13 16 45 COc1ccc(CCCNC(=O)COc2ccc(OC)cc2)cc1 ZINC000217839598 EF In-Stock Unstable SCN2A 25 46 COc1ccc(CCCNC(=O)COc2ccc(OC)cc2)cc1 ZINC000217839598 EF In-Stock Unstable HDAC8 21 53 COc1ccc(CCCNC(=O)COc2ccc(OC)cc2)cc1 ZINC000217839598 EF In-Stock Unstable MTNR1A 94 45 COc1ccc(CCCNC(=O)COc2ccc(OC)cc2)cc1 ZINC000217839598 EF In-Stock Unstable MTNR1B 66 50 COc1ccc(CCCNC(=O)COc2ccc(OC)cc2)cc1 ZINC000217839598 EF In-Stock Unstable MMP3 19 40 COc1ccc(CCCNC(=O)COc2ccc(OC)cc2)cc1 ZINC000217839598 EF In-Stock Unstable PLA2G4B 67 38 COc1ccc(CCCNC(=O)COc2ccc(OC)cc2)cc1 ZINC000217839598 EF In-Stock Unstable FAAH 21 42 COc1ccc(CCCNC(=O)COc2ccc(OC)cc2)cc1 ZINC000217839598 EF In-Stock Unstable CA9 21 51 COc1ccc(CCCNC(=O)COc2ccc(OC)cc2)cc1 ZINC000217839598 EF In-Stock Unstable MMP1 26 42 COc1ccc(CCCNC(=O)COc2ccc(OC)cc2)cc1 ZINC000217839598 EF In-Stock Unstable FFAR4 24 40 COc1ccc(CCCNC(=O)COc2ccc(OC)cc2)cc1 ZINC000217839598 EF In-Stock Unstable CRTM 47 45 COc1ccc(CCCNC(=O)COc2ccc(OC)cc2)cc1 ZINC000217839598 EF In-Stock Unstable PROKR1 55 34 CC[C@H](N)[C@H](N1C[C@@H](C)Cc2ccccc21)C(F)(F)F ZINC000217839614 CG For-Sale Unstable TPP2 54 34 CCOCC(=O)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217839636 ED In-Stock Unstable BMP1 17 43 CCC[C@@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217839657 CD For-Sale Unstable CTSC 24 41 CCC[C@@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217839657 CD For-Sale Unstable MAN1B1 52 33 Cc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1C ZINC000217839665 DH For-Sale Unstable DRD2 35 40 Cc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1C ZINC000217839665 DH For-Sale Unstable DRD4 17 45 Cc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1C ZINC000217839665 DH For-Sale Unstable HCRTR1 17 41 Cc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1C ZINC000217839665 DH For-Sale Unstable MAPK14 26 44 Cc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1C ZINC000217839665 DH For-Sale Unstable PREP 16 41 Cc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1C ZINC000217839665 DH For-Sale Unstable CACNA1I 50 35 Cc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1C ZINC000217839665 DH For-Sale Unstable ACKR3 60 39 COc1ccc2[nH]cc(CCNC(=O)Cn3ccc4c(NC(C)=O)cccc43)c2c1 ZINC000217839721 HG In-Stock Unstable ACHE 24 41 COc1ccc2[nH]cc(CCNC(=O)Cn3ccc4c(NC(C)=O)cccc43)c2c1 ZINC000217839721 HG In-Stock Unstable HTR1D 31 42 COc1ccc2[nH]cc(CCNC(=O)Cn3ccc4c(NC(C)=O)cccc43)c2c1 ZINC000217839721 HG In-Stock Unstable HTR1B 30 42 COc1ccc2[nH]cc(CCNC(=O)Cn3ccc4c(NC(C)=O)cccc43)c2c1 ZINC000217839721 HG In-Stock Unstable NQO2 40 46 COc1ccc2[nH]cc(CCNC(=O)Cn3ccc4c(NC(C)=O)cccc43)c2c1 ZINC000217839721 HG In-Stock Unstable MTNR1A 125 61 COc1ccc2[nH]cc(CCNC(=O)Cn3ccc4c(NC(C)=O)cccc43)c2c1 ZINC000217839721 HG In-Stock Unstable MTNR1B 101 61 COc1ccc2[nH]cc(CCNC(=O)Cn3ccc4c(NC(C)=O)cccc43)c2c1 ZINC000217839721 HG In-Stock Unstable ABCG2 26 42 O=C(c1ccc2c(c1)OCO2)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217839722 GE In-Stock Unstable SSTR3 62 35 COc1ccc(OCC(=O)N[C@@H](C)COc2ccc(OC)cc2)cc1 ZINC000217839727 EF In-Stock Unstable SDH1 0 43 COc1ccc(OCC(=O)N[C@@H](C)COc2ccc(OC)cc2)cc1 ZINC000217839727 EF In-Stock Unstable ACACA 34 40 COc1ccc(OCC(=O)N[C@@H](C)COc2ccc(OC)cc2)cc1 ZINC000217839727 EF In-Stock Unstable ACACB 19 40 COc1ccc(OCC(=O)N[C@@H](C)COc2ccc(OC)cc2)cc1 ZINC000217839727 EF In-Stock Unstable DXR 25 45 O=C(N[C@@H]1CCc2ccccc21)[C@H]1CCCC[C@H]1C(=O)O ZINC000217839740 CF On-Demand Unstable P2RX7 20 40 O=C(N[C@@H]1CCc2ccccc21)[C@H]1CCCC[C@H]1C(=O)O ZINC000217839740 CF On-Demand Unstable XIAP 21 44 O=C(N[C@@H]1CCc2ccccc21)[C@H]1CCCC[C@H]1C(=O)O ZINC000217839740 CF On-Demand Unstable BIRC3 34 40 O=C(N[C@@H]1CCc2ccccc21)[C@H]1CCCC[C@H]1C(=O)O ZINC000217839740 CF On-Demand Unstable BIRC2 27 40 CCC[C@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217839751 CD For-Sale Unstable CTSC 24 41 CCC[C@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217839751 CD For-Sale Unstable MAN1B1 52 33 Cc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1C ZINC000217839759 DH For-Sale Unstable DRD2 35 40 Cc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1C ZINC000217839759 DH For-Sale Unstable DRD4 17 45 Cc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1C ZINC000217839759 DH For-Sale Unstable HCRTR1 17 41 Cc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1C ZINC000217839759 DH For-Sale Unstable MAPK14 26 44 Cc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1C ZINC000217839759 DH For-Sale Unstable PREP 16 41 Cc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1C ZINC000217839759 DH For-Sale Unstable CACNA1I 50 35 Cc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1C ZINC000217839759 DH For-Sale Unstable ACKR3 60 39 COc1ccc(OCC(=O)N[C@H](C)COc2ccc(OC)cc2)cc1 ZINC000217839786 EF In-Stock Unstable SDH1 0 43 COc1ccc(OCC(=O)N[C@H](C)COc2ccc(OC)cc2)cc1 ZINC000217839786 EF In-Stock Unstable ACACA 34 40 COc1ccc(OCC(=O)N[C@H](C)COc2ccc(OC)cc2)cc1 ZINC000217839786 EF In-Stock Unstable ACACB 19 40 COc1ccc(OCC(=O)N[C@H](C)COc2ccc(OC)cc2)cc1 ZINC000217839786 EF In-Stock Unstable DXR 25 45 O=C(c1ccc2c(c1)OCO2)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217839796 GE In-Stock Unstable SSTR3 62 35 O=C(O)/C=C\c1ccc(OCCN2C(=O)CCC2=O)cc1 ZINC000217839797 CD For-Sale Unstable 17HSDCL 0 43 O=C(O)[C@@H]1CCCC[C@H]1C(=O)N[C@@H]1CCc2ccccc21 ZINC000217839807 CF For-Sale Unstable P2RX7 20 40 O=C(O)[C@@H]1CCCC[C@H]1C(=O)N[C@@H]1CCc2ccccc21 ZINC000217839807 CF For-Sale Unstable XIAP 21 44 O=C(O)[C@@H]1CCCC[C@H]1C(=O)N[C@@H]1CCc2ccccc21 ZINC000217839807 CF For-Sale Unstable BIRC3 34 40 O=C(O)[C@@H]1CCCC[C@H]1C(=O)N[C@@H]1CCc2ccccc21 ZINC000217839807 CF For-Sale Unstable BIRC2 27 40 Cn1ccnc1Sc1ccc(NC(=O)c2ccc(=O)n(Cc3ccccc3Cl)c2)cc1 ZINC000217839849 JJ On-Demand Unstable NOD2 40 37 O=C(N/C=C/c1ccccc1Br)N1CCCc2ccccc21 ZINC000217839853 FJ For-Sale Unstable AVPR2 36 45 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(I)cc1 ZINC000217839855 HH For-Sale Unstable PREP 15 43 COC(=O)C[C@H](c1ccc(O)cc1)c1c(O)c2ccccc2oc1=O ZINC000217839865 EF In-Stock Unstable CYP2C9 17 40 COC(=O)C[C@H](c1ccc(O)cc1)c1c(O)c2ccccc2oc1=O ZINC000217839865 EF In-Stock Unstable NQO1 61 56 COc1ccc(OCC(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217839872 FH In-Stock Unstable ADORA2B 28 42 COc1ccc(OCC(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217839872 FH In-Stock Unstable BDKRB1 0 43 COc1ccc(OCC(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217839872 FH In-Stock Unstable HDAC8 19 43 COc1ccc(OCC(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217839872 FH In-Stock Unstable PPARD 0 43 COc1ccc(OCC(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217839872 FH In-Stock Unstable PLA2G4B 49 33 COc1ccc(OCC(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217839872 FH In-Stock Unstable ABCB1 0 40 COc1ccc(OCC(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217839872 FH In-Stock Unstable MAPK10 0 42 COc1ccc(OCC(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217839872 FH In-Stock Unstable TUBB2B 26 40 COc1ccc(OCC(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217839872 FH In-Stock Unstable HCAR2 30 49 COc1ccc(OCC(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217839872 FH In-Stock Unstable LUCI_LUCLA 16 43 COc1ccc(OCC(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217839872 FH In-Stock Unstable YOPH 0 40 COc1ccc(OCC(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217839872 FH In-Stock Unstable AKR1C2 57 46 COc1ccc(OCC(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217839872 FH In-Stock Unstable ISPD 0 48 COc1ccc(OCC(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217839872 FH In-Stock Unstable FAS 42 44 COc1ccc(OCC(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217839872 FH In-Stock Unstable ADIPOR1 0 40 COc1ccc(OCC(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217839872 FH In-Stock Unstable ADIPOR2 0 40 COc1ccc(/C=C\C(=O)O)cc1CN1C(=O)CCC1=O ZINC000217839905 CD For-Sale Unstable PTGER2 0 41 COc1ccc(/C=C\C(=O)O)cc1CN1C(=O)CCC1=O ZINC000217839905 CD For-Sale Unstable AKR1C3 22 41 CCCN(CC)CCNC(=O)CCCC(=O)O ZINC000217839919 BD For-Sale Unstable DNM1 0 49 O=C(c1ccccc1C(F)(F)F)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217839920 HH In-Stock Unstable P2RX7 23 41 O=C(c1ccccc1C(F)(F)F)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217839920 HH In-Stock Unstable RBP4 28 40 CN1CCO[C@H]([C@@H](O)C[C@@H]2CCCc3ccccc32)C1 ZINC000217839946 CE For-Sale Unstable EBP 19 40 COC(=O)C[C@@H](c1ccc(O)cc1)c1c(O)c2ccccc2oc1=O ZINC000217839951 EF In-Stock Unstable CYP2C9 17 40 COC(=O)C[C@@H](c1ccc(O)cc1)c1c(O)c2ccccc2oc1=O ZINC000217839951 EF In-Stock Unstable NQO1 61 56 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(I)cc1 ZINC000217839952 HH For-Sale Unstable PREP 15 43 Cc1nc2ccccc2cc1C(=O)Nc1ccc(Sc2nccn2C)cc1 ZINC000217839969 FJ On-Demand Unstable GCK 17 44 COc1ccc(OCC(=O)NCCCc2cccc(OC(C)C)c2)cc1 ZINC000217839971 FH In-Stock Unstable HRH2 30 41 COc1ccc(OCC(=O)NCCCc2cccc(OC(C)C)c2)cc1 ZINC000217839971 FH In-Stock Unstable PTAFR 23 40 COc1ccc(OCC(=O)NCCCc2cccc(OC(C)C)c2)cc1 ZINC000217839971 FH In-Stock Unstable NQO2 18 42 COc1ccc(OCC(=O)NCCCc2cccc(OC(C)C)c2)cc1 ZINC000217839971 FH In-Stock Unstable FDFT1 24 49 COc1ccc(OCC(=O)NCCCc2cccc(OC(C)C)c2)cc1 ZINC000217839971 FH In-Stock Unstable SCN2A 15 40 COc1ccc(OCC(=O)NCCCc2cccc(OC(C)C)c2)cc1 ZINC000217839971 FH In-Stock Unstable HDAC8 20 46 COc1ccc(OCC(=O)NCCCc2cccc(OC(C)C)c2)cc1 ZINC000217839971 FH In-Stock Unstable MTNR1A 98 52 COc1ccc(OCC(=O)NCCCc2cccc(OC(C)C)c2)cc1 ZINC000217839971 FH In-Stock Unstable MTNR1B 77 44 COc1ccc(OCC(=O)NCCCc2cccc(OC(C)C)c2)cc1 ZINC000217839971 FH In-Stock Unstable AMP1_PLAFQ 20 42 COc1ccc(OCC(=O)NCCCc2cccc(OC(C)C)c2)cc1 ZINC000217839971 FH In-Stock Unstable CRTM 79 49 COc1ccc(OCC(=O)NCCCc2cccc(OC(C)C)c2)cc1 ZINC000217839971 FH In-Stock Unstable CRTH2 0 47 COc1ccc(OCC(=O)NCCCc2cccc(OC(C)C)c2)cc1 ZINC000217839971 FH In-Stock Unstable PDS 40 37 O=C(N/C=C/c1ccccc1Br)NCCc1ccccc1 ZINC000217839972 EH For-Sale Unstable HDAC8 15 46 O=C(N/C=C/c1ccccc1Br)NCCc1ccccc1 ZINC000217839972 EH For-Sale Unstable CA5B 24 43 O=C(N/C=C/c1ccccc1Br)NCCc1ccccc1 ZINC000217839972 EH For-Sale Unstable CA5A 23 43 O=C(N/C=C/c1ccccc1Br)NCCc1ccccc1 ZINC000217839972 EH For-Sale Unstable AMP1_PLAFQ 31 42 C[C@H]1Cc2ccccc2N(C[C@@H](O)c2cccc(N)c2)C1 ZINC000217840004 CG For-Sale Unstable TPP2 50 30 O=C(c1ccccc1C(F)(F)F)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217840012 HH In-Stock Unstable P2RX7 23 41 O=C(c1ccccc1C(F)(F)F)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217840012 HH In-Stock Unstable RBP4 28 40 O=C(N/C=C/c1ccccc1Br)NC1CCCC1 ZINC000217840049 DH For-Sale Unstable EPHX2 21 45 COc1ccc(OCC(=O)NCCCc2ccc(OC(C)C)cc2)cc1 ZINC000217840084 FH In-Stock Unstable ADRB1 16 45 COc1ccc(OCC(=O)NCCCc2ccc(OC(C)C)cc2)cc1 ZINC000217840084 FH In-Stock Unstable ADRB3 16 45 COc1ccc(OCC(=O)NCCCc2ccc(OC(C)C)cc2)cc1 ZINC000217840084 FH In-Stock Unstable HDAC8 15 49 COc1ccc(OCC(=O)NCCCc2ccc(OC(C)C)cc2)cc1 ZINC000217840084 FH In-Stock Unstable MTNR1A 63 40 COc1ccc(OCC(=O)NCCCc2ccc(OC(C)C)cc2)cc1 ZINC000217840084 FH In-Stock Unstable MTNR1B 41 46 COc1ccc(OCC(=O)NCCCc2ccc(OC(C)C)cc2)cc1 ZINC000217840084 FH In-Stock Unstable PLA2G4B 43 33 COc1ccc(OCC(=O)NCCCc2ccc(OC(C)C)cc2)cc1 ZINC000217840084 FH In-Stock Unstable CA9 16 44 COc1ccc(OCC(=O)NCCCc2ccc(OC(C)C)cc2)cc1 ZINC000217840084 FH In-Stock Unstable CRTM 42 39 COc1ccc(OCC(=O)NCCCc2ccc(OC(C)C)cc2)cc1 ZINC000217840084 FH In-Stock Unstable PROKR1 43 31 C[C@@H]1Cc2ccccc2N(C[C@@H](O)c2cccc(N)c2)C1 ZINC000217840124 CG For-Sale Unstable TPP2 50 30 CN1C(=O)C(=O)N(Cc2ccccc2/C=C\C(=O)O)C1=O ZINC000217840170 CC For-Sale Unstable PTGER2 45 47 CN1C(=O)C(=O)N(Cc2ccccc2/C=C\C(=O)O)C1=O ZINC000217840170 CC For-Sale Unstable PTGER4 0 47 CN1C(=O)C(=O)N(Cc2ccccc2/C=C\C(=O)O)C1=O ZINC000217840170 CC For-Sale Unstable PTGER3 17 47 CCOc1ccc(CCCNC(=O)COc2ccc(OC)cc2)cc1 ZINC000217840184 EG In-Stock Unstable SCNN1A 39 40 CCOc1ccc(CCCNC(=O)COc2ccc(OC)cc2)cc1 ZINC000217840184 EG In-Stock Unstable SCN2A 29 46 CCOc1ccc(CCCNC(=O)COc2ccc(OC)cc2)cc1 ZINC000217840184 EG In-Stock Unstable HDAC8 16 49 CCOc1ccc(CCCNC(=O)COc2ccc(OC)cc2)cc1 ZINC000217840184 EG In-Stock Unstable S1PR3 19 40 CCOc1ccc(CCCNC(=O)COc2ccc(OC)cc2)cc1 ZINC000217840184 EG In-Stock Unstable MTNR1A 82 45 CCOc1ccc(CCCNC(=O)COc2ccc(OC)cc2)cc1 ZINC000217840184 EG In-Stock Unstable MTNR1B 61 45 CCOc1ccc(CCCNC(=O)COc2ccc(OC)cc2)cc1 ZINC000217840184 EG In-Stock Unstable PLA2G4B 71 36 CCOc1ccc(CCCNC(=O)COc2ccc(OC)cc2)cc1 ZINC000217840184 EG In-Stock Unstable CA9 21 47 CCOc1ccc(CCCNC(=O)COc2ccc(OC)cc2)cc1 ZINC000217840184 EG In-Stock Unstable CRTM 44 41 CCOc1ccc(CCCNC(=O)COc2ccc(OC)cc2)cc1 ZINC000217840184 EG In-Stock Unstable PROKR1 53 32 C[C@H]1Cc2ccccc2N(C[C@@H](O)c2ccccc2N)C1 ZINC000217840209 CG For-Sale Unstable TPP2 51 31 O=C(/C=C\c1ccccc1)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217840213 GG In-Stock Unstable BMP1 15 41 Cn1c(=O)c2c(ncn2CC(=O)NC[C@@H]2CCCN2c2ccccc2)n(C)c1=O ZINC000217840228 GC For-Sale Unstable ADORA2A 15 40 BrC[C@@H]1CC(c2cccs2)=NO1 ZINC000217840252 BF In-Stock Unstable LUCI_PHOPY 78 39 COc1ccc(CCNC(=O)N/C=C/c2ccccc2Br)cc1OC ZINC000217840262 HH For-Sale Unstable MTNR1A 15 40 COc1ccc(CCNC(=O)N/C=C/c2ccccc2Br)cc1OC ZINC000217840262 HH For-Sale Unstable MTNR1B 16 44 COc1ccc(CCNC(=O)N/C=C/c2ccccc2Br)cc1OC ZINC000217840262 HH For-Sale Unstable NCE103 16 45 COc1ccc(CCNC(=O)N/C=C/c2ccccc2Br)cc1OC ZINC000217840262 HH For-Sale Unstable ABCG2 16 43 O=C(Cl)Cc1ccc(OCc2ccc(F)cc2)cc1 ZINC000217840291 CH For-Sale Unstable MAOB 34 47 O=C(Cl)Cc1ccc(OCc2ccc(F)cc2)cc1 ZINC000217840291 CH For-Sale Unstable ACE2 16 44 O=C(Cl)Cc1ccc(OCc2ccc(F)cc2)cc1 ZINC000217840291 CH For-Sale Unstable ACR 17 43 O=C(Cl)Cc1ccc(OCc2ccc(F)cc2)cc1 ZINC000217840291 CH For-Sale Unstable FFAR1 47 52 O=C(Cl)Cc1ccc(OCc2ccc(F)cc2)cc1 ZINC000217840291 CH For-Sale Unstable ENPP2 47 42 O=C(Cl)Cc1ccc(OCc2ccc(F)cc2)cc1 ZINC000217840291 CH For-Sale Unstable FFAR4 50 46 CCCOc1ccccc1CCCNC(=O)COc1ccc(OC)cc1 ZINC000217840295 FH In-Stock Unstable MTNR1A 94 49 CCCOc1ccccc1CCCNC(=O)COc1ccc(OC)cc1 ZINC000217840295 FH In-Stock Unstable MTNR1B 74 51 CCCOc1ccccc1CCCNC(=O)COc1ccc(OC)cc1 ZINC000217840295 FH In-Stock Unstable PLA2G4B 76 35 CCCOc1ccccc1CCCNC(=O)COc1ccc(OC)cc1 ZINC000217840295 FH In-Stock Unstable ABCB1 0 40 C[C@@H]1Cc2ccccc2N(C[C@@H](O)c2ccccc2N)C1 ZINC000217840304 CG For-Sale Unstable TPP2 51 31 COc1cc(CN2CC[C@@H](C)C[C@@H]2C)ccc1O ZINC000217840311 BG For-Sale Unstable SHBG 19 45 COc1cc(CN2CC[C@@H](C)C[C@@H]2C)ccc1O ZINC000217840311 BG For-Sale Unstable CAN2 0 43 Cn1c(=O)c2c(ncn2CC(=O)NC[C@H]2CCCN2c2ccccc2)n(C)c1=O ZINC000217840325 GC For-Sale Unstable ADORA2A 15 40 BrC[C@H]1CC(c2cccs2)=NO1 ZINC000217840341 BF In-Stock Unstable LUCI_PHOPY 78 39 C[C@H]1Cc2ccccc2N(C[C@@H](O)c2ccc(N)cc2)C1 ZINC000217840384 CG For-Sale Unstable TPP2 51 31 COc1cc(CN2CC[C@H](C)C[C@@H]2C)ccc1O ZINC000217840396 BG For-Sale Unstable SHBG 19 45 COc1cc(CN2CC[C@H](C)C[C@@H]2C)ccc1O ZINC000217840396 BG For-Sale Unstable CAN2 0 43 COc1ccc(Cl)cc1NS(=O)(=O)[C@@H](C)CO ZINC000217840423 CD For-Sale Unstable CPT1A 44 31 COc1ccc(Cl)cc1NS(=O)(=O)[C@@H](C)CO ZINC000217840423 CD For-Sale Unstable QRFPR 15 44 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc2nccnc2c1 ZINC000217840429 EG For-Sale Unstable HCRTR1 20 42 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc2nccnc2c1 ZINC000217840429 EG For-Sale Unstable HCRTR2 16 42 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc2nccnc2c1 ZINC000217840429 EG For-Sale Unstable ACKR3 51 32 COc1ccc(CN[C@@H]2CCN(C)C2=O)cc1O ZINC000217840431 CC For-Sale Unstable CDK4 0 41 COc1ccc(OCC(=O)N[C@@H](C)COc2ccc(C)cc2)cc1 ZINC000217840432 EF In-Stock Unstable SDH1 0 40 COc1ccc(OCC(=O)N[C@@H](C)COc2ccc(C)cc2)cc1 ZINC000217840432 EF In-Stock Unstable DXR 28 41 C[C@@H]1Cc2ccccc2N(C[C@@H](O)c2ccc(N)cc2)C1 ZINC000217840460 CG For-Sale Unstable TPP2 51 31 COC(=O)C[C@H](c1ccc(OC)cc1OC)c1c(O)c2ccccc2oc1=O ZINC000217840471 GG In-Stock Unstable NQO1 52 54 Cc1ccc(C2=NO[C@@H](CBr)C2)cc1 ZINC000217840481 CF In-Stock Unstable LUCI_PHOPY 100 49 COc1ccc(OCC(=O)N[C@H](C)COc2ccc(C)cc2)cc1 ZINC000217840487 EF In-Stock Unstable SDH1 0 40 COc1ccc(OCC(=O)N[C@H](C)COc2ccc(C)cc2)cc1 ZINC000217840487 EF In-Stock Unstable DXR 28 41 COc1ccc(Cl)cc1NS(=O)(=O)[C@H](C)CO ZINC000217840490 CD For-Sale Unstable CPT1A 44 31 COc1ccc(Cl)cc1NS(=O)(=O)[C@H](C)CO ZINC000217840490 CD For-Sale Unstable QRFPR 15 44 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc2nccnc2c1 ZINC000217840504 EG For-Sale Unstable HCRTR1 20 42 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc2nccnc2c1 ZINC000217840504 EG For-Sale Unstable HCRTR2 16 42 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc2nccnc2c1 ZINC000217840504 EG For-Sale Unstable ACKR3 51 32 COc1ccc(CN[C@H]2CCN(C)C2=O)cc1O ZINC000217840505 CC For-Sale Unstable CDK4 0 41 O=C(COc1ccc(Cl)cc1Cl)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217840522 IH In-Stock Unstable PRCP 19 41 Cc1ccc(C2=NO[C@H](CBr)C2)cc1 ZINC000217840558 CF In-Stock Unstable LUCI_PHOPY 100 49 COC(=O)C[C@@H](c1ccc(OC)cc1OC)c1c(O)c2ccccc2oc1=O ZINC000217840572 GG In-Stock Unstable NQO1 46 42 O=C(COc1ccc(Cl)cc1Cl)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217840593 IH In-Stock Unstable PRCP 19 41 O=C(N/C=C/c1ccccc1Br)NCc1cccnc1 ZINC000217840597 EG For-Sale Unstable PTAFR 26 41 O=C(N/C=C/c1ccccc1Br)NCc1cccnc1 ZINC000217840597 EG For-Sale Unstable NAMPT 71 51 CCOc1cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc(OCC)c1OCC ZINC000217840598 HI For-Sale Unstable DRD2 36 42 CCOc1cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc(OCC)c1OCC ZINC000217840598 HI For-Sale Unstable DRD3 17 42 CCOc1cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc(OCC)c1OCC ZINC000217840598 HI For-Sale Unstable HCRTR1 19 41 CCOc1cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc(OCC)c1OCC ZINC000217840598 HI For-Sale Unstable SSTR5 47 36 CCOc1cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc(OCC)c1OCC ZINC000217840598 HI For-Sale Unstable CACNA1I 69 36 CCOc1cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc(OCC)c1OCC ZINC000217840598 HI For-Sale Unstable HCN1 53 36 CCOc1cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc(OCC)c1OCC ZINC000217840598 HI For-Sale Unstable HCN4 46 36 CCOc1cc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc(OCC)c1OCC ZINC000217840598 HI For-Sale Unstable ACKR3 70 37 COc1ccc(OCC(=O)N[C@@H](C)c2ccc(N3CCC(C)CC3)cc2)cc1 ZINC000217840605 GI In-Stock Unstable ACACA 52 44 COc1ccc(OCC(=O)N[C@@H](C)c2ccc(N3CCC(C)CC3)cc2)cc1 ZINC000217840605 GI In-Stock Unstable ACACB 28 44 CS[C@@H]1CCC[C@@H]1NC(=O)c1ccc(Br)c(Cl)c1 ZINC000217840641 EI For-Sale Unstable SSTR3 29 40 CCOc1cc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc(OCC)c1OCC ZINC000217840667 HI For-Sale Unstable DRD2 36 42 CCOc1cc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc(OCC)c1OCC ZINC000217840667 HI For-Sale Unstable DRD3 17 42 CCOc1cc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc(OCC)c1OCC ZINC000217840667 HI For-Sale Unstable HCRTR1 19 41 CCOc1cc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc(OCC)c1OCC ZINC000217840667 HI For-Sale Unstable SSTR5 47 36 CCOc1cc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc(OCC)c1OCC ZINC000217840667 HI For-Sale Unstable CACNA1I 69 36 CCOc1cc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc(OCC)c1OCC ZINC000217840667 HI For-Sale Unstable HCN1 53 36 CCOc1cc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc(OCC)c1OCC ZINC000217840667 HI For-Sale Unstable HCN4 46 36 CCOc1cc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc(OCC)c1OCC ZINC000217840667 HI For-Sale Unstable ACKR3 70 37 COc1ccc(OCC(=O)N[C@H](C)c2ccc(N3CCC(C)CC3)cc2)cc1 ZINC000217840673 GI In-Stock Unstable ACACA 52 44 COc1ccc(OCC(=O)N[C@H](C)c2ccc(N3CCC(C)CC3)cc2)cc1 ZINC000217840673 GI In-Stock Unstable ACACB 28 44 O=C(Nc1cccc2cccnc12)c1nn(-c2ccccc2)cc1O ZINC000217840684 EG On-Demand Anodyne TNKS 22 45 O=C(Nc1cccc2cccnc12)c1nn(-c2ccccc2)cc1O ZINC000217840684 EG On-Demand Anodyne EGLN1 0 41 CC(C)(Oc1ccc(Cl)cc1)C(=O)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217840696 IH In-Stock Unstable HRH3 15 40 COc1cccc(C2=NO[C@@H](CBr)C2)c1 ZINC000217840701 CF In-Stock Unstable LUCI_PHOPY 108 71 C[C@@H](COc1cccc(Br)c1)N=C=O ZINC000217840738 CF For-Sale Unstable PDS 48 43 COc1ccc(OCC(=O)N[C@@H](C)c2ccc(N3CCC[C@@H](C)C3)cc2)cc1 ZINC000217840741 GI In-Stock Unstable ACACA 45 42 COc1ccc(OCC(=O)N[C@@H](C)c2ccc(N3CCC[C@@H](C)C3)cc2)cc1 ZINC000217840741 GI In-Stock Unstable ACACB 25 42 COc1ccc(OCC(=O)N[C@@H](C)c2ccc(N3CCC[C@@H](C)C3)cc2)cc1 ZINC000217840741 GI In-Stock Unstable RORC 42 44 CS[C@H]1CCC[C@@H]1NC(=O)c1ccc(Br)c(Cl)c1 ZINC000217840752 EI For-Sale Unstable SSTR3 29 40 Cc1cccc(C)c1OCc1ccccc1/C=C\C(=O)O ZINC000217840753 CH For-Sale Unstable PTGER2 33 70 Cc1cccc(C)c1OCc1ccccc1/C=C\C(=O)O ZINC000217840753 CH For-Sale Unstable PTGER4 39 63 Cc1cccc(C)c1OCc1ccccc1/C=C\C(=O)O ZINC000217840753 CH For-Sale Unstable PTGER3 30 70 Cc1cccc(C)c1OCc1ccccc1/C=C\C(=O)O ZINC000217840753 CH For-Sale Unstable PTGDR 0 50 CN1CCO[C@@H]([C@@H](O)Cc2cccc(Br)c2)C1 ZINC000217840755 DD For-Sale Unstable VACHT_TETCF 0 44 COc1cccc(C2=NO[C@H](CBr)C2)c1 ZINC000217840758 CF In-Stock Unstable LUCI_PHOPY 108 71 CC(C)(Oc1ccc(Cl)cc1)C(=O)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217840777 IH In-Stock Unstable HRH3 15 40 CN1CC[C@@H](NCc2ccc(OCC(N)=O)cc2)C1=O ZINC000217840784 CB For-Sale Unstable LTA4H 21 40 CN1CC[C@@H](NCc2ccc(OCC(N)=O)cc2)C1=O ZINC000217840784 CB For-Sale Unstable HRH3 26 41 CC(C)C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217840798 BE For-Sale Unstable ACE 52 36 CC(C)C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217840798 BE For-Sale Unstable DPP4 15 42 CC(C)C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217840798 BE For-Sale Unstable PREP 30 41 CC(C)C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217840798 BE For-Sale Unstable MTNR1A 19 41 CC(C)C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217840798 BE For-Sale Unstable MTNR1B 25 42 CC(C)C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217840798 BE For-Sale Unstable XIAP 43 35 CC(C)C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217840798 BE For-Sale Unstable BIRC2 45 34 CS[C@@H]1CCC[C@H]1NC(=O)c1ccc(Br)c(Cl)c1 ZINC000217840815 EI For-Sale Unstable SSTR3 29 40 CN1CCO[C@H]([C@@H](O)Cc2cccc(Br)c2)C1 ZINC000217840823 DD For-Sale Unstable VACHT_TETCF 0 44 COc1ccc(OCC(=O)N[C@H](C)c2ccc(N3CCC[C@@H](C)C3)cc2)cc1 ZINC000217840825 GI In-Stock Unstable ACACA 45 42 COc1ccc(OCC(=O)N[C@H](C)c2ccc(N3CCC[C@@H](C)C3)cc2)cc1 ZINC000217840825 GI In-Stock Unstable ACACB 25 42 COc1ccc(OCC(=O)N[C@H](C)c2ccc(N3CCC[C@@H](C)C3)cc2)cc1 ZINC000217840825 GI In-Stock Unstable RORC 42 44 C[C@H](COc1cccc(Br)c1)N=C=O ZINC000217840828 CF For-Sale Unstable PDS 48 43 O=C(N/C=C/c1ccccc1Br)N1CCC(Cc2ccccc2)CC1 ZINC000217840839 GK For-Sale Unstable GRIN2B 80 50 O=C(N/C=C/c1ccccc1Br)N1CCC(Cc2ccccc2)CC1 ZINC000217840839 GK For-Sale Unstable SIGMAR1 21 44 O=C(N/C=C/c1ccccc1Br)N1CCC(Cc2ccccc2)CC1 ZINC000217840839 GK For-Sale Unstable CCR3 48 43 O=C(N/C=C/c1ccccc1Br)N1CCC(Cc2ccccc2)CC1 ZINC000217840839 GK For-Sale Unstable GPR183 0 40 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217840840 JE In-Stock Unstable MC5R 35 40 CC(C)C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217840863 BE For-Sale Unstable ACE 52 36 CC(C)C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217840863 BE For-Sale Unstable DPP4 15 42 CC(C)C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217840863 BE For-Sale Unstable PREP 30 41 CC(C)C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217840863 BE For-Sale Unstable MTNR1A 19 41 CC(C)C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217840863 BE For-Sale Unstable MTNR1B 25 42 CC(C)C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217840863 BE For-Sale Unstable XIAP 43 35 CC(C)C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217840863 BE For-Sale Unstable BIRC2 45 34 CC[C@@H](N)[C@H](c1ccsc1)N1C[C@@H](C)Cc2ccccc21 ZINC000217840865 DI For-Sale Unstable TPP2 43 31 CN1CC[C@H](NCc2ccc(OCC(N)=O)cc2)C1=O ZINC000217840867 CB For-Sale Unstable LTA4H 21 40 CN1CC[C@H](NCc2ccc(OCC(N)=O)cc2)C1=O ZINC000217840867 CB For-Sale Unstable HRH3 26 41 Cc1cccc(C)c1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217840868 CH For-Sale Unstable PTGER2 30 62 Cc1cccc(C)c1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217840868 CH For-Sale Unstable PTGER4 30 46 Cc1cccc(C)c1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217840868 CH For-Sale Unstable PTGER3 22 58 Cc1cccc(C)c1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217840868 CH For-Sale Unstable PTGDR 0 43 Cc1cccc(C)c1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217840868 CH For-Sale Unstable FFAR1 37 40 Cc1cccc(C)c1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217840868 CH For-Sale Unstable AKR1C3 35 47 Cc1cccc(C)c1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217840868 CH For-Sale Unstable AKR1B10 15 43 Cc1ccccc1OCC(=O)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217840885 GF In-Stock Unstable COLA 73 38 Cc1ccccc1OCC(=O)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217840885 GF In-Stock Unstable CPT1A 67 38 BrC[C@@H]1CC(c2cccnc2)=NO1 ZINC000217840892 BD In-Stock Unstable CYP2E1 48 35 BrC[C@@H]1CC(c2cccnc2)=NO1 ZINC000217840892 BD In-Stock Unstable CYP2A6 41 35 BrC[C@@H]1CC(c2cccnc2)=NO1 ZINC000217840892 BD In-Stock Unstable LUCI_PHOPY 75 40 CC[C@H](N)[C@H](c1ccsc1)N1C[C@@H](C)Cc2ccccc21 ZINC000217840900 DI For-Sale Unstable TPP2 43 31 CS[C@H]1CCC[C@H]1NC(=O)c1ccc(Br)c(Cl)c1 ZINC000217840904 EI For-Sale Unstable SSTR3 29 40 C[C@@H]1C(=O)NC(=O)CN1C(=O)/C=C\c1ccc(Br)cc1 ZINC000217840906 ED For-Sale Unstable GPR183 0 40 Cc1cccc(C)c1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217840907 CH For-Sale Unstable PTGER2 29 71 Cc1cccc(C)c1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217840907 CH For-Sale Unstable PTGER4 26 45 Cc1cccc(C)c1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217840907 CH For-Sale Unstable PTGER3 23 57 Cc1cccc(C)c1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217840907 CH For-Sale Unstable LTB4R 15 47 Cc1cccc(C)c1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217840907 CH For-Sale Unstable KCNA3 26 41 Cc1cccc(C)c1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217840907 CH For-Sale Unstable PTGDR 0 42 Cc1cccc(C)c1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217840907 CH For-Sale Unstable HCAR2 0 41 Cc1cccc(C)c1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217840907 CH For-Sale Unstable FFAR1 53 44 Cc1cccc(C)c1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217840907 CH For-Sale Unstable AKR1C3 38 47 COc1ccc(OCC(=O)N[C@@H]2CC(C)(C)Oc3ccc(C)cc32)cc1 ZINC000217840955 FH In-Stock Unstable TRAR 32 40 O=C(COc1cccnc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217840967 DE For-Sale Unstable CHRNA7 61 42 O=C(COc1cccnc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217840967 DE For-Sale Unstable COLA 84 40 O=C(COc1cccnc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217840967 DE For-Sale Unstable CPT1A 83 37 O=C(COc1cccnc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217840967 DE For-Sale Unstable ACHP_LYMST 24 40 O=C(COc1cccnc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217840967 DE For-Sale Unstable VCP 56 36 O=C(COc1cccnc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217840967 DE For-Sale Unstable NAMPT 15 44 BrC[C@H]1CC(c2cccnc2)=NO1 ZINC000217840978 BD In-Stock Unstable CYP2E1 48 35 BrC[C@H]1CC(c2cccnc2)=NO1 ZINC000217840978 BD In-Stock Unstable CYP2A6 41 35 BrC[C@H]1CC(c2cccnc2)=NO1 ZINC000217840978 BD In-Stock Unstable LUCI_PHOPY 75 40 Cc1ccccc1OCC(=O)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217840984 GF In-Stock Unstable COLA 73 38 Cc1ccccc1OCC(=O)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217840984 GF In-Stock Unstable CPT1A 67 38 CC[C@@H](N)[C@@H](c1ccsc1)N1C[C@@H](C)Cc2ccccc21 ZINC000217840986 DI For-Sale Unstable TPP2 43 31 C[C@H]1C(=O)NC(=O)CN1C(=O)/C=C\c1ccc(Br)cc1 ZINC000217840998 ED For-Sale Unstable GPR183 0 40 COc1ccc(OCC(=O)N[C@H]2CC(C)(C)Oc3ccc(C)cc32)cc1 ZINC000217841007 FH In-Stock Unstable TRAR 32 40 O=C(COc1cccnc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217841052 DE For-Sale Unstable CHRNA7 61 42 O=C(COc1cccnc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217841052 DE For-Sale Unstable COLA 84 40 O=C(COc1cccnc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217841052 DE For-Sale Unstable CPT1A 83 37 O=C(COc1cccnc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217841052 DE For-Sale Unstable ACHP_LYMST 24 40 O=C(COc1cccnc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217841052 DE For-Sale Unstable VCP 56 36 O=C(COc1cccnc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217841052 DE For-Sale Unstable NAMPT 15 44 Cc1cccc(OCc2ccccc2/C=C\C(=O)O)c1C ZINC000217841053 CH For-Sale Unstable PTGER2 30 57 Cc1cccc(OCc2ccccc2/C=C\C(=O)O)c1C ZINC000217841053 CH For-Sale Unstable PTGER4 43 53 Cc1cccc(OCc2ccccc2/C=C\C(=O)O)c1C ZINC000217841053 CH For-Sale Unstable PTGER3 32 57 Cc1cccc(OCc2ccccc2/C=C\C(=O)O)c1C ZINC000217841053 CH For-Sale Unstable PTGDR 0 47 CC[C@H](N)[C@@H](c1ccsc1)N1C[C@@H](C)Cc2ccccc21 ZINC000217841067 DI For-Sale Unstable TPP2 43 31 COc1ccc(CCNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217841071 GH For-Sale Unstable BMP1 38 41 COc1ccc(CCNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217841071 GH For-Sale Unstable MMP16 0 40 COc1ccc(CCNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217841071 GH For-Sale Unstable MTNR1A 61 45 COc1ccc(CCNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217841071 GH For-Sale Unstable MTNR1B 54 45 COc1ccc(CCNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217841071 GH For-Sale Unstable CA9 22 47 Clc1ccccc1C1=NO[C@@H](CBr)C1 ZINC000217841074 CG In-Stock Unstable LUCI_PHOPY 95 69 COc1ccc(OCC(=O)N[C@@H]2CC(C)(C)Oc3cc(C)ccc32)cc1 ZINC000217841103 FH In-Stock Unstable TRAR 36 40 O=C(COc1ccccc1F)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217841109 GF In-Stock Unstable COLA 68 37 O=C(COc1ccccc1F)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217841109 GF In-Stock Unstable CPT1A 62 37 Clc1ccccc1C1=NO[C@H](CBr)C1 ZINC000217841127 CG In-Stock Unstable LUCI_PHOPY 95 69 COc1ccc(O)c(CN2CC[C@@H](C)C[C@@H]2C)c1 ZINC000217841128 BG For-Sale Unstable EBP 41 37 Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1C ZINC000217841152 CH For-Sale Unstable PTGER2 28 50 Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1C ZINC000217841152 CH For-Sale Unstable PTGER1 24 42 Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1C ZINC000217841152 CH For-Sale Unstable PTGER4 38 45 Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1C ZINC000217841152 CH For-Sale Unstable PTGER3 26 46 Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1C ZINC000217841152 CH For-Sale Unstable LTB4R 24 40 Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1C ZINC000217841152 CH For-Sale Unstable PTGDR 0 40 Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1C ZINC000217841152 CH For-Sale Unstable AKR1C3 38 50 Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1C ZINC000217841152 CH For-Sale Unstable AKR1B10 19 41 O=C(Cc1cccc2ccccc12)NC[C@H]1CCCN1c1ccccc1 ZINC000217841157 EI For-Sale Unstable PREP 21 51 NC1(c2ccc(Br)cc2C(=O)O)CC1 ZINC000217841160 CE For-Sale Unstable RARA 42 32 NC1(c2ccc(Br)cc2C(=O)O)CC1 ZINC000217841160 CE For-Sale Unstable RXRG 43 37 NC1(c2ccc(Br)cc2C(=O)O)CC1 ZINC000217841160 CE For-Sale Unstable RXRB 45 37 NC1(c2ccc(Br)cc2C(=O)O)CC1 ZINC000217841160 CE For-Sale Unstable PRS 59 36 O=C(O)CCCCCCNC(=O)[C@@H]1C[C@@H]2CCCC[C@@H]2N1 ZINC000217841174 CE For-Sale Unstable EPHX2 16 40 COc1ccc(OCC(=O)N[C@H]2CC(C)(C)Oc3cc(C)ccc32)cc1 ZINC000217841183 FH In-Stock Unstable TRAR 36 40 O=C(COc1ccccc1F)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217841192 GF In-Stock Unstable COLA 68 37 O=C(COc1ccccc1F)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217841192 GF In-Stock Unstable CPT1A 62 37 COc1ccc(O)c(CN2CC[C@H](C)C[C@@H]2C)c1 ZINC000217841208 BG For-Sale Unstable EBP 41 37 O=C(Cc1cccc2ccccc12)NC[C@@H]1CCCN1c1ccccc1 ZINC000217841230 EI For-Sale Unstable PREP 21 51 O=C(O)CCCCCCNC(=O)[C@@H]1C[C@H]2CCCC[C@@H]2N1 ZINC000217841236 CE For-Sale Unstable EPHX2 16 40 Clc1cccc(C2=NO[C@@H](CBr)C2)c1 ZINC000217841252 CG In-Stock Unstable LUCI_PHOPY 99 69 COC(=O)C[C@H](c1cccnc1)c1oc(CN2CCOCC2)cc(=O)c1O ZINC000217841254 FD In-Stock Unstable CASR 42 40 COC(=O)C[C@H](c1cccnc1)c1oc(CN2CCOCC2)cc(=O)c1O ZINC000217841254 FD In-Stock Unstable KCNA5 44 39 COc1cc(N)cc(S(=O)(=O)c2ccccc2)c1 ZINC000217841257 CE For-Sale Unstable HTR6 19 46 NC1(c2ccc(C(=O)O)cc2Br)CC1 ZINC000217841265 CE For-Sale Unstable RARA 75 42 NC1(c2ccc(C(=O)O)cc2Br)CC1 ZINC000217841265 CE For-Sale Unstable RARG 91 42 NC1(c2ccc(C(=O)O)cc2Br)CC1 ZINC000217841265 CE For-Sale Unstable RXRG 66 43 NC1(c2ccc(C(=O)O)cc2Br)CC1 ZINC000217841265 CE For-Sale Unstable RARB 84 42 NC1(c2ccc(C(=O)O)cc2Br)CC1 ZINC000217841265 CE For-Sale Unstable RXRA 52 43 NC1(c2ccc(C(=O)O)cc2Br)CC1 ZINC000217841265 CE For-Sale Unstable RXRB 66 43 COc1ccc(OCC(=O)N[C@@H]2CC(C)(C)Oc3ccc(OC)cc32)cc1 ZINC000217841302 FH In-Stock Unstable TRAR 33 42 O=C(CSCc1ccccc1)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217841303 HG In-Stock Unstable COLA 41 37 Clc1cccc(C2=NO[C@H](CBr)C2)c1 ZINC000217841306 CG In-Stock Unstable LUCI_PHOPY 99 69 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(Br)c(C)c2)[C@@H](C)O)cc1 ZINC000217841311 IF On-Demand Unstable CA1 15 41 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(Br)c(C)c2)[C@@H](C)O)cc1 ZINC000217841311 IF On-Demand Unstable MMP13 42 50 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(Br)c(C)c2)[C@@H](C)O)cc1 ZINC000217841311 IF On-Demand Unstable CA14 16 40 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(Br)c(C)c2)[C@@H](C)O)cc1 ZINC000217841311 IF On-Demand Unstable MMP2 27 49 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(Br)c(C)c2)[C@@H](C)O)cc1 ZINC000217841311 IF On-Demand Unstable MMP9 15 44 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(Br)c(C)c2)[C@@H](C)O)cc1 ZINC000217841311 IF On-Demand Unstable MMP12 73 50 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(Br)c(C)c2)[C@@H](C)O)cc1 ZINC000217841311 IF On-Demand Unstable MMP7 23 50 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(Br)c(C)c2)[C@@H](C)O)cc1 ZINC000217841311 IF On-Demand Unstable ADAMTS4 57 37 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(Br)c(C)c2)[C@@H](C)O)cc1 ZINC000217841311 IF On-Demand Unstable LEF 59 42 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(Br)c(C)c2)[C@@H](C)O)cc1 ZINC000217841311 IF On-Demand Unstable IDO1 38 52 COC(=O)C[C@@H](c1cccnc1)c1oc(CN2CCOCC2)cc(=O)c1O ZINC000217841319 FD In-Stock Unstable CASR 42 40 COC(=O)C[C@@H](c1cccnc1)c1oc(CN2CCOCC2)cc(=O)c1O ZINC000217841319 FD In-Stock Unstable KCNA5 44 39 COc1cc(O)c(C)c(Br)c1OC ZINC000217841358 BE For-Sale Unstable TUBB1 48 38 O=C(N/C=C/c1ccccc1Br)NCc1ccc(Cl)cc1 ZINC000217841364 FJ For-Sale Unstable AMP1_PLAFQ 23 42 O=C(Cc1c[nH]c2ccccc12)NC[C@H]1CCCN1c1ccccc1 ZINC000217841373 EG For-Sale Unstable ACE 16 40 O=C(Cc1c[nH]c2ccccc12)NC[C@H]1CCCN1c1ccccc1 ZINC000217841373 EG For-Sale Unstable DRD2 22 42 O=C(Cc1c[nH]c2ccccc12)NC[C@H]1CCCN1c1ccccc1 ZINC000217841373 EG For-Sale Unstable HTR1D 44 40 O=C(Cc1c[nH]c2ccccc12)NC[C@H]1CCCN1c1ccccc1 ZINC000217841373 EG For-Sale Unstable HTR1B 35 40 O=C(Cc1c[nH]c2ccccc12)NC[C@H]1CCCN1c1ccccc1 ZINC000217841373 EG For-Sale Unstable SSTR2 38 42 O=C(Cc1c[nH]c2ccccc12)NC[C@H]1CCCN1c1ccccc1 ZINC000217841373 EG For-Sale Unstable DRD3 15 43 O=C(Cc1c[nH]c2ccccc12)NC[C@H]1CCCN1c1ccccc1 ZINC000217841373 EG For-Sale Unstable HTR4 15 40 O=C(Cc1c[nH]c2ccccc12)NC[C@H]1CCCN1c1ccccc1 ZINC000217841373 EG For-Sale Unstable EDNRA 44 42 O=C(Cc1c[nH]c2ccccc12)NC[C@H]1CCCN1c1ccccc1 ZINC000217841373 EG For-Sale Unstable TACR1 43 46 O=C(Cc1c[nH]c2ccccc12)NC[C@H]1CCCN1c1ccccc1 ZINC000217841373 EG For-Sale Unstable MC4R 44 42 O=C(Cc1c[nH]c2ccccc12)NC[C@H]1CCCN1c1ccccc1 ZINC000217841373 EG For-Sale Unstable TACR2 49 38 O=C(Cc1c[nH]c2ccccc12)NC[C@H]1CCCN1c1ccccc1 ZINC000217841373 EG For-Sale Unstable CCKAR 59 49 O=C(Cc1c[nH]c2ccccc12)NC[C@H]1CCCN1c1ccccc1 ZINC000217841373 EG For-Sale Unstable HTR6 16 40 O=C(Cc1c[nH]c2ccccc12)NC[C@H]1CCCN1c1ccccc1 ZINC000217841373 EG For-Sale Unstable BRS3 24 40 O=C(Cc1c[nH]c2ccccc12)NC[C@H]1CCCN1c1ccccc1 ZINC000217841373 EG For-Sale Unstable NMBR 60 37 O=C(Cc1c[nH]c2ccccc12)NC[C@H]1CCCN1c1ccccc1 ZINC000217841373 EG For-Sale Unstable MC3R 20 42 O=C(Cc1c[nH]c2ccccc12)NC[C@H]1CCCN1c1ccccc1 ZINC000217841373 EG For-Sale Unstable MC5R 32 43 O=C(Cc1c[nH]c2ccccc12)NC[C@H]1CCCN1c1ccccc1 ZINC000217841373 EG For-Sale Unstable MMP14 41 33 O=C(Cc1c[nH]c2ccccc12)NC[C@H]1CCCN1c1ccccc1 ZINC000217841373 EG For-Sale Unstable ECE1 47 39 O=C(Cc1c[nH]c2ccccc12)NC[C@H]1CCCN1c1ccccc1 ZINC000217841373 EG For-Sale Unstable SSTR3 30 42 O=C(Cc1c[nH]c2ccccc12)NC[C@H]1CCCN1c1ccccc1 ZINC000217841373 EG For-Sale Unstable CCKBR 73 40 O=C(Cc1c[nH]c2ccccc12)NC[C@H]1CCCN1c1ccccc1 ZINC000217841373 EG For-Sale Unstable GHSR 40 35 O=C(Cc1c[nH]c2ccccc12)NC[C@H]1CCCN1c1ccccc1 ZINC000217841373 EG For-Sale Unstable MC1R 22 42 O=C(Cc1c[nH]c2ccccc12)NC[C@H]1CCCN1c1ccccc1 ZINC000217841373 EG For-Sale Unstable C5AR1 56 33 COc1ccc(OCC(=O)N[C@H]2CC(C)(C)Oc3ccc(OC)cc32)cc1 ZINC000217841380 FH In-Stock Unstable TRAR 33 42 O=C(CSCc1ccccc1)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217841382 HG In-Stock Unstable COLA 41 37 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(Br)c(C)c2)[C@@H](C)O)cc1 ZINC000217841389 IF On-Demand Unstable CA1 15 41 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(Br)c(C)c2)[C@@H](C)O)cc1 ZINC000217841389 IF On-Demand Unstable MMP13 42 50 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(Br)c(C)c2)[C@@H](C)O)cc1 ZINC000217841389 IF On-Demand Unstable CA14 16 40 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(Br)c(C)c2)[C@@H](C)O)cc1 ZINC000217841389 IF On-Demand Unstable MMP2 27 49 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(Br)c(C)c2)[C@@H](C)O)cc1 ZINC000217841389 IF On-Demand Unstable MMP9 15 44 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(Br)c(C)c2)[C@@H](C)O)cc1 ZINC000217841389 IF On-Demand Unstable MMP12 73 50 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(Br)c(C)c2)[C@@H](C)O)cc1 ZINC000217841389 IF On-Demand Unstable MMP7 23 50 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(Br)c(C)c2)[C@@H](C)O)cc1 ZINC000217841389 IF On-Demand Unstable ADAMTS4 57 37 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(Br)c(C)c2)[C@@H](C)O)cc1 ZINC000217841389 IF On-Demand Unstable LEF 59 42 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(Br)c(C)c2)[C@@H](C)O)cc1 ZINC000217841389 IF On-Demand Unstable IDO1 38 52 O=C(Cc1c[nH]c2ccccc12)NC[C@@H]1CCCN1c1ccccc1 ZINC000217841411 EG For-Sale Unstable ACE 16 40 O=C(Cc1c[nH]c2ccccc12)NC[C@@H]1CCCN1c1ccccc1 ZINC000217841411 EG For-Sale Unstable DRD2 22 42 O=C(Cc1c[nH]c2ccccc12)NC[C@@H]1CCCN1c1ccccc1 ZINC000217841411 EG For-Sale Unstable HTR1D 44 40 O=C(Cc1c[nH]c2ccccc12)NC[C@@H]1CCCN1c1ccccc1 ZINC000217841411 EG For-Sale Unstable HTR1B 35 40 O=C(Cc1c[nH]c2ccccc12)NC[C@@H]1CCCN1c1ccccc1 ZINC000217841411 EG For-Sale Unstable SSTR2 38 42 O=C(Cc1c[nH]c2ccccc12)NC[C@@H]1CCCN1c1ccccc1 ZINC000217841411 EG For-Sale Unstable DRD3 15 43 O=C(Cc1c[nH]c2ccccc12)NC[C@@H]1CCCN1c1ccccc1 ZINC000217841411 EG For-Sale Unstable HTR4 15 40 O=C(Cc1c[nH]c2ccccc12)NC[C@@H]1CCCN1c1ccccc1 ZINC000217841411 EG For-Sale Unstable EDNRA 44 42 O=C(Cc1c[nH]c2ccccc12)NC[C@@H]1CCCN1c1ccccc1 ZINC000217841411 EG For-Sale Unstable TACR1 43 46 O=C(Cc1c[nH]c2ccccc12)NC[C@@H]1CCCN1c1ccccc1 ZINC000217841411 EG For-Sale Unstable MC4R 44 42 O=C(Cc1c[nH]c2ccccc12)NC[C@@H]1CCCN1c1ccccc1 ZINC000217841411 EG For-Sale Unstable TACR2 49 38 O=C(Cc1c[nH]c2ccccc12)NC[C@@H]1CCCN1c1ccccc1 ZINC000217841411 EG For-Sale Unstable CCKAR 59 49 O=C(Cc1c[nH]c2ccccc12)NC[C@@H]1CCCN1c1ccccc1 ZINC000217841411 EG For-Sale Unstable HTR6 16 40 O=C(Cc1c[nH]c2ccccc12)NC[C@@H]1CCCN1c1ccccc1 ZINC000217841411 EG For-Sale Unstable BRS3 24 40 O=C(Cc1c[nH]c2ccccc12)NC[C@@H]1CCCN1c1ccccc1 ZINC000217841411 EG For-Sale Unstable NMBR 60 37 O=C(Cc1c[nH]c2ccccc12)NC[C@@H]1CCCN1c1ccccc1 ZINC000217841411 EG For-Sale Unstable MC3R 20 42 O=C(Cc1c[nH]c2ccccc12)NC[C@@H]1CCCN1c1ccccc1 ZINC000217841411 EG For-Sale Unstable MC5R 32 43 O=C(Cc1c[nH]c2ccccc12)NC[C@@H]1CCCN1c1ccccc1 ZINC000217841411 EG For-Sale Unstable MMP14 41 33 O=C(Cc1c[nH]c2ccccc12)NC[C@@H]1CCCN1c1ccccc1 ZINC000217841411 EG For-Sale Unstable ECE1 47 39 O=C(Cc1c[nH]c2ccccc12)NC[C@@H]1CCCN1c1ccccc1 ZINC000217841411 EG For-Sale Unstable SSTR3 30 42 O=C(Cc1c[nH]c2ccccc12)NC[C@@H]1CCCN1c1ccccc1 ZINC000217841411 EG For-Sale Unstable CCKBR 73 40 O=C(Cc1c[nH]c2ccccc12)NC[C@@H]1CCCN1c1ccccc1 ZINC000217841411 EG For-Sale Unstable GHSR 40 35 O=C(Cc1c[nH]c2ccccc12)NC[C@@H]1CCCN1c1ccccc1 ZINC000217841411 EG For-Sale Unstable MC1R 22 42 O=C(Cc1c[nH]c2ccccc12)NC[C@@H]1CCCN1c1ccccc1 ZINC000217841411 EG For-Sale Unstable C5AR1 56 33 Fc1ccccc1C1=NO[C@@H](CBr)C1 ZINC000217841436 CF In-Stock Unstable MIF 17 44 Fc1ccccc1C1=NO[C@@H](CBr)C1 ZINC000217841436 CF In-Stock Unstable LUCI_PHOPY 96 69 COc1ccc(CCOc2cccc([C@H](CC(=O)N3CCOCC3)c3c(O)c(O)c(O)c4c(=O)cc(-c5ccccc5)oc34)c2)cc1 ZINC000217841437 KK In-Stock Unstable RORC 48 38 C[C@@H](NC(=O)N/C=C/c1ccccc1Br)c1ccccc1 ZINC000217841456 EI For-Sale Unstable KCNQ2 50 37 C[C@@H]1C(=O)NC(=O)CN1C(=O)/C=C\c1ccc(F)c(Cl)c1 ZINC000217841468 DD For-Sale Unstable ITGAL 15 40 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(Br)c(C)c2)[C@H](C)O)cc1 ZINC000217841476 IF On-Demand Unstable CA1 15 41 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(Br)c(C)c2)[C@H](C)O)cc1 ZINC000217841476 IF On-Demand Unstable MMP13 42 50 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(Br)c(C)c2)[C@H](C)O)cc1 ZINC000217841476 IF On-Demand Unstable CA14 16 40 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(Br)c(C)c2)[C@H](C)O)cc1 ZINC000217841476 IF On-Demand Unstable MMP2 27 49 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(Br)c(C)c2)[C@H](C)O)cc1 ZINC000217841476 IF On-Demand Unstable MMP9 15 44 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(Br)c(C)c2)[C@H](C)O)cc1 ZINC000217841476 IF On-Demand Unstable MMP12 73 50 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(Br)c(C)c2)[C@H](C)O)cc1 ZINC000217841476 IF On-Demand Unstable MMP7 23 50 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(Br)c(C)c2)[C@H](C)O)cc1 ZINC000217841476 IF On-Demand Unstable ADAMTS4 57 37 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(Br)c(C)c2)[C@H](C)O)cc1 ZINC000217841476 IF On-Demand Unstable LEF 59 42 Cc1ccc(S(=O)(=O)N[C@@H](C(=O)Nc2ccc(Br)c(C)c2)[C@H](C)O)cc1 ZINC000217841476 IF On-Demand Unstable IDO1 38 52 O=C(Cc1cccs1)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217841482 FF In-Stock Unstable ETHR 41 48 COc1ccc(OCC(=O)N[C@@H]2CC(C)(C)Oc3cc(OC)ccc32)cc1 ZINC000217841485 FH In-Stock Unstable TRPV1 0 48 COc1ccc(OCC(=O)N[C@@H]2CC(C)(C)Oc3cc(OC)ccc32)cc1 ZINC000217841485 FH In-Stock Unstable MTNR1A 47 34 COc1ccc(OCC(=O)N[C@@H]2CC(C)(C)Oc3cc(OC)ccc32)cc1 ZINC000217841485 FH In-Stock Unstable HIF1A 19 40 COc1ccc(OCC(=O)N[C@@H]2CC(C)(C)Oc3cc(OC)ccc32)cc1 ZINC000217841485 FH In-Stock Unstable TRAR 38 42 Fc1ccccc1C1=NO[C@H](CBr)C1 ZINC000217841495 CF In-Stock Unstable MIF 17 44 Fc1ccccc1C1=NO[C@H](CBr)C1 ZINC000217841495 CF In-Stock Unstable LUCI_PHOPY 96 69 COc1ccc(CCOc2cccc([C@@H](CC(=O)N3CCOCC3)c3c(O)c(O)c(O)c4c(=O)cc(-c5ccccc5)oc34)c2)cc1 ZINC000217841507 KK In-Stock Unstable RORC 48 38 O=C(O)/C=C\c1ccccc1CN1CCCCCCC1 ZINC000217841545 CH For-Sale Unstable SLC6A1 87 42 O=C(O)/C=C\c1ccccc1CN1CCCCCCC1 ZINC000217841545 CH For-Sale Unstable PTGER2 48 51 O=C(O)/C=C\c1ccccc1CN1CCCCCCC1 ZINC000217841545 CH For-Sale Unstable PTGER4 25 51 O=C(O)/C=C\c1ccccc1CN1CCCCCCC1 ZINC000217841545 CH For-Sale Unstable FABP4 28 42 O=C(O)/C=C\c1ccccc1CN1CCCCCCC1 ZINC000217841545 CH For-Sale Unstable SIGMAR1 23 40 O=C(O)/C=C\c1ccccc1CN1CCCCCCC1 ZINC000217841545 CH For-Sale Unstable PTGER3 23 51 O=C(O)/C=C\c1ccccc1CN1CCCCCCC1 ZINC000217841545 CH For-Sale Unstable PTGDR 0 47 C[C@H](NC(=O)N/C=C/c1ccccc1Br)c1ccccc1 ZINC000217841549 EI For-Sale Unstable KCNQ2 50 37 C[C@H]1C(=O)NC(=O)CN1C(=O)/C=C\c1ccc(F)c(Cl)c1 ZINC000217841553 DD For-Sale Unstable ITGAL 15 40 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(Br)c(C)c2)[C@H](C)O)cc1 ZINC000217841554 IF On-Demand Unstable CA1 15 41 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(Br)c(C)c2)[C@H](C)O)cc1 ZINC000217841554 IF On-Demand Unstable MMP13 42 50 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(Br)c(C)c2)[C@H](C)O)cc1 ZINC000217841554 IF On-Demand Unstable CA14 16 40 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(Br)c(C)c2)[C@H](C)O)cc1 ZINC000217841554 IF On-Demand Unstable MMP2 27 49 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(Br)c(C)c2)[C@H](C)O)cc1 ZINC000217841554 IF On-Demand Unstable MMP9 15 44 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(Br)c(C)c2)[C@H](C)O)cc1 ZINC000217841554 IF On-Demand Unstable MMP12 73 50 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(Br)c(C)c2)[C@H](C)O)cc1 ZINC000217841554 IF On-Demand Unstable MMP7 23 50 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(Br)c(C)c2)[C@H](C)O)cc1 ZINC000217841554 IF On-Demand Unstable ADAMTS4 57 37 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(Br)c(C)c2)[C@H](C)O)cc1 ZINC000217841554 IF On-Demand Unstable LEF 59 42 Cc1ccc(S(=O)(=O)N[C@H](C(=O)Nc2ccc(Br)c(C)c2)[C@H](C)O)cc1 ZINC000217841554 IF On-Demand Unstable IDO1 38 52 CCOc1c(OC)ccc(Br)c1O ZINC000217841561 BF For-Sale Unstable TUBB1 22 43 COc1ccc(OCC(=O)N[C@H]2CC(C)(C)Oc3cc(OC)ccc32)cc1 ZINC000217841567 FH In-Stock Unstable TRPV1 0 48 COc1ccc(OCC(=O)N[C@H]2CC(C)(C)Oc3cc(OC)ccc32)cc1 ZINC000217841567 FH In-Stock Unstable MTNR1A 47 34 COc1ccc(OCC(=O)N[C@H]2CC(C)(C)Oc3cc(OC)ccc32)cc1 ZINC000217841567 FH In-Stock Unstable HIF1A 19 40 COc1ccc(OCC(=O)N[C@H]2CC(C)(C)Oc3cc(OC)ccc32)cc1 ZINC000217841567 FH In-Stock Unstable TRAR 38 42 O=C(Cc1cccs1)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217841572 FF In-Stock Unstable ETHR 41 48 C[C@@H](c1ccccc1Cl)N(C)C[C@@H](N)c1ccccc1 ZINC000217841574 CI For-Sale Unstable AOC3 30 46 Fc1cccc(C2=NO[C@@H](CBr)C2)c1 ZINC000217841592 CF In-Stock Unstable MIF 17 40 Fc1cccc(C2=NO[C@@H](CBr)C2)c1 ZINC000217841592 CF In-Stock Unstable LUCI_PHOPY 100 69 O=C(O)/C=C\c1ccc(CN2CCCCCCC2)cc1 ZINC000217841623 CH For-Sale Unstable HRH3 33 53 O=C(O)/C=C\c1ccc(CN2CCCCCCC2)cc1 ZINC000217841623 CH For-Sale Unstable SIGMAR1 38 48 O=C(O)/C=C\c1ccc(CN2CCCCCCC2)cc1 ZINC000217841623 CH For-Sale Unstable CXCR4 19 41 C[C@H](c1ccccc1Cl)N(C)C[C@@H](N)c1ccccc1 ZINC000217841639 CI For-Sale Unstable AOC3 30 46 COc1ccccc1CCN1C(=O)N[C@@H](CC(=O)NC[C@@H]2CCCN3CCCC[C@H]23)C1=O ZINC000217841648 ID In-Stock Unstable MBTPS1 53 36 Fc1cccc(C2=NO[C@H](CBr)C2)c1 ZINC000217841681 CF In-Stock Unstable MIF 17 40 Fc1cccc(C2=NO[C@H](CBr)C2)c1 ZINC000217841681 CF In-Stock Unstable LUCI_PHOPY 100 69 O=C(CCCc1ccccc1)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217841693 GG In-Stock Unstable COLA 49 36 O=C(CCCc1ccccc1)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217841693 GG In-Stock Unstable CPT1A 46 36 O=C(CCCc1ccccc1)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217841693 GG In-Stock Unstable PREP 58 42 O=C(CCCc1ccccc1)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217841693 GG In-Stock Unstable FAAH 45 41 O=C(CCCc1ccccc1)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217841693 GG In-Stock Unstable CES1 43 35 Cc1c(C(=O)NC[C@@H]2CCCN2c2ccccc2)cnn1-c1ccccc1 ZINC000217841697 FH For-Sale Unstable P2RY12 42 36 Cc1csc(CNC(=O)c2cc(N3CCCCC3)ccc2Cl)n1 ZINC000217841700 EI In-Stock Unstable P2RX7 0 43 CC[C@@H](NC(=O)COc1ccc(OC)cc1)c1ccc(C)c(C)c1 ZINC000217841704 EH In-Stock Unstable MTNR1A 40 38 CC[C@@H](NC(=O)COc1ccc(OC)cc1)c1ccc(C)c(C)c1 ZINC000217841704 EH In-Stock Unstable DXR 23 40 CCCN(CC)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217841740 CG For-Sale Unstable ACHE 0 43 CCCN(CC)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217841740 CG For-Sale Unstable PTGER2 0 41 CCCN(CC)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217841740 CG For-Sale Unstable TUBB1 47 38 CCCN(CC)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217841740 CG For-Sale Unstable AKR1C3 30 40 CCCN(CC)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217841740 CG For-Sale Unstable ABCG2 15 40 COc1cc(C)c(Br)c(O)c1OC ZINC000217841747 BE For-Sale Unstable TUBB1 41 35 COc1ccc(CNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217841751 FH For-Sale Unstable CA9 22 45 COc1ccc(CNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217841751 FH For-Sale Unstable KCNJ2 0 41 COc1ccc(CNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217841751 FH For-Sale Unstable GPR183 0 40 Cc1c(C(=O)NC[C@H]2CCCN2c2ccccc2)cnn1-c1ccccc1 ZINC000217841767 FH For-Sale Unstable P2RY12 42 36 CC[C@H](NC(=O)COc1ccc(OC)cc1)c1ccc(C)c(C)c1 ZINC000217841779 EH In-Stock Unstable MTNR1A 40 38 CC[C@H](NC(=O)COc1ccc(OC)cc1)c1ccc(C)c(C)c1 ZINC000217841779 EH In-Stock Unstable DXR 23 40 O=C(CCCc1ccccc1)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217841785 GG In-Stock Unstable COLA 49 36 O=C(CCCc1ccccc1)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217841785 GG In-Stock Unstable CPT1A 44 36 O=C(CCCc1ccccc1)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217841785 GG In-Stock Unstable PREP 53 42 O=C(CCCc1ccccc1)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217841785 GG In-Stock Unstable FAAH 38 41 O=C(CCCc1ccccc1)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217841785 GG In-Stock Unstable CES1 43 35 Fc1ccc(C2=NO[C@@H](CBr)C2)cc1 ZINC000217841809 CF In-Stock Unstable MIF 17 40 Fc1ccc(C2=NO[C@@H](CBr)C2)cc1 ZINC000217841809 CF In-Stock Unstable LUCI_PHOPY 106 64 CCCN(CC)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217841828 CG For-Sale Unstable ACHE 0 47 CCCN(CC)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217841828 CG For-Sale Unstable PTGER2 30 43 CCCN(CC)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217841828 CG For-Sale Unstable PTGER4 0 43 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841862 EG For-Sale Unstable HTR1A 21 49 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841862 EG For-Sale Unstable DRD2 56 49 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841862 EG For-Sale Unstable DRD4 41 32 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841862 EG For-Sale Unstable OXTR 26 40 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841862 EG For-Sale Unstable DRD3 41 46 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841862 EG For-Sale Unstable HTR3A 21 40 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841862 EG For-Sale Unstable HTR4 48 40 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841862 EG For-Sale Unstable SIGMAR1 15 45 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841862 EG For-Sale Unstable KCNA3 47 38 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841862 EG For-Sale Unstable MTNR1A 51 35 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841862 EG For-Sale Unstable MTNR1B 55 35 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841862 EG For-Sale Unstable CHRNA10 40 38 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841862 EG For-Sale Unstable MCHR1 22 60 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841862 EG For-Sale Unstable AKR1C2 45 33 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841862 EG For-Sale Unstable HCN1 67 36 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841862 EG For-Sale Unstable HCN4 50 35 COc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841862 EG For-Sale Unstable ACKR3 73 38 Fc1ccc(C2=NO[C@H](CBr)C2)cc1 ZINC000217841900 CF In-Stock Unstable MIF 17 40 Fc1ccc(C2=NO[C@H](CBr)C2)cc1 ZINC000217841900 CF In-Stock Unstable LUCI_PHOPY 106 64 COc1cc(Br)c(O)c(C)c1OC ZINC000217841921 BE For-Sale Unstable TUBB1 42 35 COc1ccc(CN(C)C2CCCC2)cc1/C=C\C(=O)O ZINC000217841930 CG For-Sale Unstable PTGER2 35 42 COc1ccc(CN(C)C2CCCC2)cc1/C=C\C(=O)O ZINC000217841930 CG For-Sale Unstable PTGER4 22 42 COc1ccc(CN(C)C2CCCC2)cc1/C=C\C(=O)O ZINC000217841930 CG For-Sale Unstable PTGER3 16 42 O=C(N/C=C/c1ccccc1Br)NCc1ccc2c(c1)OCO2 ZINC000217841941 GH For-Sale Unstable PDE5A 28 41 O=C(N/C=C/c1ccccc1Br)NCc1ccc2c(c1)OCO2 ZINC000217841941 GH For-Sale Unstable BMP1 44 39 O=C(N/C=C/c1ccccc1Br)NCc1ccc2c(c1)OCO2 ZINC000217841941 GH For-Sale Unstable SCN9A 23 43 O=C(N/C=C/c1ccccc1Br)NCc1ccc2c(c1)OCO2 ZINC000217841941 GH For-Sale Unstable NOS2 84 34 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841946 EG For-Sale Unstable HTR1A 21 49 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841946 EG For-Sale Unstable DRD2 56 49 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841946 EG For-Sale Unstable DRD4 41 32 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841946 EG For-Sale Unstable OXTR 26 40 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841946 EG For-Sale Unstable DRD3 41 46 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841946 EG For-Sale Unstable HTR3A 21 40 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841946 EG For-Sale Unstable HTR4 48 40 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841946 EG For-Sale Unstable SIGMAR1 15 45 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841946 EG For-Sale Unstable KCNA3 47 38 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841946 EG For-Sale Unstable MTNR1A 51 35 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841946 EG For-Sale Unstable MTNR1B 55 35 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841946 EG For-Sale Unstable CHRNA10 40 38 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841946 EG For-Sale Unstable MCHR1 22 60 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841946 EG For-Sale Unstable AKR1C2 45 33 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841946 EG For-Sale Unstable HCN1 67 36 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841946 EG For-Sale Unstable HCN4 50 35 COc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217841946 EG For-Sale Unstable ACKR3 73 38 O=C(NC[C@@H]1COCCO1)c1cccc(CN2CCCCCC2)c1 ZINC000217841998 EE In-Stock Unstable CHRM3 16 42 O=C(NC[C@@H]1COCCO1)c1cccc(CN2CCCCCC2)c1 ZINC000217841998 EE In-Stock Unstable BDKRB1 29 44 CCc1ccc(C2=NO[C@@H](CBr)C2)cc1 ZINC000217842003 CG In-Stock Unstable LUCI_PHOPY 102 49 COc1cc(C)c(O)c(Br)c1OC ZINC000217842024 BE For-Sale Unstable TUBB1 41 35 NS(=O)(=O)c1ccc(N[C@@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217842025 CD For-Sale Unstable CA2 35 43 NS(=O)(=O)c1ccc(N[C@@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217842025 CD For-Sale Unstable CA1 31 43 NS(=O)(=O)c1ccc(N[C@@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217842025 CD For-Sale Unstable CA7 23 41 NS(=O)(=O)c1ccc(N[C@@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217842025 CD For-Sale Unstable CA12 30 41 NS(=O)(=O)c1ccc(N[C@@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217842025 CD For-Sale Unstable CA9 30 41 NS(=O)(=O)c1ccc(N[C@@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217842025 CD For-Sale Unstable CAH_METTE 18 41 NS(=O)(=O)c1ccc(N[C@@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217842025 CD For-Sale Unstable MTCA1 41 36 NS(=O)(=O)c1ccc(N[C@@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217842025 CD For-Sale Unstable P96878_MYCTU 51 36 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217842039 GF For-Sale Unstable CA2 98 57 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217842039 GF For-Sale Unstable CA1 96 57 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217842039 GF For-Sale Unstable CA7 43 49 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217842039 GF For-Sale Unstable CA5B 55 49 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217842039 GF For-Sale Unstable CA4 70 57 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217842039 GF For-Sale Unstable CA5A 63 49 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217842039 GF For-Sale Unstable CA14 31 49 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217842039 GF For-Sale Unstable CA12 81 57 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217842039 GF For-Sale Unstable CA9 84 52 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217842039 GF For-Sale Unstable UREA_CANEN 27 40 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217842039 GF For-Sale Unstable NCE103 45 47 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217842039 GF For-Sale Unstable MTCA1 64 57 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217842039 GF For-Sale Unstable P96878_MYCTU 80 57 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc2ccccc2c1 ZINC000217842041 EI For-Sale Unstable DRD4 18 44 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc2ccccc2c1 ZINC000217842041 EI For-Sale Unstable DRD3 20 45 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc2ccccc2c1 ZINC000217842041 EI For-Sale Unstable HCRTR1 24 43 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc2ccccc2c1 ZINC000217842041 EI For-Sale Unstable PLD1 36 43 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc2ccccc2c1 ZINC000217842041 EI For-Sale Unstable PREP 19 40 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc2ccccc2c1 ZINC000217842041 EI For-Sale Unstable CAPN2 59 37 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc2ccccc2c1 ZINC000217842041 EI For-Sale Unstable PLD2 45 43 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc2ccccc2c1 ZINC000217842041 EI For-Sale Unstable HCRTR2 17 43 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc2ccccc2c1 ZINC000217842041 EI For-Sale Unstable MCHR1 15 48 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc2ccccc2c1 ZINC000217842041 EI For-Sale Unstable CACNA1I 48 34 CC[C@@H](NC(=O)COc1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217842053 FG In-Stock Unstable PLA2G4B 39 40 CC[C@@H](NC(=O)COc1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217842053 FG In-Stock Unstable DXR 25 43 CC[C@@H](NC(=O)COc1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217842053 FG In-Stock Unstable ENPP1 60 36 CCc1ccc(C2=NO[C@H](CBr)C2)cc1 ZINC000217842080 CG In-Stock Unstable LUCI_PHOPY 102 49 O=C(NC[C@H]1COCCO1)c1cccc(CN2CCCCCC2)c1 ZINC000217842083 EE In-Stock Unstable CHRM3 16 42 O=C(NC[C@H]1COCCO1)c1cccc(CN2CCCCCC2)c1 ZINC000217842083 EE In-Stock Unstable BDKRB1 29 44 O=C(c1ccc(Br)cc1CO)N1CCOCC1 ZINC000217842093 DD For-Sale Unstable AKR1C3 31 44 COc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)NCCc1c[nH]cn1)C(=O)OC2 ZINC000217842106 HF In-Stock Unstable IMPDH1 0 70 COc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)NCCc1c[nH]cn1)C(=O)OC2 ZINC000217842106 HF In-Stock Unstable HRH3 19 41 COc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)NCCc1c[nH]cn1)C(=O)OC2 ZINC000217842106 HF In-Stock Unstable IMPDH2 0 70 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc2ccccc2c1 ZINC000217842113 EI For-Sale Unstable DRD3 20 45 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc2ccccc2c1 ZINC000217842113 EI For-Sale Unstable HCRTR1 24 43 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc2ccccc2c1 ZINC000217842113 EI For-Sale Unstable PLD1 36 43 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc2ccccc2c1 ZINC000217842113 EI For-Sale Unstable PREP 19 40 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc2ccccc2c1 ZINC000217842113 EI For-Sale Unstable PLD2 45 43 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc2ccccc2c1 ZINC000217842113 EI For-Sale Unstable MCHR1 15 48 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc2ccccc2c1 ZINC000217842113 EI For-Sale Unstable CACNA1I 48 34 NS(=O)(=O)c1ccc(N[C@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217842115 CD For-Sale Unstable CA2 35 43 NS(=O)(=O)c1ccc(N[C@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217842115 CD For-Sale Unstable CA1 31 43 NS(=O)(=O)c1ccc(N[C@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217842115 CD For-Sale Unstable CA7 23 41 NS(=O)(=O)c1ccc(N[C@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217842115 CD For-Sale Unstable CA12 30 41 NS(=O)(=O)c1ccc(N[C@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217842115 CD For-Sale Unstable CA9 30 41 NS(=O)(=O)c1ccc(N[C@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217842115 CD For-Sale Unstable CAH_METTE 18 41 NS(=O)(=O)c1ccc(N[C@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217842115 CD For-Sale Unstable MTCA1 41 36 NS(=O)(=O)c1ccc(N[C@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217842115 CD For-Sale Unstable P96878_MYCTU 51 36 CC[C@H](NC(=O)COc1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217842128 FG In-Stock Unstable PLA2G4B 39 40 CC[C@H](NC(=O)COc1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217842128 FG In-Stock Unstable DXR 25 43 CC[C@H](NC(=O)COc1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217842128 FG In-Stock Unstable ENPP1 60 36 COc1cc(Br)c(C)c(O)c1OC ZINC000217842138 BE For-Sale Unstable TUBB1 41 35 C[C@@H](c1ccccc1Cl)N(C)C[C@@H](N)Cc1ccccc1 ZINC000217842147 DH For-Sale Unstable AOC3 18 44 COc1ccc(/C=C\C(=O)O)cc1CN(C)CC(C)C ZINC000217842174 CF For-Sale Unstable AKR1C3 41 43 O=C(N/C=C/c1ccccc1Br)NCc1ccccc1 ZINC000217842175 EH For-Sale Unstable ANPEP 26 43 O=C(N/C=C/c1ccccc1Br)NCc1ccccc1 ZINC000217842175 EH For-Sale Unstable CA5B 16 40 O=C(N/C=C/c1ccccc1Br)NCc1ccccc1 ZINC000217842175 EH For-Sale Unstable CA5A 19 40 O=C(N/C=C/c1ccccc1Br)NCc1ccccc1 ZINC000217842175 EH For-Sale Unstable AMP1_PLAFQ 42 39 BrC[C@@H]1CC(c2ccco2)=NO1 ZINC000217842179 BE In-Stock Unstable LUCI_PHOPY 82 40 COC(=O)c1ccccc1C(=O)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217842183 HE In-Stock Unstable BMP1 15 40 CO[C@@H]1C[C@H](C(=O)O)N(C(=O)C[C@@H](N)c2ccccc2)C1 ZINC000217842193 CC For-Sale Unstable ACE 43 48 CO[C@@H]1C[C@H](C(=O)O)N(C(=O)C[C@@H](N)c2ccccc2)C1 ZINC000217842193 CC For-Sale Unstable AGTR2 101 35 CC[C@H](NC(=O)[C@@H](NS(=O)(=O)c1ccc(C)cc1)[C@@H](C)O)c1ccc(Cl)cc1 ZINC000217842197 HF On-Demand Unstable MMP13 22 49 CC[C@H](NC(=O)[C@@H](NS(=O)(=O)c1ccc(C)cc1)[C@@H](C)O)c1ccc(Cl)cc1 ZINC000217842197 HF On-Demand Unstable MMP2 17 49 CC[C@H](NC(=O)[C@@H](NS(=O)(=O)c1ccc(C)cc1)[C@@H](C)O)c1ccc(Cl)cc1 ZINC000217842197 HF On-Demand Unstable MMP12 20 44 CC[C@H](NC(=O)[C@@H](NS(=O)(=O)c1ccc(C)cc1)[C@@H](C)O)c1ccc(Cl)cc1 ZINC000217842197 HF On-Demand Unstable MMP7 18 44 CC[C@H](NC(=O)[C@@H](NS(=O)(=O)c1ccc(C)cc1)[C@@H](C)O)c1ccc(Cl)cc1 ZINC000217842197 HF On-Demand Unstable ADAMTS4 50 36 CC[C@H](NC(=O)[C@@H](NS(=O)(=O)c1ccc(C)cc1)[C@@H](C)O)c1ccc(Cl)cc1 ZINC000217842197 HF On-Demand Unstable LEF 49 44 NS(=O)(=O)c1ccc(N[C@@H]2C[C@H]3CC=C[C@H]32)cc1 ZINC000217842199 CD For-Sale Unstable CA2 35 43 NS(=O)(=O)c1ccc(N[C@@H]2C[C@H]3CC=C[C@H]32)cc1 ZINC000217842199 CD For-Sale Unstable CA1 31 43 NS(=O)(=O)c1ccc(N[C@@H]2C[C@H]3CC=C[C@H]32)cc1 ZINC000217842199 CD For-Sale Unstable CA7 23 41 NS(=O)(=O)c1ccc(N[C@@H]2C[C@H]3CC=C[C@H]32)cc1 ZINC000217842199 CD For-Sale Unstable CA12 30 41 NS(=O)(=O)c1ccc(N[C@@H]2C[C@H]3CC=C[C@H]32)cc1 ZINC000217842199 CD For-Sale Unstable CA9 30 41 NS(=O)(=O)c1ccc(N[C@@H]2C[C@H]3CC=C[C@H]32)cc1 ZINC000217842199 CD For-Sale Unstable CAH_METTE 18 41 NS(=O)(=O)c1ccc(N[C@@H]2C[C@H]3CC=C[C@H]32)cc1 ZINC000217842199 CD For-Sale Unstable MTCA1 41 36 NS(=O)(=O)c1ccc(N[C@@H]2C[C@H]3CC=C[C@H]32)cc1 ZINC000217842199 CD For-Sale Unstable P96878_MYCTU 51 36 CO[C@H]1C[C@H](C(=O)O)N(C(=O)C[C@@H](N)c2ccccc2)C1 ZINC000217842230 CC For-Sale Unstable ACE 43 48 CO[C@H]1C[C@H](C(=O)O)N(C(=O)C[C@@H](N)c2ccccc2)C1 ZINC000217842230 CC For-Sale Unstable AGTR2 101 35 COC(=O)c1ccccc1C(=O)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217842245 HE In-Stock Unstable BMP1 15 40 C[C@H](c1ccccc1Cl)N(C)C[C@@H](N)Cc1ccccc1 ZINC000217842251 DH For-Sale Unstable AOC3 18 44 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc2ccccc2n1 ZINC000217842256 EH For-Sale Unstable SMO 41 39 CC[C@@H](NC(=O)COc1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217842259 GF In-Stock Unstable BMP1 45 40 CC[C@@H](NC(=O)COc1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217842259 GF In-Stock Unstable MMP13 41 43 CC[C@@H](NC(=O)COc1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217842259 GF In-Stock Unstable ADAM17 21 40 CC[C@@H](NC(=O)COc1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217842259 GF In-Stock Unstable MMP2 25 43 CC[C@@H](NC(=O)COc1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217842259 GF In-Stock Unstable MMP8 26 40 CC[C@@H](NC(=O)COc1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217842259 GF In-Stock Unstable MMP9 35 40 CC[C@@H](NC(=O)COc1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217842259 GF In-Stock Unstable MMP1 38 40 NS(=O)(=O)c1ccc(N[C@H]2C[C@H]3CC=C[C@@H]23)cc1 ZINC000217842268 CD For-Sale Unstable CA2 35 43 NS(=O)(=O)c1ccc(N[C@H]2C[C@H]3CC=C[C@@H]23)cc1 ZINC000217842268 CD For-Sale Unstable CA1 31 43 NS(=O)(=O)c1ccc(N[C@H]2C[C@H]3CC=C[C@@H]23)cc1 ZINC000217842268 CD For-Sale Unstable CA7 23 41 NS(=O)(=O)c1ccc(N[C@H]2C[C@H]3CC=C[C@@H]23)cc1 ZINC000217842268 CD For-Sale Unstable CA12 30 41 NS(=O)(=O)c1ccc(N[C@H]2C[C@H]3CC=C[C@@H]23)cc1 ZINC000217842268 CD For-Sale Unstable CA9 30 41 NS(=O)(=O)c1ccc(N[C@H]2C[C@H]3CC=C[C@@H]23)cc1 ZINC000217842268 CD For-Sale Unstable CAH_METTE 18 41 NS(=O)(=O)c1ccc(N[C@H]2C[C@H]3CC=C[C@@H]23)cc1 ZINC000217842268 CD For-Sale Unstable MTCA1 41 36 NS(=O)(=O)c1ccc(N[C@H]2C[C@H]3CC=C[C@@H]23)cc1 ZINC000217842268 CD For-Sale Unstable P96878_MYCTU 51 36 BrC[C@H]1CC(c2ccco2)=NO1 ZINC000217842277 BE In-Stock Unstable LUCI_PHOPY 82 40 COc1ccc(CN(C)CC(C)C)cc1/C=C\C(=O)O ZINC000217842286 CF For-Sale Unstable PTGER2 28 43 COc1ccc(CN(C)CC(C)C)cc1/C=C\C(=O)O ZINC000217842286 CF For-Sale Unstable PTGER4 0 43 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc2ccccc2n1 ZINC000217842308 EH For-Sale Unstable SMO 41 39 C[C@H]1Cc2ccccc2N([C@@H](c2ccccc2)[C@H](C)N)C1 ZINC000217842313 CH For-Sale Unstable TPP2 42 30 CC[C@H](NC(=O)COc1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217842325 GF In-Stock Unstable PTGS2 15 47 CC[C@H](NC(=O)COc1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217842325 GF In-Stock Unstable BMP1 45 40 CC[C@H](NC(=O)COc1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217842325 GF In-Stock Unstable MMP13 49 43 CC[C@H](NC(=O)COc1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217842325 GF In-Stock Unstable ADAM17 21 40 CC[C@H](NC(=O)COc1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217842325 GF In-Stock Unstable MMP2 33 43 CC[C@H](NC(=O)COc1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217842325 GF In-Stock Unstable MMP3 41 39 CC[C@H](NC(=O)COc1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217842325 GF In-Stock Unstable MMP8 33 40 CC[C@H](NC(=O)COc1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217842325 GF In-Stock Unstable MMP9 44 40 CC[C@H](NC(=O)COc1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217842325 GF In-Stock Unstable MMP12 28 40 CC[C@H](NC(=O)COc1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217842325 GF In-Stock Unstable MMP1 39 40 CO[C@@H]1C[C@@H](C(=O)O)N(C(=O)C[C@@H](N)c2ccccc2)C1 ZINC000217842331 CC For-Sale Unstable ACE 43 48 CO[C@@H]1C[C@@H](C(=O)O)N(C(=O)C[C@@H](N)c2ccccc2)C1 ZINC000217842331 CC For-Sale Unstable AGTR2 101 35 CC[C@H](NC(=O)[C@H](NS(=O)(=O)c1ccc(C)cc1)[C@@H](C)O)c1ccc(Cl)cc1 ZINC000217842345 HF On-Demand Unstable MMP13 22 49 CC[C@H](NC(=O)[C@H](NS(=O)(=O)c1ccc(C)cc1)[C@@H](C)O)c1ccc(Cl)cc1 ZINC000217842345 HF On-Demand Unstable MMP2 17 49 CC[C@H](NC(=O)[C@H](NS(=O)(=O)c1ccc(C)cc1)[C@@H](C)O)c1ccc(Cl)cc1 ZINC000217842345 HF On-Demand Unstable MMP12 20 44 CC[C@H](NC(=O)[C@H](NS(=O)(=O)c1ccc(C)cc1)[C@@H](C)O)c1ccc(Cl)cc1 ZINC000217842345 HF On-Demand Unstable MMP7 18 44 CC[C@H](NC(=O)[C@H](NS(=O)(=O)c1ccc(C)cc1)[C@@H](C)O)c1ccc(Cl)cc1 ZINC000217842345 HF On-Demand Unstable ADAMTS4 50 36 CC[C@H](NC(=O)[C@H](NS(=O)(=O)c1ccc(C)cc1)[C@@H](C)O)c1ccc(Cl)cc1 ZINC000217842345 HF On-Demand Unstable LEF 49 44 Clc1ccc(C2=NO[C@@H](CBr)C2)c(Cl)c1 ZINC000217842369 DH In-Stock Unstable LUCI_PHOPY 78 48 C[C@H]1Cc2ccccc2N([C@H](c2ccccc2)[C@@H](C)N)C1 ZINC000217842388 CH For-Sale Unstable TPP2 42 30 CO[C@H]1C[C@@H](C(=O)O)N(C(=O)C[C@@H](N)c2ccccc2)C1 ZINC000217842404 CC For-Sale Unstable ACE 43 48 CO[C@H]1C[C@@H](C(=O)O)N(C(=O)C[C@@H](N)c2ccccc2)C1 ZINC000217842404 CC For-Sale Unstable AGTR2 101 35 COc1ccc(/C=C\C(=O)O)cc1CN(C)CC(N)=O ZINC000217842416 CC For-Sale Unstable PTGER2 0 41 COc1ccc(/C=C\C(=O)O)cc1CN(C)CC(N)=O ZINC000217842416 CC For-Sale Unstable AKR1C3 22 41 COc1cc2c(c(OC)c1OC)-c1ccc(NCCCCCC(=O)NCc3ccccn3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217842419 KJ In-Stock Unstable TUBA1A 17 61 COc1ccc(OCC(=O)NCc2nc(-c3cccc(OC)c3)no2)cc1 ZINC000217842426 FE In-Stock Unstable ADORA1 0 45 COc1ccc(OCC(=O)NCc2nc(-c3cccc(OC)c3)no2)cc1 ZINC000217842426 FE In-Stock Unstable NQO2 28 40 COc1ccc(OCC(=O)NCc2nc(-c3cccc(OC)c3)no2)cc1 ZINC000217842426 FE In-Stock Unstable COLA 60 40 COc1ccc(OCC(=O)NCc2nc(-c3cccc(OC)c3)no2)cc1 ZINC000217842426 FE In-Stock Unstable CPT1A 44 40 COc1ccc(OCC(=O)NCc2nc(-c3cccc(OC)c3)no2)cc1 ZINC000217842426 FE In-Stock Unstable MTNR1A 85 42 COc1ccc(OCC(=O)NCc2nc(-c3cccc(OC)c3)no2)cc1 ZINC000217842426 FE In-Stock Unstable MTNR1B 68 38 Cc1ccc(OCC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217842428 DG For-Sale Unstable COLA 69 36 Cc1ccc(OCC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217842428 DG For-Sale Unstable CPT1A 64 35 Cc1ccc(OCC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217842428 DG For-Sale Unstable CHRNA10 40 39 Clc1ccc(C2=NO[C@H](CBr)C2)c(Cl)c1 ZINC000217842450 DH In-Stock Unstable LUCI_PHOPY 78 48 C[C@H]1Cc2ccccc2N([C@H](c2ccccc2)[C@H](C)N)C1 ZINC000217842468 CH For-Sale Unstable TPP2 42 30 Cc1ccc(OCC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217842491 DG For-Sale Unstable COLA 69 36 Cc1ccc(OCC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217842491 DG For-Sale Unstable CPT1A 64 35 Cc1ccc(OCC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217842491 DG For-Sale Unstable CHRNA10 40 39 COc1ccc(OCC(=O)NCc2nc(-c3ccc(OC)cc3OC)no2)cc1 ZINC000217842522 GE In-Stock Unstable MTNR1A 73 41 COc1ccc(OCC(=O)NCc2nc(-c3ccc(OC)cc3OC)no2)cc1 ZINC000217842522 GE In-Stock Unstable MTNR1B 54 41 O=C1C[C@@H](c2ccc3c(c2)OCO3)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217842527 II In-Stock Unstable AKR1B1 0 43 O=C1C[C@@H](c2ccc3c(c2)OCO3)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217842527 II In-Stock Unstable CYP1B1 16 40 O=C1C[C@@H](c2ccc3c(c2)OCO3)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217842527 II In-Stock Unstable CYP1A1 17 40 C[C@H]1C[C@H](C)CCN1Cc1cccc(O)c1 ZINC000217842536 BG For-Sale Unstable OPRM1 27 42 C[C@H]1C[C@H](C)CCN1Cc1cccc(O)c1 ZINC000217842536 BG For-Sale Unstable OPRD1 27 42 C[C@H]1C[C@H](C)CCN1Cc1cccc(O)c1 ZINC000217842536 BG For-Sale Unstable OPRK1 28 42 O=C(Cc1ccccc1Cl)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217842566 GG In-Stock Unstable PRCP 19 40 O=C(Cc1ccccc1Cl)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217842566 GG In-Stock Unstable COLA 57 37 O=C(Cc1ccccc1Cl)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217842566 GG In-Stock Unstable CPT1A 52 37 O=[N+]([O-])c1ccccc1C1=NO[C@@H](CBr)C1 ZINC000217842570 CE In-Stock Unstable LUCI_PHOPY 76 46 O=C(COc1ccc(Cl)cc1Cl)NC[C@H]1CCCN1c1ccccc1 ZINC000217842582 GI For-Sale Unstable PTGDR2 32 45 NS(=O)(=O)c1cccc(N[C@@H]2C[C@@H]3CC=C[C@H]32)c1 ZINC000217842600 CD For-Sale Unstable CA4 17 40 O=C1C[C@H](c2ccc3c(c2)OCO3)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217842613 II In-Stock Unstable AKR1B1 0 43 O=C1C[C@H](c2ccc3c(c2)OCO3)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217842613 II In-Stock Unstable CYP1B1 16 40 O=C1C[C@H](c2ccc3c(c2)OCO3)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217842613 II In-Stock Unstable CYP1A1 17 40 COc1ccc(OCC(=O)NCc2nc(-c3ccccc3Cl)no2)cc1 ZINC000217842620 FG In-Stock Unstable COLA 34 40 COc1ccc(OCC(=O)NCc2nc(-c3ccccc3Cl)no2)cc1 ZINC000217842620 FG In-Stock Unstable MTNR1A 54 38 COc1ccc(OCC(=O)NCc2nc(-c3ccccc3Cl)no2)cc1 ZINC000217842620 FG In-Stock Unstable PIM3 0 41 COc1ccc(OCC(=O)NCc2nc(-c3ccccc3Cl)no2)cc1 ZINC000217842620 FG In-Stock Unstable GPBAR1 18 45 O=C(Cc1ccccc1Cl)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217842639 GG In-Stock Unstable PRCP 19 40 O=C(Cc1ccccc1Cl)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217842639 GG In-Stock Unstable COLA 57 37 O=C(Cc1ccccc1Cl)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217842639 GG In-Stock Unstable CPT1A 52 37 C[C@H]1CCN(Cc2cccc(O)c2)[C@@H](C)C1 ZINC000217842642 BG For-Sale Unstable OPRM1 27 42 C[C@H]1CCN(Cc2cccc(O)c2)[C@@H](C)C1 ZINC000217842642 BG For-Sale Unstable OPRD1 27 42 C[C@H]1CCN(Cc2cccc(O)c2)[C@@H](C)C1 ZINC000217842642 BG For-Sale Unstable OPRK1 28 42 O=[N+]([O-])c1ccccc1C1=NO[C@H](CBr)C1 ZINC000217842649 CE In-Stock Unstable LUCI_PHOPY 76 46 O=C(COc1ccc(Cl)cc1Cl)NC[C@@H]1CCCN1c1ccccc1 ZINC000217842662 GI For-Sale Unstable PTGDR2 32 45 NS(=O)(=O)c1cccc(N[C@H]2C[C@@H]3CC=C[C@H]32)c1 ZINC000217842671 CD For-Sale Unstable CA4 17 40 C#CCCCNC(=O)c1ccc(F)c(OC)c1 ZINC000217842697 BD On-Demand Unstable DRD2 18 43 C#CCCCNC(=O)c1ccc(F)c(OC)c1 ZINC000217842697 BD On-Demand Unstable DRD4 42 33 C#CCCCNC(=O)c1ccc(F)c(OC)c1 ZINC000217842697 BD On-Demand Unstable DRD3 32 42 COc1ccc(OCC(=O)NCc2nc(-c3cccc(Br)c3)no2)cc1 ZINC000217842747 HG In-Stock Unstable MTNR1A 67 39 COc1ccc(OCC(=O)NCc2nc(-c3cccc(Br)c3)no2)cc1 ZINC000217842747 HG In-Stock Unstable MTNR1B 49 37 O=[N+]([O-])c1cccc(C2=NO[C@@H](CBr)C2)c1 ZINC000217842751 CE In-Stock Unstable LUCI_PHOPY 86 53 NS(=O)(=O)c1cccc(N[C@@H]2C[C@H]3CC=C[C@H]32)c1 ZINC000217842752 CD For-Sale Unstable CA4 17 40 CC(C)(C)c1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217842789 EI For-Sale Unstable HCRTR1 18 45 CC(C)(C)c1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217842789 EI For-Sale Unstable PLA2G4A 48 31 CC(C)(C)c1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217842789 EI For-Sale Unstable PREP 16 45 CC(C)(C)c1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217842789 EI For-Sale Unstable HCRTR2 15 45 CC(C)(C)c1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217842789 EI For-Sale Unstable CACNA1I 64 38 CC(C)(C)c1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217842789 EI For-Sale Unstable CYP2J2 47 41 CCOC(=O)/C(C)=N/Nc1ccc([N+](=O)[O-])cc1Br ZINC000217842827 EF For-Sale Unstable CACNA1C 44 35 CCOC(=O)/C(C)=N/Nc1ccc([N+](=O)[O-])cc1Br ZINC000217842827 EF For-Sale Unstable CACNA1D 61 34 O=[N+]([O-])c1cccc(C2=NO[C@H](CBr)C2)c1 ZINC000217842836 CE In-Stock Unstable LUCI_PHOPY 86 53 NS(=O)(=O)c1cccc(N[C@H]2C[C@H]3CC=C[C@@H]23)c1 ZINC000217842842 CD For-Sale Unstable CA4 17 40 CN(Cc1ccccn1)Cc1ccccc1/C=C\C(=O)O ZINC000217842858 CF For-Sale Unstable PTGER2 45 45 CN(Cc1ccccn1)Cc1ccccc1/C=C\C(=O)O ZINC000217842858 CF For-Sale Unstable PTGER4 23 45 CN(Cc1ccccn1)Cc1ccccc1/C=C\C(=O)O ZINC000217842858 CF For-Sale Unstable PTGER3 18 45 N[C@H](CCl)Cc1ccc(Cl)nc1 ZINC000217842860 BD For-Sale Unstable Q8WSF8_APLCA 31 40 N[C@H](CCl)Cc1ccc(Cl)nc1 ZINC000217842860 BD For-Sale Unstable NACHRBETA2 47 34 COc1ccc(OCC(=O)N(C)Cc2nc(-c3cccc(OC)c3)no2)cc1 ZINC000217842863 GF In-Stock Unstable COLA 54 40 COc1ccc(OCC(=O)N(C)Cc2nc(-c3cccc(OC)c3)no2)cc1 ZINC000217842863 GF In-Stock Unstable CPT1A 47 40 COc1ccc(OCC(=O)N(C)Cc2nc(-c3cccc(OC)c3)no2)cc1 ZINC000217842863 GF In-Stock Unstable HSD17B2 20 43 COC(=O)[C@@H](NC(=O)Cn1ccc2c(NC(C)=O)cccc21)C(C)C ZINC000217842869 ED In-Stock Unstable ELANE 48 39 CC(C)(C)c1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217842873 EI For-Sale Unstable HCRTR1 18 45 CC(C)(C)c1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217842873 EI For-Sale Unstable PLA2G4A 48 31 CC(C)(C)c1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217842873 EI For-Sale Unstable PREP 16 45 CC(C)(C)c1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217842873 EI For-Sale Unstable HCRTR2 15 45 CC(C)(C)c1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217842873 EI For-Sale Unstable CACNA1I 64 38 CC(C)(C)c1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217842873 EI For-Sale Unstable CYP2J2 47 41 N[C@@H](CCl)Cc1ccc(Cl)nc1 ZINC000217842930 BD For-Sale Unstable Q8WSF8_APLCA 31 40 N[C@@H](CCl)Cc1ccc(Cl)nc1 ZINC000217842930 BD For-Sale Unstable NACHRBETA2 47 34 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1 ZINC000217842955 II In-Stock Unstable AKR1B1 24 47 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1 ZINC000217842955 II In-Stock Unstable CYP1B1 53 50 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1 ZINC000217842955 II In-Stock Unstable CYP1A1 43 50 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1 ZINC000217842955 II In-Stock Unstable CYP1A2 33 50 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1 ZINC000217842955 II In-Stock Unstable ABCG2 0 40 O=[N+]([O-])c1ccc(C2=NO[C@@H](CBr)C2)cc1 ZINC000217842961 CE In-Stock Unstable LUCI_PHOPY 90 68 Cn1cc(C[C@H](N)C(=O)O)cc1Br ZINC000217842978 BC For-Sale Unstable TPH1 60 32 O=C(NC[C@H]1CCCN1c1ccccc1)C1CCCCC1 ZINC000217842982 CG For-Sale Unstable SLC6A1 55 34 O=C(NC[C@H]1CCCN1c1ccccc1)C1CCCCC1 ZINC000217842982 CG For-Sale Unstable HCRTR1 15 41 O=C(NC[C@H]1CCCN1c1ccccc1)C1CCCCC1 ZINC000217842982 CG For-Sale Unstable PREP 28 40 O=C(NC[C@H]1CCCN1c1ccccc1)C1CCCCC1 ZINC000217842982 CG For-Sale Unstable EPHX2 25 40 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1 ZINC000217843023 II In-Stock Unstable AKR1B1 24 47 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1 ZINC000217843023 II In-Stock Unstable CYP1B1 53 50 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1 ZINC000217843023 II In-Stock Unstable CYP1A1 43 50 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1 ZINC000217843023 II In-Stock Unstable CYP1A2 33 50 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1 ZINC000217843023 II In-Stock Unstable ABCG2 0 40 O=[N+]([O-])c1ccc(C2=NO[C@H](CBr)C2)cc1 ZINC000217843038 CE In-Stock Unstable LUCI_PHOPY 90 68 Cn1cc(C[C@@H](N)C(=O)O)cc1Br ZINC000217843039 BC For-Sale Unstable TPH1 60 32 CC[C@@H](N)[C@@H](N1C[C@@H](C)Cc2ccccc21)C(C)(C)C ZINC000217843042 CH For-Sale Unstable TPP2 55 35 O=C(NC[C@@H]1CCCN1c1ccccc1)C1CCCCC1 ZINC000217843045 CG For-Sale Unstable SLC6A1 55 34 O=C(NC[C@@H]1CCCN1c1ccccc1)C1CCCCC1 ZINC000217843045 CG For-Sale Unstable HCRTR1 15 41 O=C(NC[C@@H]1CCCN1c1ccccc1)C1CCCCC1 ZINC000217843045 CG For-Sale Unstable PREP 28 40 O=C(NC[C@@H]1CCCN1c1ccccc1)C1CCCCC1 ZINC000217843045 CG For-Sale Unstable EPHX2 25 40 CC[C@@H](CCO)NCCOc1ccccc1 ZINC000217843057 BD For-Sale Unstable DRD4 17 42 CN(Cc1cccc(/C=C\C(=O)O)c1)Cc1ccccn1 ZINC000217843083 CF For-Sale Unstable PTGER2 27 42 CN(Cc1cccc(/C=C\C(=O)O)c1)Cc1ccccn1 ZINC000217843083 CF For-Sale Unstable AKR1C3 43 42 CC[C@H](N)[C@@H](N1C[C@@H](C)Cc2ccccc21)C(C)(C)C ZINC000217843128 CH For-Sale Unstable TPP2 55 35 CC[C@H](CCO)NCCOc1ccccc1 ZINC000217843162 BD For-Sale Unstable DRD4 17 42 O=C(C[C@@H]1NC(=O)N(Cc2ccc3c(c2)OCO3)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217843171 IC In-Stock Unstable NPY1R 24 40 O=C(C[C@@H]1NC(=O)N(Cc2ccc3c(c2)OCO3)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217843171 IC In-Stock Unstable NOS2 53 32 O=C(C[C@@H]1NC(=O)N(Cc2ccc3c(c2)OCO3)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217843171 IC In-Stock Unstable SSTR3 72 33 O=C(C[C@@H]1NC(=O)N(Cc2ccc3c(c2)OCO3)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217843171 IC In-Stock Unstable MCHR1 20 43 Cc1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217843183 CG For-Sale Unstable DRD4 43 36 Cc1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217843183 CG For-Sale Unstable DRD3 19 45 Cc1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217843183 CG For-Sale Unstable HCRTR1 30 44 Cc1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217843183 CG For-Sale Unstable CTSL 16 41 Cc1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217843183 CG For-Sale Unstable PREP 26 43 Cc1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217843183 CG For-Sale Unstable HCRTR2 24 44 Cc1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217843183 CG For-Sale Unstable CACNA1I 50 38 Cc1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217843183 CG For-Sale Unstable ACKR3 53 36 Cc1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217843183 CG For-Sale Unstable KCNK3 64 42 Cc1cccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217843183 CG For-Sale Unstable KCNK9 46 42 COc1ccc(/C=C\C(=O)O)cc1Cn1cccnc1=O ZINC000217843187 CD For-Sale Unstable TSHR 53 32 COc1ccc(/C=C\C(=O)O)cc1Cn1cccnc1=O ZINC000217843187 CD For-Sale Unstable AKR1C3 30 40 COc1ccccc1C1=NO[C@@H](CBr)C1 ZINC000217843194 CF In-Stock Unstable LUCI_PHOPY 102 71 CC[C@@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)c1cccs1 ZINC000217843212 DG For-Sale Unstable ACE2 43 36 CC[C@@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)c1cccs1 ZINC000217843212 DG For-Sale Unstable CTSC 38 41 CC[C@@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)c1cccs1 ZINC000217843212 DG For-Sale Unstable XIAP 51 40 CC[C@@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)c1cccs1 ZINC000217843212 DG For-Sale Unstable SLC15A2 0 44 CC[C@@H](N)[C@H](N1C[C@@H](C)Cc2ccccc21)C(C)(C)C ZINC000217843218 CH For-Sale Unstable TPP2 55 35 COc1ccc(CN2C(=O)CCC2=O)cc1/C=C\C(=O)O ZINC000217843240 CD For-Sale Unstable PTGER2 38 43 COc1ccc(CN2C(=O)CCC2=O)cc1/C=C\C(=O)O ZINC000217843240 CD For-Sale Unstable PTGER4 22 43 COc1ccc(CN2C(=O)CCC2=O)cc1/C=C\C(=O)O ZINC000217843240 CD For-Sale Unstable PTGER3 26 43 C[C@@H](c1ccc(Cl)cc1)N(C)CC[C@@H](O)c1ccccc1 ZINC000217843250 DI On-Demand Unstable AOC3 29 48 C[C@@H](c1ccc(Cl)cc1)N(C)CC[C@@H](O)c1ccccc1 ZINC000217843250 DI On-Demand Unstable UTS2 49 41 Cc1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217843251 CG For-Sale Unstable DRD4 43 36 Cc1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217843251 CG For-Sale Unstable DRD3 19 45 Cc1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217843251 CG For-Sale Unstable HCRTR1 30 44 Cc1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217843251 CG For-Sale Unstable CTSL 16 41 Cc1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217843251 CG For-Sale Unstable PREP 26 43 Cc1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217843251 CG For-Sale Unstable HCRTR2 24 44 Cc1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217843251 CG For-Sale Unstable CACNA1I 50 38 Cc1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217843251 CG For-Sale Unstable ACKR3 53 36 Cc1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217843251 CG For-Sale Unstable KCNK3 64 42 Cc1cccc(C(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217843251 CG For-Sale Unstable KCNK9 46 42 COc1ccccc1C1=NO[C@H](CBr)C1 ZINC000217843253 CF In-Stock Unstable LUCI_PHOPY 102 71 O=C1C[C@@H](c2ccc(O)c(Cl)c2)c2c(c3ccccc3oc2=O)O1 ZINC000217843275 EH In-Stock Unstable NQO1 22 42 O=C(O)CCCCCNC(=O)N/C=C/c1ccccc1Br ZINC000217843287 FG For-Sale Unstable HDAC1 17 48 O=C(O)CCCCCNC(=O)N/C=C/c1ccccc1Br ZINC000217843287 FG For-Sale Unstable HDAC2 17 41 O=C(O)CCCCCNC(=O)N/C=C/c1ccccc1Br ZINC000217843287 FG For-Sale Unstable HDAC4 15 41 O=C(O)CCCCCNC(=O)N/C=C/c1ccccc1Br ZINC000217843287 FG For-Sale Unstable EPHX2 0 40 O=C(O)CCCCCNC(=O)N/C=C/c1ccccc1Br ZINC000217843287 FG For-Sale Unstable HDAC9 36 41 O=C(O)CCCCCNC(=O)N/C=C/c1ccccc1Br ZINC000217843287 FG For-Sale Unstable HDAC7 32 41 O=C(O)CCCCCNC(=O)N/C=C/c1ccccc1Br ZINC000217843287 FG For-Sale Unstable HDA106 0 46 CC[C@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)c1cccs1 ZINC000217843296 DG For-Sale Unstable ACE2 43 36 CC[C@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)c1cccs1 ZINC000217843296 DG For-Sale Unstable CTSC 38 41 CC[C@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)c1cccs1 ZINC000217843296 DG For-Sale Unstable XIAP 51 40 CC[C@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)c1cccs1 ZINC000217843296 DG For-Sale Unstable SLC15A2 0 44 CC[C@H](N)[C@H](N1C[C@@H](C)Cc2ccccc21)C(C)(C)C ZINC000217843299 CH For-Sale Unstable TPP2 55 35 COc1ccc(OCC(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217843300 EH In-Stock Unstable ADRB1 17 45 COc1ccc(OCC(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217843300 EH In-Stock Unstable SCNN1A 40 41 COc1ccc(OCC(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217843300 EH In-Stock Unstable ADRB3 22 45 COc1ccc(OCC(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217843300 EH In-Stock Unstable BMP1 35 42 COc1ccc(OCC(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217843300 EH In-Stock Unstable SCN2A 15 41 COc1ccc(OCC(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217843300 EH In-Stock Unstable MTNR1A 63 40 COc1ccc(OCC(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217843300 EH In-Stock Unstable MTNR1B 41 46 COc1ccc(OCC(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217843300 EH In-Stock Unstable CA9 16 44 COc1ccc(OCC(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217843300 EH In-Stock Unstable MMP1 18 40 COc1ccc(OCC(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217843300 EH In-Stock Unstable DXR 23 43 COc1ccc(OCC(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217843300 EH In-Stock Unstable FFAR1 15 41 COc1ccc(OCC(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217843300 EH In-Stock Unstable CRTM 43 39 COc1ccc(OCC(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217843300 EH In-Stock Unstable PROKR1 51 31 C[C@H](c1ccc(Cl)cc1)N(C)CC[C@@H](O)c1ccccc1 ZINC000217843312 DI On-Demand Unstable AOC3 29 48 C[C@H](c1ccc(Cl)cc1)N(C)CC[C@@H](O)c1ccccc1 ZINC000217843312 DI On-Demand Unstable UTS2 49 41 COc1ccc(C2=NO[C@@H](CBr)C2)cc1 ZINC000217843344 CF In-Stock Unstable LUCI_PHOPY 117 67 CCCC(CCC)C(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217843349 DH For-Sale Unstable ACE 42 38 O=C1C[C@H](c2ccc(O)c(Cl)c2)c2c(c3ccccc3oc2=O)O1 ZINC000217843371 EH In-Stock Unstable NQO1 22 42 C[C@H]1Cc2ccccc2N([C@@H](c2ccco2)[C@H](C)N)C1 ZINC000217843374 CG For-Sale Unstable TPP2 43 30 COc1ccc(OCC(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217843387 FG In-Stock Unstable DRD2 32 41 COc1ccc(OCC(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217843387 FG In-Stock Unstable DRD4 42 35 COc1ccc(OCC(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217843387 FG In-Stock Unstable HTR2A 20 42 COc1ccc(OCC(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217843387 FG In-Stock Unstable DRD3 45 42 COc1ccc(OCC(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217843387 FG In-Stock Unstable AVPR1A 23 41 COc1ccc(OCC(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217843387 FG In-Stock Unstable MTNR1A 45 37 COc1ccc(OCC(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217843387 FG In-Stock Unstable MTNR1B 38 42 COc1ccc(OCC(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217843387 FG In-Stock Unstable MTNR1C 0 40 COc1ccc(OCC(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217843387 FG In-Stock Unstable TYRO3 22 41 COc1ccc(C2=NO[C@H](CBr)C2)cc1 ZINC000217843399 CF In-Stock Unstable LUCI_PHOPY 117 67 CCCC(CCC)C(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217843404 DH For-Sale Unstable ACE 42 38 C[C@@H](c1ccc(Cl)cc1)N(C)CC[C@@H](O)C(C)(C)C ZINC000217843408 CI For-Sale Unstable UTS2 43 35 O=C(N1CCCO[C@@H](CN2CCCCC2)C1)C1(c2ccccc2)CC1 ZINC000217843452 EF In-Stock Unstable FABP4 44 35 O=C(N1CCCO[C@@H](CN2CCCCC2)C1)C1(c2ccccc2)CC1 ZINC000217843452 EF In-Stock Unstable HSD11B1 0 49 C[C@H]1Cc2ccccc2N([C@H](c2ccco2)[C@@H](C)N)C1 ZINC000217843459 CG For-Sale Unstable TPP2 43 30 C[C@H](c1ccc(Cl)cc1)N(C)CC[C@@H](O)C(C)(C)C ZINC000217843472 CI For-Sale Unstable UTS2 43 35 O=C(N1CCCO[C@H](CN2CCCCC2)C1)C1(c2ccccc2)CC1 ZINC000217843483 EF In-Stock Unstable FABP4 44 35 O=C(N1CCCO[C@H](CN2CCCCC2)C1)C1(c2ccccc2)CC1 ZINC000217843483 EF In-Stock Unstable HSD11B1 0 49 O=C(N[C@H](c1ccccc1)c1cccs1)[C@@H]1C[C@@H](O)CN1 ZINC000217843512 DD For-Sale Unstable XIAP 43 37 O=C(N[C@H](c1ccccc1)c1cccs1)[C@@H]1C[C@@H](O)CN1 ZINC000217843512 DD For-Sale Unstable BIRC8 45 33 Cc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217843517 CG For-Sale Unstable DRD2 28 42 Cc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217843517 CG For-Sale Unstable DRD4 17 42 Cc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217843517 CG For-Sale Unstable HCRTR1 25 46 Cc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217843517 CG For-Sale Unstable PREP 20 45 Cc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217843517 CG For-Sale Unstable HCRTR2 19 46 Cc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217843517 CG For-Sale Unstable CACNA1I 52 40 Cc1ccc(C(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217843517 CG For-Sale Unstable ACKR3 40 33 Fc1cccc(Cl)c1C1=NO[C@@H](CBr)C1 ZINC000217843526 CG In-Stock Unstable LUCI_PHOPY 84 44 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable ACE 113 54 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable OPRM1 45 41 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable OPRD1 49 43 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable MME 180 54 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable LTA4H 20 41 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable ANPEP 75 43 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable EDNRA 22 53 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable TACR1 26 42 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable CTSD 50 48 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable PGC 53 36 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable CTRA_BOVIN 28 46 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable FCER2 99 38 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable CASP3 32 42 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable TACR2 51 40 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable RNPEP 24 41 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable CTSB 56 51 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable PAPA1_CARPA 69 43 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable CYSP_TRYCR 64 60 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable RIR1_HHV11 32 44 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable CTSK 21 48 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable CTSL 43 48 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable CPA1 48 47 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable PGA 41 36 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable NPFFR2 45 31 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable HLA-A 68 46 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable ITGA4 52 38 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable NAALAD2 30 43 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable CAPNS1 66 40 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable MMP2 23 40 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable MMP3 36 44 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable MMP8 23 40 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable ECE1 82 42 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable HLA-DRB1 88 43 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable REN 59 48 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable REN1 42 35 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable LNPEP 24 41 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable CTSS 38 57 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable CTSH 26 44 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable CAPN1 94 53 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable MMP9 26 40 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable CASP1 47 44 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable CAPN2 76 44 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable CTSE 41 39 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable ACE2 122 47 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable BACE1 20 46 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable PGA5 51 39 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable LAP3 20 40 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable MMP1 41 40 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable FPR1 92 46 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable NPR 61 40 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable AMP1_PLAFQ 34 41 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable XIAP 37 46 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable PSMB2 44 39 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable BLA1_STEMA 80 41 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable PSMB8 69 42 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable DLG4 41 33 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable Q9N6S8_PLAFA 28 49 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable BRCA1 80 45 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable NPFFR1 54 31 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843533 GC On-Demand Unstable Q6PRC7_IXORI 56 43 CCOC(=O)[C@@H]1CCCN1S(=O)(=O)NC[C@@H](N)CC(C)C ZINC000217843541 DC For-Sale Unstable RHODESAIN 0 40 C[C@H]1Cc2ccccc2N([C@H](c2ccco2)[C@H](C)N)C1 ZINC000217843551 CG For-Sale Unstable TPP2 43 30 COc1ccc(C(=O)NCCCc2ccccc2OC)cc1 ZINC000217843554 CG In-Stock Unstable HTR1A 19 47 COc1ccc(C(=O)NCCCc2ccccc2OC)cc1 ZINC000217843554 CG In-Stock Unstable DRD2 32 48 COc1ccc(C(=O)NCCCc2ccccc2OC)cc1 ZINC000217843554 CG In-Stock Unstable DRD1 15 47 COc1ccc(C(=O)NCCCc2ccccc2OC)cc1 ZINC000217843554 CG In-Stock Unstable DRD4 44 34 COc1ccc(C(=O)NCCCc2ccccc2OC)cc1 ZINC000217843554 CG In-Stock Unstable ACHE 0 49 COc1ccc(C(=O)NCCCc2ccccc2OC)cc1 ZINC000217843554 CG In-Stock Unstable DRD3 49 47 COc1ccc(C(=O)NCCCc2ccccc2OC)cc1 ZINC000217843554 CG In-Stock Unstable PTAFR 16 44 COc1ccc(C(=O)NCCCc2ccccc2OC)cc1 ZINC000217843554 CG In-Stock Unstable NQO2 31 55 COc1ccc(C(=O)NCCCc2ccccc2OC)cc1 ZINC000217843554 CG In-Stock Unstable TRPV1 22 47 COc1ccc(C(=O)NCCCc2ccccc2OC)cc1 ZINC000217843554 CG In-Stock Unstable BCHE 40 34 COc1ccc(C(=O)NCCCc2ccccc2OC)cc1 ZINC000217843554 CG In-Stock Unstable KCNA3 23 44 COc1ccc(C(=O)NCCCc2ccccc2OC)cc1 ZINC000217843554 CG In-Stock Unstable PPARD 15 43 COc1ccc(C(=O)NCCCc2ccccc2OC)cc1 ZINC000217843554 CG In-Stock Unstable CA14 0 44 COc1ccc(C(=O)NCCCc2ccccc2OC)cc1 ZINC000217843554 CG In-Stock Unstable MTNR1A 98 42 COc1ccc(C(=O)NCCCc2ccccc2OC)cc1 ZINC000217843554 CG In-Stock Unstable MTNR1B 88 55 COc1ccc(C(=O)NCCCc2ccccc2OC)cc1 ZINC000217843554 CG In-Stock Unstable SLC6A5 20 46 COc1ccc(C(=O)NCCCc2ccccc2OC)cc1 ZINC000217843554 CG In-Stock Unstable ITGAV 18 40 COc1ccc(C(=O)NCCCc2ccccc2OC)cc1 ZINC000217843554 CG In-Stock Unstable MCHR1 17 40 COc1ccc(C(=O)NCCCc2ccccc2OC)cc1 ZINC000217843554 CG In-Stock Unstable TAAR1 22 49 COc1ccc(C(=O)NCCCc2ccccc2OC)cc1 ZINC000217843554 CG In-Stock Unstable TBK1 23 42 COc1ccc(C(=O)NCCCc2ccccc2OC)cc1 ZINC000217843554 CG In-Stock Unstable MBTPS1 43 38 Cc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217843581 CG For-Sale Unstable DRD2 28 42 Cc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217843581 CG For-Sale Unstable DRD4 17 42 Cc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217843581 CG For-Sale Unstable HCRTR1 25 46 Cc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217843581 CG For-Sale Unstable PREP 20 45 Cc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217843581 CG For-Sale Unstable HCRTR2 19 46 Cc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217843581 CG For-Sale Unstable CACNA1I 52 40 Cc1ccc(C(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217843581 CG For-Sale Unstable ACKR3 40 33 O=C(N[C@H](c1ccccc1)c1cccs1)[C@H]1C[C@@H](O)CN1 ZINC000217843596 DD For-Sale Unstable XIAP 43 37 O=C(N[C@H](c1ccccc1)c1cccs1)[C@H]1C[C@@H](O)CN1 ZINC000217843596 DD For-Sale Unstable BIRC8 45 33 CN1C(=O)C(=O)N(Cc2cccc(/C=C\C(=O)O)c2)C1=O ZINC000217843598 CC For-Sale Unstable HDAC8 32 40 CN1C(=O)C(=O)N(Cc2cccc(/C=C\C(=O)O)c2)C1=O ZINC000217843598 CC For-Sale Unstable HDAC6 24 40 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable ACE 113 54 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable OPRM1 45 41 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable OPRD1 49 43 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable MME 180 54 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable LTA4H 20 41 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable ANPEP 75 43 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable EDNRA 22 53 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable TACR1 26 42 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable CTSD 50 48 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable PGC 53 36 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable CTRA_BOVIN 28 46 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable FCER2 99 38 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable CASP3 32 42 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable TACR2 51 40 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable RNPEP 24 41 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable CTSB 56 51 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable PAPA1_CARPA 69 43 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable CYSP_TRYCR 64 60 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable RIR1_HHV11 32 44 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable CTSK 21 48 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable CTSL 43 48 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable CPA1 48 47 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable PGA 41 36 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable NPFFR2 45 31 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable HLA-A 68 46 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable ITGA4 52 38 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable NAALAD2 30 43 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable CAPNS1 66 40 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable MMP2 23 40 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable MMP3 36 44 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable MMP8 23 40 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable ECE1 82 42 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable HLA-DRB1 88 43 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable REN 59 48 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable REN1 42 35 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable LNPEP 24 41 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable CTSS 38 57 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable CTSH 26 44 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable CAPN1 94 53 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable MMP9 26 40 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable CASP1 47 44 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable CAPN2 76 44 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable CTSE 41 39 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable ACE2 122 47 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable BACE1 20 46 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable PGA5 51 39 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable LAP3 20 40 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable MMP1 41 40 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable FPR1 92 46 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable NPR 61 40 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable AMP1_PLAFQ 34 41 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable XIAP 37 46 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable PSMB2 44 39 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable BLA1_STEMA 80 41 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable PSMB8 69 42 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable DLG4 41 33 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable Q9N6S8_PLAFA 28 49 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable BRCA1 80 45 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable NPFFR1 54 31 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000217843606 GC On-Demand Unstable Q6PRC7_IXORI 56 43 Fc1cccc(Cl)c1C1=NO[C@H](CBr)C1 ZINC000217843610 CG In-Stock Unstable LUCI_PHOPY 84 44 C[C@@H](c1cccc(Cl)c1)N(C)C[C@@H](N)c1ccccc1 ZINC000217843617 CI For-Sale Unstable OPRL1 0 44 C[C@@H](c1cccc(Cl)c1)N(C)C[C@@H](N)c1ccccc1 ZINC000217843617 CI For-Sale Unstable AOC3 32 48 CCOc1ccc(CCCNC(=O)c2ccc(OC)cc2)cc1 ZINC000217843630 DG In-Stock Unstable DRD4 40 31 CCOc1ccc(CCCNC(=O)c2ccc(OC)cc2)cc1 ZINC000217843630 DG In-Stock Unstable SCNN1A 39 40 CCOc1ccc(CCCNC(=O)c2ccc(OC)cc2)cc1 ZINC000217843630 DG In-Stock Unstable PTAFR 21 46 CCOc1ccc(CCCNC(=O)c2ccc(OC)cc2)cc1 ZINC000217843630 DG In-Stock Unstable KCNQ1 0 46 CCOc1ccc(CCCNC(=O)c2ccc(OC)cc2)cc1 ZINC000217843630 DG In-Stock Unstable TRPV1 0 42 CCOc1ccc(CCCNC(=O)c2ccc(OC)cc2)cc1 ZINC000217843630 DG In-Stock Unstable SCN2A 30 51 CCOc1ccc(CCCNC(=O)c2ccc(OC)cc2)cc1 ZINC000217843630 DG In-Stock Unstable MTNR1A 59 39 CCOc1ccc(CCCNC(=O)c2ccc(OC)cc2)cc1 ZINC000217843630 DG In-Stock Unstable MTNR1B 42 45 CCOc1ccc(CCCNC(=O)c2ccc(OC)cc2)cc1 ZINC000217843630 DG In-Stock Unstable SLC2A1 0 40 CCOc1ccc(CCCNC(=O)c2ccc(OC)cc2)cc1 ZINC000217843630 DG In-Stock Unstable PLA2G4B 41 35 CCOc1ccc(CCCNC(=O)c2ccc(OC)cc2)cc1 ZINC000217843630 DG In-Stock Unstable CA9 18 43 CCOc1ccc(CCCNC(=O)c2ccc(OC)cc2)cc1 ZINC000217843630 DG In-Stock Unstable HDA106 0 54 CCOc1ccc(CCCNC(=O)c2ccc(OC)cc2)cc1 ZINC000217843630 DG In-Stock Unstable HT1 0 40 CCOc1ccc(CCCNC(=O)c2ccc(OC)cc2)cc1 ZINC000217843630 DG In-Stock Unstable CRTM 40 35 CCOc1ccc(CCCNC(=O)c2ccc(OC)cc2)cc1 ZINC000217843630 DG In-Stock Unstable AP2S1 0 41 CCOc1ccc(CCCNC(=O)c2ccc(OC)cc2)cc1 ZINC000217843630 DG In-Stock Unstable LMGT2 0 40 CCOC(=O)[C@H]1CCCN1S(=O)(=O)NC[C@@H](N)CC(C)C ZINC000217843632 DC For-Sale Unstable RHODESAIN 0 40 CC[C@@H](N)[C@H](c1ccco1)N1C[C@@H](C)Cc2ccccc21 ZINC000217843644 CH For-Sale Unstable TPP2 54 34 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable ACE 113 54 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable OPRM1 45 41 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable OPRD1 49 43 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable MME 180 54 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable LTA4H 20 41 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable ANPEP 75 43 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable EDNRA 22 53 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable TACR1 26 42 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable CTSD 50 48 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable PGC 53 36 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable CTRA_BOVIN 28 46 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable FCER2 99 38 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable CASP3 32 42 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable TACR2 51 40 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable RNPEP 24 41 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable CTSB 56 51 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable PAPA1_CARPA 69 43 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable CYSP_TRYCR 64 60 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable RIR1_HHV11 32 44 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable CTSK 21 48 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable CTSL 43 48 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable CPA1 48 47 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable PGA 41 36 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable NPFFR2 45 31 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable HLA-A 68 46 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable ITGA4 52 38 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable NAALAD2 30 43 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable CAPNS1 66 40 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable MMP2 23 40 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable MMP3 36 44 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable MMP8 23 40 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable ECE1 82 42 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable HLA-DRB1 88 43 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable REN 59 48 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable REN1 42 35 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable LNPEP 24 41 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable CTSS 38 57 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable CTSH 26 44 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable CAPN1 94 53 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable MMP9 26 40 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable CASP1 47 44 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable CAPN2 76 44 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable CTSE 41 39 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable ACE2 122 47 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable BACE1 20 46 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable PGA5 51 39 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable LAP3 20 40 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable MMP1 41 40 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable FPR1 92 46 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable NPR 61 40 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable AMP1_PLAFQ 34 41 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable XIAP 37 46 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable PSMB2 44 39 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable BLA1_STEMA 80 41 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable PSMB8 69 42 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable DLG4 41 33 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable Q9N6S8_PLAFA 28 49 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable BRCA1 80 45 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable NPFFR1 54 31 CC(C)[C@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843688 GC On-Demand Unstable Q6PRC7_IXORI 56 43 O=C(CCS(=O)(=O)c1ccccc1)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217843689 IE In-Stock Unstable CPT1A 43 35 C[C@H](c1cccc(Cl)c1)N(C)C[C@@H](N)c1ccccc1 ZINC000217843697 CI For-Sale Unstable OPRL1 0 44 C[C@H](c1cccc(Cl)c1)N(C)C[C@@H](N)c1ccccc1 ZINC000217843697 CI For-Sale Unstable AOC3 32 48 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217843702 HF For-Sale Unstable EPHX2 15 43 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217843702 HF For-Sale Unstable TGM2 76 47 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217843702 HF For-Sale Unstable CACNA1I 44 31 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217843702 HF For-Sale Unstable F13A1 72 40 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217843702 HF For-Sale Unstable AKR1C3 28 40 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217843702 HF For-Sale Unstable SFRP1 43 40 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217843702 HF For-Sale Unstable AKR1C1 21 42 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217843702 HF For-Sale Unstable NAMPT 43 44 CCCOc1ccccc1CCCNC(=O)c1ccc(OC)cc1 ZINC000217843713 EH In-Stock Unstable DRD2 21 44 CCCOc1ccccc1CCCNC(=O)c1ccc(OC)cc1 ZINC000217843713 EH In-Stock Unstable DRD1 0 41 CCCOc1ccccc1CCCNC(=O)c1ccc(OC)cc1 ZINC000217843713 EH In-Stock Unstable DRD4 40 31 CCCOc1ccccc1CCCNC(=O)c1ccc(OC)cc1 ZINC000217843713 EH In-Stock Unstable DRD3 36 42 CCCOc1ccccc1CCCNC(=O)c1ccc(OC)cc1 ZINC000217843713 EH In-Stock Unstable PPARG 22 41 CCCOc1ccccc1CCCNC(=O)c1ccc(OC)cc1 ZINC000217843713 EH In-Stock Unstable PTAFR 17 40 CCCOc1ccccc1CCCNC(=O)c1ccc(OC)cc1 ZINC000217843713 EH In-Stock Unstable KCNQ1 0 44 CCCOc1ccccc1CCCNC(=O)c1ccc(OC)cc1 ZINC000217843713 EH In-Stock Unstable NQO2 21 49 CCCOc1ccccc1CCCNC(=O)c1ccc(OC)cc1 ZINC000217843713 EH In-Stock Unstable SCN2A 18 40 CCCOc1ccccc1CCCNC(=O)c1ccc(OC)cc1 ZINC000217843713 EH In-Stock Unstable MTNR1A 82 44 CCCOc1ccccc1CCCNC(=O)c1ccc(OC)cc1 ZINC000217843713 EH In-Stock Unstable MTNR1B 74 51 CCCOc1ccccc1CCCNC(=O)c1ccc(OC)cc1 ZINC000217843713 EH In-Stock Unstable ABCB1 0 40 CCCOc1ccccc1CCCNC(=O)c1ccc(OC)cc1 ZINC000217843713 EH In-Stock Unstable SLC6A5 15 42 CCCOc1ccccc1CCCNC(=O)c1ccc(OC)cc1 ZINC000217843713 EH In-Stock Unstable TBK1 20 41 CCCOc1ccccc1CCCNC(=O)c1ccc(OC)cc1 ZINC000217843713 EH In-Stock Unstable AP2S1 0 44 CC[C@H](N)[C@H](c1ccco1)N1C[C@@H](C)Cc2ccccc21 ZINC000217843716 CH For-Sale Unstable TPP2 54 34 Clc1cccc(C2=NO[C@@H](CBr)C2)c1Cl ZINC000217843732 DH In-Stock Unstable LUCI_PHOPY 86 55 COc1ccc2cc(CNC[C@@](C)(O)CSC)ccc2c1 ZINC000217843739 DG On-Demand Unstable SLC6A13 0 40 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217843742 FG For-Sale Unstable ACE 15 42 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217843742 FG For-Sale Unstable FOLH1 60 40 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217843742 FG For-Sale Unstable MME 41 45 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217843742 FG For-Sale Unstable ANPEP 49 48 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217843742 FG For-Sale Unstable RNPEP 24 42 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217843742 FG For-Sale Unstable PAPA1_CARPA 44 35 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217843742 FG For-Sale Unstable CTSK 21 40 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217843742 FG For-Sale Unstable CAPNS1 51 34 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217843742 FG For-Sale Unstable CAPN1 51 42 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217843742 FG For-Sale Unstable CAPN2 44 34 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217843742 FG For-Sale Unstable FPR1 83 44 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217843742 FG For-Sale Unstable NPR 65 36 CC(C)C[C@@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217843742 FG For-Sale Unstable AMP1_PLAFQ 22 42 O=C(CCS(=O)(=O)c1ccccc1)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217843762 IE In-Stock Unstable CPT1A 43 35 COc1ccc(Cn2cc(C)cn2)cc1/C=C\C(=O)O ZINC000217843770 CE For-Sale Unstable PTGER2 33 41 COc1ccc(Cn2cc(C)cn2)cc1/C=C\C(=O)O ZINC000217843770 CE For-Sale Unstable PTGER4 18 41 COc1ccc(Cn2cc(C)cn2)cc1/C=C\C(=O)O ZINC000217843770 CE For-Sale Unstable PTGER3 18 40 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable ACE 113 54 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable OPRM1 45 41 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable OPRD1 49 43 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable MME 180 54 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable LTA4H 20 41 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable ANPEP 75 43 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable EDNRA 22 53 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable TACR1 26 42 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable CTSD 50 48 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable PGC 53 36 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable CTRA_BOVIN 28 46 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable FCER2 99 38 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable CASP3 32 42 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable TACR2 51 40 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable RNPEP 24 41 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable CTSB 56 51 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable PAPA1_CARPA 69 43 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable CYSP_TRYCR 64 60 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable RIR1_HHV11 32 44 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable CTSK 21 48 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable CTSL 43 48 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable CPA1 48 47 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable PGA 41 36 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable NPFFR2 45 31 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable HLA-A 68 46 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable ITGA4 52 38 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable NAALAD2 30 43 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable CAPNS1 66 40 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable MMP2 23 40 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable MMP3 36 44 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable MMP8 23 40 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable ECE1 82 42 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable HLA-DRB1 88 43 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable REN 59 48 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable REN1 42 35 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable LNPEP 24 41 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable CTSS 38 57 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable CTSH 26 44 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable CAPN1 94 53 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable MMP9 26 40 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable CASP1 47 44 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable CAPN2 76 44 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable CTSE 41 39 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable ACE2 122 47 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable BACE1 20 46 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable PGA5 51 39 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable LAP3 20 40 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable MMP1 41 40 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable FPR1 92 46 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable NPR 61 40 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable AMP1_PLAFQ 34 41 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable XIAP 37 46 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable PSMB2 44 39 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable BLA1_STEMA 80 41 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable PSMB8 69 42 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable DLG4 41 33 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable Q9N6S8_PLAFA 28 49 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable BRCA1 80 45 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable NPFFR1 54 31 CC(C)[C@@H](NC(=O)N1CCOCC1)C(=O)N[C@H](Cc1ccccc1)C(=O)O ZINC000217843776 GC On-Demand Unstable Q6PRC7_IXORI 56 43 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217843777 HF For-Sale Unstable EPHX2 15 43 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217843777 HF For-Sale Unstable TGM2 76 47 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217843777 HF For-Sale Unstable CACNA1I 44 31 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217843777 HF For-Sale Unstable F13A1 72 40 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217843777 HF For-Sale Unstable AKR1C3 28 40 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217843777 HF For-Sale Unstable SFRP1 43 40 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217843777 HF For-Sale Unstable AKR1C1 21 42 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217843777 HF For-Sale Unstable NAMPT 43 44 COc1ccc2cc(CNC[C@](C)(O)CSC)ccc2c1 ZINC000217843801 DG On-Demand Unstable SLC6A13 0 40 Clc1cccc(C2=NO[C@H](CBr)C2)c1Cl ZINC000217843802 DH In-Stock Unstable LUCI_PHOPY 86 55 COCC[C@H](N)CN(C)[C@@H](C)c1cccc(Cl)c1 ZINC000217843806 CF For-Sale Unstable AOC3 16 49 CC[C@@H](N)[C@@H](c1ccco1)N1C[C@@H](C)Cc2ccccc21 ZINC000217843810 CH For-Sale Unstable TPP2 54 34 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217843811 FG For-Sale Unstable ACE 15 42 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217843811 FG For-Sale Unstable FOLH1 60 40 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217843811 FG For-Sale Unstable MME 41 45 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217843811 FG For-Sale Unstable ANPEP 49 48 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217843811 FG For-Sale Unstable RNPEP 24 42 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217843811 FG For-Sale Unstable PAPA1_CARPA 44 35 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217843811 FG For-Sale Unstable CTSK 21 40 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217843811 FG For-Sale Unstable CAPNS1 51 34 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217843811 FG For-Sale Unstable CAPN1 51 42 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217843811 FG For-Sale Unstable CAPN2 44 34 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217843811 FG For-Sale Unstable FPR1 83 44 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217843811 FG For-Sale Unstable NPR 65 36 CC(C)C[C@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217843811 FG For-Sale Unstable AMP1_PLAFQ 22 42 CC[C@H](N)[C@@H](c1ccco1)N1C[C@@H](C)Cc2ccccc21 ZINC000217843875 CH For-Sale Unstable TPP2 54 34 CSCC[C@@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217843898 FF For-Sale Unstable FOLH1 24 42 CSCC[C@@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217843898 FF For-Sale Unstable NAALAD2 44 36 CSCC[C@@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217843898 FF For-Sale Unstable PAM 0 42 CSCC[C@@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217843898 FF For-Sale Unstable FPR1 42 41 CSCC[C@@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217843898 FF For-Sale Unstable SLC15A2 0 41 CSCC[C@@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217843898 FF For-Sale Unstable FPRL2 0 41 COC(=O)C[C@H](c1ccc(O)c(Cl)c1)c1c(O)c2ccccc2oc1=O ZINC000217843915 FH In-Stock Unstable NQO1 49 38 Fc1cc(F)cc(C2=NO[C@@H](CBr)C2)c1 ZINC000217843927 CF In-Stock Unstable LUCI_PHOPY 88 49 Nc1[nH]nc(C(=O)N2CCC[C@@H]2c2nc3cc(F)ccc3[nH]2)c1Cl ZINC000217843940 EF In-Stock Unstable PRCP 61 45 Cc1ccc(OCc2ccccc2/C=C\C(=O)O)c(C)c1 ZINC000217843975 CH For-Sale Unstable PTGER2 30 64 Cc1ccc(OCc2ccccc2/C=C\C(=O)O)c(C)c1 ZINC000217843975 CH For-Sale Unstable PTGER4 44 59 Cc1ccc(OCc2ccccc2/C=C\C(=O)O)c(C)c1 ZINC000217843975 CH For-Sale Unstable PTGER3 33 64 Cc1ccc(OCc2ccccc2/C=C\C(=O)O)c(C)c1 ZINC000217843975 CH For-Sale Unstable PTGDR 0 46 Cc1ccc(OCc2ccccc2/C=C\C(=O)O)c(C)c1 ZINC000217843975 CH For-Sale Unstable AKR1C3 32 44 COc1ccc(C(=O)N[C@@H](C)c2ccc(N3CCC[C@@H](C)C3)cc2)cc1 ZINC000217843995 FI In-Stock Unstable ELANE 21 42 COc1ccc(C(=O)N[C@@H](C)c2ccc(N3CCC[C@@H](C)C3)cc2)cc1 ZINC000217843995 FI In-Stock Unstable GRM3 15 42 COc1ccc(C(=O)N[C@@H](C)c2ccc(N3CCC[C@@H](C)C3)cc2)cc1 ZINC000217843995 FI In-Stock Unstable RORC 37 43 CC[C@@H](C)N(C)CCNC(=O)[C@@H]1CCC[C@@H]1C(=O)O ZINC000217843999 CD For-Sale Unstable ACE 0 42 CSCC[C@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217844003 FF For-Sale Unstable FOLH1 24 42 CSCC[C@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217844003 FF For-Sale Unstable NAALAD2 44 36 CSCC[C@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217844003 FF For-Sale Unstable PAM 0 42 CSCC[C@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217844003 FF For-Sale Unstable FPR1 42 41 CSCC[C@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217844003 FF For-Sale Unstable SLC15A2 0 41 CSCC[C@H](NC(=O)N/C=C/c1ccccc1Br)C(=O)O ZINC000217844003 FF For-Sale Unstable FPRL2 0 41 Fc1cc(F)cc(C2=NO[C@H](CBr)C2)c1 ZINC000217844009 CF In-Stock Unstable LUCI_PHOPY 88 49 Nc1[nH]nc(C(=O)N2CCC[C@H]2c2nc3cc(F)ccc3[nH]2)c1Cl ZINC000217844024 EF In-Stock Unstable PRCP 61 45 COC(=O)C[C@@H](c1ccc(O)c(Cl)c1)c1c(O)c2ccccc2oc1=O ZINC000217844028 FH In-Stock Unstable NQO1 49 38 CC[C@H](C)N(C)CCNC(=O)[C@@H]1CCC[C@@H]1C(=O)O ZINC000217844067 CD For-Sale Unstable ACE 0 42 Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)c(C)c1 ZINC000217844069 CH For-Sale Unstable PTGER2 24 55 Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)c(C)c1 ZINC000217844069 CH For-Sale Unstable PTGER4 32 46 Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)c(C)c1 ZINC000217844069 CH For-Sale Unstable PTGER3 23 55 Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)c(C)c1 ZINC000217844069 CH For-Sale Unstable AKR1C3 39 58 Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)c(C)c1 ZINC000217844069 CH For-Sale Unstable AKR1B10 21 41 COc1ccc(C(=O)N[C@H](C)c2ccc(N3CCC[C@@H](C)C3)cc2)cc1 ZINC000217844070 FI In-Stock Unstable ELANE 21 42 COc1ccc(C(=O)N[C@H](C)c2ccc(N3CCC[C@@H](C)C3)cc2)cc1 ZINC000217844070 FI In-Stock Unstable GRM3 15 42 BrC[C@@H]1CC(c2ccc3c(c2)OCO3)=NO1 ZINC000217844102 CE In-Stock Unstable DYRK1A 40 35 BrC[C@@H]1CC(c2ccc3c(c2)OCO3)=NO1 ZINC000217844102 CE In-Stock Unstable CLK1 40 35 BrC[C@@H]1CC(c2ccc3c(c2)OCO3)=NO1 ZINC000217844102 CE In-Stock Unstable CLK2 48 35 BrC[C@@H]1CC(c2ccc3c(c2)OCO3)=NO1 ZINC000217844102 CE In-Stock Unstable CLK4 73 35 BrC[C@@H]1CC(c2ccc3c(c2)OCO3)=NO1 ZINC000217844102 CE In-Stock Unstable LUCI_PHOPY 86 42 COc1ccc([C@@H](C)NC(=O)N/C=C/c2ccccc2Br)cc1OC ZINC000217844105 HI For-Sale Unstable KCNQ2 50 38 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)c(C)c1 ZINC000217844127 CH For-Sale Unstable MAOB 17 45 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)c(C)c1 ZINC000217844127 CH For-Sale Unstable PTGER2 31 56 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)c(C)c1 ZINC000217844127 CH For-Sale Unstable PTGER1 40 42 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)c(C)c1 ZINC000217844127 CH For-Sale Unstable PTGER4 32 46 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)c(C)c1 ZINC000217844127 CH For-Sale Unstable PTGER3 25 56 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)c(C)c1 ZINC000217844127 CH For-Sale Unstable LTB4R 28 44 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)c(C)c1 ZINC000217844127 CH For-Sale Unstable KCNA3 0 40 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)c(C)c1 ZINC000217844127 CH For-Sale Unstable HCAR2 0 40 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)c(C)c1 ZINC000217844127 CH For-Sale Unstable FFAR1 43 43 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)c(C)c1 ZINC000217844127 CH For-Sale Unstable AKR1C3 45 56 O=C(NCC1C[C@@H]2CC[C@H](C1)N2)NC1CCCCC1 ZINC000217844136 CE For-Sale Unstable EPHX2 19 48 COc1ccc(C(=O)N[C@@H]2CC(C)(C)Oc3ccc(C)cc32)cc1 ZINC000217844154 EI In-Stock Unstable NAAA 23 45 CC(C)[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(Cc2ccc3c(c2)OCO3)C1=O ZINC000217844157 GC In-Stock Unstable NOS2 57 34 CC(C)[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(Cc2ccc3c(c2)OCO3)C1=O ZINC000217844157 GC In-Stock Unstable SSTR3 76 32 CC(C)[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(Cc2ccc3c(c2)OCO3)C1=O ZINC000217844157 GC In-Stock Unstable MCHR1 21 40 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000217844176 IG For-Sale Unstable EPHX2 16 44 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000217844176 IG For-Sale Unstable TGM2 72 46 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000217844176 IG For-Sale Unstable F13A1 66 39 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000217844176 IG For-Sale Unstable AKR1C3 30 42 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000217844176 IG For-Sale Unstable AKR1C1 21 41 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000217844176 IG For-Sale Unstable NAMPT 42 46 BrC[C@H]1CC(c2ccc3c(c2)OCO3)=NO1 ZINC000217844187 CE In-Stock Unstable DYRK1A 40 35 BrC[C@H]1CC(c2ccc3c(c2)OCO3)=NO1 ZINC000217844187 CE In-Stock Unstable CLK1 40 35 BrC[C@H]1CC(c2ccc3c(c2)OCO3)=NO1 ZINC000217844187 CE In-Stock Unstable CLK2 48 35 BrC[C@H]1CC(c2ccc3c(c2)OCO3)=NO1 ZINC000217844187 CE In-Stock Unstable CLK4 73 35 BrC[C@H]1CC(c2ccc3c(c2)OCO3)=NO1 ZINC000217844187 CE In-Stock Unstable LUCI_PHOPY 86 42 COc1cccc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217844203 CG For-Sale Unstable PTGER2 25 49 COc1cccc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217844203 CG For-Sale Unstable PTGER4 46 55 COc1cccc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217844203 CG For-Sale Unstable PTGER3 40 56 COc1cccc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217844203 CG For-Sale Unstable LTB4R 32 41 COc1cccc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217844203 CG For-Sale Unstable MTNR1A 37 42 COc1cccc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217844203 CG For-Sale Unstable MTNR1B 39 42 COc1cccc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217844203 CG For-Sale Unstable ABCB1 0 42 COc1cccc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217844203 CG For-Sale Unstable AKR1C3 35 44 COc1ccc([C@H](C)NC(=O)N/C=C/c2ccccc2Br)cc1OC ZINC000217844217 HI For-Sale Unstable KCNQ2 50 38 COc1ccc(C(=O)N[C@H]2CC(C)(C)Oc3ccc(C)cc32)cc1 ZINC000217844224 EI In-Stock Unstable NAAA 23 45 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000217844232 IG For-Sale Unstable EPHX2 16 44 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000217844232 IG For-Sale Unstable TGM2 72 46 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000217844232 IG For-Sale Unstable F13A1 66 39 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000217844232 IG For-Sale Unstable AKR1C3 26 40 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000217844232 IG For-Sale Unstable AKR1C1 21 41 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000217844232 IG For-Sale Unstable NAMPT 42 46 BrC[C@@H]1CC(c2ccccn2)=NO1 ZINC000217844280 BD In-Stock Unstable LUCI_PHOPY 72 38 COc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217844287 CG For-Sale Unstable ALOX5 23 50 COc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217844287 CG For-Sale Unstable MAOB 41 57 COc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217844287 CG For-Sale Unstable PTGS2 0 47 COc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217844287 CG For-Sale Unstable PTGER2 24 46 COc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217844287 CG For-Sale Unstable PTGER4 44 53 COc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217844287 CG For-Sale Unstable CYP1B1 37 40 COc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217844287 CG For-Sale Unstable PTPN2 0 41 COc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217844287 CG For-Sale Unstable PTGER3 39 53 COc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217844287 CG For-Sale Unstable DRTS_LEIMA 27 40 COc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217844287 CG For-Sale Unstable LTB4R 37 46 COc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217844287 CG For-Sale Unstable MTNR1A 30 43 COc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217844287 CG For-Sale Unstable MTNR1B 35 43 COc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217844287 CG For-Sale Unstable CYP1A1 27 40 COc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217844287 CG For-Sale Unstable 17HSDCL 0 40 COc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217844287 CG For-Sale Unstable CYP24A1 16 42 COc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217844287 CG For-Sale Unstable TAAR1 15 42 COc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217844287 CG For-Sale Unstable FFAR1 60 43 COc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217844287 CG For-Sale Unstable AKR1C3 46 55 COc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217844287 CG For-Sale Unstable ABCG2 26 47 COc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217844287 CG For-Sale Unstable CYP27B1 25 42 COc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217844287 CG For-Sale Unstable PDS 22 40 COc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217844287 CG For-Sale Unstable GPR183 0 42 C[C@H]1Cc2ccccc2N(C[C@@H](O)Cn2cc(N)cn2)C1 ZINC000217844312 CD For-Sale Unstable TPP2 50 30 COc1ccc([C@@H](C)NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217844317 GI For-Sale Unstable KCNQ2 47 36 COc1ccc([C@@H](C)NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217844317 GI For-Sale Unstable ACACA 48 41 COc1ccc([C@@H](C)NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217844317 GI For-Sale Unstable ACACB 17 41 BrC[C@H]1CC(c2ccccn2)=NO1 ZINC000217844337 BD In-Stock Unstable LUCI_PHOPY 72 38 C[C@@H](c1cccc(Cl)c1)N(C)C[C@@H](N)Cc1ccccc1 ZINC000217844346 DH For-Sale Unstable AOC3 25 44 COc1ccc(C(=O)N[C@@H]2CC(C)(C)Oc3cc(C)ccc32)cc1 ZINC000217844365 EI In-Stock Unstable NAAA 24 45 CC(=O)Nc1cccc(N[C@@H]2C[C@@H]3CC=C[C@H]32)c1 ZINC000217844367 BG For-Sale Unstable KCNK3 50 33 COc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217844368 CG For-Sale Unstable ALOX5 24 44 COc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217844368 CG For-Sale Unstable MAOA 16 42 COc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217844368 CG For-Sale Unstable MAOB 66 51 COc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217844368 CG For-Sale Unstable PTGER2 24 50 COc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217844368 CG For-Sale Unstable CYSLTR1 16 40 COc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217844368 CG For-Sale Unstable PTGER4 38 53 COc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217844368 CG For-Sale Unstable G6PC 23 40 COc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217844368 CG For-Sale Unstable PTGER3 36 53 COc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217844368 CG For-Sale Unstable DRTS_LEIMA 27 40 COc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217844368 CG For-Sale Unstable LTB4R 35 45 COc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217844368 CG For-Sale Unstable KCNA3 25 42 COc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217844368 CG For-Sale Unstable AHR 23 40 COc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217844368 CG For-Sale Unstable MTNR1A 45 46 COc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217844368 CG For-Sale Unstable MTNR1B 51 46 COc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217844368 CG For-Sale Unstable NR1H4 66 39 COc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217844368 CG For-Sale Unstable HSD17B2 20 40 COc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217844368 CG For-Sale Unstable 17HSDCL 0 40 COc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217844368 CG For-Sale Unstable FFAR1 76 46 COc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217844368 CG For-Sale Unstable AKR1C3 47 61 COc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217844368 CG For-Sale Unstable ABCG2 19 48 COc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217844368 CG For-Sale Unstable ADCYAP1R1 40 36 COc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217844368 CG For-Sale Unstable PDS 45 42 Cc1n[nH]c([C@@H]2CCCN2C(=O)Cc2ccncc2)n1 ZINC000217844393 CD In-Stock Unstable PRCP 46 42 Cc1n[nH]c([C@@H]2CCCN2C(=O)Cc2ccncc2)n1 ZINC000217844393 CD In-Stock Unstable CPT1A 101 46 Cc1n[nH]c([C@@H]2CCCN2C(=O)Cc2ccncc2)n1 ZINC000217844393 CD In-Stock Unstable FAP 0 43 CCNS(=O)(=O)CCNCc1ccc(Br)c(F)c1 ZINC000217844398 ED On-Demand Unstable LEF 46 37 N#Cc1ccccc1-c1ccccc1C(=O)Nc1ccc2nc(N3CCCC3)sc2c1 ZINC000217844402 HK On-Demand Unstable NPY2R 32 42 N#Cc1ccccc1-c1ccccc1C(=O)Nc1ccc2nc(N3CCCC3)sc2c1 ZINC000217844402 HK On-Demand Unstable NR2E3 65 36 C[C@@H]1Cc2ccccc2N(C[C@@H](O)Cn2cc(N)cn2)C1 ZINC000217844404 CD For-Sale Unstable TPP2 50 30 COc1ccc([C@H](C)NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217844407 GI For-Sale Unstable KCNQ2 47 36 COc1ccc([C@H](C)NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217844407 GI For-Sale Unstable ACACA 48 41 COc1ccc([C@H](C)NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217844407 GI For-Sale Unstable ACACB 17 41 C[C@H](c1cccc(Cl)c1)N(C)C[C@@H](N)Cc1ccccc1 ZINC000217844423 DH For-Sale Unstable AOC3 25 44 COc1ccc(C(=O)N[C@H]2CC(C)(C)Oc3cc(C)ccc32)cc1 ZINC000217844432 EI In-Stock Unstable NAAA 24 45 O=C(O)/C=C\c1ccccc1COc1ccccc1F ZINC000217844434 CH For-Sale Unstable PTGER2 25 56 O=C(O)/C=C\c1ccccc1COc1ccccc1F ZINC000217844434 CH For-Sale Unstable PTGER4 38 56 O=C(O)/C=C\c1ccccc1COc1ccccc1F ZINC000217844434 CH For-Sale Unstable CXCL8 20 47 O=C(O)/C=C\c1ccccc1COc1ccccc1F ZINC000217844434 CH For-Sale Unstable FABP4 19 46 O=C(O)/C=C\c1ccccc1COc1ccccc1F ZINC000217844434 CH For-Sale Unstable PTGER3 31 56 O=C(O)/C=C\c1ccccc1COc1ccccc1F ZINC000217844434 CH For-Sale Unstable CDC25B 22 41 O=C(O)/C=C\c1ccccc1COc1ccccc1F ZINC000217844434 CH For-Sale Unstable PTGDR 0 47 O=C(O)/C=C\c1ccccc1COc1ccccc1F ZINC000217844434 CH For-Sale Unstable AKR1C3 30 48 CC(=O)Nc1cccc(N[C@H]2C[C@@H]3CC=C[C@H]32)c1 ZINC000217844439 BG For-Sale Unstable KCNK3 50 33 Nc1ccccc1C1=NO[C@@H](CBr)C1 ZINC000217844454 CE In-Stock Unstable LUCI_PHOPY 87 48 O=[N+]([O-])c1ccc(OC(=S)c2cccc(Cl)c2)cc1 ZINC000217844461 CI For-Sale Anodyne ACR 24 42 O=[N+]([O-])c1ccc(OC(=S)c2cccc(Cl)c2)cc1 ZINC000217844461 CI For-Sale Anodyne PPOX1 15 46 Cn1nc(-c2ccc(F)cc2)cc1C(=O)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217844468 IG In-Stock Unstable CCR3 45 31 Cc1n[nH]c([C@H]2CCCN2C(=O)Cc2ccncc2)n1 ZINC000217844481 CD In-Stock Unstable PRCP 46 42 Cc1n[nH]c([C@H]2CCCN2C(=O)Cc2ccncc2)n1 ZINC000217844481 CD In-Stock Unstable CPT1A 101 46 Cc1n[nH]c([C@H]2CCCN2C(=O)Cc2ccncc2)n1 ZINC000217844481 CD In-Stock Unstable FAP 0 43 Nc1ccccc1C1=NO[C@H](CBr)C1 ZINC000217844513 CE In-Stock Unstable LUCI_PHOPY 87 48 O=C(NC[C@H]1CCCN1c1ccccc1)c1cc(-c2ccc(F)cc2)n[nH]1 ZINC000217844517 FH For-Sale Unstable HCRTR1 24 46 O=C(NC[C@H]1CCCN1c1ccccc1)c1cc(-c2ccc(F)cc2)n[nH]1 ZINC000217844517 FH For-Sale Unstable TACR3 16 40 O=C(NC[C@H]1CCCN1c1ccccc1)c1cc(-c2ccc(F)cc2)n[nH]1 ZINC000217844517 FH For-Sale Unstable ALPL 54 37 O=C(NC[C@H]1CCCN1c1ccccc1)c1cc(-c2ccc(F)cc2)n[nH]1 ZINC000217844517 FH For-Sale Unstable HCRTR2 23 46 CN1CCN(C(=O)c2ccc(B(O)O)c(F)c2)CC1 ZINC000217844518 CA In-Stock Unstable HRH4 32 49 CN1CCN(C(=O)c2ccc(B(O)O)c(F)c2)CC1 ZINC000217844518 CA In-Stock Unstable L3MBTL1 0 43 CN1CCN(C(=O)c2ccc(B(O)O)c(F)c2)CC1 ZINC000217844518 CA In-Stock Unstable L3MBTL3 52 43 O=C(O)/C=C\c1ccc(COc2ccccc2F)cc1 ZINC000217844520 CH For-Sale Unstable PTGER2 24 50 O=C(O)/C=C\c1ccc(COc2ccccc2F)cc1 ZINC000217844520 CH For-Sale Unstable PTGER1 42 42 O=C(O)/C=C\c1ccc(COc2ccccc2F)cc1 ZINC000217844520 CH For-Sale Unstable PTGER4 38 50 O=C(O)/C=C\c1ccc(COc2ccccc2F)cc1 ZINC000217844520 CH For-Sale Unstable CXCL8 18 43 O=C(O)/C=C\c1ccc(COc2ccccc2F)cc1 ZINC000217844520 CH For-Sale Unstable PTPN2 0 42 O=C(O)/C=C\c1ccc(COc2ccccc2F)cc1 ZINC000217844520 CH For-Sale Unstable PTGER3 28 50 O=C(O)/C=C\c1ccc(COc2ccccc2F)cc1 ZINC000217844520 CH For-Sale Unstable LTB4R 0 44 O=C(O)/C=C\c1ccc(COc2ccccc2F)cc1 ZINC000217844520 CH For-Sale Unstable CDC25B 22 42 O=C(O)/C=C\c1ccc(COc2ccccc2F)cc1 ZINC000217844520 CH For-Sale Unstable PTGDR 0 42 O=C(O)/C=C\c1ccc(COc2ccccc2F)cc1 ZINC000217844520 CH For-Sale Unstable AKR1C3 40 57 O=C(O)/C=C\c1ccc(COc2ccccc2F)cc1 ZINC000217844520 CH For-Sale Unstable AKR1B10 17 46 CC(=O)Nc1cccc(N[C@@H]2C[C@H]3CC=C[C@H]32)c1 ZINC000217844533 BG For-Sale Unstable KCNK3 50 33 Cn1nc(-c2ccc(F)cc2)cc1C(=O)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217844545 IG In-Stock Unstable CCR3 45 31 COc1ccc(C(=O)N[C@@H]2CC(C)(C)Oc3ccc(OC)cc32)cc1 ZINC000217844551 EH In-Stock Unstable NAAA 24 50 Cc1ccc(-n2ncc(C(=O)Nc3ccc4nc(N5CCCC5)sc4c3)c2C(F)(F)F)cc1 ZINC000217844592 JK On-Demand Unstable MST1R 57 42 Nc1cccc(C2=NO[C@@H](CBr)C2)c1 ZINC000217844596 CE In-Stock Unstable LUCI_PHOPY 92 48 CC(=O)Nc1cccc(N[C@H]2C[C@H]3CC=C[C@@H]23)c1 ZINC000217844613 BG For-Sale Unstable KCNK3 50 33 COc1ccc(C(=O)N[C@H]2CC(C)(C)Oc3ccc(OC)cc32)cc1 ZINC000217844618 EH In-Stock Unstable NAAA 24 50 O=C(O)/C=C\c1ccc(COc2ccccc2F)c(F)c1 ZINC000217844621 CH For-Sale Unstable PTGER2 51 44 O=C(O)/C=C\c1ccc(COc2ccccc2F)c(F)c1 ZINC000217844621 CH For-Sale Unstable PTGER1 35 42 O=C(O)/C=C\c1ccc(COc2ccccc2F)c(F)c1 ZINC000217844621 CH For-Sale Unstable PTGER4 26 42 O=C(O)/C=C\c1ccc(COc2ccccc2F)c(F)c1 ZINC000217844621 CH For-Sale Unstable CXCL8 18 43 O=C(O)/C=C\c1ccc(COc2ccccc2F)c(F)c1 ZINC000217844621 CH For-Sale Unstable PTGER3 22 43 O=C(O)/C=C\c1ccc(COc2ccccc2F)c(F)c1 ZINC000217844621 CH For-Sale Unstable CDC25B 23 42 O=C(O)/C=C\c1ccc(COc2ccccc2F)c(F)c1 ZINC000217844621 CH For-Sale Unstable AKR1C3 37 59 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cc(-c2ccc(F)cc2)n[nH]1 ZINC000217844626 FH For-Sale Unstable HCRTR1 24 46 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cc(-c2ccc(F)cc2)n[nH]1 ZINC000217844626 FH For-Sale Unstable TACR3 16 40 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cc(-c2ccc(F)cc2)n[nH]1 ZINC000217844626 FH For-Sale Unstable ALPL 54 37 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cc(-c2ccc(F)cc2)n[nH]1 ZINC000217844626 FH For-Sale Unstable HCRTR2 23 46 Nc1cccc(C2=NO[C@H](CBr)C2)c1 ZINC000217844676 CE In-Stock Unstable LUCI_PHOPY 92 48 C[C@H](NCC(C)(C)N)C(=O)O ZINC000217844689 AB For-Sale Unstable SLC15A2 0 43 C[C@H](NCC(C)(C)N)C(=O)O ZINC000217844689 AB For-Sale Unstable BHMT2 46 30 C[C@@H](c1ccccc1Cl)N(C)CC[C@@H](O)c1ccccc1 ZINC000217844717 DI On-Demand Unstable AOC3 23 48 COc1ccc(C(=O)N[C@@H]2CC(C)(C)Oc3cc(OC)ccc32)cc1 ZINC000217844725 EH In-Stock Unstable TRPV1 0 40 COc1ccc(C(=O)N[C@@H]2CC(C)(C)Oc3cc(OC)ccc32)cc1 ZINC000217844725 EH In-Stock Unstable NAAA 25 50 O=C1OCCN1Cc1nc(-c2ccco2)nn1Cc1ccc2c(c1)OCO2 ZINC000217844733 FE In-Stock Unstable ADORA1 0 44 O=C1OCCN1Cc1nc(-c2ccco2)nn1Cc1ccc2c(c1)OCO2 ZINC000217844733 FE In-Stock Unstable ADORA2A 34 44 O=C(O)/C=C\c1ccc(OCCN2CCNC(=O)C2)cc1 ZINC000217844735 CC For-Sale Unstable LTA4H 39 43 O=C(O)/C=C\c1ccc(OCCN2CCNC(=O)C2)cc1 ZINC000217844735 CC For-Sale Unstable THRB 0 46 O=C(O)/C=C\c1ccc(OCCN2CCNC(=O)C2)cc1 ZINC000217844735 CC For-Sale Unstable HRH3 16 46 O=C(O)/C=C\c1ccc(OCCN2CCNC(=O)C2)cc1 ZINC000217844735 CC For-Sale Unstable PSMB2 47 37 O=C(O)/C=C\c1ccc(OCCN2CCNC(=O)C2)cc1 ZINC000217844735 CC For-Sale Unstable PSMB1 41 37 C[C@@H](NCC(C)(C)N)C(=O)O ZINC000217844770 AB For-Sale Unstable SLC15A2 0 43 C[C@@H](NCC(C)(C)N)C(=O)O ZINC000217844770 AB For-Sale Unstable BHMT2 46 30 BrC[C@@H]1CC(c2ccc(Br)cc2)=NO1 ZINC000217844779 DG In-Stock Unstable LUCI_PHOPY 98 49 COc1ccc(C(=O)N[C@H]2CC(C)(C)Oc3cc(OC)ccc32)cc1 ZINC000217844797 EH In-Stock Unstable TRPV1 0 40 COc1ccc(C(=O)N[C@H]2CC(C)(C)Oc3cc(OC)ccc32)cc1 ZINC000217844797 EH In-Stock Unstable NAAA 25 50 C[C@H](c1ccccc1Cl)N(C)CC[C@@H](O)c1ccccc1 ZINC000217844801 DI On-Demand Unstable AOC3 23 48 COc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)Nc1c(C)nn(C(C)C)c1C)C(=O)OC2 ZINC000217844824 JJ In-Stock Unstable IMPDH1 0 68 COc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)Nc1c(C)nn(C(C)C)c1C)C(=O)OC2 ZINC000217844824 JJ In-Stock Unstable IMPDH2 0 68 CC[C@@H](C)[C@@H](N)C(=O)N[C@H](c1cccs1)C(C)C ZINC000217844837 CF For-Sale Unstable CTSC 32 41 CCc1ccc([C@@H](C)NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217844863 FK For-Sale Unstable KCNQ2 47 36 BrC[C@H]1CC(c2ccc(Br)cc2)=NO1 ZINC000217844871 DG In-Stock Unstable LUCI_PHOPY 98 49 O=C(O)/C=C\c1cccc(CN2CCCCCCC2)c1 ZINC000217844909 CH For-Sale Unstable DRD2 16 44 O=C(O)/C=C\c1cccc(CN2CCCCCCC2)c1 ZINC000217844909 CH For-Sale Unstable ACHE 22 45 O=C(O)/C=C\c1cccc(CN2CCCCCCC2)c1 ZINC000217844909 CH For-Sale Unstable HRH2 37 44 O=C(O)/C=C\c1cccc(CN2CCCCCCC2)c1 ZINC000217844909 CH For-Sale Unstable PTGER2 26 40 O=C(O)/C=C\c1cccc(CN2CCCCCCC2)c1 ZINC000217844909 CH For-Sale Unstable CHRM3 18 43 O=C(O)/C=C\c1cccc(CN2CCCCCCC2)c1 ZINC000217844909 CH For-Sale Unstable HRH3 23 44 O=C(O)/C=C\c1cccc(CN2CCCCCCC2)c1 ZINC000217844909 CH For-Sale Unstable SIGMAR1 50 48 O=C(O)/C=C\c1cccc(CN2CCCCCCC2)c1 ZINC000217844909 CH For-Sale Unstable BDKRB1 41 41 O=C(O)/C=C\c1cccc(CN2CCCCCCC2)c1 ZINC000217844909 CH For-Sale Unstable HDAC8 41 40 O=C(O)/C=C\c1cccc(CN2CCCCCCC2)c1 ZINC000217844909 CH For-Sale Unstable HDAC1 19 44 O=C(O)/C=C\c1cccc(CN2CCCCCCC2)c1 ZINC000217844909 CH For-Sale Unstable HDAC6 27 40 O=C(O)/C=C\c1cccc(CN2CCCCCCC2)c1 ZINC000217844909 CH For-Sale Unstable ABCB1 18 40 O=C(O)/C=C\c1cccc(CN2CCCCCCC2)c1 ZINC000217844909 CH For-Sale Unstable AKR1C3 32 40 CC[C@H](C)[C@@H](N)C(=O)N[C@H](c1cccs1)C(C)C ZINC000217844921 CF For-Sale Unstable CTSC 32 41 COC(=O)C[C@@H](c1c(O)c2ccccc2oc1=O)c1cc2cc(OC)ccc2n(CC(C)C)c1=O ZINC000217844930 JI In-Stock Unstable NQO1 25 48 CC[C@@H](NC(=O)c1ccc(OC)cc1)c1ccc(C)c(C)c1 ZINC000217844932 CI In-Stock Unstable CTSL 20 44 CC[C@@H](NC(=O)c1ccc(OC)cc1)c1ccc(C)c(C)c1 ZINC000217844932 CI In-Stock Unstable TACR3 42 38 CC[C@@H](NC(=O)c1ccc(OC)cc1)c1ccc(C)c(C)c1 ZINC000217844932 CI In-Stock Unstable UTS2 79 52 CCc1ccc([C@H](C)NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217844941 FK For-Sale Unstable KCNQ2 47 36 Cc1ccccc1-n1cc(CNC(=O)c2noc(C)c2CO)cn1 ZINC000217844962 ED In-Stock Unstable PANC 41 34 O=C(O)/C=C\c1cc(F)ccc1CN1CCCCCCC1 ZINC000217844978 CH For-Sale Unstable SLC6A1 49 42 COC(=O)C[C@H](c1c(O)c2ccccc2oc1=O)c1cc2cc(OC)ccc2n(CC(C)C)c1=O ZINC000217844995 JI In-Stock Unstable NQO1 25 48 CC[C@H](NC(=O)c1ccc(OC)cc1)c1ccc(C)c(C)c1 ZINC000217844996 CI In-Stock Unstable CTSL 20 44 CC[C@H](NC(=O)c1ccc(OC)cc1)c1ccc(C)c(C)c1 ZINC000217844996 CI In-Stock Unstable TACR3 42 38 CC[C@H](NC(=O)c1ccc(OC)cc1)c1ccc(C)c(C)c1 ZINC000217844996 CI In-Stock Unstable UTS2 79 52 Cc1nc2ccccc2c(-c2ccccc2)c1CC(=O)N1CCc2ccc([N+](=O)[O-])cc21 ZINC000217845011 HK On-Demand Unstable F2RL3 49 37 Cc1nc2ccccc2c(-c2ccccc2)c1CC(=O)N1CCc2ccc([N+](=O)[O-])cc21 ZINC000217845011 HK On-Demand Unstable EIF2AK3 42 35 ClC[C@@H]1CC(c2cccs2)=NO1 ZINC000217845021 BE In-Stock Unstable LUCI_PHOPY 80 39 C[C@@H](NC(=O)N/C=C/c1ccccc1Br)c1ccc2c(c1)CCCC2 ZINC000217845061 GK For-Sale Unstable KCNQ2 49 40 ClC[C@H]1CC(c2cccs2)=NO1 ZINC000217845067 BE In-Stock Unstable LUCI_PHOPY 80 39 COC(=O)C[C@H](c1cc(OC)c2c(c1)OCO2)c1c(O)c2ccccc2oc1=O ZINC000217845114 GF In-Stock Unstable NQO1 48 45 CC[C@@H](NC(=O)c1ccc(OC)cc1)c1ccc(C)cc1C ZINC000217845138 CI In-Stock Unstable CTSL 24 47 CC[C@@H](NC(=O)c1ccc(OC)cc1)c1ccc(C)cc1C ZINC000217845138 CI In-Stock Unstable CTSS 15 47 CC[C@@H](NC(=O)c1ccc(OC)cc1)c1ccc(C)cc1C ZINC000217845138 CI In-Stock Unstable UTS2 59 51 O=C(Cn1cnc2ccccc2c1=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217845142 FE For-Sale Unstable HTR7 17 45 C[C@H](NC(=O)N/C=C/c1ccccc1Br)c1ccc2c(c1)CCCC2 ZINC000217845151 GK For-Sale Unstable KCNQ2 49 40 C[C@@H](c1cccc(Cl)c1)N(C)C[C@@](C)(N)C1CC1 ZINC000217845153 CG For-Sale Unstable OPRL1 0 40 COC(=O)Cc1ccc(C#N)cc1F ZINC000217845160 AD For-Sale Unstable CYSP_TRYCR 27 40 COC(=O)Cc1ccc(C#N)cc1F ZINC000217845160 AD For-Sale Unstable CTSF 30 40 O=C(/C=C/c1ccccc1)N1CCn2nc([C@@H](O)CO)cc2C1 ZINC000217845164 DC In-Stock Unstable GPR183 0 40 ClC[C@@H]1CC(c2ccccn2)=NO1 ZINC000217845185 AD In-Stock Unstable LUCI_PHOPY 88 42 COC(=O)C[C@@H](c1cc(OC)c2c(c1)OCO2)c1c(O)c2ccccc2oc1=O ZINC000217845187 GF In-Stock Unstable NQO1 48 45 CC[C@H](NC(=O)c1ccc(OC)cc1)c1ccc(C)cc1C ZINC000217845218 CI In-Stock Unstable CTSL 24 47 CC[C@H](NC(=O)c1ccc(OC)cc1)c1ccc(C)cc1C ZINC000217845218 CI In-Stock Unstable CTSS 15 47 CC[C@H](NC(=O)c1ccc(OC)cc1)c1ccc(C)cc1C ZINC000217845218 CI In-Stock Unstable UTS2 59 51 O=C(Cn1cnc2ccccc2c1=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217845223 FE For-Sale Unstable HTR7 17 45 C[C@H](c1cccc(Cl)c1)N(C)C[C@@](C)(N)C1CC1 ZINC000217845230 CG For-Sale Unstable OPRL1 0 40 C[C@H]1C[C@H](C)CCN1[C@@H](C)c1cccc(O)c1 ZINC000217845238 BH For-Sale Unstable OPRM1 20 46 C[C@H]1C[C@H](C)CCN1[C@@H](C)c1cccc(O)c1 ZINC000217845238 BH For-Sale Unstable OPRD1 15 46 O=C(/C=C/c1ccccc1)N1CCn2nc([C@H](O)CO)cc2C1 ZINC000217845253 DC In-Stock Unstable GPR183 0 40 ClC[C@H]1CC(c2ccccn2)=NO1 ZINC000217845261 AD In-Stock Unstable LUCI_PHOPY 88 42 CN1CCO[C@@H]([C@@H](O)Cc2ccc3ccccc3n2)C1 ZINC000217845286 CD For-Sale Unstable SMO 42 35 Oc1cccc(-c2ncsc2Br)c1 ZINC000217845308 CG For-Sale Anodyne HSD17B1 53 46 Oc1cccc(-c2ncsc2Br)c1 ZINC000217845308 CG For-Sale Anodyne HSD17B2 30 43 CC[C@@H](NC(=O)c1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217845318 EH In-Stock Unstable PPARD 22 41 CC[C@@H](NC(=O)c1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217845318 EH In-Stock Unstable TACR3 42 38 CC[C@@H](NC(=O)c1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217845318 EH In-Stock Unstable TUBB2B 15 41 CC[C@@H](NC(=O)c1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217845318 EH In-Stock Unstable MT-ND1 27 44 CC[C@@H](NC(=O)c1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217845318 EH In-Stock Unstable DXR 25 42 CC[C@@H](NC(=O)c1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217845318 EH In-Stock Unstable ENPP1 55 33 CC[C@@H](NC(=O)c1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217845318 EH In-Stock Unstable UTS2 71 52 O=C(NC[C@H]1CCCN1c1ccccc1)c1cc(-c2ccc3c(c2)OCO3)n[nH]1 ZINC000217845319 GG For-Sale Unstable NOS2 63 37 C[C@H]1C[C@H](C)CCN1[C@H](C)c1cccc(O)c1 ZINC000217845322 BH For-Sale Unstable OPRM1 20 46 C[C@H]1C[C@H](C)CCN1[C@H](C)c1cccc(O)c1 ZINC000217845322 BH For-Sale Unstable OPRD1 15 46 O=C(N/C=C/c1ccccc1Br)Nc1ccc(Oc2ccccc2)cc1 ZINC000217845349 HK For-Sale Anodyne CA1 43 47 O=C(N/C=C/c1ccccc1Br)Nc1ccc(Oc2ccccc2)cc1 ZINC000217845349 HK For-Sale Anodyne RAF1 29 40 O=C(N/C=C/c1ccccc1Br)Nc1ccc(Oc2ccccc2)cc1 ZINC000217845349 HK For-Sale Anodyne CA12 17 50 O=C(N/C=C/c1ccccc1Br)Nc1ccc(Oc2ccccc2)cc1 ZINC000217845349 HK For-Sale Anodyne CA9 17 47 O=C(N/C=C/c1ccccc1Br)Nc1ccc(Oc2ccccc2)cc1 ZINC000217845349 HK For-Sale Anodyne Q8MMZ8_EIMTE 34 40 O=C(N/C=C/c1ccccc1Br)Nc1ccc(Oc2ccccc2)cc1 ZINC000217845349 HK For-Sale Anodyne F13A1 15 40 O=C(N/C=C/c1ccccc1Br)Nc1ccc(Oc2ccccc2)cc1 ZINC000217845349 HK For-Sale Anodyne P96878_MYCTU 15 50 CN1CCO[C@H]([C@@H](O)Cc2ccc3ccccc3n2)C1 ZINC000217845355 CD For-Sale Unstable SMO 42 35 CO[C@@H]1CC[C@@H](NC(=O)c2cccc(-c3ccc(F)cc3)c2)CC1 ZINC000217845362 EI In-Stock Unstable PDE4B 41 36 CO[C@@H]1CC[C@@H](NC(=O)c2cccc(-c3ccc(F)cc3)c2)CC1 ZINC000217845362 EI In-Stock Unstable FAAH 0 49 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cc(-c2ccc3c(c2)OCO3)n[nH]1 ZINC000217845378 GG For-Sale Unstable NOS2 63 37 CC[C@H](NC(=O)c1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217845382 EH In-Stock Unstable PPARD 22 41 CC[C@H](NC(=O)c1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217845382 EH In-Stock Unstable TACR3 42 38 CC[C@H](NC(=O)c1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217845382 EH In-Stock Unstable TUBB2B 15 41 CC[C@H](NC(=O)c1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217845382 EH In-Stock Unstable MT-ND1 27 44 CC[C@H](NC(=O)c1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217845382 EH In-Stock Unstable DXR 25 42 CC[C@H](NC(=O)c1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217845382 EH In-Stock Unstable ENPP1 55 33 CC[C@H](NC(=O)c1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217845382 EH In-Stock Unstable UTS2 71 52 ClC[C@@H]1CC(c2ccncc2)=NO1 ZINC000217845397 AD In-Stock Unstable LUCI_PHOPY 95 49 CC[C@@H](C)N(CC)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217845398 CG For-Sale Unstable AKR1C3 29 40 CC[C@@H](C)N(CC)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217845398 CG For-Sale Unstable PDS 46 33 COc1cccc(C(=O)N2CCNC[C@H]2C)n1 ZINC000217845408 BC For-Sale Unstable ALS 43 33 ClC[C@H]1CC(c2ccncc2)=NO1 ZINC000217845439 AD In-Stock Unstable LUCI_PHOPY 95 49 CC[C@@H](NC(=O)c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217845449 EF In-Stock Unstable CA2 24 44 CC[C@@H](NC(=O)c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217845449 EF In-Stock Unstable PTGS2 24 49 CC[C@@H](NC(=O)c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217845449 EF In-Stock Unstable BMP1 54 39 CC[C@@H](NC(=O)c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217845449 EF In-Stock Unstable MMP13 41 44 CC[C@@H](NC(=O)c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217845449 EF In-Stock Unstable TACR3 45 39 CC[C@@H](NC(=O)c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217845449 EF In-Stock Unstable MMP3 42 39 CC[C@@H](NC(=O)c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217845449 EF In-Stock Unstable MMP1 47 41 CC[C@@H](NC(=O)c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217845449 EF In-Stock Unstable LOX1.1 43 37 CC[C@@H](NC(=O)c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217845449 EF In-Stock Unstable UTS2 64 51 CC[C@@H](NC(=O)c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217845449 EF In-Stock Unstable GPR88 0 40 CC[C@H](C)N(CC)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217845469 CG For-Sale Unstable AKR1C3 29 40 CC[C@H](C)N(CC)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217845469 CG For-Sale Unstable PDS 46 33 COc1cccc(C(=O)N2CCNC[C@@H]2C)n1 ZINC000217845506 BC For-Sale Unstable ALS 43 33 CC[C@H](NC(=O)c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217845531 EF In-Stock Unstable CA2 24 44 CC[C@H](NC(=O)c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217845531 EF In-Stock Unstable PTGS2 24 49 CC[C@H](NC(=O)c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217845531 EF In-Stock Unstable BMP1 54 39 CC[C@H](NC(=O)c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217845531 EF In-Stock Unstable MMP13 41 44 CC[C@H](NC(=O)c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217845531 EF In-Stock Unstable TACR3 45 39 CC[C@H](NC(=O)c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217845531 EF In-Stock Unstable MMP3 42 39 CC[C@H](NC(=O)c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217845531 EF In-Stock Unstable MMP1 47 41 CC[C@H](NC(=O)c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217845531 EF In-Stock Unstable LOX1.1 43 37 CC[C@H](NC(=O)c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217845531 EF In-Stock Unstable UTS2 64 51 CC[C@H](NC(=O)c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217845531 EF In-Stock Unstable GPR88 0 40 COc1ccc(CN(C)CC(N)=O)cc1/C=C\C(=O)O ZINC000217845564 CC For-Sale Unstable PTGER2 28 43 COc1ccc(CN(C)CC(N)=O)cc1/C=C\C(=O)O ZINC000217845564 CC For-Sale Unstable PTGER4 0 43 COc1ccc(CN(C)CC(N)=O)cc1/C=C\C(=O)O ZINC000217845564 CC For-Sale Unstable DRTS_TRYCR 44 32 CC[C@@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)c1ccco1 ZINC000217845565 CF For-Sale Unstable ACE2 43 36 CC[C@@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)c1ccco1 ZINC000217845565 CF For-Sale Unstable XIAP 44 38 COc1ccc(OC)c(NC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217845573 GI For-Sale Unstable CYP1B1 40 40 COc1ccc(OC)c(NC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217845573 GI For-Sale Unstable MTNR1A 19 45 COc1ccc(OC)c(NC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217845573 GI For-Sale Unstable MTNR1B 20 48 COc1ccc(OC)c(NC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217845573 GI For-Sale Unstable ABCG2 21 42 COc1ccc(OC)c(NC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217845573 GI For-Sale Unstable AKR1C2 45 36 CC[C@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)c1ccco1 ZINC000217845649 CF For-Sale Unstable ACE2 43 36 CC[C@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)c1ccco1 ZINC000217845649 CF For-Sale Unstable XIAP 44 38 COc1ccc(C(=O)NCc2nc(-c3ccc(OC)cc3OC)no2)cc1 ZINC000217845681 FF In-Stock Unstable GRIN2B 22 42 COc1ccc(C(=O)NCc2nc(-c3ccc(OC)cc3OC)no2)cc1 ZINC000217845681 FF In-Stock Unstable HRH3 18 40 COc1ccc(C(=O)NCc2nc(-c3ccc(OC)cc3OC)no2)cc1 ZINC000217845681 FF In-Stock Unstable MT-ND1 24 42 C[C@@H](CO)NC(=O)c1ccccc1-c1ccc(-c2cnc(N)nc2)c(F)c1 ZINC000217845689 FF Annotated Unstable MTTP 84 35 ClC[C@@H]1CC(c2ccc3c(c2)OCO3)=NO1 ZINC000217845782 BE In-Stock Unstable DYRK1A 40 37 ClC[C@@H]1CC(c2ccc3c(c2)OCO3)=NO1 ZINC000217845782 BE In-Stock Unstable CLK1 41 37 ClC[C@@H]1CC(c2ccc3c(c2)OCO3)=NO1 ZINC000217845782 BE In-Stock Unstable CLK2 49 37 ClC[C@@H]1CC(c2ccc3c(c2)OCO3)=NO1 ZINC000217845782 BE In-Stock Unstable CLK4 74 37 ClC[C@@H]1CC(c2ccc3c(c2)OCO3)=NO1 ZINC000217845782 BE In-Stock Unstable LUCI_PHOPY 87 42 COc1ccc(C(=O)NCc2nc(-c3cccc(Br)c3)no2)cc1 ZINC000217845793 GG In-Stock Unstable KCNQ1 0 42 COc1ccc(C(=O)NCc2nc(-c3cccc(Br)c3)no2)cc1 ZINC000217845793 GG In-Stock Unstable NQO2 17 40 COc1ccc(C(=O)NCc2nc(-c3cccc(Br)c3)no2)cc1 ZINC000217845793 GG In-Stock Unstable MMP13 20 43 COc1ccc(C(=O)NCc2nc(-c3cccc(Br)c3)no2)cc1 ZINC000217845793 GG In-Stock Unstable MT-ND1 17 40 COCc1cc(=O)c(O)c([C@H](CC(N)=O)c2coc3ccc(OC)cc3c2=O)o1 ZINC000217845829 HD In-Stock Unstable ALDH2 53 32 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccoc1 ZINC000217845846 CF For-Sale Unstable HCRTR1 18 43 O=C(NC[C@H]1CCCN1c1ccccc1)c1ccoc1 ZINC000217845846 CF For-Sale Unstable PREP 15 40 C[C@@H](c1cccc(Cl)c1)N(C)CC[C@@H](O)c1ccccc1 ZINC000217845868 DI On-Demand Unstable ADRB1 24 41 C[C@@H](c1cccc(Cl)c1)N(C)CC[C@@H](O)c1ccccc1 ZINC000217845868 DI On-Demand Unstable ADRB3 37 41 C[C@@H](c1cccc(Cl)c1)N(C)CC[C@@H](O)c1ccccc1 ZINC000217845868 DI On-Demand Unstable AOC3 28 40 ClC[C@H]1CC(c2ccc3c(c2)OCO3)=NO1 ZINC000217845870 BE In-Stock Unstable DYRK1A 40 37 ClC[C@H]1CC(c2ccc3c(c2)OCO3)=NO1 ZINC000217845870 BE In-Stock Unstable CLK1 41 37 ClC[C@H]1CC(c2ccc3c(c2)OCO3)=NO1 ZINC000217845870 BE In-Stock Unstable CLK2 49 37 ClC[C@H]1CC(c2ccc3c(c2)OCO3)=NO1 ZINC000217845870 BE In-Stock Unstable CLK4 74 37 ClC[C@H]1CC(c2ccc3c(c2)OCO3)=NO1 ZINC000217845870 BE In-Stock Unstable LUCI_PHOPY 87 42 COc1ccc(C(=O)N(C)Cc2nc(-c3ccc(OC)cc3OC)no2)cc1 ZINC000217845871 GG In-Stock Unstable MT-ND1 23 42 COc1cc(C(=O)Nc2ccc(N3CCCC3)nc2)ccc1OCC(C)C ZINC000217845883 FH On-Demand Unstable PDGFRB 41 37 COc1cc(C(=O)Nc2ccc(N3CCCC3)nc2)ccc1OCC(C)C ZINC000217845883 FH On-Demand Unstable PTGER1 22 40 COc1cc(C(=O)Nc2ccc(N3CCCC3)nc2)ccc1OCC(C)C ZINC000217845883 FH On-Demand Unstable COLA 72 38 COc1cc(C(=O)Nc2ccc(N3CCCC3)nc2)ccc1OCC(C)C ZINC000217845883 FH On-Demand Unstable CPT1A 66 36 COc1cc(C(=O)Nc2ccc(N3CCCC3)nc2)ccc1OCC(C)C ZINC000217845883 FH On-Demand Unstable CPT2 45 34 COc1cc(C(=O)Nc2ccc(N3CCCC3)nc2)ccc1OCC(C)C ZINC000217845883 FH On-Demand Unstable PRNP 52 46 COc1cc(C(=O)Nc2ccc(N3CCCC3)nc2)ccc1OCC(C)C ZINC000217845883 FH On-Demand Unstable F3 41 35 COc1cc(C(=O)Nc2ccc(N3CCCC3)nc2)ccc1OCC(C)C ZINC000217845883 FH On-Demand Unstable CPT1B 53 35 COc1cc(C(=O)Nc2ccc(N3CCCC3)nc2)ccc1OCC(C)C ZINC000217845883 FH On-Demand Unstable ENPP1 58 33 COc1cc(C(=O)Nc2ccc(N3CCCC3)nc2)ccc1OCC(C)C ZINC000217845883 FH On-Demand Unstable DGAT1 52 44 COCc1cc(=O)c(O)c([C@@H](CC(N)=O)c2coc3ccc(OC)cc3c2=O)o1 ZINC000217845898 HD In-Stock Unstable ALDH2 53 32 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccoc1 ZINC000217845922 CF For-Sale Unstable HCRTR1 18 43 O=C(NC[C@@H]1CCCN1c1ccccc1)c1ccoc1 ZINC000217845922 CF For-Sale Unstable PREP 15 40 C[C@H](c1cccc(Cl)c1)N(C)CC[C@@H](O)c1ccccc1 ZINC000217845969 DI On-Demand Unstable ADRB1 24 41 C[C@H](c1cccc(Cl)c1)N(C)CC[C@@H](O)c1ccccc1 ZINC000217845969 DI On-Demand Unstable ADRB3 37 41 C[C@H](c1cccc(Cl)c1)N(C)CC[C@@H](O)c1ccccc1 ZINC000217845969 DI On-Demand Unstable AOC3 28 40 ClC[C@@H]1CC(c2ccco2)=NO1 ZINC000217845978 AE In-Stock Unstable LUCI_PHOPY 83 40 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217845993 DI In-Stock Unstable DRD4 42 32 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217845993 DI In-Stock Unstable PTGS2 0 40 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217845993 DI In-Stock Unstable DRD3 28 42 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217845993 DI In-Stock Unstable SCNN1A 47 41 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217845993 DI In-Stock Unstable GCGR 46 40 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217845993 DI In-Stock Unstable TBXAS1 17 41 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217845993 DI In-Stock Unstable PTAFR 23 48 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217845993 DI In-Stock Unstable BMP1 35 42 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217845993 DI In-Stock Unstable NQO2 21 43 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217845993 DI In-Stock Unstable TRPV1 0 46 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217845993 DI In-Stock Unstable CTSL 19 52 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217845993 DI In-Stock Unstable SCN2A 16 46 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217845993 DI In-Stock Unstable MTNR1A 56 43 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217845993 DI In-Stock Unstable MTNR1B 50 43 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217845993 DI In-Stock Unstable MMP3 17 41 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217845993 DI In-Stock Unstable MMP8 16 41 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217845993 DI In-Stock Unstable SLC6A5 25 45 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217845993 DI In-Stock Unstable CA9 18 43 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217845993 DI In-Stock Unstable MMP1 19 47 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217845993 DI In-Stock Unstable HDA106 0 53 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217845993 DI In-Stock Unstable VIPR2 0 40 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217845993 DI In-Stock Unstable UTS2 33 40 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217845993 DI In-Stock Unstable AP2S1 0 42 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217845993 DI In-Stock Unstable DUSP2 0 40 O=C(N/C=C/c1ccccc1Br)Nc1ccc(F)cc1 ZINC000217845994 EI For-Sale Anodyne MTCA1 19 42 O=C(N/C=C/c1ccccc1Br)Nc1ccc(F)cc1 ZINC000217845994 EI For-Sale Anodyne P96878_MYCTU 22 42 O=C1[C@H]2ON(c3ccccc3)[C@H](c3cccc([N+](=O)[O-])c3)[C@@H]2C(=O)N1c1ccc([N+](=O)[O-])cc1 ZINC000217846028 JH In-Stock Bother ACHE 18 71 CCC(CC)N(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217846037 CG For-Sale Unstable PDS 45 35 O=C(NC[C@H]1CCCN1c1ccccc1)c1cccc(I)c1 ZINC000217846044 HH For-Sale Unstable PREP 21 41 O=C(NC[C@H]1CCCN1c1ccccc1)c1cccc(I)c1 ZINC000217846044 HH For-Sale Unstable CCR2 15 41 ClC[C@H]1CC(c2ccco2)=NO1 ZINC000217846062 AE In-Stock Unstable LUCI_PHOPY 83 40 O=C(N/C=C/c1ccccc1Br)Nc1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217846110 GJ For-Sale Bother IMDH_CRYPV 24 45 O=C(N/C=C/c1ccccc1Br)Nc1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217846110 GJ For-Sale Bother BLM 0 46 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217846117 DG In-Stock Unstable HTR1A 39 50 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217846117 DG In-Stock Unstable ADRA2A 15 50 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217846117 DG In-Stock Unstable DRD2 49 48 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217846117 DG In-Stock Unstable DRD1 29 48 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217846117 DG In-Stock Unstable DRD4 54 44 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217846117 DG In-Stock Unstable ADRA1D 19 44 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217846117 DG In-Stock Unstable HTR2A 36 44 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217846117 DG In-Stock Unstable HTR2C 33 44 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217846117 DG In-Stock Unstable AVPR2 36 45 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217846117 DG In-Stock Unstable ADRA1A 28 42 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217846117 DG In-Stock Unstable ADRA1B 17 44 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217846117 DG In-Stock Unstable DRD3 77 48 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217846117 DG In-Stock Unstable AVPR1A 32 43 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217846117 DG In-Stock Unstable DRD5 21 48 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217846117 DG In-Stock Unstable PLD1 24 44 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217846117 DG In-Stock Unstable MMP1 18 40 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217846117 DG In-Stock Unstable TYRO3 28 42 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217846117 DG In-Stock Unstable NOD1 26 43 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217846117 DG In-Stock Unstable NOD2 41 43 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217846117 DG In-Stock Unstable AP2S1 0 46 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217846117 DG In-Stock Unstable ALPHA-1A 0 45 O=C1[C@H]2[C@@H](c3cccc([N+](=O)[O-])c3)N(c3ccccc3)O[C@H]2C(=O)N1c1ccc([N+](=O)[O-])cc1 ZINC000217846126 JH In-Stock Bother ACHE 18 71 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cccc(I)c1 ZINC000217846133 HH For-Sale Unstable PREP 21 41 O=C(NC[C@@H]1CCCN1c1ccccc1)c1cccc(I)c1 ZINC000217846133 HH For-Sale Unstable CCR2 15 41 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable TOP1 0 82 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable CNR1 21 62 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable PPARG 0 85 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable PPARA 0 56 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable PLA2G4C 0 47 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable FABP2 0 63 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable FABP4 32 85 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable PLA2G2C 0 43 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable PLA2G4A 0 53 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable LPAR1 23 49 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable PPARD 0 85 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable PLA2G4B 54 47 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable FAAH 25 71 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable PRKCA 15 43 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable EPHX2 32 66 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable CDC25C 0 51 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable PLCG1 0 40 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable Q6UB75_PIG 0 42 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable LPAR3 40 40 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable FABP3 66 85 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable FABP5 28 85 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable LOX1.1 17 77 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable FFAR1 0 77 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable ENPP2 19 40 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable FABP1 28 85 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable SLC22A20 0 63 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable LPAR4 0 40 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable LPAR5 0 40 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable ACAT 0 45 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable LASR 52 35 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable NOD1 42 36 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable SAE1 0 40 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable OXER1 39 53 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable CQSS 60 37 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable SLCO2A1 54 40 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable LPAR6 0 40 CCCCCC/C=C\CCCC(=O)CCCCCC(=O)O ZINC000217846142 CK Annotated Unstable EST1 0 42 O=[N+]([O-])c1ccccc1C1=NO[C@@H](CCl)C1 ZINC000217846196 BE In-Stock Unstable LUCI_PHOPY 79 46 CCOc1ccc(CNC(=O)c2ccccc2Cl)cc1OCC ZINC000217846211 EI In-Stock Unstable ECR 45 35 CCOc1ccc(CNC(=O)c2ccccc2Cl)cc1OCC ZINC000217846211 EI In-Stock Unstable PDE6A 40 31 CCOc1ccc(CNC(=O)c2ccccc2Cl)cc1OCC ZINC000217846211 EI In-Stock Unstable U38 0 47 CCOc1ccc(CNC(=O)c2ccccc2Cl)cc1OCC ZINC000217846211 EI In-Stock Unstable HCN1 49 37 CCOc1ccc(CNC(=O)c2ccccc2Cl)cc1OCC ZINC000217846211 EI In-Stock Unstable HCN4 46 36 CCOc1ccc(CNC(=O)c2ccccc2Cl)cc1OCC ZINC000217846211 EI In-Stock Unstable KCNK3 39 41 CCOc1ccc(CNC(=O)c2ccccc2Cl)cc1OCC ZINC000217846211 EI In-Stock Unstable KCNK9 25 41 CCOc1ccc(CNC(=O)c2ccccc2Cl)cc1OCC ZINC000217846211 EI In-Stock Unstable PDS 43 38 CCc1ccc(-c2nc(CC(=O)Nc3ccc(N4CCCC4)nc3)cs2)cc1 ZINC000217846214 GJ On-Demand Unstable DGAT1 37 41 CCc1ccc(-c2nc(CC(=O)Nc3ccc(N4CCCC4)nc3)cs2)cc1 ZINC000217846214 GJ On-Demand Unstable SLC27A1 46 39 COc1cc([N+](=O)[O-])ccc1NC(=O)N/C=C/c1ccccc1Br ZINC000217846220 GI For-Sale Unstable EPHX1 0 53 COc1cc([N+](=O)[O-])ccc1NC(=O)N/C=C/c1ccccc1Br ZINC000217846220 GI For-Sale Unstable KCNMA1 24 53 O=C(c1ccc(C(F)(F)F)nc1)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217846224 HG In-Stock Unstable BMP1 21 43 O=C(CNC(=O)OCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217846233 FF For-Sale Unstable CELA1 20 42 O=C(CNC(=O)OCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217846233 FF For-Sale Unstable GRIN2B 18 40 O=C(CNC(=O)OCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217846233 FF For-Sale Unstable CTRA_BOVIN 53 32 O=C(CNC(=O)OCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217846233 FF For-Sale Unstable CTSB 32 41 O=C(CNC(=O)OCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217846233 FF For-Sale Unstable CTSG 41 32 O=C(CNC(=O)OCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217846233 FF For-Sale Unstable CTSK 29 41 O=C(CNC(=O)OCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217846233 FF For-Sale Unstable PREP 43 42 O=C(CNC(=O)OCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217846233 FF For-Sale Unstable CAPNS1 46 31 O=C(CNC(=O)OCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217846233 FF For-Sale Unstable CELA2A 41 32 O=C(CNC(=O)OCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217846233 FF For-Sale Unstable CTSS 16 40 O=C(CNC(=O)OCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217846233 FF For-Sale Unstable CAPN1 48 38 O=C(CNC(=O)OCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217846233 FF For-Sale Unstable CAPN2 75 38 O=C(CNC(=O)OCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217846233 FF For-Sale Unstable KLK5 40 38 O=C(CNC(=O)OCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217846233 FF For-Sale Unstable NPR 61 35 O=C(CNC(=O)OCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217846233 FF For-Sale Unstable NPFFR1 40 32 O=C(CNC(=O)OCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217846233 FF For-Sale Unstable SLC12A5 49 36 COc1ccc(Cn2cccnc2=O)cc1/C=C\C(=O)O ZINC000217846234 CD For-Sale Unstable PTGER2 39 47 COc1ccc(Cn2cccnc2=O)cc1/C=C\C(=O)O ZINC000217846234 CD For-Sale Unstable PTGER4 25 47 COc1ccc(Cn2cccnc2=O)cc1/C=C\C(=O)O ZINC000217846234 CD For-Sale Unstable PTGER3 31 47 O=[N+]([O-])c1ccccc1C1=NO[C@H](CCl)C1 ZINC000217846266 BE In-Stock Unstable LUCI_PHOPY 79 46 O=C(c1ccc(C(F)(F)F)nc1)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217846277 HG In-Stock Unstable BMP1 21 43 O=C(CNC(=O)OCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217846295 FF For-Sale Unstable CELA1 20 42 O=C(CNC(=O)OCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217846295 FF For-Sale Unstable GRIN2B 18 40 O=C(CNC(=O)OCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217846295 FF For-Sale Unstable CTRA_BOVIN 53 32 O=C(CNC(=O)OCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217846295 FF For-Sale Unstable CTSB 32 41 O=C(CNC(=O)OCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217846295 FF For-Sale Unstable CTSG 41 32 O=C(CNC(=O)OCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217846295 FF For-Sale Unstable CTSK 29 41 O=C(CNC(=O)OCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217846295 FF For-Sale Unstable PREP 43 42 O=C(CNC(=O)OCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217846295 FF For-Sale Unstable CAPNS1 46 31 O=C(CNC(=O)OCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217846295 FF For-Sale Unstable CELA2A 41 32 O=C(CNC(=O)OCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217846295 FF For-Sale Unstable CTSS 16 40 O=C(CNC(=O)OCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217846295 FF For-Sale Unstable CAPN1 48 38 O=C(CNC(=O)OCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217846295 FF For-Sale Unstable CAPN2 75 38 O=C(CNC(=O)OCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217846295 FF For-Sale Unstable KLK5 40 38 O=C(CNC(=O)OCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217846295 FF For-Sale Unstable NPR 61 35 O=C(CNC(=O)OCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217846295 FF For-Sale Unstable NPFFR1 40 32 O=C(CNC(=O)OCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217846295 FF For-Sale Unstable SLC12A5 49 36 COc1ccccc1CCCNC(=O)c1ccccc1Cl ZINC000217846317 DH In-Stock Unstable DRD2 35 43 COc1ccccc1CCCNC(=O)c1ccccc1Cl ZINC000217846317 DH In-Stock Unstable DRD1 0 40 COc1ccccc1CCCNC(=O)c1ccccc1Cl ZINC000217846317 DH In-Stock Unstable DRD3 49 41 COc1ccccc1CCCNC(=O)c1ccccc1Cl ZINC000217846317 DH In-Stock Unstable HTR4 22 42 COc1ccccc1CCCNC(=O)c1ccccc1Cl ZINC000217846317 DH In-Stock Unstable ECR 41 44 COc1ccccc1CCCNC(=O)c1ccccc1Cl ZINC000217846317 DH In-Stock Unstable KCNA3 41 42 COc1ccccc1CCCNC(=O)c1ccccc1Cl ZINC000217846317 DH In-Stock Unstable MTNR1B 46 46 COc1ccccc1CCCNC(=O)c1ccccc1Cl ZINC000217846317 DH In-Stock Unstable SLC6A5 44 41 COc1ccccc1CCCNC(=O)c1ccccc1Cl ZINC000217846317 DH In-Stock Unstable TYRO3 17 43 O=C(N/C=C/c1ccccc1Br)Nc1ccc([N+](=O)[O-])cc1 ZINC000217846318 FI For-Sale Bother NADE 0 40 O=C(N/C=C/c1ccccc1Br)Nc1ccc([N+](=O)[O-])cc1 ZINC000217846318 FI For-Sale Bother NMBR 41 31 O=C(N/C=C/c1ccccc1Br)Nc1ccc([N+](=O)[O-])cc1 ZINC000217846318 FI For-Sale Bother MTCA1 23 40 O=C(N/C=C/c1ccccc1Br)Nc1ccc([N+](=O)[O-])cc1 ZINC000217846318 FI For-Sale Bother P96878_MYCTU 26 40 O=[N+]([O-])c1cccc(C2=NO[C@@H](CCl)C2)c1 ZINC000217846373 BE In-Stock Unstable LUCI_PHOPY 87 53 O=C(N/C=C/c1ccccc1Br)Nc1cccc([N+](=O)[O-])c1 ZINC000217846395 FI For-Sale Bother DDX3X 0 51 O=C(N/C=C/c1ccccc1Br)Nc1cccc([N+](=O)[O-])c1 ZINC000217846395 FI For-Sale Bother HISG 0 40 O=C(N/C=C/c1ccccc1Br)Nc1cccc([N+](=O)[O-])c1 ZINC000217846395 FI For-Sale Bother OSIGBA0132E09-OSIGBA0108L24.11 0 42 O=C(CCl)Cc1ccc(Br)cc1F ZINC000217846403 CF For-Sale Unstable AKR1B1 15 41 O=C(NC[C@H]1CCCN1c1ccccc1)Nc1ccc(Cl)c(Cl)c1 ZINC000217846406 FJ For-Sale Unstable NPY2R 42 37 O=C(NC[C@H]1CCCN1c1ccccc1)Nc1ccc(Cl)c(Cl)c1 ZINC000217846406 FJ For-Sale Unstable CCR3 53 38 O=C(NC[C@H]1CCCN1c1ccccc1)Nc1ccc(Cl)c(Cl)c1 ZINC000217846406 FJ For-Sale Unstable RAF1 19 40 O=C(NC[C@H]1CCCN1c1ccccc1)Nc1ccc(Cl)c(Cl)c1 ZINC000217846406 FJ For-Sale Unstable EPHX2 27 48 O=C(NC[C@H]1CCCN1c1ccccc1)Nc1ccc(Cl)c(Cl)c1 ZINC000217846406 FJ For-Sale Unstable MCHR1 19 43 CCOc1ccc(CCCNC(=O)c2ccccc2Cl)cc1 ZINC000217846407 DI In-Stock Unstable SCNN1A 45 37 CCOc1ccc(CCCNC(=O)c2ccccc2Cl)cc1 ZINC000217846407 DI In-Stock Unstable SDH1 0 52 CCOc1ccc(CCCNC(=O)c2ccccc2Cl)cc1 ZINC000217846407 DI In-Stock Unstable ECR 49 45 CCOc1ccc(CCCNC(=O)c2ccccc2Cl)cc1 ZINC000217846407 DI In-Stock Unstable SCN2A 29 49 CCOc1ccc(CCCNC(=O)c2ccccc2Cl)cc1 ZINC000217846407 DI In-Stock Unstable FAAH 19 40 CCOc1ccc(CCCNC(=O)c2ccccc2Cl)cc1 ZINC000217846407 DI In-Stock Unstable SLC6A5 37 47 CCOc1ccc(CCCNC(=O)c2ccccc2Cl)cc1 ZINC000217846407 DI In-Stock Unstable CRTM 50 39 CCOc1ccc(CCCNC(=O)c2ccccc2Cl)cc1 ZINC000217846407 DI In-Stock Unstable HCN1 48 32 CCOc1ccc(CCCNC(=O)c2ccccc2Cl)cc1 ZINC000217846407 DI In-Stock Unstable HCN4 40 31 CCOc1ccc(CCCNC(=O)c2ccccc2Cl)cc1 ZINC000217846407 DI In-Stock Unstable E3UJZ5_SPOLI 37 45 CCOc1ccc(CCCNC(=O)c2ccccc2Cl)cc1 ZINC000217846407 DI In-Stock Unstable PDS 41 37 O=C(Cc1cccc(C(F)(F)F)c1)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217846411 IH In-Stock Unstable CCR2 44 43 O=C(NC[C@@H]1CCCN1c1ccccc1)Nc1ccc(Cl)c(Cl)c1 ZINC000217846473 FJ For-Sale Unstable NPY2R 42 37 O=C(NC[C@@H]1CCCN1c1ccccc1)Nc1ccc(Cl)c(Cl)c1 ZINC000217846473 FJ For-Sale Unstable CCR3 53 38 O=C(NC[C@@H]1CCCN1c1ccccc1)Nc1ccc(Cl)c(Cl)c1 ZINC000217846473 FJ For-Sale Unstable RAF1 19 40 O=C(NC[C@@H]1CCCN1c1ccccc1)Nc1ccc(Cl)c(Cl)c1 ZINC000217846473 FJ For-Sale Unstable EPHX2 27 48 O=C(NC[C@@H]1CCCN1c1ccccc1)Nc1ccc(Cl)c(Cl)c1 ZINC000217846473 FJ For-Sale Unstable MCHR1 19 43 O=[N+]([O-])c1cccc(C2=NO[C@H](CCl)C2)c1 ZINC000217846484 BE In-Stock Unstable LUCI_PHOPY 87 53 O=C(O)/C=C\c1cc(CN2C(=O)CCC2=O)ccc1F ZINC000217846488 CD For-Sale Unstable PTGER3 35 40 O=C(Cc1cccc(C(F)(F)F)c1)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217846490 IH In-Stock Unstable CCR2 44 43 CCCOc1ccccc1CCCNC(=O)c1ccccc1Cl ZINC000217846500 EI In-Stock Unstable MTNR1B 47 40 COc1ccc(CNC[C@@](C)(O)CSC)cc1 ZINC000217846507 CD On-Demand Unstable KCNJ2 0 41 O=C(OCc1ccccc1)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217846559 GG In-Stock Unstable GRIN2B 19 44 O=C(OCc1ccccc1)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217846559 GG In-Stock Unstable BMP1 22 43 O=C(OCc1ccccc1)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217846559 GG In-Stock Unstable COLA 75 38 O=C(OCc1ccccc1)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217846559 GG In-Stock Unstable CPT1A 62 38 O=C(OCc1ccccc1)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217846559 GG In-Stock Unstable PREP 28 40 O=C(NC[C@@H]1CCCN1c1ccccc1)Nc1ccccc1 ZINC000217846564 CG For-Sale Unstable LPL 45 37 O=C(NC[C@@H]1CCCN1c1ccccc1)Nc1ccccc1 ZINC000217846564 CG For-Sale Unstable CCR3 44 44 O=C(NC[C@@H]1CCCN1c1ccccc1)Nc1ccccc1 ZINC000217846564 CG For-Sale Unstable EPHX2 35 45 O=[N+]([O-])c1ccc(C2=NO[C@@H](CCl)C2)cc1 ZINC000217846582 BE In-Stock Unstable LUCI_PHOPY 92 68 O=C(O)/C=C\c1ccc(OCCN2CCCCC2=O)cc1 ZINC000217846583 CE For-Sale Unstable LTA4H 42 38 O=C(O)/C=C\c1ccc(OCCN2CCCCC2=O)cc1 ZINC000217846583 CE For-Sale Unstable HRH3 30 49 O=C(O)/C=C\c1ccc(OCCN2CCCCC2=O)cc1 ZINC000217846583 CE For-Sale Unstable PSMB2 48 38 O=C(O)/C=C\c1ccc(OCCN2CCCCC2=O)cc1 ZINC000217846583 CE For-Sale Unstable PSMB1 43 38 COc1ccc(CNC[C@](C)(O)CSC)cc1 ZINC000217846602 CD On-Demand Unstable KCNJ2 0 41 CC1CCN(c2ccc([C@@H](C)NC(=O)c3ccccc3Cl)cc2)CC1 ZINC000217846622 FK In-Stock Unstable PRCP 23 41 COc1cccc(OC[C@@H]2CCCN(C(=O)c3cc(=O)cc(C)o3)C2)c1 ZINC000217846626 FF In-Stock Unstable DRD4 40 32 O=[N+]([O-])c1ccc(C2=NO[C@H](CCl)C2)cc1 ZINC000217846655 BE In-Stock Unstable LUCI_PHOPY 92 68 COc1ccc(/C=C\C(=O)O)cc1CN1CCCCC1=O ZINC000217846657 CE For-Sale Unstable PTGER2 15 44 O=C(OCc1ccccc1)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217846663 GG In-Stock Unstable GRIN2B 21 49 O=C(OCc1ccccc1)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217846663 GG In-Stock Unstable BMP1 23 43 O=C(OCc1ccccc1)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217846663 GG In-Stock Unstable COLA 75 38 O=C(OCc1ccccc1)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217846663 GG In-Stock Unstable CPT1A 69 38 O=C(OCc1ccccc1)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217846663 GG In-Stock Unstable PREP 36 41 O=C(NC[C@H]1CCCN1c1ccccc1)Nc1ccccc1 ZINC000217846664 CG For-Sale Unstable LPL 45 37 O=C(NC[C@H]1CCCN1c1ccccc1)Nc1ccccc1 ZINC000217846664 CG For-Sale Unstable CCR3 44 44 O=C(NC[C@H]1CCCN1c1ccccc1)Nc1ccccc1 ZINC000217846664 CG For-Sale Unstable EPHX2 35 45 CC1CCN(c2ccc([C@H](C)NC(=O)c3ccccc3Cl)cc2)CC1 ZINC000217846695 FK In-Stock Unstable PRCP 23 41 COc1cccc(OC[C@H]2CCCN(C(=O)c3cc(=O)cc(C)o3)C2)c1 ZINC000217846696 FF In-Stock Unstable DRD4 40 32 COc1ccccc1CNC[C@@](C)(O)CSC ZINC000217846721 CD On-Demand Unstable PHES 0 42 COc1ccccc1CNC[C@@](C)(O)CSC ZINC000217846721 CD On-Demand Unstable GPM3 0 49 COc1ccc(Cn2nc(C)nc2C)cc1/C=C\C(=O)O ZINC000217846741 CE For-Sale Unstable PTGER2 32 41 COc1ccc(Cn2nc(C)nc2C)cc1/C=C\C(=O)O ZINC000217846741 CE For-Sale Unstable PTGER4 20 41 COc1ccc(Cn2nc(C)nc2C)cc1/C=C\C(=O)O ZINC000217846741 CE For-Sale Unstable PTGER3 19 40 CCOC(=O)N1CCN(C(=O)CC/C(C)=C/Cc2c(O)c3c(c(C)c2OC)COC3=O)CC1 ZINC000217846754 JF In-Stock Unstable IMPDH1 0 70 CCOC(=O)N1CCN(C(=O)CC/C(C)=C/Cc2c(O)c3c(c(C)c2OC)COC3=O)CC1 ZINC000217846754 JF In-Stock Unstable IMPDH2 0 70 O=C(O)[C@@H]1CC(Cc2ccccc2)=NO1 ZINC000217846755 BD In-Stock Unstable LUCI_PHOPY 59 33 O=C(NC[C@H]1CCCN1c1ccccc1)Nc1ccc(Cl)cc1 ZINC000217846767 EI For-Sale Unstable CCR3 25 43 O=C(NC[C@H]1CCCN1c1ccccc1)Nc1ccc(Cl)cc1 ZINC000217846767 EI For-Sale Unstable EPHX2 42 43 O=C(NC[C@H]1CCCN1c1ccccc1)Nc1ccc(Cl)cc1 ZINC000217846767 EI For-Sale Unstable MCHR1 15 47 O=C(NC[C@H]1CCCN1c1ccccc1)Nc1ccc(Cl)cc1 ZINC000217846767 EI For-Sale Unstable FPR2 46 45 COc1ccccc1CNC[C@](C)(O)CSC ZINC000217846809 CD On-Demand Unstable PHES 0 42 COc1ccccc1CNC[C@](C)(O)CSC ZINC000217846809 CD On-Demand Unstable GPM3 0 49 O=C(O)[C@H]1CC(Cc2ccccc2)=NO1 ZINC000217846842 BD In-Stock Unstable LUCI_PHOPY 59 33 O=C(NC[C@@H]1CCCN1c1ccccc1)Nc1ccc(Cl)cc1 ZINC000217846853 EI For-Sale Unstable CCR3 25 43 O=C(NC[C@@H]1CCCN1c1ccccc1)Nc1ccc(Cl)cc1 ZINC000217846853 EI For-Sale Unstable EPHX2 42 43 O=C(NC[C@@H]1CCCN1c1ccccc1)Nc1ccc(Cl)cc1 ZINC000217846853 EI For-Sale Unstable MCHR1 15 47 O=C(NC[C@@H]1CCCN1c1ccccc1)Nc1ccc(Cl)cc1 ZINC000217846853 EI For-Sale Unstable FPR2 46 45 O=C(N/C=C/c1ccccc1Br)N1CCN(c2ccc(F)cc2)CC1 ZINC000217846859 HI For-Sale Unstable AKR1C3 0 43 CCc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217846903 CH For-Sale Unstable OPRL1 0 42 CCc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217846903 CH For-Sale Unstable PTGER2 27 49 CCc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217846903 CH For-Sale Unstable PPARA 19 40 CCc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217846903 CH For-Sale Unstable PTGER4 44 48 CCc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217846903 CH For-Sale Unstable PTPN2 0 40 CCc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217846903 CH For-Sale Unstable PTGER3 38 60 CCc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217846903 CH For-Sale Unstable CDC25B 22 42 CCc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217846903 CH For-Sale Unstable PTGDR 0 60 CCc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217846903 CH For-Sale Unstable FFAR1 42 44 CCc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217846903 CH For-Sale Unstable FFAR4 52 42 CCCCCCCCCN[C@@H](CC)CCO ZINC000217846910 BG For-Sale Unstable CQSS 40 31 CCC[C@@](C)(O)CNC(=O)c1cccc(Cl)c1F ZINC000217846944 CF On-Demand Unstable ECR 44 41 CCC[C@@](C)(O)CNC(=O)c1cccc(Cl)c1F ZINC000217846944 CF On-Demand Unstable E3UJZ5_SPOLI 42 40 CCc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217846992 CH For-Sale Unstable MAOB 20 55 CCc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217846992 CH For-Sale Unstable PTGER2 38 47 CCc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217846992 CH For-Sale Unstable PPARA 17 41 CCc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217846992 CH For-Sale Unstable PTGER4 31 43 CCc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217846992 CH For-Sale Unstable PTGER3 16 46 CCc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217846992 CH For-Sale Unstable PTGDR 0 46 CCc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217846992 CH For-Sale Unstable FFAR1 40 43 CCc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217846992 CH For-Sale Unstable AKR1C3 33 43 CCc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217846992 CH For-Sale Unstable FFAR4 43 35 CCCCCCCCCN[C@H](CC)CCO ZINC000217847000 BG For-Sale Unstable CQSS 40 31 CCC[C@](C)(O)CNC(=O)c1cccc(Cl)c1F ZINC000217847026 CF On-Demand Unstable ECR 44 41 CCC[C@](C)(O)CNC(=O)c1cccc(Cl)c1F ZINC000217847026 CF On-Demand Unstable E3UJZ5_SPOLI 42 40 CCc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217847069 CH For-Sale Unstable ALOX5 26 50 CCc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217847069 CH For-Sale Unstable MAOB 68 48 CCc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217847069 CH For-Sale Unstable PPARG 19 41 CCc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217847069 CH For-Sale Unstable PTGER2 23 50 CCc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217847069 CH For-Sale Unstable PPARA 22 40 CCc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217847069 CH For-Sale Unstable LTA4H 24 41 CCc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217847069 CH For-Sale Unstable PTGER4 30 47 CCc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217847069 CH For-Sale Unstable PTPN2 0 40 CCc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217847069 CH For-Sale Unstable PTGER3 35 48 CCc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217847069 CH For-Sale Unstable LTB4R 34 45 CCc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217847069 CH For-Sale Unstable NR1H4 65 35 CCc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217847069 CH For-Sale Unstable GYS1 47 35 CCc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217847069 CH For-Sale Unstable PTGDR 0 48 CCc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217847069 CH For-Sale Unstable HCAR2 0 42 CCc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217847069 CH For-Sale Unstable FFAR1 86 47 CCc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217847069 CH For-Sale Unstable AKR1C3 37 48 CCc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217847069 CH For-Sale Unstable FFAR4 46 45 CCOc1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217847072 FJ For-Sale Unstable CA1 42 40 CCOc1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217847072 FJ For-Sale Unstable CA12 18 40 CCOc1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217847072 FJ For-Sale Unstable CA9 19 40 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable F2 69 47 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable ACE 53 53 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable LHCGR 47 49 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable AGTR1 34 45 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable SSTR2 81 42 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable OPRM1 68 68 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable OPRD1 50 65 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable OPRK1 0 65 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable CELA1 47 35 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable ELANE 57 38 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable MME 42 51 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable EDNRB 51 48 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable EDNRA 62 49 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable TACR1 52 57 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable TRHR 70 36 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable AGTR2 0 40 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable HLA-DRB3 45 33 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable MC4R 58 46 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable CMA1 39 42 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable CTRA_BOVIN 63 34 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable BMP1 46 45 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable TACR2 23 48 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable XPNPEP1 0 42 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable CTSB 26 41 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable TRY1_BOVIN 97 36 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable CCKAR 122 51 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable NTSR1 185 65 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable NTSR2 120 45 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable CTSG 44 34 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable BRS3 26 42 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable NPFFR2 48 47 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable TIMP3 17 47 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable C3AR1 31 59 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable HLA-A 98 59 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable NMBR 34 43 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable MC3R 76 43 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable MC5R 85 38 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable MMP2 29 46 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable MMP8 43 45 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable MMP14 26 44 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable GRPR 81 41 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable ECE1 66 49 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable HLA-DRB1 74 37 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable CELA2A 53 34 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable REN 39 58 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable REN1 81 46 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable LNPEP 32 47 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable LGMN 55 34 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable MMP11 95 43 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable SORT1 67 45 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable PEPD 0 42 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable XPNPEP2 0 42 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable CCKBR 93 63 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable GHSR 72 56 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable CAPN1 39 45 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable MMP9 29 47 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable CTRC 34 42 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable CAPN2 63 41 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable MC1R 107 43 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable ADAM9 41 42 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable NS3 0 42 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable LAP3 18 42 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable C5AR1 55 64 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable MMP7 28 43 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable MARS 42 35 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable TPP2 42 47 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable MMP1 26 45 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable KLK1 25 48 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable FPR1 27 45 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable NPR 44 49 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable XIAP 65 50 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable MAGI3 0 44 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable SLC15A2 0 45 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable KISS1R 90 42 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable ERAP2 44 44 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable PSMB8 26 41 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable Q9N6S8_PLAFA 26 51 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable ERAP1 0 44 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable BRCA1 69 39 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable NPFFR1 20 47 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable NMUR2 0 45 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable LASB 0 56 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable NMUR1 0 45 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable UBE2I 0 42 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable CD36 0 45 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable CBX7 0 45 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable TMPRSS11D 54 38 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable PSMB9 0 41 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable HPN 20 40 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable HGFAC 0 40 CC[C@H](C)[C@H](N)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(N)=O ZINC000217847078 KD Annotated Unstable DSBA 0 56 O=C(O)/C=C\c1cccc(COc2ccccc2F)c1 ZINC000217847145 CH For-Sale Unstable MAOB 15 45 O=C(O)/C=C\c1cccc(COc2ccccc2F)c1 ZINC000217847145 CH For-Sale Unstable PTGER2 26 52 O=C(O)/C=C\c1cccc(COc2ccccc2F)c1 ZINC000217847145 CH For-Sale Unstable PPIA 42 34 O=C(O)/C=C\c1cccc(COc2ccccc2F)c1 ZINC000217847145 CH For-Sale Unstable PTGER1 63 43 O=C(O)/C=C\c1cccc(COc2ccccc2F)c1 ZINC000217847145 CH For-Sale Unstable PTGER4 41 48 O=C(O)/C=C\c1cccc(COc2ccccc2F)c1 ZINC000217847145 CH For-Sale Unstable CXCL8 17 41 O=C(O)/C=C\c1cccc(COc2ccccc2F)c1 ZINC000217847145 CH For-Sale Unstable PTGER3 30 52 O=C(O)/C=C\c1cccc(COc2ccccc2F)c1 ZINC000217847145 CH For-Sale Unstable LTB4R 17 45 O=C(O)/C=C\c1cccc(COc2ccccc2F)c1 ZINC000217847145 CH For-Sale Unstable HCAR2 0 45 O=C(O)/C=C\c1cccc(COc2ccccc2F)c1 ZINC000217847145 CH For-Sale Unstable AKR1C3 42 57 COc1ccc(C(=O)NC[C@@H]2CCCN3CCCC[C@H]23)cc1-n1cccn1 ZINC000217847159 FF In-Stock Unstable FAP 0 40 COc1ccc(C(=O)NC[C@@H]2CCCN3CCCC[C@H]23)cc1-n1cccn1 ZINC000217847159 FF In-Stock Unstable ACKR3 52 35 O=C(O)/C=C\c1cc(F)ccc1COc1ccccc1F ZINC000217847222 CH For-Sale Unstable PTGER2 16 51 O=C(O)/C=C\c1cc(F)ccc1COc1ccccc1F ZINC000217847222 CH For-Sale Unstable PTGER1 30 43 O=C(O)/C=C\c1cc(F)ccc1COc1ccccc1F ZINC000217847222 CH For-Sale Unstable PTGER4 28 48 O=C(O)/C=C\c1cc(F)ccc1COc1ccccc1F ZINC000217847222 CH For-Sale Unstable CXCL8 18 41 O=C(O)/C=C\c1cc(F)ccc1COc1ccccc1F ZINC000217847222 CH For-Sale Unstable FABP4 17 42 O=C(O)/C=C\c1cc(F)ccc1COc1ccccc1F ZINC000217847222 CH For-Sale Unstable PTGER3 26 48 O=C(O)/C=C\c1cc(F)ccc1COc1ccccc1F ZINC000217847222 CH For-Sale Unstable PTGDR 0 40 O=C(O)/C=C\c1cc(F)ccc1COc1ccccc1F ZINC000217847222 CH For-Sale Unstable AKR1C3 31 47 Cc1c(Cl)cccc1C(=O)N1CCn2nc(CO)cc2C1 ZINC000217847267 DD In-Stock Unstable P2RX7 55 42 CC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217847278 FI For-Sale Unstable MTCA1 19 45 CC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217847278 FI For-Sale Unstable P96878_MYCTU 18 45 CC(=O)OC(C)(C)C(=O)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217847279 FD In-Stock Unstable BMP1 18 43 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCc1ccccc1 ZINC000217847281 IH In-Stock Unstable TOP1 0 45 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCc1ccccc1 ZINC000217847281 IH In-Stock Unstable HTR7 20 40 O=C(O)/C=C\c1cc(COc2ccccc2F)ccc1F ZINC000217847301 CH For-Sale Unstable PTGER2 24 51 O=C(O)/C=C\c1cc(COc2ccccc2F)ccc1F ZINC000217847301 CH For-Sale Unstable PTGER1 61 43 O=C(O)/C=C\c1cc(COc2ccccc2F)ccc1F ZINC000217847301 CH For-Sale Unstable PTGER4 45 50 O=C(O)/C=C\c1cc(COc2ccccc2F)ccc1F ZINC000217847301 CH For-Sale Unstable PTGER3 36 51 O=C(O)/C=C\c1cc(COc2ccccc2F)ccc1F ZINC000217847301 CH For-Sale Unstable PTGDR 0 45 O=C(O)/C=C\c1cc(COc2ccccc2F)ccc1F ZINC000217847301 CH For-Sale Unstable AKR1C3 32 47 C[C@@H](c1ccccc1F)N(C)CC[C@@H](O)c1ccccc1 ZINC000217847322 CH On-Demand Unstable AOC3 22 40 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCc1ccccc1 ZINC000217847359 IH In-Stock Unstable TOP1 0 45 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCc1ccccc1 ZINC000217847359 IH In-Stock Unstable HTR7 20 40 CC[C@@H](C)N(C)CCN[C@@H]1CCc2cc(O)ccc21 ZINC000217847360 CF For-Sale Unstable STS 47 33 CC(=O)OC(C)(C)C(=O)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217847361 FD In-Stock Unstable BMP1 18 43 COc1cccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217847364 EG For-Sale Unstable HTR1A 18 41 COc1cccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217847364 EG For-Sale Unstable DRD4 43 33 COc1cccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217847364 EG For-Sale Unstable HRH2 27 46 COc1cccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217847364 EG For-Sale Unstable DRD3 16 40 COc1cccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217847364 EG For-Sale Unstable PTGER3 17 45 COc1cccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217847364 EG For-Sale Unstable NPY1R 53 41 COc1cccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217847364 EG For-Sale Unstable CCKAR 49 47 COc1cccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217847364 EG For-Sale Unstable P2RY1 19 42 COc1cccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217847364 EG For-Sale Unstable CCR3 80 54 COc1cccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217847364 EG For-Sale Unstable MTNR1A 48 41 COc1cccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217847364 EG For-Sale Unstable MTNR1B 52 41 COc1cccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217847364 EG For-Sale Unstable SOAT1 18 43 COc1cccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217847364 EG For-Sale Unstable CCKBR 47 47 COc1cccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217847364 EG For-Sale Unstable EPHX2 40 47 COc1cccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217847364 EG For-Sale Unstable CHRNA10 41 41 COc1cccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217847364 EG For-Sale Unstable MCHR1 25 51 COc1cccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217847364 EG For-Sale Unstable ACKR3 64 33 O=C(O)/C=C\c1cccc(COc2ccccc2Cl)c1 ZINC000217847381 CI For-Sale Unstable EGFR 23 40 O=C(O)/C=C\c1cccc(COc2ccccc2Cl)c1 ZINC000217847381 CI For-Sale Unstable MAOB 26 42 O=C(O)/C=C\c1cccc(COc2ccccc2Cl)c1 ZINC000217847381 CI For-Sale Unstable PTGER2 26 55 O=C(O)/C=C\c1cccc(COc2ccccc2Cl)c1 ZINC000217847381 CI For-Sale Unstable PPIA 42 34 O=C(O)/C=C\c1cccc(COc2ccccc2Cl)c1 ZINC000217847381 CI For-Sale Unstable ERBB2 32 40 O=C(O)/C=C\c1cccc(COc2ccccc2Cl)c1 ZINC000217847381 CI For-Sale Unstable PTGER1 64 43 O=C(O)/C=C\c1cccc(COc2ccccc2Cl)c1 ZINC000217847381 CI For-Sale Unstable PTGER4 42 48 O=C(O)/C=C\c1cccc(COc2ccccc2Cl)c1 ZINC000217847381 CI For-Sale Unstable FABP4 15 42 O=C(O)/C=C\c1cccc(COc2ccccc2Cl)c1 ZINC000217847381 CI For-Sale Unstable PTGER3 29 55 O=C(O)/C=C\c1cccc(COc2ccccc2Cl)c1 ZINC000217847381 CI For-Sale Unstable LTB4R 19 45 O=C(O)/C=C\c1cccc(COc2ccccc2Cl)c1 ZINC000217847381 CI For-Sale Unstable NR1H4 45 40 O=C(O)/C=C\c1cccc(COc2ccccc2Cl)c1 ZINC000217847381 CI For-Sale Unstable 17HSDCL 0 43 O=C(O)/C=C\c1cccc(COc2ccccc2Cl)c1 ZINC000217847381 CI For-Sale Unstable FABP5 29 42 O=C(O)/C=C\c1cccc(COc2ccccc2Cl)c1 ZINC000217847381 CI For-Sale Unstable FFAR1 30 40 O=C(O)/C=C\c1cccc(COc2ccccc2Cl)c1 ZINC000217847381 CI For-Sale Unstable AKR1C3 40 53 O=C(O)/C=C\c1cccc(COc2ccccc2Cl)c1 ZINC000217847381 CI For-Sale Unstable ADCYAP1R1 44 37 O=C(O)/C=C\c1cccc(COc2ccccc2Cl)c1 ZINC000217847381 CI For-Sale Unstable PDS 17 41 C[C@H](c1ccccc1F)N(C)CC[C@@H](O)c1ccccc1 ZINC000217847391 CH On-Demand Unstable AOC3 22 40 CC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217847407 FI For-Sale Unstable CCR3 17 40 CC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217847407 FI For-Sale Unstable AKR1C3 22 43 CC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217847407 FI For-Sale Unstable PARP15 0 40 CC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217847407 FI For-Sale Unstable KCNK3 95 38 CC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217847407 FI For-Sale Unstable KCNK9 52 38 O=C(c1ccc(F)c(F)c1)N1C[C@H]2CNC[C@@H](C2)C1 ZINC000217847411 CD For-Sale Unstable CHRNA7 30 59 COc1cccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217847433 EG For-Sale Unstable HTR1A 18 41 COc1cccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217847433 EG For-Sale Unstable DRD4 43 33 COc1cccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217847433 EG For-Sale Unstable HRH2 27 46 COc1cccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217847433 EG For-Sale Unstable DRD3 16 40 COc1cccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217847433 EG For-Sale Unstable PTGER3 17 45 COc1cccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217847433 EG For-Sale Unstable NPY1R 53 41 COc1cccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217847433 EG For-Sale Unstable CCKAR 49 47 COc1cccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217847433 EG For-Sale Unstable P2RY1 19 42 COc1cccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217847433 EG For-Sale Unstable CCR3 80 54 COc1cccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217847433 EG For-Sale Unstable MTNR1A 48 41 COc1cccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217847433 EG For-Sale Unstable MTNR1B 52 41 COc1cccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217847433 EG For-Sale Unstable SOAT1 18 43 COc1cccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217847433 EG For-Sale Unstable CCKBR 47 47 COc1cccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217847433 EG For-Sale Unstable EPHX2 40 47 COc1cccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217847433 EG For-Sale Unstable CHRNA10 41 41 COc1cccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217847433 EG For-Sale Unstable MCHR1 25 51 COc1cccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217847433 EG For-Sale Unstable ACKR3 64 33 CC[C@H](C)N(C)CCN[C@@H]1CCc2cc(O)ccc21 ZINC000217847436 CF For-Sale Unstable STS 47 33 CCN(CC)CCC(=O)NCc1ccccc1 ZINC000217847455 BE For-Sale Unstable MME 23 41 CCN(CC)CCC(=O)NCc1ccccc1 ZINC000217847455 BE For-Sale Unstable AMY2 40 39 CCN(CC)CCC(=O)NCc1ccccc1 ZINC000217847455 BE For-Sale Unstable CA5B 16 43 CCN(CC)CCC(=O)NCc1ccccc1 ZINC000217847455 BE For-Sale Unstable CA5A 19 43 CCN(CC)CCC(=O)NCc1ccccc1 ZINC000217847455 BE For-Sale Unstable MTNR1B 16 40 CCN(CC)CCC(=O)NCc1ccccc1 ZINC000217847455 BE For-Sale Unstable TPSAB1 15 45 CCN(CC)CCC(=O)NCc1ccccc1 ZINC000217847455 BE For-Sale Unstable AMP1_PLAFQ 41 39 CCN(CC)CCC(=O)NCc1ccccc1 ZINC000217847455 BE For-Sale Unstable PDS 53 40 O=C(O)/C=C\c1cc(F)ccc1COc1ccccc1Cl ZINC000217847468 DI For-Sale Unstable PTGER2 21 47 O=C(O)/C=C\c1cc(F)ccc1COc1ccccc1Cl ZINC000217847468 DI For-Sale Unstable PTGER1 38 41 O=C(O)/C=C\c1cc(F)ccc1COc1ccccc1Cl ZINC000217847468 DI For-Sale Unstable PTGER4 28 46 O=C(O)/C=C\c1cc(F)ccc1COc1ccccc1Cl ZINC000217847468 DI For-Sale Unstable CXCL8 24 40 O=C(O)/C=C\c1cc(F)ccc1COc1ccccc1Cl ZINC000217847468 DI For-Sale Unstable FABP4 19 43 O=C(O)/C=C\c1cc(F)ccc1COc1ccccc1Cl ZINC000217847468 DI For-Sale Unstable PTGER3 27 47 O=C(O)/C=C\c1cc(F)ccc1COc1ccccc1Cl ZINC000217847468 DI For-Sale Unstable CDC25B 0 41 O=C(O)/C=C\c1cc(F)ccc1COc1ccccc1Cl ZINC000217847468 DI For-Sale Unstable FABP5 29 43 O=C(O)/C=C\c1cc(F)ccc1COc1ccccc1Cl ZINC000217847468 DI For-Sale Unstable AKR1C3 30 41 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1ccccc1Cl ZINC000217847544 EI In-Stock Unstable ECR 33 41 CC(C)(C)c1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217847554 FJ For-Sale Unstable TRPV1 15 42 CC(C)(C)c1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217847554 FJ For-Sale Unstable CCR3 23 41 CC(C)(C)c1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217847554 FJ For-Sale Unstable EPHX2 42 45 O=C(O)/C=C\c1cc(COc2ccccc2Cl)ccc1F ZINC000217847563 DI For-Sale Unstable PTGER2 21 51 O=C(O)/C=C\c1cc(COc2ccccc2Cl)ccc1F ZINC000217847563 DI For-Sale Unstable PTGER1 71 40 O=C(O)/C=C\c1cc(COc2ccccc2Cl)ccc1F ZINC000217847563 DI For-Sale Unstable PTGER4 40 47 O=C(O)/C=C\c1cc(COc2ccccc2Cl)ccc1F ZINC000217847563 DI For-Sale Unstable PTGER3 36 51 O=C(O)/C=C\c1cc(COc2ccccc2Cl)ccc1F ZINC000217847563 DI For-Sale Unstable PTGDR 0 42 O=C(O)/C=C\c1cc(COc2ccccc2Cl)ccc1F ZINC000217847563 DI For-Sale Unstable AKR1C3 31 47 O=C(O)/C=C\c1cc(COc2ccccc2Cl)ccc1F ZINC000217847563 DI For-Sale Unstable CYSP_PLAFA 40 32 CC(C)(C)c1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217847622 FJ For-Sale Unstable TRPV1 15 42 CC(C)(C)c1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217847622 FJ For-Sale Unstable CCR3 23 41 CC(C)(C)c1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217847622 FJ For-Sale Unstable EPHX2 42 45 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1ccccc1Cl ZINC000217847639 EI In-Stock Unstable ECR 33 41 CCC[C@@](C)(O)CNC(=O)c1cc(C)cc(Cl)c1 ZINC000217847662 CF On-Demand Unstable CACNA1I 48 36 CCC[C@](C)(O)CNC(=O)c1cc(C)cc(Cl)c1 ZINC000217847738 CF On-Demand Unstable CACNA1I 48 36 CC[C@@H](NC(=O)c1ccccc1Cl)c1ccc(C)c(C)c1 ZINC000217847746 DJ In-Stock Unstable PTGER3 52 43 CC[C@@H](NC(=O)c1ccccc1Cl)c1ccc(C)c(C)c1 ZINC000217847746 DJ In-Stock Unstable ECR 45 43 CC[C@@H](NC(=O)c1ccccc1Cl)c1ccc(C)c(C)c1 ZINC000217847746 DJ In-Stock Unstable TACR3 49 37 CC[C@@H](NC(=O)c1ccccc1Cl)c1ccc(C)c(C)c1 ZINC000217847746 DJ In-Stock Unstable UTS2 68 37 O=C1C[C@@H](c2ccc(C(=O)O)cc2)c2c(c3ccccc3oc2=O)O1 ZINC000217847763 EF In-Stock Unstable VKORC1 0 40 O=C1C[C@@H](c2ccc(C(=O)O)cc2)c2c(c3ccccc3oc2=O)O1 ZINC000217847763 EF In-Stock Unstable NQO1 15 42 O=C1C[C@@H](c2ccc(C(=O)O)cc2)c2c(c3ccccc3oc2=O)O1 ZINC000217847763 EF In-Stock Unstable TNKS 15 44 Cc1ccc2[nH]c([C@@H](C)NC(=O)c3ccc(SCCO)cc3)nc2c1 ZINC000217847790 FG In-Stock Unstable F9 23 40 O=C1C[C@H](c2ccc(C(=O)O)cc2)c2c(c3ccccc3oc2=O)O1 ZINC000217847808 EF In-Stock Unstable VKORC1 0 40 O=C1C[C@H](c2ccc(C(=O)O)cc2)c2c(c3ccccc3oc2=O)O1 ZINC000217847808 EF In-Stock Unstable NQO1 15 42 O=C1C[C@H](c2ccc(C(=O)O)cc2)c2c(c3ccccc3oc2=O)O1 ZINC000217847808 EF In-Stock Unstable TNKS 15 44 CC[C@H](NC(=O)c1ccccc1Cl)c1ccc(C)c(C)c1 ZINC000217847819 DJ In-Stock Unstable PTGER3 52 43 CC[C@H](NC(=O)c1ccccc1Cl)c1ccc(C)c(C)c1 ZINC000217847819 DJ In-Stock Unstable ECR 45 43 CC[C@H](NC(=O)c1ccccc1Cl)c1ccc(C)c(C)c1 ZINC000217847819 DJ In-Stock Unstable TACR3 49 37 CC[C@H](NC(=O)c1ccccc1Cl)c1ccc(C)c(C)c1 ZINC000217847819 DJ In-Stock Unstable UTS2 68 37 COc1ccc(CN2CCNC(=O)C2)cc1/C=C\C(=O)O ZINC000217847824 CC For-Sale Unstable PTGER2 24 41 COc1ccc(CN2CCNC(=O)C2)cc1/C=C\C(=O)O ZINC000217847824 CC For-Sale Unstable PTGER4 0 41 Cc1ccc2[nH]c([C@H](C)NC(=O)c3ccc(SCCO)cc3)nc2c1 ZINC000217847853 FG In-Stock Unstable F9 23 40 CC[C@@H](NC(=O)c1ccccc1Cl)c1ccc(C)cc1C ZINC000217847936 DJ In-Stock Unstable ECR 47 47 CC[C@@H](NC(=O)c1ccccc1Cl)c1ccc(C)cc1C ZINC000217847936 DJ In-Stock Unstable TACR3 23 40 CC[C@@H](NC(=O)c1ccccc1Cl)c1ccc(C)cc1C ZINC000217847936 DJ In-Stock Unstable UTS2 42 34 CC[C@@H](NC(=O)c1ccccc1Cl)c1ccc(C)cc1C ZINC000217847936 DJ In-Stock Unstable CTSA 52 40 CC[C@@H](NC(=O)c1ccccc1Cl)c1ccc(C)cc1C ZINC000217847936 DJ In-Stock Unstable KCNK3 31 42 Cc1cccc(NC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217847937 EJ For-Sale Unstable CCKAR 24 51 Cc1cccc(NC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217847937 EJ For-Sale Unstable KDR 17 40 Cc1cccc(NC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217847937 EJ For-Sale Unstable KCNK3 109 46 Cc1cccc(NC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217847937 EJ For-Sale Unstable KCNK9 64 46 CCCCOc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217847948 FJ For-Sale Unstable ADRB1 21 42 CCCCOc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217847948 FJ For-Sale Unstable HRH2 27 43 CCCCOc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217847948 FJ For-Sale Unstable LTA4H 50 38 CCCCOc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217847948 FJ For-Sale Unstable HRH3 26 43 CCCCOc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217847948 FJ For-Sale Unstable P2RY1 31 40 CCCCOc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217847948 FJ For-Sale Unstable PLA2G4B 74 34 CCCCOc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217847948 FJ For-Sale Unstable FAAH 24 45 CCCCOc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217847948 FJ For-Sale Unstable EPHX2 52 47 CCCCOc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217847948 FJ For-Sale Unstable NCE103 19 46 CC[C@H](NC(=O)c1ccccc1Cl)c1ccc(C)cc1C ZINC000217848016 DJ In-Stock Unstable ECR 47 47 CC[C@H](NC(=O)c1ccccc1Cl)c1ccc(C)cc1C ZINC000217848016 DJ In-Stock Unstable TACR3 23 40 CC[C@H](NC(=O)c1ccccc1Cl)c1ccc(C)cc1C ZINC000217848016 DJ In-Stock Unstable UTS2 42 34 CC[C@H](NC(=O)c1ccccc1Cl)c1ccc(C)cc1C ZINC000217848016 DJ In-Stock Unstable CTSA 52 40 CC[C@H](NC(=O)c1ccccc1Cl)c1ccc(C)cc1C ZINC000217848016 DJ In-Stock Unstable KCNK3 31 42 O=C(O)/C=C\c1cc(CN2CCCCCCC2)ccc1F ZINC000217848024 CH For-Sale Unstable HRH3 19 41 O=C(O)/C=C\c1cc(CN2CCCCCCC2)ccc1F ZINC000217848024 CH For-Sale Unstable SIGMAR1 19 41 O=C(O)/C=C\c1cc(CN2CCCCCCC2)ccc1F ZINC000217848024 CH For-Sale Unstable CCR1 0 42 CCCn1c(NC(=O)c2nn(-c3ccccc3)cc2O)nc2ccccc21 ZINC000217848027 FH On-Demand Unstable ADORA3 17 44 CCCCOc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217848028 FJ For-Sale Unstable ADRB1 21 42 CCCCOc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217848028 FJ For-Sale Unstable HRH2 27 43 CCCCOc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217848028 FJ For-Sale Unstable LTA4H 50 38 CCCCOc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217848028 FJ For-Sale Unstable HRH3 26 43 CCCCOc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217848028 FJ For-Sale Unstable P2RY1 31 40 CCCCOc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217848028 FJ For-Sale Unstable PLA2G4B 74 34 CCCCOc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217848028 FJ For-Sale Unstable FAAH 24 45 CCCCOc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217848028 FJ For-Sale Unstable EPHX2 52 47 CCCCOc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217848028 FJ For-Sale Unstable NCE103 19 46 O=C(N/C=C/c1ccccc1Br)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217848043 HK For-Sale Anodyne GUAB 0 45 O=C(N/C=C/c1ccccc1Br)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217848043 HK For-Sale Anodyne RAF1 31 45 O=C(N/C=C/c1ccccc1Br)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217848043 HK For-Sale Anodyne Q8MMZ8_EIMTE 50 45 O=C(N/C=C/c1ccccc1Br)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217848043 HK For-Sale Anodyne PTPA 0 45 O=C(N/C=C/c1ccccc1Br)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217848043 HK For-Sale Anodyne IMDH_CRYPV 31 48 O=C(N/C=C/c1ccccc1Br)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217848043 HK For-Sale Anodyne BLM 0 45 COc1ccccc1[C@H](CC(=O)N1CCc2c([nH]c3ccccc23)C1)c1oc(C)cc(=O)c1O ZINC000217848079 JI In-Stock Unstable RORC 36 41 CC[C@@H](NC(=O)c1ccccc1Cl)c1ccc(OC)c(OC)c1 ZINC000217848110 EI In-Stock Unstable PTGER3 39 46 CC[C@@H](NC(=O)c1ccccc1Cl)c1ccc(OC)c(OC)c1 ZINC000217848110 EI In-Stock Unstable TACR3 48 39 CC[C@@H](NC(=O)c1ccccc1Cl)c1ccc(OC)c(OC)c1 ZINC000217848110 EI In-Stock Unstable UTS2 66 36 CC[C@@H](NC(=O)c1ccccc1Cl)c1ccc(OC)c(OC)c1 ZINC000217848110 EI In-Stock Unstable KCNK3 43 38 O=C(NC[C@H]1CCCN1c1ccccc1)Nc1cccc(Cl)c1 ZINC000217848137 EI For-Sale Unstable PPIA 15 40 O=C(NC[C@H]1CCCN1c1ccccc1)Nc1cccc(Cl)c1 ZINC000217848137 EI For-Sale Unstable NPY1R 43 40 O=C(NC[C@H]1CCCN1c1ccccc1)Nc1cccc(Cl)c1 ZINC000217848137 EI For-Sale Unstable CCR3 54 39 O=C(NC[C@H]1CCCN1c1ccccc1)Nc1cccc(Cl)c1 ZINC000217848137 EI For-Sale Unstable GRM5 15 56 O=C(NC[C@H]1CCCN1c1ccccc1)Nc1cccc(Cl)c1 ZINC000217848137 EI For-Sale Unstable CCKBR 46 39 O=C(NC[C@H]1CCCN1c1ccccc1)Nc1cccc(Cl)c1 ZINC000217848137 EI For-Sale Unstable EPHX2 39 60 O=C(NC[C@H]1CCCN1c1ccccc1)Nc1cccc(Cl)c1 ZINC000217848137 EI For-Sale Unstable MCHR1 27 41 O=C(NC[C@H]1CCCN1c1ccccc1)Nc1cccc(Cl)c1 ZINC000217848137 EI For-Sale Unstable CACNA1I 22 47 NC(=O)[C@H]1CCCN1Cc1ccccc1/C=C\C(=O)O ZINC000217848141 CD For-Sale Unstable SLC6A1 43 37 NC(=O)[C@H]1CCCN1Cc1ccccc1/C=C\C(=O)O ZINC000217848141 CD For-Sale Unstable PTGER3 17 43 NC(=O)[C@H]1CCCN1Cc1ccccc1/C=C\C(=O)O ZINC000217848141 CD For-Sale Unstable PREP 42 36 CC[C@H](NC(=O)c1ccccc1Cl)c1ccc(OC)c(OC)c1 ZINC000217848181 EI In-Stock Unstable PTGER3 39 46 CC[C@H](NC(=O)c1ccccc1Cl)c1ccc(OC)c(OC)c1 ZINC000217848181 EI In-Stock Unstable TACR3 48 39 CC[C@H](NC(=O)c1ccccc1Cl)c1ccc(OC)c(OC)c1 ZINC000217848181 EI In-Stock Unstable UTS2 66 36 CC[C@H](NC(=O)c1ccccc1Cl)c1ccc(OC)c(OC)c1 ZINC000217848181 EI In-Stock Unstable KCNK3 43 38 COc1ccccc1[C@@H](CC(=O)N1CCc2c([nH]c3ccccc23)C1)c1oc(C)cc(=O)c1O ZINC000217848182 JI In-Stock Unstable RORC 36 41 CC(C)(C)NC(=O)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217848216 EE In-Stock Unstable BMP1 30 47 COC1(C)CCN(C(=O)c2ccc(Br)cc2)CC1 ZINC000217848240 DG On-Demand Unstable CCR5 49 44 COC1(C)CCN(C(=O)c2ccc(Br)cc2)CC1 ZINC000217848240 DG On-Demand Unstable L3MBTL3 48 36 O=C(NC[C@@H]1CCCN1c1ccccc1)Nc1cccc(Cl)c1 ZINC000217848243 EI For-Sale Unstable PPIA 15 40 O=C(NC[C@@H]1CCCN1c1ccccc1)Nc1cccc(Cl)c1 ZINC000217848243 EI For-Sale Unstable NPY1R 43 40 O=C(NC[C@@H]1CCCN1c1ccccc1)Nc1cccc(Cl)c1 ZINC000217848243 EI For-Sale Unstable CCR3 54 39 O=C(NC[C@@H]1CCCN1c1ccccc1)Nc1cccc(Cl)c1 ZINC000217848243 EI For-Sale Unstable GRM5 15 56 O=C(NC[C@@H]1CCCN1c1ccccc1)Nc1cccc(Cl)c1 ZINC000217848243 EI For-Sale Unstable CCKBR 46 39 O=C(NC[C@@H]1CCCN1c1ccccc1)Nc1cccc(Cl)c1 ZINC000217848243 EI For-Sale Unstable EPHX2 39 60 O=C(NC[C@@H]1CCCN1c1ccccc1)Nc1cccc(Cl)c1 ZINC000217848243 EI For-Sale Unstable MCHR1 27 41 O=C(NC[C@@H]1CCCN1c1ccccc1)Nc1cccc(Cl)c1 ZINC000217848243 EI For-Sale Unstable CACNA1I 22 47 CCn1nc(C)c(CNC(=O)c2cc(=O)cc(C)o2)c1C ZINC000217848245 CD In-Stock Unstable P2RX7 19 44 Cc1cc(C)c(C(=O)Nc2ccc(Cc3ccncc3)cc2)c(C)c1 ZINC000217848276 EJ On-Demand Unstable JAK1 18 42 Cc1cc(C)c(C(=O)Nc2ccc(Cc3ccncc3)cc2)c(C)c1 ZINC000217848276 EJ On-Demand Unstable FLT1 57 45 Cc1cc(C)c(C(=O)Nc2ccc(Cc3ccncc3)cc2)c(C)c1 ZINC000217848276 EJ On-Demand Unstable KDR 23 45 Cc1cc(C)c(C(=O)Nc2ccc(Cc3ccncc3)cc2)c(C)c1 ZINC000217848276 EJ On-Demand Unstable GRM4 22 42 Cc1cc(C)c(C(=O)Nc2ccc(Cc3ccncc3)cc2)c(C)c1 ZINC000217848276 EJ On-Demand Unstable TYK2 49 36 Cc1cc(C)c(C(=O)Nc2ccc(Cc3ccncc3)cc2)c(C)c1 ZINC000217848276 EJ On-Demand Unstable KCNK3 46 41 CC(C)(C)NC(=O)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217848305 EE In-Stock Unstable BMP1 30 47 CC[C@@H](NC(=O)c1ccccc1Cl)c1ccc(S(C)(=O)=O)cc1 ZINC000217848315 FH In-Stock Unstable CTSF 47 35 CC[C@@H](NC(=O)c1ccccc1Cl)c1ccc(S(C)(=O)=O)cc1 ZINC000217848315 FH In-Stock Unstable TACR3 51 40 CC[C@@H](NC(=O)c1ccccc1Cl)c1ccc(S(C)(=O)=O)cc1 ZINC000217848315 FH In-Stock Unstable UTS2 47 37 O=C(NC[C@H]1CCCN1c1ccccc1)NC1CCCCC1 ZINC000217848338 DG For-Sale Unstable EPHX2 48 52 CC[C@H](NC(=O)c1ccccc1Cl)c1ccc(S(C)(=O)=O)cc1 ZINC000217848354 FH In-Stock Unstable CTSF 47 35 CC[C@H](NC(=O)c1ccccc1Cl)c1ccc(S(C)(=O)=O)cc1 ZINC000217848354 FH In-Stock Unstable TACR3 51 40 CC[C@H](NC(=O)c1ccccc1Cl)c1ccc(S(C)(=O)=O)cc1 ZINC000217848354 FH In-Stock Unstable UTS2 47 37 CCOc1cc(CN2CCN(C)[C@@H](C)C2)cc(Br)c1O ZINC000217848391 EF For-Sale Unstable SSTR5 46 35 COC(=O)CNC(=O)CCCCCN1C(=O)c2ccccc2N2C(=O)c3c(ccc(OC)c3OC)[C@H]12 ZINC000217848408 JF In-Stock Unstable HTR7 24 40 COc1ccccc1NC(=O)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217848412 GG In-Stock Unstable BMP1 17 40 COc1ccccc1NC(=O)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217848412 GG In-Stock Unstable SMO 43 51 O=C(NC[C@@H]1CCCN1c1ccccc1)NC1CCCCC1 ZINC000217848421 DG For-Sale Unstable EPHX2 48 52 COc1ccc(-c2noc(CNC(=O)c3ccccc3Cl)n2)c(OC)c1 ZINC000217848481 FG In-Stock Unstable ECR 25 41 COc1ccc(-c2noc(CNC(=O)c3ccccc3Cl)n2)c(OC)c1 ZINC000217848481 FG In-Stock Unstable U38 0 43 COc1ccc(-c2noc(CNC(=O)c3ccccc3Cl)n2)c(OC)c1 ZINC000217848481 FG In-Stock Unstable KCNK3 30 41 COc1ccccc1NC(=O)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217848486 GG In-Stock Unstable BMP1 17 40 COc1ccccc1NC(=O)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217848486 GG In-Stock Unstable SMO 43 51 COC(=O)CNC(=O)CCCCCN1C(=O)c2ccccc2N2C(=O)c3c(ccc(OC)c3OC)[C@@H]12 ZINC000217848497 JF In-Stock Unstable HTR7 24 40 O=C(N/C=C/c1ccccc1Br)Nc1cccc(Cl)c1 ZINC000217848498 FJ For-Sale Anodyne PPIA 22 40 O=C(N/C=C/c1ccccc1Br)Nc1cccc(Cl)c1 ZINC000217848498 FJ For-Sale Anodyne KCNK3 55 44 O=C(N/C=C/c1ccccc1Br)Nc1cccc(Cl)c1 ZINC000217848498 FJ For-Sale Anodyne KCNK9 27 41 CCOc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217848533 EH For-Sale Unstable HRH2 15 44 CCOc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217848533 EH For-Sale Unstable LTA4H 43 39 CCOc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217848533 EH For-Sale Unstable CA1 43 38 CCOc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217848533 EH For-Sale Unstable NPY2R 23 45 CCOc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217848533 EH For-Sale Unstable CCR3 32 41 CCOc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217848533 EH For-Sale Unstable ITGA4 42 31 CCOc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217848533 EH For-Sale Unstable EPHX2 44 42 CCOc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217848533 EH For-Sale Unstable NOD2 25 41 O=C(O)/C=C\c1ccc(C(=O)N2CC(=O)NC(=O)C2)cc1 ZINC000217848569 CB For-Sale Unstable GPR183 0 43 O=C(Nc1ccccc1F)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217848587 GG In-Stock Unstable BMP1 20 42 O=C(Nc1ccccc1F)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217848587 GG In-Stock Unstable SMO 43 37 COc1cccc(-c2noc(CN(C)C(=O)c3ccccc3Cl)n2)c1 ZINC000217848607 FH In-Stock Unstable ECR 37 44 COc1cccc(-c2noc(CN(C)C(=O)c3ccccc3Cl)n2)c1 ZINC000217848607 FH In-Stock Unstable GRM5 16 44 COc1cccc(-c2noc(CN(C)C(=O)c3ccccc3Cl)n2)c1 ZINC000217848607 FH In-Stock Unstable HSD17B2 26 46 O=C(N/C=C/c1ccccc1Br)Nc1ccc(Cl)cc1 ZINC000217848615 FJ For-Sale Anodyne MTCA1 15 42 O=C(N/C=C/c1ccccc1Br)Nc1ccc(Cl)cc1 ZINC000217848615 FJ For-Sale Anodyne P96878_MYCTU 20 42 O=C(N/C=C/c1ccccc1Br)Nc1ccc(Cl)cc1 ZINC000217848615 FJ For-Sale Anodyne P95276_MYCTO 0 41 CCOc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217848626 EH For-Sale Unstable HRH2 15 44 CCOc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217848626 EH For-Sale Unstable LTA4H 43 39 CCOc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217848626 EH For-Sale Unstable CA1 43 38 CCOc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217848626 EH For-Sale Unstable NPY2R 23 45 CCOc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217848626 EH For-Sale Unstable CCR3 32 41 CCOc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217848626 EH For-Sale Unstable ITGA4 42 31 CCOc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217848626 EH For-Sale Unstable EPHX2 44 42 CCOc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217848626 EH For-Sale Unstable NOD2 25 41 O=C(Nc1ccccc1F)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217848664 GG In-Stock Unstable BMP1 20 42 O=C(Nc1ccccc1F)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217848664 GG In-Stock Unstable SMO 43 37 CN1CCO[C@@H]([C@@H](O)c2ccccc2C(F)(F)F)C1 ZINC000217848695 CE For-Sale Unstable RBP4 48 36 COc1ccc(-c2noc(CN(C)C(=O)c3ccccc3Cl)n2)c(OC)c1 ZINC000217848740 GH In-Stock Unstable ECR 21 40 COc1ccc(-c2noc(CN(C)C(=O)c3ccccc3Cl)n2)c(OC)c1 ZINC000217848740 GH In-Stock Unstable GPBAR1 24 42 O=C(NC[C@H]1CCCN1c1ccccc1)Nc1ccccc1Cl ZINC000217848741 EI For-Sale Unstable LPL 39 43 O=C(NC[C@H]1CCCN1c1ccccc1)Nc1ccccc1Cl ZINC000217848741 EI For-Sale Unstable KCNQ2 49 39 O=C(NC[C@H]1CCCN1c1ccccc1)Nc1ccccc1Cl ZINC000217848741 EI For-Sale Unstable EPHB3 43 37 O=C(NC[C@H]1CCCN1c1ccccc1)Nc1ccccc1Cl ZINC000217848741 EI For-Sale Unstable LIPG 15 43 C[C@@H](Cn1cncn1)NC(=O)CSc1nnc(N)s1 ZINC000217848742 CC In-Stock Unstable HIS3 83 42 Cc1noc(C)c1CSc1ncccc1C(=O)Nc1ccc(Cc2ccncc2)cc1 ZINC000217848766 IK On-Demand Unstable FLT1 21 40 O=C(Nc1cccs1)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217848773 FG In-Stock Unstable BMP1 18 42 CC(C)(C)OC(=O)NC12C[C@H]3C[C@@H](CC(N)(C3)C1)C2 ZINC000217848800 CF For-Sale Unstable EPHX2 30 44 CN1CCO[C@H]([C@@H](O)c2ccccc2C(F)(F)F)C1 ZINC000217848808 CE For-Sale Unstable RBP4 48 36 C[C@H](Cn1cncn1)NC(=O)CSc1nnc(N)s1 ZINC000217848809 CC In-Stock Unstable HIS3 83 42 O=C(NC[C@@H]1CCCN1c1ccccc1)Nc1ccccc1Cl ZINC000217848810 EI For-Sale Unstable LPL 39 43 O=C(NC[C@@H]1CCCN1c1ccccc1)Nc1ccccc1Cl ZINC000217848810 EI For-Sale Unstable KCNQ2 49 39 O=C(NC[C@@H]1CCCN1c1ccccc1)Nc1ccccc1Cl ZINC000217848810 EI For-Sale Unstable EPHB3 43 37 O=C(NC[C@@H]1CCCN1c1ccccc1)Nc1ccccc1Cl ZINC000217848810 EI For-Sale Unstable LIPG 15 43 CCOc1ccc([C@@H](C)N[C@@H]2CCCC[C@@H]2CC)cc1 ZINC000217848816 CJ For-Sale Unstable ACACA 25 40 O=C(N/C=C/c1ccccc1Br)N1CCN(Cc2ccccc2)CC1 ZINC000217848836 HH For-Sale Unstable DRD4 31 40 O=C(N/C=C/c1ccccc1Br)N1CCN(Cc2ccccc2)CC1 ZINC000217848836 HH For-Sale Unstable SIGMAR1 48 45 O=C(N/C=C/c1ccccc1Br)N1CCN(Cc2ccccc2)CC1 ZINC000217848836 HH For-Sale Unstable FAAH 26 49 O=C(N/C=C/c1ccccc1Br)N1CCN(Cc2ccccc2)CC1 ZINC000217848836 HH For-Sale Unstable MGLL 0 43 O=C(N/C=C/c1ccccc1Br)N1CCN(Cc2ccccc2)CC1 ZINC000217848836 HH For-Sale Unstable GPR183 0 44 CN(Cc1nc(-c2cccc(Br)c2)no1)C(=O)c1ccccc1Cl ZINC000217848844 HI In-Stock Unstable ECR 40 35 O=C(Nc1cccs1)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217848865 FG In-Stock Unstable BMP1 18 42 CCOc1ccc([C@@H](C)N[C@H]2CCCC[C@@H]2CC)cc1 ZINC000217848888 CJ For-Sale Unstable ACACA 25 40 O=C(NC[C@H]1CCCN1c1ccccc1)NC1CCCC1 ZINC000217848913 CF For-Sale Unstable EPHX2 44 50 CC(C)c1ccc(CCCNC(=O)c2ccccc2Cl)cc1 ZINC000217848943 DJ In-Stock Unstable ANPEP 16 43 CC(C)c1ccc(CCCNC(=O)c2ccccc2Cl)cc1 ZINC000217848943 DJ In-Stock Unstable SDH1 0 56 CC(C)c1ccc(CCCNC(=O)c2ccccc2Cl)cc1 ZINC000217848943 DJ In-Stock Unstable ECR 48 47 CC(C)c1ccc(CCCNC(=O)c2ccccc2Cl)cc1 ZINC000217848943 DJ In-Stock Unstable SLC6A5 35 46 CC(C)c1ccc(CCCNC(=O)c2ccccc2Cl)cc1 ZINC000217848943 DJ In-Stock Unstable AMP1_PLAFQ 31 43 CC(C)c1ccc(CCCNC(=O)c2ccccc2Cl)cc1 ZINC000217848943 DJ In-Stock Unstable CRTM 41 41 CC(C)c1ccc(CCCNC(=O)c2ccccc2Cl)cc1 ZINC000217848943 DJ In-Stock Unstable SMO 17 43 CC(C)c1ccc(CCCNC(=O)c2ccccc2Cl)cc1 ZINC000217848943 DJ In-Stock Unstable E3UJZ5_SPOLI 39 47 O=C(NC[C@@H]1CCCN1c1ccccc1)NC1CCCC1 ZINC000217848983 CF For-Sale Unstable EPHX2 44 50 Cc1nc2sc([C@H](c3ccccc3)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)c(O)n2n1 ZINC000217848996 IG In-Stock Unstable CHRNA4 25 41 CCOc1cc(CN2CCN(C)[C@@H](C)C2)ccc1O ZINC000217848997 CD For-Sale Unstable SSTR5 81 48 O=C(NCCc1ccccc1)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217849000 GF In-Stock Unstable BMP1 22 42 CCS(=O)(=O)N1CCC(C(=O)Nc2ccc(Cc3ccncc3)cc2)(c2ccccc2)CC1 ZINC000217849002 JH On-Demand Unstable F13A1 54 33 CCS(=O)(=O)N1CCC(C(=O)Nc2ccc(Cc3ccncc3)cc2)(c2ccccc2)CC1 ZINC000217849002 JH On-Demand Unstable NAMPT 44 35 O=C/C(=C/CO)OCc1ccccc1 ZINC000217849014 AD For-Sale Unstable KLK3 40 32 O=C(NCCCN1CCCc2ccccc21)c1ccccc1Cl ZINC000217849058 EH In-Stock Unstable DRD2 36 44 O=C(NCCCN1CCCc2ccccc21)c1ccccc1Cl ZINC000217849058 EH In-Stock Unstable DRD1 21 40 O=C(NCCCN1CCCc2ccccc21)c1ccccc1Cl ZINC000217849058 EH In-Stock Unstable HTR2A 30 42 O=C(NCCCN1CCCc2ccccc21)c1ccccc1Cl ZINC000217849058 EH In-Stock Unstable HTR2C 33 41 O=C(NCCCN1CCCc2ccccc21)c1ccccc1Cl ZINC000217849058 EH In-Stock Unstable AVPR2 41 51 O=C(NCCCN1CCCc2ccccc21)c1ccccc1Cl ZINC000217849058 EH In-Stock Unstable SLC6A4 16 42 O=C(NCCCN1CCCc2ccccc21)c1ccccc1Cl ZINC000217849058 EH In-Stock Unstable DRD3 57 43 O=C(NCCCN1CCCc2ccccc21)c1ccccc1Cl ZINC000217849058 EH In-Stock Unstable TYRO3 26 45 O=C(NCCc1ccccc1)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217849087 GF In-Stock Unstable BMP1 20 42 O=C/C(=C\CO)OCc1ccccc1 ZINC000217849089 AD For-Sale Unstable KLK3 40 32 Cc1nc2sc([C@@H](c3ccccc3)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)c(O)n2n1 ZINC000217849092 IG In-Stock Unstable CHRNA4 25 41 Cc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1C ZINC000217849104 DI For-Sale Unstable LPL 49 35 Cc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1C ZINC000217849104 DI For-Sale Unstable HRH3 21 40 Cc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1C ZINC000217849104 DI For-Sale Unstable NPY1R 44 37 Cc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1C ZINC000217849104 DI For-Sale Unstable CCR3 55 38 Cc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1C ZINC000217849104 DI For-Sale Unstable EPHX2 22 41 Cc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1C ZINC000217849104 DI For-Sale Unstable MCHR1 15 46 Cc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1C ZINC000217849104 DI For-Sale Unstable FPR2 37 40 O=C(N/C=C/c1ccccc1Br)NC1CCCCCCCCCCC1 ZINC000217849137 HK For-Sale Unstable EPHX2 24 48 COc1ccc(/C=C\C(=O)N2CC(=O)NC(=O)[C@H]2C)cc1 ZINC000217849160 CC For-Sale Unstable GPR183 0 47 COc1ccccc1CCCNC(=O)c1ccc(Cl)cc1 ZINC000217849171 DH In-Stock Unstable HTR1A 21 58 COc1ccccc1CCCNC(=O)c1ccc(Cl)cc1 ZINC000217849171 DH In-Stock Unstable DRD2 36 58 COc1ccccc1CCCNC(=O)c1ccc(Cl)cc1 ZINC000217849171 DH In-Stock Unstable DRD1 15 45 COc1ccccc1CCCNC(=O)c1ccc(Cl)cc1 ZINC000217849171 DH In-Stock Unstable DRD4 44 38 COc1ccccc1CCCNC(=O)c1ccc(Cl)cc1 ZINC000217849171 DH In-Stock Unstable DRD3 59 58 COc1ccccc1CCCNC(=O)c1ccc(Cl)cc1 ZINC000217849171 DH In-Stock Unstable F10 0 43 COc1ccccc1CCCNC(=O)c1ccc(Cl)cc1 ZINC000217849171 DH In-Stock Unstable TRPV1 0 44 COc1ccccc1CCCNC(=O)c1ccc(Cl)cc1 ZINC000217849171 DH In-Stock Unstable TSPO 19 40 COc1ccccc1CCCNC(=O)c1ccc(Cl)cc1 ZINC000217849171 DH In-Stock Unstable CPT1A 46 32 COc1ccccc1CCCNC(=O)c1ccc(Cl)cc1 ZINC000217849171 DH In-Stock Unstable PPARD 17 42 COc1ccccc1CCCNC(=O)c1ccc(Cl)cc1 ZINC000217849171 DH In-Stock Unstable MTNR1A 42 38 COc1ccccc1CCCNC(=O)c1ccc(Cl)cc1 ZINC000217849171 DH In-Stock Unstable MTNR1B 44 45 COc1ccccc1CCCNC(=O)c1ccc(Cl)cc1 ZINC000217849171 DH In-Stock Unstable SLC6A5 28 40 COc1ccccc1CCCNC(=O)c1ccc(Cl)cc1 ZINC000217849171 DH In-Stock Unstable PTGDR 24 41 COc1ccccc1CCCNC(=O)c1ccc(Cl)cc1 ZINC000217849171 DH In-Stock Unstable ITGAV 17 40 COc1ccccc1CCCNC(=O)c1ccc(Cl)cc1 ZINC000217849171 DH In-Stock Unstable PTGDR2 20 41 COc1ccccc1CCCNC(=O)c1ccc(Cl)cc1 ZINC000217849171 DH In-Stock Unstable TAAR1 19 44 COc1ccccc1CCCNC(=O)c1ccc(Cl)cc1 ZINC000217849171 DH In-Stock Unstable UTS2 43 33 COc1ccccc1CCCNC(=O)c1ccc(Cl)cc1 ZINC000217849171 DH In-Stock Unstable MBTPS1 53 35 COc1ccccc1CCCNC(=O)c1ccc(Cl)cc1 ZINC000217849171 DH In-Stock Unstable AP2S1 0 47 COc1ccccc1CCCNC(=O)c1ccc(Cl)cc1 ZINC000217849171 DH In-Stock Unstable ALPHA-1A 0 42 Cc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1C ZINC000217849190 DI For-Sale Unstable LPL 49 35 Cc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1C ZINC000217849190 DI For-Sale Unstable HRH3 21 40 Cc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1C ZINC000217849190 DI For-Sale Unstable NPY1R 44 37 Cc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1C ZINC000217849190 DI For-Sale Unstable CCR3 55 38 Cc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1C ZINC000217849190 DI For-Sale Unstable EPHX2 22 41 Cc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1C ZINC000217849190 DI For-Sale Unstable MCHR1 15 46 Cc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1C ZINC000217849190 DI For-Sale Unstable FPR2 37 40 C[C@@H]1CN(Cc2ccccc2/C=C\C(=O)O)[C@H](C)CO1 ZINC000217849195 CE For-Sale Unstable PTGER2 33 42 C[C@@H]1CN(Cc2ccccc2/C=C\C(=O)O)[C@H](C)CO1 ZINC000217849195 CE For-Sale Unstable PTGER4 17 42 C[C@@H]1CN(Cc2ccccc2/C=C\C(=O)O)[C@H](C)CO1 ZINC000217849195 CE For-Sale Unstable PTGER3 17 42 C[C@@H]1CN(Cc2ccccc2/C=C\C(=O)O)[C@H](C)CO1 ZINC000217849195 CE For-Sale Unstable PTGDR 15 41 O=C(Nc1ccccc1Cl)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217849217 GH In-Stock Unstable BMP1 22 42 O=C(Nc1ccccc1Cl)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217849217 GH In-Stock Unstable SMO 52 47 COc1ccc(/C=C\C(=O)N2CC(=O)NC(=O)[C@@H]2C)cc1 ZINC000217849249 CC For-Sale Unstable GPR183 0 47 CCOc1ccc(CCCNC(=O)c2ccc(Cl)cc2)cc1 ZINC000217849263 DI In-Stock Unstable DRD3 15 40 CCOc1ccc(CCCNC(=O)c2ccc(Cl)cc2)cc1 ZINC000217849263 DI In-Stock Unstable SCNN1A 47 35 CCOc1ccc(CCCNC(=O)c2ccc(Cl)cc2)cc1 ZINC000217849263 DI In-Stock Unstable KCNQ1 0 45 CCOc1ccc(CCCNC(=O)c2ccc(Cl)cc2)cc1 ZINC000217849263 DI In-Stock Unstable SCN2A 32 50 CCOc1ccc(CCCNC(=O)c2ccc(Cl)cc2)cc1 ZINC000217849263 DI In-Stock Unstable SCN5A 0 41 CCOc1ccc(CCCNC(=O)c2ccc(Cl)cc2)cc1 ZINC000217849263 DI In-Stock Unstable SLC6A5 46 40 CCOc1ccc(CCCNC(=O)c2ccc(Cl)cc2)cc1 ZINC000217849263 DI In-Stock Unstable CXCR3 19 41 CCOc1ccc(CCCNC(=O)c2ccc(Cl)cc2)cc1 ZINC000217849263 DI In-Stock Unstable HDA106 0 47 CCOc1ccc(CCCNC(=O)c2ccc(Cl)cc2)cc1 ZINC000217849263 DI In-Stock Unstable CRTM 42 42 CCOc1ccc(CCCNC(=O)c2ccc(Cl)cc2)cc1 ZINC000217849263 DI In-Stock Unstable UTS2 40 33 CCOc1ccc(CCCNC(=O)c2ccc(Cl)cc2)cc1 ZINC000217849263 DI In-Stock Unstable NOD2 17 40 CCOc1ccccc1NC(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217849293 EH For-Sale Unstable ITGA4 43 35 CCOc1ccccc1NC(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217849293 EH For-Sale Unstable HCN1 53 36 CCOc1ccccc1NC(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217849293 EH For-Sale Unstable HCN4 46 36 O=C(Nc1ccc(Cc2ccncc2)cc1)c1cnn(-c2ccccc2)c1C(F)(F)F ZINC000217849297 HK On-Demand Unstable FLT1 59 42 O=C(Nc1ccc(Cc2ccncc2)cc1)c1cnn(-c2ccccc2)c1C(F)(F)F ZINC000217849297 HK On-Demand Unstable KDR 23 44 O=C(Nc1ccc(Cc2ccncc2)cc1)c1cnn(-c2ccccc2)c1C(F)(F)F ZINC000217849297 HK On-Demand Unstable MST1R 67 51 O=C(N/C=C/c1ccccc1Br)NCCN1CCOCC1 ZINC000217849306 FE For-Sale Unstable CASR 48 35 O=C(N/C=C/c1ccccc1Br)NCCN1CCOCC1 ZINC000217849306 FE For-Sale Unstable EPHX2 18 47 O=C(N/C=C/c1ccccc1Br)NCCN1CCOCC1 ZINC000217849306 FE For-Sale Unstable HPGDS 23 40 O=C(Nc1ccccc1Cl)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217849329 GH In-Stock Unstable BMP1 22 42 O=C(Nc1ccccc1Cl)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217849329 GH In-Stock Unstable SMO 52 47 CCOc1ccccc1NC(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217849373 EH For-Sale Unstable ITGA4 43 35 CCOc1ccccc1NC(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217849373 EH For-Sale Unstable HCN1 53 36 CCOc1ccccc1NC(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217849373 EH For-Sale Unstable HCN4 46 36 CCCOc1ccccc1CCCNC(=O)c1ccc(Cl)cc1 ZINC000217849381 EI In-Stock Unstable DRD3 26 47 CCCOc1ccccc1CCCNC(=O)c1ccc(Cl)cc1 ZINC000217849381 EI In-Stock Unstable KCNQ1 0 40 CCCOc1ccccc1CCCNC(=O)c1ccc(Cl)cc1 ZINC000217849381 EI In-Stock Unstable MTNR1B 43 40 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc3ncccc3c2)CC(=O)O4)cc1O ZINC000217849388 JJ In-Stock Unstable CYP1A1 30 42 Cc1nc(COc2ccccc2C(=O)Nc2ccc(Cc3ccncc3)cc2)no1 ZINC000217849397 HI On-Demand Unstable PPIA 44 36 Cc1nc(COc2ccccc2C(=O)Nc2ccc(Cc3ccncc3)cc2)no1 ZINC000217849397 HI On-Demand Unstable KIT 15 40 Cc1nc(COc2ccccc2C(=O)Nc2ccc(Cc3ccncc3)cc2)no1 ZINC000217849397 HI On-Demand Unstable FLT1 43 40 Cc1nc(COc2ccccc2C(=O)Nc2ccc(Cc3ccncc3)cc2)no1 ZINC000217849397 HI On-Demand Unstable KDR 20 44 Cc1nc(COc2ccccc2C(=O)Nc2ccc(Cc3ccncc3)cc2)no1 ZINC000217849397 HI On-Demand Unstable KCNK3 53 40 Cc1nc(COc2ccccc2C(=O)Nc2ccc(Cc3ccncc3)cc2)no1 ZINC000217849397 HI On-Demand Unstable KCNK9 54 40 O=C(NCc1cccs1)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217849438 GF In-Stock Unstable BMP1 18 41 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc3ncccc3c2)CC(=O)O4)cc1O ZINC000217849464 JJ In-Stock Unstable CYP1A1 30 42 Cc1ccc(OC[C@@H](C)NC(=O)c2ccc(Cl)cc2)cc1 ZINC000217849467 DH In-Stock Unstable PTGS2 0 47 Cc1ccc(OC[C@@H](C)NC(=O)c2ccc(Cl)cc2)cc1 ZINC000217849467 DH In-Stock Unstable SDH1 0 44 Cc1ccc(OC[C@@H](C)NC(=O)c2ccc(Cl)cc2)cc1 ZINC000217849467 DH In-Stock Unstable CCR1 21 44 Cc1ccc(OC[C@@H](C)NC(=O)c2ccc(Cl)cc2)cc1 ZINC000217849467 DH In-Stock Unstable TRPA1 15 48 Cc1ccc(OC[C@@H](C)NC(=O)c2ccc(Cl)cc2)cc1 ZINC000217849467 DH In-Stock Unstable UTS2 56 47 Cc1ccc(OC[C@@H](C)NC(=O)c2ccc(Cl)cc2)cc1 ZINC000217849467 DH In-Stock Unstable GPR88 0 40 COc1cc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc(OC)c1 ZINC000217849511 FG For-Sale Unstable P2RY1 16 40 COc1cc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc(OC)c1 ZINC000217849511 FG For-Sale Unstable CCR3 57 44 COc1cc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc(OC)c1 ZINC000217849511 FG For-Sale Unstable MCHR1 15 48 COc1cc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc(OC)c1 ZINC000217849511 FG For-Sale Unstable ACKR3 61 32 O=C(Cn1nnc(-c2ccc(Cl)cc2)n1)Nc1ccc(Cc2ccncc2)cc1 ZINC000217849514 HH On-Demand Unstable FLT1 23 44 O=C(Cn1nnc(-c2ccc(Cl)cc2)n1)Nc1ccc(Cc2ccncc2)cc1 ZINC000217849514 HH On-Demand Unstable IMDH_CRYPV 18 40 O=C(Cn1nnc(-c2ccc(Cl)cc2)n1)Nc1ccc(Cc2ccncc2)cc1 ZINC000217849514 HH On-Demand Unstable SCARB1 31 41 O=C(NCc1cccs1)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217849522 GF In-Stock Unstable BMP1 18 41 CCC(CC)N(C)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217849555 CG For-Sale Unstable APP 43 40 CCC(CC)N(C)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217849555 CG For-Sale Unstable TUBB1 49 40 CCC(CC)N(C)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217849555 CG For-Sale Unstable AKR1C3 31 42 COC(=O)[C@H](Cc1ccccc1)[C@H](C)NC(C)=O ZINC000217849561 BD On-Demand Unstable PRSS1 20 54 COC(=O)[C@H](Cc1ccccc1)[C@H](C)NC(C)=O ZINC000217849561 BD On-Demand Unstable ACE 43 41 COC(=O)[C@H](Cc1ccccc1)[C@H](C)NC(C)=O ZINC000217849561 BD On-Demand Unstable OPRM1 22 40 COC(=O)[C@H](Cc1ccccc1)[C@H](C)NC(C)=O ZINC000217849561 BD On-Demand Unstable MME 96 43 COC(=O)[C@H](Cc1ccccc1)[C@H](C)NC(C)=O ZINC000217849561 BD On-Demand Unstable LTA4H 15 43 COC(=O)[C@H](Cc1ccccc1)[C@H](C)NC(C)=O ZINC000217849561 BD On-Demand Unstable ANPEP 81 38 COC(=O)[C@H](Cc1ccccc1)[C@H](C)NC(C)=O ZINC000217849561 BD On-Demand Unstable TACR1 18 48 COC(=O)[C@H](Cc1ccccc1)[C@H](C)NC(C)=O ZINC000217849561 BD On-Demand Unstable CTRA_BOVIN 17 43 COC(=O)[C@H](Cc1ccccc1)[C@H](C)NC(C)=O ZINC000217849561 BD On-Demand Unstable FCER2 81 38 COC(=O)[C@H](Cc1ccccc1)[C@H](C)NC(C)=O ZINC000217849561 BD On-Demand Unstable ACACA 16 41 COC(=O)[C@H](Cc1ccccc1)[C@H](C)NC(C)=O ZINC000217849561 BD On-Demand Unstable CTSB 54 42 COC(=O)[C@H](Cc1ccccc1)[C@H](C)NC(C)=O ZINC000217849561 BD On-Demand Unstable PAPA1_CARPA 74 55 COC(=O)[C@H](Cc1ccccc1)[C@H](C)NC(C)=O ZINC000217849561 BD On-Demand Unstable CYSP_TRYCR 48 38 COC(=O)[C@H](Cc1ccccc1)[C@H](C)NC(C)=O ZINC000217849561 BD On-Demand Unstable CTSL 34 41 COC(=O)[C@H](Cc1ccccc1)[C@H](C)NC(C)=O ZINC000217849561 BD On-Demand Unstable CPA1 57 41 COC(=O)[C@H](Cc1ccccc1)[C@H](C)NC(C)=O ZINC000217849561 BD On-Demand Unstable TIMP3 47 36 COC(=O)[C@H](Cc1ccccc1)[C@H](C)NC(C)=O ZINC000217849561 BD On-Demand Unstable CTRB1 34 44 COC(=O)[C@H](Cc1ccccc1)[C@H](C)NC(C)=O ZINC000217849561 BD On-Demand Unstable CAPNS1 61 40 COC(=O)[C@H](Cc1ccccc1)[C@H](C)NC(C)=O ZINC000217849561 BD On-Demand Unstable MMP3 24 41 COC(=O)[C@H](Cc1ccccc1)[C@H](C)NC(C)=O ZINC000217849561 BD On-Demand Unstable HLA-DRB1 56 37 COC(=O)[C@H](Cc1ccccc1)[C@H](C)NC(C)=O ZINC000217849561 BD On-Demand Unstable CTSS 23 41 COC(=O)[C@H](Cc1ccccc1)[C@H](C)NC(C)=O ZINC000217849561 BD On-Demand Unstable CAPN1 78 44 COC(=O)[C@H](Cc1ccccc1)[C@H](C)NC(C)=O ZINC000217849561 BD On-Demand Unstable CAPN2 77 38 COC(=O)[C@H](Cc1ccccc1)[C@H](C)NC(C)=O ZINC000217849561 BD On-Demand Unstable ACE2 90 41 COC(=O)[C@H](Cc1ccccc1)[C@H](C)NC(C)=O ZINC000217849561 BD On-Demand Unstable PLAU 30 42 COC(=O)[C@H](Cc1ccccc1)[C@H](C)NC(C)=O ZINC000217849561 BD On-Demand Unstable CTSC 26 40 COC(=O)[C@H](Cc1ccccc1)[C@H](C)NC(C)=O ZINC000217849561 BD On-Demand Unstable MMP1 28 42 COC(=O)[C@H](Cc1ccccc1)[C@H](C)NC(C)=O ZINC000217849561 BD On-Demand Unstable FPR1 51 37 COC(=O)[C@H](Cc1ccccc1)[C@H](C)NC(C)=O ZINC000217849561 BD On-Demand Unstable NPR 53 43 COC(=O)[C@H](Cc1ccccc1)[C@H](C)NC(C)=O ZINC000217849561 BD On-Demand Unstable AMP1_PLAFQ 54 40 Cc1ccc(OC[C@H](C)NC(=O)c2ccc(Cl)cc2)cc1 ZINC000217849562 DH In-Stock Unstable PTGS2 0 47 Cc1ccc(OC[C@H](C)NC(=O)c2ccc(Cl)cc2)cc1 ZINC000217849562 DH In-Stock Unstable SDH1 0 44 Cc1ccc(OC[C@H](C)NC(=O)c2ccc(Cl)cc2)cc1 ZINC000217849562 DH In-Stock Unstable CCR1 22 44 Cc1ccc(OC[C@H](C)NC(=O)c2ccc(Cl)cc2)cc1 ZINC000217849562 DH In-Stock Unstable TRPA1 17 48 Cc1ccc(OC[C@H](C)NC(=O)c2ccc(Cl)cc2)cc1 ZINC000217849562 DH In-Stock Unstable UTS2 68 47 Cc1ccc(OC[C@H](C)NC(=O)c2ccc(Cl)cc2)cc1 ZINC000217849562 DH In-Stock Unstable GPR88 0 40 O=C(N/C=C/c1ccccc1Br)NCCN1CCNCC1 ZINC000217849596 FD For-Sale Unstable PLD2 41 32 CCCC[C@@H](NC(=O)[C@@H]1C[C@@H](O)CN1)C(=O)O ZINC000217849598 BB For-Sale Unstable NOD1 84 40 Cc1nc2cc(NC(=O)CCCCCN3C(=O)c4ccccc4N4C(=O)c5ccccc5[C@H]34)ccc2[nH]1 ZINC000217849600 JK In-Stock Unstable GYRB 44 35 Cc1ccccc1[C@@H]1CCCN(C(=O)c2ccc(SCCO)cc2)C1 ZINC000217849601 FI In-Stock Unstable L3MBTL3 60 38 COc1cc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc(OC)c1 ZINC000217849619 FG For-Sale Unstable P2RY1 16 40 COc1cc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc(OC)c1 ZINC000217849619 FG For-Sale Unstable CCR3 57 44 COc1cc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc(OC)c1 ZINC000217849619 FG For-Sale Unstable MCHR1 15 48 COc1cc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc(OC)c1 ZINC000217849619 FG For-Sale Unstable ACKR3 61 32 O=C(Nc1ccc(C(F)(F)F)cc1)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217849641 II In-Stock Unstable BMP1 22 43 O=C(Nc1ccc(C(F)(F)F)cc1)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217849641 II In-Stock Unstable TRPV1 17 42 O=C(Nc1ccc(C(F)(F)F)cc1)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217849641 II In-Stock Unstable EPHX2 31 52 COC(=O)[C@@H](Cc1ccccc1)[C@@H](C)NC(C)=O ZINC000217849649 BD On-Demand Unstable PRSS1 20 54 COC(=O)[C@@H](Cc1ccccc1)[C@@H](C)NC(C)=O ZINC000217849649 BD On-Demand Unstable ACE 43 41 COC(=O)[C@@H](Cc1ccccc1)[C@@H](C)NC(C)=O ZINC000217849649 BD On-Demand Unstable OPRM1 36 44 COC(=O)[C@@H](Cc1ccccc1)[C@@H](C)NC(C)=O ZINC000217849649 BD On-Demand Unstable OPRD1 38 40 COC(=O)[C@@H](Cc1ccccc1)[C@@H](C)NC(C)=O ZINC000217849649 BD On-Demand Unstable MME 96 43 COC(=O)[C@@H](Cc1ccccc1)[C@@H](C)NC(C)=O ZINC000217849649 BD On-Demand Unstable LTA4H 15 43 COC(=O)[C@@H](Cc1ccccc1)[C@@H](C)NC(C)=O ZINC000217849649 BD On-Demand Unstable ANPEP 81 38 COC(=O)[C@@H](Cc1ccccc1)[C@@H](C)NC(C)=O ZINC000217849649 BD On-Demand Unstable TACR1 19 41 COC(=O)[C@@H](Cc1ccccc1)[C@@H](C)NC(C)=O ZINC000217849649 BD On-Demand Unstable CTRA_BOVIN 17 43 COC(=O)[C@@H](Cc1ccccc1)[C@@H](C)NC(C)=O ZINC000217849649 BD On-Demand Unstable FCER2 81 38 COC(=O)[C@@H](Cc1ccccc1)[C@@H](C)NC(C)=O ZINC000217849649 BD On-Demand Unstable ACACA 38 41 COC(=O)[C@@H](Cc1ccccc1)[C@@H](C)NC(C)=O ZINC000217849649 BD On-Demand Unstable CTSB 54 42 COC(=O)[C@@H](Cc1ccccc1)[C@@H](C)NC(C)=O ZINC000217849649 BD On-Demand Unstable PAPA1_CARPA 74 55 COC(=O)[C@@H](Cc1ccccc1)[C@@H](C)NC(C)=O ZINC000217849649 BD On-Demand Unstable CYSP_TRYCR 48 38 COC(=O)[C@@H](Cc1ccccc1)[C@@H](C)NC(C)=O ZINC000217849649 BD On-Demand Unstable CTSL 34 41 COC(=O)[C@@H](Cc1ccccc1)[C@@H](C)NC(C)=O ZINC000217849649 BD On-Demand Unstable CPA1 57 41 COC(=O)[C@@H](Cc1ccccc1)[C@@H](C)NC(C)=O ZINC000217849649 BD On-Demand Unstable TIMP3 47 36 COC(=O)[C@@H](Cc1ccccc1)[C@@H](C)NC(C)=O ZINC000217849649 BD On-Demand Unstable CTRB1 34 44 COC(=O)[C@@H](Cc1ccccc1)[C@@H](C)NC(C)=O ZINC000217849649 BD On-Demand Unstable CAPNS1 61 40 COC(=O)[C@@H](Cc1ccccc1)[C@@H](C)NC(C)=O ZINC000217849649 BD On-Demand Unstable MMP3 24 41 COC(=O)[C@@H](Cc1ccccc1)[C@@H](C)NC(C)=O ZINC000217849649 BD On-Demand Unstable HLA-DRB1 56 37 COC(=O)[C@@H](Cc1ccccc1)[C@@H](C)NC(C)=O ZINC000217849649 BD On-Demand Unstable CTSS 23 41 COC(=O)[C@@H](Cc1ccccc1)[C@@H](C)NC(C)=O ZINC000217849649 BD On-Demand Unstable CAPN1 78 44 COC(=O)[C@@H](Cc1ccccc1)[C@@H](C)NC(C)=O ZINC000217849649 BD On-Demand Unstable CAPN2 77 38 COC(=O)[C@@H](Cc1ccccc1)[C@@H](C)NC(C)=O ZINC000217849649 BD On-Demand Unstable ACE2 90 41 COC(=O)[C@@H](Cc1ccccc1)[C@@H](C)NC(C)=O ZINC000217849649 BD On-Demand Unstable PLAU 30 42 COC(=O)[C@@H](Cc1ccccc1)[C@@H](C)NC(C)=O ZINC000217849649 BD On-Demand Unstable CTSC 26 40 COC(=O)[C@@H](Cc1ccccc1)[C@@H](C)NC(C)=O ZINC000217849649 BD On-Demand Unstable MMP1 28 42 COC(=O)[C@@H](Cc1ccccc1)[C@@H](C)NC(C)=O ZINC000217849649 BD On-Demand Unstable FPR1 51 37 COC(=O)[C@@H](Cc1ccccc1)[C@@H](C)NC(C)=O ZINC000217849649 BD On-Demand Unstable NPR 53 43 COC(=O)[C@@H](Cc1ccccc1)[C@@H](C)NC(C)=O ZINC000217849649 BD On-Demand Unstable AMP1_PLAFQ 54 40 Cc1ccccc1[C@H]1CCCN(C(=O)c2ccc(SCCO)cc2)C1 ZINC000217849664 FI In-Stock Unstable L3MBTL3 60 38 CCCC[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1)C(=O)O ZINC000217849667 BB For-Sale Unstable NOD1 84 40 Cc1nc2cc(NC(=O)CCCCCN3C(=O)c4ccccc4N4C(=O)c5ccccc5[C@@H]34)ccc2[nH]1 ZINC000217849668 JK In-Stock Unstable GYRB 44 35 CC1CCN(c2ccc([C@@H](C)NC(=O)c3ccc(Cl)cc3)cc2)CC1 ZINC000217849677 FK In-Stock Unstable F10 20 42 CC1CCN(c2ccc([C@@H](C)NC(=O)c3ccc(Cl)cc3)cc2)CC1 ZINC000217849677 FK In-Stock Unstable PTGER4 25 41 CC1CCN(c2ccc([C@@H](C)NC(=O)c3ccc(Cl)cc3)cc2)CC1 ZINC000217849677 FK In-Stock Unstable SDH1 0 44 CC1CCN(c2ccc([C@@H](C)NC(=O)c3ccc(Cl)cc3)cc2)CC1 ZINC000217849677 FK In-Stock Unstable PRCP 22 42 CC1CCN(c2ccc([C@@H](C)NC(=O)c3ccc(Cl)cc3)cc2)CC1 ZINC000217849677 FK In-Stock Unstable CCR1 42 43 CC1CCN(c2ccc([C@@H](C)NC(=O)c3ccc(Cl)cc3)cc2)CC1 ZINC000217849677 FK In-Stock Unstable PRNP 47 38 CC1CCN(c2ccc([C@@H](C)NC(=O)c3ccc(Cl)cc3)cc2)CC1 ZINC000217849677 FK In-Stock Unstable UTS2 47 38 CCC(CC)N(C)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217849678 CG For-Sale Unstable PTGER2 28 43 CCC(CC)N(C)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217849678 CG For-Sale Unstable PTGER4 0 43 Cc1ccc(CNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217849718 EI For-Sale Unstable ANPEP 17 43 O=C(Nc1ccc(C(F)(F)F)cc1)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217849725 II In-Stock Unstable BMP1 22 43 O=C(Nc1ccc(C(F)(F)F)cc1)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217849725 II In-Stock Unstable TRPV1 17 42 O=C(Nc1ccc(C(F)(F)F)cc1)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217849725 II In-Stock Unstable EPHX2 31 52 COc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217849727 EG For-Sale Unstable ADRB1 15 41 COc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217849727 EG For-Sale Unstable TSHR 48 32 COc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217849727 EG For-Sale Unstable LPL 38 41 COc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217849727 EG For-Sale Unstable LTA4H 29 40 COc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217849727 EG For-Sale Unstable CA1 47 35 COc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217849727 EG For-Sale Unstable HRH3 15 43 COc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217849727 EG For-Sale Unstable NPY1R 28 41 COc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217849727 EG For-Sale Unstable P2RY1 40 38 COc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217849727 EG For-Sale Unstable CCR3 37 48 COc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217849727 EG For-Sale Unstable CHRNA7 15 41 COc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217849727 EG For-Sale Unstable MTNR1B 33 41 COc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217849727 EG For-Sale Unstable MTOR 45 34 COc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217849727 EG For-Sale Unstable EPHX2 48 46 COc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217849727 EG For-Sale Unstable CA12 20 40 COc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217849727 EG For-Sale Unstable CA9 19 40 COc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217849727 EG For-Sale Unstable MCHR1 19 54 COc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217849727 EG For-Sale Unstable LIPG 15 41 CC1CCN(c2ccc([C@H](C)NC(=O)c3ccc(Cl)cc3)cc2)CC1 ZINC000217849749 FK In-Stock Unstable F10 20 42 CC1CCN(c2ccc([C@H](C)NC(=O)c3ccc(Cl)cc3)cc2)CC1 ZINC000217849749 FK In-Stock Unstable PTGER4 25 41 CC1CCN(c2ccc([C@H](C)NC(=O)c3ccc(Cl)cc3)cc2)CC1 ZINC000217849749 FK In-Stock Unstable SDH1 0 44 CC1CCN(c2ccc([C@H](C)NC(=O)c3ccc(Cl)cc3)cc2)CC1 ZINC000217849749 FK In-Stock Unstable PRCP 22 42 CC1CCN(c2ccc([C@H](C)NC(=O)c3ccc(Cl)cc3)cc2)CC1 ZINC000217849749 FK In-Stock Unstable CCR1 42 43 CC1CCN(c2ccc([C@H](C)NC(=O)c3ccc(Cl)cc3)cc2)CC1 ZINC000217849749 FK In-Stock Unstable PRNP 47 38 CC1CCN(c2ccc([C@H](C)NC(=O)c3ccc(Cl)cc3)cc2)CC1 ZINC000217849749 FK In-Stock Unstable UTS2 47 38 CCCC[C@@H](NC(=O)[C@H]1C[C@@H](O)CN1)C(=O)O ZINC000217849754 BB For-Sale Unstable NOD1 84 40 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](CC(C)C)C(=O)Nc3ccc(C(N)=O)cc3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217849786 KI In-Stock Unstable TUBA1A 17 63 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](CC(C)C)C(=O)Nc3ccc(C(N)=O)cc3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217849786 KI In-Stock Unstable TPPP 0 60 COc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217849815 EG For-Sale Unstable ADRB1 15 41 COc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217849815 EG For-Sale Unstable TSHR 48 32 COc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217849815 EG For-Sale Unstable LPL 38 41 COc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217849815 EG For-Sale Unstable LTA4H 29 40 COc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217849815 EG For-Sale Unstable CA1 47 35 COc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217849815 EG For-Sale Unstable HRH3 15 43 COc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217849815 EG For-Sale Unstable NPY1R 28 41 COc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217849815 EG For-Sale Unstable P2RY1 40 38 COc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217849815 EG For-Sale Unstable CCR3 37 48 COc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217849815 EG For-Sale Unstable CHRNA7 15 41 COc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217849815 EG For-Sale Unstable MTNR1B 33 41 COc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217849815 EG For-Sale Unstable MTOR 45 34 COc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217849815 EG For-Sale Unstable EPHX2 48 46 COc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217849815 EG For-Sale Unstable CA12 20 40 COc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217849815 EG For-Sale Unstable CA9 19 40 COc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217849815 EG For-Sale Unstable MCHR1 19 54 COc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217849815 EG For-Sale Unstable LIPG 15 41 CCCC[C@H](NC(=O)[C@H]1C[C@@H](O)CN1)C(=O)O ZINC000217849835 BB For-Sale Unstable NOD1 84 40 Cc1ccccc1NC(=O)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217849842 GG In-Stock Unstable BMP1 23 43 Cc1ccccc1NC(=O)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217849842 GG In-Stock Unstable SMO 47 46 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)c3ccc(Cl)cc3)cc2)C1 ZINC000217849843 FK In-Stock Unstable F10 15 42 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)c3ccc(Cl)cc3)cc2)C1 ZINC000217849843 FK In-Stock Unstable SDH1 0 41 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)c3ccc(Cl)cc3)cc2)C1 ZINC000217849843 FK In-Stock Unstable HRH3 33 42 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)c3ccc(Cl)cc3)cc2)C1 ZINC000217849843 FK In-Stock Unstable PRCP 18 40 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)c3ccc(Cl)cc3)cc2)C1 ZINC000217849843 FK In-Stock Unstable CCR1 40 41 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)c3ccc(Cl)cc3)cc2)C1 ZINC000217849843 FK In-Stock Unstable ADAM17 0 40 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)c3ccc(Cl)cc3)cc2)C1 ZINC000217849843 FK In-Stock Unstable UTS2 48 38 O=C(O)/C=C\c1cc(Cn2cccnc2=O)ccc1F ZINC000217849880 CD For-Sale Unstable PTGER2 23 45 O=C(O)/C=C\c1cc(Cn2cccnc2=O)ccc1F ZINC000217849880 CD For-Sale Unstable PTGER4 0 45 O=C(O)/C=C\c1cc(Cn2cccnc2=O)ccc1F ZINC000217849880 CD For-Sale Unstable PTGER3 34 45 COc1cccc([C@@H]2CCCN2C(=O)c2cc3ccccc3cc2O)c1 ZINC000217849898 EJ On-Demand Unstable ADAM17 26 45 COc1cccc([C@@H]2CCCN2C(=O)c2cc3ccccc3cc2O)c1 ZINC000217849898 EJ On-Demand Unstable COLA 80 36 COc1cccc([C@@H]2CCCN2C(=O)c2cc3ccccc3cc2O)c1 ZINC000217849898 EJ On-Demand Unstable CPT1A 76 36 COc1cccc([C@@H]2CCCN2C(=O)c2cc3ccccc3cc2O)c1 ZINC000217849898 EJ On-Demand Unstable EBP 30 41 COc1cccc([C@@H]2CCCN2C(=O)c2cc3ccccc3cc2O)c1 ZINC000217849898 EJ On-Demand Unstable GPBAR1 0 44 COc1cccc([C@@H]2CCCN2C(=O)c2cc3ccccc3cc2O)c1 ZINC000217849898 EJ On-Demand Unstable NR1D1 28 42 Cc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217849922 DH For-Sale Unstable LPL 57 37 Cc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217849922 DH For-Sale Unstable CCR3 33 45 Cc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217849922 DH For-Sale Unstable MTOR 62 38 Cc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217849922 DH For-Sale Unstable EPHX2 38 42 C[C@H](NC(=O)c1ccc(Cl)cc1)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217849936 FK In-Stock Unstable F10 15 42 C[C@H](NC(=O)c1ccc(Cl)cc1)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217849936 FK In-Stock Unstable SDH1 0 41 C[C@H](NC(=O)c1ccc(Cl)cc1)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217849936 FK In-Stock Unstable HRH3 33 42 C[C@H](NC(=O)c1ccc(Cl)cc1)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217849936 FK In-Stock Unstable PRCP 18 40 C[C@H](NC(=O)c1ccc(Cl)cc1)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217849936 FK In-Stock Unstable CCR1 40 41 C[C@H](NC(=O)c1ccc(Cl)cc1)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217849936 FK In-Stock Unstable ADAM17 0 40 C[C@H](NC(=O)c1ccc(Cl)cc1)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217849936 FK In-Stock Unstable UTS2 48 38 Cc1ccccc1NC(=O)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217849940 GG In-Stock Unstable BMP1 23 43 Cc1ccccc1NC(=O)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217849940 GG In-Stock Unstable SMO 47 46 COc1cccc([C@H]2CCCN2C(=O)c2cc3ccccc3cc2O)c1 ZINC000217849983 EJ On-Demand Unstable ADAM17 26 45 COc1cccc([C@H]2CCCN2C(=O)c2cc3ccccc3cc2O)c1 ZINC000217849983 EJ On-Demand Unstable COLA 80 36 COc1cccc([C@H]2CCCN2C(=O)c2cc3ccccc3cc2O)c1 ZINC000217849983 EJ On-Demand Unstable CPT1A 76 36 COc1cccc([C@H]2CCCN2C(=O)c2cc3ccccc3cc2O)c1 ZINC000217849983 EJ On-Demand Unstable EBP 30 41 COc1cccc([C@H]2CCCN2C(=O)c2cc3ccccc3cc2O)c1 ZINC000217849983 EJ On-Demand Unstable GPBAR1 0 44 COc1cccc([C@H]2CCCN2C(=O)c2cc3ccccc3cc2O)c1 ZINC000217849983 EJ On-Demand Unstable NR1D1 28 42 Cc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217850000 DH For-Sale Unstable LPL 57 37 Cc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217850000 DH For-Sale Unstable CCR3 33 45 Cc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217850000 DH For-Sale Unstable MTOR 62 38 Cc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217850000 DH For-Sale Unstable EPHX2 38 42 O=C(N/C=C/c1ccccc1Br)NCCCN1CCOCC1 ZINC000217850029 FE For-Sale Unstable TACR2 27 40 O=C(N/C=C/c1ccccc1Br)NCCCN1CCOCC1 ZINC000217850029 FE For-Sale Unstable EPHX2 21 44 O=C(NCc1ccc(F)cc1)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217850035 GF In-Stock Unstable BMP1 17 42 O=C(NCc1ccc(F)cc1)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217850035 GF In-Stock Unstable CCR3 64 34 O=C(NCc1ccc(F)cc1)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217850035 GF In-Stock Unstable NAMPT 43 39 Cc1ccc2c(c1)[C@@H](NC(=O)c1ccc(Cl)cc1)CC(C)(C)O2 ZINC000217850047 EJ In-Stock Unstable ABCC9 40 48 Cc1ccc2c(c1)[C@@H](NC(=O)c1ccc(Cl)cc1)CC(C)(C)O2 ZINC000217850047 EJ In-Stock Unstable HCRTR2 0 43 CC(C)(F)COc1cccc(Br)c1 ZINC000217850048 BH For-Sale Unstable HMOX2 19 40 COc1ccc(Cn2ccnc2C)cc1/C=C\C(=O)O ZINC000217850049 CE For-Sale Unstable PTGER3 24 42 COc1cccc([C@@H]2CCCN2C(=O)c2cc(Br)ccc2O)c1 ZINC000217850106 GI On-Demand Unstable ADAM17 0 43 O=C(NCCCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217850113 EH For-Sale Unstable FKBP1A 32 45 O=C(NCCCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217850113 EH For-Sale Unstable SLC18A2 43 38 O=C(NCCCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217850113 EH For-Sale Unstable CCR3 18 44 O=C(NCCCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217850113 EH For-Sale Unstable PREP 64 38 O=C(NCc1ccc(F)cc1)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217850115 GF In-Stock Unstable BMP1 17 42 O=C(NCc1ccc(F)cc1)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217850115 GF In-Stock Unstable CCR3 64 34 O=C(NCc1ccc(F)cc1)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217850115 GF In-Stock Unstable NAMPT 43 39 Cc1ccc2c(c1)[C@H](NC(=O)c1ccc(Cl)cc1)CC(C)(C)O2 ZINC000217850126 EJ In-Stock Unstable ABCC9 40 48 Cc1ccc2c(c1)[C@H](NC(=O)c1ccc(Cl)cc1)CC(C)(C)O2 ZINC000217850126 EJ In-Stock Unstable HCRTR2 0 43 COc1ccc(CN2CCCCC2=O)cc1/C=C\C(=O)O ZINC000217850135 CE For-Sale Unstable PTGER2 31 55 COc1ccc(CN2CCCCC2=O)cc1/C=C\C(=O)O ZINC000217850135 CE For-Sale Unstable PTGER4 19 41 COc1cccc([C@H]2CCCN2C(=O)c2cc(Br)ccc2O)c1 ZINC000217850159 GI On-Demand Unstable ADAM17 0 43 C[C@H](F)CCOc1cccc(Br)c1 ZINC000217850184 BH On-Demand Unstable HMOX2 20 42 COCCNC(=O)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217850188 ED In-Stock Unstable BMP1 18 43 COCCNC(=O)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217850188 ED In-Stock Unstable PA 19 43 O=C(NCCCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217850211 EH For-Sale Unstable FKBP1A 32 45 O=C(NCCCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217850211 EH For-Sale Unstable SLC18A2 43 38 O=C(NCCCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217850211 EH For-Sale Unstable CCR3 18 44 O=C(NCCCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217850211 EH For-Sale Unstable PREP 64 38 Cc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1ccc(Cl)cc1 ZINC000217850230 EJ In-Stock Unstable ABCC9 32 43 COCCNC(=O)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217850261 ED In-Stock Unstable BMP1 18 43 COCCNC(=O)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217850261 ED In-Stock Unstable PA 19 43 C[C@@H](F)CCOc1cccc(Br)c1 ZINC000217850263 BH On-Demand Unstable HMOX2 20 42 Cc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1ccc(Cl)cc1 ZINC000217850301 EJ In-Stock Unstable ABCC9 32 43 CC[C@@H](C)N(C)CCNC(=O)CCCCC(=O)O ZINC000217850325 CD For-Sale Unstable DNM1 0 51 CC[C@@H](C)N(C)CCNC(=O)CCCCC(=O)O ZINC000217850325 CD For-Sale Unstable Q6UB75_PIG 0 40 COc1ccccc1NC(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217850328 EG For-Sale Unstable HTR1A 22 40 COc1ccccc1NC(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217850328 EG For-Sale Unstable DRD2 38 41 COc1ccccc1NC(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217850328 EG For-Sale Unstable CCR3 24 41 COc1ccccc1NC(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217850328 EG For-Sale Unstable ITGA4 34 42 COc1ccccc1NC(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217850328 EG For-Sale Unstable ACKR3 65 35 Cc1cccc(=O)n1Cc1ccccc1/C=C\C(=O)O ZINC000217850367 CE For-Sale Unstable PTGER2 48 49 Cc1cccc(=O)n1Cc1ccccc1/C=C\C(=O)O ZINC000217850367 CE For-Sale Unstable PTGER4 21 47 Cc1cccc(=O)n1Cc1ccccc1/C=C\C(=O)O ZINC000217850367 CE For-Sale Unstable PTGER3 22 49 Cc1cccc(=O)n1Cc1ccccc1/C=C\C(=O)O ZINC000217850367 CE For-Sale Unstable PTGDR 17 45 CC[C@H](C)N(C)CCNC(=O)CCCCC(=O)O ZINC000217850401 CD For-Sale Unstable DNM1 0 51 CC[C@H](C)N(C)CCNC(=O)CCCCC(=O)O ZINC000217850401 CD For-Sale Unstable Q6UB75_PIG 0 40 COc1ccccc1NC(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217850407 EG For-Sale Unstable HTR1A 22 40 COc1ccccc1NC(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217850407 EG For-Sale Unstable DRD2 38 41 COc1ccccc1NC(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217850407 EG For-Sale Unstable CCR3 24 41 COc1ccccc1NC(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217850407 EG For-Sale Unstable ITGA4 34 42 COc1ccccc1NC(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217850407 EG For-Sale Unstable ACKR3 65 35 COc1ccc2c(c1)[C@@H](NC(=O)c1ccc(Cl)cc1)CC(C)(C)O2 ZINC000217850426 EI In-Stock Unstable ABCC9 39 45 COc1ccc2c(c1)[C@@H](NC(=O)c1ccc(Cl)cc1)CC(C)(C)O2 ZINC000217850426 EI In-Stock Unstable PTGS2 31 41 COc1ccc2c(c1)[C@@H](NC(=O)c1ccc(Cl)cc1)CC(C)(C)O2 ZINC000217850426 EI In-Stock Unstable HCRTR2 0 45 COc1ccc2c(c1)[C@@H](NC(=O)c1ccc(Cl)cc1)CC(C)(C)O2 ZINC000217850426 EI In-Stock Unstable NAAA 22 44 COc1cccc([C@@H]2CCCN2C(=O)c2[nH]c3c(c2C)C(=O)CC(C)(C)C3)c1 ZINC000217850445 GI On-Demand Unstable GPBAR1 27 40 C[C@H]1CN([C@H](C)c2cccc(O)c2)CCN1C ZINC000217850464 BE For-Sale Unstable OPRM1 15 52 Cc1cccc(=O)n1Cc1ccc(/C=C\C(=O)O)cc1 ZINC000217850466 CE For-Sale Unstable PTGER2 20 40 COCCNC(=O)[C@H](CC(C)C)Nc1ccc2c(cc1=O)[C@@H](NC(C)=O)CCc1cc(OC)c(OC)c(OC)c1-2 ZINC000217850484 KG In-Stock Unstable TUBA1A 18 68 COCCNC(=O)[C@H](CC(C)C)Nc1ccc2c(cc1=O)[C@@H](NC(C)=O)CCc1cc(OC)c(OC)c(OC)c1-2 ZINC000217850484 KG In-Stock Unstable TPPP 0 64 CCN(C)C(=O)CNC(=O)c1cc(N)ccc1OC ZINC000217850485 CC For-Sale Unstable HTR4 29 45 COc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217850494 FG For-Sale Unstable HTR1A 15 40 COc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217850494 FG For-Sale Unstable DRD2 36 41 COc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217850494 FG For-Sale Unstable CCR3 21 40 COc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217850494 FG For-Sale Unstable ITGA4 50 41 COc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217850494 FG For-Sale Unstable MTNR1A 51 36 COc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217850494 FG For-Sale Unstable MTNR1B 53 36 COc1ccc(NC(=O)NC[C@@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217850494 FG For-Sale Unstable ACKR3 68 36 COc1ccc2c(c1)[C@H](NC(=O)c1ccc(Cl)cc1)CC(C)(C)O2 ZINC000217850505 EI In-Stock Unstable ABCC9 39 45 COc1ccc2c(c1)[C@H](NC(=O)c1ccc(Cl)cc1)CC(C)(C)O2 ZINC000217850505 EI In-Stock Unstable PTGS2 31 41 COc1ccc2c(c1)[C@H](NC(=O)c1ccc(Cl)cc1)CC(C)(C)O2 ZINC000217850505 EI In-Stock Unstable HCRTR2 0 45 COc1ccc2c(c1)[C@H](NC(=O)c1ccc(Cl)cc1)CC(C)(C)O2 ZINC000217850505 EI In-Stock Unstable NAAA 22 44 COc1cccc([C@H]2CCCN2C(=O)c2[nH]c3c(c2C)C(=O)CC(C)(C)C3)c1 ZINC000217850519 GI On-Demand Unstable GPBAR1 27 40 Cc1csc(NC(=O)N/C=C/c2ccccc2Br)n1 ZINC000217850559 EI For-Sale Unstable UL26 17 40 Cc1csc(NC(=O)N/C=C/c2ccccc2Br)n1 ZINC000217850559 EI For-Sale Unstable U53 0 40 Cc1csc(NC(=O)N/C=C/c2ccccc2Br)n1 ZINC000217850559 EI For-Sale Unstable SCAF_EBVB9 18 40 Cc1csc(NC(=O)N/C=C/c2ccccc2Br)n1 ZINC000217850559 EI For-Sale Unstable GCK 17 43 COc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217850574 FG For-Sale Unstable HTR1A 15 40 COc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217850574 FG For-Sale Unstable DRD2 36 41 COc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217850574 FG For-Sale Unstable CCR3 21 40 COc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217850574 FG For-Sale Unstable ITGA4 50 41 COc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217850574 FG For-Sale Unstable MTNR1A 51 36 COc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217850574 FG For-Sale Unstable MTNR1B 53 36 COc1ccc(NC(=O)NC[C@H]2CCCN2c2ccccc2)c(OC)c1 ZINC000217850574 FG For-Sale Unstable ACKR3 68 36 COC(=O)c1nc(NC(=O)CNc2ccc3c(cc2=O)[C@@H](NC(C)=O)CCc2cc(OC)c(OC)c(OC)c2-3)sc1-c1ccccc1 ZINC000217850603 KJ In-Stock Unstable TUBA1A 16 58 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1ccc(Cl)cc1 ZINC000217850604 EI In-Stock Unstable ABCC9 31 41 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1ccc(Cl)cc1 ZINC000217850604 EI In-Stock Unstable PTGS2 36 41 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1ccc(Cl)cc1 ZINC000217850604 EI In-Stock Unstable HCRTR2 0 41 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1ccc(Cl)cc1 ZINC000217850604 EI In-Stock Unstable NAAA 22 44 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1ccc(Cl)cc1 ZINC000217850686 EI In-Stock Unstable ABCC9 31 41 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1ccc(Cl)cc1 ZINC000217850686 EI In-Stock Unstable PTGS2 36 41 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1ccc(Cl)cc1 ZINC000217850686 EI In-Stock Unstable HCRTR2 0 41 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1ccc(Cl)cc1 ZINC000217850686 EI In-Stock Unstable NAAA 22 44 COc1ccc(CNC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217850689 FG For-Sale Unstable DRD2 43 42 COc1ccc(CNC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217850689 FG For-Sale Unstable ACHE 17 43 COc1ccc(CNC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217850689 FG For-Sale Unstable DRD3 26 41 COc1ccc(CNC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217850689 FG For-Sale Unstable HCRTR1 34 44 COc1ccc(CNC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217850689 FG For-Sale Unstable BCHE 17 43 COc1ccc(CNC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217850689 FG For-Sale Unstable NOS2 22 46 COc1ccc(CNC(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217850689 FG For-Sale Unstable ACKR3 69 39 CCc1ccc(-c2nc(CC(=O)N3CCC[C@@H]3c3cccc(OC)c3)cs2)cc1 ZINC000217850703 HK On-Demand Unstable AVPR1B 23 42 CCc1ccc(-c2nc(CC(=O)N3CCC[C@@H]3c3cccc(OC)c3)cs2)cc1 ZINC000217850703 HK On-Demand Unstable ADAM17 30 44 CCc1ccc(-c2nc(CC(=O)N3CCC[C@@H]3c3cccc(OC)c3)cs2)cc1 ZINC000217850703 HK On-Demand Unstable COLA 118 48 CCc1ccc(-c2nc(CC(=O)N3CCC[C@@H]3c3cccc(OC)c3)cs2)cc1 ZINC000217850703 HK On-Demand Unstable CPT1A 112 48 COc1cccc(NC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217850757 EI For-Sale Unstable CCKAR 0 40 COc1cccc(NC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217850757 EI For-Sale Unstable MTNR1A 22 45 COc1cccc(NC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217850757 EI For-Sale Unstable MTNR1B 28 45 COc1cccc(NC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217850757 EI For-Sale Unstable TAAR1 32 48 COc1cccc(NC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217850757 EI For-Sale Unstable AKR1C3 15 41 COc1cccc(NC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217850757 EI For-Sale Unstable KCNK3 81 47 COc1cccc(NC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217850757 EI For-Sale Unstable KCNK9 65 38 CC[C@@H](CO)NC(=O)c1cnn2ccccc12 ZINC000217850767 BC On-Demand Unstable JAK1 18 40 CC[C@@H](CO)NC(=O)c1cnn2ccccc12 ZINC000217850767 BC On-Demand Unstable TYK2 32 40 CC[C@@H](CO)NC(=O)c1cnn2ccccc12 ZINC000217850767 BC On-Demand Unstable EPHB3 37 51 COc1ccc(CNC(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217850772 FG For-Sale Unstable DRD2 43 42 COc1ccc(CNC(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217850772 FG For-Sale Unstable ACHE 17 43 COc1ccc(CNC(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217850772 FG For-Sale Unstable DRD3 26 41 COc1ccc(CNC(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217850772 FG For-Sale Unstable HCRTR1 34 44 COc1ccc(CNC(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217850772 FG For-Sale Unstable BCHE 17 43 COc1ccc(CNC(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217850772 FG For-Sale Unstable NOS2 22 46 COc1ccc(CNC(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217850772 FG For-Sale Unstable ACKR3 69 39 CCc1ccc(-c2nc(CC(=O)N3CCC[C@H]3c3cccc(OC)c3)cs2)cc1 ZINC000217850782 HK On-Demand Unstable AVPR1B 23 42 CCc1ccc(-c2nc(CC(=O)N3CCC[C@H]3c3cccc(OC)c3)cs2)cc1 ZINC000217850782 HK On-Demand Unstable ADAM17 30 44 CCc1ccc(-c2nc(CC(=O)N3CCC[C@H]3c3cccc(OC)c3)cs2)cc1 ZINC000217850782 HK On-Demand Unstable COLA 118 48 CCc1ccc(-c2nc(CC(=O)N3CCC[C@H]3c3cccc(OC)c3)cs2)cc1 ZINC000217850782 HK On-Demand Unstable CPT1A 112 48 CC[C@@H](NC(=O)c1ccc(Cl)cc1)c1ccc(C)c(C)c1 ZINC000217850796 DJ In-Stock Unstable UTS2 87 50 O=C(O)/C=C\c1ccccc1COc1ccccc1Cl ZINC000217850843 CI For-Sale Unstable PTGER2 25 56 O=C(O)/C=C\c1ccccc1COc1ccccc1Cl ZINC000217850843 CI For-Sale Unstable PTGER4 42 56 O=C(O)/C=C\c1ccccc1COc1ccccc1Cl ZINC000217850843 CI For-Sale Unstable CXCL8 38 47 O=C(O)/C=C\c1ccccc1COc1ccccc1Cl ZINC000217850843 CI For-Sale Unstable FABP4 22 50 O=C(O)/C=C\c1ccccc1COc1ccccc1Cl ZINC000217850843 CI For-Sale Unstable PTGER3 32 56 O=C(O)/C=C\c1ccccc1COc1ccccc1Cl ZINC000217850843 CI For-Sale Unstable PTGDR 0 47 O=C(O)/C=C\c1ccccc1COc1ccccc1Cl ZINC000217850843 CI For-Sale Unstable FABP5 34 50 O=C(N/C=C/c1ccccc1Br)Nc1cc(Cl)ccc1O ZINC000217850863 FJ For-Sale Anodyne KCNMA1 26 48 CC[C@H](NC(=O)c1ccc(Cl)cc1)c1ccc(C)c(C)c1 ZINC000217850865 DJ In-Stock Unstable UTS2 87 50 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)Nc3cccc(C)n3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217850873 KH In-Stock Unstable TUBA1A 19 68 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)Nc3cccc(C)n3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217850873 KH In-Stock Unstable TPPP 0 64 O=C(O)/C=C\c1ccc(COc2ccccc2Cl)cc1 ZINC000217850908 CI For-Sale Unstable PTGER2 24 51 O=C(O)/C=C\c1ccc(COc2ccccc2Cl)cc1 ZINC000217850908 CI For-Sale Unstable PPIA 41 32 O=C(O)/C=C\c1ccc(COc2ccccc2Cl)cc1 ZINC000217850908 CI For-Sale Unstable PTGER1 51 42 O=C(O)/C=C\c1ccc(COc2ccccc2Cl)cc1 ZINC000217850908 CI For-Sale Unstable PTGER4 42 50 O=C(O)/C=C\c1ccc(COc2ccccc2Cl)cc1 ZINC000217850908 CI For-Sale Unstable CXCL8 24 40 O=C(O)/C=C\c1ccc(COc2ccccc2Cl)cc1 ZINC000217850908 CI For-Sale Unstable FABP4 15 41 O=C(O)/C=C\c1ccc(COc2ccccc2Cl)cc1 ZINC000217850908 CI For-Sale Unstable PTGER3 30 51 O=C(O)/C=C\c1ccc(COc2ccccc2Cl)cc1 ZINC000217850908 CI For-Sale Unstable LTB4R 17 48 O=C(O)/C=C\c1ccc(COc2ccccc2Cl)cc1 ZINC000217850908 CI For-Sale Unstable PTGDR 0 42 O=C(O)/C=C\c1ccc(COc2ccccc2Cl)cc1 ZINC000217850908 CI For-Sale Unstable 17HSDCL 0 45 O=C(O)/C=C\c1ccc(COc2ccccc2Cl)cc1 ZINC000217850908 CI For-Sale Unstable FABP5 28 41 O=C(O)/C=C\c1ccc(COc2ccccc2Cl)cc1 ZINC000217850908 CI For-Sale Unstable AKR1C3 37 55 O=C(O)/C=C\c1ccc(COc2ccccc2Cl)cc1 ZINC000217850908 CI For-Sale Unstable AKR1B10 17 46 CC(=O)Nc1ccc(S(=O)(=O)N2CCC[C@H](Cc3nc(-c4cnccn4)no3)C2)cc1 ZINC000217850931 IE In-Stock Unstable BMP1 29 43 CC(=O)Nc1ccc(S(=O)(=O)N2CCC[C@H](Cc3nc(-c4cnccn4)no3)C2)cc1 ZINC000217850931 IE In-Stock Unstable IKBKB 17 43 CC(=O)Nc1ccc(S(=O)(=O)N2CCC[C@H](Cc3nc(-c4cnccn4)no3)C2)cc1 ZINC000217850931 IE In-Stock Unstable TGM2 40 35 CC(=O)Nc1ccc(S(=O)(=O)N2CCC[C@H](Cc3nc(-c4cnccn4)no3)C2)cc1 ZINC000217850931 IE In-Stock Unstable F13A1 62 35 CC(=O)Nc1ccc(S(=O)(=O)N2CCC[C@H](Cc3nc(-c4cnccn4)no3)C2)cc1 ZINC000217850931 IE In-Stock Unstable NAMPT 53 38 COc1cccc([C@@H]2CCCN2C(=O)CNC(=O)c2ccc(Br)cc2)c1 ZINC000217850934 HH On-Demand Unstable DRD4 48 37 COc1cccc([C@@H]2CCCN2C(=O)CNC(=O)c2ccc(Br)cc2)c1 ZINC000217850934 HH On-Demand Unstable CPT1A 87 39 COc1cccc([C@@H]2CCCN2C(=O)CNC(=O)c2ccc(Br)cc2)c1 ZINC000217850934 HH On-Demand Unstable DPP4 15 45 COc1cccc([C@@H]2CCCN2C(=O)CNC(=O)c2ccc(Br)cc2)c1 ZINC000217850934 HH On-Demand Unstable PREP 42 40 CC[C@@H](NC(=O)c1ccc(Cl)cc1)c1ccc(C)cc1C ZINC000217850968 DJ In-Stock Unstable CTSV 22 42 CC[C@@H](NC(=O)c1ccc(Cl)cc1)c1ccc(C)cc1C ZINC000217850968 DJ In-Stock Unstable UTS2 59 49 COc1cccc([C@H]2CCCN2C(=O)CNC(=O)c2ccc(Br)cc2)c1 ZINC000217850978 HH On-Demand Unstable DRD4 48 37 COc1cccc([C@H]2CCCN2C(=O)CNC(=O)c2ccc(Br)cc2)c1 ZINC000217850978 HH On-Demand Unstable CPT1A 87 39 COc1cccc([C@H]2CCCN2C(=O)CNC(=O)c2ccc(Br)cc2)c1 ZINC000217850978 HH On-Demand Unstable DPP4 15 45 COc1cccc([C@H]2CCCN2C(=O)CNC(=O)c2ccc(Br)cc2)c1 ZINC000217850978 HH On-Demand Unstable PREP 42 40 CC(=O)Nc1ccc(S(=O)(=O)N2CCC[C@@H](Cc3nc(-c4cnccn4)no3)C2)cc1 ZINC000217850993 IE In-Stock Unstable BMP1 29 43 CC(=O)Nc1ccc(S(=O)(=O)N2CCC[C@@H](Cc3nc(-c4cnccn4)no3)C2)cc1 ZINC000217850993 IE In-Stock Unstable IKBKB 17 43 CC(=O)Nc1ccc(S(=O)(=O)N2CCC[C@@H](Cc3nc(-c4cnccn4)no3)C2)cc1 ZINC000217850993 IE In-Stock Unstable TGM2 40 35 CC(=O)Nc1ccc(S(=O)(=O)N2CCC[C@@H](Cc3nc(-c4cnccn4)no3)C2)cc1 ZINC000217850993 IE In-Stock Unstable F13A1 62 35 CC(=O)Nc1ccc(S(=O)(=O)N2CCC[C@@H](Cc3nc(-c4cnccn4)no3)C2)cc1 ZINC000217850993 IE In-Stock Unstable NAMPT 53 38 O=C(O)/C=C\c1ccc(COc2ccccc2Cl)c(F)c1 ZINC000217851003 DI For-Sale Unstable PTGER2 46 43 O=C(O)/C=C\c1ccc(COc2ccccc2Cl)c(F)c1 ZINC000217851003 DI For-Sale Unstable PTGER1 50 43 O=C(O)/C=C\c1ccc(COc2ccccc2Cl)c(F)c1 ZINC000217851003 DI For-Sale Unstable PTGER4 21 42 O=C(O)/C=C\c1ccc(COc2ccccc2Cl)c(F)c1 ZINC000217851003 DI For-Sale Unstable FABP4 19 42 O=C(O)/C=C\c1ccc(COc2ccccc2Cl)c(F)c1 ZINC000217851003 DI For-Sale Unstable PTGER3 19 43 O=C(O)/C=C\c1ccc(COc2ccccc2Cl)c(F)c1 ZINC000217851003 DI For-Sale Unstable CDC25B 23 42 O=C(O)/C=C\c1ccc(COc2ccccc2Cl)c(F)c1 ZINC000217851003 DI For-Sale Unstable FABP5 28 42 O=C(O)/C=C\c1ccc(COc2ccccc2Cl)c(F)c1 ZINC000217851003 DI For-Sale Unstable AKR1C3 35 53 CC[C@H](NC(=O)c1ccc(Cl)cc1)c1ccc(C)cc1C ZINC000217851033 DJ In-Stock Unstable CTSV 22 42 CC[C@H](NC(=O)c1ccc(Cl)cc1)c1ccc(C)cc1C ZINC000217851033 DJ In-Stock Unstable UTS2 70 49 CC(C)S(=O)(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217851066 CD For-Sale Unstable NPY2R 21 42 CC(C)S(=O)(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217851066 CD For-Sale Unstable GRIA4 29 40 O=C(N/C=C/c1ccccc1Br)Nc1nccs1 ZINC000217851068 DH For-Sale Anodyne MAP1 114 39 O=C(O)/C=C\c1ccccc1COc1ccc(Cl)cc1 ZINC000217851081 CI For-Sale Unstable PTGER2 22 47 O=C(O)/C=C\c1ccccc1COc1ccc(Cl)cc1 ZINC000217851081 CI For-Sale Unstable PTGER4 30 47 O=C(O)/C=C\c1ccccc1COc1ccc(Cl)cc1 ZINC000217851081 CI For-Sale Unstable PTGER3 30 57 O=C(O)/C=C\c1ccccc1COc1ccc(Cl)cc1 ZINC000217851081 CI For-Sale Unstable CDC25B 24 43 O=C(O)/C=C\c1ccccc1COc1ccc(Cl)cc1 ZINC000217851081 CI For-Sale Unstable PTGDR 0 56 O=C(O)/C=C\c1ccccc1COc1ccc(Cl)cc1 ZINC000217851081 CI For-Sale Unstable FFAR1 24 48 O=C(O)/C=C\c1ccccc1COc1ccc(Cl)cc1 ZINC000217851081 CI For-Sale Unstable FFAR4 47 48 O=S(=O)(c1ccc2c(c1)OCCO2)N1CCC[C@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217851127 ID In-Stock Unstable PKM 35 41 CSc1cccc(NC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217851134 FJ For-Sale Unstable KCNK3 50 33 CC(C)S(=O)(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217851138 CD For-Sale Unstable NPY2R 21 42 CC(C)S(=O)(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217851138 CD For-Sale Unstable GRIA4 29 40 CC[C@@H](NC(=O)c1ccc(Cl)cc1)c1ccc(OC)c(OC)c1 ZINC000217851140 EI In-Stock Unstable PTGS2 0 40 CC[C@@H](NC(=O)c1ccc(Cl)cc1)c1ccc(OC)c(OC)c1 ZINC000217851140 EI In-Stock Unstable CMA1 27 42 CC[C@@H](NC(=O)c1ccc(Cl)cc1)c1ccc(OC)c(OC)c1 ZINC000217851140 EI In-Stock Unstable COLA 59 35 CC[C@@H](NC(=O)c1ccc(Cl)cc1)c1ccc(OC)c(OC)c1 ZINC000217851140 EI In-Stock Unstable CPT1A 55 33 CC[C@@H](NC(=O)c1ccc(Cl)cc1)c1ccc(OC)c(OC)c1 ZINC000217851140 EI In-Stock Unstable CPT1B 51 32 CC[C@@H](NC(=O)c1ccc(Cl)cc1)c1ccc(OC)c(OC)c1 ZINC000217851140 EI In-Stock Unstable UTS2 74 46 O=C(O)/C=C\c1ccc(COc2ccc(Cl)cc2)cc1 ZINC000217851160 CI For-Sale Unstable MAOB 29 52 O=C(O)/C=C\c1ccc(COc2ccc(Cl)cc2)cc1 ZINC000217851160 CI For-Sale Unstable PTGER2 41 44 O=C(O)/C=C\c1ccc(COc2ccc(Cl)cc2)cc1 ZINC000217851160 CI For-Sale Unstable PTGER4 28 43 O=C(O)/C=C\c1ccc(COc2ccc(Cl)cc2)cc1 ZINC000217851160 CI For-Sale Unstable PTPN2 0 46 O=C(O)/C=C\c1ccc(COc2ccc(Cl)cc2)cc1 ZINC000217851160 CI For-Sale Unstable PTGER3 19 46 O=C(O)/C=C\c1ccc(COc2ccc(Cl)cc2)cc1 ZINC000217851160 CI For-Sale Unstable CDC25B 22 44 O=C(O)/C=C\c1ccc(COc2ccc(Cl)cc2)cc1 ZINC000217851160 CI For-Sale Unstable PTGDR 0 46 O=C(O)/C=C\c1ccc(COc2ccc(Cl)cc2)cc1 ZINC000217851160 CI For-Sale Unstable ADAMTS4 24 41 O=C(O)/C=C\c1ccc(COc2ccc(Cl)cc2)cc1 ZINC000217851160 CI For-Sale Unstable 17HSDCL 0 41 O=C(O)/C=C\c1ccc(COc2ccc(Cl)cc2)cc1 ZINC000217851160 CI For-Sale Unstable FFAR1 37 43 O=C(O)/C=C\c1ccc(COc2ccc(Cl)cc2)cc1 ZINC000217851160 CI For-Sale Unstable AKR1C3 32 54 O=C(O)/C=C\c1ccc(COc2ccc(Cl)cc2)cc1 ZINC000217851160 CI For-Sale Unstable FFAR4 40 42 O=C(O)/C=C\c1ccc(COc2ccc(Cl)cc2)cc1 ZINC000217851160 CI For-Sale Unstable GPR183 0 42 O=S(=O)(c1ccc2c(c1)OCCO2)N1CCC[C@@H](Cc2nc(-c3cnccn3)no2)C1 ZINC000217851187 ID In-Stock Unstable PKM 35 41 CC[C@H](NC(=O)c1ccc(Cl)cc1)c1ccc(OC)c(OC)c1 ZINC000217851194 EI In-Stock Unstable PTGS2 0 40 CC[C@H](NC(=O)c1ccc(Cl)cc1)c1ccc(OC)c(OC)c1 ZINC000217851194 EI In-Stock Unstable CMA1 27 42 CC[C@H](NC(=O)c1ccc(Cl)cc1)c1ccc(OC)c(OC)c1 ZINC000217851194 EI In-Stock Unstable COLA 59 35 CC[C@H](NC(=O)c1ccc(Cl)cc1)c1ccc(OC)c(OC)c1 ZINC000217851194 EI In-Stock Unstable CPT1A 46 32 CC[C@H](NC(=O)c1ccc(Cl)cc1)c1ccc(OC)c(OC)c1 ZINC000217851194 EI In-Stock Unstable CPT1B 51 32 CC[C@H](NC(=O)c1ccc(Cl)cc1)c1ccc(OC)c(OC)c1 ZINC000217851194 EI In-Stock Unstable UTS2 74 46 O=C(N/C=C/c1ccccc1Br)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217851225 KH For-Sale Unstable LPL 55 44 O=C(N/C=C/c1ccccc1Br)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217851225 KH For-Sale Unstable LIPG 22 44 O=C(O)/C=C\c1ccc(COc2ccc(Cl)cc2)c(F)c1 ZINC000217851233 DI For-Sale Unstable PTGER4 28 44 O=C(O)/C=C\c1ccc(COc2ccc(Cl)cc2)c(F)c1 ZINC000217851233 DI For-Sale Unstable CDC25B 25 48 O=C(O)/C=C\c1ccc(COc2ccc(Cl)cc2)c(F)c1 ZINC000217851233 DI For-Sale Unstable FFAR1 15 40 O=C(O)/C=C\c1ccc(COc2ccc(Cl)cc2)c(F)c1 ZINC000217851233 DI For-Sale Unstable AKR1C3 32 46 O=C(O)/C=C\c1ccc(COc2ccc(Cl)cc2)c(F)c1 ZINC000217851233 DI For-Sale Unstable FFAR4 43 40 CC[C@@H](NC(=O)c1ccc(Cl)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217851250 FH In-Stock Unstable PTGS2 26 47 CC[C@@H](NC(=O)c1ccc(Cl)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217851250 FH In-Stock Unstable CA1 18 43 CC[C@@H](NC(=O)c1ccc(Cl)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217851250 FH In-Stock Unstable LOX1.1 43 41 CC[C@@H](NC(=O)c1ccc(Cl)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217851250 FH In-Stock Unstable O49150_SOLTU 51 41 CC[C@@H](NC(=O)c1ccc(Cl)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217851250 FH In-Stock Unstable UTS2 66 49 Cc1ccc(CN2CCN(CCC(=O)O)C[C@@H](O)C2)c(C)c1 ZINC000217851253 DD In-Stock Unstable SLC6A1 45 33 Cc1ccc2ccc(N3CCN[C@H](C(C)C)C3)nc2n1 ZINC000217851279 CE For-Sale Unstable PRKCQ 28 46 COc1cn(CC(=O)Nc2ccc(C(C)C)cc2)c(CO)cc1=O ZINC000217851301 EE In-Stock Unstable NR5A1 23 40 COc1cn(CC(=O)Nc2ccc(C(C)C)cc2)c(CO)cc1=O ZINC000217851301 EE In-Stock Unstable ENPP1 57 33 CC[C@H](NC(=O)c1ccc(Cl)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217851307 FH In-Stock Unstable PTGS2 26 47 CC[C@H](NC(=O)c1ccc(Cl)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217851307 FH In-Stock Unstable CA1 18 43 CC[C@H](NC(=O)c1ccc(Cl)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217851307 FH In-Stock Unstable LOX1.1 43 41 CC[C@H](NC(=O)c1ccc(Cl)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217851307 FH In-Stock Unstable O49150_SOLTU 51 41 CC[C@H](NC(=O)c1ccc(Cl)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217851307 FH In-Stock Unstable UTS2 66 49 Cc1cccc(C(=O)/C=C/c2ccc(F)cc2)c1O ZINC000217851309 CH For-Sale Unstable MAOB 15 50 Cc1ccc(C)c(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217851322 CH For-Sale Unstable PTGER2 30 61 Cc1ccc(C)c(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217851322 CH For-Sale Unstable PTGER4 44 56 Cc1ccc(C)c(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217851322 CH For-Sale Unstable PTGER3 34 61 Cc1ccc(C)c(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217851322 CH For-Sale Unstable PTGDR 0 46 Cc1ccc(C)c(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217851322 CH For-Sale Unstable AKR1C3 31 41 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217851343 HF For-Sale Unstable CA2 110 58 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217851343 HF For-Sale Unstable CA1 95 58 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217851343 HF For-Sale Unstable CA7 57 55 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217851343 HF For-Sale Unstable CA5B 65 55 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217851343 HF For-Sale Unstable CA4 74 56 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217851343 HF For-Sale Unstable CA5A 70 55 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217851343 HF For-Sale Unstable CA14 41 49 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217851343 HF For-Sale Unstable CA12 72 58 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217851343 HF For-Sale Unstable CA9 80 58 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217851343 HF For-Sale Unstable CYNT 29 43 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217851343 HF For-Sale Unstable NCE103 37 40 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217851343 HF For-Sale Unstable LIG1 0 40 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217851343 HF For-Sale Unstable MTCA1 47 53 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217851343 HF For-Sale Unstable P96878_MYCTU 60 53 Cc1ccc2ccc(N3CCN[C@@H](C(C)C)C3)nc2n1 ZINC000217851366 CE For-Sale Unstable PRKCQ 28 46 Cc1ccc([C@@H](C)N2CC[C@@H](N3CCCC3)C2)c(O)c1 ZINC000217851384 CF For-Sale Unstable L3MBTL3 54 35 Cc1ccc([C@@H](C)N2CC[C@@H](N3CCCC3)C2)c(O)c1 ZINC000217851384 CF For-Sale Unstable MBTD1 0 42 Cc1ccc(C)c(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217851394 CH For-Sale Unstable PTGER2 24 52 Cc1ccc(C)c(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217851394 CH For-Sale Unstable PTGER4 33 43 Cc1ccc(C)c(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217851394 CH For-Sale Unstable PTGER3 25 52 Cc1ccc(C)c(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217851394 CH For-Sale Unstable AKR1C3 37 55 O=C(CCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)Nc1nc2c(s1)CCC2 ZINC000217851403 IH In-Stock Unstable SLC27A1 32 45 CCCCS(=O)(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217851405 CE For-Sale Unstable ADAMTS5 32 40 O=C(N/C=C/c1ccccc1Br)Nc1cccnc1Cl ZINC000217851439 FI For-Sale Anodyne G2YM83_BOTF4 45 33 COc1ccc(-c2noc(CNC(=O)c3ccc(Cl)cc3)n2)c(OC)c1 ZINC000217851444 FG In-Stock Unstable PTGS2 38 42 COc1ccc(-c2noc(CNC(=O)c3ccc(Cl)cc3)n2)c(OC)c1 ZINC000217851444 FG In-Stock Unstable F10 47 32 COc1ccc(-c2noc(CNC(=O)c3ccc(Cl)cc3)n2)c(OC)c1 ZINC000217851444 FG In-Stock Unstable HRH3 19 40 COc1ccc(-c2noc(CNC(=O)c3ccc(Cl)cc3)n2)c(OC)c1 ZINC000217851444 FG In-Stock Unstable COLA 52 33 COc1ccc(-c2noc(CNC(=O)c3ccc(Cl)cc3)n2)c(OC)c1 ZINC000217851444 FG In-Stock Unstable CPT1A 48 33 COc1ccc(-c2noc(CNC(=O)c3ccc(Cl)cc3)n2)c(OC)c1 ZINC000217851444 FG In-Stock Unstable PPARD 20 44 COc1ccc(-c2noc(CNC(=O)c3ccc(Cl)cc3)n2)c(OC)c1 ZINC000217851444 FG In-Stock Unstable CPT1B 49 33 COc1ccc(-c2noc(CNC(=O)c3ccc(Cl)cc3)n2)c(OC)c1 ZINC000217851444 FG In-Stock Unstable PDK1 29 42 COc1ccc(-c2noc(CNC(=O)c3ccc(Cl)cc3)n2)c(OC)c1 ZINC000217851444 FG In-Stock Unstable MT-ND1 18 45 COc1ccc(-c2noc(CNC(=O)c3ccc(Cl)cc3)n2)c(OC)c1 ZINC000217851444 FG In-Stock Unstable U38 0 42 Cc1ccc([C@H](C)N2CC[C@@H](N3CCCC3)C2)c(O)c1 ZINC000217851451 CF For-Sale Unstable L3MBTL3 54 35 Cc1ccc([C@H](C)N2CC[C@@H](N3CCCC3)C2)c(O)c1 ZINC000217851451 CF For-Sale Unstable MBTD1 0 42 CCCCS(=O)(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217851479 CE For-Sale Unstable ADAMTS5 32 40 O=C(CCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)Nc1nc2c(s1)CCC2 ZINC000217851490 IH In-Stock Unstable SLC27A1 32 45 Cc1ccc(C)c(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217851492 CH For-Sale Unstable MAOB 18 45 Cc1ccc(C)c(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217851492 CH For-Sale Unstable PTGER2 29 54 Cc1ccc(C)c(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217851492 CH For-Sale Unstable PTGER1 25 40 Cc1ccc(C)c(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217851492 CH For-Sale Unstable PTGER4 36 44 Cc1ccc(C)c(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217851492 CH For-Sale Unstable PTGER3 28 53 Cc1ccc(C)c(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217851492 CH For-Sale Unstable LTB4R 17 44 Cc1ccc(C)c(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217851492 CH For-Sale Unstable KCNA3 0 40 Cc1ccc(C)c(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217851492 CH For-Sale Unstable FFAR1 42 43 Cc1ccc(C)c(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217851492 CH For-Sale Unstable AKR1C3 43 53 Oc1ccc2c(c1)CCC[C@@H]2N1CC[C@@H](N2CCCC2)C1 ZINC000217851551 CF For-Sale Unstable SLC6A1 0 41 Oc1ccc2c(c1)CCC[C@@H]2N1CC[C@@H](N2CCCC2)C1 ZINC000217851551 CF For-Sale Unstable DRD5 20 50 Oc1ccc2c(c1)CCC[C@@H]2N1CC[C@@H](N2CCCC2)C1 ZINC000217851551 CF For-Sale Unstable L3MBTL3 75 36 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccccc1 ZINC000217851618 DF For-Sale Unstable NPY1R 42 35 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccccc1 ZINC000217851618 DF For-Sale Unstable NPY2R 49 39 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccccc1 ZINC000217851618 DF For-Sale Unstable ADAMTS5 37 46 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccccc1 ZINC000217851618 DF For-Sale Unstable SFRP1 76 33 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccccc1 ZINC000217851618 DF For-Sale Unstable WNT3 53 32 Oc1ccc2c(c1)CCC[C@H]2N1CC[C@@H](N2CCCC2)C1 ZINC000217851642 CF For-Sale Unstable SLC6A1 0 41 Oc1ccc2c(c1)CCC[C@H]2N1CC[C@@H](N2CCCC2)C1 ZINC000217851642 CF For-Sale Unstable DRD5 20 50 Oc1ccc2c(c1)CCC[C@H]2N1CC[C@@H](N2CCCC2)C1 ZINC000217851642 CF For-Sale Unstable L3MBTL3 75 36 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1 ZINC000217851671 DF For-Sale Unstable NPY1R 42 35 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1 ZINC000217851671 DF For-Sale Unstable NPY2R 49 39 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1 ZINC000217851671 DF For-Sale Unstable ADAMTS5 37 46 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1 ZINC000217851671 DF For-Sale Unstable SFRP1 76 33 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1 ZINC000217851671 DF For-Sale Unstable WNT3 53 32 CC(C)c1ccc(CCCNC(=O)c2ccc(Cl)cc2)cc1 ZINC000217851725 DJ In-Stock Unstable GCGR 42 39 CC(C)c1ccc(CCCNC(=O)c2ccc(Cl)cc2)cc1 ZINC000217851725 DJ In-Stock Unstable TBXAS1 0 40 CC(C)c1ccc(CCCNC(=O)c2ccc(Cl)cc2)cc1 ZINC000217851725 DJ In-Stock Unstable ECR 29 40 CC(C)c1ccc(CCCNC(=O)c2ccc(Cl)cc2)cc1 ZINC000217851725 DJ In-Stock Unstable HDA106 0 50 CC(C)c1ccc(CCCNC(=O)c2ccc(Cl)cc2)cc1 ZINC000217851725 DJ In-Stock Unstable MCL1 0 45 CC(C)c1ccc(CCCNC(=O)c2ccc(Cl)cc2)cc1 ZINC000217851725 DJ In-Stock Unstable UTS2 50 40 CC(C)c1ccc(CCCNC(=O)c2ccc(Cl)cc2)cc1 ZINC000217851725 DJ In-Stock Unstable E3UJZ5_SPOLI 30 40 Oc1cccc2c1CC[C@@H]2N1CC[C@@H](N2CCCC2)C1 ZINC000217851756 CF For-Sale Unstable SLC6A1 0 40 Oc1cccc2c1CC[C@@H]2N1CC[C@@H](N2CCCC2)C1 ZINC000217851756 CF For-Sale Unstable L3MBTL3 101 40 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1cccs1 ZINC000217851765 DF For-Sale Unstable ADAMTS5 32 41 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1cccs1 ZINC000217851765 DF For-Sale Unstable GCKR 34 41 CCN1CCC[C@@H]1CNC(=O)CCN1C(=O)c2ccccc2N2C(=O)c3c(ccc(OC)c3OC)[C@H]12 ZINC000217851768 JF In-Stock Unstable DRD2 39 45 CCN1CCC[C@@H]1CNC(=O)CCN1C(=O)c2ccccc2N2C(=O)c3c(ccc(OC)c3OC)[C@H]12 ZINC000217851768 JF In-Stock Unstable ACKR3 50 31 C[C@@H](C(=O)NCc1cnn(C)c1)c1ccc(-c2ccccc2)c(F)c1 ZINC000217851770 EH In-Stock Unstable TRPV1 102 41 C[C@@H](C(=O)NCc1cnn(C)c1)c1ccc(-c2ccccc2)c(F)c1 ZINC000217851770 EH In-Stock Unstable BCHE 23 49 CCOC(=O)CN1C[C@]2(CCCN2C(C)=O)C1=O ZINC000217851806 CB For-Sale Unstable SLC12A5 52 34 C[C@H](C(=O)NCc1cnn(C)c1)c1ccc(-c2ccccc2)c(F)c1 ZINC000217851812 EH In-Stock Unstable TRPV1 102 41 C[C@H](C(=O)NCc1cnn(C)c1)c1ccc(-c2ccccc2)c(F)c1 ZINC000217851812 EH In-Stock Unstable BCHE 23 49 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1cccs1 ZINC000217851822 DF For-Sale Unstable ADAMTS5 32 41 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1cccs1 ZINC000217851822 DF For-Sale Unstable GCKR 34 41 Oc1cccc2c1CC[C@H]2N1CC[C@@H](N2CCCC2)C1 ZINC000217851830 CF For-Sale Unstable SLC6A1 0 40 Oc1cccc2c1CC[C@H]2N1CC[C@@H](N2CCCC2)C1 ZINC000217851830 CF For-Sale Unstable L3MBTL3 101 40 CCN1CCC[C@H]1CNC(=O)CCN1C(=O)c2ccccc2N2C(=O)c3c(ccc(OC)c3OC)[C@H]12 ZINC000217851833 JF In-Stock Unstable DRD2 39 45 CCN1CCC[C@H]1CNC(=O)CCN1C(=O)c2ccccc2N2C(=O)c3c(ccc(OC)c3OC)[C@H]12 ZINC000217851833 JF In-Stock Unstable ACKR3 50 31 O=C(NCCCN1CCCc2ccccc21)c1ccc(Cl)cc1 ZINC000217851863 EH In-Stock Unstable HTR1A 20 44 O=C(NCCCN1CCCc2ccccc21)c1ccc(Cl)cc1 ZINC000217851863 EH In-Stock Unstable DRD2 37 51 O=C(NCCCN1CCCc2ccccc21)c1ccc(Cl)cc1 ZINC000217851863 EH In-Stock Unstable DRD1 29 42 O=C(NCCCN1CCCc2ccccc21)c1ccc(Cl)cc1 ZINC000217851863 EH In-Stock Unstable DRD4 46 37 O=C(NCCCN1CCCc2ccccc21)c1ccc(Cl)cc1 ZINC000217851863 EH In-Stock Unstable HTR2C 28 52 O=C(NCCCN1CCCc2ccccc21)c1ccc(Cl)cc1 ZINC000217851863 EH In-Stock Unstable AVPR2 43 44 O=C(NCCCN1CCCc2ccccc21)c1ccc(Cl)cc1 ZINC000217851863 EH In-Stock Unstable DRD3 63 51 O=C(NCCCN1CCCc2ccccc21)c1ccc(Cl)cc1 ZINC000217851863 EH In-Stock Unstable APP 33 40 O=C(NCCCN1CCCc2ccccc21)c1ccc(Cl)cc1 ZINC000217851863 EH In-Stock Unstable HTR3B 0 41 O=C(NCCCN1CCCc2ccccc21)c1ccc(Cl)cc1 ZINC000217851863 EH In-Stock Unstable PLD2 53 42 O=C(NCCCN1CCCc2ccccc21)c1ccc(Cl)cc1 ZINC000217851863 EH In-Stock Unstable TYRO3 23 40 O=C(NCCCN1CCCc2ccccc21)c1ccc(Cl)cc1 ZINC000217851863 EH In-Stock Unstable NOD1 26 41 CCOC(=O)CN1C[C@@]2(CCCN2C(C)=O)C1=O ZINC000217851877 CB For-Sale Unstable SLC12A5 52 34 C[C@@H](c1ccc(O)cc1)N1CC[C@@H](N2CCCC2)C1 ZINC000217851927 CF For-Sale Unstable CHRM2 19 42 C[C@@H](c1ccc(O)cc1)N1CC[C@@H](N2CCCC2)C1 ZINC000217851927 CF For-Sale Unstable L3MBTL3 76 38 NC(=O)[C@H]1CCCN1Cc1cccc(/C=C\C(=O)O)c1 ZINC000217851950 CD For-Sale Unstable PREP 53 37 COc1ccccc1CCCNC(=O)c1cccc(Cl)c1 ZINC000217851997 DH In-Stock Unstable HTR1A 25 48 COc1ccccc1CCCNC(=O)c1cccc(Cl)c1 ZINC000217851997 DH In-Stock Unstable DRD2 38 53 COc1ccccc1CCCNC(=O)c1cccc(Cl)c1 ZINC000217851997 DH In-Stock Unstable DRD1 23 46 COc1ccccc1CCCNC(=O)c1cccc(Cl)c1 ZINC000217851997 DH In-Stock Unstable DRD4 51 41 COc1ccccc1CCCNC(=O)c1cccc(Cl)c1 ZINC000217851997 DH In-Stock Unstable ACHE 22 43 COc1ccccc1CCCNC(=O)c1cccc(Cl)c1 ZINC000217851997 DH In-Stock Unstable DRD3 66 48 COc1ccccc1CCCNC(=O)c1cccc(Cl)c1 ZINC000217851997 DH In-Stock Unstable NQO2 19 46 COc1ccccc1CCCNC(=O)c1cccc(Cl)c1 ZINC000217851997 DH In-Stock Unstable ECR 27 40 COc1ccccc1CCCNC(=O)c1cccc(Cl)c1 ZINC000217851997 DH In-Stock Unstable CTSL 21 42 COc1ccccc1CCCNC(=O)c1cccc(Cl)c1 ZINC000217851997 DH In-Stock Unstable CPT1A 46 32 COc1ccccc1CCCNC(=O)c1cccc(Cl)c1 ZINC000217851997 DH In-Stock Unstable MTNR1A 57 40 COc1ccccc1CCCNC(=O)c1cccc(Cl)c1 ZINC000217851997 DH In-Stock Unstable MTNR1B 57 45 COc1ccccc1CCCNC(=O)c1cccc(Cl)c1 ZINC000217851997 DH In-Stock Unstable CCKBR 0 43 COc1ccccc1CCCNC(=O)c1cccc(Cl)c1 ZINC000217851997 DH In-Stock Unstable SLC6A5 31 40 COc1ccccc1CCCNC(=O)c1cccc(Cl)c1 ZINC000217851997 DH In-Stock Unstable CTSV 29 42 COc1ccccc1CCCNC(=O)c1cccc(Cl)c1 ZINC000217851997 DH In-Stock Unstable PTGDR 27 41 COc1ccccc1CCCNC(=O)c1cccc(Cl)c1 ZINC000217851997 DH In-Stock Unstable MCHR1 15 46 COc1ccccc1CCCNC(=O)c1cccc(Cl)c1 ZINC000217851997 DH In-Stock Unstable PTGDR2 19 41 COc1ccccc1CCCNC(=O)c1cccc(Cl)c1 ZINC000217851997 DH In-Stock Unstable CACNA1I 38 42 COc1ccccc1CCCNC(=O)c1cccc(Cl)c1 ZINC000217851997 DH In-Stock Unstable MBTPS1 48 32 COc1ccccc1CCCNC(=O)c1cccc(Cl)c1 ZINC000217851997 DH In-Stock Unstable AP2S1 0 42 COc1ccccc1CCCNC(=O)c1cccc(Cl)c1 ZINC000217851997 DH In-Stock Unstable ALPHA-1A 0 44 COc1ccccc1CCCNC(=O)c1cccc(Cl)c1 ZINC000217851997 DH In-Stock Unstable KCNK3 50 39 COc1ccccc1CCCNC(=O)c1cccc(Cl)c1 ZINC000217851997 DH In-Stock Unstable KCNK9 43 39 COc1ccccc1CCCNC(=O)c1cccc(Cl)c1 ZINC000217851997 DH In-Stock Unstable LMGT2 0 45 C[C@H](c1ccc(O)cc1)N1CC[C@@H](N2CCCC2)C1 ZINC000217852031 CF For-Sale Unstable CHRM2 19 42 C[C@H](c1ccc(O)cc1)N1CC[C@@H](N2CCCC2)C1 ZINC000217852031 CF For-Sale Unstable L3MBTL3 76 38 C[C@@H](c1ccc(F)cc1O)N1CC[C@@H](N2CCCC2)C1 ZINC000217852108 CF For-Sale Unstable L3MBTL3 55 34 C[C@@H](c1ccc(F)cc1O)N1CC[C@@H](N2CCCC2)C1 ZINC000217852108 CF For-Sale Unstable MBTD1 0 41 COc1ccc(F)cc1-c1ccnc2[nH]c([C@]3(O)CCNC3)cc12 ZINC000217852111 EF For-Sale Unstable CSNK1G2 44 32 CCCOc1ccccc1CCCNC(=O)c1cccc(Cl)c1 ZINC000217852112 EI In-Stock Unstable DRD4 43 34 CCCOc1ccccc1CCCNC(=O)c1cccc(Cl)c1 ZINC000217852112 EI In-Stock Unstable DRD3 37 40 CCCOc1ccccc1CCCNC(=O)c1cccc(Cl)c1 ZINC000217852112 EI In-Stock Unstable MTNR1B 53 40 CCCOc1ccccc1CCCNC(=O)c1cccc(Cl)c1 ZINC000217852112 EI In-Stock Unstable ALPHA-1A 0 40 CCCOc1ccccc1CCCNC(=O)c1cccc(Cl)c1 ZINC000217852112 EI In-Stock Unstable LMGT2 0 42 Cc1cccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217852130 EF For-Sale Unstable NPY2R 51 40 Cc1cccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217852130 EF For-Sale Unstable ADAMTS5 32 40 COc1cc([C@@H]2CC(=O)Oc3c2c2nc4ccccc4nc2c2ccccc32)ccc1OCC(=O)O ZINC000217852131 JJ In-Stock Unstable PTGIR 42 34 CCN(Cc1cc(/C=C\C(=O)O)ccc1OC)C1CC1 ZINC000217852166 CF For-Sale Unstable PTGER2 0 42 CCN(Cc1cc(/C=C\C(=O)O)ccc1OC)C1CC1 ZINC000217852166 CF For-Sale Unstable AKR1C3 37 40 COc1ccc(F)cc1-c1ccnc2[nH]c([C@@]3(O)CCNC3)cc12 ZINC000217852187 EF For-Sale Unstable CSNK1G2 44 32 C[C@H](c1ccc(F)cc1O)N1CC[C@@H](N2CCCC2)C1 ZINC000217852189 CF For-Sale Unstable L3MBTL3 55 34 C[C@H](c1ccc(F)cc1O)N1CC[C@@H](N2CCCC2)C1 ZINC000217852189 CF For-Sale Unstable MBTD1 0 41 Cc1cccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217852201 EF For-Sale Unstable NPY2R 51 40 Cc1cccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217852201 EF For-Sale Unstable ADAMTS5 32 40 COc1cc([C@H]2CC(=O)Oc3c2c2nc4ccccc4nc2c2ccccc32)ccc1OCC(=O)O ZINC000217852231 JJ In-Stock Unstable PTGIR 42 34 CC1CCN(c2ccc([C@@H](C)NC(=O)c3cccc(Cl)c3)cc2)CC1 ZINC000217852232 FK In-Stock Unstable F10 15 42 CC1CCN(c2ccc([C@@H](C)NC(=O)c3cccc(Cl)c3)cc2)CC1 ZINC000217852232 FK In-Stock Unstable PTGER4 24 41 CC1CCN(c2ccc([C@@H](C)NC(=O)c3cccc(Cl)c3)cc2)CC1 ZINC000217852232 FK In-Stock Unstable PRKD1 30 40 CC1CCN(c2ccc([C@@H](C)NC(=O)c3cccc(Cl)c3)cc2)CC1 ZINC000217852232 FK In-Stock Unstable CCKBR 0 42 CC1CCN(c2ccc([C@@H](C)NC(=O)c3cccc(Cl)c3)cc2)CC1 ZINC000217852232 FK In-Stock Unstable PTGDR 0 40 CC[C@@H](C)N(CC)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217852270 CG For-Sale Unstable TUBB1 42 38 CC[C@@H](C)N(CC)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217852270 CG For-Sale Unstable AKR1C3 31 42 C[C@@H](Cc1ccc(O)cc1)N1CC[C@@H](N2CCCC2)C1 ZINC000217852279 CE For-Sale Unstable L3MBTL3 85 37 CN1CCO[C@@H]([C@@H](O)Cc2ccc(F)cc2Cl)C1 ZINC000217852282 CD For-Sale Unstable P2RX7 47 39 Cc1cccc2[nH]c(-c3ccc(O)c(O)c3)nc12 ZINC000217852295 BF For-Sale Unstable PARP2 42 39 Cc1cccc2[nH]c(-c3ccc(O)c(O)c3)nc12 ZINC000217852295 BF For-Sale Unstable HPSE 16 51 Cc1cccc2[nH]c(-c3ccc(O)c(O)c3)nc12 ZINC000217852295 BF For-Sale Unstable PARP1 39 50 Cc1cccc2[nH]c(-c3ccc(O)c(O)c3)nc12 ZINC000217852295 BF For-Sale Unstable TNKS 39 47 Cc1cccc2[nH]c(-c3ccc(O)c(O)c3)nc12 ZINC000217852295 BF For-Sale Unstable TNKS2 25 47 CC1CCN(c2ccc([C@H](C)NC(=O)c3cccc(Cl)c3)cc2)CC1 ZINC000217852298 FK In-Stock Unstable F10 15 42 CC1CCN(c2ccc([C@H](C)NC(=O)c3cccc(Cl)c3)cc2)CC1 ZINC000217852298 FK In-Stock Unstable PTGER4 24 41 CC1CCN(c2ccc([C@H](C)NC(=O)c3cccc(Cl)c3)cc2)CC1 ZINC000217852298 FK In-Stock Unstable PRKD1 30 40 CC1CCN(c2ccc([C@H](C)NC(=O)c3cccc(Cl)c3)cc2)CC1 ZINC000217852298 FK In-Stock Unstable CCKBR 0 42 CC1CCN(c2ccc([C@H](C)NC(=O)c3cccc(Cl)c3)cc2)CC1 ZINC000217852298 FK In-Stock Unstable PTGDR 0 40 CCO[C@@H](CN)CN1C[C@@H](C)Cc2ccccc21 ZINC000217852304 BE For-Sale Unstable TPP2 57 32 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccccc1F ZINC000217852323 EF For-Sale Unstable NPY1R 43 35 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccccc1F ZINC000217852323 EF For-Sale Unstable NPY2R 47 37 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccccc1F ZINC000217852323 EF For-Sale Unstable ADAMTS5 35 40 O=C(C[C@@H](c1coc2ccccc2c1=O)c1c(O)c(O)c(O)c2c(=O)cc(-c3ccccc3)oc12)N1CCOCC1 ZINC000217852340 KI In-Stock Unstable PRKDC 34 41 CC[C@H](C)N(CC)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217852356 CG For-Sale Unstable TUBB1 42 38 CC[C@H](C)N(CC)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217852356 CG For-Sale Unstable AKR1C3 31 42 CN1CCO[C@H]([C@@H](O)Cc2ccc(F)cc2Cl)C1 ZINC000217852360 CD For-Sale Unstable P2RX7 47 39 C[C@H](Cc1ccc(O)cc1)N1CC[C@@H](N2CCCC2)C1 ZINC000217852375 CE For-Sale Unstable L3MBTL3 85 37 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1F ZINC000217852383 EF For-Sale Unstable NPY1R 43 35 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1F ZINC000217852383 EF For-Sale Unstable NPY2R 47 37 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1F ZINC000217852383 EF For-Sale Unstable ADAMTS5 35 40 CCO[C@H](CN)CN1C[C@@H](C)Cc2ccccc21 ZINC000217852394 BE For-Sale Unstable TPP2 57 32 O=C(C[C@H](c1coc2ccccc2c1=O)c1c(O)c(O)c(O)c2c(=O)cc(-c3ccccc3)oc12)N1CCOCC1 ZINC000217852422 KI In-Stock Unstable PRKDC 34 41 CCC[C@@H](NC(=O)[C@@H]1C[C@@H](O)CN1)C(=O)O ZINC000217852430 BB For-Sale Unstable NOD1 59 35 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)c3cccc(Cl)c3)cc2)C1 ZINC000217852431 FK In-Stock Unstable HRH3 30 44 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)c3cccc(Cl)c3)cc2)C1 ZINC000217852431 FK In-Stock Unstable CCR1 15 40 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)c3cccc(Cl)c3)cc2)C1 ZINC000217852431 FK In-Stock Unstable ADAM17 27 44 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)c3cccc(Cl)c3)cc2)C1 ZINC000217852431 FK In-Stock Unstable PRKD1 27 40 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)c3cccc(Cl)c3)cc2)C1 ZINC000217852431 FK In-Stock Unstable CCKBR 62 44 CCO[C@@H](CN)CCN1C[C@@H](C)Cc2ccccc21 ZINC000217852466 CE For-Sale Unstable TPP2 50 30 CC[C@@H](C)N(CC)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217852475 CG For-Sale Unstable PTGER2 27 43 CC[C@@H](C)N(CC)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217852475 CG For-Sale Unstable PTGER4 0 43 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc(F)cc1 ZINC000217852480 EF For-Sale Unstable ADAMTS5 38 46 CC[C@@H](c1ccccc1O)N1CC[C@@H](N2CCCC2)C1 ZINC000217852500 CG On-Demand Unstable L3MBTL1 0 40 CC[C@@H](c1ccccc1O)N1CC[C@@H](N2CCCC2)C1 ZINC000217852500 CG On-Demand Unstable L3MBTL3 79 37 CC[C@@H](c1ccccc1O)N1CC[C@@H](N2CCCC2)C1 ZINC000217852500 CG On-Demand Unstable TP53BP1 0 40 CCC[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1)C(=O)O ZINC000217852505 BB For-Sale Unstable NOD1 59 35 C[C@H](NC(=O)c1cccc(Cl)c1)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217852536 FK In-Stock Unstable HRH3 30 44 C[C@H](NC(=O)c1cccc(Cl)c1)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217852536 FK In-Stock Unstable CCR1 15 40 C[C@H](NC(=O)c1cccc(Cl)c1)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217852536 FK In-Stock Unstable ADAM17 27 44 C[C@H](NC(=O)c1cccc(Cl)c1)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217852536 FK In-Stock Unstable PRKD1 27 40 C[C@H](NC(=O)c1cccc(Cl)c1)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217852536 FK In-Stock Unstable CCKBR 62 44 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc(F)cc1 ZINC000217852545 EF For-Sale Unstable ADAMTS5 38 46 CC[C@H](C)N(CC)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217852548 CG For-Sale Unstable PTGER2 27 43 CC[C@H](C)N(CC)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217852548 CG For-Sale Unstable PTGER4 0 43 CCO[C@H](CN)CCN1C[C@@H](C)Cc2ccccc21 ZINC000217852562 CE For-Sale Unstable TPP2 50 30 CCC[C@@H](NC(=O)[C@H]1C[C@@H](O)CN1)C(=O)O ZINC000217852588 BB For-Sale Unstable NOD1 59 35 CC[C@H](c1ccccc1O)N1CC[C@@H](N2CCCC2)C1 ZINC000217852590 CG On-Demand Unstable L3MBTL1 0 40 CC[C@H](c1ccccc1O)N1CC[C@@H](N2CCCC2)C1 ZINC000217852590 CG On-Demand Unstable L3MBTL3 79 37 CC[C@H](c1ccccc1O)N1CC[C@@H](N2CCCC2)C1 ZINC000217852590 CG On-Demand Unstable TP53BP1 0 40 CCC[C@H](NC(=O)[C@H]1C[C@@H](O)CN1)C(=O)O ZINC000217852641 BB For-Sale Unstable NOD1 59 35 Cc1ccc2c(c1)[C@@H](NC(=O)c1cccc(Cl)c1)CC(C)(C)O2 ZINC000217852655 EJ In-Stock Unstable ABCC9 43 50 Cc1ccc2c(c1)[C@@H](NC(=O)c1cccc(Cl)c1)CC(C)(C)O2 ZINC000217852655 EJ In-Stock Unstable KCNK9 27 43 CSC[C@@](C)(O)CNCc1cc(C)nc2ccccc12 ZINC000217852656 CF For-Sale Unstable ADAM17 60 34 CSC[C@@](C)(O)CNCc1cc(C)nc2ccccc12 ZINC000217852656 CF For-Sale Unstable METG 73 39 C[C@@H](c1cc(Br)ccc1O)N1CC[C@@H](N2CCCC2)C1 ZINC000217852685 EG For-Sale Unstable L3MBTL1 0 41 C[C@@H](c1cc(Br)ccc1O)N1CC[C@@H](N2CCCC2)C1 ZINC000217852685 EG For-Sale Unstable L3MBTL3 65 39 C[C@@H](c1cc(Br)ccc1O)N1CC[C@@H](N2CCCC2)C1 ZINC000217852685 EG For-Sale Unstable MBTD1 0 52 CC[C@@H](CCN)N1C[C@@H](C)Cc2ccccc21 ZINC000217852709 BF For-Sale Unstable TPP2 53 33 CSC[C@](C)(O)CNCc1cc(C)nc2ccccc12 ZINC000217852714 CF For-Sale Unstable ADAM17 60 34 CSC[C@](C)(O)CNCc1cc(C)nc2ccccc12 ZINC000217852714 CF For-Sale Unstable METG 73 39 CCCCCNC(=O)N/C=C/c1ccccc1Br ZINC000217852730 DH For-Sale Unstable EPHX2 24 42 CCCCCNC(=O)N/C=C/c1ccccc1Br ZINC000217852730 DH For-Sale Unstable ASAH1 60 34 O=C(c1cc(CO)ccn1)N1CCN(c2ccc(Cl)cn2)CC1 ZINC000217852735 ED In-Stock Unstable NPBWR1 49 36 C[C@H](c1cc(Br)ccc1O)N1CC[C@@H](N2CCCC2)C1 ZINC000217852752 EG For-Sale Unstable L3MBTL1 0 41 C[C@H](c1cc(Br)ccc1O)N1CC[C@@H](N2CCCC2)C1 ZINC000217852752 EG For-Sale Unstable L3MBTL3 65 39 C[C@H](c1cc(Br)ccc1O)N1CC[C@@H](N2CCCC2)C1 ZINC000217852752 EG For-Sale Unstable MBTD1 0 52 Cc1ccc2c(c1)[C@H](NC(=O)c1cccc(Cl)c1)CC(C)(C)O2 ZINC000217852765 EJ In-Stock Unstable ABCC9 43 50 Cc1ccc2c(c1)[C@H](NC(=O)c1cccc(Cl)c1)CC(C)(C)O2 ZINC000217852765 EJ In-Stock Unstable KCNK9 27 43 CC[C@H](CCN)N1C[C@@H](C)Cc2ccccc21 ZINC000217852775 BF For-Sale Unstable TPP2 53 33 O=C(N/C=C/c1ccccc1Br)Nc1ccccc1 ZINC000217852817 DI For-Sale Anodyne EPHX1 0 48 O=C(N/C=C/c1ccccc1Br)Nc1ccccc1 ZINC000217852817 DI For-Sale Anodyne P95276_MYCTO 0 48 C[C@@H](CCc1ccc(O)cc1)N1CC[C@@H](N2CCCC2)C1 ZINC000217852850 CF For-Sale Unstable L3MBTL3 89 39 Cc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1cccc(Cl)c1 ZINC000217852854 EJ In-Stock Unstable ABCC9 33 47 Cc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1cccc(Cl)c1 ZINC000217852854 EJ In-Stock Unstable KCNK3 24 44 Cc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1cccc(Cl)c1 ZINC000217852854 EJ In-Stock Unstable KCNK9 32 44 Cc1cccc2[nH]c(-c3ccc(F)c(Br)c3)nc12 ZINC000217852869 DI For-Sale Unstable PARP1 35 40 Cc1cccc2[nH]c(-c3ccc(F)c(Br)c3)nc12 ZINC000217852869 DI For-Sale Unstable TNKS 35 45 Cc1cccc2[nH]c(-c3ccc(F)c(Br)c3)nc12 ZINC000217852869 DI For-Sale Unstable TNKS2 25 45 CCOC(=O)[C@@H]1CCCN(C(=O)N/C=C/c2ccccc2Br)C1 ZINC000217852932 GG For-Sale Unstable SLC6A1 70 35 C[C@H](CCc1ccc(O)cc1)N1CC[C@@H](N2CCCC2)C1 ZINC000217852947 CF For-Sale Unstable L3MBTL3 89 39 Cc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1cccc(Cl)c1 ZINC000217852952 EJ In-Stock Unstable ABCC9 33 47 Cc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1cccc(Cl)c1 ZINC000217852952 EJ In-Stock Unstable KCNK9 32 44 CNC(=O)CN(C)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217852972 CC For-Sale Unstable LTA4H 32 40 CCOC(=O)[C@H]1CCCN(C(=O)N/C=C/c2ccccc2Br)C1 ZINC000217853009 GG For-Sale Unstable SLC6A1 70 35 CCc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217853017 EG For-Sale Unstable ADAMTS5 39 49 C[C@@H](c1ccccc1O)N1CC[C@@H](N2CCCC2)C1 ZINC000217853045 CF For-Sale Unstable L3MBTL1 0 42 C[C@@H](c1ccccc1O)N1CC[C@@H](N2CCCC2)C1 ZINC000217853045 CF For-Sale Unstable L3MBTL3 92 42 C[C@@H](c1ccccc1O)N1CC[C@@H](N2CCCC2)C1 ZINC000217853045 CF For-Sale Unstable MBTD1 0 45 C[C@@H](c1ccccc1O)N1CC[C@@H](N2CCCC2)C1 ZINC000217853045 CF For-Sale Unstable TP53BP1 0 42 COc1ccc2c(c1)[C@@H](NC(=O)c1cccc(Cl)c1)CC(C)(C)O2 ZINC000217853057 EI In-Stock Unstable ABCC9 35 48 COc1ccc2c(c1)[C@@H](NC(=O)c1cccc(Cl)c1)CC(C)(C)O2 ZINC000217853057 EI In-Stock Unstable DRD4 43 34 CCc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217853096 EG For-Sale Unstable ADAMTS5 39 49 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217853099 IE In-Stock Unstable ACE 17 43 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217853099 IE In-Stock Unstable HTR1D 26 41 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217853099 IE In-Stock Unstable HTR1B 17 41 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217853099 IE In-Stock Unstable TACR1 33 40 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217853099 IE In-Stock Unstable MC4R 45 37 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217853099 IE In-Stock Unstable TACR2 23 42 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217853099 IE In-Stock Unstable CCKAR 78 45 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217853099 IE In-Stock Unstable BRS3 26 41 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217853099 IE In-Stock Unstable MC3R 69 37 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217853099 IE In-Stock Unstable MC5R 62 36 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217853099 IE In-Stock Unstable GRPR 43 33 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217853099 IE In-Stock Unstable ECE1 49 40 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217853099 IE In-Stock Unstable HDAC2 15 40 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217853099 IE In-Stock Unstable HDAC3 15 40 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217853099 IE In-Stock Unstable SSTR3 52 38 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217853099 IE In-Stock Unstable MMP11 94 35 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217853099 IE In-Stock Unstable CCKBR 72 45 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217853099 IE In-Stock Unstable GHSR 67 40 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217853099 IE In-Stock Unstable MC1R 94 37 O=C(CC[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217853099 IE In-Stock Unstable KISS1R 60 33 C[C@H](c1ccccc1O)N1CC[C@@H](N2CCCC2)C1 ZINC000217853111 CF For-Sale Unstable L3MBTL1 0 42 C[C@H](c1ccccc1O)N1CC[C@@H](N2CCCC2)C1 ZINC000217853111 CF For-Sale Unstable L3MBTL3 92 42 C[C@H](c1ccccc1O)N1CC[C@@H](N2CCCC2)C1 ZINC000217853111 CF For-Sale Unstable MBTD1 0 45 C[C@H](c1ccccc1O)N1CC[C@@H](N2CCCC2)C1 ZINC000217853111 CF For-Sale Unstable TP53BP1 0 42 COc1ccc2c(c1)[C@H](NC(=O)c1cccc(Cl)c1)CC(C)(C)O2 ZINC000217853137 EI In-Stock Unstable ABCC9 35 48 COc1ccc2c(c1)[C@H](NC(=O)c1cccc(Cl)c1)CC(C)(C)O2 ZINC000217853137 EI In-Stock Unstable DRD4 43 34 Cc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1C ZINC000217853200 EG For-Sale Unstable HTR7 17 41 Cc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1C ZINC000217853200 EG For-Sale Unstable ADAMTS5 34 49 Cc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1C ZINC000217853200 EG For-Sale Unstable SFRP1 54 35 Cc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1C ZINC000217853200 EG For-Sale Unstable WNT3 49 31 Cn1c(C(=O)N2CCc3c([nH]c4ccccc34)C2)cc2ccc(Cl)cc21 ZINC000217853201 FJ In-Stock Unstable FABI 55 38 Cn1c(C(=O)N2CCc3c([nH]c4ccccc34)C2)cc2ccc(Cl)cc21 ZINC000217853201 FJ In-Stock Unstable QRFPR 18 42 C[C@@H](c1cc(F)ccc1O)N1CC[C@@H](N2CCCC2)C1 ZINC000217853221 CF For-Sale Unstable L3MBTL3 67 39 C[C@@H](c1cc(F)ccc1O)N1CC[C@@H](N2CCCC2)C1 ZINC000217853221 CF For-Sale Unstable MBTD1 0 41 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1cccc(Cl)c1 ZINC000217853233 EI In-Stock Unstable ABCC9 32 45 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1cccc(Cl)c1 ZINC000217853233 EI In-Stock Unstable DRD4 44 35 Cc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1C ZINC000217853279 EG For-Sale Unstable HTR7 17 41 Cc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1C ZINC000217853279 EG For-Sale Unstable ADAMTS5 34 49 Cc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1C ZINC000217853279 EG For-Sale Unstable SFRP1 54 35 Cc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1C ZINC000217853279 EG For-Sale Unstable WNT3 49 31 C[C@H](c1cc(F)ccc1O)N1CC[C@@H](N2CCCC2)C1 ZINC000217853308 CF For-Sale Unstable L3MBTL3 67 39 C[C@H](c1cc(F)ccc1O)N1CC[C@@H](N2CCCC2)C1 ZINC000217853308 CF For-Sale Unstable MBTD1 0 41 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1cccc(Cl)c1 ZINC000217853321 EI In-Stock Unstable ABCC9 32 45 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1cccc(Cl)c1 ZINC000217853321 EI In-Stock Unstable DRD4 44 35 N#Cc1ccc2[nH]c(-c3ccc(F)c(Br)c3)nc2c1 ZINC000217853345 DI On-Demand Mild CHEK2 63 41 N#Cc1ccc2[nH]c(-c3ccc(F)c(Br)c3)nc2c1 ZINC000217853345 DI On-Demand Mild NR2E3 52 36 N#Cc1ccc2[nH]c(-c3ccc(F)c(Br)c3)nc2c1 ZINC000217853345 DI On-Demand Mild DGAT1 15 41 Cc1ccc(O)c([C@@H](C)N2CC[C@@H](N3CCCC3)C2)c1 ZINC000217853377 CF For-Sale Unstable L3MBTL1 0 40 Cc1ccc(O)c([C@@H](C)N2CC[C@@H](N3CCCC3)C2)c1 ZINC000217853377 CF For-Sale Unstable L3MBTL3 69 40 Cc1ccc(O)c([C@@H](C)N2CC[C@@H](N3CCCC3)C2)c1 ZINC000217853377 CF For-Sale Unstable MBTD1 0 42 Cc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)c(C)c1 ZINC000217853393 EG For-Sale Unstable EPHX2 17 40 Cc1ccc(/C=C/S(=O)(=O)N2CCC[C@H](Cc3nc(-c4cnccn4)no3)C2)cc1 ZINC000217853426 IG In-Stock Unstable BMP1 16 40 CC[C@@H](NC(=O)c1cccc(Cl)c1)c1ccc(C)c(C)c1 ZINC000217853431 DJ In-Stock Unstable CTSL 21 46 CC[C@@H](NC(=O)c1cccc(Cl)c1)c1ccc(C)c(C)c1 ZINC000217853431 DJ In-Stock Unstable CCKBR 0 44 CC[C@@H](NC(=O)c1cccc(Cl)c1)c1ccc(C)c(C)c1 ZINC000217853431 DJ In-Stock Unstable CTSS 17 46 CC[C@@H](NC(=O)c1cccc(Cl)c1)c1ccc(C)c(C)c1 ZINC000217853431 DJ In-Stock Unstable CTSV 37 46 CC[C@@H](NC(=O)c1cccc(Cl)c1)c1ccc(C)c(C)c1 ZINC000217853431 DJ In-Stock Unstable UTS2 68 45 CC[C@@H](NC(=O)c1cccc(Cl)c1)c1ccc(C)c(C)c1 ZINC000217853431 DJ In-Stock Unstable KCNK3 39 40 CC[C@@H](NC(=O)c1cccc(Cl)c1)c1ccc(C)c(C)c1 ZINC000217853431 DJ In-Stock Unstable KCNK9 27 43 O=C(CSc1nnc(N2CCCCC2)n1Cc1ccco1)c1cccc([N+](=O)[O-])c1 ZINC000217853451 IH On-Demand Unstable HCRTR2 20 41 Cc1ccc(O)c([C@H](C)N2CC[C@@H](N3CCCC3)C2)c1 ZINC000217853458 CF For-Sale Unstable L3MBTL1 0 40 Cc1ccc(O)c([C@H](C)N2CC[C@@H](N3CCCC3)C2)c1 ZINC000217853458 CF For-Sale Unstable L3MBTL3 69 40 Cc1ccc(O)c([C@H](C)N2CC[C@@H](N3CCCC3)C2)c1 ZINC000217853458 CF For-Sale Unstable MBTD1 0 42 Cc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)c(C)c1 ZINC000217853477 EG For-Sale Unstable EPHX2 17 40 COc1ccc2[nH]c3c(c2c1)CCC[C@@H]3NC(=O)c1cc(-c2ccccn2)n[nH]1 ZINC000217853490 GH In-Stock Unstable MAPKAPK2 0 42 Cc1ccc(/C=C/S(=O)(=O)N2CCC[C@@H](Cc3nc(-c4cnccn4)no3)C2)cc1 ZINC000217853494 IG In-Stock Unstable BMP1 16 40 CC[C@H](NC(=O)c1cccc(Cl)c1)c1ccc(C)c(C)c1 ZINC000217853498 DJ In-Stock Unstable CTSL 21 46 CC[C@H](NC(=O)c1cccc(Cl)c1)c1ccc(C)c(C)c1 ZINC000217853498 DJ In-Stock Unstable CCKBR 0 44 CC[C@H](NC(=O)c1cccc(Cl)c1)c1ccc(C)c(C)c1 ZINC000217853498 DJ In-Stock Unstable CTSS 17 46 CC[C@H](NC(=O)c1cccc(Cl)c1)c1ccc(C)c(C)c1 ZINC000217853498 DJ In-Stock Unstable CTSV 37 46 CC[C@H](NC(=O)c1cccc(Cl)c1)c1ccc(C)c(C)c1 ZINC000217853498 DJ In-Stock Unstable UTS2 68 45 CC[C@H](NC(=O)c1cccc(Cl)c1)c1ccc(C)c(C)c1 ZINC000217853498 DJ In-Stock Unstable KCNK3 39 40 CC[C@H](NC(=O)c1cccc(Cl)c1)c1ccc(C)c(C)c1 ZINC000217853498 DJ In-Stock Unstable KCNK9 27 43 Oc1ccc2c(c1)OC[C@@H]2N1CC[C@@H](N2CCCC2)C1 ZINC000217853551 CD For-Sale Unstable L3MBTL3 61 36 O=S(=O)(CCc1ccccc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217853577 EF For-Sale Unstable SLC18A2 41 36 COc1ccc2[nH]c3c(c2c1)CCC[C@H]3NC(=O)c1cc(-c2ccccn2)n[nH]1 ZINC000217853586 GH In-Stock Unstable MAPKAPK2 0 42 CC[C@@H](NC(=O)c1cccc(Cl)c1)c1ccc(C)cc1C ZINC000217853606 DJ In-Stock Unstable CTSL 26 47 CC[C@@H](NC(=O)c1cccc(Cl)c1)c1ccc(C)cc1C ZINC000217853606 DJ In-Stock Unstable CCKBR 22 45 CC[C@@H](NC(=O)c1cccc(Cl)c1)c1ccc(C)cc1C ZINC000217853606 DJ In-Stock Unstable CTSS 20 49 CC[C@@H](NC(=O)c1cccc(Cl)c1)c1ccc(C)cc1C ZINC000217853606 DJ In-Stock Unstable CTSV 46 49 CC[C@@H](NC(=O)c1cccc(Cl)c1)c1ccc(C)cc1C ZINC000217853606 DJ In-Stock Unstable UTS2 53 44 CC[C@@H](NC(=O)c1cccc(Cl)c1)c1ccc(C)cc1C ZINC000217853606 DJ In-Stock Unstable KCNK3 48 39 CC[C@@H](NC(=O)c1cccc(Cl)c1)c1ccc(C)cc1C ZINC000217853606 DJ In-Stock Unstable KCNK9 40 48 CC[C@@H](NC(=O)c1cccc(Cl)c1)c1ccc(C)cc1C ZINC000217853606 DJ In-Stock Unstable PDS 24 40 COC(=O)c1ccc(S(=O)(=O)N2CCC[C@H](Cc3nc(-c4cnccn4)no3)C2)cc1 ZINC000217853613 ID In-Stock Unstable BMP1 21 41 Oc1ccc2c(c1)OC[C@H]2N1CC[C@@H](N2CCCC2)C1 ZINC000217853624 CD For-Sale Unstable L3MBTL3 61 36 O=S(=O)(CCc1ccccc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217853628 EF For-Sale Unstable SLC18A2 41 36 CC[C@H](NC(=O)c1cccc(Cl)c1)c1ccc(C)cc1C ZINC000217853680 DJ In-Stock Unstable CTSL 28 49 CC[C@H](NC(=O)c1cccc(Cl)c1)c1ccc(C)cc1C ZINC000217853680 DJ In-Stock Unstable CCKBR 22 45 CC[C@H](NC(=O)c1cccc(Cl)c1)c1ccc(C)cc1C ZINC000217853680 DJ In-Stock Unstable CTSS 20 49 CC[C@H](NC(=O)c1cccc(Cl)c1)c1ccc(C)cc1C ZINC000217853680 DJ In-Stock Unstable CTSV 46 49 CC[C@H](NC(=O)c1cccc(Cl)c1)c1ccc(C)cc1C ZINC000217853680 DJ In-Stock Unstable UTS2 61 44 CC[C@H](NC(=O)c1cccc(Cl)c1)c1ccc(C)cc1C ZINC000217853680 DJ In-Stock Unstable CTSA 28 40 CC[C@H](NC(=O)c1cccc(Cl)c1)c1ccc(C)cc1C ZINC000217853680 DJ In-Stock Unstable KCNK3 56 48 CC[C@H](NC(=O)c1cccc(Cl)c1)c1ccc(C)cc1C ZINC000217853680 DJ In-Stock Unstable KCNK9 40 48 CC[C@H](NC(=O)c1cccc(Cl)c1)c1ccc(C)cc1C ZINC000217853680 DJ In-Stock Unstable PDS 30 40 C[C@@H](CO)NC(=O)CC[C@@H]1NC(=O)N(CCc2ccccc2)C1=O ZINC000217853688 EC In-Stock Unstable GALR1 45 32 Oc1ccc(-c2nc3cc(Cl)ccc3[nH]2)cc1O ZINC000217853698 CG For-Sale Clean CHEK2 79 52 Oc1ccc(-c2nc3cc(Cl)ccc3[nH]2)cc1O ZINC000217853698 CG For-Sale Clean NR2E3 72 40 Oc1ccc(-c2nc3cc(Cl)ccc3[nH]2)cc1O ZINC000217853698 CG For-Sale Clean SCD1 18 42 Oc1ccc(-c2nc3cc(Cl)ccc3[nH]2)cc1O ZINC000217853698 CG For-Sale Clean SCD 0 42 Oc1ccc(-c2nc3cc(Cl)ccc3[nH]2)cc1O ZINC000217853698 CG For-Sale Clean DGAT1 28 43 COC(=O)c1ccc(S(=O)(=O)N2CCC[C@@H](Cc3nc(-c4cnccn4)no3)C2)cc1 ZINC000217853702 ID In-Stock Unstable BMP1 21 41 CC1(C)CC(NC(=O)N/C=C/c2ccccc2Br)CC(C)(C)N1 ZINC000217853730 GI For-Sale Unstable EZH2 53 42 CC1(C)CC(NC(=O)N/C=C/c2ccccc2Br)CC(C)(C)N1 ZINC000217853730 GI For-Sale Unstable HIV1_ENV 0 40 CC[C@@H](NC(=O)c1cccc(Cl)c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217853772 FH In-Stock Unstable TACR3 41 37 CC[C@@H](NC(=O)c1cccc(Cl)c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217853772 FH In-Stock Unstable CCKBR 0 42 CC[C@@H](NC(=O)c1cccc(Cl)c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217853772 FH In-Stock Unstable CTSV 33 44 CC[C@@H](NC(=O)c1cccc(Cl)c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217853772 FH In-Stock Unstable UTS2 69 46 CC[C@H](NC(=O)c1cccc(Cl)c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217853821 FH In-Stock Unstable TACR3 41 37 CC[C@H](NC(=O)c1cccc(Cl)c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217853821 FH In-Stock Unstable CCKBR 0 42 CC[C@H](NC(=O)c1cccc(Cl)c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217853821 FH In-Stock Unstable CTSV 33 44 CC[C@H](NC(=O)c1cccc(Cl)c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217853821 FH In-Stock Unstable UTS2 69 46 C[C@@H](c1ccc(Cl)cc1)N(C)CCN[C@H](C)C1CC1 ZINC000217853830 CH For-Sale Unstable UTS2 40 33 O=C(c1cc2ccccc2cc1O)N1CCC[C@@H]1c1ccccc1 ZINC000217853838 DJ On-Demand Unstable COLA 73 33 O=C(c1cc2ccccc2cc1O)N1CCC[C@@H]1c1ccccc1 ZINC000217853838 DJ On-Demand Unstable CPT1A 69 33 O=C(c1cc2ccccc2cc1O)N1CCC[C@@H]1c1ccccc1 ZINC000217853838 DJ On-Demand Unstable PREP 41 34 OC[C@@H]1CCC[C@@H]1NCc1ccc(Br)c(F)c1 ZINC000217853861 DF On-Demand Unstable SSTR3 0 41 CC[C@@H](c1ccc(O)cc1)N1CC[C@@H](N2CCCC2)C1 ZINC000217853895 CG For-Sale Unstable L3MBTL3 65 36 O=C(c1cc2ccccc2cc1O)N1CCC[C@H]1c1ccccc1 ZINC000217853917 DJ On-Demand Unstable COLA 73 33 O=C(c1cc2ccccc2cc1O)N1CCC[C@H]1c1ccccc1 ZINC000217853917 DJ On-Demand Unstable CPT1A 70 33 O=C(c1cc2ccccc2cc1O)N1CCC[C@H]1c1ccccc1 ZINC000217853917 DJ On-Demand Unstable PREP 53 37 OC[C@H]1CCC[C@@H]1NCc1ccc(Br)c(F)c1 ZINC000217853924 DF For-Sale Unstable SSTR3 22 41 COc1ccc(-c2noc(CNC(=O)c3cccc(Cl)c3)n2)c(OC)c1 ZINC000217853970 FG In-Stock Unstable DRD4 46 37 COc1ccc(-c2noc(CNC(=O)c3cccc(Cl)c3)n2)c(OC)c1 ZINC000217853970 FG In-Stock Unstable PDK1 24 40 CC(C)[C@H](NC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)C(=O)N1CCc2ccccc2C1 ZINC000217853976 IF In-Stock Unstable CHRNA4 26 43 OC[C@@H]1CCC[C@H]1NCc1ccc(Br)c(F)c1 ZINC000217853996 DF For-Sale Unstable SSTR3 22 41 CC[C@H](c1ccc(O)cc1)N1CC[C@@H](N2CCCC2)C1 ZINC000217854004 CG For-Sale Unstable L3MBTL3 65 36 O=C(c1cc(Br)ccc1O)N1CCC[C@@H]1c1ccccc1 ZINC000217854021 EI On-Demand Unstable UTS2R 43 29 OC[C@H]1CCC[C@H]1NCc1ccc(Br)c(F)c1 ZINC000217854053 DF For-Sale Unstable SSTR3 22 41 CN1CC(=O)N(Cc2ccccc2/C=C\C(=O)O)C1=O ZINC000217854058 CD For-Sale Unstable PTGER2 44 46 CN1CC(=O)N(Cc2ccccc2/C=C\C(=O)O)C1=O ZINC000217854058 CD For-Sale Unstable PTGER4 0 46 CN1CC(=O)N(Cc2ccccc2/C=C\C(=O)O)C1=O ZINC000217854058 CD For-Sale Unstable PTGER3 22 46 C[C@@H](c1cc(Cl)ccc1O)N1CC[C@@H](N2CCCC2)C1 ZINC000217854066 CG For-Sale Unstable L3MBTL3 66 39 C[C@@H](c1cc(Cl)ccc1O)N1CC[C@@H](N2CCCC2)C1 ZINC000217854066 CG For-Sale Unstable MBTD1 0 41 O=C(NCc1nc(-c2cccc(Br)c2)no1)c1cccc(Cl)c1 ZINC000217854079 GI In-Stock Unstable GRM5 26 42 Oc1cc([C@@H]2CCCNC2)ccc1Br ZINC000217854092 CF For-Sale Unstable DRD2 17 55 O=C(c1cc(Br)ccc1O)N1CCC[C@H]1c1ccccc1 ZINC000217854119 EI On-Demand Unstable UTS2R 43 29 COc1cccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217854135 EF For-Sale Unstable NPY2R 76 43 COc1cccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217854135 EF For-Sale Unstable ADAMTS5 31 43 Oc1cc([C@H]2CCCNC2)ccc1Br ZINC000217854151 CF For-Sale Unstable DRD2 17 55 C[C@H](c1cc(Cl)ccc1O)N1CC[C@@H](N2CCCC2)C1 ZINC000217854157 CG For-Sale Unstable L3MBTL3 66 39 C[C@H](c1cc(Cl)ccc1O)N1CC[C@@H](N2CCCC2)C1 ZINC000217854157 CG For-Sale Unstable MBTD1 0 41 COc1cccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217854192 EF For-Sale Unstable NPY2R 76 43 COc1cccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217854192 EF For-Sale Unstable ADAMTS5 31 43 CC(C)(C)OC[C@H](NS(=O)(=O)Cc1ccc(C#N)cc1)C(=O)O ZINC000217854259 ED On-Demand Unstable CTRB_BOVIN 50 38 CC(C)(C)OC[C@H](NS(=O)(=O)Cc1ccc(C#N)cc1)C(=O)O ZINC000217854259 ED On-Demand Unstable TMPRSS11D 47 33 COc1cc(C(=O)N2CCC[C@@H]2c2ccccc2)ccc1OCC(C)C ZINC000217854260 FJ On-Demand Unstable FKBP1A 42 36 COc1cc(C(=O)N2CCC[C@@H]2c2ccccc2)ccc1OCC(C)C ZINC000217854260 FJ On-Demand Unstable ADAM17 15 40 COc1cc(C(=O)N2CCC[C@@H]2c2ccccc2)ccc1OCC(C)C ZINC000217854260 FJ On-Demand Unstable CPT1A 62 36 COc1cc(C(=O)N2CCC[C@@H]2c2ccccc2)ccc1OCC(C)C ZINC000217854260 FJ On-Demand Unstable MTNR1B 22 41 COc1cc(C(=O)N2CCC[C@@H]2c2ccccc2)ccc1OCC(C)C ZINC000217854260 FJ On-Demand Unstable BRCA1 42 30 COc1cc(C(=O)N2CCC[C@@H]2c2ccccc2)ccc1OCC(C)C ZINC000217854260 FJ On-Demand Unstable ACKR3 62 39 Fc1ccc(-c2nc3cc(Cl)ccc3[nH]2)cc1Br ZINC000217854275 EJ For-Sale Anodyne GYRB 0 45 Fc1ccc(-c2nc3cc(Cl)ccc3[nH]2)cc1Br ZINC000217854275 EJ For-Sale Anodyne CHEK2 58 48 Fc1ccc(-c2nc3cc(Cl)ccc3[nH]2)cc1Br ZINC000217854275 EJ For-Sale Anodyne NR2E3 68 41 Fc1ccc(-c2nc3cc(Cl)ccc3[nH]2)cc1Br ZINC000217854275 EJ For-Sale Anodyne SCD1 17 43 Fc1ccc(-c2nc3cc(Cl)ccc3[nH]2)cc1Br ZINC000217854275 EJ For-Sale Anodyne DGAT1 21 40 Oc1cccc2c1CCC[C@@H]2N1CC[C@@H](N2CCCC2)C1 ZINC000217854284 CF For-Sale Unstable SLC6A1 0 42 Oc1cccc2c1CCC[C@@H]2N1CC[C@@H](N2CCCC2)C1 ZINC000217854284 CF For-Sale Unstable L3MBTL3 75 39 O=S(=O)(NCCCCCO)c1ccccc1-c1ccccc1 ZINC000217854310 DF On-Demand Unstable CASP1 19 46 COc1ccccc1S(=O)(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217854312 EF For-Sale Unstable NPY1R 44 35 COc1ccccc1S(=O)(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217854312 EF For-Sale Unstable NPY2R 60 40 COc1ccccc1S(=O)(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217854312 EF For-Sale Unstable ADAMTS5 33 43 COc1cc(C(=O)N2CCC[C@H]2c2ccccc2)ccc1OCC(C)C ZINC000217854350 FJ On-Demand Unstable FKBP1A 42 36 COc1cc(C(=O)N2CCC[C@H]2c2ccccc2)ccc1OCC(C)C ZINC000217854350 FJ On-Demand Unstable ADAM17 15 40 COc1cc(C(=O)N2CCC[C@H]2c2ccccc2)ccc1OCC(C)C ZINC000217854350 FJ On-Demand Unstable CPT1A 62 36 COc1cc(C(=O)N2CCC[C@H]2c2ccccc2)ccc1OCC(C)C ZINC000217854350 FJ On-Demand Unstable MTNR1B 22 41 COc1cc(C(=O)N2CCC[C@H]2c2ccccc2)ccc1OCC(C)C ZINC000217854350 FJ On-Demand Unstable BRCA1 42 30 COc1cc(C(=O)N2CCC[C@H]2c2ccccc2)ccc1OCC(C)C ZINC000217854350 FJ On-Demand Unstable ACKR3 62 39 Cc1cccc(=O)n1Cc1cccc(/C=C\C(=O)O)c1 ZINC000217854351 CE For-Sale Unstable HDAC8 34 41 Cc1cccc(=O)n1Cc1cccc(/C=C\C(=O)O)c1 ZINC000217854351 CE For-Sale Unstable HDAC6 28 41 Oc1cccc2c1CCC[C@H]2N1CC[C@@H](N2CCCC2)C1 ZINC000217854366 CF For-Sale Unstable SLC6A1 0 42 Oc1cccc2c1CCC[C@H]2N1CC[C@@H](N2CCCC2)C1 ZINC000217854366 CF For-Sale Unstable L3MBTL3 75 39 CCN(Cc1ccccc1)C(=O)N/C=C/c1ccccc1Br ZINC000217854382 FJ For-Sale Unstable PTGES 0 41 COc1ccccc1S(=O)(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217854392 EF For-Sale Unstable NPY1R 44 35 COc1ccccc1S(=O)(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217854392 EF For-Sale Unstable NPY2R 60 40 COc1ccccc1S(=O)(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217854392 EF For-Sale Unstable ADAMTS5 33 43 CN(Cc1nc(-c2ccccc2Cl)no1)C(=O)c1cccc(Cl)c1 ZINC000217854393 FI In-Stock Unstable GPBAR1 31 42 CC[C@@H](CCO)NC[C@@H](O)COC(C)C ZINC000217854431 BC On-Demand Unstable ADRB2 0 58 O=C1C[C@@H](c2cccc(OC(F)F)c2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217854432 JJ In-Stock Unstable AKR1B1 0 41 C[C@@H](c1cccc(O)c1)N1CC[C@@H](N2CCCC2)C1 ZINC000217854472 CF For-Sale Unstable L3MBTL3 78 38 CN(Cc1nc(-c2cccc(Br)c2)no1)C(=O)c1cccc(Cl)c1 ZINC000217854493 HI In-Stock Unstable GRM5 17 43 CN(Cc1nc(-c2cccc(Br)c2)no1)C(=O)c1cccc(Cl)c1 ZINC000217854493 HI In-Stock Unstable GPBAR1 15 40 CC[C@H](CCO)NC[C@@H](O)COC(C)C ZINC000217854497 BC On-Demand Unstable ADRB2 0 58 O=C1C[C@H](c2cccc(OC(F)F)c2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217854525 JJ In-Stock Unstable AKR1B1 0 41 C[C@H](c1cccc(O)c1)N1CC[C@@H](N2CCCC2)C1 ZINC000217854553 CF For-Sale Unstable L3MBTL3 78 38 CC[C@@H](CCO)NC[C@H](O)COC(C)C ZINC000217854586 BC On-Demand Unstable ADRB2 0 58 O=C(NCCCN1CCCc2ccccc21)c1cccc(Cl)c1 ZINC000217854603 EH In-Stock Unstable HTR1A 27 44 O=C(NCCCN1CCCc2ccccc21)c1cccc(Cl)c1 ZINC000217854603 EH In-Stock Unstable DRD2 39 44 O=C(NCCCN1CCCc2ccccc21)c1cccc(Cl)c1 ZINC000217854603 EH In-Stock Unstable DRD1 25 44 O=C(NCCCN1CCCc2ccccc21)c1cccc(Cl)c1 ZINC000217854603 EH In-Stock Unstable DRD4 53 44 O=C(NCCCN1CCCc2ccccc21)c1cccc(Cl)c1 ZINC000217854603 EH In-Stock Unstable HTR2A 38 40 O=C(NCCCN1CCCc2ccccc21)c1cccc(Cl)c1 ZINC000217854603 EH In-Stock Unstable HTR2C 36 46 O=C(NCCCN1CCCc2ccccc21)c1cccc(Cl)c1 ZINC000217854603 EH In-Stock Unstable AVPR2 35 55 O=C(NCCCN1CCCc2ccccc21)c1cccc(Cl)c1 ZINC000217854603 EH In-Stock Unstable DRD3 65 45 O=C(NCCCN1CCCc2ccccc21)c1cccc(Cl)c1 ZINC000217854603 EH In-Stock Unstable HRP1_PLAFA 26 40 O=C(NCCCN1CCCc2ccccc21)c1cccc(Cl)c1 ZINC000217854603 EH In-Stock Unstable CCKBR 22 40 O=C(NCCCN1CCCc2ccccc21)c1cccc(Cl)c1 ZINC000217854603 EH In-Stock Unstable PLD2 43 39 O=C(NCCCN1CCCc2ccccc21)c1cccc(Cl)c1 ZINC000217854603 EH In-Stock Unstable CACNA1I 44 43 O=C(NCCCN1CCCc2ccccc21)c1cccc(Cl)c1 ZINC000217854603 EH In-Stock Unstable TYRO3 23 42 CC(=O)c1cn(CCNC(=O)CC[C@@H]2NC(=O)c3ccccc3NC2=O)c2ccccc12 ZINC000217854606 IE In-Stock Unstable CNR1 15 40 CC(=O)c1cn(CCNC(=O)CC[C@@H]2NC(=O)c3ccccc3NC2=O)c2ccccc12 ZINC000217854606 IE In-Stock Unstable CNR2 22 40 O=C(O)/C=C\c1cccc(COc2ccc(Cl)cc2)c1 ZINC000217854648 CI For-Sale Unstable ALOX5 15 48 O=C(O)/C=C\c1cccc(COc2ccc(Cl)cc2)c1 ZINC000217854648 CI For-Sale Unstable MAOA 16 44 O=C(O)/C=C\c1cccc(COc2ccc(Cl)cc2)c1 ZINC000217854648 CI For-Sale Unstable MAOB 80 46 O=C(O)/C=C\c1cccc(COc2ccc(Cl)cc2)c1 ZINC000217854648 CI For-Sale Unstable PTGER2 54 48 O=C(O)/C=C\c1cccc(COc2ccc(Cl)cc2)c1 ZINC000217854648 CI For-Sale Unstable CYSLTR1 20 41 O=C(O)/C=C\c1cccc(COc2ccc(Cl)cc2)c1 ZINC000217854648 CI For-Sale Unstable LTA4H 16 40 O=C(O)/C=C\c1cccc(COc2ccc(Cl)cc2)c1 ZINC000217854648 CI For-Sale Unstable PTGER1 47 38 O=C(O)/C=C\c1cccc(COc2ccc(Cl)cc2)c1 ZINC000217854648 CI For-Sale Unstable PTGER4 29 48 O=C(O)/C=C\c1cccc(COc2ccc(Cl)cc2)c1 ZINC000217854648 CI For-Sale Unstable PTPN2 0 40 O=C(O)/C=C\c1cccc(COc2ccc(Cl)cc2)c1 ZINC000217854648 CI For-Sale Unstable PTGER3 32 48 O=C(O)/C=C\c1cccc(COc2ccc(Cl)cc2)c1 ZINC000217854648 CI For-Sale Unstable LTB4R 22 43 O=C(O)/C=C\c1cccc(COc2ccc(Cl)cc2)c1 ZINC000217854648 CI For-Sale Unstable KCNA3 0 49 O=C(O)/C=C\c1cccc(COc2ccc(Cl)cc2)c1 ZINC000217854648 CI For-Sale Unstable CDC25B 22 43 O=C(O)/C=C\c1cccc(COc2ccc(Cl)cc2)c1 ZINC000217854648 CI For-Sale Unstable NR1H4 50 41 O=C(O)/C=C\c1cccc(COc2ccc(Cl)cc2)c1 ZINC000217854648 CI For-Sale Unstable GYS1 49 36 O=C(O)/C=C\c1cccc(COc2ccc(Cl)cc2)c1 ZINC000217854648 CI For-Sale Unstable ACR 22 40 O=C(O)/C=C\c1cccc(COc2ccc(Cl)cc2)c1 ZINC000217854648 CI For-Sale Unstable PTGDR 0 46 O=C(O)/C=C\c1cccc(COc2ccc(Cl)cc2)c1 ZINC000217854648 CI For-Sale Unstable ADAMTS4 24 41 O=C(O)/C=C\c1cccc(COc2ccc(Cl)cc2)c1 ZINC000217854648 CI For-Sale Unstable HCAR2 0 40 O=C(O)/C=C\c1cccc(COc2ccc(Cl)cc2)c1 ZINC000217854648 CI For-Sale Unstable 17HSDCL 0 41 O=C(O)/C=C\c1cccc(COc2ccc(Cl)cc2)c1 ZINC000217854648 CI For-Sale Unstable FFAR1 68 44 O=C(O)/C=C\c1cccc(COc2ccc(Cl)cc2)c1 ZINC000217854648 CI For-Sale Unstable AKR1C3 40 54 O=C(O)/C=C\c1cccc(COc2ccc(Cl)cc2)c1 ZINC000217854648 CI For-Sale Unstable FFAR4 32 43 O=C(O)/C=C\c1cccc(COc2ccc(Cl)cc2)c1 ZINC000217854648 CI For-Sale Unstable ADCYAP1R1 35 41 O=C(O)/C=C\c1cccc(COc2ccc(Cl)cc2)c1 ZINC000217854648 CI For-Sale Unstable TUBA4A 0 40 O=C(O)/C=C\c1cccc(COc2ccc(Cl)cc2)c1 ZINC000217854648 CI For-Sale Unstable GPR183 0 45 CC[C@H](CCO)NC[C@H](O)COC(C)C ZINC000217854665 BC On-Demand Unstable ADRB2 0 58 CC[C@@H]1CCCCN1C(=O)N/C=C/c1ccccc1Br ZINC000217854671 EI For-Sale Unstable ABHD11 0 40 Cc1c(C(=O)N2CCC[C@@H]2c2ccccc2)[nH]c2c1C(=O)CC(C)(C)C2 ZINC000217854680 FI On-Demand Unstable HSP90AA1 47 35 CCOc1ccc(CNC(=O)c2ccc(Cl)cc2Cl)cc1OCC ZINC000217854707 FJ In-Stock Unstable PYGL 17 40 CCOc1ccc(CNC(=O)c2ccc(Cl)cc2Cl)cc1OCC ZINC000217854707 FJ In-Stock Unstable PPARD 24 42 CCOc1ccc(CNC(=O)c2ccc(Cl)cc2Cl)cc1OCC ZINC000217854707 FJ In-Stock Unstable SLC6A9 45 36 CCOc1ccc(CNC(=O)c2ccc(Cl)cc2Cl)cc1OCC ZINC000217854707 FJ In-Stock Unstable UL54 57 34 CCOc1ccc(CNC(=O)c2ccc(Cl)cc2Cl)cc1OCC ZINC000217854707 FJ In-Stock Unstable U38 0 45 CCOc1ccc(CNC(=O)c2ccc(Cl)cc2Cl)cc1OCC ZINC000217854707 FJ In-Stock Unstable PTGDR2 19 44 CCOc1ccc(CNC(=O)c2ccc(Cl)cc2Cl)cc1OCC ZINC000217854707 FJ In-Stock Unstable ENR 0 45 COc1cc(OC)c([C@@H]2CC(=O)Oc3ccc4c(c32)OC(C)(C)CC4=O)cc1OC ZINC000217854710 HH In-Stock Unstable MT-ND4 52 32 O=C(O)/C=C\c1cc(F)ccc1COc1ccc(Cl)cc1 ZINC000217854728 DI For-Sale Unstable PTGER2 40 44 O=C(O)/C=C\c1cc(F)ccc1COc1ccc(Cl)cc1 ZINC000217854728 DI For-Sale Unstable PTGER3 25 44 O=C(O)/C=C\c1cc(F)ccc1COc1ccc(Cl)cc1 ZINC000217854728 DI For-Sale Unstable CDC25B 23 41 O=C(O)/C=C\c1cc(F)ccc1COc1ccc(Cl)cc1 ZINC000217854728 DI For-Sale Unstable PTGDR 0 42 O=C(O)/C=C\c1cc(F)ccc1COc1ccc(Cl)cc1 ZINC000217854728 DI For-Sale Unstable FFAR4 29 40 Cc1c(C(=O)N2CCC[C@H]2c2ccccc2)[nH]c2c1C(=O)CC(C)(C)C2 ZINC000217854761 FI On-Demand Unstable HSP90AA1 47 35 CC[C@H]1CCCCN1C(=O)N/C=C/c1ccccc1Br ZINC000217854780 EI For-Sale Unstable ABHD11 0 40 COc1ccccc1CCCNC(=O)c1ccc(Cl)cc1Cl ZINC000217854788 EI In-Stock Unstable DRD2 27 43 COc1ccccc1CCCNC(=O)c1ccc(Cl)cc1Cl ZINC000217854788 EI In-Stock Unstable DRD1 0 41 COc1ccccc1CCCNC(=O)c1ccc(Cl)cc1Cl ZINC000217854788 EI In-Stock Unstable DRD3 36 42 COc1ccccc1CCCNC(=O)c1ccc(Cl)cc1Cl ZINC000217854788 EI In-Stock Unstable CPT1A 43 30 COc1ccccc1CCCNC(=O)c1ccc(Cl)cc1Cl ZINC000217854788 EI In-Stock Unstable PYGL 23 46 COc1ccccc1CCCNC(=O)c1ccc(Cl)cc1Cl ZINC000217854788 EI In-Stock Unstable MTNR1B 40 44 COc1ccccc1CCCNC(=O)c1ccc(Cl)cc1Cl ZINC000217854788 EI In-Stock Unstable SLC6A9 44 36 COc1ccccc1CCCNC(=O)c1ccc(Cl)cc1Cl ZINC000217854788 EI In-Stock Unstable SLC6A5 25 40 COc1ccccc1CCCNC(=O)c1ccc(Cl)cc1Cl ZINC000217854788 EI In-Stock Unstable ALPL 45 41 COc1ccccc1CCCNC(=O)c1ccc(Cl)cc1Cl ZINC000217854788 EI In-Stock Unstable U38 0 44 COc1cc(OC)c([C@H]2CC(=O)Oc3ccc4c(c32)OC(C)(C)CC4=O)cc1OC ZINC000217854796 HH In-Stock Unstable MT-ND4 52 32 O=C(O)/C=C\c1cc(COc2ccc(Cl)cc2)ccc1F ZINC000217854815 DI For-Sale Unstable PTGER2 49 47 O=C(O)/C=C\c1cc(COc2ccc(Cl)cc2)ccc1F ZINC000217854815 DI For-Sale Unstable PTGER4 24 44 O=C(O)/C=C\c1cc(COc2ccc(Cl)cc2)ccc1F ZINC000217854815 DI For-Sale Unstable PTPN2 0 41 O=C(O)/C=C\c1cc(COc2ccc(Cl)cc2)ccc1F ZINC000217854815 DI For-Sale Unstable PTGER3 34 48 O=C(O)/C=C\c1cc(COc2ccc(Cl)cc2)ccc1F ZINC000217854815 DI For-Sale Unstable CDC25B 23 41 O=C(O)/C=C\c1cc(COc2ccc(Cl)cc2)ccc1F ZINC000217854815 DI For-Sale Unstable GYS1 49 34 O=C(O)/C=C\c1cc(COc2ccc(Cl)cc2)ccc1F ZINC000217854815 DI For-Sale Unstable PTGDR 0 48 O=C(O)/C=C\c1cc(COc2ccc(Cl)cc2)ccc1F ZINC000217854815 DI For-Sale Unstable FFAR1 52 40 O=C(O)/C=C\c1cc(COc2ccc(Cl)cc2)ccc1F ZINC000217854815 DI For-Sale Unstable AKR1C3 27 43 O=C(N/C=C/c1ccccc1Br)N(Cc1ccccc1)Cc1ccccc1 ZINC000217854877 HK For-Sale Unstable PTGES 0 44 Cc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1C ZINC000217854888 CH For-Sale Unstable TSHR 47 31 Cc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1C ZINC000217854888 CH For-Sale Unstable PTGER2 31 54 Cc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1C ZINC000217854888 CH For-Sale Unstable PTGER4 41 49 Cc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1C ZINC000217854888 CH For-Sale Unstable PTGER3 32 59 Cc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1C ZINC000217854888 CH For-Sale Unstable PPARD 22 42 Cc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1C ZINC000217854888 CH For-Sale Unstable CDC25B 22 41 Cc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1C ZINC000217854888 CH For-Sale Unstable PTGDR 0 59 Cc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1C ZINC000217854888 CH For-Sale Unstable FFAR4 41 36 CN1CCO[C@@H]([C@@H](O)Cc2cc(F)ccc2F)C1 ZINC000217854912 CD For-Sale Unstable DPP4 31 42 CCOc1ccc(CCCNC(=O)c2ccc(Cl)cc2Cl)cc1 ZINC000217854939 FJ In-Stock Unstable ADRB3 17 40 CCOc1ccc(CCCNC(=O)c2ccc(Cl)cc2Cl)cc1 ZINC000217854939 FJ In-Stock Unstable SCN2A 26 42 CCOc1ccc(CCCNC(=O)c2ccc(Cl)cc2Cl)cc1 ZINC000217854939 FJ In-Stock Unstable SLC6A9 45 36 CCOc1ccc(CCCNC(=O)c2ccc(Cl)cc2Cl)cc1 ZINC000217854939 FJ In-Stock Unstable ALPL 42 37 CCOc1ccc(CCCNC(=O)c2ccc(Cl)cc2Cl)cc1 ZINC000217854939 FJ In-Stock Unstable CRTM 46 40 CCOc1ccc(CCCNC(=O)c2ccc(Cl)cc2Cl)cc1 ZINC000217854939 FJ In-Stock Unstable PDS 42 36 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCC[C@@H]2c2ccccc2)[C@@H](C)O)cc1 ZINC000217854966 HE On-Demand Unstable F2 30 40 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCC[C@@H]2c2ccccc2)[C@@H](C)O)cc1 ZINC000217854966 HE On-Demand Unstable ELANE 43 42 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCC[C@@H]2c2ccccc2)[C@@H](C)O)cc1 ZINC000217854966 HE On-Demand Unstable MMP13 40 45 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCC[C@@H]2c2ccccc2)[C@@H](C)O)cc1 ZINC000217854966 HE On-Demand Unstable ADAM17 53 43 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCC[C@@H]2c2ccccc2)[C@@H](C)O)cc1 ZINC000217854966 HE On-Demand Unstable MMP2 33 45 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCC[C@@H]2c2ccccc2)[C@@H](C)O)cc1 ZINC000217854966 HE On-Demand Unstable MMP3 17 45 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCC[C@@H]2c2ccccc2)[C@@H](C)O)cc1 ZINC000217854966 HE On-Demand Unstable CAPN1 16 40 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCC[C@@H]2c2ccccc2)[C@@H](C)O)cc1 ZINC000217854966 HE On-Demand Unstable ADAMTS4 60 38 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCC[C@@H]2c2ccccc2)[C@@H](C)O)cc1 ZINC000217854966 HE On-Demand Unstable XIAP 41 39 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCC[C@@H]2c2ccccc2)[C@@H](C)O)cc1 ZINC000217854966 HE On-Demand Unstable WNT3 42 36 Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1C ZINC000217854995 CH For-Sale Unstable ESR1 15 43 Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1C ZINC000217854995 CH For-Sale Unstable ALOX5 15 51 Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1C ZINC000217854995 CH For-Sale Unstable MAOB 47 40 Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1C ZINC000217854995 CH For-Sale Unstable PTGER2 23 46 Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1C ZINC000217854995 CH For-Sale Unstable PTGER4 28 45 Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1C ZINC000217854995 CH For-Sale Unstable PTGER3 23 49 Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1C ZINC000217854995 CH For-Sale Unstable PPARD 26 40 Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1C ZINC000217854995 CH For-Sale Unstable PTGDR 0 49 Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1C ZINC000217854995 CH For-Sale Unstable FFAR1 61 40 Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1C ZINC000217854995 CH For-Sale Unstable AKR1C3 34 46 CN1CCO[C@H]([C@@H](O)Cc2cc(F)ccc2F)C1 ZINC000217855038 CD For-Sale Unstable DPP4 31 42 CCCOc1ccccc1CCCNC(=O)c1ccc(Cl)cc1Cl ZINC000217855049 FK In-Stock Unstable SLC6A9 45 39 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1cccc(Cl)c1 ZINC000217855056 FG For-Sale Unstable HTR7 20 47 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1cccc(Cl)c1 ZINC000217855056 FG For-Sale Unstable NPY2R 41 39 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1cccc(Cl)c1 ZINC000217855056 FG For-Sale Unstable HTR6 27 47 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1cccc(Cl)c1 ZINC000217855056 FG For-Sale Unstable FBP1 22 44 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1cccc(Cl)c1 ZINC000217855056 FG For-Sale Unstable ADAMTS5 35 48 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1cccc(Cl)c1 ZINC000217855056 FG For-Sale Unstable AKR1C3 15 40 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1cccc(Cl)c1 ZINC000217855056 FG For-Sale Unstable SFRP1 44 36 COc1ccc(NC(=O)N/C=C/c2ccccc2Br)c(OC)c1 ZINC000217855076 GI For-Sale Unstable CYP1B1 30 46 COc1ccc(NC(=O)N/C=C/c2ccccc2Br)c(OC)c1 ZINC000217855076 GI For-Sale Unstable MTNR1A 20 45 COc1ccc(NC(=O)N/C=C/c2ccccc2Br)c(OC)c1 ZINC000217855076 GI For-Sale Unstable MTNR1B 19 45 COc1ccc(NC(=O)N/C=C/c2ccccc2Br)c(OC)c1 ZINC000217855076 GI For-Sale Unstable AKR1C2 41 35 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1C ZINC000217855080 CH For-Sale Unstable ALOX5 20 46 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1C ZINC000217855080 CH For-Sale Unstable TSHR 41 32 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1C ZINC000217855080 CH For-Sale Unstable MAOB 75 48 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1C ZINC000217855080 CH For-Sale Unstable PTGER2 26 55 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1C ZINC000217855080 CH For-Sale Unstable EDNRA 0 43 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1C ZINC000217855080 CH For-Sale Unstable PTGER4 29 49 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1C ZINC000217855080 CH For-Sale Unstable PTGER3 30 49 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1C ZINC000217855080 CH For-Sale Unstable LTB4R 23 44 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1C ZINC000217855080 CH For-Sale Unstable PPARD 27 41 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1C ZINC000217855080 CH For-Sale Unstable NR1H4 49 38 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1C ZINC000217855080 CH For-Sale Unstable GYS1 40 35 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1C ZINC000217855080 CH For-Sale Unstable PTGDR 0 47 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1C ZINC000217855080 CH For-Sale Unstable FFAR1 93 46 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1C ZINC000217855080 CH For-Sale Unstable AKR1C3 38 47 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCC[C@H]2c2ccccc2)[C@@H](C)O)cc1 ZINC000217855103 HE On-Demand Unstable F2 30 40 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCC[C@H]2c2ccccc2)[C@@H](C)O)cc1 ZINC000217855103 HE On-Demand Unstable ELANE 43 42 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCC[C@H]2c2ccccc2)[C@@H](C)O)cc1 ZINC000217855103 HE On-Demand Unstable MMP13 40 45 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCC[C@H]2c2ccccc2)[C@@H](C)O)cc1 ZINC000217855103 HE On-Demand Unstable ADAM17 53 43 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCC[C@H]2c2ccccc2)[C@@H](C)O)cc1 ZINC000217855103 HE On-Demand Unstable MMP2 33 45 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCC[C@H]2c2ccccc2)[C@@H](C)O)cc1 ZINC000217855103 HE On-Demand Unstable MMP3 17 45 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCC[C@H]2c2ccccc2)[C@@H](C)O)cc1 ZINC000217855103 HE On-Demand Unstable CAPN1 16 40 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCC[C@H]2c2ccccc2)[C@@H](C)O)cc1 ZINC000217855103 HE On-Demand Unstable ADAMTS4 60 38 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCC[C@H]2c2ccccc2)[C@@H](C)O)cc1 ZINC000217855103 HE On-Demand Unstable XIAP 41 39 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCC[C@H]2c2ccccc2)[C@@H](C)O)cc1 ZINC000217855103 HE On-Demand Unstable WNT3 42 36 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1cccc(Cl)c1 ZINC000217855120 FG For-Sale Unstable HTR7 20 47 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1cccc(Cl)c1 ZINC000217855120 FG For-Sale Unstable NPY2R 41 39 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1cccc(Cl)c1 ZINC000217855120 FG For-Sale Unstable HTR6 27 47 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1cccc(Cl)c1 ZINC000217855120 FG For-Sale Unstable FBP1 22 44 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1cccc(Cl)c1 ZINC000217855120 FG For-Sale Unstable ADAMTS5 35 48 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1cccc(Cl)c1 ZINC000217855120 FG For-Sale Unstable AKR1C3 15 40 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1cccc(Cl)c1 ZINC000217855120 FG For-Sale Unstable SFRP1 44 36 Cc1ccccc1OC[C@H](C)NC(=O)c1ccc(Cl)cc1Cl ZINC000217855129 EI In-Stock Unstable SDH1 0 45 Cc1ccccc1OC[C@H](C)NC(=O)c1ccc(Cl)cc1Cl ZINC000217855129 EI In-Stock Unstable SLC6A9 34 41 Cc1ccccc1OC[C@H](C)NC(=O)c1ccc(Cl)cc1Cl ZINC000217855129 EI In-Stock Unstable ALPL 32 40 CC[C@@H](CCO)NCCCCCC(=O)O ZINC000217855145 BD For-Sale Unstable FABP2 0 42 CC[C@@H](CCO)NCCCCCC(=O)O ZINC000217855145 BD For-Sale Unstable PLA2G2C 0 40 CC[C@@H](CCO)NCCCCCC(=O)O ZINC000217855145 BD For-Sale Unstable Q6UB75_PIG 0 42 CC[C@@H](CCO)NCCCCCC(=O)O ZINC000217855145 BD For-Sale Unstable SLC22A20 0 42 CC[C@@H](CCO)NCCCCCC(=O)O ZINC000217855145 BD For-Sale Unstable CQSS 40 30 Cc1cccc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217855156 CH For-Sale Unstable PTGER2 31 55 Cc1cccc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217855156 CH For-Sale Unstable PTGER4 51 56 Cc1cccc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217855156 CH For-Sale Unstable PTGER3 41 57 Cc1cccc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217855156 CH For-Sale Unstable PTGDR 0 57 Cc1cccc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217855156 CH For-Sale Unstable FFAR1 29 44 Cc1cccc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217855156 CH For-Sale Unstable FFAR4 40 37 Cc1cccc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217855156 CH For-Sale Unstable PDS 25 40 Cn1ccnc1CN1CCN(C(=O)c2ccc(-n3cnnn3)cc2O)CC1 ZINC000217855159 FC In-Stock Unstable KCNJ1 60 39 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccccc1Cl ZINC000217855205 FG For-Sale Unstable NPY1R 43 35 CCc1ccc(-c2nc(CC(=O)N3CCC[C@@H]3c3ccccc3)cs2)cc1 ZINC000217855211 GK On-Demand Unstable PRCP 30 41 CCc1ccc(-c2nc(CC(=O)N3CCC[C@@H]3c3ccccc3)cs2)cc1 ZINC000217855211 GK On-Demand Unstable ADAM17 41 45 CCc1ccc(-c2nc(CC(=O)N3CCC[C@@H]3c3ccccc3)cs2)cc1 ZINC000217855211 GK On-Demand Unstable COLA 114 49 CCc1ccc(-c2nc(CC(=O)N3CCC[C@@H]3c3ccccc3)cs2)cc1 ZINC000217855211 GK On-Demand Unstable CPT1A 108 49 CCc1ccc(-c2nc(CC(=O)N3CCC[C@@H]3c3ccccc3)cs2)cc1 ZINC000217855211 GK On-Demand Unstable PREP 53 32 CC[C@H](CCO)NCCCCCC(=O)O ZINC000217855223 BD For-Sale Unstable FABP2 0 42 CC[C@H](CCO)NCCCCCC(=O)O ZINC000217855223 BD For-Sale Unstable PLA2G2C 0 40 CC[C@H](CCO)NCCCCCC(=O)O ZINC000217855223 BD For-Sale Unstable Q6UB75_PIG 0 42 CC[C@H](CCO)NCCCCCC(=O)O ZINC000217855223 BD For-Sale Unstable SLC22A20 0 42 CC[C@H](CCO)NCCCCCC(=O)O ZINC000217855223 BD For-Sale Unstable CQSS 40 30 Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217855234 CH For-Sale Unstable ALOX5 21 51 Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217855234 CH For-Sale Unstable MAOB 46 41 Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217855234 CH For-Sale Unstable PTGER2 29 48 Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217855234 CH For-Sale Unstable PTGER4 47 54 Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217855234 CH For-Sale Unstable CA7 0 40 Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217855234 CH For-Sale Unstable PTGER3 40 54 Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217855234 CH For-Sale Unstable DRTS_LEIMA 30 41 Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217855234 CH For-Sale Unstable LTB4R 26 40 Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217855234 CH For-Sale Unstable PTGDR 0 49 Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217855234 CH For-Sale Unstable FFAR1 64 50 Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217855234 CH For-Sale Unstable AKR1C3 40 51 Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217855234 CH For-Sale Unstable AKR1B10 24 42 Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217855234 CH For-Sale Unstable PDS 29 40 COc1ccc(-c2coc3ccc(OC/C=C/c4ccccc4)cc23)cc1 ZINC000217855253 FK In-Stock Unstable ALDH2 65 38 COc1ccc(-c2coc3ccc(OC/C=C/c4ccccc4)cc23)cc1 ZINC000217855253 FK In-Stock Unstable SHC 17 42 CC1CCN(c2ccc([C@@H](C)NC(=O)c3ccc(Cl)cc3Cl)cc2)CC1 ZINC000217855262 GK In-Stock Unstable PTGER4 20 40 CC1CCN(c2ccc([C@@H](C)NC(=O)c3ccc(Cl)cc3Cl)cc2)CC1 ZINC000217855262 GK In-Stock Unstable SDH1 0 41 CCc1ccc(-c2nc(CC(=O)N3CCC[C@H]3c3ccccc3)cs2)cc1 ZINC000217855276 GK On-Demand Unstable PRCP 30 41 CCc1ccc(-c2nc(CC(=O)N3CCC[C@H]3c3ccccc3)cs2)cc1 ZINC000217855276 GK On-Demand Unstable ADAM17 41 45 CCc1ccc(-c2nc(CC(=O)N3CCC[C@H]3c3ccccc3)cs2)cc1 ZINC000217855276 GK On-Demand Unstable COLA 114 49 CCc1ccc(-c2nc(CC(=O)N3CCC[C@H]3c3ccccc3)cs2)cc1 ZINC000217855276 GK On-Demand Unstable CPT1A 108 49 CCc1ccc(-c2nc(CC(=O)N3CCC[C@H]3c3ccccc3)cs2)cc1 ZINC000217855276 GK On-Demand Unstable PREP 53 32 Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2F)c1 ZINC000217855286 CH For-Sale Unstable PTGER2 44 42 Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2F)c1 ZINC000217855286 CH For-Sale Unstable PTGER4 28 41 Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2F)c1 ZINC000217855286 CH For-Sale Unstable PTGER3 22 41 Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2F)c1 ZINC000217855286 CH For-Sale Unstable CDC25B 24 41 Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2F)c1 ZINC000217855286 CH For-Sale Unstable FFAR1 28 40 Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2F)c1 ZINC000217855286 CH For-Sale Unstable AKR1C3 33 46 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1Cl ZINC000217855303 FG For-Sale Unstable NPY1R 43 35 CC1CCN(c2ccc([C@H](C)NC(=O)c3ccc(Cl)cc3Cl)cc2)CC1 ZINC000217855341 GK In-Stock Unstable PTGER4 20 40 CC1CCN(c2ccc([C@H](C)NC(=O)c3ccc(Cl)cc3Cl)cc2)CC1 ZINC000217855341 GK In-Stock Unstable SDH1 0 41 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(O)c(Cl)c2)CC(=O)O4)cc1O ZINC000217855357 JJ In-Stock Unstable AKR1B1 0 49 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(O)c(Cl)c2)CC(=O)O4)cc1O ZINC000217855357 JJ In-Stock Unstable CYP1B1 59 39 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(O)c(Cl)c2)CC(=O)O4)cc1O ZINC000217855357 JJ In-Stock Unstable CYP1A1 45 47 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc(F)c(F)c1 ZINC000217855397 FF For-Sale Unstable HTR7 15 41 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc(F)c(F)c1 ZINC000217855397 FF For-Sale Unstable ADAMTS5 38 42 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc(F)c(F)c1 ZINC000217855397 FF For-Sale Unstable SFRP1 99 34 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc(F)c(F)c1 ZINC000217855397 FF For-Sale Unstable WNT3 83 34 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(O)c(Cl)c2)CC(=O)O4)cc1O ZINC000217855418 JJ In-Stock Unstable AKR1B1 0 49 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(O)c(Cl)c2)CC(=O)O4)cc1O ZINC000217855418 JJ In-Stock Unstable CYP1B1 59 39 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(O)c(Cl)c2)CC(=O)O4)cc1O ZINC000217855418 JJ In-Stock Unstable CYP1A1 45 47 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)c3ccc(Cl)cc3Cl)cc2)C1 ZINC000217855436 GK In-Stock Unstable HRH3 0 40 CCN1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217855443 CD For-Sale Unstable PTGER2 48 49 CCN1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217855443 CD For-Sale Unstable PTGER4 24 49 CCN1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217855443 CD For-Sale Unstable PTGER3 22 49 O=C(CN1CCN(C(=O)c2cc(N3CCCC3)ccn2)CC1)NCc1ccccc1 ZINC000217855459 HD On-Demand Unstable HTR1A 17 41 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc(F)c(F)c1 ZINC000217855468 FF For-Sale Unstable HTR7 15 41 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc(F)c(F)c1 ZINC000217855468 FF For-Sale Unstable ADAMTS5 38 42 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc(F)c(F)c1 ZINC000217855468 FF For-Sale Unstable SFRP1 99 34 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc(F)c(F)c1 ZINC000217855468 FF For-Sale Unstable WNT3 83 34 CC[C@@H]1CCN(c2ccc(CBr)cc2C(F)(F)F)C1 ZINC000217855481 EJ For-Sale Unstable LIPG 31 41 C[C@H]1CN(C(=O)c2ncn(-c3ccccc3)n2)CCN1 ZINC000217855497 CC On-Demand Unstable REN 35 48 C[C@H](NC(=O)c1ccc(Cl)cc1Cl)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217855523 GK In-Stock Unstable HRH3 0 40 CN1CCCC[C@@H]1CCOc1cc(Cl)ccc1Cl ZINC000217855537 CI For-Sale Unstable HRH1 22 48 CN1CCCC[C@@H]1CCOc1cc(Cl)ccc1Cl ZINC000217855537 CI For-Sale Unstable CHRNA10 78 51 CN1CCCC[C@@H]1CCOc1cc(Cl)ccc1Cl ZINC000217855537 CI For-Sale Unstable ACKR3 68 34 CCN1CCN(Cc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217855556 CD For-Sale Unstable SIGMAR1 32 48 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1cc(F)ccc1F ZINC000217855560 FF For-Sale Unstable NPY1R 41 33 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1cc(F)ccc1F ZINC000217855560 FF For-Sale Unstable NPY2R 56 35 CC[C@H]1CCN(c2ccc(CBr)cc2C(F)(F)F)C1 ZINC000217855583 EJ For-Sale Unstable LIPG 31 41 CN1CCCC[C@H]1CCOc1cc(Cl)ccc1Cl ZINC000217855618 CI For-Sale Unstable HRH1 22 48 CN1CCCC[C@H]1CCOc1cc(Cl)ccc1Cl ZINC000217855618 CI For-Sale Unstable CHRNA10 78 51 CN1CCCC[C@H]1CCOc1cc(Cl)ccc1Cl ZINC000217855618 CI For-Sale Unstable ACKR3 68 34 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1cc(F)ccc1F ZINC000217855623 FF For-Sale Unstable NPY1R 41 33 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1cc(F)ccc1F ZINC000217855623 FF For-Sale Unstable NPY2R 56 35 O=C(O)CCCc1ccc2cnn(-c3ccc(F)cc3)c2c1 ZINC000217855641 CH For-Sale Unstable NR3C1 28 41 O=C(O)CCCc1ccc2cnn(-c3ccc(F)cc3)c2c1 ZINC000217855641 CH For-Sale Unstable PLA2G4A 25 40 Cc1ccc2c(c1)[C@@H](NC(=O)c1ccc(Cl)cc1Cl)CC(C)(C)O2 ZINC000217855643 FK In-Stock Unstable CNR1 16 47 Cc1ccc2c(c1)[C@H](NC(=O)c1ccc(Cl)cc1Cl)CC(C)(C)O2 ZINC000217855745 FK In-Stock Unstable CNR1 16 47 CCOC(=O)CCCc1ccc2cnn(-c3ccc(F)cc3)c2c1 ZINC000217855758 EI For-Sale Unstable NR3C1 31 40 Cc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1ccc(Cl)cc1Cl ZINC000217855822 FK In-Stock Unstable CNR1 17 47 Cc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1ccc(Cl)cc1Cl ZINC000217855822 FK In-Stock Unstable SLC6A9 46 36 CCCCNC(=O)[C@@H](C)N[C@@H](CC)CCO ZINC000217855860 BD For-Sale Unstable DPP7 0 40 O=C1CCCc2cc3c(cnn3-c3ccc(F)cc3)cc2C1 ZINC000217855867 CH For-Sale Unstable NR3C1 30 41 CCCCN(CCCC)Cc1ccccc1/C=C\C(=O)O ZINC000217855878 CI For-Sale Unstable PTGER2 22 44 CCCCN(CCCC)Cc1ccccc1/C=C\C(=O)O ZINC000217855878 CI For-Sale Unstable PTGER4 23 50 CCCCN(CCCC)Cc1ccccc1/C=C\C(=O)O ZINC000217855878 CI For-Sale Unstable PTGER3 19 50 CCCCN(CCCC)Cc1ccccc1/C=C\C(=O)O ZINC000217855878 CI For-Sale Unstable PTGDR 0 48 CCCCN(CCCC)Cc1ccccc1/C=C\C(=O)O ZINC000217855878 CI For-Sale Unstable PLM2_PLAFA 32 40 Cc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1ccc(Cl)cc1Cl ZINC000217855884 FK In-Stock Unstable CNR1 17 47 Cc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1ccc(Cl)cc1Cl ZINC000217855884 FK In-Stock Unstable SLC6A9 43 36 CCCCNC(=O)[C@H](C)N[C@@H](CC)CCO ZINC000217855947 BD For-Sale Unstable DPP7 0 40 CC[C@H]1C(=O)CCCc2cc3c(cnn3-c3ccc(F)cc3)cc21 ZINC000217855968 DJ For-Sale Unstable NR3C1 46 41 CCCCN(CCCC)Cc1ccc(/C=C\C(=O)O)cc1 ZINC000217855991 CI For-Sale Unstable PLM2_PLAFA 37 41 CCCCN(CCCC)Cc1ccc(/C=C\C(=O)O)cc1 ZINC000217855991 CI For-Sale Unstable AKR1C3 27 40 CCCCN(CCCC)Cc1ccc(/C=C\C(=O)O)cc1 ZINC000217855991 CI For-Sale Unstable TRPM2 0 40 CCCCNC(=O)[C@@H](C)N[C@H](CC)CCO ZINC000217856018 BD For-Sale Unstable DPP7 0 40 CC[C@@H]1C(=O)CCCc2cc3c(cnn3-c3ccc(F)cc3)cc21 ZINC000217856032 DJ For-Sale Unstable NR3C1 46 41 CCCCNC(=O)[C@H](C)N[C@H](CC)CCO ZINC000217856081 BD For-Sale Unstable DPP7 0 40 CCN(Cc1ccc(OC)c(/C=C\C(=O)O)c1)C1CC1 ZINC000217856110 CF For-Sale Unstable PTGER2 34 41 CCN(Cc1ccc(OC)c(/C=C\C(=O)O)c1)C1CC1 ZINC000217856110 CF For-Sale Unstable PTGER4 0 41 CCN(Cc1ccc(OC)c(/C=C\C(=O)O)c1)C1CC1 ZINC000217856110 CF For-Sale Unstable PTGER3 15 41 CC(=O)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217856111 FF For-Sale Unstable ADAMTS5 39 42 CC(=O)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217856111 FF For-Sale Unstable SFRP1 106 35 CC(=O)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217856111 FF For-Sale Unstable LIMK2 29 41 CC(=O)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217856111 FF For-Sale Unstable WNT3 70 32 COc1ccccc1-n1c(C[C@@H]2CCCN(C(=O)/C=C/c3ccco3)C2)n[nH]c1=O ZINC000217856146 HF In-Stock Unstable HTR1A 41 37 COc1ccccc1-n1c(C[C@@H]2CCCN(C(=O)/C=C/c3ccco3)C2)n[nH]c1=O ZINC000217856146 HF In-Stock Unstable DRD2 23 47 COc1ccccc1-n1c(C[C@@H]2CCCN(C(=O)/C=C/c3ccco3)C2)n[nH]c1=O ZINC000217856146 HF In-Stock Unstable DRD3 27 47 COc1cc2oc(=O)cc(-c3ccccc3)c2cc1CCC(=O)N[C@H](CO)c1ccccc1 ZINC000217856168 II In-Stock Unstable CMA1 15 44 COc1cc2oc(=O)cc(-c3ccccc3)c2cc1CCC(=O)N[C@H](CO)c1ccccc1 ZINC000217856168 II In-Stock Unstable GPR88 0 40 O[C@@H]1CN(Cc2ccoc2)CCN(Cc2nc3ccccc3[nH]2)C1 ZINC000217856177 ED In-Stock Unstable DRD4 15 53 CSC[C@@](C)(O)CNCc1ccc(C(F)(F)F)cc1 ZINC000217856178 CF On-Demand Unstable PETD 0 40 CC(=O)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217856186 FF For-Sale Unstable ADAMTS5 39 42 CC(=O)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217856186 FF For-Sale Unstable SFRP1 106 35 CC(=O)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217856186 FF For-Sale Unstable LIMK2 29 41 CC(=O)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217856186 FF For-Sale Unstable WNT3 70 32 COc1ccccc1-n1c(C[C@H]2CCCN(C(=O)/C=C/c3ccco3)C2)n[nH]c1=O ZINC000217856232 HF In-Stock Unstable HTR1A 41 37 COc1ccccc1-n1c(C[C@H]2CCCN(C(=O)/C=C/c3ccco3)C2)n[nH]c1=O ZINC000217856232 HF In-Stock Unstable DRD2 23 47 COc1ccccc1-n1c(C[C@H]2CCCN(C(=O)/C=C/c3ccco3)C2)n[nH]c1=O ZINC000217856232 HF In-Stock Unstable DRD3 27 47 CSC[C@](C)(O)CNCc1ccc(C(F)(F)F)cc1 ZINC000217856242 CF On-Demand Unstable PETD 0 40 COc1cccc([C@@H]2CC(=O)Oc3c(C(C)=O)c(O)c4c(C)cc(=O)oc4c32)c1OCc1ccccc1 ZINC000217856248 KK In-Stock Unstable KCNA3 40 38 CC[C@@H](NC(=O)c1ccc(Cl)cc1Cl)c1ccc(C)c(C)c1 ZINC000217856300 EK In-Stock Unstable UTS2 48 37 COc1ccccc1-n1c(C[C@@H]2CCCN(C(=O)c3ccco3)C2)n[nH]c1=O ZINC000217856304 GE In-Stock Unstable HTR1A 50 47 COc1ccccc1-n1c(C[C@@H]2CCCN(C(=O)c3ccco3)C2)n[nH]c1=O ZINC000217856304 GE In-Stock Unstable DRD2 34 45 COc1ccccc1-n1c(C[C@@H]2CCCN(C(=O)c3ccco3)C2)n[nH]c1=O ZINC000217856304 GE In-Stock Unstable ADRA1D 37 47 COc1ccccc1-n1c(C[C@@H]2CCCN(C(=O)c3ccco3)C2)n[nH]c1=O ZINC000217856304 GE In-Stock Unstable ADRA1A 31 47 CC(=O)c1cccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217856306 FF For-Sale Unstable NPY2R 48 36 CC(=O)c1cccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217856306 FF For-Sale Unstable AKR1C3 60 38 CC(=O)c1cccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217856306 FF For-Sale Unstable SFRP1 113 38 CC(=O)c1cccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217856306 FF For-Sale Unstable WNT3 76 33 COc1cccc([C@H]2CC(=O)Oc3c(C(C)=O)c(O)c4c(C)cc(=O)oc4c32)c1OCc1ccccc1 ZINC000217856314 KK In-Stock Unstable KCNA3 40 38 COc1cccc(C[C@H](O)[C@@H]2CN(C)CCO2)c1 ZINC000217856321 CC For-Sale Unstable VACHT_TETCF 0 47 CC(=O)c1cccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217856360 FF For-Sale Unstable NPY2R 48 36 CC(=O)c1cccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217856360 FF For-Sale Unstable AKR1C3 60 38 CC(=O)c1cccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217856360 FF For-Sale Unstable SFRP1 113 38 CC(=O)c1cccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217856360 FF For-Sale Unstable WNT3 76 33 CC[C@H](NC(=O)c1ccc(Cl)cc1Cl)c1ccc(C)c(C)c1 ZINC000217856365 EK In-Stock Unstable UTS2 48 37 COc1ccccc1-n1c(C[C@H]2CCCN(C(=O)c3ccco3)C2)n[nH]c1=O ZINC000217856377 GE In-Stock Unstable HTR1A 63 47 COc1ccccc1-n1c(C[C@H]2CCCN(C(=O)c3ccco3)C2)n[nH]c1=O ZINC000217856377 GE In-Stock Unstable DRD2 40 45 COc1ccccc1-n1c(C[C@H]2CCCN(C(=O)c3ccco3)C2)n[nH]c1=O ZINC000217856377 GE In-Stock Unstable ADRA1D 42 47 COc1ccccc1-n1c(C[C@H]2CCCN(C(=O)c3ccco3)C2)n[nH]c1=O ZINC000217856377 GE In-Stock Unstable ADRA1A 39 47 COc1ccccc1-n1c(C[C@H]2CCCN(C(=O)c3ccco3)C2)n[nH]c1=O ZINC000217856377 GE In-Stock Unstable ADRA1B 33 47 COc1ccccc1-n1c(C[C@H]2CCCN(C(=O)c3ccco3)C2)n[nH]c1=O ZINC000217856377 GE In-Stock Unstable DRD3 41 39 COc1cccc(C[C@H](O)[C@H]2CN(C)CCO2)c1 ZINC000217856387 CC For-Sale Unstable VACHT_TETCF 0 47 COc1ccc(-c2n[nH]cc2C(=O)NC[C@@H]2CCCN3CCCC[C@H]23)cc1Cl ZINC000217856423 HH In-Stock Unstable PDE5A 24 41 COc1ccc(-c2n[nH]cc2C(=O)NC[C@@H]2CCCN3CCCC[C@H]23)cc1Cl ZINC000217856423 HH In-Stock Unstable HTR4 41 55 CC[C@@H](NC(=O)c1ccc(Cl)cc1Cl)c1ccc(C)cc1C ZINC000217856461 EK In-Stock Unstable SLC6A9 40 38 CC[C@@H](NC(=O)c1ccc(Cl)cc1Cl)c1ccc(C)cc1C ZINC000217856461 EK In-Stock Unstable UTS2 40 32 COc1ccccc1-n1c(C[C@H]2CCCN(C(=O)c3cc(C)oc3C)C2)n[nH]c1=O ZINC000217856481 HF In-Stock Unstable HTR1A 56 37 COc1ccccc1-n1c(C[C@H]2CCCN(C(=O)c3cc(C)oc3C)C2)n[nH]c1=O ZINC000217856481 HF In-Stock Unstable DRD3 40 38 COc1ccccc1-n1c(C[C@H]2CCCN(C(=O)c3cc(C)oc3C)C2)n[nH]c1=O ZINC000217856481 HF In-Stock Unstable TACR3 20 40 CCCc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217856482 FH For-Sale Unstable ADAMTS5 27 57 CC(C)[C@H](NC(=O)COc1ccc2c(-c3ccccc3)cc(=O)oc2c1)c1nc2ccccc2n1C ZINC000217856514 JK In-Stock Unstable ALDH2 52 32 CC(C)[C@H](NC(=O)COc1ccc2c(-c3ccccc3)cc(=O)oc2c1)c1nc2ccccc2n1C ZINC000217856514 JK In-Stock Unstable MAOA 39 41 CC(C)[C@H](NC(=O)COc1ccc2c(-c3ccccc3)cc(=O)oc2c1)c1nc2ccccc2n1C ZINC000217856514 JK In-Stock Unstable MAOB 30 46 CC(C)[C@H](NC(=O)COc1ccc2c(-c3ccccc3)cc(=O)oc2c1)c1nc2ccccc2n1C ZINC000217856514 JK In-Stock Unstable BCHE 21 43 CC[C@H](NC(=O)c1ccc(Cl)cc1Cl)c1ccc(C)cc1C ZINC000217856532 EK In-Stock Unstable SLC6A9 40 38 CC[C@H](NC(=O)c1ccc(Cl)cc1Cl)c1ccc(C)cc1C ZINC000217856532 EK In-Stock Unstable UTS2 40 32 CCCc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217856572 FH For-Sale Unstable ADAMTS5 43 58 COc1ccccc1-n1c(C[C@@H]2CCCN(C(=O)c3cc(C)oc3C)C2)n[nH]c1=O ZINC000217856574 HF In-Stock Unstable HTR1A 56 37 COc1ccccc1-n1c(C[C@@H]2CCCN(C(=O)c3cc(C)oc3C)C2)n[nH]c1=O ZINC000217856574 HF In-Stock Unstable DRD3 40 38 COc1ccccc1-n1c(C[C@@H]2CCCN(C(=O)c3cc(C)oc3C)C2)n[nH]c1=O ZINC000217856574 HF In-Stock Unstable TACR3 20 40 CC(C)C[C@H](NC(=O)c1ccc2c(ccn2C)c1)C(=O)O ZINC000217856637 CE In-Stock Unstable CA2 15 51 CC(C)C[C@H](NC(=O)c1ccc2c(ccn2C)c1)C(=O)O ZINC000217856637 CE In-Stock Unstable CCKAR 0 40 CC(C)C[C@H](NC(=O)c1ccc2c(ccn2C)c1)C(=O)O ZINC000217856637 CE In-Stock Unstable NTSR1 27 40 CC(C)C[C@H](NC(=O)c1ccc2c(ccn2C)c1)C(=O)O ZINC000217856637 CE In-Stock Unstable CTSK 19 41 CC(C)C[C@H](NC(=O)c1ccc2c(ccn2C)c1)C(=O)O ZINC000217856637 CE In-Stock Unstable CTSL 23 41 CC(C)C[C@H](NC(=O)c1ccc2c(ccn2C)c1)C(=O)O ZINC000217856637 CE In-Stock Unstable CCKBR 34 40 CC(C)C[C@H](NC(=O)c1ccc2c(ccn2C)c1)C(=O)O ZINC000217856637 CE In-Stock Unstable CAPN2 0 40 CC(C)C[C@H](NC(=O)c1ccc2c(ccn2C)c1)C(=O)O ZINC000217856637 CE In-Stock Unstable FPR1 45 34 CC[C@@H](NC(=O)c1ccc(Cl)cc1Cl)c1ccc(OC)c(OC)c1 ZINC000217856641 FJ In-Stock Unstable CMA1 31 42 CC[C@@H](NC(=O)c1ccc(Cl)cc1Cl)c1ccc(OC)c(OC)c1 ZINC000217856641 FJ In-Stock Unstable PTGER3 22 41 CC[C@@H](NC(=O)c1ccc(Cl)cc1Cl)c1ccc(OC)c(OC)c1 ZINC000217856641 FJ In-Stock Unstable PYGL 19 46 CC[C@@H](NC(=O)c1ccc(Cl)cc1Cl)c1ccc(OC)c(OC)c1 ZINC000217856641 FJ In-Stock Unstable TTR 0 41 CC[C@@H](NC(=O)c1ccc(Cl)cc1Cl)c1ccc(OC)c(OC)c1 ZINC000217856641 FJ In-Stock Unstable UTS2 54 38 CC[C@@H](NC(=O)c1ccc(Cl)cc1Cl)c1ccc(OC)c(OC)c1 ZINC000217856641 FJ In-Stock Unstable CYSP_PLAFA 34 41 Cc1cc(C)c(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)c(C)c1 ZINC000217856689 FH For-Sale Unstable NR3C2 25 40 Cc1nc2ccccc2c(-c2ccccc2)c1CC(=O)N1CCN(C(=O)CN2CCOCC2)CC1 ZINC000217856700 JF On-Demand Unstable TSPO 17 52 Cc1nc2ccccc2c(-c2ccccc2)c1CC(=O)N1CCN(C(=O)CN2CCOCC2)CC1 ZINC000217856700 JF On-Demand Unstable PTGDS 41 35 O=C(c1cc(-c2ccccc2)n[nH]1)N1CCC[C@H](Cc2n[nH]c(=O)n2-c2ccccc2F)C1 ZINC000217856701 IG In-Stock Unstable TACR3 21 45 CC[C@H](NC(=O)c1ccc(Cl)cc1Cl)c1ccc(OC)c(OC)c1 ZINC000217856723 FJ In-Stock Unstable CMA1 31 42 CC[C@H](NC(=O)c1ccc(Cl)cc1Cl)c1ccc(OC)c(OC)c1 ZINC000217856723 FJ In-Stock Unstable PTGER3 22 41 CC[C@H](NC(=O)c1ccc(Cl)cc1Cl)c1ccc(OC)c(OC)c1 ZINC000217856723 FJ In-Stock Unstable PYGL 19 46 CC[C@H](NC(=O)c1ccc(Cl)cc1Cl)c1ccc(OC)c(OC)c1 ZINC000217856723 FJ In-Stock Unstable TTR 0 41 CC[C@H](NC(=O)c1ccc(Cl)cc1Cl)c1ccc(OC)c(OC)c1 ZINC000217856723 FJ In-Stock Unstable UTS2 54 38 CC[C@H](NC(=O)c1ccc(Cl)cc1Cl)c1ccc(OC)c(OC)c1 ZINC000217856723 FJ In-Stock Unstable CYSP_PLAFA 34 41 O=C(c1cc(-c2ccccc2)n[nH]1)N1CCC[C@@H](Cc2n[nH]c(=O)n2-c2ccccc2F)C1 ZINC000217856775 IG In-Stock Unstable TACR3 21 45 Cc1cc(C)c(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)c(C)c1 ZINC000217856778 FH For-Sale Unstable NR3C2 25 40 CNC(=O)CN(C)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217856793 CC For-Sale Unstable TUBB1 41 36 CNC(=O)CN(C)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217856793 CC For-Sale Unstable AKR1C3 21 40 CCc1ccc(-c2nc(CC(=O)N3CCN(C(=O)CN4CCOCC4)CC3)cs2)cc1 ZINC000217856800 ID On-Demand Unstable LTA4H 16 41 CC[C@@H](NC(=O)c1ccc(Cl)cc1Cl)c1ccc(S(C)(=O)=O)cc1 ZINC000217856822 GI In-Stock Unstable PTGS2 21 43 CC[C@@H](NC(=O)c1ccc(Cl)cc1Cl)c1ccc(S(C)(=O)=O)cc1 ZINC000217856822 GI In-Stock Unstable SLC6A9 49 41 CC[C@@H](NC(=O)c1ccc(Cl)cc1Cl)c1ccc(S(C)(=O)=O)cc1 ZINC000217856822 GI In-Stock Unstable UTS2 47 38 CNC(=O)CN(C)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217856891 CC For-Sale Unstable PTGER2 27 41 CNC(=O)CN(C)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217856891 CC For-Sale Unstable PTGER4 0 41 Cc1cc(C)c(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1C ZINC000217856892 FH For-Sale Unstable NPY1R 40 32 O=C(O)CC[C@@H](NC(=O)[C@@H]1C[C@@H]2CCCC[C@@H]2N1)C(=O)O ZINC000217856905 CC For-Sale Unstable FOLH1 41 43 O=C(O)CC[C@@H](NC(=O)[C@@H]1C[C@@H]2CCCC[C@@H]2N1)C(=O)O ZINC000217856905 CC For-Sale Unstable NAALAD2 53 43 CC[C@H](NC(=O)c1ccc(Cl)cc1Cl)c1ccc(S(C)(=O)=O)cc1 ZINC000217856912 GI In-Stock Unstable SLC6A9 47 41 CC[C@H](NC(=O)c1ccc(Cl)cc1Cl)c1ccc(S(C)(=O)=O)cc1 ZINC000217856912 GI In-Stock Unstable UTS2 47 38 Cc1cc(C)c(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1C ZINC000217856957 FH For-Sale Unstable NPY1R 40 32 O=C(O)CC[C@H](NC(=O)[C@@H]1C[C@@H]2CCCC[C@@H]2N1)C(=O)O ZINC000217856968 CC For-Sale Unstable FOLH1 41 43 O=C(O)CC[C@H](NC(=O)[C@@H]1C[C@@H]2CCCC[C@@H]2N1)C(=O)O ZINC000217856968 CC For-Sale Unstable NAALAD2 53 43 COc1ccc(-c2noc(CNC(=O)c3ccc(Cl)cc3Cl)n2)c(OC)c1 ZINC000217857016 HH In-Stock Unstable COLA 46 34 COc1ccc(-c2noc(CNC(=O)c3ccc(Cl)cc3Cl)n2)c(OC)c1 ZINC000217857016 HH In-Stock Unstable CPT1A 46 34 COc1ccc(-c2noc(CNC(=O)c3ccc(Cl)cc3Cl)n2)c(OC)c1 ZINC000217857016 HH In-Stock Unstable SLC6A9 42 36 COc1ccc(-c2noc(CNC(=O)c3ccc(Cl)cc3Cl)n2)c(OC)c1 ZINC000217857016 HH In-Stock Unstable CPT1B 49 31 COc1ccc(-c2noc(CNC(=O)c3ccc(Cl)cc3Cl)n2)c(OC)c1 ZINC000217857016 HH In-Stock Unstable PDK1 37 45 COc1ccc(-c2noc(CNC(=O)c3ccc(Cl)cc3Cl)n2)c(OC)c1 ZINC000217857016 HH In-Stock Unstable U38 0 42 COc1ccc(-c2noc(CNC(=O)c3ccc(Cl)cc3Cl)n2)c(OC)c1 ZINC000217857016 HH In-Stock Unstable CYSP_PLAFA 33 43 O=C(N/C=C/c1ccccc1Br)Nc1ccc(Nc2ccccc2)cc1 ZINC000217857038 HK For-Sale Anodyne EPHX1 0 43 O=C(N/C=C/c1ccccc1Br)Nc1ccc(Nc2ccccc2)cc1 ZINC000217857038 HK For-Sale Anodyne MTCA1 15 40 O=C(N/C=C/c1ccccc1Br)Nc1ccc(Nc2ccccc2)cc1 ZINC000217857038 HK For-Sale Anodyne P96878_MYCTU 22 40 O=C(N/C=C/c1ccccc1Br)Nc1ccc(Nc2ccccc2)cc1 ZINC000217857038 HK For-Sale Anodyne P95276_MYCTO 0 43 C[C@@H]1CN(Cc2ccc(F)c(/C=C\C(=O)O)c2)[C@H](C)CO1 ZINC000217857052 CF For-Sale Unstable CCR1 24 42 O=C(O)CC[C@@H](NC(=O)[C@H]1C[C@@H]2CCCC[C@@H]2N1)C(=O)O ZINC000217857054 CC For-Sale Unstable FOLH1 41 43 O=C(O)CC[C@@H](NC(=O)[C@H]1C[C@@H]2CCCC[C@@H]2N1)C(=O)O ZINC000217857054 CC For-Sale Unstable NAALAD2 53 43 CC[C@@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C1CC1 ZINC000217857059 CF For-Sale Unstable ACE 33 44 CC[C@@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C1CC1 ZINC000217857059 CF For-Sale Unstable MME 42 44 CC[C@@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C1CC1 ZINC000217857059 CF For-Sale Unstable TACR3 29 41 CC[C@@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C1CC1 ZINC000217857059 CF For-Sale Unstable CAPN2 61 40 CC[C@@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C1CC1 ZINC000217857059 CF For-Sale Unstable ACE2 56 37 CC[C@@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C1CC1 ZINC000217857059 CF For-Sale Unstable XIAP 82 41 CC[C@@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C1CC1 ZINC000217857059 CF For-Sale Unstable BIRC8 43 31 CC(C)(C)OC(=O)N1CCC(c2cc(C(N)=O)n[nH]2)CC1 ZINC000217857070 CD In-Stock Unstable GPR119 39 44 CC(C)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217857077 FH For-Sale Unstable ADAMTS5 37 45 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC1CCOCC1 ZINC000217857088 BG On-Demand Unstable TRPM8 15 40 CC[C@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C1CC1 ZINC000217857131 CF For-Sale Unstable ACE 33 44 CC[C@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C1CC1 ZINC000217857131 CF For-Sale Unstable MME 42 44 CC[C@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C1CC1 ZINC000217857131 CF For-Sale Unstable TACR3 29 41 CC[C@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C1CC1 ZINC000217857131 CF For-Sale Unstable CAPN2 61 40 CC[C@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C1CC1 ZINC000217857131 CF For-Sale Unstable ACE2 56 37 CC[C@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C1CC1 ZINC000217857131 CF For-Sale Unstable XIAP 82 41 CC[C@H](C)[C@@H](N)C(=O)N[C@H](c1ccccc1)C1CC1 ZINC000217857131 CF For-Sale Unstable BIRC8 43 31 CC(C)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217857153 FH For-Sale Unstable ADAMTS5 37 45 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC1CCOCC1 ZINC000217857174 BG On-Demand Unstable TRPM8 15 40 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC1CCOCC1 ZINC000217857236 BG For-Sale Unstable TRPM8 15 40 Cc1cccc(NC(=O)N/C=C/c2ccccc2Br)n1 ZINC000217857250 EH For-Sale Unstable GRM5 17 46 Cc1cccc(NC(=O)N/C=C/c2ccccc2Br)n1 ZINC000217857250 EH For-Sale Unstable SORT1 16 42 CCOc1ccccc1S(=O)(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217857255 FG For-Sale Unstable NPY1R 42 34 CCOc1ccccc1S(=O)(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217857255 FG For-Sale Unstable NPY2R 43 39 CCOc1ccccc1S(=O)(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217857255 FG For-Sale Unstable ADAMTS5 32 41 COc1ccc(-c2noc(CN(C)C(=O)c3ccc(Cl)cc3Cl)n2)c(OC)c1 ZINC000217857257 HI In-Stock Unstable CYSP_PLAFA 32 42 CCN(Cc1ccccc1/C=C\C(=O)O)C1CCCC1 ZINC000217857260 CH For-Sale Unstable PTGER2 43 48 CCN(Cc1ccccc1/C=C\C(=O)O)C1CCCC1 ZINC000217857260 CH For-Sale Unstable PTGER4 0 48 CCN(Cc1ccccc1/C=C\C(=O)O)C1CCCC1 ZINC000217857260 CH For-Sale Unstable PTGER3 16 48 CCN(Cc1ccccc1/C=C\C(=O)O)C1CCCC1 ZINC000217857260 CH For-Sale Unstable PTGDR 0 46 CN1CCN(C(=O)C[C@@H](c2coc3ccccc3c2=O)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)CC1 ZINC000217857261 KH In-Stock Unstable TNKS 19 42 O=C(N[C@H](c1ccccc1)C1CC1)[C@@H]1C[C@@H](O)CN1 ZINC000217857288 CC For-Sale Unstable CTSC 21 40 CC1CCN(c2nnc(SCC(=O)c3cccc([N+](=O)[O-])c3)n2Cc2ccco2)CC1 ZINC000217857291 II On-Demand Unstable HCRTR2 20 41 O=C1CCCc2cc3c(cnn3-c3ccc(F)cc3)cc21 ZINC000217857301 CH For-Sale Unstable NR3C1 32 44 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC1CCOCC1 ZINC000217857324 BG For-Sale Unstable TRPM8 15 40 CN1CCN(C(=O)C[C@H](c2coc3ccccc3c2=O)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)CC1 ZINC000217857326 KH In-Stock Unstable TNKS 19 42 CCOc1ccccc1S(=O)(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217857329 FG For-Sale Unstable NPY1R 42 34 CCOc1ccccc1S(=O)(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217857329 FG For-Sale Unstable NPY2R 43 39 CCOc1ccccc1S(=O)(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217857329 FG For-Sale Unstable ADAMTS5 32 41 COc1ccc(Br)c(C(=O)NCCn2ccnc2-c2ccccn2)c1 ZINC000217857357 HG In-Stock Unstable DRD4 46 36 COc1ccc(Br)c(C(=O)NCCn2ccnc2-c2ccccn2)c1 ZINC000217857357 HG In-Stock Unstable DRD3 28 43 CCN(Cc1ccc(/C=C\C(=O)O)cc1)C1CCCC1 ZINC000217857364 CH For-Sale Unstable NR1H4 26 40 O=C(N[C@H](c1ccccc1)C1CC1)[C@H]1C[C@@H](O)CN1 ZINC000217857377 CC For-Sale Unstable CTSC 21 40 CC(C)c1ccc(CCCNC(=O)c2ccc(Cl)cc2Cl)cc1 ZINC000217857381 FK In-Stock Unstable CNR1 17 40 CC(C)c1ccc(CCCNC(=O)c2ccc(Cl)cc2Cl)cc1 ZINC000217857381 FK In-Stock Unstable SDH1 0 43 CC(C)c1ccc(CCCNC(=O)c2ccc(Cl)cc2Cl)cc1 ZINC000217857381 FK In-Stock Unstable SLC6A9 44 35 CC(C)c1ccc(CCCNC(=O)c2ccc(Cl)cc2Cl)cc1 ZINC000217857381 FK In-Stock Unstable SLC6A5 22 42 CC(C)c1ccc(CCCNC(=O)c2ccc(Cl)cc2Cl)cc1 ZINC000217857381 FK In-Stock Unstable ALPL 45 39 CC(C)c1ccc(CCCNC(=O)c2ccc(Cl)cc2Cl)cc1 ZINC000217857381 FK In-Stock Unstable MCL1 0 49 COc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1C ZINC000217857444 FF For-Sale Unstable NPY2R 42 36 COc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1C ZINC000217857444 FF For-Sale Unstable ADAMTS5 31 43 O=C(NCCCN1CCCc2ccccc21)c1ccc(Cl)cc1Cl ZINC000217857513 FJ In-Stock Unstable DRD2 30 42 O=C(NCCCN1CCCc2ccccc21)c1ccc(Cl)cc1Cl ZINC000217857513 FJ In-Stock Unstable CNR1 53 33 O=C(NCCCN1CCCc2ccccc21)c1ccc(Cl)cc1Cl ZINC000217857513 FJ In-Stock Unstable HTR2C 28 46 O=C(NCCCN1CCCc2ccccc21)c1ccc(Cl)cc1Cl ZINC000217857513 FJ In-Stock Unstable AVPR2 41 44 O=C(NCCCN1CCCc2ccccc21)c1ccc(Cl)cc1Cl ZINC000217857513 FJ In-Stock Unstable DRD3 44 41 O=C(NCCCN1CCCc2ccccc21)c1ccc(Cl)cc1Cl ZINC000217857513 FJ In-Stock Unstable AVPR1A 16 40 O=C(NCCCN1CCCc2ccccc21)c1ccc(Cl)cc1Cl ZINC000217857513 FJ In-Stock Unstable HRP1_PLAFA 26 41 O=C(NCCCN1CCCc2ccccc21)c1ccc(Cl)cc1Cl ZINC000217857513 FJ In-Stock Unstable SLC6A9 48 38 O=C(NCCCN1CCCc2ccccc21)c1ccc(Cl)cc1Cl ZINC000217857513 FJ In-Stock Unstable TYRO3 28 44 O=C(O)/C=C\c1cccc(OCCN2C(=O)CNC2=O)c1 ZINC000217857525 CC For-Sale Unstable 17HSDCL 0 40 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1C ZINC000217857526 FF For-Sale Unstable NPY2R 42 36 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1C ZINC000217857526 FF For-Sale Unstable ADAMTS5 31 43 O=C(N/C=C/c1ccccc1Br)Nc1cccnc1 ZINC000217857554 DH For-Sale Anodyne NAMPT 22 46 COc1ccc(CN(C)C(=O)c2ccc(C(C)(C)C)cc2)cc1 ZINC000217857604 DI In-Stock Unstable PTGDR 17 40 COc1ccc(CN(C)C(=O)c2ccc(C(C)(C)C)cc2)cc1 ZINC000217857604 DI In-Stock Unstable MT-ND1 39 70 COc1ccc(CN(C)C(=O)c2ccc(C(C)(C)C)cc2)cc1 ZINC000217857604 DI In-Stock Unstable HSD17B2 20 51 COc1ccc(CN(C)C(=O)c2ccc(C(C)(C)C)cc2)cc1 ZINC000217857604 DI In-Stock Unstable AOC3 15 44 COc1ccc(CN(C)C(=O)c2ccc(C(C)(C)C)cc2)cc1 ZINC000217857604 DI In-Stock Unstable MLYCD 18 51 COc1ccc(CN(C)C(=O)c2ccc(C(C)(C)C)cc2)cc1 ZINC000217857604 DI In-Stock Unstable LIMK2 39 45 COc1ccc(CN(C)C(=O)c2ccc(C(C)(C)C)cc2)cc1 ZINC000217857604 DI In-Stock Unstable E3UJZ5_SPOLI 27 40 O=C(O)/C=C\c1ccc(OCCN2C(=O)CNC2=O)cc1 ZINC000217857623 CC For-Sale Unstable 17HSDCL 0 41 COc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)c(C)c1 ZINC000217857649 FF For-Sale Unstable NPY1R 40 31 COc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)c(C)c1 ZINC000217857649 FF For-Sale Unstable NPY2R 58 41 COc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)c(C)c1 ZINC000217857649 FF For-Sale Unstable ADAMTS5 29 42 COc1ccc(/C=C\C(=O)O)cc1Cn1ccccc1=O ZINC000217857689 CE For-Sale Unstable TSHR 66 33 COc1ccc(/C=C\C(=O)O)cc1Cn1ccccc1=O ZINC000217857689 CE For-Sale Unstable PTGER3 17 43 COc1ccc(/C=C\C(=O)O)cc1Cn1ccccc1=O ZINC000217857689 CE For-Sale Unstable AKR1C3 31 40 Cc1ccc([C@@H](C)N2CC[C@@H](N3CCCCC3)C2)c(O)c1 ZINC000217857691 CG For-Sale Unstable L3MBTL3 53 34 Cc1ccc([C@@H](C)N2CC[C@@H](N3CCCCC3)C2)c(O)c1 ZINC000217857691 CG For-Sale Unstable MBTD1 0 41 CCS(=O)(=O)c1ccc(NC(=O)c2csc(-c3cccc(Cl)c3)n2)cc1 ZINC000217857694 HJ On-Demand Unstable CPT1A 45 35 CCS(=O)(=O)c1ccc(NC(=O)c2csc(-c3cccc(Cl)c3)n2)cc1 ZINC000217857694 HJ On-Demand Unstable GRM4 38 44 CCS(=O)(=O)c1ccc(NC(=O)c2csc(-c3cccc(Cl)c3)n2)cc1 ZINC000217857694 HJ On-Demand Unstable PFK 0 41 CCS(=O)(=O)c1ccc(NC(=O)c2csc(-c3cccc(Cl)c3)n2)cc1 ZINC000217857694 HJ On-Demand Unstable SMO 0 42 CCS(=O)(=O)c1ccc(NC(=O)c2csc(-c3cccc(Cl)c3)n2)cc1 ZINC000217857694 HJ On-Demand Unstable RORC 76 49 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)c(C)c1 ZINC000217857726 FF For-Sale Unstable NPY1R 40 31 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)c(C)c1 ZINC000217857726 FF For-Sale Unstable NPY2R 58 41 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)c(C)c1 ZINC000217857726 FF For-Sale Unstable ADAMTS5 29 42 COc1ccccc1CCCNC(=O)c1ccc(C(C)(C)C)cc1 ZINC000217857738 EI In-Stock Unstable DRD2 28 58 COc1ccccc1CCCNC(=O)c1ccc(C(C)(C)C)cc1 ZINC000217857738 EI In-Stock Unstable DRD1 0 46 COc1ccccc1CCCNC(=O)c1ccc(C(C)(C)C)cc1 ZINC000217857738 EI In-Stock Unstable DRD3 43 46 COc1ccccc1CCCNC(=O)c1ccc(C(C)(C)C)cc1 ZINC000217857738 EI In-Stock Unstable EDNRB 0 40 COc1ccccc1CCCNC(=O)c1ccc(C(C)(C)C)cc1 ZINC000217857738 EI In-Stock Unstable KCNQ1 0 43 COc1ccccc1CCCNC(=O)c1ccc(C(C)(C)C)cc1 ZINC000217857738 EI In-Stock Unstable TRPV1 29 41 COc1ccccc1CCCNC(=O)c1ccc(C(C)(C)C)cc1 ZINC000217857738 EI In-Stock Unstable MTNR1B 45 45 COc1ccccc1CCCNC(=O)c1ccc(C(C)(C)C)cc1 ZINC000217857738 EI In-Stock Unstable MT-ND1 34 51 COc1ccccc1CCCNC(=O)c1ccc(C(C)(C)C)cc1 ZINC000217857738 EI In-Stock Unstable CYNT 25 43 COc1ccccc1CCCNC(=O)c1ccc(C(C)(C)C)cc1 ZINC000217857738 EI In-Stock Unstable MBTPS1 41 33 COc1ccccc1CCCNC(=O)c1ccc(C(C)(C)C)cc1 ZINC000217857738 EI In-Stock Unstable AP2S1 0 47 COc1ccccc1CCCNC(=O)c1ccc(C(C)(C)C)cc1 ZINC000217857738 EI In-Stock Unstable ALPHA-1A 0 42 Cc1ccc([C@H](C)N2CC[C@@H](N3CCCCC3)C2)c(O)c1 ZINC000217857768 CG For-Sale Unstable L3MBTL3 53 34 Cc1ccc([C@H](C)N2CC[C@@H](N3CCCCC3)C2)c(O)c1 ZINC000217857768 CG For-Sale Unstable MBTD1 0 41 O=C(NCCn1ccnc1-c1ccccn1)C1CC1 ZINC000217857779 CD In-Stock Unstable GPBAR1 15 40 COc1ccc(Cn2ccccc2=O)cc1/C=C\C(=O)O ZINC000217857789 CE For-Sale Unstable PTGER4 23 46 COc1ccc(Cn2ccccc2=O)cc1/C=C\C(=O)O ZINC000217857789 CE For-Sale Unstable PTGER3 32 43 COc1ccc(Cn2ccccc2=O)cc1/C=C\C(=O)O ZINC000217857789 CE For-Sale Unstable AKR1B10 29 40 O=C(Cc1csc(-c2ccccn2)n1)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217857796 FG In-Stock Unstable COLA 0 46 O=C(Cc1csc(-c2ccccn2)n1)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217857796 FG In-Stock Unstable CPT1A 18 46 COc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1F ZINC000217857833 FF For-Sale Unstable NPY2R 53 36 COc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1F ZINC000217857833 FF For-Sale Unstable ADAMTS5 34 40 COc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1F ZINC000217857833 FF For-Sale Unstable SFRP1 53 31 COc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1F ZINC000217857833 FF For-Sale Unstable ACKR3 62 32 CC(C)(C)c1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217857834 FK In-Stock Unstable SRD5A2 26 50 CC(C)(C)c1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217857834 FK In-Stock Unstable PPARA 0 49 CC(C)(C)c1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217857834 FK In-Stock Unstable F10 0 46 CC(C)(C)c1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217857834 FK In-Stock Unstable TRPV1 18 49 CC(C)(C)c1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217857834 FK In-Stock Unstable ECR 71 43 CC(C)(C)c1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217857834 FK In-Stock Unstable PRNP 45 38 CC(C)(C)c1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217857834 FK In-Stock Unstable PPARD 0 56 CC(C)(C)c1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217857834 FK In-Stock Unstable NR1H4 34 65 CC(C)(C)c1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217857834 FK In-Stock Unstable HDAC1 49 49 CC(C)(C)c1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217857834 FK In-Stock Unstable HDAC2 28 42 CC(C)(C)c1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217857834 FK In-Stock Unstable HDAC3 0 49 CC(C)(C)c1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217857834 FK In-Stock Unstable ABCB1 0 42 CC(C)(C)c1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217857834 FK In-Stock Unstable FABH 0 47 CC(C)(C)c1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217857834 FK In-Stock Unstable MAP3K5 56 42 CC(C)(C)c1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217857834 FK In-Stock Unstable AKR1C3 26 43 CC(C)(C)c1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217857834 FK In-Stock Unstable CYNT 25 41 CC(C)(C)c1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217857834 FK In-Stock Unstable PAGA 0 55 CC(C)(C)c1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217857834 FK In-Stock Unstable E3UJZ5_SPOLI 60 38 CC(C)(C)c1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217857834 FK In-Stock Unstable KCNK3 83 46 Oc1cccc2c1CC[C@@H]2N1CC[C@@H](N2CCCCC2)C1 ZINC000217857870 CF For-Sale Unstable SLC6A1 0 41 Oc1cccc2c1CC[C@@H]2N1CC[C@@H](N2CCCCC2)C1 ZINC000217857870 CF For-Sale Unstable L3MBTL3 91 39 CCc1ccc(-c2nc(CC(=O)NCc3ccccc3S(=O)(=O)N(C)C)cs2)cc1 ZINC000217857916 IG On-Demand Unstable AVPR1B 35 40 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1F ZINC000217857918 FF For-Sale Unstable NPY2R 53 36 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1F ZINC000217857918 FF For-Sale Unstable ADAMTS5 34 40 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1F ZINC000217857918 FF For-Sale Unstable SFRP1 53 31 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1F ZINC000217857918 FF For-Sale Unstable ACKR3 62 32 CC(C)[C@@H]1CN(c2ccc3ccccc3n2)CCN1 ZINC000217857938 CF For-Sale Unstable PRKCD 15 49 CC(C)[C@@H]1CN(c2ccc3ccccc3n2)CCN1 ZINC000217857938 CF For-Sale Unstable PRKCQ 32 49 CCOc1ccc(CCCNC(=O)c2ccc(C(C)(C)C)cc2)cc1 ZINC000217857941 EJ In-Stock Unstable KCNQ1 0 51 CCOc1ccc(CCCNC(=O)c2ccc(C(C)(C)C)cc2)cc1 ZINC000217857941 EJ In-Stock Unstable SCN2A 23 50 CCOc1ccc(CCCNC(=O)c2ccc(C(C)(C)C)cc2)cc1 ZINC000217857941 EJ In-Stock Unstable PLA2G4B 47 36 CCOc1ccc(CCCNC(=O)c2ccc(C(C)(C)C)cc2)cc1 ZINC000217857941 EJ In-Stock Unstable MT-ND1 34 40 CCOc1ccc(CCCNC(=O)c2ccc(C(C)(C)C)cc2)cc1 ZINC000217857941 EJ In-Stock Unstable HDA106 0 42 CCOc1ccc(CCCNC(=O)c2ccc(C(C)(C)C)cc2)cc1 ZINC000217857941 EJ In-Stock Unstable GIPR 20 40 CCOc1ccc(CCCNC(=O)c2ccc(C(C)(C)C)cc2)cc1 ZINC000217857941 EJ In-Stock Unstable CYNT 27 52 CCOc1ccc(CCCNC(=O)c2ccc(C(C)(C)C)cc2)cc1 ZINC000217857941 EJ In-Stock Unstable CRTM 40 36 Oc1cccc2c1CC[C@H]2N1CC[C@@H](N2CCCCC2)C1 ZINC000217857965 CF For-Sale Unstable SLC6A1 0 41 Oc1cccc2c1CC[C@H]2N1CC[C@@H](N2CCCCC2)C1 ZINC000217857965 CF For-Sale Unstable L3MBTL3 91 39 O=C(NCCn1ccnc1-c1ccccn1)c1ccccc1 ZINC000217857985 CE In-Stock Unstable DRD4 40 31 O=C(NCCn1ccnc1-c1ccccn1)c1ccccc1 ZINC000217857985 CE In-Stock Unstable KDM4E 24 42 Cc1nc2ccc(CNC(=O)Cc3ccc(N(C)C)cc3)cc2[nH]1 ZINC000217857986 DF In-Stock Unstable TYMS 83 42 Cc1nc2ccc(CNC(=O)Cc3ccc(N(C)C)cc3)cc2[nH]1 ZINC000217857986 DF In-Stock Unstable NAMPT 49 34 O=C(CSc1nnc(-c2ccccc2Cl)o1)Nc1ccc(N2CCCCC2)nc1 ZINC000217858026 IJ On-Demand Unstable ALOX15 51 35 O=C(CSc1nnc(-c2ccccc2Cl)o1)Nc1ccc(N2CCCCC2)nc1 ZINC000217858026 IJ On-Demand Unstable DGAT1 43 45 O=C(CSc1nnc(-c2ccccc2Cl)o1)Nc1ccc(N2CCCCC2)nc1 ZINC000217858026 IJ On-Demand Unstable CPB 0 42 Cc1c(Cl)cccc1S(=O)(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217858028 FH For-Sale Unstable NPY2R 40 41 C[C@@H](c1ccc(O)cc1)N1CC[C@@H](N2CCCCC2)C1 ZINC000217858031 CG For-Sale Unstable CHRM2 18 44 C[C@@H](c1ccc(O)cc1)N1CC[C@@H](N2CCCCC2)C1 ZINC000217858031 CG For-Sale Unstable L3MBTL3 70 38 C[C@@H](c1ccc(O)cc1)N1CC[C@@H](N2CCCCC2)C1 ZINC000217858031 CG For-Sale Unstable MBTD1 0 48 CC(C)[C@H]1CN(c2ccc3ccccc3n2)CCN1 ZINC000217858032 CF On-Demand Unstable PRKCD 15 49 CC(C)[C@H]1CN(c2ccc3ccccc3n2)CCN1 ZINC000217858032 CF On-Demand Unstable PRKCQ 32 49 CCCOc1ccccc1CCCNC(=O)c1ccc(C(C)(C)C)cc1 ZINC000217858053 FK In-Stock Unstable KCNQ1 0 45 CCCOc1ccccc1CCCNC(=O)c1ccc(C(C)(C)C)cc1 ZINC000217858053 FK In-Stock Unstable TRPV1 0 40 CCCOc1ccccc1CCCNC(=O)c1ccc(C(C)(C)C)cc1 ZINC000217858053 FK In-Stock Unstable PPARD 18 41 CCCOc1ccccc1CCCNC(=O)c1ccc(C(C)(C)C)cc1 ZINC000217858053 FK In-Stock Unstable MTNR1B 43 40 CCCOc1ccccc1CCCNC(=O)c1ccc(C(C)(C)C)cc1 ZINC000217858053 FK In-Stock Unstable CYNT 18 40 CCOc1ccc(C(=O)NCCn2ccnc2-c2ccccn2)cc1 ZINC000217858084 EF In-Stock Unstable DRD4 42 32 CCOc1ccc(C(=O)NCCn2ccnc2-c2ccccn2)cc1 ZINC000217858084 EF In-Stock Unstable DRD3 18 42 CCOc1ccc(C(=O)NCCn2ccnc2-c2ccccn2)cc1 ZINC000217858084 EF In-Stock Unstable PRNP 41 36 CCOc1ccc(C(=O)NCCn2ccnc2-c2ccccn2)cc1 ZINC000217858084 EF In-Stock Unstable SMO 21 40 C[C@H](c1ccc(O)cc1)N1CC[C@@H](N2CCCCC2)C1 ZINC000217858103 CG For-Sale Unstable CHRM2 18 44 C[C@H](c1ccc(O)cc1)N1CC[C@@H](N2CCCCC2)C1 ZINC000217858103 CG For-Sale Unstable L3MBTL3 70 38 C[C@H](c1ccc(O)cc1)N1CC[C@@H](N2CCCCC2)C1 ZINC000217858103 CG For-Sale Unstable MBTD1 0 48 Cc1c(Cl)cccc1S(=O)(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217858119 FH For-Sale Unstable NPY2R 40 41 O=C(C[C@H](c1cc2ccccc2[nH]c1=O)c1c(O)c(O)c(O)c2c(=O)cc(-c3ccccc3)oc12)N1CCOCC1 ZINC000217858120 KH In-Stock Unstable PRKDC 17 41 Cc1ccccc1OC[C@@H](C)NC(=O)c1ccc(C(C)(C)C)cc1 ZINC000217858153 EI In-Stock Unstable ADRB2 0 44 Cc1ccccc1OC[C@@H](C)NC(=O)c1ccc(C(C)(C)C)cc1 ZINC000217858153 EI In-Stock Unstable VDR 54 40 Cc1ccccc1OC[C@@H](C)NC(=O)c1ccc(C(C)(C)C)cc1 ZINC000217858153 EI In-Stock Unstable SDH1 0 44 C[C@@H](c1ccc(F)cc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217858185 CG For-Sale Unstable L3MBTL3 49 33 C[C@@H](c1ccc(F)cc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217858185 CG For-Sale Unstable MBTD1 0 40 O=C(C[C@@H](c1cc2ccccc2[nH]c1=O)c1c(O)c(O)c(O)c2c(=O)cc(-c3ccccc3)oc12)N1CCOCC1 ZINC000217858199 KH In-Stock Unstable PRKDC 17 41 O=C(NCCn1ccnc1-c1ccccn1)c1ccc2c(c1)OCO2 ZINC000217858200 EE In-Stock Unstable DRD4 41 32 O=C(NCCn1ccnc1-c1ccccn1)c1ccc2c(c1)OCO2 ZINC000217858200 EE In-Stock Unstable DRD3 18 40 O=C(NCCn1ccnc1-c1ccccn1)c1ccc2c(c1)OCO2 ZINC000217858200 EE In-Stock Unstable TGFBR1 19 41 O=C(NCCn1ccnc1-c1ccccn1)c1ccc2c(c1)OCO2 ZINC000217858200 EE In-Stock Unstable DYRK2 40 34 Cc1c[nH]c(C(=O)N2CC[C@@H](c3ccc(F)cc3)C2)n1 ZINC000217858226 CE In-Stock Unstable HSD11B1 28 44 Cc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1Cl ZINC000217858227 FH For-Sale Unstable ADAMTS5 37 43 Cc1ccccc1OC[C@H](C)NC(=O)c1ccc(C(C)(C)C)cc1 ZINC000217858235 EI In-Stock Unstable ADRB2 0 44 Cc1ccccc1OC[C@H](C)NC(=O)c1ccc(C(C)(C)C)cc1 ZINC000217858235 EI In-Stock Unstable VDR 54 40 Cc1ccccc1OC[C@H](C)NC(=O)c1ccc(C(C)(C)C)cc1 ZINC000217858235 EI In-Stock Unstable SDH1 0 44 O=C(NC[C@@H](O)C(F)(F)F)c1cccc(Cl)c1F ZINC000217858257 CE On-Demand Unstable E3UJZ5_SPOLI 43 37 C[C@H](c1ccc(F)cc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217858268 CG For-Sale Unstable L3MBTL3 49 33 C[C@H](c1ccc(F)cc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217858268 CG For-Sale Unstable MBTD1 0 40 Cc1ccc(NCCN2CCC[C@@H]3CCCC[C@H]32)cc1 ZINC000217858279 CI For-Sale Unstable HRH3 0 44 Cc1c[nH]c(C(=O)N2CC[C@H](c3ccc(F)cc3)C2)n1 ZINC000217858282 CE In-Stock Unstable HSD11B1 28 44 Cc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1Cl ZINC000217858289 FH For-Sale Unstable ADAMTS5 37 43 CCNc1nc(Cl)nc(NCC#N)n1 ZINC000217858301 BC For-Sale Unstable PETD 0 73 CCNc1nc(Cl)nc(NCC#N)n1 ZINC000217858301 BC For-Sale Unstable Q31945_CHEAL 0 58 CCNc1nc(Cl)nc(NCC#N)n1 ZINC000217858301 BC For-Sale Unstable PPX1 0 73 O=C(NCCn1ccnc1-c1ccccn1)c1ccccc1Cl ZINC000217858303 EG In-Stock Unstable HTR2A 15 48 O=C(NCCn1ccnc1-c1ccccn1)c1ccccc1Cl ZINC000217858303 EG In-Stock Unstable DRD3 18 43 O=C(NCCn1ccnc1-c1ccccn1)c1ccccc1Cl ZINC000217858303 EG In-Stock Unstable SHH 19 45 Cc1cccc(=O)n1Cc1ccc(F)c(/C=C\C(=O)O)c1 ZINC000217858313 CE For-Sale Unstable PTGER3 40 35 Cc1cccc(=O)n1Cc1ccc(F)c(/C=C\C(=O)O)c1 ZINC000217858313 CE For-Sale Unstable PTGES2 62 33 O=C(NC[C@H](O)C(F)(F)F)c1cccc(Cl)c1F ZINC000217858314 CE On-Demand Unstable E3UJZ5_SPOLI 43 37 Cc1ccc(OC[C@@H](C)NC(=O)c2ccc(C(C)(C)C)cc2)cc1 ZINC000217858336 EI In-Stock Unstable SDH1 0 44 Cc1ccc(OC[C@@H](C)NC(=O)c2ccc(C(C)(C)C)cc2)cc1 ZINC000217858336 EI In-Stock Unstable MAP3K5 40 37 Cc1ccc(OC[C@@H](C)NC(=O)c2ccc(C(C)(C)C)cc2)cc1 ZINC000217858336 EI In-Stock Unstable UTS2 26 40 Cc1ccc(OC[C@@H](C)NC(=O)c2ccc(C(C)(C)C)cc2)cc1 ZINC000217858336 EI In-Stock Unstable GPR88 0 40 Cc1ccc(NCCN2CCC[C@H]3CCCC[C@H]32)cc1 ZINC000217858365 CI For-Sale Unstable HRH3 0 44 C[C@@H](Cc1ccc(O)cc1)N1CC[C@@H](N2CCCCC2)C1 ZINC000217858378 CF For-Sale Unstable L3MBTL3 80 36 Cc1ccc(Cl)cc1S(=O)(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217858386 FH For-Sale Unstable ADAMTS5 35 40 Cc1ccc(OC[C@H](C)NC(=O)c2ccc(C(C)(C)C)cc2)cc1 ZINC000217858396 EI In-Stock Unstable SDH1 0 44 Cc1ccc(OC[C@H](C)NC(=O)c2ccc(C(C)(C)C)cc2)cc1 ZINC000217858396 EI In-Stock Unstable MAP3K5 40 37 Cc1ccc(OC[C@H](C)NC(=O)c2ccc(C(C)(C)C)cc2)cc1 ZINC000217858396 EI In-Stock Unstable UTS2 26 40 Cc1ccc(OC[C@H](C)NC(=O)c2ccc(C(C)(C)C)cc2)cc1 ZINC000217858396 EI In-Stock Unstable GPR88 0 40 CC(=O)Nc1cccc(NC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217858454 FI For-Sale Unstable KCNK3 108 39 CC(=O)Nc1cccc(NC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217858454 FI For-Sale Unstable KCNK9 70 39 Cc1ccc(Cl)cc1S(=O)(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217858461 FH For-Sale Unstable ADAMTS5 35 40 C[C@H](Cc1ccc(O)cc1)N1CC[C@@H](N2CCCCC2)C1 ZINC000217858478 CF For-Sale Unstable L3MBTL3 80 36 CC1CCN(c2ccc([C@@H](C)NC(=O)c3ccc(C(C)(C)C)cc3)cc2)CC1 ZINC000217858481 GK In-Stock Unstable PRNP 46 38 O=C(NCCn1ccnc1-c1ccccn1)c1c(F)cccc1Cl ZINC000217858519 EG In-Stock Unstable HTR2A 15 45 O=C(NCCn1ccnc1-c1ccccn1)c1c(F)cccc1Cl ZINC000217858519 EG In-Stock Unstable DRD3 17 42 CCC[C@@H](O)CNCCCn1ccnc1 ZINC000217858536 BD For-Sale Unstable TBXAS1 33 50 CCC[C@@H](O)CNCCCn1ccnc1 ZINC000217858536 BD For-Sale Unstable HMOX2 44 32 CCC[C@@H](O)CNCCCn1ccnc1 ZINC000217858536 BD For-Sale Unstable CAMC 0 40 CCC[C@@H](O)CNCCCn1ccnc1 ZINC000217858536 BD For-Sale Unstable QPCT 44 39 CC[C@@H](c1ccccc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217858544 CG For-Sale Unstable L3MBTL3 93 39 CC1CCN(c2ccc([C@H](C)NC(=O)c3ccc(C(C)(C)C)cc3)cc2)CC1 ZINC000217858547 GK In-Stock Unstable PRNP 46 38 CCc1nccn1Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217858576 CF For-Sale Unstable PTGER2 29 42 CCc1nccn1Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217858576 CF For-Sale Unstable PTGER4 0 42 CCc1nccn1Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217858576 CF For-Sale Unstable PTGER3 16 43 CCC[C@H](O)CNCCCn1ccnc1 ZINC000217858618 BD For-Sale Unstable TBXAS1 33 50 CCC[C@H](O)CNCCCn1ccnc1 ZINC000217858618 BD For-Sale Unstable HMOX2 44 32 CCC[C@H](O)CNCCCn1ccnc1 ZINC000217858618 BD For-Sale Unstable CAMC 0 40 CCC[C@H](O)CNCCCn1ccnc1 ZINC000217858618 BD For-Sale Unstable QPCT 44 39 CC[C@H](c1ccccc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217858620 CG For-Sale Unstable L3MBTL3 93 39 O=C(NCCn1ccnc1-c1ccccn1)c1ccccc1C(F)(F)F ZINC000217858645 FG In-Stock Unstable P2RX7 34 43 COCCn1c([C@H](C)NC(=O)COc2ccc3c(C)cc(=O)oc3c2)nc2ccccc21 ZINC000217858651 IG In-Stock Unstable MAOA 60 51 COCCn1c([C@H](C)NC(=O)COc2ccc3c(C)cc(=O)oc3c2)nc2ccccc21 ZINC000217858651 IG In-Stock Unstable ACHE 19 46 COCCn1c([C@H](C)NC(=O)COc2ccc3c(C)cc(=O)oc3c2)nc2ccccc21 ZINC000217858651 IG In-Stock Unstable MAOB 42 51 COCCn1c([C@H](C)NC(=O)COc2ccc3c(C)cc(=O)oc3c2)nc2ccccc21 ZINC000217858651 IG In-Stock Unstable BCHE 24 46 C[C@@H](c1cc(Br)ccc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217858718 FH For-Sale Unstable L3MBTL1 0 40 C[C@@H](c1cc(Br)ccc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217858718 FH For-Sale Unstable L3MBTL3 58 38 C[C@@H](c1cc(Br)ccc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217858718 FH For-Sale Unstable MBTD1 0 51 O=C(NC1CCN(C(=O)N2CCOCC2)CC1)[C@@H]1C[C@H]1c1ccccc1 ZINC000217858734 FD In-Stock Unstable EPHX2 35 45 O=C(NC1CCN(C(=O)N2CCOCC2)CC1)[C@@H]1C[C@H]1c1ccccc1 ZINC000217858734 FD In-Stock Unstable AKR1C3 32 46 Cc1cc(C)cc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217858746 CH For-Sale Unstable PTGER2 30 53 Cc1cc(C)cc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217858746 CH For-Sale Unstable PTGER4 45 48 Cc1cc(C)cc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217858746 CH For-Sale Unstable PTGER3 37 55 Cc1cc(C)cc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217858746 CH For-Sale Unstable PTGDR 0 55 Cc1cc(C)cc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217858746 CH For-Sale Unstable FFAR1 20 40 O=C(/C=C/c1ccccc1)NCCn1ccnc1-c1ccccn1 ZINC000217858748 DF In-Stock Unstable HDAC8 45 35 O=C(/C=C/c1ccccc1)NCCn1ccnc1-c1ccccn1 ZINC000217858748 DF In-Stock Unstable HDAC6 37 40 COC(=O)C[C@H](c1ccc(OC)c(O)c1)c1c(O)c2ccccc2oc1=O ZINC000217858750 FF In-Stock Unstable RORC 41 33 COc1cc(C(=O)NC[C@@H](O)C(F)(F)F)ccc1F ZINC000217858767 CD On-Demand Unstable CYSLTR1 44 35 COc1cc(C(=O)NC[C@@H](O)C(F)(F)F)ccc1F ZINC000217858767 CD On-Demand Unstable PPARD 24 40 O=S(=O)(Cc1cccc(Cl)c1)NC[C@H]1CCCN1c1ccccc1 ZINC000217858777 FG For-Sale Unstable HTR1A 15 40 C[C@H](c1cc(Br)ccc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217858802 FH For-Sale Unstable L3MBTL1 0 40 C[C@H](c1cc(Br)ccc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217858802 FH For-Sale Unstable L3MBTL3 58 38 C[C@H](c1cc(Br)ccc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217858802 FH For-Sale Unstable MBTD1 0 51 COc1cc(C(=O)NC[C@H](O)C(F)(F)F)ccc1F ZINC000217858836 CD On-Demand Unstable CYSLTR1 44 35 COc1cc(C(=O)NC[C@H](O)C(F)(F)F)ccc1F ZINC000217858836 CD On-Demand Unstable PPARD 24 40 COC(=O)C[C@@H](c1ccc(OC)c(O)c1)c1c(O)c2ccccc2oc1=O ZINC000217858841 FF In-Stock Unstable RORC 41 33 Cc1cc(C)cc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217858843 CH For-Sale Unstable PTGER2 22 45 Cc1cc(C)cc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217858843 CH For-Sale Unstable PTGER4 35 44 Cc1cc(C)cc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217858843 CH For-Sale Unstable PTGER3 32 45 Cc1cc(C)cc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217858843 CH For-Sale Unstable PTGDR 0 45 Cc1cc(C)cc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217858843 CH For-Sale Unstable FFAR1 35 41 Cc1cc(C)cc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217858843 CH For-Sale Unstable AKR1C3 35 50 Cc1cc(C)cc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217858843 CH For-Sale Unstable AKR1B10 19 40 O=S(=O)(Cc1cccc(Cl)c1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217858847 FG For-Sale Unstable HTR1A 15 40 O=C(COc1ccc(Cl)cc1Cl)NCCn1ccnc1-c1ccccn1 ZINC000217858861 GG In-Stock Unstable MCHR2 21 40 C[C@@H](c1ccccc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217858892 CG For-Sale Unstable L3MBTL1 0 41 C[C@@H](c1ccccc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217858892 CG For-Sale Unstable L3MBTL3 94 41 C[C@@H](c1ccccc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217858892 CG For-Sale Unstable MBTD1 0 44 C[C@@H](c1ccccc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217858892 CG For-Sale Unstable TP53BP1 0 41 Cc1cc(C)cc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217858910 CH For-Sale Unstable MAOB 50 45 Cc1cc(C)cc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217858910 CH For-Sale Unstable PTGER2 26 54 Cc1cc(C)cc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217858910 CH For-Sale Unstable PTGER4 40 48 Cc1cc(C)cc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217858910 CH For-Sale Unstable PTGER3 40 48 Cc1cc(C)cc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217858910 CH For-Sale Unstable LTB4R 21 46 Cc1cc(C)cc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217858910 CH For-Sale Unstable NR1H4 43 35 Cc1cc(C)cc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217858910 CH For-Sale Unstable HCAR2 0 40 Cc1cc(C)cc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217858910 CH For-Sale Unstable FFAR1 76 47 Cc1cc(C)cc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217858910 CH For-Sale Unstable AKR1C3 40 48 Cc1cccc(C)c1NC(=O)[C@H](C)Sc1nnc(N2C[C@H](C)C[C@@H](C)C2)n1Cc1ccco1 ZINC000217858922 JK On-Demand Unstable HCRTR2 20 40 O=C(O)CC[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217858926 CC For-Sale Unstable CTSC 21 41 O=C(O)CC[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217858926 CC For-Sale Unstable MAN1B1 52 33 Cc1cc(Cl)cc(C(=O)NC[C@@H](O)C(F)(F)F)c1 ZINC000217858932 CE On-Demand Unstable CACNA1I 50 36 C[C@H](c1ccccc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217858950 CG For-Sale Unstable L3MBTL1 0 41 C[C@H](c1ccccc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217858950 CG For-Sale Unstable L3MBTL3 94 41 C[C@H](c1ccccc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217858950 CG For-Sale Unstable MBTD1 0 44 C[C@H](c1ccccc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217858950 CG For-Sale Unstable TP53BP1 0 41 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc(F)c(Cl)c1 ZINC000217858968 FG For-Sale Unstable HTR7 19 41 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc(F)c(Cl)c1 ZINC000217858968 FG For-Sale Unstable HTR6 17 41 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc(F)c(Cl)c1 ZINC000217858968 FG For-Sale Unstable ADAMTS5 37 41 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc(F)c(Cl)c1 ZINC000217858968 FG For-Sale Unstable SFRP1 65 34 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc(F)c(Cl)c1 ZINC000217858968 FG For-Sale Unstable WNT3 44 31 Cc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217858990 CH For-Sale Unstable ALOX5 22 45 Cc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217858990 CH For-Sale Unstable MAOA 16 41 Cc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217858990 CH For-Sale Unstable MAOB 68 50 Cc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217858990 CH For-Sale Unstable PTGER2 28 54 Cc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217858990 CH For-Sale Unstable CYSLTR1 15 41 Cc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217858990 CH For-Sale Unstable PTGER4 41 54 Cc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217858990 CH For-Sale Unstable PTGER3 37 54 Cc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217858990 CH For-Sale Unstable DRTS_LEIMA 30 41 Cc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217858990 CH For-Sale Unstable LTB4R 21 46 Cc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217858990 CH For-Sale Unstable KCNA3 0 40 Cc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217858990 CH For-Sale Unstable NR1H4 53 36 Cc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217858990 CH For-Sale Unstable PTGDR 0 46 Cc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217858990 CH For-Sale Unstable HCAR2 0 40 Cc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217858990 CH For-Sale Unstable FFAR1 83 53 Cc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217858990 CH For-Sale Unstable AKR1C3 41 51 Cc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217858990 CH For-Sale Unstable FFAR4 16 40 Cc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217858990 CH For-Sale Unstable PDS 48 43 Cc1cc(Cl)cc(C(=O)NC[C@H](O)C(F)(F)F)c1 ZINC000217859007 CE On-Demand Unstable CACNA1I 50 36 O=C(O)CC[C@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217859015 CC For-Sale Unstable CTSC 21 41 O=C(O)CC[C@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217859015 CC For-Sale Unstable MAN1B1 52 33 Cc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1ccc(C(C)(C)C)cc1 ZINC000217859021 FK In-Stock Unstable KCNK3 15 42 CSC[C@@](C)(O)CNCc1ccc(O)c(Cl)c1 ZINC000217859022 CE For-Sale Unstable NCE103 27 45 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc(F)c(Cl)c1 ZINC000217859046 FG For-Sale Unstable HTR7 19 41 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc(F)c(Cl)c1 ZINC000217859046 FG For-Sale Unstable HTR6 17 41 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc(F)c(Cl)c1 ZINC000217859046 FG For-Sale Unstable ADAMTS5 37 41 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc(F)c(Cl)c1 ZINC000217859046 FG For-Sale Unstable SFRP1 65 34 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc(F)c(Cl)c1 ZINC000217859046 FG For-Sale Unstable WNT3 44 31 CSc1ccc(C(=O)O[C@H]2C[C@H]3CC[C@@]2(C)C3(C)C)cc1 ZINC000217859048 DJ For-Sale Unstable ELANE 0 47 C[C@@H](c1cc(F)ccc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217859061 CG For-Sale Unstable L3MBTL3 64 38 C[C@@H](c1cc(F)ccc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217859061 CG For-Sale Unstable MBTD1 0 40 Cc1cccc(OCc2ccc(F)cc2/C=C\C(=O)O)c1 ZINC000217859069 CH For-Sale Unstable PTGER2 60 47 Cc1cccc(OCc2ccc(F)cc2/C=C\C(=O)O)c1 ZINC000217859069 CH For-Sale Unstable PTGER4 39 47 Cc1cccc(OCc2ccc(F)cc2/C=C\C(=O)O)c1 ZINC000217859069 CH For-Sale Unstable PTGER3 31 47 Cc1cccc(OCc2ccc(F)cc2/C=C\C(=O)O)c1 ZINC000217859069 CH For-Sale Unstable PTGDR 0 43 C[C@@H]1C[C@@H](C)CN(c2nnc(SCC(=O)c3cccc([N+](=O)[O-])c3)n2Cc2ccco2)C1 ZINC000217859080 JI On-Demand Unstable HCRTR2 20 41 CSC[C@](C)(O)CNCc1ccc(O)c(Cl)c1 ZINC000217859109 CE For-Sale Unstable NCE103 27 45 Cc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1ccc(C(C)(C)C)cc1 ZINC000217859131 FK In-Stock Unstable KCNK3 15 42 C[C@H](c1cc(F)ccc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217859133 CG For-Sale Unstable L3MBTL3 64 38 C[C@H](c1cc(F)ccc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217859133 CG For-Sale Unstable MBTD1 0 40 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc2c(c1)CCCC2 ZINC000217859147 FH For-Sale Unstable NPY1R 50 41 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc2c(c1)CCCC2 ZINC000217859147 FH For-Sale Unstable NPY2R 57 41 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc2c(c1)CCCC2 ZINC000217859147 FH For-Sale Unstable ADAMTS5 32 41 Cc1cccc(OCc2ccc(F)c(/C=C\C(=O)O)c2)c1 ZINC000217859148 CH For-Sale Unstable MAOB 41 40 Cc1cccc(OCc2ccc(F)c(/C=C\C(=O)O)c2)c1 ZINC000217859148 CH For-Sale Unstable PTGER2 23 46 Cc1cccc(OCc2ccc(F)c(/C=C\C(=O)O)c2)c1 ZINC000217859148 CH For-Sale Unstable PTGER4 41 52 Cc1cccc(OCc2ccc(F)c(/C=C\C(=O)O)c2)c1 ZINC000217859148 CH For-Sale Unstable PTGER3 52 39 Cc1cccc(OCc2ccc(F)c(/C=C\C(=O)O)c2)c1 ZINC000217859148 CH For-Sale Unstable GYS1 51 34 Cc1cccc(OCc2ccc(F)c(/C=C\C(=O)O)c2)c1 ZINC000217859148 CH For-Sale Unstable PTGDR 0 47 Cc1cccc(OCc2ccc(F)c(/C=C\C(=O)O)c2)c1 ZINC000217859148 CH For-Sale Unstable FFAR1 78 48 Cc1cccc(OCc2ccc(F)c(/C=C\C(=O)O)c2)c1 ZINC000217859148 CH For-Sale Unstable AKR1C3 32 41 Cc1ccccc1OCC(=O)NCCn1ccnc1-c1ccccn1 ZINC000217859157 EE In-Stock Unstable CYSP_TRYCR 0 48 C[C@H]1C[C@@H](C)CN(c2nnc(SCC(=O)c3cccc([N+](=O)[O-])c3)n2Cc2ccco2)C1 ZINC000217859173 JI On-Demand Unstable HCRTR2 20 41 NS(=O)(=O)c1ccc(CCNC(=S)Nc2ccc(I)cc2)cc1 ZINC000217859194 JE For-Sale Unstable CA2 156 87 NS(=O)(=O)c1ccc(CCNC(=S)Nc2ccc(I)cc2)cc1 ZINC000217859194 JE For-Sale Unstable ADRB2 15 51 NS(=O)(=O)c1ccc(CCNC(=S)Nc2ccc(I)cc2)cc1 ZINC000217859194 JE For-Sale Unstable ADRB1 18 51 NS(=O)(=O)c1ccc(CCNC(=S)Nc2ccc(I)cc2)cc1 ZINC000217859194 JE For-Sale Unstable ADRB3 20 51 NS(=O)(=O)c1ccc(CCNC(=S)Nc2ccc(I)cc2)cc1 ZINC000217859194 JE For-Sale Unstable CA6 29 44 NS(=O)(=O)c1ccc(CCNC(=S)Nc2ccc(I)cc2)cc1 ZINC000217859194 JE For-Sale Unstable CA1 144 87 NS(=O)(=O)c1ccc(CCNC(=S)Nc2ccc(I)cc2)cc1 ZINC000217859194 JE For-Sale Unstable CA7 73 52 NS(=O)(=O)c1ccc(CCNC(=S)Nc2ccc(I)cc2)cc1 ZINC000217859194 JE For-Sale Unstable CA13 27 44 NS(=O)(=O)c1ccc(CCNC(=S)Nc2ccc(I)cc2)cc1 ZINC000217859194 JE For-Sale Unstable CA5B 58 50 NS(=O)(=O)c1ccc(CCNC(=S)Nc2ccc(I)cc2)cc1 ZINC000217859194 JE For-Sale Unstable CA4 108 76 NS(=O)(=O)c1ccc(CCNC(=S)Nc2ccc(I)cc2)cc1 ZINC000217859194 JE For-Sale Unstable CA5A 60 50 NS(=O)(=O)c1ccc(CCNC(=S)Nc2ccc(I)cc2)cc1 ZINC000217859194 JE For-Sale Unstable CA14 72 49 NS(=O)(=O)c1ccc(CCNC(=S)Nc2ccc(I)cc2)cc1 ZINC000217859194 JE For-Sale Unstable CA12 110 87 NS(=O)(=O)c1ccc(CCNC(=S)Nc2ccc(I)cc2)cc1 ZINC000217859194 JE For-Sale Unstable CA9 124 87 NS(=O)(=O)c1ccc(CCNC(=S)Nc2ccc(I)cc2)cc1 ZINC000217859194 JE For-Sale Unstable CAH_METTE 29 43 NS(=O)(=O)c1ccc(CCNC(=S)Nc2ccc(I)cc2)cc1 ZINC000217859194 JE For-Sale Unstable UREA_CANEN 30 44 NS(=O)(=O)c1ccc(CCNC(=S)Nc2ccc(I)cc2)cc1 ZINC000217859194 JE For-Sale Unstable CYNT 52 47 NS(=O)(=O)c1ccc(CCNC(=S)Nc2ccc(I)cc2)cc1 ZINC000217859194 JE For-Sale Unstable NCE103 64 61 NS(=O)(=O)c1ccc(CCNC(=S)Nc2ccc(I)cc2)cc1 ZINC000217859194 JE For-Sale Unstable ALPI 16 50 NS(=O)(=O)c1ccc(CCNC(=S)Nc2ccc(I)cc2)cc1 ZINC000217859194 JE For-Sale Unstable CA15 20 44 NS(=O)(=O)c1ccc(CCNC(=S)Nc2ccc(I)cc2)cc1 ZINC000217859194 JE For-Sale Unstable MTCA1 61 61 NS(=O)(=O)c1ccc(CCNC(=S)Nc2ccc(I)cc2)cc1 ZINC000217859194 JE For-Sale Unstable P96878_MYCTU 77 61 NS(=O)(=O)c1ccc(CCNC(=S)Nc2ccc(I)cc2)cc1 ZINC000217859194 JE For-Sale Unstable A6YCJ1_9METZ 34 53 CCOC(=O)c1sc(NC(=O)CCCNc2ccc3c(cc2=O)[C@@H](NC(C)=O)CCc2cc(OC)c(OC)c(OC)c2-3)nc1C ZINC000217859203 KJ In-Stock Unstable TUBA1A 15 57 Cc1ccc(O)c([C@@H](C)N2CC[C@@H](N3CCCCC3)C2)c1 ZINC000217859210 CG For-Sale Unstable L3MBTL3 65 39 Cc1ccc(O)c([C@@H](C)N2CC[C@@H](N3CCCCC3)C2)c1 ZINC000217859210 CG For-Sale Unstable MBTD1 0 41 Cc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217859214 CH For-Sale Unstable ALOX5 17 48 Cc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217859214 CH For-Sale Unstable MAOB 23 40 Cc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217859214 CH For-Sale Unstable PTGER2 32 62 Cc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217859214 CH For-Sale Unstable PPIA 42 34 Cc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217859214 CH For-Sale Unstable PTGER1 49 42 Cc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217859214 CH For-Sale Unstable PTGER4 47 48 Cc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217859214 CH For-Sale Unstable PTGER3 35 52 Cc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217859214 CH For-Sale Unstable LTB4R 27 48 Cc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217859214 CH For-Sale Unstable PTGDR 0 43 Cc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217859214 CH For-Sale Unstable FFAR1 53 46 Cc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217859214 CH For-Sale Unstable AKR1C3 42 55 CC1(C)[C@H]2CC[C@@]1(C)[C@@H](OC(=O)CCc1cccs1)C2 ZINC000217859215 CI For-Sale Unstable ELANE 0 43 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc2c(c1)CCCC2 ZINC000217859221 FH For-Sale Unstable NPY1R 50 41 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc2c(c1)CCCC2 ZINC000217859221 FH For-Sale Unstable NPY2R 57 41 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc2c(c1)CCCC2 ZINC000217859221 FH For-Sale Unstable ADAMTS5 32 41 COc1ccc2c(c1)[C@@H](NC(=O)c1ccc(C(C)(C)C)cc1)CC(C)(C)O2 ZINC000217859252 FK In-Stock Unstable MT-ND1 31 42 COc1ccc2c(c1)[C@@H](NC(=O)c1ccc(C(C)(C)C)cc1)CC(C)(C)O2 ZINC000217859252 FK In-Stock Unstable NAAA 22 44 C[C@H]1C[C@H](C)CN(c2nnc(SCC(=O)c3cccc([N+](=O)[O-])c3)n2Cc2ccco2)C1 ZINC000217859283 JI On-Demand Unstable HCRTR2 20 41 Cc1ccc(O)c([C@H](C)N2CC[C@@H](N3CCCCC3)C2)c1 ZINC000217859304 CG For-Sale Unstable L3MBTL3 65 39 Cc1ccc(O)c([C@H](C)N2CC[C@@H](N3CCCCC3)C2)c1 ZINC000217859304 CG For-Sale Unstable MBTD1 0 41 COc1ccc2c(c1)[C@H](NC(=O)c1ccc(C(C)(C)C)cc1)CC(C)(C)O2 ZINC000217859311 FK In-Stock Unstable MT-ND1 31 42 COc1ccc2c(c1)[C@H](NC(=O)c1ccc(C(C)(C)C)cc1)CC(C)(C)O2 ZINC000217859311 FK In-Stock Unstable NAAA 22 44 Cc1ccccc1OCc1ccc(F)cc1/C=C\C(=O)O ZINC000217859322 CH For-Sale Unstable PTGER2 25 47 Cc1ccccc1OCc1ccc(F)cc1/C=C\C(=O)O ZINC000217859322 CH For-Sale Unstable PTGER4 38 46 Cc1ccccc1OCc1ccc(F)cc1/C=C\C(=O)O ZINC000217859322 CH For-Sale Unstable PTGER3 31 50 Cc1ccccc1OCc1ccc(F)cc1/C=C\C(=O)O ZINC000217859322 CH For-Sale Unstable PTGDR 0 41 Cc1ccccc1OCc1ccc(F)cc1/C=C\C(=O)O ZINC000217859322 CH For-Sale Unstable AKR1C3 31 41 CC(C)(C)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217859337 FH For-Sale Unstable NPY1R 40 33 CC(C)(C)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217859337 FH For-Sale Unstable NPY2R 42 37 CC(C)(C)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217859337 FH For-Sale Unstable ADAMTS5 38 51 CC(C)[C@H](NC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)C(=O)NCCc1ccco1 ZINC000217859343 ID In-Stock Unstable CHRNA4 26 42 Oc1ccc2c(c1)OC[C@@H]2N1CC[C@@H](N2CCCCC2)C1 ZINC000217859394 CE For-Sale Unstable L3MBTL3 55 35 CC(C)(C)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217859404 FH For-Sale Unstable NPY1R 40 33 CC(C)(C)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217859404 FH For-Sale Unstable NPY2R 42 37 CC(C)(C)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217859404 FH For-Sale Unstable ADAMTS5 38 51 Cc1ccccc1OCc1ccc(F)c(/C=C\C(=O)O)c1 ZINC000217859424 CH For-Sale Unstable PTGER2 26 48 Cc1ccccc1OCc1ccc(F)c(/C=C\C(=O)O)c1 ZINC000217859424 CH For-Sale Unstable PTGER1 65 40 Cc1ccccc1OCc1ccc(F)c(/C=C\C(=O)O)c1 ZINC000217859424 CH For-Sale Unstable PTGER4 50 47 Cc1ccccc1OCc1ccc(F)c(/C=C\C(=O)O)c1 ZINC000217859424 CH For-Sale Unstable PTGER3 42 51 Cc1ccccc1OCc1ccc(F)c(/C=C\C(=O)O)c1 ZINC000217859424 CH For-Sale Unstable PTGDR 0 45 Cc1ccccc1OCc1ccc(F)c(/C=C\C(=O)O)c1 ZINC000217859424 CH For-Sale Unstable FFAR1 37 41 Cc1ccccc1OCc1ccc(F)c(/C=C\C(=O)O)c1 ZINC000217859424 CH For-Sale Unstable AKR1C3 33 44 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1ccc(C(C)(C)C)cc1 ZINC000217859429 FK In-Stock Unstable MT-ND1 31 42 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1ccc(C(C)(C)C)cc1 ZINC000217859429 FK In-Stock Unstable NAAA 22 44 CCNc1c(O)cccc1[N+](=O)[O-] ZINC000217859432 AD For-Sale Unstable COLA 64 37 CCNc1c(O)cccc1[N+](=O)[O-] ZINC000217859432 AD For-Sale Unstable PQSD 0 41 O=C(O)CN(C(=O)[C@@H]1C[C@@H]2CCCC[C@@H]2N1)C1CC1 ZINC000217859447 CC For-Sale Unstable ACE 49 35 CC[C@H](Sc1nnc(N2C[C@H](C)C[C@@H](C)C2)n1Cc1ccco1)C(=O)NCc1ccccc1 ZINC000217859465 JJ On-Demand Unstable HCRTR2 0 42 Oc1ccc2c(c1)OC[C@H]2N1CC[C@@H](N2CCCCC2)C1 ZINC000217859478 CE For-Sale Unstable L3MBTL3 55 35 O=C(O)CN(C(=O)[C@@H]1C[C@H]2CCCC[C@@H]2N1)C1CC1 ZINC000217859497 CC For-Sale Unstable ACE 49 35 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1ccc(C(C)(C)C)cc1 ZINC000217859518 FK In-Stock Unstable MT-ND1 31 42 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1ccc(C(C)(C)C)cc1 ZINC000217859518 FK In-Stock Unstable NAAA 22 44 CCC[C@@H](O)CNCCc1ccsc1 ZINC000217859537 BE For-Sale Unstable ADRB2 16 40 CCC[C@@H](O)CNCCc1ccsc1 ZINC000217859537 BE For-Sale Unstable ADRB1 23 43 CCC[C@@H](O)CNCCc1ccsc1 ZINC000217859537 BE For-Sale Unstable ADRB3 26 43 CCN1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217859539 CD For-Sale Unstable DRD2 19 40 CCN1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217859539 CD For-Sale Unstable ACHE 19 40 CCN1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217859539 CD For-Sale Unstable CHRM3 18 44 CCN1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217859539 CD For-Sale Unstable SIGMAR1 44 48 CCN1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217859539 CD For-Sale Unstable HDAC8 43 39 CCN1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217859539 CD For-Sale Unstable HDAC1 18 43 CCN1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217859539 CD For-Sale Unstable FAAH 17 40 CCN1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217859539 CD For-Sale Unstable MCHR2 41 32 CCN1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217859539 CD For-Sale Unstable AKR1C3 33 42 CC[C@@H](c1ccc(O)cc1)N1CC[C@@H](N2CCCCC2)C1 ZINC000217859555 CG For-Sale Unstable L3MBTL3 62 35 CC[C@H](C(=O)NCCn1ccnc1-c1ccccn1)c1ccccc1 ZINC000217859577 EG In-Stock Unstable KCNQ2 40 38 CC[C@@H](NC(=O)c1ccc(C(C)(C)C)cc1)c1ccc(C)c(C)c1 ZINC000217859618 DK In-Stock Unstable TRPV1 16 41 CC[C@@H](NC(=O)c1ccc(C(C)(C)C)cc1)c1ccc(C)c(C)c1 ZINC000217859618 DK In-Stock Unstable UTS2 64 38 CCC[C@H](O)CNCCc1ccsc1 ZINC000217859637 BE For-Sale Unstable ADRB2 16 40 CCC[C@H](O)CNCCc1ccsc1 ZINC000217859637 BE For-Sale Unstable ADRB1 23 43 CCC[C@H](O)CNCCc1ccsc1 ZINC000217859637 BE For-Sale Unstable ADRB3 26 43 CC[C@H](c1ccc(O)cc1)N1CC[C@@H](N2CCCCC2)C1 ZINC000217859644 CG For-Sale Unstable L3MBTL3 62 35 CSC[C@@](C)(O)CNCc1ccccc1OC(F)F ZINC000217859650 CE On-Demand Unstable PHES 0 45 O=C(CSc1nnc(N2CCCC2)n1Cc1ccco1)c1cccc([N+](=O)[O-])c1 ZINC000217859653 HG On-Demand Unstable HCRTR2 20 42 CC[C@@H](C(=O)NCCn1ccnc1-c1ccccn1)c1ccccc1 ZINC000217859680 EG In-Stock Unstable KCNQ2 40 38 C[C@@H](c1cc(Cl)ccc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217859700 DH For-Sale Unstable L3MBTL3 64 38 C[C@@H](c1cc(Cl)ccc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217859700 DH For-Sale Unstable MBTD1 0 40 CC[C@H](NC(=O)c1ccc(C(C)(C)C)cc1)c1ccc(C)c(C)c1 ZINC000217859708 DK In-Stock Unstable TRPV1 16 41 CC[C@H](NC(=O)c1ccc(C(C)(C)C)cc1)c1ccc(C)c(C)c1 ZINC000217859708 DK In-Stock Unstable UTS2 64 38 CSC[C@](C)(O)CNCc1ccccc1OC(F)F ZINC000217859711 CE On-Demand Unstable PHES 0 45 COc1cccc(-c2ccc(C(=O)NCC3(C)COC3)cc2)c1 ZINC000217859722 DG In-Stock Unstable DRD4 48 38 COc1cccc(-c2ccc(C(=O)NCC3(C)COC3)cc2)c1 ZINC000217859722 DG In-Stock Unstable DHODH 24 45 COc1cccc(-c2ccc(C(=O)NCC3(C)COC3)cc2)c1 ZINC000217859722 DG In-Stock Unstable MTNR1A 43 36 COc1cccc(-c2ccc(C(=O)NCC3(C)COC3)cc2)c1 ZINC000217859722 DG In-Stock Unstable ROCK2 41 36 COc1cccc(-c2ccc(C(=O)NCC3(C)COC3)cc2)c1 ZINC000217859722 DG In-Stock Unstable HSD17B2 22 48 COc1cccc(-c2ccc(C(=O)NCC3(C)COC3)cc2)c1 ZINC000217859722 DG In-Stock Unstable FIMH 30 40 CC(=O)Nc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217859754 FF For-Sale Unstable CA2 15 42 CC(=O)Nc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217859754 FF For-Sale Unstable CA1 18 41 CC(=O)Nc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217859754 FF For-Sale Unstable NPY2R 17 43 CC(=O)Nc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217859754 FF For-Sale Unstable TGM2 27 43 CC(=O)Nc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217859754 FF For-Sale Unstable ADAMTS5 39 41 CC(=O)Nc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217859754 FF For-Sale Unstable F13A1 48 43 CC(=O)Nc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217859754 FF For-Sale Unstable IDO1 32 45 CC(=O)Nc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217859754 FF For-Sale Unstable SFRP1 87 32 CC(=O)Nc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217859754 FF For-Sale Unstable WNT3 69 32 CCN1CCN(Cc2ccc(F)c(/C=C\C(=O)O)c2)CC1 ZINC000217859765 CE For-Sale Unstable SIGMAR1 16 40 CCN1CCN(Cc2ccc(F)c(/C=C\C(=O)O)c2)CC1 ZINC000217859765 CE For-Sale Unstable CCR1 19 45 O=C(N/C=C/c1ccccc1Br)Nc1ccccc1N1CCOCC1 ZINC000217859769 HI For-Sale Unstable KCNQ2 80 40 O=C(N/C=C/c1ccccc1Br)Nc1ccccc1N1CCOCC1 ZINC000217859769 HI For-Sale Unstable AKR1C3 0 40 C[C@H](c1cc(Cl)ccc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217859784 DH For-Sale Unstable L3MBTL3 64 38 C[C@H](c1cc(Cl)ccc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217859784 DH For-Sale Unstable MBTD1 0 40 O=C(Cc1cccs1)NCCn1ccnc1-c1ccccn1 ZINC000217859787 DE In-Stock Unstable CA5B 30 41 O=C(Cc1cccs1)NCCn1ccnc1-c1ccccn1 ZINC000217859787 DE In-Stock Unstable FAAH 15 42 COC(C)(C)C[C@@H](C)N[C@@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217859788 CI For-Sale Unstable TRPM8 0 42 COC(C)(C)C[C@@H](C)N[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217859818 CI For-Sale Unstable TRPM8 0 42 CC(=O)Nc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217859848 FF For-Sale Unstable CA2 15 42 CC(=O)Nc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217859848 FF For-Sale Unstable CA1 18 41 CC(=O)Nc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217859848 FF For-Sale Unstable NPY2R 17 43 CC(=O)Nc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217859848 FF For-Sale Unstable TGM2 27 43 CC(=O)Nc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217859848 FF For-Sale Unstable ADAMTS5 39 41 CC(=O)Nc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217859848 FF For-Sale Unstable F13A1 48 43 CC(=O)Nc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217859848 FF For-Sale Unstable IDO1 32 45 CC(=O)Nc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217859848 FF For-Sale Unstable SFRP1 87 32 CC(=O)Nc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217859848 FF For-Sale Unstable WNT3 69 32 CN1CCN(c2ccc(NC(=O)N/C=C/c3ccccc3Br)cc2)CC1 ZINC000217859852 HH For-Sale Unstable PRNP 41 48 CN1CCN(c2ccc(NC(=O)N/C=C/c3ccccc3Br)cc2)CC1 ZINC000217859852 HH For-Sale Unstable MTOR 24 42 CC[C@@H](NC(=O)c1ccc(C(C)(C)C)cc1)c1ccc(C)cc1C ZINC000217859866 DK In-Stock Unstable MAP3K5 31 40 CC[C@@H](NC(=O)c1ccc(C(C)(C)C)cc1)c1ccc(C)cc1C ZINC000217859866 DK In-Stock Unstable UTS2 43 38 CCCCN(CCCC)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217859885 CI For-Sale Unstable PTGER2 27 41 CCCCN(CCCC)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217859885 CI For-Sale Unstable AKR1C3 31 47 C[C@@H](c1cccc(O)c1)N1CC[C@@H](N2CCCCC2)C1 ZINC000217859886 CG For-Sale Unstable L3MBTL3 70 37 C[C@@H](c1cccc(O)c1)N1CC[C@@H](N2CCCCC2)C1 ZINC000217859886 CG For-Sale Unstable MBTD1 0 60 COC(C)(C)C[C@H](C)N[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217859916 CI For-Sale Unstable TRPM8 0 42 CC[C@H](NC(=O)c1ccc(C(C)(C)C)cc1)c1ccc(C)cc1C ZINC000217859925 DK In-Stock Unstable MAP3K5 31 40 CC[C@H](NC(=O)c1ccc(C(C)(C)C)cc1)c1ccc(C)cc1C ZINC000217859925 DK In-Stock Unstable UTS2 43 38 O=C(N/C=C/c1ccccc1Br)Nc1ccc(N2CCCCC2)cc1 ZINC000217859948 HK For-Sale Unstable KCNQ2 15 41 CCC[C@@H]1CCN(c2ccc(CBr)cc2C(F)(F)F)C1 ZINC000217859961 FK For-Sale Unstable LIPG 28 40 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc2c(c1)OCCO2 ZINC000217859970 FE For-Sale Unstable PKM 38 45 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc2c(c1)OCCO2 ZINC000217859970 FE For-Sale Unstable SFRP1 63 32 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc2c(c1)OCCO2 ZINC000217859970 FE For-Sale Unstable WNT3 52 32 C[C@H](c1cccc(O)c1)N1CC[C@@H](N2CCCCC2)C1 ZINC000217859975 CG For-Sale Unstable L3MBTL3 70 37 C[C@H](c1cccc(O)c1)N1CC[C@@H](N2CCCCC2)C1 ZINC000217859975 CG For-Sale Unstable MBTD1 0 60 CC[C@@H](C)N(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217859993 CF For-Sale Unstable NR1H4 40 39 CC[C@@H](C)N(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217859993 CF For-Sale Unstable PDS 45 35 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc2c(c1)OCCO2 ZINC000217860031 FE For-Sale Unstable PKM 38 45 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc2c(c1)OCCO2 ZINC000217860031 FE For-Sale Unstable SFRP1 63 32 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc2c(c1)OCCO2 ZINC000217860031 FE For-Sale Unstable WNT3 52 32 CCC[C@@H](C)CN[C@@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217860038 BI For-Sale Unstable TRPM8 0 41 CCC[C@H]1CCN(c2ccc(CBr)cc2C(F)(F)F)C1 ZINC000217860040 FK For-Sale Unstable LIPG 28 40 CC[C@@H](NC(=O)c1ccc(C(C)(C)C)cc1)c1ccc(OC)c(OC)c1 ZINC000217860047 FJ In-Stock Unstable PPARA 17 47 CC[C@@H](NC(=O)c1ccc(C(C)(C)C)cc1)c1ccc(OC)c(OC)c1 ZINC000217860047 FJ In-Stock Unstable TRPV1 28 44 CC[C@@H](NC(=O)c1ccc(C(C)(C)C)cc1)c1ccc(OC)c(OC)c1 ZINC000217860047 FJ In-Stock Unstable PPARD 20 47 CC[C@@H](NC(=O)c1ccc(C(C)(C)C)cc1)c1ccc(OC)c(OC)c1 ZINC000217860047 FJ In-Stock Unstable MT-ND1 36 45 CC[C@@H](NC(=O)c1ccc(C(C)(C)C)cc1)c1ccc(OC)c(OC)c1 ZINC000217860047 FJ In-Stock Unstable UTS2 66 41 CC[C@H](C)N(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217860077 CF For-Sale Unstable NR1H4 40 39 CC[C@H](C)N(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217860077 CF For-Sale Unstable PDS 45 35 CCC[C@H](C)CN[C@@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217860105 BI For-Sale Unstable TRPM8 0 41 CC[C@H](NC(=O)c1ccc(C(C)(C)C)cc1)c1ccc(OC)c(OC)c1 ZINC000217860128 FJ In-Stock Unstable PPARA 17 47 CC[C@H](NC(=O)c1ccc(C(C)(C)C)cc1)c1ccc(OC)c(OC)c1 ZINC000217860128 FJ In-Stock Unstable TRPV1 28 44 CC[C@H](NC(=O)c1ccc(C(C)(C)C)cc1)c1ccc(OC)c(OC)c1 ZINC000217860128 FJ In-Stock Unstable PPARD 20 47 CC[C@H](NC(=O)c1ccc(C(C)(C)C)cc1)c1ccc(OC)c(OC)c1 ZINC000217860128 FJ In-Stock Unstable MT-ND1 36 45 CC[C@H](NC(=O)c1ccc(C(C)(C)C)cc1)c1ccc(OC)c(OC)c1 ZINC000217860128 FJ In-Stock Unstable UTS2 66 41 Nc1cnc(N2CCOCC2)cc1N ZINC000217860133 AC In-Stock Unstable ADK 50 41 COc1cc(C)c(C)cc1S(=O)(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217860157 FG For-Sale Unstable NPY1R 40 32 COc1cc(C)c(C)cc1S(=O)(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217860157 FG For-Sale Unstable NPY2R 47 37 O=C(NCCn1ccnc1-c1ccccn1)c1cccs1 ZINC000217860161 CE In-Stock Unstable SIRT2 21 40 CCC[C@@H](C)CN[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217860177 BI For-Sale Unstable TRPM8 0 41 COc1cc(C)c(C)cc1S(=O)(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217860228 FG For-Sale Unstable NPY1R 40 32 COc1cc(C)c(C)cc1S(=O)(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217860228 FG For-Sale Unstable NPY2R 47 37 CC[C@@H](NC(=O)c1ccc(C(C)(C)C)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217860230 FI In-Stock Unstable CA2 30 43 CC[C@@H](NC(=O)c1ccc(C(C)(C)C)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217860230 FI In-Stock Unstable TRPV1 15 41 CC[C@@H](NC(=O)c1ccc(C(C)(C)C)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217860230 FI In-Stock Unstable CTSF 52 35 CC[C@@H](NC(=O)c1ccc(C(C)(C)C)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217860230 FI In-Stock Unstable LOX1.1 42 38 CC[C@@H](NC(=O)c1ccc(C(C)(C)C)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217860230 FI In-Stock Unstable O49150_SOLTU 50 38 CC[C@@H](NC(=O)c1ccc(C(C)(C)C)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217860230 FI In-Stock Unstable CYNT 46 43 CC[C@@H](NC(=O)c1ccc(C(C)(C)C)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217860230 FI In-Stock Unstable UTS2 56 38 CCC[C@H](C)CN[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217860235 BI For-Sale Unstable TRPM8 0 41 COc1ccc(CCN2C(=O)N[C@@H](CC(=O)NCCc3ccc(O)cc3)C2=O)cc1 ZINC000217860271 HD In-Stock Unstable ADRB1 22 40 COc1ccc(CCN2C(=O)N[C@@H](CC(=O)NCCc3ccc(O)cc3)C2=O)cc1 ZINC000217860271 HD In-Stock Unstable ADRB3 19 40 O=C(NCCn1ccnc1-c1ccccn1)c1cc2ccccc2oc1=O ZINC000217860293 FE In-Stock Unstable POLR1A 46 34 CC[C@H](NC(=O)c1ccc(C(C)(C)C)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217860310 FI In-Stock Unstable CA2 30 43 CC[C@H](NC(=O)c1ccc(C(C)(C)C)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217860310 FI In-Stock Unstable CTSF 48 35 CC[C@H](NC(=O)c1ccc(C(C)(C)C)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217860310 FI In-Stock Unstable LOX1.1 42 38 CC[C@H](NC(=O)c1ccc(C(C)(C)C)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217860310 FI In-Stock Unstable O49150_SOLTU 50 38 CC[C@H](NC(=O)c1ccc(C(C)(C)C)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217860310 FI In-Stock Unstable CYNT 46 43 CC[C@H](NC(=O)c1ccc(C(C)(C)C)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217860310 FI In-Stock Unstable UTS2 46 38 CNc1ccccc1C(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217860355 CE On-Demand Unstable SLC18A3 51 40 Cc1ccc([C@H](C)N[C@H]2C[C@H](C)CC[C@H]2C(C)C)c(O)c1 ZINC000217860372 CJ For-Sale Unstable TRPM8 18 52 CCCN(CCOc1cccc(/C=C\C(=O)O)c1)C(C)C ZINC000217860382 CG For-Sale Unstable AKR1C3 29 41 COc1ccccc1CCN1C(=O)N[C@@H](CCC(=O)NCc2cccnc2)C1=O ZINC000217860395 GD In-Stock Unstable HTR7 19 42 COc1ccccc1CCN1C(=O)N[C@@H](CCC(=O)NCc2cccnc2)C1=O ZINC000217860395 GD In-Stock Unstable MBTPS1 41 32 CNc1ccccc1C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217860427 CE On-Demand Unstable SLC18A3 51 40 Cc1cncc(NC(=O)c2ccc(Br)c(Cl)c2)c1 ZINC000217860444 EI On-Demand Unstable MAOB 18 40 Cc1cncc(NC(=O)c2ccc(Br)c(Cl)c2)c1 ZINC000217860444 EI On-Demand Unstable SCN10A 44 47 Cc1cncc(NC(=O)c2ccc(Br)c(Cl)c2)c1 ZINC000217860444 EI On-Demand Unstable CSF1R 27 46 Cc1cncc(NC(=O)c2ccc(Br)c(Cl)c2)c1 ZINC000217860444 EI On-Demand Unstable TAAR1 21 48 Cc1cncc(NC(=O)c2ccc(Br)c(Cl)c2)c1 ZINC000217860444 EI On-Demand Unstable NAMPT 17 40 Cc1cncc(NC(=O)c2ccc(Br)c(Cl)c2)c1 ZINC000217860444 EI On-Demand Unstable KCNK3 76 42 Cc1cncc(NC(=O)c2ccc(Br)c(Cl)c2)c1 ZINC000217860444 EI On-Demand Unstable KCNK9 44 40 Cc1ccc([C@H](C)N[C@H]2C[C@@H](C)CC[C@H]2C(C)C)c(O)c1 ZINC000217860445 CJ For-Sale Unstable TRPM8 18 52 COc1ccc(-c2noc(CNC(=O)c3ccc(C(C)(C)C)cc3)n2)c(OC)c1 ZINC000217860473 GH In-Stock Unstable PPARA 19 43 COc1ccc(-c2noc(CNC(=O)c3ccc(C(C)(C)C)cc3)n2)c(OC)c1 ZINC000217860473 GH In-Stock Unstable GRIN2B 0 40 COc1ccc(-c2noc(CNC(=O)c3ccc(C(C)(C)C)cc3)n2)c(OC)c1 ZINC000217860473 GH In-Stock Unstable TRPV1 39 40 COc1ccc(-c2noc(CNC(=O)c3ccc(C(C)(C)C)cc3)n2)c(OC)c1 ZINC000217860473 GH In-Stock Unstable PPARD 21 43 COc1ccc(-c2noc(CNC(=O)c3ccc(C(C)(C)C)cc3)n2)c(OC)c1 ZINC000217860473 GH In-Stock Unstable MT-ND1 38 58 COc1ccc(-c2noc(CNC(=O)c3ccc(C(C)(C)C)cc3)n2)c(OC)c1 ZINC000217860473 GH In-Stock Unstable MAP3K5 41 33 COc1cc2c(c(OC)c1OC)-c1ccc(NCCCCCC(=O)Nc3ccc(Cn4cncn4)cc3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217860503 KK In-Stock Unstable TUBA1A 15 56 COc1ccc(CCC(=O)NCCn2ccnc2-c2ccccn2)cc1 ZINC000217860506 FF In-Stock Unstable FAAH 47 48 COc1ccc(CCC(=O)NCCn2ccnc2-c2ccccn2)cc1 ZINC000217860506 FF In-Stock Unstable CES1 28 45 COc1ccc(CCC(=O)NCCn2ccnc2-c2ccccn2)cc1 ZINC000217860506 FF In-Stock Unstable PROKR1 42 30 CCOc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1C ZINC000217860514 FG For-Sale Unstable ADAMTS5 31 42 COC(=O)c1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217860517 GI For-Sale Unstable ACR 47 39 CCCN(CCOc1ccc(/C=C\C(=O)O)cc1)C(C)C ZINC000217860520 CG For-Sale Unstable AHR 15 43 CCCN(CCOc1ccc(/C=C\C(=O)O)cc1)C(C)C ZINC000217860520 CG For-Sale Unstable PLA2G4B 61 33 CCCN(CCOc1ccc(/C=C\C(=O)O)cc1)C(C)C ZINC000217860520 CG For-Sale Unstable AKR1C3 22 40 Cc1ccc([C@H](C)N[C@H]2C[C@@H](C)CC[C@@H]2C(C)C)c(O)c1 ZINC000217860534 CJ For-Sale Unstable TRPM8 18 52 Cc1cncc(NC(=O)c2cc(C)ccc2Br)c1 ZINC000217860563 DH On-Demand Unstable F12 0 40 Cc1cncc(NC(=O)c2cc(C)ccc2Br)c1 ZINC000217860563 DH On-Demand Unstable CSF1R 18 41 Cc1cncc(NC(=O)c2cc(C)ccc2Br)c1 ZINC000217860563 DH On-Demand Unstable KCNK3 52 35 Cc1cncc(NC(=O)c2cc(C)ccc2Br)c1 ZINC000217860563 DH On-Demand Unstable KCNK9 59 36 CCOc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1C ZINC000217860577 FG For-Sale Unstable ADAMTS5 31 42 CC(C)(C)c1ccc(C(=O)NCc2nc(-c3cccc(Br)c3)no2)cc1 ZINC000217860604 HJ In-Stock Unstable KCNQ1 0 47 CC(C)(C)c1ccc(C(=O)NCc2nc(-c3cccc(Br)c3)no2)cc1 ZINC000217860604 HJ In-Stock Unstable MAP3K5 42 37 COc1ccc(O)c(CN[C@H]2C[C@@H](C)CC[C@@H]2C(C)C)c1 ZINC000217860652 CH For-Sale Unstable TRPM8 17 47 CCC1(CNC(=O)c2cc(C)ccc2Br)CCC1 ZINC000217860680 DI On-Demand Unstable HCN1 53 33 CCC1(CNC(=O)c2cc(C)ccc2Br)CCC1 ZINC000217860680 DI On-Demand Unstable HCN4 50 32 COc1c(C)cc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1C ZINC000217860723 FG For-Sale Unstable NPY2R 65 37 COc1c(C)cc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1C ZINC000217860723 FG For-Sale Unstable ADAMTS5 31 40 COc1c(C)cc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1C ZINC000217860723 FG For-Sale Unstable SFRP1 48 31 COc1ccc(-c2noc(CN(C)C(=O)c3ccc(C(C)(C)C)cc3)n2)c(OC)c1 ZINC000217860730 HI In-Stock Unstable MT-ND1 32 44 O=C(N/C=C/c1ccccc1Br)Nc1ccc2ccccc2c1 ZINC000217860737 FK For-Sale Anodyne IMDH_CRYPV 28 40 COc1ccc(O)c(CN[C@H]2C[C@H](C)CC[C@@H]2C(C)C)c1 ZINC000217860746 CH For-Sale Unstable TRPM8 17 47 O=C(NCCn1ccnc1-c1ccccn1)c1cc(=O)c2ccccc2o1 ZINC000217860749 FE In-Stock Unstable BCHE 27 42 COc1c(C)cc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1C ZINC000217860803 FG For-Sale Unstable NPY2R 65 37 COc1c(C)cc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1C ZINC000217860803 FG For-Sale Unstable ADAMTS5 31 40 COc1c(C)cc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1C ZINC000217860803 FG For-Sale Unstable SFRP1 48 31 CC(C)c1ccc(CCCNC(=O)c2ccc(C(C)(C)C)cc2)cc1 ZINC000217860842 EK In-Stock Unstable GCGR 46 42 CC(C)c1ccc(CCCNC(=O)c2ccc(C(C)(C)C)cc2)cc1 ZINC000217860842 EK In-Stock Unstable TRPV1 36 40 CC(C)c1ccc(CCCNC(=O)c2ccc(C(C)(C)C)cc2)cc1 ZINC000217860842 EK In-Stock Unstable ECR 37 42 CC(C)c1ccc(CCCNC(=O)c2ccc(C(C)(C)C)cc2)cc1 ZINC000217860842 EK In-Stock Unstable CYNT 28 54 CC(C)c1ccc(CCCNC(=O)c2ccc(C(C)(C)C)cc2)cc1 ZINC000217860842 EK In-Stock Unstable E3UJZ5_SPOLI 31 42 Cc1nc([C@H](C)N[C@H]2C[C@H](C)CC[C@H]2C(C)C)c(C)s1 ZINC000217860886 CJ For-Sale Unstable TRPM8 0 40 CCc1ccc(OC)c(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217860893 FG For-Sale Unstable ADAMTS5 33 42 O=C(NCCn1ccnc1-c1ccccn1)[C@H]1COc2ccccc2O1 ZINC000217860936 FD In-Stock Unstable ADRA2B 18 41 CN(CCCNC(=O)c1ccc(C(C)(C)C)cc1)c1ccccc1 ZINC000217860942 DI In-Stock Unstable GCGR 19 40 CN(CCCNC(=O)c1ccc(C(C)(C)C)cc1)c1ccccc1 ZINC000217860942 DI In-Stock Unstable KCNQ1 0 48 CN(CCCNC(=O)c1ccc(C(C)(C)C)cc1)c1ccccc1 ZINC000217860942 DI In-Stock Unstable ECR 44 39 CN(CCCNC(=O)c1ccc(C(C)(C)C)cc1)c1ccccc1 ZINC000217860942 DI In-Stock Unstable KCNA3 25 46 CN(CCCNC(=O)c1ccc(C(C)(C)C)cc1)c1ccccc1 ZINC000217860942 DI In-Stock Unstable AMY2 44 32 CN(CCCNC(=O)c1ccc(C(C)(C)C)cc1)c1ccccc1 ZINC000217860942 DI In-Stock Unstable NR1H4 0 50 CN(CCCNC(=O)c1ccc(C(C)(C)C)cc1)c1ccccc1 ZINC000217860942 DI In-Stock Unstable HDA106 0 44 CN(CCCNC(=O)c1ccc(C(C)(C)C)cc1)c1ccccc1 ZINC000217860942 DI In-Stock Unstable CYNT 25 42 CN(CCCNC(=O)c1ccc(C(C)(C)C)cc1)c1ccccc1 ZINC000217860942 DI In-Stock Unstable E3UJZ5_SPOLI 58 38 CCc1ccc(OC)c(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217860961 FG For-Sale Unstable ADAMTS5 33 42 Cc1nc([C@H](C)N[C@H]2C[C@@H](C)CC[C@H]2C(C)C)c(C)s1 ZINC000217860962 CJ For-Sale Unstable TRPM8 0 40 C[C@H](O)[C@@H](NC(=O)N(C)[C@@H](C)c1ccccc1Cl)C(=O)O ZINC000217860977 DD For-Sale Unstable CXCL8 36 40 CSC[C@@](C)(O)CNCc1ccccc1N1CCCC1 ZINC000217861009 CE For-Sale Unstable KCNQ2 68 38 Cc1nc([C@H](C)N[C@H]2C[C@@H](C)CC[C@@H]2C(C)C)c(C)s1 ZINC000217861022 CJ For-Sale Unstable TRPM8 0 40 O=C(NCCn1ccnc1-c1ccccn1)[C@@H]1COc2ccccc2O1 ZINC000217861024 FD In-Stock Unstable ADRA2B 18 41 NC[C@H]1COC[C@H]1c1ccccc1Br ZINC000217861045 CE For-Sale Unstable HTR2B 16 72 CC(C)(C)c1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217861050 FJ In-Stock Unstable HTR1A 21 42 CC(C)(C)c1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217861050 FJ In-Stock Unstable DRD2 35 53 CC(C)(C)c1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217861050 FJ In-Stock Unstable DRD1 23 42 CC(C)(C)c1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217861050 FJ In-Stock Unstable DRD4 43 35 CC(C)(C)c1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217861050 FJ In-Stock Unstable HTR2C 27 41 CC(C)(C)c1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217861050 FJ In-Stock Unstable AVPR2 40 43 CC(C)(C)c1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217861050 FJ In-Stock Unstable DRD3 56 42 CC(C)(C)c1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217861050 FJ In-Stock Unstable HTR3B 0 41 CC(C)(C)c1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217861050 FJ In-Stock Unstable CYNT 24 40 CC(C)(C)c1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217861050 FJ In-Stock Unstable TYRO3 23 40 CC(C)(C)c1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217861050 FJ In-Stock Unstable AP2S1 0 40 CC(C)(C)c1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217861050 FJ In-Stock Unstable ALPHA-1A 0 41 COc1ccc(CCS(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217861055 FF For-Sale Unstable MMP13 37 50 COc1ccc(CCS(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217861055 FF For-Sale Unstable MMP8 18 50 COc1ccc(CCS(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217861055 FF For-Sale Unstable MMP12 20 50 COc1ccc(CCS(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217861055 FF For-Sale Unstable ADAMTS5 25 42 Cc1cc2ncc(N3CCN[C@H](C(C)C)C3)nc2cc1C ZINC000217861063 CF For-Sale Unstable PRKCQ 15 43 C[C@H](O)[C@H](NC(=O)N(C)[C@@H](C)c1ccccc1Cl)C(=O)O ZINC000217861067 DD For-Sale Unstable CXCL8 36 40 CSC[C@](C)(O)CNCc1ccccc1N1CCCC1 ZINC000217861092 CE For-Sale Unstable KCNQ2 68 38 COc1cc(Br)c2[nH]cc(CCN)c2c1 ZINC000217861100 CE For-Sale Unstable HTR1D 35 63 COc1cc(Br)c2[nH]cc(CCN)c2c1 ZINC000217861100 CE For-Sale Unstable HTR1B 34 45 COc1cc(Br)c2[nH]cc(CCN)c2c1 ZINC000217861100 CE For-Sale Unstable MPO 40 42 COc1cc(Br)c2[nH]cc(CCN)c2c1 ZINC000217861100 CE For-Sale Unstable HTR1E 16 41 Cc1cc2ncc(N3CCN[C@@H](C(C)C)C3)nc2cc1C ZINC000217861120 CF For-Sale Unstable PRKCQ 15 43 COc1ccc(CCS(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217861128 FF For-Sale Unstable MMP13 37 50 COc1ccc(CCS(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217861128 FF For-Sale Unstable MMP8 18 50 COc1ccc(CCS(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217861128 FF For-Sale Unstable MMP12 20 50 COc1ccc(CCS(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217861128 FF For-Sale Unstable ADAMTS5 25 42 NC[C@H]1COC[C@@H]1c1ccccc1Br ZINC000217861144 CE For-Sale Unstable HTR2B 16 72 COc1ccc(CNC(=O)c2ccc([N+](=O)[O-])cc2)c(OC)c1OC ZINC000217861175 EF In-Stock Unstable PPARD 21 42 COc1ccc(CNC(=O)c2ccc([N+](=O)[O-])cc2)c(OC)c1OC ZINC000217861175 EF In-Stock Unstable SLC9A1 61 38 COc1ccc(CNC(=O)c2ccc([N+](=O)[O-])cc2)c(OC)c1OC ZINC000217861175 EF In-Stock Unstable KCNMA1 19 40 COc1ccc(CNC(=O)c2ccc([N+](=O)[O-])cc2)c(OC)c1OC ZINC000217861175 EF In-Stock Unstable MT-ND1 18 44 COc1ccc(CNC(=O)c2ccc([N+](=O)[O-])cc2)c(OC)c1OC ZINC000217861175 EF In-Stock Unstable U38 0 40 CNc1ccccc1C(=O)N[C@@H]1CCN2CCC[C@@H]12 ZINC000217861200 CD For-Sale Unstable SLC18A3 44 38 NC[C@@H]1COC[C@H]1c1ccccc1Br ZINC000217861204 CE For-Sale Unstable HTR2B 16 72 COc1ccc(OC)c(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217861249 GF For-Sale Unstable DRD2 19 42 COc1ccc(OC)c(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217861249 GF For-Sale Unstable ADRA1D 15 42 COc1ccc(OC)c(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217861249 GF For-Sale Unstable NPY1R 40 31 COc1ccc(OC)c(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217861249 GF For-Sale Unstable NPY2R 61 41 COc1ccc(OC)c(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217861249 GF For-Sale Unstable NPY5R 16 41 COc1ccc(OC)c(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)c1 ZINC000217861249 GF For-Sale Unstable ADAMTS5 31 44 CCOc1ccc(CNC(=O)c2ccc([N+](=O)[O-])cc2)cc1OCC ZINC000217861276 EG In-Stock Unstable PPARA 15 43 CCOc1ccc(CNC(=O)c2ccc([N+](=O)[O-])cc2)cc1OCC ZINC000217861276 EG In-Stock Unstable CCR3 0 47 CCOc1ccc(CNC(=O)c2ccc([N+](=O)[O-])cc2)cc1OCC ZINC000217861276 EG In-Stock Unstable ACR 23 41 CCOc1ccc(CNC(=O)c2ccc([N+](=O)[O-])cc2)cc1OCC ZINC000217861276 EG In-Stock Unstable MT-ND1 25 46 CCOc1ccc(CNC(=O)c2ccc([N+](=O)[O-])cc2)cc1OCC ZINC000217861276 EG In-Stock Unstable U38 0 44 CCOc1ccc(CNC(=O)c2ccc([N+](=O)[O-])cc2)cc1OCC ZINC000217861276 EG In-Stock Unstable ENR 0 41 NC[C@@H]1COC[C@@H]1c1ccccc1Br ZINC000217861278 CE For-Sale Unstable HTR2B 16 72 CNc1ccccc1C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217861307 CD For-Sale Unstable SLC18A3 44 38 COc1ccc(OC)c(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217861328 GF For-Sale Unstable DRD2 19 42 COc1ccc(OC)c(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217861328 GF For-Sale Unstable ADRA1D 15 42 COc1ccc(OC)c(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217861328 GF For-Sale Unstable NPY1R 40 31 COc1ccc(OC)c(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217861328 GF For-Sale Unstable NPY2R 61 41 COc1ccc(OC)c(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217861328 GF For-Sale Unstable NPY5R 16 41 COc1ccc(OC)c(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)c1 ZINC000217861328 GF For-Sale Unstable ADAMTS5 31 44 CS(=O)(=O)N1CCC(C(=O)NCCn2ccnc2-c2ccccn2)CC1 ZINC000217861335 GC In-Stock Unstable EPHX2 42 43 CNNC(=O)c1cc(C)cc(C)c1 ZINC000217861345 AD For-Sale Unstable ECR 41 38 CNNC(=O)c1cc(C)cc(C)c1 ZINC000217861345 AD For-Sale Unstable E3UJZ5_SPOLI 47 38 CCN(Cc1cccc(/C=C\C(=O)O)c1)C1CCCC1 ZINC000217861346 CH For-Sale Unstable PTGER2 0 40 CCN(Cc1cccc(/C=C\C(=O)O)c1)C1CCCC1 ZINC000217861346 CH For-Sale Unstable NR1H4 42 40 COc1cccc2c1ccn2CCNC(=O)CCc1c[nH]c2ccccc12 ZINC000217861360 FH In-Stock Unstable ACHE 29 42 COc1cccc2c1ccn2CCNC(=O)CCc1c[nH]c2ccccc12 ZINC000217861360 FH In-Stock Unstable TACR1 38 40 COc1cccc2c1ccn2CCNC(=O)CCc1c[nH]c2ccccc12 ZINC000217861360 FH In-Stock Unstable BRS3 22 41 COc1cccc2c1ccn2CCNC(=O)CCc1c[nH]c2ccccc12 ZINC000217861360 FH In-Stock Unstable NMBR 31 40 COc1cccc2c1ccn2CCNC(=O)CCc1c[nH]c2ccccc12 ZINC000217861360 FH In-Stock Unstable MC5R 28 40 COc1cccc2c1ccn2CCNC(=O)CCc1c[nH]c2ccccc12 ZINC000217861360 FH In-Stock Unstable GHSR 47 36 COc1ccccc1CCCNC(=O)c1ccc([N+](=O)[O-])cc1 ZINC000217861416 DF In-Stock Unstable DRD2 21 44 COc1ccccc1CCCNC(=O)c1ccc([N+](=O)[O-])cc1 ZINC000217861416 DF In-Stock Unstable DRD1 0 43 COc1ccccc1CCCNC(=O)c1ccc([N+](=O)[O-])cc1 ZINC000217861416 DF In-Stock Unstable DRD3 33 43 COc1ccccc1CCCNC(=O)c1ccc([N+](=O)[O-])cc1 ZINC000217861416 DF In-Stock Unstable MTNR1B 41 42 COc1ccccc1CCCNC(=O)c1ccc([N+](=O)[O-])cc1 ZINC000217861416 DF In-Stock Unstable KCNMA1 19 41 COc1ccccc1CCCNC(=O)c1ccc([N+](=O)[O-])cc1 ZINC000217861416 DF In-Stock Unstable HDA106 0 51 COc1ccccc1CCCNC(=O)c1ccc([N+](=O)[O-])cc1 ZINC000217861416 DF In-Stock Unstable AP2S1 0 44 O=C(NCCn1ccnc1-c1ccccn1)c1cc(-c2ccccc2)on1 ZINC000217861432 FG In-Stock Unstable HDAC10 18 51 COc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217861437 GF For-Sale Unstable DRD2 19 41 COc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217861437 GF For-Sale Unstable NPY2R 49 37 COc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217861437 GF For-Sale Unstable HTR6 26 45 COc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217861437 GF For-Sale Unstable ADAMTS5 32 42 COc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217861437 GF For-Sale Unstable SFRP1 43 30 COc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1OC ZINC000217861437 GF For-Sale Unstable ACKR3 41 35 C[C@@H]1CCCN(c2ccccn2)C1 ZINC000217861454 AE On-Demand Unstable DRD4 26 43 C[C@@H]1CCCN(c2ccccn2)C1 ZINC000217861454 AE On-Demand Unstable EBP 30 43 CSc1ccc(CN[C@H]2C[C@@H](C)CC[C@@H]2C(C)C)cc1 ZINC000217861474 CJ For-Sale Unstable TRPM8 16 42 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217861496 GF For-Sale Unstable DRD2 19 41 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217861496 GF For-Sale Unstable NPY2R 49 37 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217861496 GF For-Sale Unstable HTR6 26 45 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217861496 GF For-Sale Unstable ADAMTS5 32 42 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217861496 GF For-Sale Unstable SFRP1 43 30 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1OC ZINC000217861496 GF For-Sale Unstable ACKR3 41 35 C[C@H]1CCCC[C@H]1N[C@H](C)CC(C)(C)c1ccccc1 ZINC000217861525 CJ For-Sale Unstable AMY2 44 30 CCOc1ccc(CCCNC(=O)c2ccc([N+](=O)[O-])cc2)cc1 ZINC000217861528 EG In-Stock Unstable KCNQ1 0 42 CCOc1ccc(CCCNC(=O)c2ccc([N+](=O)[O-])cc2)cc1 ZINC000217861528 EG In-Stock Unstable CCR3 0 43 CCOc1ccc(CCCNC(=O)c2ccc([N+](=O)[O-])cc2)cc1 ZINC000217861528 EG In-Stock Unstable SCN2A 16 47 CCOc1ccc(CCCNC(=O)c2ccc([N+](=O)[O-])cc2)cc1 ZINC000217861528 EG In-Stock Unstable ACR 24 43 CCOc1ccc(CCCNC(=O)c2ccc([N+](=O)[O-])cc2)cc1 ZINC000217861528 EG In-Stock Unstable HDA106 0 51 CSc1ccc(CN[C@H]2C[C@H](C)CC[C@@H]2C(C)C)cc1 ZINC000217861550 CJ For-Sale Unstable TRPM8 16 42 C[C@H]1CCCN(c2ccccn2)C1 ZINC000217861552 AE On-Demand Unstable DRD4 26 43 C[C@H]1CCCN(c2ccccn2)C1 ZINC000217861552 AE On-Demand Unstable EBP 30 43 COc1nn(C)cc1C(=O)NCCn1ccnc1-c1ccccn1 ZINC000217861557 ED In-Stock Unstable DRD4 40 31 Cc1nc(NC(=O)OC(C)(C)C)sc1C(=O)NCc1ccccc1 ZINC000217861563 EH On-Demand Unstable CHRM4 30 45 Cc1nc(NC(=O)OC(C)(C)C)sc1C(=O)NCc1ccccc1 ZINC000217861563 EH On-Demand Unstable SCD1 50 51 Cc1nc(NC(=O)OC(C)(C)C)sc1C(=O)NCc1ccccc1 ZINC000217861563 EH On-Demand Unstable SCD 43 50 Cc1nc(NC(=O)OC(C)(C)C)sc1C(=O)NCc1ccccc1 ZINC000217861563 EH On-Demand Unstable PDS 41 33 C[C@H]1CCCC[C@@H]1N[C@H](C)CC(C)(C)c1ccccc1 ZINC000217861582 CJ For-Sale Unstable AMY2 44 30 COC(=O)c1sccc1S(=O)(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217861600 GE For-Sale Unstable ADAMTS5 34 40 CSC[C@@](C)(O)CNCc1ccccc1[N+](=O)[O-] ZINC000217861605 CD On-Demand Unstable COLA 99 40 CSC[C@@](C)(O)CNCc1ccccc1[N+](=O)[O-] ZINC000217861605 CD On-Demand Unstable PQSD 0 44 CCCOc1ccccc1CCCNC(=O)c1ccc([N+](=O)[O-])cc1 ZINC000217861610 EH In-Stock Unstable CCR3 0 41 CC1(C)C[C@H]2C[C@@](C)(CN2C(=O)N/C=C/c2ccccc2Br)C1 ZINC000217861638 GK For-Sale Unstable AVPR2 16 44 CC1(C)C[C@H]2C[C@@](C)(CN2C(=O)N/C=C/c2ccccc2Br)C1 ZINC000217861638 GK For-Sale Unstable AVPR1A 38 44 CCC[C@@H](O)CNCCc1cccnc1 ZINC000217861639 BD For-Sale Unstable ADRB2 63 42 CCC[C@@H](O)CNCCc1cccnc1 ZINC000217861639 BD For-Sale Unstable ADRB3 99 45 CCC[C@@H](O)CNCCc1cccnc1 ZINC000217861639 BD For-Sale Unstable FDFT1 0 41 COC(=O)C[C@H](C1=C(O)C(=O)c2ccccc2C1=O)c1cc2cc(OC)ccc2[nH]c1=O ZINC000217861642 IG In-Stock Unstable TUBB2B 39 43 COC(=O)c1sccc1S(=O)(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217861669 GE For-Sale Unstable ADAMTS5 34 40 CSC[C@](C)(O)CNCc1ccccc1[N+](=O)[O-] ZINC000217861686 CD On-Demand Unstable COLA 99 40 CSC[C@](C)(O)CNCc1ccccc1[N+](=O)[O-] ZINC000217861686 CD On-Demand Unstable PQSD 0 44 O=C(O)/C=C\c1cc(Cn2ccccc2=O)ccc1F ZINC000217861691 CE For-Sale Unstable PTGER2 30 40 O=C(O)/C=C\c1cc(Cn2ccccc2=O)ccc1F ZINC000217861691 CE For-Sale Unstable PTGER4 18 40 O=C(O)/C=C\c1cc(Cn2ccccc2=O)ccc1F ZINC000217861691 CE For-Sale Unstable PTGER3 40 40 CC1CCN(c2ccc([C@@H](C)NC(=O)c3ccc([N+](=O)[O-])cc3)cc2)CC1 ZINC000217861716 FI In-Stock Unstable SSTR2 35 42 CC(C)(C)OC(=O)Nc1nc(CN2CCOCC2)c(C(=O)NCc2ccccc2)s1 ZINC000217861723 IG For-Sale Unstable CASR 41 36 CC(C)(C)OC(=O)Nc1nc(CN2CCOCC2)c(C(=O)NCc2ccccc2)s1 ZINC000217861723 IG For-Sale Unstable SCD1 25 42 CC(C)(C)OC(=O)Nc1nc(CN2CCOCC2)c(C(=O)NCc2ccccc2)s1 ZINC000217861723 IG For-Sale Unstable SCD 23 40 CCC[C@H](O)CNCCc1cccnc1 ZINC000217861725 BD For-Sale Unstable ADRB2 63 42 CCC[C@H](O)CNCCc1cccnc1 ZINC000217861725 BD For-Sale Unstable ADRB3 99 45 CCC[C@H](O)CNCCc1cccnc1 ZINC000217861725 BD For-Sale Unstable FDFT1 0 41 COC(=O)C[C@@H](C1=C(O)C(=O)c2ccccc2C1=O)c1cc2cc(OC)ccc2[nH]c1=O ZINC000217861729 IG In-Stock Unstable TUBB2B 39 43 COc1ccc(Cl)cc1S(=O)(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217861762 GG For-Sale Unstable ADRA1D 23 43 COc1ccc(Cl)cc1S(=O)(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217861762 GG For-Sale Unstable ADRA1A 18 43 COc1ccc(Cl)cc1S(=O)(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217861762 GG For-Sale Unstable ADRA1B 20 43 COc1ccc(Cl)cc1S(=O)(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217861762 GG For-Sale Unstable NPY2R 51 35 COc1ccc(Cl)cc1S(=O)(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217861762 GG For-Sale Unstable COLA 79 51 COc1ccc(Cl)cc1S(=O)(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217861762 GG For-Sale Unstable CPT1A 74 51 COc1ccc(Cl)cc1S(=O)(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217861762 GG For-Sale Unstable CPT2 48 36 COc1ccc(Cl)cc1S(=O)(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217861762 GG For-Sale Unstable CPT1B 62 37 NC[C@H]1COC[C@H]1c1cccc(Br)c1 ZINC000217861766 CE For-Sale Unstable HTR2B 15 69 O=C(CCSc1ccccc1)NCCn1ccnc1-c1ccccn1 ZINC000217861767 FG In-Stock Unstable FAAH 15 45 CC1CCN(c2ccc([C@H](C)NC(=O)c3ccc([N+](=O)[O-])cc3)cc2)CC1 ZINC000217861795 FI In-Stock Unstable SSTR2 35 42 COc1ccc(Cn2nc(C)cc2C)cc1/C=C\C(=O)O ZINC000217861804 CF For-Sale Unstable PTGER2 34 41 COc1ccc(Cn2nc(C)cc2C)cc1/C=C\C(=O)O ZINC000217861804 CF For-Sale Unstable PTGER4 0 41 COc1ccc(Cn2nc(C)cc2C)cc1/C=C\C(=O)O ZINC000217861804 CF For-Sale Unstable PTGER3 15 41 O=C(C[C@@H]1NC(=O)c2ccccc2NC1=O)NC1CCN(C(=O)c2cc3ccccc3[nH]2)CC1 ZINC000217861813 JE In-Stock Unstable GRIN2B 29 44 O=C(C[C@@H]1NC(=O)c2ccccc2NC1=O)NC1CCN(C(=O)c2cc3ccccc3[nH]2)CC1 ZINC000217861813 JE In-Stock Unstable HRH4 19 45 O=C(C[C@@H]1NC(=O)c2ccccc2NC1=O)NC1CCN(C(=O)c2cc3ccccc3[nH]2)CC1 ZINC000217861813 JE In-Stock Unstable AKR1C3 20 49 C#CCCNC[C@@H](O)CCC ZINC000217861815 AC For-Sale Unstable CYP4A4 45 29 CN(C)c1cccc(NC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217861822 FI For-Sale Unstable KCNK3 56 42 NC[C@H]1COC[C@@H]1c1cccc(Br)c1 ZINC000217861833 CE For-Sale Unstable HTR2B 15 69 COc1ccc(Cl)cc1S(=O)(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217861840 GG For-Sale Unstable ADRA1D 23 43 COc1ccc(Cl)cc1S(=O)(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217861840 GG For-Sale Unstable ADRA1A 18 43 COc1ccc(Cl)cc1S(=O)(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217861840 GG For-Sale Unstable ADRA1B 20 43 COc1ccc(Cl)cc1S(=O)(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217861840 GG For-Sale Unstable NPY2R 51 35 COc1ccc(Cl)cc1S(=O)(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217861840 GG For-Sale Unstable COLA 79 51 COc1ccc(Cl)cc1S(=O)(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217861840 GG For-Sale Unstable CPT1A 74 51 COc1ccc(Cl)cc1S(=O)(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217861840 GG For-Sale Unstable CPT2 48 36 COc1ccc(Cl)cc1S(=O)(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217861840 GG For-Sale Unstable CPT1B 62 37 C#CCCNC[C@H](O)CCC ZINC000217861853 AC For-Sale Unstable CYP4A4 45 29 Cn1ncc2c(SCCOc3cc(Cl)ccc3Cl)ncnc21 ZINC000217861862 FH On-Demand Unstable Q9M629_MAIZE 53 37 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1N[C@@H](C)c1ccc(F)c(Cl)c1 ZINC000217861863 DK For-Sale Unstable TRPM8 16 50 CC[C@@H](C)N(C)CCNC(=O)CCCC(=O)O ZINC000217861887 BD On-Demand Unstable DNM1 0 48 CCCCCCCCCCCCCCCCCCOC[C@@H](CO[P@@](=O)(O)OCCBr)OC(N)=O ZINC000217861892 KK For-Sale Unstable PTAFR 20 60 CCCCCCCCCCCCCCCCCCOC[C@@H](CO[P@@](=O)(O)OCCBr)OC(N)=O ZINC000217861892 KK For-Sale Unstable LPAR1 15 50 CCCCCCCCCCCCCCCCCCOC[C@@H](CO[P@@](=O)(O)OCCBr)OC(N)=O ZINC000217861892 KK For-Sale Unstable LPAR3 51 50 CN1CCc2nc(NC(=O)N/C=C/c3ccccc3Br)sc2C1 ZINC000217861897 GH For-Sale Unstable F10 23 45 NC[C@@H]1COC[C@H]1c1cccc(Br)c1 ZINC000217861911 CE For-Sale Unstable HTR2B 15 69 COc1ccc([C@@H](C)N[C@@H]2CCCC[C@@H]2C)c(F)c1 ZINC000217861941 CI For-Sale Unstable CASR 0 41 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1N[C@@H](C)c1ccc(F)c(Cl)c1 ZINC000217861950 DK For-Sale Unstable TRPM8 16 50 CC[C@H](C)N(C)CCNC(=O)CCCC(=O)O ZINC000217861956 BD On-Demand Unstable DNM1 0 48 CCCCCCCCCCCCCCCCCCOC[C@H](CO[P@@](=O)(O)OCCBr)OC(N)=O ZINC000217861958 KK For-Sale Unstable PTAFR 20 60 CCCCCCCCCCCCCCCCCCOC[C@H](CO[P@@](=O)(O)OCCBr)OC(N)=O ZINC000217861958 KK For-Sale Unstable LPAR1 15 50 CCCCCCCCCCCCCCCCCCOC[C@H](CO[P@@](=O)(O)OCCBr)OC(N)=O ZINC000217861958 KK For-Sale Unstable LPAR3 51 50 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc(C(F)(F)F)cc1 ZINC000217861960 GH For-Sale Unstable ADAMTS5 36 59 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc(C(F)(F)F)cc1 ZINC000217861960 GH For-Sale Unstable SFRP1 126 40 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc(C(F)(F)F)cc1 ZINC000217861960 GH For-Sale Unstable WNT3 86 36 NC[C@@H]1COC[C@@H]1c1cccc(Br)c1 ZINC000217861972 CE For-Sale Unstable HTR2B 15 69 COc1ccc(CNC[C@@](C)(O)CSC)cc1C ZINC000217861979 CE On-Demand Unstable MT-ND1 15 40 CC[C@@H]1c2ccsc2CCN1C(=O)CSc1ncn(-c2ccccc2)n1 ZINC000217862008 GH On-Demand Unstable TRPM8 17 45 COc1ccc([C@@H](C)N[C@H]2CCCC[C@@H]2C)c(F)c1 ZINC000217862030 CI For-Sale Unstable CASR 0 41 COc1ccc(CNC[C@](C)(O)CSC)cc1C ZINC000217862038 CE On-Demand Unstable MT-ND1 15 40 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1N[C@@H](C)c1ccc(F)c(Cl)c1 ZINC000217862045 DK For-Sale Unstable TRPM8 16 50 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc(C(F)(F)F)cc1 ZINC000217862053 GH For-Sale Unstable ADAMTS5 36 59 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc(C(F)(F)F)cc1 ZINC000217862053 GH For-Sale Unstable SFRP1 126 40 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc(C(F)(F)F)cc1 ZINC000217862053 GH For-Sale Unstable WNT3 86 36 O=C(NCCc1ccccc1F)c1cc(I)ccc1O ZINC000217862060 GG For-Sale Unstable SLC6A5 40 34 CC[C@H]1c2ccsc2CCN1C(=O)CSc1ncn(-c2ccccc2)n1 ZINC000217862081 GH On-Demand Unstable TRPM8 17 45 O=C(NCCn1ccnc1-c1ccccn1)c1ccc(Cl)s1 ZINC000217862092 EG In-Stock Unstable F10 29 46 CC(C)[C@H]1CC[C@H](C)C[C@@H]1N[C@@H](C)c1ccc(F)c(Cl)c1 ZINC000217862122 DK For-Sale Unstable TRPM8 16 50 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1cccc(C(F)(F)F)c1 ZINC000217862162 GH For-Sale Unstable CACNA1B 54 37 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1cccc(C(F)(F)F)c1 ZINC000217862162 GH For-Sale Unstable CCR2 26 43 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1cccc(C(F)(F)F)c1 ZINC000217862162 GH For-Sale Unstable ADAMTS5 32 48 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1cccc(C(F)(F)F)c1 ZINC000217862162 GH For-Sale Unstable SFRP1 130 39 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1cccc(C(F)(F)F)c1 ZINC000217862162 GH For-Sale Unstable WNT3 87 36 NC(=O)c1ccccc1NC(=O)N/C=C/c1ccccc1Br ZINC000217862205 FG For-Sale Unstable PAGA 0 45 Cc1cccc(OC[C@@H]2CCCN(C(=O)Cn3nc(C)cc3N)C2)c1 ZINC000217862212 EE In-Stock Unstable CHRNA10 42 37 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1cccc(C(F)(F)F)c1 ZINC000217862246 GH For-Sale Unstable CACNA1B 54 37 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1cccc(C(F)(F)F)c1 ZINC000217862246 GH For-Sale Unstable CCR2 26 43 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1cccc(C(F)(F)F)c1 ZINC000217862246 GH For-Sale Unstable ADAMTS5 32 48 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1cccc(C(F)(F)F)c1 ZINC000217862246 GH For-Sale Unstable SFRP1 130 39 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1cccc(C(F)(F)F)c1 ZINC000217862246 GH For-Sale Unstable WNT3 87 36 Cc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1ccc([N+](=O)[O-])cc1 ZINC000217862287 EH In-Stock Unstable CACNA1D 52 34 Cc1cccc(OC[C@H]2CCCN(C(=O)Cn3nc(C)cc3N)C2)c1 ZINC000217862298 EE In-Stock Unstable CHRNA10 42 37 Cc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1ccc([N+](=O)[O-])cc1 ZINC000217862355 EH In-Stock Unstable CACNA1D 52 34 O=C(NCCn1ccnc1-c1ccccn1)c1cccc(OC(F)(F)F)c1 ZINC000217862367 GG In-Stock Unstable DRD4 49 38 O=C(NCCn1ccnc1-c1ccccn1)c1cccc(OC(F)(F)F)c1 ZINC000217862367 GG In-Stock Unstable SCN1A 0 46 O=C(NCCn1ccnc1-c1ccccn1)c1cccc(OC(F)(F)F)c1 ZINC000217862367 GG In-Stock Unstable GCGR 18 41 O=C(NCCn1ccnc1-c1ccccn1)c1cccc(OC(F)(F)F)c1 ZINC000217862367 GG In-Stock Unstable SCN8A 0 46 COc1cccc(N2CCN(C(=O)COc3coc(CN4CCc5cc(OC)c(OC)cc5C4)cc3=O)CC2)c1 ZINC000217862376 KF In-Stock Unstable DRD4 41 33 COc1cccc(N2CCN(C(=O)COc3coc(CN4CCc5cc(OC)c(OC)cc5C4)cc3=O)CC2)c1 ZINC000217862376 KF In-Stock Unstable ABCB1B 53 33 COc1cccc(N2CCN(C(=O)COc3coc(CN4CCc5cc(OC)c(OC)cc5C4)cc3=O)CC2)c1 ZINC000217862376 KF In-Stock Unstable ABCB1 28 43 COc1cccc(N2CCN(C(=O)COc3coc(CN4CCc5cc(OC)c(OC)cc5C4)cc3=O)CC2)c1 ZINC000217862376 KF In-Stock Unstable ABCG2 29 41 CS(=O)(=O)c1cc(F)cc([C@H](N)C(=O)O)c1 ZINC000217862379 BC For-Sale Unstable CACNA2D1 19 43 O=C(N/C=C/c1ccccc1Br)Nc1cccc(Br)c1 ZINC000217862407 GK For-Sale Anodyne KCNK3 73 34 CS(=O)(=O)c1cc(F)cc([C@@H](N)C(=O)O)c1 ZINC000217862441 BC For-Sale Unstable CACNA2D1 19 43 COc1ccc2c(c1)[C@@H](NC(=O)c1ccc([N+](=O)[O-])cc1)CC(C)(C)O2 ZINC000217862444 FH In-Stock Unstable NAAA 18 42 O=C(NCCn1ccnc1-c1ccccn1)Nc1cccc(Cl)c1 ZINC000217862460 EG In-Stock Unstable PPIA 23 43 O=C(NCCn1ccnc1-c1ccccn1)Nc1cccc(Cl)c1 ZINC000217862460 EG In-Stock Unstable PTGER3 17 42 O=C(NCCn1ccnc1-c1ccccn1)Nc1cccc(Cl)c1 ZINC000217862460 EG In-Stock Unstable GRM5 15 43 O=C(NCCn1ccnc1-c1ccccn1)Nc1cccc(Cl)c1 ZINC000217862460 EG In-Stock Unstable CCKBR 38 41 O=C(NCCn1ccnc1-c1ccccn1)Nc1cccc(Cl)c1 ZINC000217862460 EG In-Stock Unstable EPHB4 28 41 O=C(CCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCc1ccc2c(c1)OCO2 ZINC000217862461 JG In-Stock Unstable NOS2 86 35 COc1ccc2c(c1)[C@H](NC(=O)c1ccc([N+](=O)[O-])cc1)CC(C)(C)O2 ZINC000217862519 FH In-Stock Unstable NAAA 18 42 Cc1ccccc1OCc1ccccc1/C=C\C(=O)O ZINC000217862536 CH For-Sale Unstable PTGER2 31 57 Cc1ccccc1OCc1ccccc1/C=C\C(=O)O ZINC000217862536 CH For-Sale Unstable PTGER4 48 56 Cc1ccccc1OCc1ccccc1/C=C\C(=O)O ZINC000217862536 CH For-Sale Unstable PTGER3 36 57 Cc1ccccc1OCc1ccccc1/C=C\C(=O)O ZINC000217862536 CH For-Sale Unstable PTGDR 0 50 Cc1ccccc1OCc1ccccc1/C=C\C(=O)O ZINC000217862536 CH For-Sale Unstable MT-CYB 22 46 O=C(CCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCc1ccc2c(c1)OCO2 ZINC000217862538 JG In-Stock Unstable NOS2 86 35 CC(C)COc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217862551 GH For-Sale Unstable NPY2R 42 35 CC(C)COc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217862551 GH For-Sale Unstable ADAMTS5 34 43 COc1cccc(NC(=O)NCCn2ccnc2-c2ccccn2)c1 ZINC000217862579 EF In-Stock Unstable DRD4 47 36 COc1cccc(NC(=O)NCCn2ccnc2-c2ccccn2)c1 ZINC000217862579 EF In-Stock Unstable HRH2 45 45 COc1cccc(NC(=O)NCCn2ccnc2-c2ccccn2)c1 ZINC000217862579 EF In-Stock Unstable PTGER3 21 44 COc1cccc(NC(=O)NCCn2ccnc2-c2ccccn2)c1 ZINC000217862579 EF In-Stock Unstable CCKAR 35 41 COc1cccc(NC(=O)NCCn2ccnc2-c2ccccn2)c1 ZINC000217862579 EF In-Stock Unstable CCR3 37 44 COc1cccc(NC(=O)NCCn2ccnc2-c2ccccn2)c1 ZINC000217862579 EF In-Stock Unstable CCKBR 37 43 COc1cccc(NC(=O)NCCn2ccnc2-c2ccccn2)c1 ZINC000217862579 EF In-Stock Unstable ZAP70 43 40 COc1cccc(NC(=O)NCCn2ccnc2-c2ccccn2)c1 ZINC000217862579 EF In-Stock Unstable ACAT 0 47 COc1cccc(NC(=O)NCCn2ccnc2-c2ccccn2)c1 ZINC000217862579 EF In-Stock Unstable SLC11A2 17 46 COc1cccc(NC(=O)NCCn2ccnc2-c2ccccn2)c1 ZINC000217862579 EF In-Stock Unstable KCNK3 42 35 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCc1cc(F)ccc1F ZINC000217862599 CJ For-Sale Unstable TRPM8 16 49 CC(C)COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217862621 GH For-Sale Unstable NPY2R 42 35 CC(C)COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217862621 GH For-Sale Unstable ADAMTS5 34 43 Cc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217862624 CH For-Sale Unstable PTGER2 31 52 Cc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217862624 CH For-Sale Unstable PPIA 42 33 Cc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217862624 CH For-Sale Unstable PTGER1 37 41 Cc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217862624 CH For-Sale Unstable PTGER4 45 50 Cc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217862624 CH For-Sale Unstable PTGER3 33 50 Cc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217862624 CH For-Sale Unstable PTGDR 0 44 Cc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217862624 CH For-Sale Unstable FFAR1 30 40 Cc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217862624 CH For-Sale Unstable AKR1C3 39 55 Cc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217862624 CH For-Sale Unstable AKR1B10 22 43 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1ccc([N+](=O)[O-])cc1 ZINC000217862640 FH In-Stock Unstable CACNA1D 63 36 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1ccc([N+](=O)[O-])cc1 ZINC000217862640 FH In-Stock Unstable NAAA 21 42 CC(C)[C@H](NC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)C(=O)NCCn1ccc2ccccc21 ZINC000217862643 JF In-Stock Unstable CHRNA4 27 44 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCc1cc(F)ccc1F ZINC000217862672 CJ For-Sale Unstable TRPM8 16 49 O=C(NCCn1ccnc1-c1ccccn1)Nc1c(F)cccc1F ZINC000217862679 EG In-Stock Unstable ACAT 0 43 CC(C)(C)c1ccc(NC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217862698 FK For-Sale Unstable TRPV1 19 46 Cc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1F ZINC000217862708 CH For-Sale Unstable PTGER2 22 47 Cc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1F ZINC000217862708 CH For-Sale Unstable PTGER1 36 40 Cc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1F ZINC000217862708 CH For-Sale Unstable PTGER4 25 42 Cc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1F ZINC000217862708 CH For-Sale Unstable PTGER3 22 42 Cc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1F ZINC000217862708 CH For-Sale Unstable AKR1C3 37 53 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1ccc([N+](=O)[O-])cc1 ZINC000217862714 FH In-Stock Unstable CACNA1D 63 36 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1ccc([N+](=O)[O-])cc1 ZINC000217862714 FH In-Stock Unstable NAAA 21 42 CCCOc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1C ZINC000217862718 GH For-Sale Unstable ADAMTS5 32 43 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCc1cc(F)ccc1F ZINC000217862750 CJ For-Sale Unstable TRPM8 16 49 C[C@H](Sc1nnc(Cc2ccccc2)n1-c1ccccc1)C(=O)N[C@@H]1CCCC[C@@H]1C ZINC000217862753 IK For-Sale Anodyne BIRC2 45 36 Cc1ccc(NC(=O)NCCn2ccnc2-c2ccccn2)cc1C ZINC000217862782 EG In-Stock Unstable QPCT 17 40 Cc1ccc(NC(=O)NCCn2ccnc2-c2ccccn2)cc1C ZINC000217862782 EG In-Stock Unstable PRMT3 44 34 O=C(O)/C=C\c1ccccc1COc1ccc(F)cc1 ZINC000217862793 CH For-Sale Unstable PTGER2 23 50 O=C(O)/C=C\c1ccccc1COc1ccc(F)cc1 ZINC000217862793 CH For-Sale Unstable PTGER4 31 50 O=C(O)/C=C\c1ccccc1COc1ccc(F)cc1 ZINC000217862793 CH For-Sale Unstable PTGER3 29 56 O=C(O)/C=C\c1ccccc1COc1ccc(F)cc1 ZINC000217862793 CH For-Sale Unstable CDC25B 23 43 O=C(O)/C=C\c1ccccc1COc1ccc(F)cc1 ZINC000217862793 CH For-Sale Unstable GYS1 51 34 O=C(O)/C=C\c1ccccc1COc1ccc(F)cc1 ZINC000217862793 CH For-Sale Unstable PTGDR 0 56 O=C(O)/C=C\c1ccccc1COc1ccc(F)cc1 ZINC000217862793 CH For-Sale Unstable FFAR1 24 48 O=C(O)/C=C\c1ccccc1COc1ccc(F)cc1 ZINC000217862793 CH For-Sale Unstable FFAR4 46 48 CCCOc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1C ZINC000217862810 GH For-Sale Unstable ADAMTS5 32 43 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCc1cc(F)ccc1F ZINC000217862819 CJ For-Sale Unstable TRPM8 16 49 C[C@H](Sc1nnc(Cc2ccccc2)n1-c1ccccc1)C(=O)N[C@H]1CCCC[C@@H]1C ZINC000217862825 IK For-Sale Anodyne BIRC2 45 36 CC[C@@H](NC(=O)c1ccc([N+](=O)[O-])cc1)c1ccc(C)c(C)c1 ZINC000217862828 DI In-Stock Unstable PGR 17 41 CC[C@@H](NC(=O)c1ccc([N+](=O)[O-])cc1)c1ccc(C)c(C)c1 ZINC000217862828 DI In-Stock Unstable AR 0 42 CC[C@@H](NC(=O)c1ccc([N+](=O)[O-])cc1)c1ccc(C)c(C)c1 ZINC000217862828 DI In-Stock Unstable UTS2 64 37 O=C(O)/C=C\c1ccc(COc2ccc(F)cc2)cc1 ZINC000217862862 CH For-Sale Unstable MAOB 19 70 O=C(O)/C=C\c1ccc(COc2ccc(F)cc2)cc1 ZINC000217862862 CH For-Sale Unstable PTGER2 37 46 O=C(O)/C=C\c1ccc(COc2ccc(F)cc2)cc1 ZINC000217862862 CH For-Sale Unstable PTGER4 26 46 O=C(O)/C=C\c1ccc(COc2ccc(F)cc2)cc1 ZINC000217862862 CH For-Sale Unstable PTPN2 0 46 O=C(O)/C=C\c1ccc(COc2ccc(F)cc2)cc1 ZINC000217862862 CH For-Sale Unstable PTGER3 17 46 O=C(O)/C=C\c1ccc(COc2ccc(F)cc2)cc1 ZINC000217862862 CH For-Sale Unstable CDC25B 0 45 O=C(O)/C=C\c1ccc(COc2ccc(F)cc2)cc1 ZINC000217862862 CH For-Sale Unstable ACE2 15 43 O=C(O)/C=C\c1ccc(COc2ccc(F)cc2)cc1 ZINC000217862862 CH For-Sale Unstable PTGDR 0 46 O=C(O)/C=C\c1ccc(COc2ccc(F)cc2)cc1 ZINC000217862862 CH For-Sale Unstable FFAR1 39 50 O=C(O)/C=C\c1ccc(COc2ccc(F)cc2)cc1 ZINC000217862862 CH For-Sale Unstable AKR1C3 35 54 O=C(O)/C=C\c1ccc(COc2ccc(F)cc2)cc1 ZINC000217862862 CH For-Sale Unstable ENPP2 47 43 O=C(O)/C=C\c1ccc(COc2ccc(F)cc2)cc1 ZINC000217862862 CH For-Sale Unstable FFAR4 42 42 O=C(O)/C=C\c1ccc(COc2ccc(F)cc2)cc1 ZINC000217862862 CH For-Sale Unstable HPGD 24 40 O=C(NCCn1ccnc1-c1ccccn1)NCc1ccc(Cl)cc1 ZINC000217862875 FG In-Stock Unstable GPR39 0 47 CN1CCN(C)[C@@H](Cc2ncnn2-c2cccc(C(F)(F)F)c2)C1 ZINC000217862879 EE In-Stock Unstable CHRNA10 17 43 CC[C@H](NC(=O)c1ccc([N+](=O)[O-])cc1)c1ccc(C)c(C)c1 ZINC000217862898 DI In-Stock Unstable PGR 17 41 CC[C@H](NC(=O)c1ccc([N+](=O)[O-])cc1)c1ccc(C)c(C)c1 ZINC000217862898 DI In-Stock Unstable AR 0 42 CC[C@H](NC(=O)c1ccc([N+](=O)[O-])cc1)c1ccc(C)c(C)c1 ZINC000217862898 DI In-Stock Unstable CCR3 0 47 CC[C@H](NC(=O)c1ccc([N+](=O)[O-])cc1)c1ccc(C)c(C)c1 ZINC000217862898 DI In-Stock Unstable UTS2 64 37 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccccc1Br ZINC000217862939 GG For-Sale Unstable NPY1R 44 35 NC(=O)CC[C@H](NC(=O)[C@@H]1C[C@H]2CCCC[C@@H]2N1)C(=O)O ZINC000217862960 CB For-Sale Unstable SLC5A1 20 46 O=C(O)/C=C\c1ccc(COc2ccc(F)cc2)c(F)c1 ZINC000217862968 CH For-Sale Unstable CDC25B 24 47 O=C(O)/C=C\c1ccc(COc2ccc(F)cc2)c(F)c1 ZINC000217862968 CH For-Sale Unstable FFAR1 17 41 O=C(O)/C=C\c1ccc(COc2ccc(F)cc2)c(F)c1 ZINC000217862968 CH For-Sale Unstable AKR1C3 33 47 O=C(O)/C=C\c1ccc(COc2ccc(F)cc2)c(F)c1 ZINC000217862968 CH For-Sale Unstable FFAR4 42 41 COc1ccc(CNC(=O)NCCn2ccnc2-c2ccccn2)cc1OC ZINC000217862974 GE In-Stock Unstable DRTS_TRYCR 45 31 CC[C@@H](C)N(C)CCNC(=O)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217862975 DF On-Demand Unstable GSTM2 25 41 CC[C@@H](NC(=O)c1ccc([N+](=O)[O-])cc1)c1ccc(C)cc1C ZINC000217863014 DI In-Stock Unstable PGR 15 40 CC[C@@H](NC(=O)c1ccc([N+](=O)[O-])cc1)c1ccc(C)cc1C ZINC000217863014 DI In-Stock Unstable AR 0 42 CC[C@@H](NC(=O)c1ccc([N+](=O)[O-])cc1)c1ccc(C)cc1C ZINC000217863014 DI In-Stock Unstable TRPA1 15 47 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1Br ZINC000217863016 GG For-Sale Unstable NPY1R 44 35 CC[C@H](C)N(C)CCNC(=O)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217863029 DF On-Demand Unstable GSTM2 25 41 COC(=O)c1c(O)c(O)cn1Cc1ccccc1 ZINC000217863059 BD For-Sale Unstable MAPK8 18 46 COC(=O)c1c(O)c(O)cn1Cc1ccccc1 ZINC000217863059 BD For-Sale Unstable FAS 40 35 C[C@H]1CCC[C@@H](C)N1Cc1ccccc1/C=C\C(=O)O ZINC000217863060 CH For-Sale Unstable PTGER2 44 47 C[C@H]1CCC[C@@H](C)N1Cc1ccccc1/C=C\C(=O)O ZINC000217863060 CH For-Sale Unstable PTGER4 0 47 C[C@H]1CCC[C@@H](C)N1Cc1ccccc1/C=C\C(=O)O ZINC000217863060 CH For-Sale Unstable PTGER3 17 48 C[C@H]1CCC[C@@H](C)N1Cc1ccccc1/C=C\C(=O)O ZINC000217863060 CH For-Sale Unstable PTGDR 0 48 O=C(NCCn1ccnc1-c1ccccn1)Nc1ccc(C(F)(F)F)cc1 ZINC000217863068 GH In-Stock Unstable TRPV1 18 43 O=C(NCCn1ccnc1-c1ccccn1)Nc1ccc(C(F)(F)F)cc1 ZINC000217863068 GH In-Stock Unstable P2RY1 32 40 O=C(NCCn1ccnc1-c1ccccn1)Nc1ccc(C(F)(F)F)cc1 ZINC000217863068 GH In-Stock Unstable FLT1 17 47 O=C(NCCn1ccnc1-c1ccccn1)Nc1ccc(C(F)(F)F)cc1 ZINC000217863068 GH In-Stock Unstable EPHX2 32 44 O=C(NCCn1ccnc1-c1ccccn1)Nc1ccc(C(F)(F)F)cc1 ZINC000217863068 GH In-Stock Unstable SLC11A2 23 43 CC[C@H](NC(=O)c1ccc([N+](=O)[O-])cc1)c1ccc(C)cc1C ZINC000217863098 DI In-Stock Unstable PGR 15 40 CC[C@H](NC(=O)c1ccc([N+](=O)[O-])cc1)c1ccc(C)cc1C ZINC000217863098 DI In-Stock Unstable AR 0 42 CC[C@H](NC(=O)c1ccc([N+](=O)[O-])cc1)c1ccc(C)cc1C ZINC000217863098 DI In-Stock Unstable TRPA1 15 47 CCOc1ccc(CC(=O)NC[C@@H]2CCCN3CCCC[C@H]23)cc1 ZINC000217863105 EG In-Stock Unstable CACNA1I 21 41 CCOc1ccc(CC(=O)NC[C@@H]2CCCN3CCCC[C@H]23)cc1 ZINC000217863105 EG In-Stock Unstable HCN1 41 33 CCOc1ccc(CC(=O)NC[C@@H]2CCCN3CCCC[C@H]23)cc1 ZINC000217863105 EG In-Stock Unstable HCN4 42 35 O=C(NCCc1ccccc1F)C(F)F ZINC000217863164 BD On-Demand Unstable CXCL8 23 40 O=C(NCCc1ccccc1F)C(F)F ZINC000217863164 BD On-Demand Unstable NQO2 39 40 O=C(NCCc1ccccc1F)C(F)F ZINC000217863164 BD On-Demand Unstable CPA1 21 41 O=C(NCCc1ccccc1F)C(F)F ZINC000217863164 BD On-Demand Unstable MTNR1A 48 40 O=C(NCCc1ccccc1F)C(F)F ZINC000217863164 BD On-Demand Unstable TAAR1 20 59 CC[C@@H](NC(=O)c1ccc([N+](=O)[O-])cc1)c1ccc(OC)c(OC)c1 ZINC000217863224 EG In-Stock Unstable PGR 15 42 CC[C@@H](NC(=O)c1ccc([N+](=O)[O-])cc1)c1ccc(OC)c(OC)c1 ZINC000217863224 EG In-Stock Unstable AR 0 48 CC[C@@H](NC(=O)c1ccc([N+](=O)[O-])cc1)c1ccc(OC)c(OC)c1 ZINC000217863224 EG In-Stock Unstable CCR3 0 46 CC[C@@H](NC(=O)c1ccc([N+](=O)[O-])cc1)c1ccc(OC)c(OC)c1 ZINC000217863224 EG In-Stock Unstable KCNMA1 24 41 CC[C@@H](NC(=O)c1ccc([N+](=O)[O-])cc1)c1ccc(OC)c(OC)c1 ZINC000217863224 EG In-Stock Unstable UTS2 56 38 CC[C@H](NC(=O)c1ccc([N+](=O)[O-])cc1)c1ccc(OC)c(OC)c1 ZINC000217863302 EG In-Stock Unstable PGR 15 42 CC[C@H](NC(=O)c1ccc([N+](=O)[O-])cc1)c1ccc(OC)c(OC)c1 ZINC000217863302 EG In-Stock Unstable AR 0 48 CC[C@H](NC(=O)c1ccc([N+](=O)[O-])cc1)c1ccc(OC)c(OC)c1 ZINC000217863302 EG In-Stock Unstable CCR3 0 46 CC[C@H](NC(=O)c1ccc([N+](=O)[O-])cc1)c1ccc(OC)c(OC)c1 ZINC000217863302 EG In-Stock Unstable KCNMA1 24 41 CC[C@H](NC(=O)c1ccc([N+](=O)[O-])cc1)c1ccc(OC)c(OC)c1 ZINC000217863302 EG In-Stock Unstable UTS2 56 38 CSC[C@@](C)(O)CNCc1ccc(F)c(C)c1 ZINC000217863312 CE On-Demand Unstable LEF 31 43 CSC[C@](C)(O)CNCc1ccc(F)c(C)c1 ZINC000217863352 CE On-Demand Unstable LEF 31 43 COc1cccc(C(=O)C(Cl)Cl)c1 ZINC000217863361 BF For-Sale Unstable DRD4 50 38 COc1cccc(C(=O)C(Cl)Cl)c1 ZINC000217863361 BF For-Sale Unstable MTNR1A 37 44 COc1cccc(C(=O)C(Cl)Cl)c1 ZINC000217863361 BF For-Sale Unstable MTNR1B 39 46 COc1cccc(C(=O)C(Cl)Cl)c1 ZINC000217863361 BF For-Sale Unstable TUBB2B 50 49 COc1cccc(C(=O)C(Cl)Cl)c1 ZINC000217863361 BF For-Sale Unstable HSD17B2 25 43 COc1cccc(C(=O)C(Cl)Cl)c1 ZINC000217863361 BF For-Sale Unstable TAAR1 33 45 COc1cccc(C(=O)C(Cl)Cl)c1 ZINC000217863361 BF For-Sale Unstable AKR1C3 29 43 COc1cccc(C(=O)C(Cl)Cl)c1 ZINC000217863361 BF For-Sale Unstable KCNK3 23 49 COCCNC(=O)NCCn1ccnc1-c1ccccn1 ZINC000217863364 CC In-Stock Unstable ACAT 0 40 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217863375 HF For-Sale Unstable CA2 105 60 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217863375 HF For-Sale Unstable CA6 17 40 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217863375 HF For-Sale Unstable CA1 93 60 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217863375 HF For-Sale Unstable CA7 55 57 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217863375 HF For-Sale Unstable CA13 22 40 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217863375 HF For-Sale Unstable CA5B 63 57 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217863375 HF For-Sale Unstable CA4 67 58 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217863375 HF For-Sale Unstable CA5A 65 57 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217863375 HF For-Sale Unstable CA14 40 54 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217863375 HF For-Sale Unstable CA12 72 60 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217863375 HF For-Sale Unstable CA9 82 60 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217863375 HF For-Sale Unstable CYNT 26 45 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217863375 HF For-Sale Unstable NCE103 35 55 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217863375 HF For-Sale Unstable LIG1 0 51 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217863375 HF For-Sale Unstable MTCA1 43 40 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217863375 HF For-Sale Unstable P96878_MYCTU 56 44 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217863375 HF For-Sale Unstable CA 0 41 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217863375 HF For-Sale Unstable A6YCJ1_9METZ 25 51 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217863375 HF For-Sale Unstable Q5TU56_ANOGA 0 40 CC[C@@H](NC(=O)c1ccc([N+](=O)[O-])cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217863397 FF In-Stock Unstable PGR 18 40 CC[C@@H](NC(=O)c1ccc([N+](=O)[O-])cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217863397 FF In-Stock Unstable CCR3 24 45 CC[C@H](NC(=O)c1ccc([N+](=O)[O-])cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217863432 FF In-Stock Unstable PGR 18 40 CC[C@H](NC(=O)c1ccc([N+](=O)[O-])cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217863432 FF In-Stock Unstable CCR3 24 45 COC(=O)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217863468 FE For-Sale Unstable TBXA2R 17 40 COC(=O)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217863468 FE For-Sale Unstable NPY2R 55 36 COC(=O)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217863468 FE For-Sale Unstable ADAMTS5 38 42 COC(=O)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217863468 FE For-Sale Unstable SFRP1 119 36 COC(=O)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217863468 FE For-Sale Unstable WNT3 82 33 O=S(=O)(NCCn1ccnc1-c1ccccn1)c1ccc2c(c1)OCCO2 ZINC000217863487 GD In-Stock Unstable PKM 33 45 Cc1cc(C)c(-c2csc(NC(=O)CSc3nnc(C(C)(C)C)[nH]3)n2)cc1C ZINC000217863491 HJ On-Demand Unstable ENPP1 69 35 N#CCOc1ccc(NC(=O)C(F)F)cc1 ZINC000217863494 BD For-Sale Unstable DHODH 44 33 O=C(N/C=C/c1ccccc1Br)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217863502 JK For-Sale Anodyne PTPA 0 45 CC[C@@H](C)N(C)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217863572 CG For-Sale Unstable TUBB1 49 40 CC[C@@H](C)N(C)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217863572 CG For-Sale Unstable AKR1C3 31 42 COC(=O)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217863587 FE For-Sale Unstable TBXA2R 17 40 COC(=O)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217863587 FE For-Sale Unstable NPY2R 55 36 COC(=O)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217863587 FE For-Sale Unstable ADAMTS5 38 42 COC(=O)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217863587 FE For-Sale Unstable SFRP1 119 36 COC(=O)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217863587 FE For-Sale Unstable WNT3 82 33 Cc1ccc(-c2noc(CNC(=O)c3ccc([N+](=O)[O-])cc3)n2)cc1 ZINC000217863634 EF In-Stock Unstable KCNQ1 0 42 CC[C@H](C)N(C)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217863638 CG For-Sale Unstable TUBB1 49 40 CC[C@H](C)N(C)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217863638 CG For-Sale Unstable AKR1C3 31 42 O=S(=O)(Cc1ccc(C(F)(F)F)cc1)NC[C@H]1CCCN1c1ccccc1 ZINC000217863709 GH For-Sale Unstable ADAMTS5 30 49 COc1cccc(-c2noc(CNC(=O)c3ccc([N+](=O)[O-])cc3)n2)c1 ZINC000217863732 FF In-Stock Unstable DRD4 40 31 COc1cccc(-c2noc(CNC(=O)c3ccc([N+](=O)[O-])cc3)n2)c1 ZINC000217863732 FF In-Stock Unstable U38 0 45 CCCN(Cc1cc(/C=C\C(=O)O)ccc1OC)C(C)C ZINC000217863739 CG For-Sale Unstable AKR1C3 30 41 O=S(=O)(Cc1ccc(C(F)(F)F)cc1)NC[C@@H]1CCCN1c1ccccc1 ZINC000217863796 GH For-Sale Unstable ADAMTS5 30 49 O=C(c1ccccc1-c1ccc(F)cc1)N1CCC[C@@H](c2ccncn2)C1 ZINC000217863817 FI In-Stock Unstable HCRTR1 23 43 O=C(c1ccccc1-c1ccc(F)cc1)N1CCC[C@@H](c2ccncn2)C1 ZINC000217863817 FI In-Stock Unstable MLNR 18 43 O=C(c1ccccc1-c1ccc(F)cc1)N1CCC[C@@H](c2ccncn2)C1 ZINC000217863817 FI In-Stock Unstable HCRTR2 23 43 O=C(c1ccccc1-c1ccc(F)cc1)N1CCC[C@@H](c2ccncn2)C1 ZINC000217863817 FI In-Stock Unstable SLC6A7 0 42 O=C(O)CCSS(=O)(=O)O ZINC000217863849 AB For-Sale Unstable ASD 0 43 COc1ccc(-c2noc(CNC(=O)c3ccc([N+](=O)[O-])cc3)n2)c(OC)c1 ZINC000217863855 GF In-Stock Unstable MT-ND1 17 42 COc1ccc(-c2noc(CNC(=O)c3ccc([N+](=O)[O-])cc3)n2)c(OC)c1 ZINC000217863855 GF In-Stock Unstable U38 0 46 COc1ccc(-c2noc(CNC(=O)c3ccc([N+](=O)[O-])cc3)n2)c(OC)c1 ZINC000217863855 GF In-Stock Unstable ABCG2 26 42 CCCN(Cc1ccc(OC)c(/C=C\C(=O)O)c1)C(C)C ZINC000217863861 CG For-Sale Unstable PTGER2 26 41 CCCN(Cc1ccc(OC)c(/C=C\C(=O)O)c1)C(C)C ZINC000217863861 CG For-Sale Unstable PTGER4 0 41 O=C(c1ccccc1-c1ccc(F)cc1)N1CCC[C@H](c2ccncn2)C1 ZINC000217863903 FI In-Stock Unstable HCRTR1 23 43 O=C(c1ccccc1-c1ccc(F)cc1)N1CCC[C@H](c2ccncn2)C1 ZINC000217863903 FI In-Stock Unstable MLNR 18 43 O=C(c1ccccc1-c1ccc(F)cc1)N1CCC[C@H](c2ccncn2)C1 ZINC000217863903 FI In-Stock Unstable HCRTR2 23 43 O=C(c1ccccc1-c1ccc(F)cc1)N1CCC[C@H](c2ccncn2)C1 ZINC000217863903 FI In-Stock Unstable SLC6A7 0 42 CCOc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217863921 FG For-Sale Unstable NPY2R 54 36 CCOc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217863921 FG For-Sale Unstable CHRNA10 40 39 CCOc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217863921 FG For-Sale Unstable ADAMTS5 36 44 O=C(N/C=C/c1ccccc1Br)Nc1ccc(F)c(Cl)c1 ZINC000217863922 FK For-Sale Anodyne P95276_MYCTO 0 42 CCOc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217863982 FG For-Sale Unstable CHRNA10 40 39 CCOc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217863982 FG For-Sale Unstable ADAMTS5 30 44 O=C(NCc1nc(-c2cccc(Br)c2)no1)c1ccc([N+](=O)[O-])cc1 ZINC000217864001 HG In-Stock Unstable U38 0 40 O=C(N/C=C/c1ccccc1Br)NCc1ccc(F)cc1 ZINC000217864012 EI For-Sale Unstable AMP1_PLAFQ 16 44 CCN(C)C(=O)CNC(=O)c1ccc(Cl)c(N)c1 ZINC000217864048 CD For-Sale Unstable CA2 19 43 CCN(C)C(=O)CNC(=O)c1ccc(Cl)c(N)c1 ZINC000217864048 CD For-Sale Unstable PYGL 23 40 SCCCCCCCCCN1CCN2CCCC[C@@H]2C1 ZINC000217864050 CH For-Sale Unstable EBP 15 46 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2Br)CC1 ZINC000217864099 HH For-Sale Unstable HTR1A 87 50 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2Br)CC1 ZINC000217864099 HH For-Sale Unstable DRD2 64 48 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2Br)CC1 ZINC000217864099 HH For-Sale Unstable DRD4 34 46 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2Br)CC1 ZINC000217864099 HH For-Sale Unstable ADRA1D 61 39 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2Br)CC1 ZINC000217864099 HH For-Sale Unstable HTR1D 23 42 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2Br)CC1 ZINC000217864099 HH For-Sale Unstable HTR1B 18 50 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2Br)CC1 ZINC000217864099 HH For-Sale Unstable HTR2A 34 43 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2Br)CC1 ZINC000217864099 HH For-Sale Unstable ADRA1A 56 39 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2Br)CC1 ZINC000217864099 HH For-Sale Unstable ADRA1B 50 39 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2Br)CC1 ZINC000217864099 HH For-Sale Unstable DRD3 70 48 COc1ccccc1N1CCN(C(=O)N/C=C/c2ccccc2Br)CC1 ZINC000217864099 HH For-Sale Unstable HTR7 56 43 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc(F)cc1F ZINC000217864101 FF For-Sale Unstable NPY2R 40 35 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCc1cccc(Cl)c1Cl ZINC000217864102 DK For-Sale Unstable TRPM8 16 46 CC[C@@H](C)[C@@H](CO)NC(=O)[C@H](Cc1ccccc1)N1Cc2ccccc2C1=O ZINC000217864116 GF In-Stock Unstable MME 68 41 CC[C@@H](C)[C@@H](CO)NC(=O)[C@H](Cc1ccccc1)N1Cc2ccccc2C1=O ZINC000217864116 GF In-Stock Unstable CTSB 19 44 CC[C@@H](C)[C@@H](CO)NC(=O)[C@H](Cc1ccccc1)N1Cc2ccccc2C1=O ZINC000217864116 GF In-Stock Unstable PAPA1_CARPA 40 31 CC[C@@H](C)[C@@H](CO)NC(=O)[C@H](Cc1ccccc1)N1Cc2ccccc2C1=O ZINC000217864116 GF In-Stock Unstable REN 18 48 CC[C@@H](C)[C@@H](CO)NC(=O)[C@H](Cc1ccccc1)N1Cc2ccccc2C1=O ZINC000217864116 GF In-Stock Unstable ACE2 58 39 CC[C@@H](C)[C@@H](CO)NC(=O)[C@H](Cc1ccccc1)N1Cc2ccccc2C1=O ZINC000217864116 GF In-Stock Unstable POL 0 40 CC[C@@H](C)[C@@H](CO)NC(=O)[C@H](Cc1ccccc1)N1Cc2ccccc2C1=O ZINC000217864116 GF In-Stock Unstable DERP1 0 44 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable ACE 94 51 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable FOLH1 79 53 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable MME 134 57 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable LTA4H 29 40 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable ANPEP 106 44 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable CTSB 29 43 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable PAPA1_CARPA 40 35 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable CCKAR 56 47 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable CTSK 19 43 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable CTSL 33 43 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable CPA1 59 45 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable TIMP3 66 36 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable HDAC8 24 40 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable CTRB1 26 40 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable NAALAD2 81 52 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable MMP2 40 55 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable MMP3 78 55 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable MMP8 22 40 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable HDAC1 15 40 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable CCKBR 18 47 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable CTSS 15 43 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable CAPN1 36 41 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable MMP9 26 57 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable CAPN2 33 40 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable EPHX2 15 48 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable ACE2 76 47 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable HDAC11 41 34 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable LAP3 63 39 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable MMP1 34 57 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable FPR1 69 60 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable NPR 51 39 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable AMP1_PLAFQ 51 42 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable BLA1_STEMA 74 36 O=C(Nc1ccccc1)N[C@@H](CCc1ccccc1)C(=O)O ZINC000217864121 CF For-Sale Unstable NCE103 21 42 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCc1cccc(Cl)c1Cl ZINC000217864169 DK For-Sale Unstable TRPM8 16 46 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc(F)cc1F ZINC000217864172 FF For-Sale Unstable NPY2R 40 35 COC1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217864188 CE For-Sale Unstable SIGMAR1 36 41 COC1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217864188 CE For-Sale Unstable PTGER3 22 45 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCc1cccc(Cl)c1Cl ZINC000217864256 DK For-Sale Unstable TRPM8 16 46 CN(Cc1cc(-c2ccccc2)on1)C(=O)c1nc2ccccc2c(=O)[nH]1 ZINC000217864262 FF In-Stock Unstable TSPO 36 40 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1cc(F)cc(F)c1 ZINC000217864292 FF For-Sale Unstable HTR7 17 40 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1cc(F)cc(F)c1 ZINC000217864292 FF For-Sale Unstable ADAMTS5 38 43 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1cc(F)cc(F)c1 ZINC000217864292 FF For-Sale Unstable SFRP1 60 33 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1cc(F)cc(F)c1 ZINC000217864292 FF For-Sale Unstable WNT3 47 33 COC1CCN(Cc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217864296 CE For-Sale Unstable DRD2 17 41 COC1CCN(Cc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217864296 CE For-Sale Unstable DRD4 43 38 COC1CCN(Cc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217864296 CE For-Sale Unstable OPRK1 17 44 COC1CCN(Cc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217864296 CE For-Sale Unstable SIGMAR1 50 52 CN(Cc1ccc2ccccc2c1)C(=O)C(F)F ZINC000217864300 BG On-Demand Unstable ALOX5 16 49 CN(Cc1ccc2ccccc2c1)C(=O)C(F)F ZINC000217864300 BG On-Demand Unstable TACR1 15 43 CN(Cc1ccc2ccccc2c1)C(=O)C(F)F ZINC000217864300 BG On-Demand Unstable MTTP 40 33 CN(Cc1ccc2ccccc2c1)C(=O)C(F)F ZINC000217864300 BG On-Demand Unstable CYP2A5 0 43 CSC[C@@](C)(O)CNCc1cccc([N+](=O)[O-])c1 ZINC000217864314 CD On-Demand Unstable CACNA1C 49 37 CSC[C@@](C)(O)CNCc1cccc([N+](=O)[O-])c1 ZINC000217864314 CD On-Demand Unstable CACNA1D 82 37 O=S(=O)(NCCn1ccnc1-c1ccccn1)c1ccc(F)c(Cl)c1 ZINC000217864332 GF In-Stock Unstable HTR7 19 46 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCc1cccc(Cl)c1Cl ZINC000217864336 DK For-Sale Unstable TRPM8 16 46 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1cc(F)cc(F)c1 ZINC000217864371 FF For-Sale Unstable HTR7 17 40 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1cc(F)cc(F)c1 ZINC000217864371 FF For-Sale Unstable ADAMTS5 38 43 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1cc(F)cc(F)c1 ZINC000217864371 FF For-Sale Unstable SFRP1 60 33 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1cc(F)cc(F)c1 ZINC000217864371 FF For-Sale Unstable WNT3 47 33 CSC[C@](C)(O)CNCc1cccc([N+](=O)[O-])c1 ZINC000217864382 CD On-Demand Unstable CACNA1C 49 37 CSC[C@](C)(O)CNCc1cccc([N+](=O)[O-])c1 ZINC000217864382 CD On-Demand Unstable CACNA1D 82 37 O=C(CN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCCc1c[nH]cn1 ZINC000217864396 HD In-Stock Unstable HRH1 17 40 O=C(CN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCCc1c[nH]cn1 ZINC000217864396 HD In-Stock Unstable HRH3 42 46 COC1CCN(Cc2ccc(/C=C\C(=O)O)cc2F)CC1 ZINC000217864401 CF For-Sale Unstable CCR2 54 40 Cc1ccc(CN[C@H]2C[C@H](C)CC[C@H]2C(C)C)c(C)c1 ZINC000217864452 CJ For-Sale Unstable TRPM8 16 46 O=C(CN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCCc1c[nH]cn1 ZINC000217864476 HD In-Stock Unstable HRH1 17 40 O=C(CN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCCc1c[nH]cn1 ZINC000217864476 HD In-Stock Unstable HRH3 42 46 O=C(N/C=C/c1ccccc1Br)NC1CCCCCC1 ZINC000217864479 EI For-Sale Unstable EPHX2 24 48 O=C(O)CC[C@H](NC(=O)[C@@H]1C[C@H]2CCCC[C@@H]2N1)C(=O)O ZINC000217864497 CC For-Sale Unstable FOLH1 41 43 O=C(O)CC[C@H](NC(=O)[C@@H]1C[C@H]2CCCC[C@@H]2N1)C(=O)O ZINC000217864497 CC For-Sale Unstable NAALAD2 53 43 Cc1ccc(CN[C@H]2C[C@@H](C)CC[C@H]2C(C)C)c(C)c1 ZINC000217864515 CJ For-Sale Unstable TRPM8 16 46 CC(C)c1ccc(CCCNC(=O)c2ccc([N+](=O)[O-])cc2)cc1 ZINC000217864579 EI In-Stock Unstable CCR3 0 40 CC(C)c1ccc(CCCNC(=O)c2ccc([N+](=O)[O-])cc2)cc1 ZINC000217864579 EI In-Stock Unstable COLA 27 45 CC(C)c1ccc(CCCNC(=O)c2ccc([N+](=O)[O-])cc2)cc1 ZINC000217864579 EI In-Stock Unstable HDA106 0 53 CC[C@@H]1CN(Cc2ccccc2/C=C\C(=O)O)CCO1 ZINC000217864586 CE For-Sale Unstable PTGER2 40 42 CC[C@@H]1CN(Cc2ccccc2/C=C\C(=O)O)CCO1 ZINC000217864586 CE For-Sale Unstable PTGER4 18 42 CC[C@@H]1CN(Cc2ccccc2/C=C\C(=O)O)CCO1 ZINC000217864586 CE For-Sale Unstable PTGER3 15 42 CC[C@@H]1CN(Cc2ccccc2/C=C\C(=O)O)CCO1 ZINC000217864586 CE For-Sale Unstable PTGDR 15 41 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCc1ccc(O)cc1 ZINC000217864628 CH For-Sale Unstable TRPM8 17 46 CC[C@H]1CN(Cc2ccccc2/C=C\C(=O)O)CCO1 ZINC000217864671 CE For-Sale Unstable PTGER2 40 42 CC[C@H]1CN(Cc2ccccc2/C=C\C(=O)O)CCO1 ZINC000217864671 CE For-Sale Unstable PTGER4 18 42 CC[C@H]1CN(Cc2ccccc2/C=C\C(=O)O)CCO1 ZINC000217864671 CE For-Sale Unstable PTGER3 15 42 CC[C@H]1CN(Cc2ccccc2/C=C\C(=O)O)CCO1 ZINC000217864671 CE For-Sale Unstable PTGDR 15 41 CCC[C@@H](O)CNCCc1cccs1 ZINC000217864677 BE For-Sale Unstable ADAM17 0 46 O=C(NCCCN1CCCc2ccccc21)c1ccc([N+](=O)[O-])cc1 ZINC000217864693 EG In-Stock Unstable DRD2 22 40 O=C(NCCCN1CCCc2ccccc21)c1ccc([N+](=O)[O-])cc1 ZINC000217864693 EG In-Stock Unstable ADRA1D 20 43 O=C(NCCCN1CCCc2ccccc21)c1ccc([N+](=O)[O-])cc1 ZINC000217864693 EG In-Stock Unstable HTR1D 23 43 O=C(NCCCN1CCCc2ccccc21)c1ccc([N+](=O)[O-])cc1 ZINC000217864693 EG In-Stock Unstable AVPR2 29 46 O=C(NCCCN1CCCc2ccccc21)c1ccc([N+](=O)[O-])cc1 ZINC000217864693 EG In-Stock Unstable ADRA1A 32 42 O=C(NCCCN1CCCc2ccccc21)c1ccc([N+](=O)[O-])cc1 ZINC000217864693 EG In-Stock Unstable ADRA1B 26 43 O=C(NCCCN1CCCc2ccccc21)c1ccc([N+](=O)[O-])cc1 ZINC000217864693 EG In-Stock Unstable DRD3 34 40 O=C(NCCCN1CCCc2ccccc21)c1ccc([N+](=O)[O-])cc1 ZINC000217864693 EG In-Stock Unstable ADRA2B 23 43 O=C(NCCCN1CCCc2ccccc21)c1ccc([N+](=O)[O-])cc1 ZINC000217864693 EG In-Stock Unstable ADRA2C 18 43 O=C(N/C=C/c1ccccc1Br)Nc1cc(Cl)cc(Cl)c1 ZINC000217864694 GK For-Sale Anodyne PPIA 16 42 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1cccc(F)c1 ZINC000217864700 EF For-Sale Unstable NPY2R 47 39 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1cccc(F)c1 ZINC000217864700 EF For-Sale Unstable HTR6 40 39 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1cccc(F)c1 ZINC000217864700 EF For-Sale Unstable ADAMTS5 36 42 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1cccc(F)c1 ZINC000217864700 EF For-Sale Unstable SFRP1 90 35 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1cccc(F)c1 ZINC000217864700 EF For-Sale Unstable WNT3 68 32 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCc1ccc(O)cc1 ZINC000217864723 CH For-Sale Unstable TRPM8 17 46 CC(=O)N1CCN(Cc2ccc(OCCCn3ccnc3)cc2)CC1 ZINC000217864751 EE In-Stock Unstable CYP11B1 41 39 CC(=O)N1CCN(Cc2ccc(OCCCn3ccnc3)cc2)CC1 ZINC000217864751 EE In-Stock Unstable LTA4H 41 37 CC(=O)N1CCN(Cc2ccc(OCCCn3ccnc3)cc2)CC1 ZINC000217864751 EE In-Stock Unstable TBXAS1 69 52 CC(=O)N1CCN(Cc2ccc(OCCCn3ccnc3)cc2)CC1 ZINC000217864751 EE In-Stock Unstable HRH3 48 45 CC(=O)N1CCN(Cc2ccc(OCCCn3ccnc3)cc2)CC1 ZINC000217864751 EE In-Stock Unstable CYP11B2 46 39 CC(=O)N1CCN(Cc2ccc(OCCCn3ccnc3)cc2)CC1 ZINC000217864751 EE In-Stock Unstable FAAH 23 41 CC(=O)N1CCN(Cc2ccc(OCCCn3ccnc3)cc2)CC1 ZINC000217864751 EE In-Stock Unstable HMOX1 56 52 CC(=O)N1CCN(Cc2ccc(OCCCn3ccnc3)cc2)CC1 ZINC000217864751 EE In-Stock Unstable CYP17A1 22 41 CC(=O)N1CCN(Cc2ccc(OCCCn3ccnc3)cc2)CC1 ZINC000217864751 EE In-Stock Unstable HMOX2 60 51 CC(=O)N1CCN(Cc2ccc(OCCCn3ccnc3)cc2)CC1 ZINC000217864751 EE In-Stock Unstable MGLL 0 50 CC(=O)N1CCN(Cc2ccc(OCCCn3ccnc3)cc2)CC1 ZINC000217864751 EE In-Stock Unstable QPCT 39 41 O=S(=O)(NCCn1ccnc1-c1ccccn1)c1ccc2c(c1)CCCC2 ZINC000217864762 GF In-Stock Unstable HTR7 16 43 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1cccc(F)c1 ZINC000217864776 EF For-Sale Unstable NPY2R 47 39 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1cccc(F)c1 ZINC000217864776 EF For-Sale Unstable ADAMTS5 36 42 CC[C@@H]1CN(Cc2ccc(/C=C\C(=O)O)cc2)CCO1 ZINC000217864780 CE For-Sale Unstable DRD4 28 49 CC[C@@H]1CN(Cc2ccc(/C=C\C(=O)O)cc2)CCO1 ZINC000217864780 CE For-Sale Unstable SIGMAR1 20 43 CCC[C@H](O)CNCCc1cccs1 ZINC000217864795 BE For-Sale Unstable ADAM17 0 46 COc1ccc(CNC(=O)c2cccc([N+](=O)[O-])c2)c(OC)c1OC ZINC000217864799 EF In-Stock Unstable DRD4 41 31 COc1ccc(CNC(=O)c2cccc([N+](=O)[O-])c2)c(OC)c1OC ZINC000217864799 EF In-Stock Unstable CACNA1C 52 37 COc1ccc(CNC(=O)c2cccc([N+](=O)[O-])c2)c(OC)c1OC ZINC000217864799 EF In-Stock Unstable CACNA1D 86 37 COc1ccc(CNC(=O)c2cccc([N+](=O)[O-])c2)c(OC)c1OC ZINC000217864799 EF In-Stock Unstable PYGL 22 41 COc1ccc(CNC(=O)c2cccc([N+](=O)[O-])c2)c(OC)c1OC ZINC000217864799 EF In-Stock Unstable PPARD 15 43 COc1ccc(CNC(=O)c2cccc([N+](=O)[O-])c2)c(OC)c1OC ZINC000217864799 EF In-Stock Unstable SLC9A1 61 39 COc1ccc(CNC(=O)c2cccc([N+](=O)[O-])c2)c(OC)c1OC ZINC000217864799 EF In-Stock Unstable KCNMA1 19 42 COc1ccc(CNC(=O)c2cccc([N+](=O)[O-])c2)c(OC)c1OC ZINC000217864799 EF In-Stock Unstable E1 0 42 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCc1ccc(O)cc1 ZINC000217864824 CH For-Sale Unstable TRPM8 17 46 CC[C@H]1CN(Cc2ccc(/C=C\C(=O)O)cc2)CCO1 ZINC000217864873 CE For-Sale Unstable DRD4 28 49 CC[C@H]1CN(Cc2ccc(/C=C\C(=O)O)cc2)CCO1 ZINC000217864873 CE For-Sale Unstable SIGMAR1 20 43 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc2ccccc2c1 ZINC000217864886 FH For-Sale Unstable NPY1R 56 52 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc2ccccc2c1 ZINC000217864886 FH For-Sale Unstable NPY2R 56 52 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc2ccccc2c1 ZINC000217864886 FH For-Sale Unstable ADAMTS5 34 49 CCOc1ccc(CNC(=O)c2cccc([N+](=O)[O-])c2)cc1OCC ZINC000217864894 EG In-Stock Unstable TYMS 17 40 CCOc1ccc(CNC(=O)c2cccc([N+](=O)[O-])c2)cc1OCC ZINC000217864894 EG In-Stock Unstable CACNA1C 54 38 CCOc1ccc(CNC(=O)c2cccc([N+](=O)[O-])c2)cc1OCC ZINC000217864894 EG In-Stock Unstable CACNA1D 87 38 CCOc1ccc(CNC(=O)c2cccc([N+](=O)[O-])c2)cc1OCC ZINC000217864894 EG In-Stock Unstable CCR3 0 42 CCOc1ccc(CNC(=O)c2cccc([N+](=O)[O-])c2)cc1OCC ZINC000217864894 EG In-Stock Unstable PYGL 23 41 CCOc1ccc(CNC(=O)c2cccc([N+](=O)[O-])c2)cc1OCC ZINC000217864894 EG In-Stock Unstable U38 0 40 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCc1ccc(O)cc1 ZINC000217864903 CH For-Sale Unstable TRPM8 17 46 Cc1cc(C)cc(NC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217864914 EJ For-Sale Unstable KCNK3 42 35 Cc1ccccc1CCNC(=O)C(F)F ZINC000217864916 BD On-Demand Unstable ANPEP 18 41 COc1ccc(CN2C(=O)CNC2=O)cc1/C=C\C(=O)O ZINC000217864945 CC For-Sale Unstable PTGER2 28 41 COc1ccc(CN2C(=O)CNC2=O)cc1/C=C\C(=O)O ZINC000217864945 CC For-Sale Unstable PTGER4 0 41 COc1ccc(CN2C(=O)CNC2=O)cc1/C=C\C(=O)O ZINC000217864945 CC For-Sale Unstable PTGER3 18 41 COc1ccc(S(=O)(=O)NCCn2ccnc2-c2ccccn2)cc1F ZINC000217864962 GE In-Stock Unstable HTR7 16 42 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc2ccccc2c1 ZINC000217864968 FH For-Sale Unstable NPY1R 56 52 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc2ccccc2c1 ZINC000217864968 FH For-Sale Unstable NPY2R 56 52 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc2ccccc2c1 ZINC000217864968 FH For-Sale Unstable ADAMTS5 34 49 COc1ccccc1CCCNC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217865000 DF In-Stock Unstable DRD2 21 43 COc1ccccc1CCCNC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217865000 DF In-Stock Unstable DRD1 0 41 COc1ccccc1CCCNC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217865000 DF In-Stock Unstable DRD4 46 36 COc1ccccc1CCCNC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217865000 DF In-Stock Unstable ADRA1B 17 41 COc1ccccc1CCCNC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217865000 DF In-Stock Unstable DRD3 31 43 COc1ccccc1CCCNC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217865000 DF In-Stock Unstable CACNA1C 47 39 COc1ccccc1CCCNC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217865000 DF In-Stock Unstable CACNA1D 82 36 COc1ccccc1CCCNC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217865000 DF In-Stock Unstable PYGL 24 43 COc1ccccc1CCCNC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217865000 DF In-Stock Unstable MTNR1B 47 42 COc1ccccc1CCCNC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217865000 DF In-Stock Unstable KCNMA1 24 41 COc1ccccc1CCCNC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217865000 DF In-Stock Unstable ALPHA-1A 0 40 COc1cc(CN[C@H]2C[C@@H](C)CC[C@@H]2C(C)C)ccc1O ZINC000217865019 CH For-Sale Unstable TRPV1 0 74 COc1cc(CN[C@H]2C[C@@H](C)CC[C@@H]2C(C)C)ccc1O ZINC000217865019 CH For-Sale Unstable TRPM8 16 42 COc1ccc(OCCNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217865020 GH For-Sale Unstable MTNR1A 37 45 COc1ccc(OCCNC(=O)N/C=C/c2ccccc2Br)cc1 ZINC000217865020 GH For-Sale Unstable MTNR1B 28 45 O=C(NCCc1cccc(Cl)c1)C(F)F ZINC000217865061 BE On-Demand Unstable ANPEP 20 46 O=C(NCCc1cccc(Cl)c1)C(F)F ZINC000217865061 BE On-Demand Unstable CTSL 26 43 O=C(NCCc1cccc(Cl)c1)C(F)F ZINC000217865061 BE On-Demand Unstable CTSS 16 43 O=C(NCCc1cccc(Cl)c1)C(F)F ZINC000217865061 BE On-Demand Unstable CTSV 41 43 O=C(NCCc1cccc(Cl)c1)C(F)F ZINC000217865061 BE On-Demand Unstable AMP1_PLAFQ 44 41 O=C(NCCc1cccc(Cl)c1)C(F)F ZINC000217865061 BE On-Demand Unstable LEF 56 33 O=C(NCCc1cccc(Cl)c1)C(F)F ZINC000217865061 BE On-Demand Unstable HT1 0 53 O=C(NCCc1cccc(Cl)c1)C(F)F ZINC000217865061 BE On-Demand Unstable NCE103 29 41 O=C(NCCc1cccc(Cl)c1)C(F)F ZINC000217865061 BE On-Demand Unstable P96878_MYCTU 17 41 O=C(NCCc1cccc(Cl)c1)C(F)F ZINC000217865061 BE On-Demand Unstable CAN2 0 41 O=C(NCCc1cccc(Cl)c1)C(F)F ZINC000217865061 BE On-Demand Unstable PDS 58 38 O=C(NCCc1cccc(Cl)c1)C(F)F ZINC000217865061 BE On-Demand Unstable LMGT2 0 53 Cc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217865083 EF For-Sale Unstable NPY2R 41 40 Cc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217865083 EF For-Sale Unstable ADAMTS5 38 44 COc1cc(CN[C@H]2C[C@H](C)CC[C@@H]2C(C)C)ccc1O ZINC000217865107 CH For-Sale Unstable TRPV1 0 74 COc1cc(CN[C@H]2C[C@H](C)CC[C@@H]2C(C)C)ccc1O ZINC000217865107 CH For-Sale Unstable TRPM8 16 42 CCOc1ccc(CCCNC(=O)c2cccc([N+](=O)[O-])c2)cc1 ZINC000217865114 EG In-Stock Unstable DRD4 43 32 CCOc1ccc(CCCNC(=O)c2cccc([N+](=O)[O-])c2)cc1 ZINC000217865114 EG In-Stock Unstable CACNA1C 50 41 CCOc1ccc(CCCNC(=O)c2cccc([N+](=O)[O-])c2)cc1 ZINC000217865114 EG In-Stock Unstable P2RX7 0 42 CCOc1ccc(CCCNC(=O)c2cccc([N+](=O)[O-])c2)cc1 ZINC000217865114 EG In-Stock Unstable CACNA1D 82 41 CCOc1ccc(CCCNC(=O)c2cccc([N+](=O)[O-])c2)cc1 ZINC000217865114 EG In-Stock Unstable SCN2A 18 44 CCOc1ccc(CCCNC(=O)c2cccc([N+](=O)[O-])c2)cc1 ZINC000217865114 EG In-Stock Unstable PYGL 26 40 CCOc1ccc(CCCNC(=O)c2cccc([N+](=O)[O-])c2)cc1 ZINC000217865114 EG In-Stock Unstable CRTM 41 34 CCOc1ccc(CCCNC(=O)c2cccc([N+](=O)[O-])c2)cc1 ZINC000217865114 EG In-Stock Unstable PDS 16 42 Cn1ccc2c(C(=O)N[C@@H](Cc3ccccc3)C(=O)O)cccc21 ZINC000217865124 DF In-Stock Unstable ACE 49 43 Cn1ccc2c(C(=O)N[C@@H](Cc3ccccc3)C(=O)O)cccc21 ZINC000217865124 DF In-Stock Unstable MME 108 47 Cn1ccc2c(C(=O)N[C@@H](Cc3ccccc3)C(=O)O)cccc21 ZINC000217865124 DF In-Stock Unstable ANPEP 74 41 Cn1ccc2c(C(=O)N[C@@H](Cc3ccccc3)C(=O)O)cccc21 ZINC000217865124 DF In-Stock Unstable CTSB 34 44 Cn1ccc2c(C(=O)N[C@@H](Cc3ccccc3)C(=O)O)cccc21 ZINC000217865124 DF In-Stock Unstable PAPA1_CARPA 47 39 Cn1ccc2c(C(=O)N[C@@H](Cc3ccccc3)C(=O)O)cccc21 ZINC000217865124 DF In-Stock Unstable CPA1 52 43 Cn1ccc2c(C(=O)N[C@@H](Cc3ccccc3)C(=O)O)cccc21 ZINC000217865124 DF In-Stock Unstable CCR3 19 43 Cn1ccc2c(C(=O)N[C@@H](Cc3ccccc3)C(=O)O)cccc21 ZINC000217865124 DF In-Stock Unstable NPFFR2 19 41 Cn1ccc2c(C(=O)N[C@@H](Cc3ccccc3)C(=O)O)cccc21 ZINC000217865124 DF In-Stock Unstable NAALAD2 32 45 Cn1ccc2c(C(=O)N[C@@H](Cc3ccccc3)C(=O)O)cccc21 ZINC000217865124 DF In-Stock Unstable ECE1 57 39 Cn1ccc2c(C(=O)N[C@@H](Cc3ccccc3)C(=O)O)cccc21 ZINC000217865124 DF In-Stock Unstable CAPN1 42 44 Cn1ccc2c(C(=O)N[C@@H](Cc3ccccc3)C(=O)O)cccc21 ZINC000217865124 DF In-Stock Unstable ACE2 100 42 Cn1ccc2c(C(=O)N[C@@H](Cc3ccccc3)C(=O)O)cccc21 ZINC000217865124 DF In-Stock Unstable CTSV 42 35 Cn1ccc2c(C(=O)N[C@@H](Cc3ccccc3)C(=O)O)cccc21 ZINC000217865124 DF In-Stock Unstable FPR1 60 41 Cn1ccc2c(C(=O)N[C@@H](Cc3ccccc3)C(=O)O)cccc21 ZINC000217865124 DF In-Stock Unstable POL 0 42 Cn1ccc2c(C(=O)N[C@@H](Cc3ccccc3)C(=O)O)cccc21 ZINC000217865124 DF In-Stock Unstable SLC15A2 0 45 Cn1ccc2c(C(=O)N[C@@H](Cc3ccccc3)C(=O)O)cccc21 ZINC000217865124 DF In-Stock Unstable BLA1_STEMA 75 40 Cc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217865173 EF For-Sale Unstable NPY2R 41 40 Cc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217865173 EF For-Sale Unstable ADAMTS5 38 44 CCOc1ccc(NC(=O)C(F)F)cc1OC ZINC000217865183 BE On-Demand Unstable GRM4 17 40 CCOc1ccc(NC(=O)C(F)F)cc1OC ZINC000217865183 BE On-Demand Unstable PDGFRA 45 37 CCOc1ccc(NC(=O)C(F)F)cc1OC ZINC000217865183 BE On-Demand Unstable ENPP1 80 40 CCOc1ccc(NC(=O)C(F)F)cc1OC ZINC000217865183 BE On-Demand Unstable DRTS_TRYCR 45 32 CCOc1ccc(NC(=O)C(F)F)cc1OC ZINC000217865183 BE On-Demand Unstable KCNK3 47 46 CCOc1ccc(NC(=O)C(F)F)cc1OC ZINC000217865183 BE On-Demand Unstable KCNK9 40 46 CC(=O)Nc1ccc(S(=O)(=O)NCCn2ccnc2-c2ccccn2)c(C)c1 ZINC000217865186 GE In-Stock Unstable GPR39 0 40 Cc1cc(C)n(Cc2ccc(F)cc2/C=C\C(=O)O)n1 ZINC000217865217 CF For-Sale Unstable PTGER1 21 41 CCCOc1ccccc1CCCNC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217865225 EH In-Stock Unstable CACNA1C 46 38 CCCOc1ccccc1CCCNC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217865225 EH In-Stock Unstable CACNA1D 78 38 CCCOc1ccccc1CCCNC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217865225 EH In-Stock Unstable PYGL 23 40 CCCOc1ccccc1CCCNC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217865225 EH In-Stock Unstable MTNR1B 42 38 CCCOc1ccccc1CCCNC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217865225 EH In-Stock Unstable ACAT 0 40 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCc1ccc(Cl)c(Cl)c1 ZINC000217865231 DK For-Sale Unstable SSTR3 18 45 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCc1ccc(Cl)c(Cl)c1 ZINC000217865231 DK For-Sale Unstable TRPM8 18 48 CC(=O)NCCNC(=O)N/C=C/c1ccccc1Br ZINC000217865233 ED For-Sale Unstable MTNR1A 23 48 CC(=O)NCCNC(=O)N/C=C/c1ccccc1Br ZINC000217865233 ED For-Sale Unstable MTNR1B 20 48 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCc1ccc2c(c1)OCO2 ZINC000217865237 JH In-Stock Unstable NOS2 84 35 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1 ZINC000217865271 FG For-Sale Unstable TBXA2R 41 35 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1 ZINC000217865271 FG For-Sale Unstable HTR7 16 40 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1 ZINC000217865271 FG For-Sale Unstable NPY2R 37 40 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1 ZINC000217865271 FG For-Sale Unstable APP 41 38 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1 ZINC000217865271 FG For-Sale Unstable ADAMTS5 43 46 CSC[C@@](C)(O)CNCc1cccc2cccnc12 ZINC000217865298 CE On-Demand Unstable METAP2 15 40 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCc1ccc2c(c1)OCO2 ZINC000217865305 JH In-Stock Unstable NOS2 84 35 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCc1ccc(Cl)c(Cl)c1 ZINC000217865312 DK For-Sale Unstable SSTR3 18 45 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCc1ccc(Cl)c(Cl)c1 ZINC000217865312 DK For-Sale Unstable TRPM8 18 48 Cc1ccccc1CNC(=O)C(F)F ZINC000217865343 AD On-Demand Unstable ANPEP 31 52 Cc1ccccc1CNC(=O)C(F)F ZINC000217865343 AD On-Demand Unstable P2RX7 36 48 Cc1ccccc1CNC(=O)C(F)F ZINC000217865343 AD On-Demand Unstable AMP1_PLAFQ 43 57 Cc1ccc(OC[C@@H](C)NC(=O)c2cccc([N+](=O)[O-])c2)cc1 ZINC000217865349 DG In-Stock Unstable CACNA1C 49 35 Cc1ccc(OC[C@@H](C)NC(=O)c2cccc([N+](=O)[O-])c2)cc1 ZINC000217865349 DG In-Stock Unstable SDH1 0 41 Cc1ccc(OC[C@@H](C)NC(=O)c2cccc([N+](=O)[O-])c2)cc1 ZINC000217865349 DG In-Stock Unstable P2RX7 0 43 Cc1ccc(OC[C@@H](C)NC(=O)c2cccc([N+](=O)[O-])c2)cc1 ZINC000217865349 DG In-Stock Unstable CACNA1D 83 36 Cc1ccc(OC[C@@H](C)NC(=O)c2cccc([N+](=O)[O-])c2)cc1 ZINC000217865349 DG In-Stock Unstable PYGL 27 47 Cc1ccc(OC[C@@H](C)NC(=O)c2cccc([N+](=O)[O-])c2)cc1 ZINC000217865349 DG In-Stock Unstable IRAK4 19 40 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1 ZINC000217865368 FG For-Sale Unstable TBXA2R 41 35 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1 ZINC000217865368 FG For-Sale Unstable HTR7 16 40 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1 ZINC000217865368 FG For-Sale Unstable NPY2R 37 40 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1 ZINC000217865368 FG For-Sale Unstable APP 41 38 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)cc1 ZINC000217865368 FG For-Sale Unstable ADAMTS5 43 46 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCc1ccc(Cl)c(Cl)c1 ZINC000217865372 DK For-Sale Unstable SSTR3 18 45 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCc1ccc(Cl)c(Cl)c1 ZINC000217865372 DK For-Sale Unstable TRPM8 18 48 CSC[C@](C)(O)CNCc1cccc2cccnc12 ZINC000217865385 CE On-Demand Unstable METAP2 15 40 Cc1ccc(OC[C@H](C)NC(=O)c2cccc([N+](=O)[O-])c2)cc1 ZINC000217865435 DG In-Stock Unstable CACNA1C 49 35 Cc1ccc(OC[C@H](C)NC(=O)c2cccc([N+](=O)[O-])c2)cc1 ZINC000217865435 DG In-Stock Unstable SDH1 0 41 Cc1ccc(OC[C@H](C)NC(=O)c2cccc([N+](=O)[O-])c2)cc1 ZINC000217865435 DG In-Stock Unstable P2RX7 0 43 Cc1ccc(OC[C@H](C)NC(=O)c2cccc([N+](=O)[O-])c2)cc1 ZINC000217865435 DG In-Stock Unstable CACNA1D 83 36 Cc1ccc(OC[C@H](C)NC(=O)c2cccc([N+](=O)[O-])c2)cc1 ZINC000217865435 DG In-Stock Unstable PYGL 27 47 Cc1ccc(OC[C@H](C)NC(=O)c2cccc([N+](=O)[O-])c2)cc1 ZINC000217865435 DG In-Stock Unstable IRAK4 19 40 O=C(N/C=C/c1ccccc1Br)NC12CC3CC(CC(C3)C1)C2 ZINC000217865449 GJ For-Sale Unstable EPHX2 100 50 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCc1ccc(Cl)c(Cl)c1 ZINC000217865454 DK For-Sale Unstable SSTR3 18 45 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCc1ccc(Cl)c(Cl)c1 ZINC000217865454 DK For-Sale Unstable TRPM8 18 48 COc1ccc(C(=O)N[C@@H](C)CCCO)c(F)c1 ZINC000217865465 CD On-Demand Unstable GPR35 20 41 O=C(O)[C@@H]1CCCN1C(=O)[C@@H]1C[C@H]2CCCC[C@@H]2N1 ZINC000217865472 CC For-Sale Unstable ACE 24 49 O=C(O)[C@@H]1CCCN1C(=O)[C@@H]1C[C@H]2CCCC[C@@H]2N1 ZINC000217865472 CC For-Sale Unstable MME 0 47 COc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217865476 EF For-Sale Unstable CASR 26 42 COc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217865476 EF For-Sale Unstable KCNA5 18 40 COc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217865476 EF For-Sale Unstable NPY1R 44 39 COc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217865476 EF For-Sale Unstable NPY2R 78 41 COc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217865476 EF For-Sale Unstable HTR6 16 41 COc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217865476 EF For-Sale Unstable ADAMTS5 36 53 O=C1CCc2cc(S(=O)(=O)NCCn3ccnc3-c3ccccn3)cc3c2N1CC3 ZINC000217865506 HD In-Stock Unstable CYP11B1 28 40 O=C1CCc2cc(S(=O)(=O)NCCn3ccnc3-c3ccccn3)cc3c2N1CC3 ZINC000217865506 HD In-Stock Unstable CYP11B2 28 40 COc1ccc2c(c1)N(CCN1CCC(NC(=O)OC(C)(C)C)CC1)C(=O)CC2 ZINC000217865551 HF For-Sale Unstable CHRM1 15 51 COc1ccc2c(c1)N(CCN1CCC(NC(=O)OC(C)(C)C)CC1)C(=O)CC2 ZINC000217865551 HF For-Sale Unstable DRD4 40 32 COc1ccc2c(c1)N(CCN1CCC(NC(=O)OC(C)(C)C)CC1)C(=O)CC2 ZINC000217865551 HF For-Sale Unstable SIGMAR1 15 43 O=C(N/C=C/c1ccccc1Br)Nc1cccc2cccnc12 ZINC000217865555 FJ For-Sale Anodyne PFHDAC1 0 43 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217865568 EF For-Sale Unstable CASR 26 42 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217865568 EF For-Sale Unstable HTR7 25 46 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217865568 EF For-Sale Unstable CASP3 43 39 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217865568 EF For-Sale Unstable KCNA5 18 40 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217865568 EF For-Sale Unstable MMP13 63 42 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217865568 EF For-Sale Unstable NPY1R 44 39 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217865568 EF For-Sale Unstable NPY2R 78 41 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217865568 EF For-Sale Unstable HTR6 21 42 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217865568 EF For-Sale Unstable MMP2 43 41 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217865568 EF For-Sale Unstable MMP3 55 41 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217865568 EF For-Sale Unstable MMP8 33 41 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217865568 EF For-Sale Unstable MMP14 19 41 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217865568 EF For-Sale Unstable NPY5R 27 41 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217865568 EF For-Sale Unstable PRTN3 49 30 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217865568 EF For-Sale Unstable MMP9 53 41 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217865568 EF For-Sale Unstable MMP12 32 41 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217865568 EF For-Sale Unstable MMP7 46 38 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217865568 EF For-Sale Unstable ADAMTS5 36 53 COc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217865568 EF For-Sale Unstable MMP1 54 41 C[C@@H](CCCO)NC(=O)c1cnn2ccccc12 ZINC000217865644 BD On-Demand Unstable TYK2 31 41 Cc1cc(C)c(CN[C@H]2C[C@H](C)CC[C@H]2C(C)C)c(C)c1 ZINC000217865698 CK For-Sale Unstable TRPM8 15 44 COc1ccc([C@@H]2CCCN2C(=O)CC[C@@H]2NC(=O)c3ccccc3NC2=O)c(OC)c1 ZINC000217865719 IF In-Stock Unstable COLA 51 35 COc1ccc([C@@H]2CCCN2C(=O)CC[C@@H]2NC(=O)c3ccccc3NC2=O)c(OC)c1 ZINC000217865719 IF In-Stock Unstable CPT1A 50 35 C[C@H](CCCO)NC(=O)c1cnn2ccccc12 ZINC000217865725 BD On-Demand Unstable TYK2 31 41 C[C@@H]1Cc2ccccc2N1C(=O)N/C=C/c1ccccc1Br ZINC000217865765 FJ For-Sale Unstable DRD4 24 41 C[C@@H]1Cc2ccccc2N1C(=O)N/C=C/c1ccccc1Br ZINC000217865765 FJ For-Sale Unstable TPP2 45 34 Cc1cc(C)c(CN[C@H]2C[C@@H](C)CC[C@H]2C(C)C)c(C)c1 ZINC000217865788 CK For-Sale Unstable TRPM8 15 44 COc1ccc([C@H]2CCCN2C(=O)CC[C@@H]2NC(=O)c3ccccc3NC2=O)c(OC)c1 ZINC000217865808 IF In-Stock Unstable COLA 51 35 COc1ccc([C@H]2CCCN2C(=O)CC[C@@H]2NC(=O)c3ccccc3NC2=O)c(OC)c1 ZINC000217865808 IF In-Stock Unstable CPT1A 50 35 O=S(=O)(c1ccccc1)n1ccc2c(-c3cccc(F)c3F)ccnc21 ZINC000217865828 FI For-Sale Anodyne HTR6 16 40 C[C@@H](CCCO)NC(=O)c1c(F)cccc1Br ZINC000217865837 DE On-Demand Unstable DAC 26 47 C[C@H]1Cc2ccccc2N1C(=O)N/C=C/c1ccccc1Br ZINC000217865852 FJ For-Sale Unstable DRD4 24 41 C[C@H]1Cc2ccccc2N1C(=O)N/C=C/c1ccccc1Br ZINC000217865852 FJ For-Sale Unstable TPP2 45 34 COc1ccc(Cn2cc(Cl)cn2)cc1/C=C\C(=O)O ZINC000217865871 CF For-Sale Unstable PTGER2 25 40 COc1ccc(Cn2cc(Cl)cn2)cc1/C=C\C(=O)O ZINC000217865871 CF For-Sale Unstable PTGER4 0 40 COc1ccc(Cn2cc(Cl)cn2)cc1/C=C\C(=O)O ZINC000217865871 CF For-Sale Unstable CYSP_PLAFA 43 39 S=C(NCCCn1ccnc1)Nc1ccncc1 ZINC000217865880 CD In-Stock Unstable CYP19A1 15 43 S=C(NCCCn1ccnc1)Nc1ccncc1 ZINC000217865880 CD In-Stock Unstable CYP11B1 20 43 S=C(NCCCn1ccnc1)Nc1ccncc1 ZINC000217865880 CD In-Stock Unstable TBXAS1 45 50 S=C(NCCCn1ccnc1)Nc1ccncc1 ZINC000217865880 CD In-Stock Unstable HMOX2 47 37 S=C(NCCCn1ccnc1)Nc1ccncc1 ZINC000217865880 CD In-Stock Unstable QPCT 132 76 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCc1c(F)cccc1F ZINC000217865913 CJ For-Sale Unstable TRPM8 17 45 Cc1ccc2c(c1)[C@@H](NC(=O)c1cccc([N+](=O)[O-])c1)CC(C)(C)O2 ZINC000217865914 EH In-Stock Unstable CACNA1C 48 36 Cc1ccc2c(c1)[C@@H](NC(=O)c1cccc([N+](=O)[O-])c1)CC(C)(C)O2 ZINC000217865914 EH In-Stock Unstable CACNA1D 79 36 Cc1ccc2c(c1)[C@@H](NC(=O)c1cccc([N+](=O)[O-])c1)CC(C)(C)O2 ZINC000217865914 EH In-Stock Unstable PYGL 0 40 C[C@H](CCCO)NC(=O)c1c(F)cccc1Br ZINC000217865918 DE On-Demand Unstable DAC 26 47 O=C(O)/C=C\c1ccccc1COc1ccc(F)cc1Cl ZINC000217865970 DI For-Sale Unstable PTGER2 24 50 O=C(O)/C=C\c1ccccc1COc1ccc(F)cc1Cl ZINC000217865970 DI For-Sale Unstable PTGER1 50 42 O=C(O)/C=C\c1ccccc1COc1ccc(F)cc1Cl ZINC000217865970 DI For-Sale Unstable PTGER4 37 52 O=C(O)/C=C\c1ccccc1COc1ccc(F)cc1Cl ZINC000217865970 DI For-Sale Unstable FABP4 19 42 O=C(O)/C=C\c1ccccc1COc1ccc(F)cc1Cl ZINC000217865970 DI For-Sale Unstable PTGER3 33 50 O=C(O)/C=C\c1ccccc1COc1ccc(F)cc1Cl ZINC000217865970 DI For-Sale Unstable PTGDR 0 45 O=C(O)/C=C\c1ccccc1COc1ccc(F)cc1Cl ZINC000217865970 DI For-Sale Unstable FABP5 29 42 O=C(O)/C=C\c1ccccc1COc1ccc(F)cc1Cl ZINC000217865970 DI For-Sale Unstable AKR1C3 31 44 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCc1c(F)cccc1F ZINC000217866004 CJ For-Sale Unstable TRPM8 17 45 Cc1ccc2c(c1)[C@H](NC(=O)c1cccc([N+](=O)[O-])c1)CC(C)(C)O2 ZINC000217866011 EH In-Stock Unstable CACNA1C 48 36 Cc1ccc2c(c1)[C@H](NC(=O)c1cccc([N+](=O)[O-])c1)CC(C)(C)O2 ZINC000217866011 EH In-Stock Unstable CACNA1D 79 36 Cc1ccc2c(c1)[C@H](NC(=O)c1cccc([N+](=O)[O-])c1)CC(C)(C)O2 ZINC000217866011 EH In-Stock Unstable PYGL 0 40 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc(OCC(C)C)c2)CC(=O)O4)cc1O ZINC000217866034 KK In-Stock Unstable AKR1B1 0 41 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc(OCC(C)C)c2)CC(=O)O4)cc1O ZINC000217866034 KK In-Stock Unstable CYP1A1 35 41 O=C(O)/C=C\c1ccc(COc2ccc(F)cc2Cl)cc1 ZINC000217866053 DI For-Sale Unstable EGFR 22 43 O=C(O)/C=C\c1ccc(COc2ccc(F)cc2Cl)cc1 ZINC000217866053 DI For-Sale Unstable ESR1 15 49 O=C(O)/C=C\c1ccc(COc2ccc(F)cc2Cl)cc1 ZINC000217866053 DI For-Sale Unstable PTGER2 21 42 O=C(O)/C=C\c1ccc(COc2ccc(F)cc2Cl)cc1 ZINC000217866053 DI For-Sale Unstable ERBB2 30 43 O=C(O)/C=C\c1ccc(COc2ccc(F)cc2Cl)cc1 ZINC000217866053 DI For-Sale Unstable PTGER1 51 40 O=C(O)/C=C\c1ccc(COc2ccc(F)cc2Cl)cc1 ZINC000217866053 DI For-Sale Unstable PTGER4 37 42 O=C(O)/C=C\c1ccc(COc2ccc(F)cc2Cl)cc1 ZINC000217866053 DI For-Sale Unstable AKR1C3 39 56 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCc1c(F)cccc1F ZINC000217866062 CJ For-Sale Unstable TRPM8 17 45 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc(OCC(C)C)c2)CC(=O)O4)cc1O ZINC000217866118 KK In-Stock Unstable AKR1B1 0 41 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc(OCC(C)C)c2)CC(=O)O4)cc1O ZINC000217866118 KK In-Stock Unstable CYP1A1 35 41 Cc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217866121 EH In-Stock Unstable CACNA1C 52 37 Cc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217866121 EH In-Stock Unstable CACNA1D 84 37 Cc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217866121 EH In-Stock Unstable PYGL 0 41 Cc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217866121 EH In-Stock Unstable IRAK4 18 41 CC(C)(C)OC(=O)NC1CCN(CCN2C(=O)COc3ccc(F)cc32)CC1 ZINC000217866136 GF For-Sale Unstable CHRM1 15 49 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2Cl)c1 ZINC000217866154 DI For-Sale Unstable EGFR 58 49 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2Cl)c1 ZINC000217866154 DI For-Sale Unstable MAOB 21 41 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2Cl)c1 ZINC000217866154 DI For-Sale Unstable PTGER2 22 46 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2Cl)c1 ZINC000217866154 DI For-Sale Unstable ERBB2 74 49 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2Cl)c1 ZINC000217866154 DI For-Sale Unstable PTGER1 66 40 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2Cl)c1 ZINC000217866154 DI For-Sale Unstable PTGER4 29 42 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2Cl)c1 ZINC000217866154 DI For-Sale Unstable PTGER3 19 46 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2Cl)c1 ZINC000217866154 DI For-Sale Unstable LTB4R 19 48 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2Cl)c1 ZINC000217866154 DI For-Sale Unstable PLK1 0 49 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2Cl)c1 ZINC000217866154 DI For-Sale Unstable HCAR2 0 47 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2Cl)c1 ZINC000217866154 DI For-Sale Unstable AKR1C3 42 60 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2Cl)c1 ZINC000217866154 DI For-Sale Unstable ADCYAP1R1 43 36 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCc1c(F)cccc1F ZINC000217866156 CJ For-Sale Unstable TRPM8 17 45 O=C(N/C=C/c1ccccc1Br)N1CCN(c2ncccn2)CC1 ZINC000217866171 GF For-Sale Unstable SLC6A7 0 46 Cc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217866205 EH In-Stock Unstable CACNA1C 52 37 Cc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217866205 EH In-Stock Unstable CACNA1D 84 37 Cc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217866205 EH In-Stock Unstable PYGL 0 41 Cc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217866205 EH In-Stock Unstable IRAK4 18 41 CCC[C@@H](O)CNCC(=O)NCCC(C)C ZINC000217866216 BC For-Sale Unstable PGA 46 40 CCC[C@@H](O)CNCC(=O)NCCC(C)C ZINC000217866216 BC For-Sale Unstable DNPEP 0 41 CCN(C)C(=O)CNC(=O)c1cc(Cl)ccc1N ZINC000217866227 CD For-Sale Unstable PYGL 52 45 Cc1ccccc1C(=O)NCCn1ccnc1-c1cccnc1 ZINC000217866239 DF In-Stock Unstable POLR1A 45 32 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2)c1 ZINC000217866240 CH For-Sale Unstable ALOX5 20 48 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2)c1 ZINC000217866240 CH For-Sale Unstable MAOA 16 41 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2)c1 ZINC000217866240 CH For-Sale Unstable MAOB 71 62 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2)c1 ZINC000217866240 CH For-Sale Unstable PTGER2 22 48 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2)c1 ZINC000217866240 CH For-Sale Unstable PTGER4 25 48 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2)c1 ZINC000217866240 CH For-Sale Unstable PTPN2 0 42 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2)c1 ZINC000217866240 CH For-Sale Unstable PTGER3 29 48 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2)c1 ZINC000217866240 CH For-Sale Unstable LTB4R 24 43 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2)c1 ZINC000217866240 CH For-Sale Unstable CDC25B 22 42 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2)c1 ZINC000217866240 CH For-Sale Unstable GYS1 65 36 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2)c1 ZINC000217866240 CH For-Sale Unstable PTGDR 0 46 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2)c1 ZINC000217866240 CH For-Sale Unstable HCAR2 0 49 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2)c1 ZINC000217866240 CH For-Sale Unstable FFAR1 72 44 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2)c1 ZINC000217866240 CH For-Sale Unstable AKR1C3 39 56 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2)c1 ZINC000217866240 CH For-Sale Unstable ENPP2 36 41 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2)c1 ZINC000217866240 CH For-Sale Unstable FFAR4 40 43 O=C(O)/C=C\c1cccc(COc2ccc(F)cc2)c1 ZINC000217866240 CH For-Sale Unstable ADCYAP1R1 30 41 COc1ccc(CN[C@H]2C[C@@H](C)CC[C@@H]2C(C)C)cc1O ZINC000217866257 CH For-Sale Unstable TRPM8 16 42 CCC[C@H](O)CNCC(=O)NCCC(C)C ZINC000217866279 BC For-Sale Unstable PGA 46 40 CCC[C@H](O)CNCC(=O)NCCC(C)C ZINC000217866279 BC For-Sale Unstable DNPEP 0 41 O=C(O)/C=C\c1cc(F)ccc1COc1ccc(F)cc1 ZINC000217866310 CH For-Sale Unstable PTGER2 46 42 O=C(O)/C=C\c1cc(F)ccc1COc1ccc(F)cc1 ZINC000217866310 CH For-Sale Unstable PTGER4 24 42 O=C(O)/C=C\c1cc(F)ccc1COc1ccc(F)cc1 ZINC000217866310 CH For-Sale Unstable PTGER3 21 45 O=C(O)/C=C\c1cc(F)ccc1COc1ccc(F)cc1 ZINC000217866310 CH For-Sale Unstable PTGDR 0 45 O=C(O)/C=C\c1cc(F)ccc1COc1ccc(F)cc1 ZINC000217866310 CH For-Sale Unstable FFAR1 24 43 O=C(O)/C=C\c1cc(F)ccc1COc1ccc(F)cc1 ZINC000217866310 CH For-Sale Unstable FFAR4 45 43 COc1ccc2c(c1)[C@@H](NC(=O)c1cccc([N+](=O)[O-])c1)CC(C)(C)O2 ZINC000217866315 FH In-Stock Unstable CACNA1C 47 39 COc1ccc2c(c1)[C@@H](NC(=O)c1cccc([N+](=O)[O-])c1)CC(C)(C)O2 ZINC000217866315 FH In-Stock Unstable CACNA1D 79 39 COc1ccc(C(=O)NCCn2ccnc2-c2cccnc2)cc1 ZINC000217866334 DE In-Stock Unstable DRD4 48 38 COc1ccc(C(=O)NCCn2ccnc2-c2cccnc2)cc1 ZINC000217866334 DE In-Stock Unstable DRD3 19 41 COc1ccc(C(=O)NCCn2ccnc2-c2cccnc2)cc1 ZINC000217866334 DE In-Stock Unstable TBXAS1 19 43 COc1ccc(C(=O)NCCn2ccnc2-c2cccnc2)cc1 ZINC000217866334 DE In-Stock Unstable PTAFR 24 49 COc1ccc(C(=O)NCCn2ccnc2-c2cccnc2)cc1 ZINC000217866334 DE In-Stock Unstable GSK3B 0 44 COc1ccc(C(=O)NCCn2ccnc2-c2cccnc2)cc1 ZINC000217866334 DE In-Stock Unstable CYP11B2 29 42 COc1ccc(C(=O)NCCn2ccnc2-c2cccnc2)cc1 ZINC000217866334 DE In-Stock Unstable IKBKE 22 42 COc1ccc(C(=O)NCCn2ccnc2-c2cccnc2)cc1 ZINC000217866334 DE In-Stock Unstable TBK1 24 42 COc1ccc(C(=O)NCCn2ccnc2-c2cccnc2)cc1 ZINC000217866334 DE In-Stock Unstable ROS1 45 38 COc1ccc(CN[C@H]2C[C@H](C)CC[C@@H]2C(C)C)cc1O ZINC000217866355 CH For-Sale Unstable TRPM8 16 42 CCOC(=O)N1CCC(NC(=O)N/C=C/c2ccccc2Br)CC1 ZINC000217866366 GG For-Sale Unstable EPHX2 35 45 CCOC(=O)N1CCC(NC(=O)N/C=C/c2ccccc2Br)CC1 ZINC000217866366 GG For-Sale Unstable CCR8 38 42 COc1ccc2c(c1)[C@H](NC(=O)c1cccc([N+](=O)[O-])c1)CC(C)(C)O2 ZINC000217866399 FH In-Stock Unstable CACNA1C 47 39 COc1ccc2c(c1)[C@H](NC(=O)c1cccc([N+](=O)[O-])c1)CC(C)(C)O2 ZINC000217866399 FH In-Stock Unstable CACNA1D 79 39 O=C(O)/C=C\c1cc(COc2ccc(F)cc2)ccc1F ZINC000217866402 CH For-Sale Unstable MAOB 19 48 O=C(O)/C=C\c1cc(COc2ccc(F)cc2)ccc1F ZINC000217866402 CH For-Sale Unstable PTGER2 45 50 O=C(O)/C=C\c1cc(COc2ccc(F)cc2)ccc1F ZINC000217866402 CH For-Sale Unstable PTGER4 0 50 O=C(O)/C=C\c1cc(COc2ccc(F)cc2)ccc1F ZINC000217866402 CH For-Sale Unstable PTGER3 30 50 O=C(O)/C=C\c1cc(COc2ccc(F)cc2)ccc1F ZINC000217866402 CH For-Sale Unstable GYS1 51 34 O=C(O)/C=C\c1cc(COc2ccc(F)cc2)ccc1F ZINC000217866402 CH For-Sale Unstable PTGDR 0 48 O=C(O)/C=C\c1cc(COc2ccc(F)cc2)ccc1F ZINC000217866402 CH For-Sale Unstable FFAR1 51 43 O=C(O)/C=C\c1cc(COc2ccc(F)cc2)ccc1F ZINC000217866402 CH For-Sale Unstable AKR1C3 26 43 CCOc1ccccc1C(=O)NCCn1ccnc1-c1cccnc1 ZINC000217866414 EF In-Stock Unstable GYRB 0 40 CCOc1ccccc1C(=O)NCCn1ccnc1-c1cccnc1 ZINC000217866414 EF In-Stock Unstable ACAT 0 44 CCOc1ccccc1C(=O)NCCn1ccnc1-c1cccnc1 ZINC000217866414 EF In-Stock Unstable HCN1 59 41 CCOc1ccccc1C(=O)NCCn1ccnc1-c1cccnc1 ZINC000217866414 EF In-Stock Unstable HCN4 49 38 O=C(CCCNc1ncccn1)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217866416 FD In-Stock Unstable CHRNA4 31 52 O=C(N/C=C/c1ccccc1Br)N1CCN(c2cccc(Cl)c2)CC1 ZINC000217866479 HJ For-Sale Unstable HTR1A 15 42 COc1ccc(COc2ccccc2)cc1/C=C\C(=O)O ZINC000217866483 CG For-Sale Unstable ALOX5 20 41 COc1ccc(COc2ccccc2)cc1/C=C\C(=O)O ZINC000217866483 CG For-Sale Unstable TSHR 56 35 COc1ccc(COc2ccccc2)cc1/C=C\C(=O)O ZINC000217866483 CG For-Sale Unstable MAOB 23 44 COc1ccc(COc2ccccc2)cc1/C=C\C(=O)O ZINC000217866483 CG For-Sale Unstable PPARG 15 42 COc1ccc(COc2ccccc2)cc1/C=C\C(=O)O ZINC000217866483 CG For-Sale Unstable PTGER2 26 58 COc1ccc(COc2ccccc2)cc1/C=C\C(=O)O ZINC000217866483 CG For-Sale Unstable PPARA 18 40 COc1ccc(COc2ccccc2)cc1/C=C\C(=O)O ZINC000217866483 CG For-Sale Unstable PTGER4 48 58 COc1ccc(COc2ccccc2)cc1/C=C\C(=O)O ZINC000217866483 CG For-Sale Unstable PTGER3 51 58 COc1ccc(COc2ccccc2)cc1/C=C\C(=O)O ZINC000217866483 CG For-Sale Unstable LTB4R 52 45 COc1ccc(COc2ccccc2)cc1/C=C\C(=O)O ZINC000217866483 CG For-Sale Unstable TNFRSF1A 35 41 COc1ccc(COc2ccccc2)cc1/C=C\C(=O)O ZINC000217866483 CG For-Sale Unstable FFAR1 59 45 COc1ccc(COc2ccccc2)cc1/C=C\C(=O)O ZINC000217866483 CG For-Sale Unstable AKR1C3 38 49 COc1ccc(COc2ccccc2)cc1/C=C\C(=O)O ZINC000217866483 CG For-Sale Unstable FFAR4 41 41 COc1ccc(COc2ccccc2)cc1/C=C\C(=O)O ZINC000217866483 CG For-Sale Unstable ABCG2 20 45 COc1ccc(COc2ccccc2)cc1/C=C\C(=O)O ZINC000217866483 CG For-Sale Unstable AKR1B10 39 45 COc1ccc(COc2ccccc2)cc1/C=C\C(=O)O ZINC000217866483 CG For-Sale Unstable CYSP_PLAFA 50 40 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1N[C@@H]1CCSC1 ZINC000217866488 BH For-Sale Unstable TRPM8 0 42 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217866493 FH In-Stock Unstable DRD4 40 31 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217866493 FH In-Stock Unstable CACNA1C 49 39 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217866493 FH In-Stock Unstable CACNA1D 83 39 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217866493 FH In-Stock Unstable PYGL 0 40 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217866493 FH In-Stock Unstable AKR1C2 15 41 CC[C@@H](C)[C@H](N)C(=O)N1C[C@H](C)O[C@@H](C)C1 ZINC000217866516 BC For-Sale Unstable DPP9 18 45 O=C(NCCn1ccnc1-c1cccnc1)c1ccc2c(c1)OCO2 ZINC000217866518 EE In-Stock Unstable DRD4 40 31 O=C(NCCn1ccnc1-c1cccnc1)c1ccc2c(c1)OCO2 ZINC000217866518 EE In-Stock Unstable NOS2 40 31 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1N[C@@H]1CCSC1 ZINC000217866541 BH On-Demand Unstable TRPM8 16 42 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217866547 FH In-Stock Unstable DRD4 40 31 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217866547 FH In-Stock Unstable CACNA1C 49 39 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217866547 FH In-Stock Unstable CACNA1D 83 39 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217866547 FH In-Stock Unstable PYGL 0 40 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1cccc([N+](=O)[O-])c1 ZINC000217866547 FH In-Stock Unstable AKR1C2 15 41 O=C(O)/C=C\c1ccc(COc2ccccc2)c(F)c1 ZINC000217866572 CH For-Sale Unstable PTGER2 49 43 O=C(O)/C=C\c1ccc(COc2ccccc2)c(F)c1 ZINC000217866572 CH For-Sale Unstable PTGER4 26 43 O=C(O)/C=C\c1ccc(COc2ccccc2)c(F)c1 ZINC000217866572 CH For-Sale Unstable PTPN2 0 43 O=C(O)/C=C\c1ccc(COc2ccccc2)c(F)c1 ZINC000217866572 CH For-Sale Unstable PTGER3 30 43 O=C(O)/C=C\c1ccc(COc2ccccc2)c(F)c1 ZINC000217866572 CH For-Sale Unstable CDC25B 25 43 O=C(O)/C=C\c1ccc(COc2ccccc2)c(F)c1 ZINC000217866572 CH For-Sale Unstable PTGDR 0 41 O=C(O)/C=C\c1ccc(COc2ccccc2)c(F)c1 ZINC000217866572 CH For-Sale Unstable AKR1C3 34 53 O=C(O)/C=C\c1ccc(COc2ccccc2)c(F)c1 ZINC000217866572 CH For-Sale Unstable FFAR4 55 37 Cc1ccc2nc(-c3ccc(NC(=O)N/C=C/c4ccccc4Br)cc3)sc2c1 ZINC000217866573 JK For-Sale Unstable APP 26 51 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1N[C@@H]1CCSC1 ZINC000217866638 BH For-Sale Unstable TRPM8 0 42 COc1ccccc1Oc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217866670 II For-Sale Unstable HTR7 23 43 COc1ccccc1Oc1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217866670 II For-Sale Unstable ADAMTS5 27 45 O=C(N/C=C/c1ccccc1Br)Nc1ccc2c(c1)OCO2 ZINC000217866681 FH For-Sale Unstable CCR2 0 42 CC[C@@H](NC(=O)c1cccc([N+](=O)[O-])c1)c1ccc(C)c(C)c1 ZINC000217866689 DI In-Stock Unstable CACNA1C 51 35 CC[C@@H](NC(=O)c1cccc([N+](=O)[O-])c1)c1ccc(C)c(C)c1 ZINC000217866689 DI In-Stock Unstable CACNA1D 82 35 CC[C@@H](NC(=O)c1cccc([N+](=O)[O-])c1)c1ccc(C)c(C)c1 ZINC000217866689 DI In-Stock Unstable CCR3 0 43 CC[C@@H](NC(=O)c1cccc([N+](=O)[O-])c1)c1ccc(C)c(C)c1 ZINC000217866689 DI In-Stock Unstable UTS2 56 40 C[C@H]1CCC[C@@H](C)N1Cc1cccc(/C=C\C(=O)O)c1 ZINC000217866696 CH For-Sale Unstable HDAC8 40 37 CC(C)[C@H]1CC[C@H](C)C[C@@H]1N[C@@H]1CCSC1 ZINC000217866717 BH For-Sale Unstable TRPM8 0 42 COc1ccc2c(c1)cc(C(=O)N[C@H]1CCCc3c1[nH]c1ccc(OC)cc31)n2C ZINC000217866729 HI In-Stock Unstable MAPKAPK2 23 49 COc1ccc2c(c1)cc(C(=O)N[C@H]1CCCc3c1[nH]c1ccc(OC)cc31)n2C ZINC000217866729 HI In-Stock Unstable MTNR1A 31 47 O=C(NCCn1ccnc1-c1cccnc1)c1ccc(F)c(F)c1 ZINC000217866740 EF In-Stock Unstable PLD2 42 39 CC[C@H](NC(=O)c1cccc([N+](=O)[O-])c1)c1ccc(C)c(C)c1 ZINC000217866755 DI In-Stock Unstable CACNA1C 51 35 CC[C@H](NC(=O)c1cccc([N+](=O)[O-])c1)c1ccc(C)c(C)c1 ZINC000217866755 DI In-Stock Unstable CACNA1D 82 35 CC[C@H](NC(=O)c1cccc([N+](=O)[O-])c1)c1ccc(C)c(C)c1 ZINC000217866755 DI In-Stock Unstable UTS2 56 40 COc1ccccc1Oc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217866764 II For-Sale Unstable HTR7 23 43 COc1ccccc1Oc1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217866764 II For-Sale Unstable ADAMTS5 27 45 COc1ccc2c(c1)cc(C(=O)N[C@@H]1CCCc3c1[nH]c1ccc(OC)cc31)n2C ZINC000217866812 HI In-Stock Unstable MAPKAPK2 23 49 COc1ccc2c(c1)cc(C(=O)N[C@@H]1CCCc3c1[nH]c1ccc(OC)cc31)n2C ZINC000217866812 HI In-Stock Unstable MTNR1A 31 47 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC1[C@@H](C)CCC[C@@H]1C ZINC000217866840 CJ For-Sale Unstable TRPM8 15 40 CC[C@@H](NC(=O)c1cccc([N+](=O)[O-])c1)c1ccc(C)cc1C ZINC000217866846 DI In-Stock Unstable CACNA1C 48 35 CC[C@@H](NC(=O)c1cccc([N+](=O)[O-])c1)c1ccc(C)cc1C ZINC000217866846 DI In-Stock Unstable CACNA1D 78 35 CC[C@@H](NC(=O)c1cccc([N+](=O)[O-])c1)c1ccc(C)cc1C ZINC000217866846 DI In-Stock Unstable PYGL 0 43 CC[C@@H](NC(=O)c1cccc([N+](=O)[O-])c1)c1ccc(C)cc1C ZINC000217866846 DI In-Stock Unstable IRAK4 20 43 CC[C@@H](NC(=O)c1cccc([N+](=O)[O-])c1)c1ccc(C)cc1C ZINC000217866846 DI In-Stock Unstable KCNK3 42 33 C[C@@H](CCCO)NC(=O)c1cc(Cl)ccc1Br ZINC000217866891 DF On-Demand Unstable ALPL 43 38 C[C@@H](CCCO)NC(=O)c1cc(Cl)ccc1Br ZINC000217866891 DF On-Demand Unstable UTS2 41 32 O=C(N/C=C/c1ccccc1Br)Nc1cccc(F)c1 ZINC000217866893 EI For-Sale Anodyne KCNK3 63 44 O=C(N/C=C/c1ccccc1Br)Nc1cccc(F)c1 ZINC000217866893 EI For-Sale Anodyne KCNK9 31 41 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC1[C@@H](C)CCC[C@@H]1C ZINC000217866907 CJ For-Sale Unstable TRPM8 15 40 CC[C@H](NC(=O)c1cccc([N+](=O)[O-])c1)c1ccc(C)cc1C ZINC000217866915 DI In-Stock Unstable CACNA1C 48 35 CC[C@H](NC(=O)c1cccc([N+](=O)[O-])c1)c1ccc(C)cc1C ZINC000217866915 DI In-Stock Unstable CACNA1D 78 35 CC[C@H](NC(=O)c1cccc([N+](=O)[O-])c1)c1ccc(C)cc1C ZINC000217866915 DI In-Stock Unstable PYGL 0 43 CC[C@H](NC(=O)c1cccc([N+](=O)[O-])c1)c1ccc(C)cc1C ZINC000217866915 DI In-Stock Unstable IRAK4 20 43 CC[C@H](NC(=O)c1cccc([N+](=O)[O-])c1)c1ccc(C)cc1C ZINC000217866915 DI In-Stock Unstable KCNK3 42 33 O=C(NCCn1ccnc1-c1cccnc1)c1cccc(C(F)(F)F)c1 ZINC000217866933 FG In-Stock Unstable ABL1 15 42 O=C(NCCn1ccnc1-c1cccnc1)c1cccc(C(F)(F)F)c1 ZINC000217866933 FG In-Stock Unstable DRD4 41 32 O=C(NCCn1ccnc1-c1cccnc1)c1cccc(C(F)(F)F)c1 ZINC000217866933 FG In-Stock Unstable KIT 0 44 O=C(NCCn1ccnc1-c1cccnc1)c1cccc(C(F)(F)F)c1 ZINC000217866933 FG In-Stock Unstable CCR2 64 45 O=C(NCCn1ccnc1-c1cccnc1)c1cccc(C(F)(F)F)c1 ZINC000217866933 FG In-Stock Unstable EPHX2 0 41 O=C(NCCn1ccnc1-c1cccnc1)c1cccc(C(F)(F)F)c1 ZINC000217866933 FG In-Stock Unstable CHEK1 41 31 O=C(NCCn1ccnc1-c1cccnc1)c1cccc(C(F)(F)F)c1 ZINC000217866933 FG In-Stock Unstable BRAF 46 43 O=C(NCCn1ccnc1-c1cccnc1)c1cccc(C(F)(F)F)c1 ZINC000217866933 FG In-Stock Unstable GPR52 0 44 C[C@H](CCCO)NC(=O)c1cc(Cl)ccc1Br ZINC000217866966 DF On-Demand Unstable ALPL 43 38 C[C@H](CCCO)NC(=O)c1cc(Cl)ccc1Br ZINC000217866966 DF On-Demand Unstable UTS2 41 32 CN(C)[C@@H]1C[C@@H](C(=O)O)N(C(=O)Cc2ccc(O)c(Cl)c2)C1 ZINC000217866971 ED In-Stock Unstable OPRK1 43 42 CN(C)[C@@H]1C[C@@H](C(=O)O)N(C(=O)Cc2ccc(O)c(Cl)c2)C1 ZINC000217866971 ED In-Stock Unstable NCE103 29 42 CN(C)[C@@H]1C[C@@H](C(=O)O)N(C(=O)Cc2ccc(O)c(Cl)c2)C1 ZINC000217866971 ED In-Stock Unstable CAN2 0 46 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC1[C@@H](C)CCC[C@@H]1C ZINC000217867009 CJ For-Sale Unstable TRPM8 15 40 CC[C@@H](NC(=O)c1cccc([N+](=O)[O-])c1)c1ccc(OC)c(OC)c1 ZINC000217867030 EG In-Stock Unstable CACNA1C 47 36 CC[C@@H](NC(=O)c1cccc([N+](=O)[O-])c1)c1ccc(OC)c(OC)c1 ZINC000217867030 EG In-Stock Unstable CACNA1D 82 36 CC[C@@H](NC(=O)c1cccc([N+](=O)[O-])c1)c1ccc(OC)c(OC)c1 ZINC000217867030 EG In-Stock Unstable CCR3 0 41 CC[C@@H](NC(=O)c1cccc([N+](=O)[O-])c1)c1ccc(OC)c(OC)c1 ZINC000217867030 EG In-Stock Unstable PYGL 22 41 CC[C@@H](NC(=O)c1cccc([N+](=O)[O-])c1)c1ccc(OC)c(OC)c1 ZINC000217867030 EG In-Stock Unstable KCNMA1 19 41 CC[C@@H](NC(=O)c1cccc([N+](=O)[O-])c1)c1ccc(OC)c(OC)c1 ZINC000217867030 EG In-Stock Unstable UTS2 55 41 CSC[C@@](C)(O)CNCc1cccc2ccccc12 ZINC000217867036 CG On-Demand Unstable KCNJ2 0 43 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC1[C@@H](C)CCC[C@@H]1C ZINC000217867072 CJ For-Sale Unstable TRPM8 15 40 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)c(C(F)(F)F)c1 ZINC000217867086 HI For-Sale Unstable ADAMTS5 31 44 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)c(C(F)(F)F)c1 ZINC000217867086 HI For-Sale Unstable SFRP1 140 41 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc(Cl)c(C(F)(F)F)c1 ZINC000217867086 HI For-Sale Unstable WNT3 93 39 CSC[C@](C)(O)CNCc1cccc2ccccc12 ZINC000217867100 CG On-Demand Unstable KCNJ2 0 43 CC[C@H](NC(=O)c1cccc([N+](=O)[O-])c1)c1ccc(OC)c(OC)c1 ZINC000217867112 EG In-Stock Unstable CACNA1C 47 36 CC[C@H](NC(=O)c1cccc([N+](=O)[O-])c1)c1ccc(OC)c(OC)c1 ZINC000217867112 EG In-Stock Unstable CACNA1D 82 36 CC[C@H](NC(=O)c1cccc([N+](=O)[O-])c1)c1ccc(OC)c(OC)c1 ZINC000217867112 EG In-Stock Unstable CCR3 0 41 CC[C@H](NC(=O)c1cccc([N+](=O)[O-])c1)c1ccc(OC)c(OC)c1 ZINC000217867112 EG In-Stock Unstable PYGL 22 41 CC[C@H](NC(=O)c1cccc([N+](=O)[O-])c1)c1ccc(OC)c(OC)c1 ZINC000217867112 EG In-Stock Unstable KCNMA1 19 41 CC[C@H](NC(=O)c1cccc([N+](=O)[O-])c1)c1ccc(OC)c(OC)c1 ZINC000217867112 EG In-Stock Unstable UTS2 55 41 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1N[C@@H]1C[C@@H]2C[C@@H]1[C@@H]1CCC[C@@H]21 ZINC000217867158 CJ For-Sale Unstable TRPM8 0 40 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)c(C(F)(F)F)c1 ZINC000217867175 HI For-Sale Unstable ADAMTS5 31 44 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)c(C(F)(F)F)c1 ZINC000217867175 HI For-Sale Unstable SFRP1 140 41 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Cl)c(C(F)(F)F)c1 ZINC000217867175 HI For-Sale Unstable WNT3 93 39 CC[C@@H]1COCCN1C[C@@H](O)COc1ccc(N)cc1 ZINC000217867202 CD For-Sale Unstable ABCB1 0 42 CC[C@@H](NC(=O)c1cccc([N+](=O)[O-])c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217867213 FF In-Stock Unstable TACR3 43 37 CC[C@@H](NC(=O)c1cccc([N+](=O)[O-])c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217867213 FF In-Stock Unstable HISG 0 41 O=C(N/C=C/c1ccccc1Br)Nc1ccc(I)cc1 ZINC000217867214 IJ For-Sale Anodyne MTCA1 15 42 O=C(N/C=C/c1ccccc1Br)Nc1ccc(I)cc1 ZINC000217867214 IJ For-Sale Anodyne P96878_MYCTU 18 42 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1N[C@@H]1C[C@@H]2C[C@@H]1[C@@H]1CCC[C@@H]21 ZINC000217867230 CJ For-Sale Unstable TRPM8 0 40 CC[C@@H](C)[C@H](N)C(=O)N1C[C@H](C)C[C@@H](C)C1 ZINC000217867267 BD For-Sale Unstable CHRNA4 0 42 CC[C@@H](C)[C@H](N)C(=O)N1C[C@H](C)C[C@@H](C)C1 ZINC000217867267 BD For-Sale Unstable TPP2 33 41 CC[C@@H](C)[C@H](N)C(=O)N1C[C@H](C)C[C@@H](C)C1 ZINC000217867267 BD For-Sale Unstable DPP9 0 46 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217867284 HI For-Sale Unstable MMP13 22 45 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217867284 HI For-Sale Unstable NPY1R 42 38 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217867284 HI For-Sale Unstable NPY2R 53 38 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217867284 HI For-Sale Unstable MMP2 22 45 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217867284 HI For-Sale Unstable MMP8 15 40 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217867284 HI For-Sale Unstable MMP14 27 45 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217867284 HI For-Sale Unstable MMP9 20 45 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217867284 HI For-Sale Unstable ADAMTS5 33 44 CC[C@H]1COCCN1C[C@@H](O)COc1ccc(N)cc1 ZINC000217867287 CD For-Sale Unstable ABCB1 0 42 CC[C@H](NC(=O)c1cccc([N+](=O)[O-])c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217867292 FF In-Stock Unstable TACR3 43 37 CC[C@H](NC(=O)c1cccc([N+](=O)[O-])c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217867292 FF In-Stock Unstable HISG 0 41 CC[C@@H](C)N(C)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217867300 CG For-Sale Unstable PTGER2 28 43 CC[C@@H](C)N(C)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217867300 CG For-Sale Unstable PTGER4 0 43 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1N[C@@H]1C[C@@H]2C[C@@H]1[C@@H]1CCC[C@@H]21 ZINC000217867310 CJ For-Sale Unstable TRPM8 0 40 COC(=O)c1nc(NC(=O)[C@H](C)Nc2ccc3c(cc2=O)[C@@H](NC(C)=O)CCc2cc(OC)c(OC)c(OC)c2-3)sc1C(C)C ZINC000217867313 KJ In-Stock Unstable TUBA1A 17 61 O=C(N/C=C/c1ccccc1Br)NCCc1c[nH]c2ccccc12 ZINC000217867326 GI For-Sale Unstable MC4R 32 47 O=C(N/C=C/c1ccccc1Br)NCCc1c[nH]c2ccccc12 ZINC000217867326 GI For-Sale Unstable CCKAR 28 42 O=C(N/C=C/c1ccccc1Br)NCCc1c[nH]c2ccccc12 ZINC000217867326 GI For-Sale Unstable MPO 36 41 O=C(N/C=C/c1ccccc1Br)NCCc1c[nH]c2ccccc12 ZINC000217867326 GI For-Sale Unstable BRS3 41 44 O=C(N/C=C/c1ccccc1Br)NCCc1c[nH]c2ccccc12 ZINC000217867326 GI For-Sale Unstable NMBR 22 44 O=C(N/C=C/c1ccccc1Br)NCCc1c[nH]c2ccccc12 ZINC000217867326 GI For-Sale Unstable HDAC7 21 42 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217867372 HI For-Sale Unstable MMP13 22 45 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217867372 HI For-Sale Unstable NPY1R 42 38 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217867372 HI For-Sale Unstable NPY2R 53 38 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217867372 HI For-Sale Unstable MMP2 22 45 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217867372 HI For-Sale Unstable MMP8 15 40 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217867372 HI For-Sale Unstable MMP14 27 45 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217867372 HI For-Sale Unstable MMP9 20 45 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Oc2ccccc2)cc1 ZINC000217867372 HI For-Sale Unstable ADAMTS5 33 44 CC[C@H](C)N(C)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217867389 CG For-Sale Unstable PTGER2 28 43 CC[C@H](C)N(C)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217867389 CG For-Sale Unstable PTGER4 0 43 C[C@@H](CCCO)NC(=O)c1ccc(Cl)cc1Br ZINC000217867392 DF On-Demand Unstable UTS2 40 32 Cc1cccc(-c2noc(CNC(=O)c3cccc([N+](=O)[O-])c3)n2)c1 ZINC000217867405 EF In-Stock Unstable CACNA1C 46 34 Cc1cccc(-c2noc(CNC(=O)c3cccc([N+](=O)[O-])c3)n2)c1 ZINC000217867405 EF In-Stock Unstable CACNA1D 74 34 Cc1cccc(-c2noc(CNC(=O)c3cccc([N+](=O)[O-])c3)n2)c1 ZINC000217867405 EF In-Stock Unstable E1 0 41 CC(C)[C@H]1CC[C@H](C)C[C@@H]1N[C@@H]1C[C@@H]2C[C@@H]1[C@@H]1CCC[C@@H]21 ZINC000217867412 CJ For-Sale Unstable TRPM8 0 40 CC[C@@H]1COCCN1C[C@@H](O)COc1cccc(N)c1 ZINC000217867438 CD For-Sale Unstable ABCB1 27 42 COc1cc([C@@H]2CC(=O)Oc3cc4c(cc32)OCO4)ccc1OCCc1ccccc1 ZINC000217867451 HI In-Stock Unstable EDNRA 24 40 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc(Br)cc1 ZINC000217867471 GG For-Sale Unstable NPY2R 35 40 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccc(Br)cc1 ZINC000217867471 GG For-Sale Unstable ADAMTS5 34 44 C[C@H](CCCO)NC(=O)c1ccc(Cl)cc1Br ZINC000217867488 DF On-Demand Unstable UTS2 40 32 Cc1ccc(-c2noc(CNC(=O)c3cccc([N+](=O)[O-])c3)n2)cc1 ZINC000217867496 EF In-Stock Unstable CACNA1C 49 35 Cc1ccc(-c2noc(CNC(=O)c3cccc([N+](=O)[O-])c3)n2)cc1 ZINC000217867496 EF In-Stock Unstable CACNA1D 81 35 Cc1ccc(-c2noc(CNC(=O)c3cccc([N+](=O)[O-])c3)n2)cc1 ZINC000217867496 EF In-Stock Unstable E1 0 41 CC[C@H]1COCCN1C[C@@H](O)COc1cccc(N)c1 ZINC000217867517 CD For-Sale Unstable ABCB1 27 42 COc1cc([C@H]2CC(=O)Oc3cc4c(cc32)OCO4)ccc1OCCc1ccccc1 ZINC000217867522 HI In-Stock Unstable EDNRA 24 40 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Br)cc1 ZINC000217867529 GG For-Sale Unstable NPY2R 35 40 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccc(Br)cc1 ZINC000217867529 GG For-Sale Unstable ADAMTS5 34 44 O=C(c1ncccc1O)N1CCCC[C@@H]1c1nc2ccccc2[nH]1 ZINC000217867559 DG In-Stock Unstable PRCP 52 40 O=C(c1ncccc1O)N1CCCC[C@@H]1c1nc2ccccc2[nH]1 ZINC000217867559 DG In-Stock Unstable COLA 79 36 O=C(c1ncccc1O)N1CCCC[C@@H]1c1nc2ccccc2[nH]1 ZINC000217867559 DG In-Stock Unstable CPT1A 72 36 O=C(c1ncccc1O)N1CCCC[C@@H]1c1nc2ccccc2[nH]1 ZINC000217867559 DG In-Stock Unstable KCNN3 31 42 O=C(c1ncccc1O)N1CCCC[C@@H]1c1nc2ccccc2[nH]1 ZINC000217867559 DG In-Stock Unstable SMO 0 42 Cc1ccc(CN[C@H]2C[C@H](C)CC[C@H]2C(C)C)o1 ZINC000217867599 BI For-Sale Unstable TRPM8 15 44 CC[C@@H]1COCCN1C[C@@H](O)COc1ccccc1N ZINC000217867609 CD For-Sale Unstable ADRB2 40 47 CC[C@@H]1COCCN1C[C@@H](O)COc1ccccc1N ZINC000217867609 CD For-Sale Unstable ADRB3 32 47 CC[C@@H]1COCCN1C[C@@H](O)COc1ccccc1N ZINC000217867609 CD For-Sale Unstable ABCB1 56 39 COc1ccc(-c2noc(CNC(=O)c3cccc([N+](=O)[O-])c3)n2)cc1 ZINC000217867624 FF In-Stock Unstable DRD4 43 34 COc1ccc(-c2noc(CNC(=O)c3cccc([N+](=O)[O-])c3)n2)cc1 ZINC000217867624 FF In-Stock Unstable CACNA1D 44 33 COc1ccc(-c2noc(CNC(=O)c3cccc([N+](=O)[O-])c3)n2)cc1 ZINC000217867624 FF In-Stock Unstable U38 0 41 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)NCc3cccnc3)[C@H]21 ZINC000217867628 JF In-Stock Unstable TSHR 40 31 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)NCc3cccnc3)[C@H]21 ZINC000217867628 JF In-Stock Unstable HTR7 18 44 O=C(c1ncccc1O)N1CCCC[C@H]1c1nc2ccccc2[nH]1 ZINC000217867637 DG In-Stock Unstable PRCP 52 40 O=C(c1ncccc1O)N1CCCC[C@H]1c1nc2ccccc2[nH]1 ZINC000217867637 DG In-Stock Unstable COLA 79 36 O=C(c1ncccc1O)N1CCCC[C@H]1c1nc2ccccc2[nH]1 ZINC000217867637 DG In-Stock Unstable CPT1A 72 36 O=C(c1ncccc1O)N1CCCC[C@H]1c1nc2ccccc2[nH]1 ZINC000217867637 DG In-Stock Unstable KCNN3 31 42 O=C(c1ncccc1O)N1CCCC[C@H]1c1nc2ccccc2[nH]1 ZINC000217867637 DG In-Stock Unstable SMO 0 42 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccccc1C(F)(F)F ZINC000217867643 GH For-Sale Unstable NPY2R 30 47 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccccc1C(F)(F)F ZINC000217867643 GH For-Sale Unstable ADAMTS5 31 44 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccccc1C(F)(F)F ZINC000217867643 GH For-Sale Unstable SFRP1 134 39 O=S(=O)(NC[C@H]1CCCN1c1ccccc1)c1ccccc1C(F)(F)F ZINC000217867643 GH For-Sale Unstable WNT3 91 38 CC[C@H]1COCCN1C[C@@H](O)COc1ccccc1N ZINC000217867696 CD For-Sale Unstable ADRB2 40 47 CC[C@H]1COCCN1C[C@@H](O)COc1ccccc1N ZINC000217867696 CD For-Sale Unstable ADRB3 32 47 CC[C@H]1COCCN1C[C@@H](O)COc1ccccc1N ZINC000217867696 CD For-Sale Unstable ABCB1 56 39 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)NCc3cccnc3)[C@@H]21 ZINC000217867712 JF In-Stock Unstable TSHR 40 31 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)NCc3cccnc3)[C@@H]21 ZINC000217867712 JF In-Stock Unstable HTR7 18 44 Cc1ccc(CN[C@H]2C[C@@H](C)CC[C@H]2C(C)C)o1 ZINC000217867721 BI For-Sale Unstable TRPM8 15 44 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1C(F)(F)F ZINC000217867722 GH For-Sale Unstable NPY2R 30 47 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1C(F)(F)F ZINC000217867722 GH For-Sale Unstable ADAMTS5 31 44 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1C(F)(F)F ZINC000217867722 GH For-Sale Unstable SFRP1 134 39 O=S(=O)(NC[C@@H]1CCCN1c1ccccc1)c1ccccc1C(F)(F)F ZINC000217867722 GH For-Sale Unstable WNT3 91 38 CC[C@@H](C)CN(C)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217867732 CG For-Sale Unstable AKR1C3 30 40 Cc1cc(-c2ccncc2)nn1CCNC(=O)/C=C/c1ccccc1Cl ZINC000217867733 FH In-Stock Unstable BOTA 26 43 COc1ccc(-c2noc(CNC(=O)c3cccc([N+](=O)[O-])c3)n2)c(OC)c1 ZINC000217867741 GF In-Stock Unstable DRD4 42 32 COc1ccc(-c2noc(CNC(=O)c3cccc([N+](=O)[O-])c3)n2)c(OC)c1 ZINC000217867741 GF In-Stock Unstable CACNA1D 63 37 COc1ccc(-c2noc(CNC(=O)c3cccc([N+](=O)[O-])c3)n2)c(OC)c1 ZINC000217867741 GF In-Stock Unstable U38 0 40 COc1ccc(-c2noc(CNC(=O)c3cccc([N+](=O)[O-])c3)n2)c(OC)c1 ZINC000217867741 GF In-Stock Unstable TAAR1 27 51 C[C@@H]1[C@H]2[C@H]3OCCN2CC[C@@]1(C)c1cc(O)ccc13 ZINC000217867754 CE For-Sale Unstable OPRM1 29 44 C[C@@H]1[C@H]2[C@H]3OCCN2CC[C@@]1(C)c1cc(O)ccc13 ZINC000217867754 CE For-Sale Unstable OPRD1 19 44 C[C@@H]1[C@H]2[C@H]3OCCN2CC[C@@]1(C)c1cc(O)ccc13 ZINC000217867754 CE For-Sale Unstable OPRK1 29 44 C[C@@H]1[C@H]2[C@H]3OCCN2CC[C@@]1(C)c1cc(O)ccc13 ZINC000217867754 CE For-Sale Unstable SIGMAR1 19 44 CCOc1c(Br)cc(Br)cc1CNC[C@@](C)(O)CSC ZINC000217867788 IH On-Demand Unstable METG 36 44 Cc1cccc(C)c1C(=O)N[C@@H](C)CCCO ZINC000217867792 BE On-Demand Unstable ACAT 0 40 CC(C)(C)OC(=O)NC1CCN(CCN2C(=O)COc3ccccc32)CC1 ZINC000217867800 GE For-Sale Unstable CHRM1 21 65 CC(C)(C)OC(=O)NC1CCN(CCN2C(=O)COc3ccccc32)CC1 ZINC000217867800 GE For-Sale Unstable DRD2 22 47 CC(C)(C)OC(=O)NC1CCN(CCN2C(=O)COc3ccccc32)CC1 ZINC000217867800 GE For-Sale Unstable UTS2R 15 59 CC[C@H](C)CN(C)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217867813 CG For-Sale Unstable AKR1C3 30 40 N#Cc1ccccc1S(=O)(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217867819 EF For-Sale Unstable NPY1R 44 35 N#Cc1ccccc1S(=O)(=O)NC[C@H]1CCCN1c1ccccc1 ZINC000217867819 EF For-Sale Unstable ADAMTS5 30 41 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@H](C(=O)Nc3cccc(-c4nc[nH]n4)c3)C(C)C)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217867820 KJ In-Stock Unstable TUBA1A 17 60 Cc1cc(-c2ccncc2)nn1CCNC(=O)c1cnn(-c2ccccc2)c1C ZINC000217867835 GG In-Stock Unstable SLC9A2 0 40 C[C@H]1[C@H]2[C@H]3OCCN2CC[C@@]1(C)c1cc(O)ccc13 ZINC000217867844 CE For-Sale Unstable OPRM1 29 44 C[C@H]1[C@H]2[C@H]3OCCN2CC[C@@]1(C)c1cc(O)ccc13 ZINC000217867844 CE For-Sale Unstable OPRD1 19 44 C[C@H]1[C@H]2[C@H]3OCCN2CC[C@@]1(C)c1cc(O)ccc13 ZINC000217867844 CE For-Sale Unstable OPRK1 29 44 C[C@H]1[C@H]2[C@H]3OCCN2CC[C@@]1(C)c1cc(O)ccc13 ZINC000217867844 CE For-Sale Unstable SIGMAR1 19 44 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCc1ccc(O)c(O)c1 ZINC000217867845 CH For-Sale Unstable TRPM8 17 45 O=C(NCc1nc(-c2cccc(Br)c2)no1)c1cccc([N+](=O)[O-])c1 ZINC000217867860 HG In-Stock Unstable E1 0 41 CCOc1c(Br)cc(Br)cc1CNC[C@](C)(O)CSC ZINC000217867868 IH On-Demand Unstable METG 36 44 Cc1cccc(C)c1C(=O)N[C@H](C)CCCO ZINC000217867882 BE On-Demand Unstable ACAT 0 40 N#Cc1ccccc1S(=O)(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217867893 EF For-Sale Unstable NPY1R 44 35 N#Cc1ccccc1S(=O)(=O)NC[C@@H]1CCCN1c1ccccc1 ZINC000217867893 EF For-Sale Unstable ADAMTS5 30 41 CC[C@@H](C)CN(C)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217867917 CG For-Sale Unstable PTGER2 24 41 CC[C@@H](C)CN(C)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217867917 CG For-Sale Unstable PTGER4 0 41 Cc1cc(-c2ccncc2)nn1CCNC(=O)c1cncc(Br)c1 ZINC000217867928 GF In-Stock Unstable SCN10A 41 33 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCc1ccc(O)c(O)c1 ZINC000217867931 CH For-Sale Unstable TRPM8 17 45 COc1cc(NC(=O)N/C=C/c2ccccc2Br)c(OC)cc1Cl ZINC000217867944 HJ For-Sale Unstable CYSP_PLAFA 40 34 CC[C@H](C)CN(C)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217867994 CG For-Sale Unstable PTGER2 24 41 CC[C@H](C)CN(C)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217867994 CG For-Sale Unstable PTGER4 0 41 COc1cccc(-c2noc(CN(C)C(=O)c3cccc([N+](=O)[O-])c3)n2)c1 ZINC000217868004 FF In-Stock Unstable GPBAR1 24 41 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCc1ccc(O)c(O)c1 ZINC000217868011 CH For-Sale Unstable TRPM8 17 45 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217868018 GD For-Sale Unstable CA2 35 49 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217868018 GD For-Sale Unstable CA6 17 40 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217868018 GD For-Sale Unstable CA1 35 49 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217868018 GD For-Sale Unstable CA7 21 40 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217868018 GD For-Sale Unstable NPY1R 40 34 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217868018 GD For-Sale Unstable CA5B 30 40 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217868018 GD For-Sale Unstable CA4 21 49 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217868018 GD For-Sale Unstable CA12 24 49 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217868018 GD For-Sale Unstable ADAMTS5 34 44 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217868018 GD For-Sale Unstable CA9 32 49 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217868018 GD For-Sale Unstable CAH_METTE 21 40 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217868018 GD For-Sale Unstable CYNT 33 40 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217868018 GD For-Sale Unstable NCE103 20 40 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217868018 GD For-Sale Unstable CA15 21 40 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217868018 GD For-Sale Unstable MTCA1 20 40 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@H]2CCCN2c2ccccc2)cc1 ZINC000217868018 GD For-Sale Unstable A6YCJ1_9METZ 27 40 CC[C@@H](C)[C@H](N)C(=O)N[C@@H]1CCC[C@@H](C)C1 ZINC000217868020 BE For-Sale Unstable TPP2 39 43 CCOc1ccc(C(=O)NCCn2nc(-c3ccncc3)cc2C)cc1OCC ZINC000217868026 GG In-Stock Unstable SSTR5 40 35 CC[C@@H](C)[C@H](N)C(=O)N[C@H]1CCC[C@@H](C)C1 ZINC000217868072 BE For-Sale Unstable TPP2 39 43 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217868074 GD For-Sale Unstable CA2 35 49 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217868074 GD For-Sale Unstable CA6 17 40 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217868074 GD For-Sale Unstable CA1 35 49 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217868074 GD For-Sale Unstable CA7 21 40 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217868074 GD For-Sale Unstable NPY1R 40 34 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217868074 GD For-Sale Unstable CA5B 30 40 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217868074 GD For-Sale Unstable CA4 21 49 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217868074 GD For-Sale Unstable CA12 24 49 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217868074 GD For-Sale Unstable ADAMTS5 34 44 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217868074 GD For-Sale Unstable CA9 32 49 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217868074 GD For-Sale Unstable CAH_METTE 21 40 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217868074 GD For-Sale Unstable CYNT 33 40 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217868074 GD For-Sale Unstable NCE103 20 40 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217868074 GD For-Sale Unstable CA15 21 40 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217868074 GD For-Sale Unstable MTCA1 20 40 NS(=O)(=O)c1ccc(S(=O)(=O)NC[C@@H]2CCCN2c2ccccc2)cc1 ZINC000217868074 GD For-Sale Unstable A6YCJ1_9METZ 27 40 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCc1ccc(O)c(O)c1 ZINC000217868086 CH For-Sale Unstable TRPM8 17 45 Cn1cc(C(=O)N2CCN(c3ccnc4nncn34)CC2)c2ccccc21 ZINC000217868145 FD In-Stock Unstable TPSAB1 27 41 CN(Cc1nc(-c2ccccc2Cl)no1)C(=O)c1cccc([N+](=O)[O-])c1 ZINC000217868206 FH In-Stock Unstable GPBAR1 28 40 CSC[C@@](C)(O)CNCc1ccc(OCC(N)=O)cc1 ZINC000217868218 CC On-Demand Unstable PLA2G4B 43 31 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCc1ccc(Br)o1 ZINC000217868222 DJ For-Sale Unstable TRPM8 15 41 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)Nc3cccc(-c4nc[nH]n4)c3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217868233 KH In-Stock Unstable TUBA1A 17 62 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)Nc3cccc(-c4nc[nH]n4)c3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217868233 KH In-Stock Unstable TPPP 0 57 COc1ccc(Cl)cc1C(=O)NCCn1nc(-c2ccncc2)cc1C ZINC000217868262 FG In-Stock Unstable CNR1 15 41 COc1ccc(Cl)cc1C(=O)NCCn1nc(-c2ccncc2)cc1C ZINC000217868262 FG In-Stock Unstable F10 48 33 COc1ccc(Cl)cc1C(=O)NCCn1nc(-c2ccncc2)cc1C ZINC000217868262 FG In-Stock Unstable CPT1A 44 33 Cn1ccnc1[C@@H]1CCCN(Cc2ccc(OCCn3ccnc3)cc2)C1 ZINC000217868286 FG In-Stock Unstable CYP11B1 0 44 Cn1ccnc1[C@@H]1CCCN(Cc2ccc(OCCn3ccnc3)cc2)C1 ZINC000217868286 FG In-Stock Unstable HRH3 35 43 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCc1ccc(Br)o1 ZINC000217868293 DJ For-Sale Unstable TRPM8 15 41 COC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217868296 CE For-Sale Unstable CHRM2 15 42 COC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217868296 CE For-Sale Unstable DRD2 27 42 COC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217868296 CE For-Sale Unstable DRD4 54 42 COC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217868296 CE For-Sale Unstable ACHE 44 44 COC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217868296 CE For-Sale Unstable HRH1 17 41 COC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217868296 CE For-Sale Unstable CHRM3 26 42 COC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217868296 CE For-Sale Unstable SIGMAR1 61 52 COC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217868296 CE For-Sale Unstable SSTR5 43 33 COC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217868296 CE For-Sale Unstable CCR3 33 41 COC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217868296 CE For-Sale Unstable MCHR1 29 42 COC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217868296 CE For-Sale Unstable CCR8 26 42 COC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217868296 CE For-Sale Unstable AKR1C3 30 41 O=C(N/C=C/c1ccccc1Br)N1CCN(c2ccccc2)CC1 ZINC000217868297 GH For-Sale Unstable ERBB2 0 41 O=C(N/C=C/c1ccccc1Br)N1CCN(c2ccccc2)CC1 ZINC000217868297 GH For-Sale Unstable AKR1C3 0 43 O=C(N/C=C/c1ccccc1Br)N1CCN(c2ccccc2)CC1 ZINC000217868297 GH For-Sale Unstable GPR183 0 41 CSC[C@](C)(O)CNCc1ccc(OCC(N)=O)cc1 ZINC000217868307 CC On-Demand Unstable PLA2G4B 43 31 C=CCNC(=O)CCCCCN1C(=O)c2ccccc2N2C(=O)c3c(ccc(OC)c3OC)[C@H]12 ZINC000217868353 JH In-Stock Unstable HTR7 23 40 Cc1cc(-c2ccncc2)nn1CCNC(=O)c1cccc(C(F)(F)F)c1 ZINC000217868358 FH In-Stock Unstable DRD4 41 33 Cc1cc(-c2ccncc2)nn1CCNC(=O)c1cccc(C(F)(F)F)c1 ZINC000217868358 FH In-Stock Unstable FLT1 23 43 Cc1cc(-c2ccncc2)nn1CCNC(=O)c1cccc(C(F)(F)F)c1 ZINC000217868358 FH In-Stock Unstable KDR 18 43 Cc1cc(-c2ccncc2)nn1CCNC(=O)c1cccc(C(F)(F)F)c1 ZINC000217868358 FH In-Stock Unstable NPY5R 15 40 Cc1cc(-c2ccncc2)nn1CCNC(=O)c1cccc(C(F)(F)F)c1 ZINC000217868358 FH In-Stock Unstable EPHB2 18 40 Cc1cc(-c2ccncc2)nn1CCNC(=O)c1cccc(C(F)(F)F)c1 ZINC000217868358 FH In-Stock Unstable CCR2 65 41 Cc1cc(-c2ccncc2)nn1CCNC(=O)c1cccc(C(F)(F)F)c1 ZINC000217868358 FH In-Stock Unstable BRAF 43 51 Cc1cc(-c2ccncc2)nn1CCNC(=O)c1cccc(C(F)(F)F)c1 ZINC000217868358 FH In-Stock Unstable EPHB4 28 42 Cc1cc(-c2ccncc2)nn1CCNC(=O)c1cccc(C(F)(F)F)c1 ZINC000217868358 FH In-Stock Unstable GPR52 0 42 Cn1ccnc1[C@H]1CCCN(Cc2ccc(OCCn3ccnc3)cc2)C1 ZINC000217868366 FG In-Stock Unstable CYP11B1 0 44 Cn1ccnc1[C@H]1CCCN(Cc2ccc(OCCn3ccnc3)cc2)C1 ZINC000217868366 FG In-Stock Unstable HRH3 35 43 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCc1ccc(Br)o1 ZINC000217868374 DJ For-Sale Unstable TRPM8 15 41 COC1CCN(Cc2ccc(F)cc2/C=C\C(=O)O)CC1 ZINC000217868384 CF For-Sale Unstable SIGMAR1 21 40 COC1CCN(Cc2ccc(F)cc2/C=C\C(=O)O)CC1 ZINC000217868384 CF For-Sale Unstable CCR3 35 40 C=CCNC(=O)CCCCCN1C(=O)c2ccccc2N2C(=O)c3c(ccc(OC)c3OC)[C@@H]12 ZINC000217868410 JH In-Stock Unstable HTR7 23 40 CC(C)c1ccc(CCCNC(=O)c2cccc([N+](=O)[O-])c2)cc1 ZINC000217868437 EI In-Stock Unstable DRD4 41 31 CC(C)c1ccc(CCCNC(=O)c2cccc([N+](=O)[O-])c2)cc1 ZINC000217868437 EI In-Stock Unstable CACNA1D 67 36 CC(C)c1ccc(CCCNC(=O)c2cccc([N+](=O)[O-])c2)cc1 ZINC000217868437 EI In-Stock Unstable COLA 25 40 Cc1cc(-c2ccncc2)nn1CCNC(=O)c1cccc2ccccc12 ZINC000217868441 FH In-Stock Unstable CCR3 0 41 Cc1cc(-c2ccncc2)nn1CCNC(=O)c1cccc2ccccc12 ZINC000217868441 FH In-Stock Unstable ROCK1 24 41 Cc1cc(-c2ccncc2)nn1CCNC(=O)c1cccc2ccccc12 ZINC000217868441 FH In-Stock Unstable POLR1A 76 41 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCc1ccc(Br)o1 ZINC000217868447 DJ For-Sale Unstable TRPM8 15 41 COC1CCN(Cc2ccc(F)c(/C=C\C(=O)O)c2)CC1 ZINC000217868519 CF For-Sale Unstable SIGMAR1 33 43 COC1CCN(Cc2ccc(F)c(/C=C\C(=O)O)c2)CC1 ZINC000217868519 CF For-Sale Unstable SSTR5 53 35 COC1CCN(Cc2ccc(F)c(/C=C\C(=O)O)c2)CC1 ZINC000217868519 CF For-Sale Unstable CCR1 0 40 COC1CCN(Cc2ccc(F)c(/C=C\C(=O)O)c2)CC1 ZINC000217868519 CF For-Sale Unstable CCR3 37 41 COC1CCN(Cc2ccc(F)c(/C=C\C(=O)O)c2)CC1 ZINC000217868519 CF For-Sale Unstable MCHR1 35 40 O=C(NCCCN1CCCc2ccccc21)c1cccc([N+](=O)[O-])c1 ZINC000217868527 EG In-Stock Unstable DRD2 22 43 O=C(NCCCN1CCCc2ccccc21)c1cccc([N+](=O)[O-])c1 ZINC000217868527 EG In-Stock Unstable DRD4 48 39 O=C(NCCCN1CCCc2ccccc21)c1cccc([N+](=O)[O-])c1 ZINC000217868527 EG In-Stock Unstable ADRA1D 19 41 O=C(NCCCN1CCCc2ccccc21)c1cccc([N+](=O)[O-])c1 ZINC000217868527 EG In-Stock Unstable AVPR2 26 58 O=C(NCCCN1CCCc2ccccc21)c1cccc([N+](=O)[O-])c1 ZINC000217868527 EG In-Stock Unstable ADRA1B 24 41 O=C(NCCCN1CCCc2ccccc21)c1cccc([N+](=O)[O-])c1 ZINC000217868527 EG In-Stock Unstable ADRA2B 0 41 O=C(NCCCN1CCCc2ccccc21)c1cccc([N+](=O)[O-])c1 ZINC000217868527 EG In-Stock Unstable ADRA2C 18 41 C[C@H](/C=C/C#N)NC(=O)OC(C)(C)C ZINC000217868538 AD For-Sale Unstable PAPA1_CARPA 53 44 C[C@H](/C=C/C#N)NC(=O)OC(C)(C)C ZINC000217868538 AD For-Sale Unstable CTSK 21 44 CN(C[C@@H]1CCCCN1C)C(=O)c1ccc(OCc2ccccc2F)cc1 ZINC000217868540 FH In-Stock Unstable CHRNA10 53 41 CN(C[C@@H]1CCCCN1C)C(=O)c1ccc(OCc2ccccc2F)cc1 ZINC000217868540 FH In-Stock Unstable NS5B 0 50 CN(C[C@@H]1CCCCN1C)C(=O)c1ccc(OCc2ccccc2F)cc1 ZINC000217868540 FH In-Stock Unstable ACKR3 73 40 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCc1ccc([C@@H]2C[C@@H]2C)o1 ZINC000217868559 CJ For-Sale Unstable TRPM8 0 40 COc1ccc([N+](=O)[O-])cc1NC(=O)N/C=C/c1ccccc1Br ZINC000217868617 GI For-Sale Unstable KCNMA1 22 53 Cc1cc(-c2ccncc2)nn1CCNC(=O)COc1ccc(F)cc1 ZINC000217868624 FF In-Stock Unstable ADORA2A 15 40 CN(C[C@H]1CCCCN1C)C(=O)c1ccc(OCc2ccccc2F)cc1 ZINC000217868627 FH In-Stock Unstable CHRNA10 53 41 CN(C[C@H]1CCCCN1C)C(=O)c1ccc(OCc2ccccc2F)cc1 ZINC000217868627 FH In-Stock Unstable NS5B 0 50 CN(C[C@H]1CCCCN1C)C(=O)c1ccc(OCc2ccccc2F)cc1 ZINC000217868627 FH In-Stock Unstable ACKR3 73 40 CCOc1ccc(CNC(=O)c2ccc(Br)cc2)cc1OCC ZINC000217868633 GI In-Stock Unstable PPARG 19 47 CCOc1ccc(CNC(=O)c2ccc(Br)cc2)cc1OCC ZINC000217868633 GI In-Stock Unstable PPARA 24 47 CCOc1ccc(CNC(=O)c2ccc(Br)cc2)cc1OCC ZINC000217868633 GI In-Stock Unstable PPARD 26 47 CCOc1ccc(CNC(=O)c2ccc(Br)cc2)cc1OCC ZINC000217868633 GI In-Stock Unstable AGPAT2 28 44 CCOc1ccc(CNC(=O)c2ccc(Br)cc2)cc1OCC ZINC000217868633 GI In-Stock Unstable MT-ND1 26 49 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCc1ccc([C@@H]2C[C@@H]2C)o1 ZINC000217868643 CJ For-Sale Unstable TRPM8 0 40 CC(C)(C)c1ccc(CCN)cc1Br ZINC000217868688 CG For-Sale Unstable TAAR1 28 44 COCc1cc(=O)c(O)c([C@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccc(OC)cc2)o1 ZINC000217868705 JI In-Stock Unstable DRD5 18 40 COCc1cc(=O)c(O)c([C@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccc(OC)cc2)o1 ZINC000217868705 JI In-Stock Unstable RORC 44 37 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCc1ccc([C@@H]2C[C@@H]2C)o1 ZINC000217868723 CJ For-Sale Unstable TRPM8 0 40 Cc1cc(-c2ccncc2)nn1CCNC(=O)C(c1ccccc1)c1ccccc1 ZINC000217868738 GI In-Stock Unstable ROCK1 23 40 Cc1cc(-c2ccncc2)nn1CCNC(=O)C(c1ccccc1)c1ccccc1 ZINC000217868738 GI In-Stock Unstable ROCK2 17 40 Cc1cc(-c2ccncc2)nn1CCNC(=O)C(c1ccccc1)c1ccccc1 ZINC000217868738 GI In-Stock Unstable SOAT1 27 44 Cc1cc(-c2ccncc2)nn1CCNC(=O)C(c1ccccc1)c1ccccc1 ZINC000217868738 GI In-Stock Unstable GPR142 50 42 COc1ccccc1CCCNC(=O)c1ccc(Br)cc1 ZINC000217868739 EH In-Stock Unstable HTR1A 15 47 COc1ccccc1CCCNC(=O)c1ccc(Br)cc1 ZINC000217868739 EH In-Stock Unstable DRD2 31 47 COc1ccccc1CCCNC(=O)c1ccc(Br)cc1 ZINC000217868739 EH In-Stock Unstable DRD1 0 46 COc1ccccc1CCCNC(=O)c1ccc(Br)cc1 ZINC000217868739 EH In-Stock Unstable DRD3 45 46 COc1ccccc1CCCNC(=O)c1ccc(Br)cc1 ZINC000217868739 EH In-Stock Unstable TRPV1 0 41 COc1ccccc1CCCNC(=O)c1ccc(Br)cc1 ZINC000217868739 EH In-Stock Unstable MTNR1B 46 45 COc1ccccc1CCCNC(=O)c1ccc(Br)cc1 ZINC000217868739 EH In-Stock Unstable ITGAV 17 40 COc1ccccc1CCCNC(=O)c1ccc(Br)cc1 ZINC000217868739 EH In-Stock Unstable HDA106 0 44 COc1ccccc1CCCNC(=O)c1ccc(Br)cc1 ZINC000217868739 EH In-Stock Unstable MBTPS1 41 33 COc1ccccc1CCCNC(=O)c1ccc(Br)cc1 ZINC000217868739 EH In-Stock Unstable AP2S1 0 47 COc1ccccc1CCCNC(=O)c1ccc(Br)cc1 ZINC000217868739 EH In-Stock Unstable ALPHA-1A 0 44 CC[C@@H]1CN(Cc2cccc(/C=C\C(=O)O)c2)CCO1 ZINC000217868769 CE For-Sale Unstable DRD4 36 49 CC[C@@H]1CN(Cc2cccc(/C=C\C(=O)O)c2)CCO1 ZINC000217868769 CE For-Sale Unstable SIGMAR1 32 43 CC[C@@H]1CN(Cc2cccc(/C=C\C(=O)O)c2)CCO1 ZINC000217868769 CE For-Sale Unstable HDAC8 39 41 CC[C@@H]1CN(Cc2cccc(/C=C\C(=O)O)c2)CCO1 ZINC000217868769 CE For-Sale Unstable HDAC1 17 41 CC[C@@H]1CN(Cc2cccc(/C=C\C(=O)O)c2)CCO1 ZINC000217868769 CE For-Sale Unstable HDAC6 28 41 COCc1cc(=O)c(O)c([C@@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccc(OC)cc2)o1 ZINC000217868775 JI In-Stock Unstable DRD5 18 40 COCc1cc(=O)c(O)c([C@@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2ccc(OC)cc2)o1 ZINC000217868775 JI In-Stock Unstable RORC 44 37 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCc1ccc([C@@H]2C[C@@H]2C)o1 ZINC000217868825 CJ For-Sale Unstable TRPM8 0 40 CC[C@H]1CN(Cc2cccc(/C=C\C(=O)O)c2)CCO1 ZINC000217868836 CE For-Sale Unstable DRD4 36 49 CC[C@H]1CN(Cc2cccc(/C=C\C(=O)O)c2)CCO1 ZINC000217868836 CE For-Sale Unstable SIGMAR1 32 43 CC[C@H]1CN(Cc2cccc(/C=C\C(=O)O)c2)CCO1 ZINC000217868836 CE For-Sale Unstable HDAC8 39 41 CC[C@H]1CN(Cc2cccc(/C=C\C(=O)O)c2)CCO1 ZINC000217868836 CE For-Sale Unstable HDAC1 17 41 CC[C@H]1CN(Cc2cccc(/C=C\C(=O)O)c2)CCO1 ZINC000217868836 CE For-Sale Unstable HDAC6 28 41 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)N[C@@H](CCSC)c3nnc4ccccn34)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217868849 KH In-Stock Unstable TUBA1A 16 55 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)N[C@@H](CCSC)c3nnc4ccccn34)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217868849 KH In-Stock Unstable TPPP 0 53 Cc1cc(-c2ccncc2)nn1CCNC(=O)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217868850 IE In-Stock Unstable GSK3B 15 41 Cc1cc(-c2ccncc2)nn1CCNC(=O)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217868850 IE In-Stock Unstable TGM2 41 42 Cc1cc(-c2ccncc2)nn1CCNC(=O)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217868850 IE In-Stock Unstable NAMPT 50 44 CCOc1ccc(CCCNC(=O)c2ccc(Br)cc2)cc1 ZINC000217868854 FI In-Stock Unstable KCNQ1 0 45 CCOc1ccc(CCCNC(=O)c2ccc(Br)cc2)cc1 ZINC000217868854 FI In-Stock Unstable SCN2A 23 50 CCOc1ccc(CCCNC(=O)c2ccc(Br)cc2)cc1 ZINC000217868854 FI In-Stock Unstable HDA106 0 44 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCc1cccc(C#N)c1 ZINC000217868918 CI On-Demand Unstable TRPM8 17 42 CCCOc1ccccc1CCCNC(=O)c1ccc(Br)cc1 ZINC000217868982 GJ In-Stock Unstable KCNQ1 0 40 CCCOc1ccccc1CCCNC(=O)c1ccc(Br)cc1 ZINC000217868982 GJ In-Stock Unstable MTNR1A 41 47 CCCOc1ccccc1CCCNC(=O)c1ccc(Br)cc1 ZINC000217868982 GJ In-Stock Unstable MTNR1B 48 40 C[C@H](C(=O)O)c1ccc(CO[C@@H]2CCCC[C@@H]2C)cc1 ZINC000217868983 CH For-Sale Unstable PTGS1 34 51 C[C@H](C(=O)O)c1ccc(CO[C@@H]2CCCC[C@@H]2C)cc1 ZINC000217868983 CH For-Sale Unstable PTGS2 23 51 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCc1cccc(C#N)c1 ZINC000217869001 CI On-Demand Unstable TRPM8 17 42 C[C@H](C(=O)O)c1ccc(CO[C@H]2CCCC[C@@H]2C)cc1 ZINC000217869061 CH For-Sale Unstable PTGS1 34 51 C[C@H](C(=O)O)c1ccc(CO[C@H]2CCCC[C@@H]2C)cc1 ZINC000217869061 CH For-Sale Unstable PTGS2 23 51 Cc1ccccc1OC[C@@H](C)NC(=O)c1ccc(Br)cc1 ZINC000217869072 EH In-Stock Unstable SDH1 0 40 COc1ccc(CCC(=O)NCCn2nc(-c3ccncc3)cc2C)cc1 ZINC000217869074 FG In-Stock Unstable MTNR1A 42 39 COc1ccc(CCC(=O)NCCn2nc(-c3ccncc3)cc2C)cc1 ZINC000217869074 FG In-Stock Unstable PTGDR 22 45 COc1ccc(CCC(=O)NCCn2nc(-c3ccncc3)cc2C)cc1 ZINC000217869074 FG In-Stock Unstable PROKR1 42 30 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCc1cccc(C#N)c1 ZINC000217869089 CI For-Sale Unstable TRPM8 17 42 COc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)Nc1cccc3c1ccn3C)C(=O)OC2 ZINC000217869148 IJ In-Stock Unstable IMPDH1 0 73 COc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)Nc1cccc3c1ccn3C)C(=O)OC2 ZINC000217869148 IJ In-Stock Unstable IMPDH2 0 73 OCc1cn(CCCCBr)nn1 ZINC000217869154 BC For-Sale Unstable GBA 15 40 Cc1cc(-c2ccncc2)nn1CCNC(=O)c1ccc(F)cc1Cl ZINC000217869170 FG In-Stock Unstable P2RX7 53 43 Cc1cc(-c2ccncc2)nn1CCNC(=O)c1ccc(F)cc1Cl ZINC000217869170 FG In-Stock Unstable PYGL 22 42 Cc1cc(-c2ccncc2)nn1CCNC(=O)c1ccc(F)cc1Cl ZINC000217869170 FG In-Stock Unstable ALPL 49 32 CC1CCN(c2ccc([C@@H](C)NC(=O)c3ccc(Br)cc3)cc2)CC1 ZINC000217869175 HK In-Stock Unstable SDH1 0 48 CC1CCN(c2ccc([C@@H](C)NC(=O)c3ccc(Br)cc3)cc2)CC1 ZINC000217869175 HK In-Stock Unstable PRNP 46 38 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCc1cccc(C#N)c1 ZINC000217869183 CI For-Sale Unstable TRPM8 17 42 O=C(O)/C=C\c1cccc(OCCN2CCCC2=O)c1 ZINC000217869236 CD For-Sale Unstable CYSLTR2 17 41 CC[C@@H](C)[C@H](N)C(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217869238 CF For-Sale Unstable DPP4 24 66 CC[C@@H](C)[C@H](N)C(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217869238 CF For-Sale Unstable PREP 18 45 CC[C@@H](C)[C@H](N)C(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217869238 CF For-Sale Unstable DPP7 37 49 CC[C@@H](C)[C@H](N)C(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217869238 CF For-Sale Unstable TPP2 50 55 CC[C@@H](C)[C@H](N)C(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217869238 CF For-Sale Unstable XIAP 17 40 CC[C@@H](C)[C@H](N)C(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217869238 CF For-Sale Unstable DPP8 31 54 CC[C@@H](C)[C@H](N)C(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217869238 CF For-Sale Unstable DPP9 19 48 CC1CCN(c2ccc([C@H](C)NC(=O)c3ccc(Br)cc3)cc2)CC1 ZINC000217869245 HK In-Stock Unstable SDH1 0 48 CC1CCN(c2ccc([C@H](C)NC(=O)c3ccc(Br)cc3)cc2)CC1 ZINC000217869245 HK In-Stock Unstable PRNP 46 38 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)C1CCC1 ZINC000217869250 DE For-Sale Unstable SCD1 16 41 Cc1cc(-c2ccncc2)nn1CCNC(=O)c1cccc(C#N)c1 ZINC000217869276 EF In-Stock Unstable DRD4 44 35 CC[C@@H](N[C@@H]1C[C@@H](C)CC[C@@H]1C(C)C)c1ccc(O)cc1 ZINC000217869324 CJ For-Sale Unstable TRPM8 16 43 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)C1CCC1 ZINC000217869327 DE For-Sale Unstable SCD1 16 41 CC[C@@H](C)[C@H](N)C(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217869329 CF For-Sale Unstable DPP4 24 66 CC[C@@H](C)[C@H](N)C(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217869329 CF For-Sale Unstable PREP 18 45 CC[C@@H](C)[C@H](N)C(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217869329 CF For-Sale Unstable DPP7 37 49 CC[C@@H](C)[C@H](N)C(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217869329 CF For-Sale Unstable TPP2 50 55 CC[C@@H](C)[C@H](N)C(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217869329 CF For-Sale Unstable XIAP 17 40 CC[C@@H](C)[C@H](N)C(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217869329 CF For-Sale Unstable DPP8 31 54 CC[C@@H](C)[C@H](N)C(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217869329 CF For-Sale Unstable DPP9 19 48 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)c3ccc(Br)cc3)cc2)C1 ZINC000217869355 HK In-Stock Unstable SDH1 0 48 Clc1cc2c(cc1Br)CCCO2 ZINC000217869367 BG For-Sale Unstable AHR 20 50 Cc1csc(C(=O)NCCn2nc(-c3ccncc3)cc2C)c1 ZINC000217869381 EG In-Stock Unstable ROCK1 22 41 CC[C@H](N[C@@H]1C[C@@H](C)CC[C@@H]1C(C)C)c1ccc(O)cc1 ZINC000217869404 CJ For-Sale Unstable TRPM8 16 43 O=C(O)/C=C\c1ccccc1Cn1cnc2ccccc21 ZINC000217869405 CG For-Sale Unstable PTGER2 47 46 O=C(O)/C=C\c1ccccc1Cn1cnc2ccccc21 ZINC000217869405 CG For-Sale Unstable PTGER4 24 46 O=C(O)/C=C\c1ccccc1Cn1cnc2ccccc21 ZINC000217869405 CG For-Sale Unstable PTGER3 23 46 O=C(COCc1nc2cc(F)ccc2[nH]1)NCc1ccc2ccccc2n1 ZINC000217869408 FG In-Stock Unstable CYSLTR1 46 34 O=C(COCc1nc2cc(F)ccc2[nH]1)NCc1ccc2ccccc2n1 ZINC000217869408 FG In-Stock Unstable CYSP_TRYCR 0 45 O=C(COCc1nc2cc(F)ccc2[nH]1)NCc1ccc2ccccc2n1 ZINC000217869408 FG In-Stock Unstable FABK 0 46 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)C1CCC1 ZINC000217869412 DE For-Sale Unstable SCD1 16 41 C[C@H](NC(=O)c1ccc(Br)cc1)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217869440 HK In-Stock Unstable SDH1 0 48 CC[C@@H](N[C@H]1C[C@@H](C)CC[C@@H]1C(C)C)c1ccc(O)cc1 ZINC000217869462 CJ For-Sale Unstable TRPM8 16 43 CC[C@@H](C)[C@H](N)C(=O)N[C@H]1CCC[C@@H](O)C1 ZINC000217869488 BC For-Sale Unstable TPP2 39 41 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)C1CCC1 ZINC000217869500 DE For-Sale Unstable SCD1 16 41 C[C@H](C(=O)O)c1ccc(CO[C@@H]2CCC[C@@H](C)C2)cc1 ZINC000217869508 CH For-Sale Unstable PTGS1 31 52 C[C@H](C(=O)O)c1ccc(CO[C@@H]2CCC[C@@H](C)C2)cc1 ZINC000217869508 CH For-Sale Unstable PTGS2 0 52 CC[C@H](N[C@H]1C[C@@H](C)CC[C@@H]1C(C)C)c1ccc(O)cc1 ZINC000217869528 CJ For-Sale Unstable TRPM8 16 43 CC[C@@H]1COCCN1C[C@@H](O)COc1ccccc1CN ZINC000217869550 CC For-Sale Unstable ADRB2 42 48 CC[C@@H]1COCCN1C[C@@H](O)COc1ccccc1CN ZINC000217869550 CC For-Sale Unstable ADRB3 37 48 CC[C@@H]1COCCN1C[C@@H](O)COc1ccccc1CN ZINC000217869550 CC For-Sale Unstable ABCB1 55 39 Cc1ccc2c(c1)[C@@H](NC(=O)c1ccc(Br)cc1)CC(C)(C)O2 ZINC000217869563 FJ In-Stock Unstable PHZR 0 43 CC[C@@H]1C[C@@H](O)[C@@H](C)N1 ZINC000217869597 AC In-Stock Unstable FUCA2 48 30 CC[C@@H]1C[C@@H](O)[C@@H](C)N1 ZINC000217869597 AC In-Stock Unstable GAL1 0 53 CC[C@H]1COCCN1C[C@@H](O)COc1ccccc1CN ZINC000217869599 CC For-Sale Unstable ADRB2 42 48 CC[C@H]1COCCN1C[C@@H](O)COc1ccccc1CN ZINC000217869599 CC For-Sale Unstable ADRB3 37 48 CC[C@H]1COCCN1C[C@@H](O)COc1ccccc1CN ZINC000217869599 CC For-Sale Unstable ABCB1 55 39 Cc1ccc2c(c1)[C@H](NC(=O)c1ccc(Br)cc1)CC(C)(C)O2 ZINC000217869607 FJ In-Stock Unstable PHZR 0 43 C[C@H](C(=O)O)c1ccc(CO[C@H]2CCC[C@@H](C)C2)cc1 ZINC000217869632 CH For-Sale Unstable PTGS1 31 52 C[C@H](C(=O)O)c1ccc(CO[C@H]2CCC[C@@H](C)C2)cc1 ZINC000217869632 CH For-Sale Unstable PTGS2 0 52 CC[C@@H](C)[C@H](N)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217869644 BC For-Sale Unstable TPP2 41 43 Cc1noc(C)c1CC(=O)NCCn1nc(-c2ccncc2)cc1C ZINC000217869663 EE In-Stock Unstable P2RX7 35 49 CC[C@@H](N[C@@H]1C[C@@H](C)CC[C@@H]1C(C)C)c1ccccc1O ZINC000217869676 CJ For-Sale Unstable TRPM8 19 45 CC[C@H]1C[C@@H](O)[C@@H](C)N1 ZINC000217869677 AC In-Stock Unstable FUCA2 48 30 CC[C@H]1C[C@@H](O)[C@@H](C)N1 ZINC000217869677 AC In-Stock Unstable GAL1 0 53 Cc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1ccc(Br)cc1 ZINC000217869721 FJ In-Stock Unstable TRPV1 0 40 Cc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1ccc(Br)cc1 ZINC000217869721 FJ In-Stock Unstable PHZR 0 43 CC[C@H](C)[C@H](N)C(=O)N[C@H]1CCN2CCC[C@@H]12 ZINC000217869727 BC For-Sale Unstable TPP2 41 43 CC[C@@H]1C[C@H](O)[C@@H](C)N1 ZINC000217869745 AC In-Stock Unstable FUCA2 48 30 CC[C@@H]1C[C@H](O)[C@@H](C)N1 ZINC000217869745 AC In-Stock Unstable GAL1 0 53 CC[C@H](N[C@@H]1C[C@@H](C)CC[C@@H]1C(C)C)c1ccccc1O ZINC000217869746 CJ For-Sale Unstable TRPM8 0 45 Cc1cc(-c2ccncc2)nn1CCNC(=O)c1ccoc1 ZINC000217869750 CE In-Stock Unstable HSPB1 0 40 Cc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1ccc(Br)cc1 ZINC000217869783 FJ In-Stock Unstable TRPV1 0 40 Cc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1ccc(Br)cc1 ZINC000217869783 FJ In-Stock Unstable PHZR 0 43 CC[C@@H]1COCCN1C[C@@H](O)COc1cccc(CN)c1 ZINC000217869790 CC For-Sale Unstable ABCB1 37 44 C[C@H](C(=O)O)c1ccc(COC[C@@H]2CC=CC[C@@H]2C)cc1 ZINC000217869819 CH For-Sale Unstable PTGS1 27 47 C[C@H](C(=O)O)c1ccc(COC[C@@H]2CC=CC[C@@H]2C)cc1 ZINC000217869819 CH For-Sale Unstable PTGS2 0 47 CC[C@@H](N[C@H]1C[C@@H](C)CC[C@@H]1C(C)C)c1ccccc1O ZINC000217869831 CJ For-Sale Unstable TRPM8 19 45 CC[C@H]1C[C@H](O)[C@@H](C)N1 ZINC000217869832 AC In-Stock Unstable FUCA2 48 30 CC[C@H]1C[C@H](O)[C@@H](C)N1 ZINC000217869832 AC In-Stock Unstable GAL1 0 53 Cn1c(CCNC(=O)c2cc(=O)n(-c3ccccc3)[nH]2)nc2ccccc21 ZINC000217869849 FE In-Stock Unstable CTSA 60 41 C[C@H](C(=O)O)c1ccc(COC[C@H]2CC=CC[C@@H]2C)cc1 ZINC000217869858 CH For-Sale Unstable PTGS1 27 47 C[C@H](C(=O)O)c1ccc(COC[C@H]2CC=CC[C@@H]2C)cc1 ZINC000217869858 CH For-Sale Unstable PTGS2 0 47 CC[C@H]1COCCN1C[C@@H](O)COc1cccc(CN)c1 ZINC000217869863 CC For-Sale Unstable ABCB1 37 44 COc1ccc2c(c1)[C@@H](NC(=O)c1ccc(Br)cc1)CC(C)(C)O2 ZINC000217869902 GI In-Stock Unstable NAAA 22 45 Cc1cc(=O)n(Cc2ccccc2/C=C\C(=O)O)cn1 ZINC000217869908 CD For-Sale Unstable PTGER2 18 41 Cc1cc(=O)n(Cc2ccccc2/C=C\C(=O)O)cn1 ZINC000217869908 CD For-Sale Unstable PTGER3 22 44 CC[C@H](N[C@H]1C[C@@H](C)CC[C@@H]1C(C)C)c1ccccc1O ZINC000217869915 CJ For-Sale Unstable TRPM8 19 45 COc1ccc2c(c1)[C@H](NC(=O)c1ccc(Br)cc1)CC(C)(C)O2 ZINC000217869942 GI In-Stock Unstable NAAA 22 45 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCc1ccc(O)cc1O ZINC000217870040 CH For-Sale Unstable TRPM8 16 45 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1ccc(Br)cc1 ZINC000217870060 GI In-Stock Unstable NAAA 23 45 COCCCOCCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217870084 CE For-Sale Unstable PLA2G4B 61 35 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCc1ccc(O)cc1O ZINC000217870109 CH For-Sale Unstable TRPM8 16 45 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1ccc(Br)cc1 ZINC000217870126 GI In-Stock Unstable NAAA 23 45 COc1cc(CN2C[C@@H]3CC[C@H](C2)[C@@H]3O)ccc1OCC=C(C)C ZINC000217870146 EG In-Stock Unstable SSTR5 46 37 Cc1cc(-c2ccncc2)nn1CCNC(=O)c1ccccc1OC(F)(F)F ZINC000217870148 GH In-Stock Unstable KCNK3 49 43 Cc1cc(-c2ccncc2)nn1CCNC(=O)c1ccccc1OC(F)(F)F ZINC000217870148 GH In-Stock Unstable KCNK9 50 44 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCc1ccc(O)cc1O ZINC000217870192 CH For-Sale Unstable TRPM8 16 45 C=C=CC[C@@H](CC(=O)OC)NC(=O)OC(C)(C)C ZINC000217870202 CE For-Sale Unstable CTSK 17 44 O=C(O)/C=C\c1cc(F)ccc1COc1ccccc1 ZINC000217870205 CH For-Sale Unstable PTGER2 58 49 O=C(O)/C=C\c1cc(F)ccc1COc1ccccc1 ZINC000217870205 CH For-Sale Unstable PTGER4 31 49 O=C(O)/C=C\c1cc(F)ccc1COc1ccccc1 ZINC000217870205 CH For-Sale Unstable PTGER3 37 49 O=C(O)/C=C\c1cc(F)ccc1COc1ccccc1 ZINC000217870205 CH For-Sale Unstable PTGDR 0 47 O=C(O)/C=C\c1cc(F)ccc1COc1ccccc1 ZINC000217870205 CH For-Sale Unstable HCAR2 0 41 O=C(O)/C=C\c1cc(F)ccc1COc1ccccc1 ZINC000217870205 CH For-Sale Unstable FFAR1 18 44 O=C(O)/C=C\c1cc(F)ccc1COc1ccccc1 ZINC000217870205 CH For-Sale Unstable FFAR4 44 44 CC[C@@H](NC(=O)c1ccc(Br)cc1)c1ccc(C)c(C)c1 ZINC000217870217 EJ In-Stock Unstable TACR3 30 40 CC[C@@H](NC(=O)c1ccc(Br)cc1)c1ccc(C)c(C)c1 ZINC000217870217 EJ In-Stock Unstable UTS2 55 38 Cc1cc(-c2ccncc2)nn1CCNC(=O)Cc1ccc(F)cc1F ZINC000217870280 FF In-Stock Unstable P2RX7 29 42 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCc1ccc(O)cc1O ZINC000217870285 CH For-Sale Unstable TRPM8 16 45 O=C(O)/C=C\c1cc(COc2ccccc2)ccc1F ZINC000217870288 CH For-Sale Unstable MAOB 20 43 O=C(O)/C=C\c1cc(COc2ccccc2)ccc1F ZINC000217870288 CH For-Sale Unstable PTGER2 22 44 O=C(O)/C=C\c1cc(COc2ccccc2)ccc1F ZINC000217870288 CH For-Sale Unstable PTGER4 37 54 O=C(O)/C=C\c1cc(COc2ccccc2)ccc1F ZINC000217870288 CH For-Sale Unstable PTGER3 52 38 O=C(O)/C=C\c1cc(COc2ccccc2)ccc1F ZINC000217870288 CH For-Sale Unstable CDC25B 23 42 O=C(O)/C=C\c1cc(COc2ccccc2)ccc1F ZINC000217870288 CH For-Sale Unstable GYS1 45 34 O=C(O)/C=C\c1cc(COc2ccccc2)ccc1F ZINC000217870288 CH For-Sale Unstable PTGDR 0 52 O=C(O)/C=C\c1cc(COc2ccccc2)ccc1F ZINC000217870288 CH For-Sale Unstable HCAR2 0 40 O=C(O)/C=C\c1cc(COc2ccccc2)ccc1F ZINC000217870288 CH For-Sale Unstable FFAR1 57 44 O=C(O)/C=C\c1cc(COc2ccccc2)ccc1F ZINC000217870288 CH For-Sale Unstable AKR1C3 31 41 O=C(O)/C=C\c1cc(COc2ccccc2)ccc1F ZINC000217870288 CH For-Sale Unstable FFAR4 47 42 CC[C@H](NC(=O)c1ccc(Br)cc1)c1ccc(C)c(C)c1 ZINC000217870296 EJ In-Stock Unstable TACR3 30 40 CC[C@H](NC(=O)c1ccc(Br)cc1)c1ccc(C)c(C)c1 ZINC000217870296 EJ In-Stock Unstable UTS2 55 38 COc1c([C@H](N)CC(=O)O)ccc(F)c1Cl ZINC000217870323 BD For-Sale Unstable HMGCR 41 38 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cc(OC)c3c(c2)OCCO3)CC(=O)O4)cc1O ZINC000217870333 KI In-Stock Unstable AKR1B1 0 49 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cc(OC)c3c(c2)OCCO3)CC(=O)O4)cc1O ZINC000217870333 KI In-Stock Unstable CYP1B1 56 35 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cc(OC)c3c(c2)OCCO3)CC(=O)O4)cc1O ZINC000217870333 KI In-Stock Unstable CYP1A1 37 44 N#Cc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217870374 CG For-Sale Unstable PTGER2 16 45 N#Cc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217870374 CG For-Sale Unstable PTGER4 25 45 N#Cc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217870374 CG For-Sale Unstable PTGER3 25 48 N#Cc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217870374 CG For-Sale Unstable FFAR4 42 37 CC[C@@H]1COCCN1C[C@@H](O)COc1ccc(CN)cc1 ZINC000217870380 CC For-Sale Unstable ABCB1 26 42 Cc1ccc([C@H](C)N[C@H]2C[C@H](C)CC[C@H]2C(C)C)cc1C ZINC000217870403 CK For-Sale Unstable TRPM8 15 43 COc1c([C@@H](N)CC(=O)O)ccc(F)c1Cl ZINC000217870421 BD For-Sale Unstable HMGCR 41 38 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cc(OC)c3c(c2)OCCO3)CC(=O)O4)cc1O ZINC000217870423 KI In-Stock Unstable AKR1B1 0 49 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cc(OC)c3c(c2)OCCO3)CC(=O)O4)cc1O ZINC000217870423 KI In-Stock Unstable CYP1B1 56 35 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cc(OC)c3c(c2)OCCO3)CC(=O)O4)cc1O ZINC000217870423 KI In-Stock Unstable CYP1A1 37 44 O=C(N/C=C/c1ccccc1Br)NC1CCN(Cc2ccccc2)CC1 ZINC000217870446 HI For-Sale Unstable CHRM2 17 46 O=C(N/C=C/c1ccccc1Br)NC1CCN(Cc2ccccc2)CC1 ZINC000217870446 HI For-Sale Unstable CHRM1 15 46 O=C(N/C=C/c1ccccc1Br)NC1CCN(Cc2ccccc2)CC1 ZINC000217870446 HI For-Sale Unstable DRD2 18 58 O=C(N/C=C/c1ccccc1Br)NC1CCN(Cc2ccccc2)CC1 ZINC000217870446 HI For-Sale Unstable DRD4 46 58 O=C(N/C=C/c1ccccc1Br)NC1CCN(Cc2ccccc2)CC1 ZINC000217870446 HI For-Sale Unstable ACHE 38 48 O=C(N/C=C/c1ccccc1Br)NC1CCN(Cc2ccccc2)CC1 ZINC000217870446 HI For-Sale Unstable DRD3 26 58 O=C(N/C=C/c1ccccc1Br)NC1CCN(Cc2ccccc2)CC1 ZINC000217870446 HI For-Sale Unstable CHRM3 23 46 O=C(N/C=C/c1ccccc1Br)NC1CCN(Cc2ccccc2)CC1 ZINC000217870446 HI For-Sale Unstable SIGMAR1 58 60 O=C(N/C=C/c1ccccc1Br)NC1CCN(Cc2ccccc2)CC1 ZINC000217870446 HI For-Sale Unstable SSTR5 41 37 O=C(N/C=C/c1ccccc1Br)NC1CCN(Cc2ccccc2)CC1 ZINC000217870446 HI For-Sale Unstable CCR3 38 48 O=C(N/C=C/c1ccccc1Br)NC1CCN(Cc2ccccc2)CC1 ZINC000217870446 HI For-Sale Unstable SLC6A5 16 43 O=C(N/C=C/c1ccccc1Br)NC1CCN(Cc2ccccc2)CC1 ZINC000217870446 HI For-Sale Unstable EPHX2 17 52 O=C(N/C=C/c1ccccc1Br)NC1CCN(Cc2ccccc2)CC1 ZINC000217870446 HI For-Sale Unstable MCHR1 46 48 O=C(N/C=C/c1ccccc1Br)NC1CCN(Cc2ccccc2)CC1 ZINC000217870446 HI For-Sale Unstable CACNA1G 18 42 O=C(N/C=C/c1ccccc1Br)NC1CCN(Cc2ccccc2)CC1 ZINC000217870446 HI For-Sale Unstable ADIPOR1 0 47 O=C(N/C=C/c1ccccc1Br)NC1CCN(Cc2ccccc2)CC1 ZINC000217870446 HI For-Sale Unstable ADIPOR2 0 47 O=C(O)/C=C\c1ccccc1COC[C@@H]1CCCCO1 ZINC000217870462 CF For-Sale Unstable PTGER2 42 42 O=C(O)/C=C\c1ccccc1COC[C@@H]1CCCCO1 ZINC000217870462 CF For-Sale Unstable PTGER4 0 42 O=C(O)/C=C\c1ccccc1COC[C@@H]1CCCCO1 ZINC000217870462 CF For-Sale Unstable PTGER3 15 42 CC[C@H]1COCCN1C[C@@H](O)COc1ccc(CN)cc1 ZINC000217870468 CC For-Sale Unstable ABCB1 26 42 Cc1ccc([C@H](C)N[C@H]2C[C@@H](C)CC[C@H]2C(C)C)cc1C ZINC000217870482 CK For-Sale Unstable TRPM8 15 43 CO[C@@H]1CCC[C@@H](OCc2ccc([C@@H](C)C(=O)O)cc2)C1 ZINC000217870484 CG For-Sale Unstable PTGS1 34 52 CO[C@@H]1CCC[C@@H](OCc2ccc([C@@H](C)C(=O)O)cc2)C1 ZINC000217870484 CG For-Sale Unstable PTGS2 23 52 CO[C@@H]1CCC[C@@H](OCc2ccc([C@@H](C)C(=O)O)cc2)C1 ZINC000217870484 CG For-Sale Unstable SLC22A20 0 48 Cc1cc(-c2ccncc2)nn1CCNC(=O)Nc1ccccc1 ZINC000217870485 DG In-Stock Unstable CCKAR 18 40 Cc1cc(-c2ccncc2)nn1CCNC(=O)Nc1ccccc1 ZINC000217870485 DG In-Stock Unstable ROCK1 27 46 Cc1cc(-c2ccncc2)nn1CCNC(=O)Nc1ccccc1 ZINC000217870485 DG In-Stock Unstable ROCK2 26 42 Cc1cc(-c2ccncc2)nn1CCNC(=O)Nc1ccccc1 ZINC000217870485 DG In-Stock Unstable CYP2C9 15 41 Cc1cc(-c2ccncc2)nn1CCNC(=O)Nc1ccccc1 ZINC000217870485 DG In-Stock Unstable QPCT 41 39 Cc1cc(-c2ccncc2)nn1CCNC(=O)Nc1ccccc1 ZINC000217870485 DG In-Stock Unstable SMG1 40 31 Cc1cc(-c2ccncc2)nn1CCNC(=O)Nc1ccccc1 ZINC000217870485 DG In-Stock Unstable GPR142 23 41 NC(=O)c1ccc(NC(=O)CC[C@@H]2NC(=O)N(CCc3ccccc3)C2=O)cc1 ZINC000217870531 GD In-Stock Unstable LTA4H 22 40 O=C(O)/C=C\c1ccccc1COC[C@H]1CCCCO1 ZINC000217870546 CF For-Sale Unstable PTGER2 42 42 O=C(O)/C=C\c1ccccc1COC[C@H]1CCCCO1 ZINC000217870546 CF For-Sale Unstable PTGER4 0 42 O=C(O)/C=C\c1ccccc1COC[C@H]1CCCCO1 ZINC000217870546 CF For-Sale Unstable PTGER3 15 42 CO[C@@H]1CCC[C@H](OCc2ccc([C@@H](C)C(=O)O)cc2)C1 ZINC000217870548 CG For-Sale Unstable PTGS1 34 52 CO[C@@H]1CCC[C@H](OCc2ccc([C@@H](C)C(=O)O)cc2)C1 ZINC000217870548 CG For-Sale Unstable PTGS2 23 52 CO[C@@H]1CCC[C@H](OCc2ccc([C@@H](C)C(=O)O)cc2)C1 ZINC000217870548 CG For-Sale Unstable SLC22A20 0 48 Cc1ccc([C@H](C)N[C@H]2C[C@@H](C)CC[C@@H]2C(C)C)cc1C ZINC000217870554 CK For-Sale Unstable TRPM8 15 43 CC[C@@H](NC(=O)c1ccc(Br)cc1)c1ccc(OC)c(OC)c1 ZINC000217870563 GI In-Stock Unstable PPARD 16 44 CC[C@@H](NC(=O)c1ccc(Br)cc1)c1ccc(OC)c(OC)c1 ZINC000217870563 GI In-Stock Unstable UTS2 66 41 COc1ccc(CNC(=O)NCCn2nc(-c3ccncc3)cc2C)cc1 ZINC000217870606 FF In-Stock Unstable ROCK1 26 43 COc1ccc(CNC(=O)NCCn2nc(-c3ccncc3)cc2C)cc1 ZINC000217870606 FF In-Stock Unstable ROCK2 28 43 COc1ccc(CNC(=O)NCCn2nc(-c3ccncc3)cc2C)cc1 ZINC000217870606 FF In-Stock Unstable PROKR1 40 31 CC[C@H](NC(=O)c1ccc(Br)cc1)c1ccc(OC)c(OC)c1 ZINC000217870632 GI In-Stock Unstable PPARD 16 44 CC[C@H](NC(=O)c1ccc(Br)cc1)c1ccc(OC)c(OC)c1 ZINC000217870632 GI In-Stock Unstable UTS2 57 41 COc1ccc([C@@H](C)N2CCC[C@@H](C)CC2)c(O)c1 ZINC000217870640 CH For-Sale Unstable RORC 40 39 COc1ccc2cc([C@@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(OC)c(O)c6)oc5c43)c(=O)[nH]c2c1 ZINC000217870648 KI In-Stock Unstable AKR1B1 0 42 COc1ccc2cc([C@@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(OC)c(O)c6)oc5c43)c(=O)[nH]c2c1 ZINC000217870648 KI In-Stock Unstable CYP1A1 30 42 CC[C@@H](NC(=O)c1ccc(Br)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217870718 GH In-Stock Unstable CA2 18 42 CC[C@@H](NC(=O)c1ccc(Br)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217870718 GH In-Stock Unstable LOX1.1 42 38 CC[C@@H](NC(=O)c1ccc(Br)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217870718 GH In-Stock Unstable O49150_SOLTU 50 38 CC[C@@H](NC(=O)c1ccc(Br)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217870718 GH In-Stock Unstable UTS2 56 38 COc1ccc2cc([C@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(OC)c(O)c6)oc5c43)c(=O)[nH]c2c1 ZINC000217870737 KI In-Stock Unstable AKR1B1 0 42 COc1ccc2cc([C@H]3CC(=O)Oc4cc(O)c5c(=O)cc(-c6ccc(OC)c(O)c6)oc5c43)c(=O)[nH]c2c1 ZINC000217870737 KI In-Stock Unstable CYP1A1 30 42 COc1cc(C[C@H](N)C(=O)O)cc(F)c1Cl ZINC000217870739 BD For-Sale Unstable CACNA2D1 29 41 O=C(N/C=C/c1ccccc1Br)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217870755 IH For-Sale Unstable BMP1 23 41 O=C(N/C=C/c1ccccc1Br)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217870755 IH For-Sale Unstable SSTR3 52 31 O=C(N/C=C/c1ccccc1Br)N1CCN(Cc2ccc3c(c2)OCO3)CC1 ZINC000217870755 IH For-Sale Unstable MCHR1 26 50 CC[C@H](NC(=O)c1ccc(Br)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217870784 GH In-Stock Unstable CA2 18 42 CC[C@H](NC(=O)c1ccc(Br)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217870784 GH In-Stock Unstable LOX1.1 42 38 CC[C@H](NC(=O)c1ccc(Br)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217870784 GH In-Stock Unstable O49150_SOLTU 50 38 CC[C@H](NC(=O)c1ccc(Br)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217870784 GH In-Stock Unstable UTS2 56 38 COc1cc(C[C@@H](N)C(=O)O)cc(F)c1Cl ZINC000217870797 BD For-Sale Unstable CACNA2D1 29 41 C[C@H](C(=O)O)c1ccc(COC2C[C@H](C)C[C@@H](C)C2)cc1 ZINC000217870800 CI For-Sale Unstable PTGS1 32 53 C[C@H](C(=O)O)c1ccc(COC2C[C@H](C)C[C@@H](C)C2)cc1 ZINC000217870800 CI For-Sale Unstable PTGS2 22 53 C[C@H](C(=O)O)c1ccc(COC2C[C@H](C)C[C@@H](C)C2)cc1 ZINC000217870800 CI For-Sale Unstable SLC22A20 0 53 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)NCCCn3ccnc3)[C@H]21 ZINC000217870827 JF In-Stock Unstable TBXAS1 20 40 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)NCCCn3ccnc3)[C@H]21 ZINC000217870827 JF In-Stock Unstable QPCT 34 45 CCOC(=O)N1CCN(C(=O)N/C=C/c2ccccc2Br)CC1 ZINC000217870832 GF For-Sale Unstable P2RY12 51 38 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)NCCCn3ccnc3)[C@@H]21 ZINC000217870873 JF In-Stock Unstable TBXAS1 20 40 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)NCCCn3ccnc3)[C@@H]21 ZINC000217870873 JF In-Stock Unstable QPCT 34 45 C[C@H](C(=O)O)c1ccc(CO[C@@H]2CC[C@@H](C)[C@@H](C)C2)cc1 ZINC000217870901 CI For-Sale Unstable PTGS1 32 50 C[C@H](C(=O)O)c1ccc(CO[C@@H]2CC[C@@H](C)[C@@H](C)C2)cc1 ZINC000217870901 CI For-Sale Unstable PTGS2 24 50 C[C@H](C(=O)O)c1ccc(CO[C@@H]2CC[C@@H](C)[C@@H](C)C2)cc1 ZINC000217870901 CI For-Sale Unstable SLC22A20 0 50 COc1ccc(-c2noc(CNC(=O)c3ccc(Br)cc3)n2)c(OC)c1 ZINC000217870926 HG In-Stock Unstable HRH3 17 40 COc1ccc(-c2noc(CNC(=O)c3ccc(Br)cc3)n2)c(OC)c1 ZINC000217870926 HG In-Stock Unstable PPARD 15 44 COc1ccc(-c2noc(CNC(=O)c3ccc(Br)cc3)n2)c(OC)c1 ZINC000217870926 HG In-Stock Unstable MT-ND1 18 45 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCc1c(Cl)cccc1Cl ZINC000217870947 DK For-Sale Unstable TRPM8 17 49 CCCCCCOCc1cc(/C=C\C(=O)O)ccc1OC ZINC000217870989 CH For-Sale Unstable PTGER2 0 42 CCCCCCOCc1cc(/C=C\C(=O)O)ccc1OC ZINC000217870989 CH For-Sale Unstable LTB4R 40 43 CCCCCCOCc1cc(/C=C\C(=O)O)ccc1OC ZINC000217870989 CH For-Sale Unstable PLA2G4B 79 41 CCCCCCOCc1cc(/C=C\C(=O)O)ccc1OC ZINC000217870989 CH For-Sale Unstable TUBB1 42 37 CCCCCCOCc1cc(/C=C\C(=O)O)ccc1OC ZINC000217870989 CH For-Sale Unstable AKR1C3 30 46 COC(=O)C[C@@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(OC)c(CO)c1 ZINC000217871014 GF In-Stock Unstable TNF 20 40 O=C(NCc1nc(-c2cccc(Br)c2)no1)c1ccc(Br)cc1 ZINC000217871029 II In-Stock Unstable KCNQ1 0 43 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCc1c(Cl)cccc1Cl ZINC000217871037 DK For-Sale Unstable TRPM8 17 49 CC[C@@H](C)[C@H](N)C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217871063 CD For-Sale Unstable TPP2 38 40 COC(=O)C[C@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(OC)c(CO)c1 ZINC000217871093 GF In-Stock Unstable TNF 20 40 C[C@@H]1CCCN([C@H](C)Cc2ccc(O)cc2)CC1 ZINC000217871097 BG For-Sale Unstable EBP 15 41 O=C(O)/C=C\c1cccc(COCCc2cccs2)c1 ZINC000217871104 CH For-Sale Unstable PTGER2 36 45 O=C(O)/C=C\c1cccc(COCCc2cccs2)c1 ZINC000217871104 CH For-Sale Unstable PTGER4 0 45 O=C(O)/C=C\c1cccc(COCCc2cccs2)c1 ZINC000217871104 CH For-Sale Unstable LTB4R 17 42 O=C(O)/C=C\c1cccc(COCCc2cccs2)c1 ZINC000217871104 CH For-Sale Unstable HCAR2 0 40 O=C(O)/C=C\c1cccc(COCCc2cccs2)c1 ZINC000217871104 CH For-Sale Unstable AKR1C3 35 44 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCc1c(Cl)cccc1Cl ZINC000217871112 DK For-Sale Unstable TRPM8 17 49 COc1cccc(-c2noc(CN(C)C(=O)c3ccc(Br)cc3)n2)c1 ZINC000217871124 HH In-Stock Unstable HSD17B2 27 54 O=C(N/C=C/c1ccccc1Br)Nc1ccc(C(F)(F)F)cc1 ZINC000217871129 GK For-Sale Anodyne EPHX2 26 41 O=C(N/C=C/c1ccccc1Br)Nc1ccc(C(F)(F)F)cc1 ZINC000217871129 GK For-Sale Anodyne PTPA 0 40 O=C(N/C=C/c1ccccc1Br)Nc1ccc(C(F)(F)F)cc1 ZINC000217871129 GK For-Sale Anodyne MTCA1 15 46 O=C(N/C=C/c1ccccc1Br)Nc1ccc(C(F)(F)F)cc1 ZINC000217871129 GK For-Sale Anodyne P96878_MYCTU 15 46 CC[C@H](C)[C@H](N)C(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217871146 CD On-Demand Unstable TPP2 38 40 O=C(O)/C=C\c1cc(F)ccc1COCCc1cccs1 ZINC000217871168 DH For-Sale Unstable PTGER2 43 45 O=C(O)/C=C\c1cc(F)ccc1COCCc1cccs1 ZINC000217871168 DH For-Sale Unstable PTGER4 25 45 O=C(O)/C=C\c1cc(F)ccc1COCCc1cccs1 ZINC000217871168 DH For-Sale Unstable PTGER3 19 45 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCc1c(Cl)cccc1Cl ZINC000217871194 DK For-Sale Unstable TRPM8 17 49 COc1cc(C[C@H](N)C(=O)O)cc(Cl)c1F ZINC000217871214 BD For-Sale Unstable CACNA2D1 28 41 O=C(O)/C=C\c1cc(COCCc2cccs2)ccc1F ZINC000217871271 DH For-Sale Unstable PTGER2 42 48 O=C(O)/C=C\c1cc(COCCc2cccs2)ccc1F ZINC000217871271 DH For-Sale Unstable PTGER4 24 48 O=C(O)/C=C\c1cc(COCCc2cccs2)ccc1F ZINC000217871271 DH For-Sale Unstable PTGER3 19 48 O=C(c1ccc2cc[nH]c2c1)N1CC(Oc2ccc(F)cc2)C1 ZINC000217871283 DG In-Stock Unstable GHSR 0 56 COc1cc(C[C@@H](N)C(=O)O)cc(Cl)c1F ZINC000217871315 BD For-Sale Unstable CACNA2D1 28 41 COc1ccc(OC)c(S(=O)(=O)NCCn2nc(-c3ccncc3)cc2C)c1 ZINC000217871355 HE In-Stock Unstable LRRK2 23 40 Cn1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cn1 ZINC000217871370 HG In-Stock Unstable AKR1B1 0 42 O=C(O)/C=C\c1cccc(OCCSc2ccccc2)c1 ZINC000217871377 DH For-Sale Unstable PTGER3 15 42 O=C(O)/C=C\c1cccc(OCCSc2ccccc2)c1 ZINC000217871377 DH For-Sale Unstable LTB4R 23 40 O=C(O)/C=C\c1cccc(OCCSc2ccccc2)c1 ZINC000217871377 DH For-Sale Unstable AKR1C3 29 40 CC(C)c1ccc(CCCNC(=O)c2ccc(Br)cc2)cc1 ZINC000217871393 FJ In-Stock Unstable SDH1 0 40 CC(C)c1ccc(CCCNC(=O)c2ccc(Br)cc2)cc1 ZINC000217871393 FJ In-Stock Unstable AMP1_PLAFQ 26 40 CC(C)c1ccc(CCCNC(=O)c2ccc(Br)cc2)cc1 ZINC000217871393 FJ In-Stock Unstable HDA106 0 40 CCCCN1C[C@@H](O)C[C@@H]1C ZINC000217871407 AD In-Stock Unstable GBA2 46 38 O=C(O)/C=C\c1ccc(OCCSc2ccccc2)cc1 ZINC000217871424 DH For-Sale Unstable PTGER2 32 42 O=C(O)/C=C\c1ccc(OCCSc2ccccc2)cc1 ZINC000217871424 DH For-Sale Unstable PTGER4 15 42 O=C(O)/C=C\c1ccc(OCCSc2ccccc2)cc1 ZINC000217871424 DH For-Sale Unstable LTB4R 20 41 O=C(O)/C=C\c1ccc(OCCSc2ccccc2)cc1 ZINC000217871424 DH For-Sale Unstable PLA2G4B 40 38 Cn1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cn1 ZINC000217871430 HG In-Stock Unstable AKR1B1 0 42 C[C@@H]1CCCN([C@H](C)CCc2ccc(O)cc2)CC1 ZINC000217871455 CH For-Sale Unstable EBP 17 43 C[C@@H]1CCCN([C@H](C)CCc2ccc(O)cc2)CC1 ZINC000217871455 CH For-Sale Unstable BIRC2 33 41 CCCCN1C[C@H](O)C[C@@H]1C ZINC000217871502 AD In-Stock Unstable GBA2 46 38 O=C(NCCCN1CCCc2ccccc21)c1ccc(Br)cc1 ZINC000217871508 FI In-Stock Unstable HTR1A 16 40 O=C(NCCCN1CCCc2ccccc21)c1ccc(Br)cc1 ZINC000217871508 FI In-Stock Unstable DRD2 29 42 O=C(NCCCN1CCCc2ccccc21)c1ccc(Br)cc1 ZINC000217871508 FI In-Stock Unstable DRD1 19 41 O=C(NCCCN1CCCc2ccccc21)c1ccc(Br)cc1 ZINC000217871508 FI In-Stock Unstable HTR2C 16 41 O=C(NCCCN1CCCc2ccccc21)c1ccc(Br)cc1 ZINC000217871508 FI In-Stock Unstable AVPR2 35 43 O=C(NCCCN1CCCc2ccccc21)c1ccc(Br)cc1 ZINC000217871508 FI In-Stock Unstable DRD3 50 42 O=C(NCCCN1CCCc2ccccc21)c1ccc(Br)cc1 ZINC000217871508 FI In-Stock Unstable AVPR1A 21 40 O=C(NCCCN1CCCc2ccccc21)c1ccc(Br)cc1 ZINC000217871508 FI In-Stock Unstable HTR3B 0 41 O=C(NCCCN1CCCc2ccccc21)c1ccc(Br)cc1 ZINC000217871508 FI In-Stock Unstable TYRO3 21 40 O=C(NCCCN1CCCc2ccccc21)c1ccc(Br)cc1 ZINC000217871508 FI In-Stock Unstable ALPHA-1A 0 41 CC[C@@H](C)[C@H](N)C(=O)N[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217871532 CF For-Sale Unstable TRPM8 18 48 Cc1ccc(SCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217871551 CI For-Sale Unstable PTGER2 27 43 Cc1ccc(SCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217871551 CI For-Sale Unstable LTB4R 18 46 Cc1ccc(SCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217871551 CI For-Sale Unstable AKR1C3 36 44 Cc1ccc(SCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217871551 CI For-Sale Unstable GPR183 0 40 COc1cccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)c1OC ZINC000217871573 JI In-Stock Unstable AKR1B1 22 48 COc1cccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)c1OC ZINC000217871573 JI In-Stock Unstable CYP1B1 68 39 COc1cccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)c1OC ZINC000217871573 JI In-Stock Unstable CYP1A1 50 47 COc1cccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)c1OC ZINC000217871573 JI In-Stock Unstable CYP1A2 43 47 O[C@]1(c2ccc(Cl)c(Cl)c2)C[C@@H]2C[C@@H]1[C@@H]1CCC[C@@H]21 ZINC000217871625 CJ For-Sale Unstable SLC6A3 0 40 COc1cccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)c1OC ZINC000217871650 JI In-Stock Unstable AKR1B1 22 48 COc1cccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)c1OC ZINC000217871650 JI In-Stock Unstable CYP1B1 68 39 COc1cccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)c1OC ZINC000217871650 JI In-Stock Unstable CYP1A1 50 47 COc1cccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)c1OC ZINC000217871650 JI In-Stock Unstable CYP1A2 43 47 O=C(O)/C=C\c1ccccc1CSc1ccccc1F ZINC000217871652 CI For-Sale Unstable PTGER2 43 50 O=C(O)/C=C\c1ccccc1CSc1ccccc1F ZINC000217871652 CI For-Sale Unstable PTGER4 0 50 O=C(O)/C=C\c1ccccc1CSc1ccccc1F ZINC000217871652 CI For-Sale Unstable PTGER3 17 51 O=C(O)/C=C\c1ccccc1CSc1ccccc1F ZINC000217871652 CI For-Sale Unstable PTGDR 0 51 CCOc1ccc(CNC(=O)c2ccc(Cl)c([N+](=O)[O-])c2)cc1OCC ZINC000217871659 GH In-Stock Unstable TAAR1 18 45 Cc1cc(-c2ccncc2)nn1CCNS(=O)(=O)c1ccc(F)c(F)c1 ZINC000217871662 GF In-Stock Unstable TBXAS1 27 41 O=C(O)/C=C\c1ccc(CSc2ccccc2F)cc1 ZINC000217871720 CI For-Sale Unstable PTGER2 29 43 O=C(O)/C=C\c1ccc(CSc2ccccc2F)cc1 ZINC000217871720 CI For-Sale Unstable PTGER4 0 43 O=C(O)/C=C\c1ccc(CSc2ccccc2F)cc1 ZINC000217871720 CI For-Sale Unstable NPY2R 0 44 O=C(O)/C=C\c1ccc(CSc2ccccc2F)cc1 ZINC000217871720 CI For-Sale Unstable PTGDR 0 41 O=C(O)/C=C\c1ccc(CSc2ccccc2F)cc1 ZINC000217871720 CI For-Sale Unstable AKR1C3 31 43 O[C@@]1(c2ccc(Cl)c(Cl)c2)C[C@@H]2C[C@@H]1[C@@H]1CCC[C@@H]21 ZINC000217871723 CJ For-Sale Unstable SLC6A3 0 40 COc1ccccc1CCCNC(=O)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217871738 EH In-Stock Unstable DRD2 23 43 COc1ccccc1CCCNC(=O)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217871738 EH In-Stock Unstable DRD1 0 42 COc1ccccc1CCCNC(=O)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217871738 EH In-Stock Unstable DRD3 39 43 COc1ccccc1CCCNC(=O)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217871738 EH In-Stock Unstable MTNR1B 24 40 COc1ccccc1CCCNC(=O)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217871738 EH In-Stock Unstable TAAR1 26 53 COc1ccccc1CCCNC(=O)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217871738 EH In-Stock Unstable AP2S1 0 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccncc1 ZINC000217871740 EE For-Sale Unstable HCRTR2 42 36 O[C@]1(c2ccc(Cl)c(Cl)c2)C[C@H]2C[C@@H]1[C@@H]1CCC[C@@H]21 ZINC000217871759 CJ For-Sale Unstable SLC6A3 0 40 O=C(N/C=C/c1ccccc1Br)N1CCN(c2ccccn2)CC1 ZINC000217871796 GG For-Sale Unstable SLC6A7 0 45 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccncc1 ZINC000217871820 EE For-Sale Unstable HCRTR2 42 36 CCC[C@@H](O)CNCCCCCO ZINC000217871828 AC For-Sale Unstable Q8WS26_TRYCR 36 41 CCC[C@@H](O)CNCCCCCO ZINC000217871828 AC For-Sale Unstable FPPS 0 41 CCC[C@@H](O)CNCCCCCO ZINC000217871828 AC For-Sale Unstable SPPS 0 41 O=C(Nc1ccccc1C(=O)c1ccccc1)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217871831 GJ In-Stock Bother PYGL 25 41 O=C(Nc1ccccc1C(=O)c1ccccc1)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217871831 GJ In-Stock Bother PPARD 0 41 O=C(Nc1ccccc1C(=O)c1ccccc1)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217871831 GJ In-Stock Bother NR1H4 0 44 O=C(Nc1ccccc1C(=O)c1ccccc1)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217871831 GJ In-Stock Bother FABH 0 43 O=C(Nc1ccccc1C(=O)c1ccccc1)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217871831 GJ In-Stock Bother TAAR1 27 52 O=C(Nc1ccccc1C(=O)c1ccccc1)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217871831 GJ In-Stock Bother AKR1C3 18 45 O=C(Nc1ccccc1C(=O)c1ccccc1)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217871831 GJ In-Stock Bother PAGA 0 42 O=C(Nc1ccccc1C(=O)c1ccccc1)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217871831 GJ In-Stock Bother SMO 17 40 O=C(Nc1ccccc1C(=O)c1ccccc1)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217871831 GJ In-Stock Bother KCNK3 48 40 O[C@@]1(c2ccc(Cl)c(Cl)c2)C[C@H]2C[C@@H]1[C@@H]1CCC[C@@H]21 ZINC000217871841 CJ For-Sale Unstable SLC6A3 0 40 COc1ccc(CSc2nncs2)cc1/C=C\C(=O)O ZINC000217871843 DF For-Sale Unstable PTGER2 25 40 COc1ccc(CSc2nncs2)cc1/C=C\C(=O)O ZINC000217871843 DF For-Sale Unstable PTGER4 16 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccncc1 ZINC000217871900 EE For-Sale Unstable HCRTR2 42 36 COc1cc([C@@H](C)N2CCC[C@@H](C)CC2)ccc1O ZINC000217871910 CH For-Sale Unstable RORC 46 39 CCC[C@H](O)CNCCCCCO ZINC000217871915 AC For-Sale Unstable Q8WS26_TRYCR 36 41 CCC[C@H](O)CNCCCCCO ZINC000217871915 AC For-Sale Unstable FPPS 0 41 CCC[C@H](O)CNCCCCCO ZINC000217871915 AC For-Sale Unstable SPPS 0 41 CSCc1ccc(C(=O)N2CCCC[C@@H]2c2ccccn2)o1 ZINC000217871921 DH In-Stock Unstable COLA 108 41 CSCc1ccc(C(=O)N2CCCC[C@@H]2c2ccccn2)o1 ZINC000217871921 DH In-Stock Unstable CPT1A 103 41 CCOc1ccc(CCCNC(=O)c2ccc(Cl)c([N+](=O)[O-])c2)cc1 ZINC000217871922 FI In-Stock Unstable TAAR1 19 46 CCOc1ccc(CCCNC(=O)c2ccc(Cl)c([N+](=O)[O-])c2)cc1 ZINC000217871922 FI In-Stock Unstable CRTM 43 36 O=C1C[C@@H](c2cccc(O)c2)c2c(ccc3c(=O)c(-c4ccc(O)cc4)coc23)O1 ZINC000217871967 HI In-Stock Unstable ALDH2 91 38 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccncc1 ZINC000217871994 EE For-Sale Unstable HCRTR2 42 36 CSCc1ccc(C(=O)N2CCCC[C@H]2c2ccccn2)o1 ZINC000217872004 DH In-Stock Unstable COLA 108 41 CSCc1ccc(C(=O)N2CCCC[C@H]2c2ccccn2)o1 ZINC000217872004 DH In-Stock Unstable CPT1A 103 41 CCCOc1ccccc1CCCNC(=O)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217872021 GI In-Stock Unstable TAAR1 21 45 O=C1C[C@H](c2cccc(O)c2)c2c(ccc3c(=O)c(-c4ccc(O)cc4)coc23)O1 ZINC000217872038 HI In-Stock Unstable ALDH2 91 38 Cc1ccccc1OC[C@@H](C)NC(=O)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217872103 EH In-Stock Unstable TAAR1 25 51 Cc1ccccc1OC[C@H](C)NC(=O)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217872188 EH In-Stock Unstable TAAR1 25 51 CC[C@@H](O)CCNCc1cccc(OC(F)(F)F)c1 ZINC000217872199 CF On-Demand Unstable CETP 0 47 CC[C@@H](O)CCNCc1cccc(OC(F)(F)F)c1 ZINC000217872199 CF On-Demand Unstable PHES 0 42 CC[C@@H](O)CCNCc1cccc(OC(F)(F)F)c1 ZINC000217872199 CF On-Demand Unstable PDS 70 37 CCN(C)C(=O)CNC(=O)c1cc(N)cc(Cl)c1 ZINC000217872262 CD For-Sale Unstable CACNA1I 42 33 Cc1ccc(OC[C@H](C)NC(=O)c2ccc(Cl)c([N+](=O)[O-])c2)cc1 ZINC000217872270 EH In-Stock Unstable TAAR1 18 48 CC[C@H](O)CCNCc1cccc(OC(F)(F)F)c1 ZINC000217872273 CF On-Demand Unstable CETP 0 47 CC[C@H](O)CCNCc1cccc(OC(F)(F)F)c1 ZINC000217872273 CF On-Demand Unstable PHES 0 42 CC[C@H](O)CCNCc1cccc(OC(F)(F)F)c1 ZINC000217872273 CF On-Demand Unstable PDS 70 37 NCc1ccc(C(=O)N[C@@H]2C[C@@H]3C[C@@H]2[C@@H]2CCC[C@@H]32)cc1 ZINC000217872284 CF For-Sale Unstable SSTR3 28 42 C[C@@H]1CCCN([C@H](C)c2cc(Cl)ccc2O)CC1 ZINC000217872316 CI For-Sale Unstable EBP 19 41 COC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217872341 GI For-Sale Unstable CCKAR 0 41 COC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217872341 GI For-Sale Unstable PARP14 0 41 COC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217872341 GI For-Sale Unstable PARP15 0 41 COC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217872341 GI For-Sale Unstable KCNK3 102 36 COC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217872341 GI For-Sale Unstable KCNK9 64 36 COC(=O)c1cccc(NC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217872341 GI For-Sale Unstable PARP10 0 41 COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc(OC)c1OC ZINC000217872345 JI In-Stock Unstable ALOX5 0 51 COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc(OC)c1OC ZINC000217872345 JI In-Stock Unstable AKR1B1 25 51 COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc(OC)c1OC ZINC000217872345 JI In-Stock Unstable CYP1B1 75 44 COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc(OC)c1OC ZINC000217872345 JI In-Stock Unstable CYP1A1 55 44 COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc(OC)c1OC ZINC000217872345 JI In-Stock Unstable CYP1A2 46 52 COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc(OC)c1OC ZINC000217872345 JI In-Stock Unstable ABCG2 0 40 NCc1ccc(C(=O)N[C@H]2C[C@@H]3C[C@@H]2[C@@H]2CCC[C@@H]32)cc1 ZINC000217872363 CF For-Sale Unstable SSTR3 28 42 COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc(OC)c1OC ZINC000217872423 JI In-Stock Unstable ALOX5 0 51 COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc(OC)c1OC ZINC000217872423 JI In-Stock Unstable AKR1B1 25 51 COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc(OC)c1OC ZINC000217872423 JI In-Stock Unstable CYP1B1 75 44 COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc(OC)c1OC ZINC000217872423 JI In-Stock Unstable CYP1A1 55 44 COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc(OC)c1OC ZINC000217872423 JI In-Stock Unstable CYP1A2 46 52 COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc(OC)c1OC ZINC000217872423 JI In-Stock Unstable ABCG2 0 40 CCN(C)C(=O)CNC(=O)c1cccc(Cl)c1N ZINC000217872434 CD For-Sale Unstable ECR 48 36 NCc1ccc(C(=O)N[C@@H]2C[C@H]3C[C@@H]2[C@@H]2CCC[C@@H]32)cc1 ZINC000217872445 CF For-Sale Unstable SSTR3 28 42 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccccc1C ZINC000217872457 FF For-Sale Unstable HCRTR1 53 37 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccccc1C ZINC000217872457 FF For-Sale Unstable HCRTR2 58 37 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccccc1C ZINC000217872513 FF For-Sale Unstable HCRTR1 53 37 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccccc1C ZINC000217872513 FF For-Sale Unstable HCRTR2 58 37 NCc1ccc(C(=O)N[C@H]2C[C@H]3C[C@@H]2[C@@H]2CCC[C@@H]32)cc1 ZINC000217872522 CF For-Sale Unstable SSTR3 28 42 COc1ccccc1-c1nc(NC(=O)CCCNc2ccc3c(cc2=O)[C@@H](NC(C)=O)CCc2cc(OC)c(OC)c(OC)c2-3)n[nH]1 ZINC000217872538 KI In-Stock Unstable TUBA1A 16 58 COc1ccccc1-c1nc(NC(=O)CCCNc2ccc3c(cc2=O)[C@@H](NC(C)=O)CCc2cc(OC)c(OC)c(OC)c2-3)n[nH]1 ZINC000217872538 KI In-Stock Unstable TPPP 0 55 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccccc1C ZINC000217872563 FF For-Sale Unstable HCRTR1 53 37 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccccc1C ZINC000217872563 FF For-Sale Unstable HCRTR2 58 37 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccccc1C ZINC000217872647 FF For-Sale Unstable HCRTR1 53 37 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccccc1C ZINC000217872647 FF For-Sale Unstable HCRTR2 58 37 COc1ncc(Br)cc1Nc1ncc([N+](=O)[O-])c(NC2CCCCC2)n1 ZINC000217872686 HI For-Sale Unstable PRKCQ 46 40 CCO[C@@H]1C[C@@H](NCc2cccc(O)c2)C1(C)C ZINC000217872751 BF For-Sale Unstable SLC6A13 0 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccccc1F ZINC000217872783 FF For-Sale Unstable HCRTR1 54 39 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccccc1F ZINC000217872783 FF For-Sale Unstable HCRTR2 59 39 Cc1ccccc1CNC(=O)N/C=C/c1ccccc1Br ZINC000217872786 EI For-Sale Unstable ANPEP 15 48 Cc1ccccc1CNC(=O)N/C=C/c1ccccc1Br ZINC000217872786 EI For-Sale Unstable AMP1_PLAFQ 18 43 CCO[C@H]1C[C@@H](NCc2cccc(O)c2)C1(C)C ZINC000217872843 BF For-Sale Unstable SLC6A13 0 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccccc1F ZINC000217872868 FF For-Sale Unstable HCRTR1 54 39 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccccc1F ZINC000217872868 FF For-Sale Unstable HCRTR2 59 39 Cc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217872877 FJ In-Stock Unstable TAAR1 17 43 C[C@H](C(=O)O)c1ccc(CS[C@@H]2CCC[C@@H](C)C2)cc1 ZINC000217872879 CJ For-Sale Unstable PTGS1 25 52 C[C@H](C(=O)O)c1ccc(CS[C@@H]2CCC[C@@H](C)C2)cc1 ZINC000217872879 CJ For-Sale Unstable SLC22A20 0 44 Cc1cc(-c2cccs2)nn1CCNC(=O)c1cncc(Br)c1 ZINC000217872885 GH In-Stock Unstable GPR142 48 31 CCO[C@@H]1C[C@H](NCc2cccc(O)c2)C1(C)C ZINC000217872921 BF For-Sale Unstable SLC6A13 0 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccccc1F ZINC000217872940 FF For-Sale Unstable HCRTR1 54 39 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccccc1F ZINC000217872940 FF For-Sale Unstable HCRTR2 59 39 Cc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217872963 FJ In-Stock Unstable TAAR1 17 43 C[C@H](C(=O)O)c1ccc(CS[C@H]2CCC[C@@H](C)C2)cc1 ZINC000217872966 CJ For-Sale Unstable PTGS1 25 52 C[C@H](C(=O)O)c1ccc(CS[C@H]2CCC[C@@H](C)C2)cc1 ZINC000217872966 CJ For-Sale Unstable SLC22A20 0 44 Cc1c(NC(=O)c2cncs2)cccc1S(N)(=O)=O ZINC000217872973 CD For-Sale Unstable CA2 19 44 Cc1c(NC(=O)c2cncs2)cccc1S(N)(=O)=O ZINC000217872973 CD For-Sale Unstable CA4 22 44 Cc1c(NC(=O)c2cncs2)cccc1S(N)(=O)=O ZINC000217872973 CD For-Sale Unstable CYNT 21 44 Cc1cccc(CNC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217872987 EI For-Sale Unstable ANPEP 21 50 CCO[C@H]1C[C@H](NCc2cccc(O)c2)C1(C)C ZINC000217873007 BF For-Sale Unstable SLC6A13 0 40 COC(=O)CSCc1cc(/C=C\C(=O)O)ccc1OC ZINC000217873019 CE For-Sale Unstable TUBB1 47 38 COC(=O)CSCc1cc(/C=C\C(=O)O)ccc1OC ZINC000217873019 CE For-Sale Unstable AKR1C3 31 40 COC(=O)CSCc1cc(/C=C\C(=O)O)ccc1OC ZINC000217873019 CE For-Sale Unstable ABCG2 15 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccccc1F ZINC000217873035 FF For-Sale Unstable HCRTR1 54 39 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccccc1F ZINC000217873035 FF For-Sale Unstable HCRTR2 59 39 COc1cccc(CNC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217873074 FH For-Sale Unstable DRD4 40 31 COc1cccc(CNC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217873074 FH For-Sale Unstable ROCK2 39 42 COc1cccc(CNC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217873074 FH For-Sale Unstable PDS 41 36 COc1ccc2c(c1)[C@@H](NC(=O)c1ccc(Cl)c([N+](=O)[O-])c1)CC(C)(C)O2 ZINC000217873078 GI In-Stock Unstable TAAR1 22 50 COc1ccc2c(c1)[C@@H](NC(=O)c1ccc(Cl)c([N+](=O)[O-])c1)CC(C)(C)O2 ZINC000217873078 GI In-Stock Unstable APLNR 0 40 CC[C@@H]1C(=O)NC(=O)CN1C(=O)/C=C\c1ccc(Br)cc1 ZINC000217873108 FD For-Sale Unstable GPR183 0 40 COC(=O)CSCc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217873111 CE For-Sale Unstable PTGER4 25 44 COC(=O)CSCc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217873111 CE For-Sale Unstable PTGER3 18 44 COC(=O)CSCc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217873111 CE For-Sale Unstable LTB4R 38 43 COc1ccc2c(c1)[C@H](NC(=O)c1ccc(Cl)c([N+](=O)[O-])c1)CC(C)(C)O2 ZINC000217873152 GI In-Stock Unstable TAAR1 24 50 COc1ccc2c(c1)[C@H](NC(=O)c1ccc(Cl)c([N+](=O)[O-])c1)CC(C)(C)O2 ZINC000217873152 GI In-Stock Unstable APLNR 0 40 Cc1cc(-c2cccs2)nn1CCNC(=O)c1ccccc1 ZINC000217873178 DG In-Stock Unstable DRD4 41 32 CC[C@H]1C(=O)NC(=O)CN1C(=O)/C=C\c1ccc(Br)cc1 ZINC000217873188 FD For-Sale Unstable GPR183 0 40 CC[C@@H](c1ccccc1O)N1C[C@@H](C)Cc2ccccc21 ZINC000217873244 CJ For-Sale Unstable TPP2 44 32 CN1CCO[C@@H]([C@@H](N)Cc2ccccc2F)C1 ZINC000217873251 BD For-Sale Unstable DPP4 15 44 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217873269 GI In-Stock Unstable TAAR1 27 55 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217873269 GI In-Stock Unstable APLNR 0 40 Cc1cc(-c2cccs2)nn1CCNC(=O)[C@@H](C)Oc1ccccc1 ZINC000217873303 FH In-Stock Unstable FABP4 22 43 COc1ccc(Br)cc1CN[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217873320 FK For-Sale Unstable TACR1 28 40 COc1ccc(Br)cc1CN[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217873320 FK For-Sale Unstable TRPM8 15 40 COc1ccc(CSc2cnn(C)c2)cc1/C=C\C(=O)O ZINC000217873321 DF For-Sale Unstable LTB4R 31 41 CC[C@H](c1ccccc1O)N1C[C@@H](C)Cc2ccccc21 ZINC000217873322 CJ For-Sale Unstable TPP2 44 32 COc1cc([C@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc(OC)c1O ZINC000217873329 KH In-Stock Unstable PRKDC 20 42 COc1cc([C@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc(OC)c1O ZINC000217873329 KH In-Stock Unstable CYP1B1 55 39 COc1cc([C@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc(OC)c1O ZINC000217873329 KH In-Stock Unstable CYP1A1 42 39 COc1cc([C@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc(OC)c1O ZINC000217873329 KH In-Stock Unstable RORC 51 36 CN1CCO[C@H]([C@@H](N)Cc2ccccc2F)C1 ZINC000217873337 BD For-Sale Unstable DPP4 15 44 CCCCN1C[C@@H](O)C[C@@H]1CC ZINC000217873346 AD In-Stock Unstable GBA2 45 37 Cc1cc(-c2cccs2)nn1CCNC(=O)[C@H](C)Oc1ccccc1 ZINC000217873376 FH In-Stock Unstable FABP4 22 43 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217873379 GI In-Stock Unstable TAAR1 26 55 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217873379 GI In-Stock Unstable APLNR 0 40 COc1ccc(Br)cc1CN[C@H]1C[C@H](C)CC[C@@H]1C(C)C ZINC000217873390 FK For-Sale Unstable TACR1 28 40 COc1ccc(Br)cc1CN[C@H]1C[C@H](C)CC[C@@H]1C(C)C ZINC000217873390 FK For-Sale Unstable TRPM8 15 40 COc1ccc(C[C@H](N)C(=O)O)c(F)c1Cl ZINC000217873393 BD For-Sale Unstable CACNA2D1 33 40 COc1cc([C@@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc(OC)c1O ZINC000217873421 KH In-Stock Unstable PRKDC 20 42 COc1cc([C@@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc(OC)c1O ZINC000217873421 KH In-Stock Unstable CYP1B1 55 39 COc1cc([C@@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc(OC)c1O ZINC000217873421 KH In-Stock Unstable CYP1A1 42 39 COc1cc([C@@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc(OC)c1O ZINC000217873421 KH In-Stock Unstable RORC 51 36 CCCCN1C[C@H](O)C[C@@H]1CC ZINC000217873425 AD In-Stock Unstable GBA2 45 37 COc1ccc(C[C@@H](N)C(=O)O)c(F)c1Cl ZINC000217873445 BD For-Sale Unstable CACNA2D1 33 40 N#Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217873454 CG For-Sale Unstable MAOB 28 45 N#Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217873454 CG For-Sale Unstable PTGER2 39 50 N#Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217873454 CG For-Sale Unstable EDNRA 0 43 N#Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217873454 CG For-Sale Unstable PTGER4 27 50 N#Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217873454 CG For-Sale Unstable PTGER3 24 50 N#Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217873454 CG For-Sale Unstable FFAR1 36 52 N#Cc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217873454 CG For-Sale Unstable AKR1C3 32 42 CC[C@@H](NC(=O)c1ccc(Cl)c([N+](=O)[O-])c1)c1ccc(C)c(C)c1 ZINC000217873467 EJ In-Stock Unstable TAAR1 19 46 CC[C@@H](NC(=O)c1ccc(Cl)c([N+](=O)[O-])c1)c1ccc(C)c(C)c1 ZINC000217873467 EJ In-Stock Unstable UTS2 53 34 CC[C@H](NC(=O)c1ccc(Cl)c([N+](=O)[O-])c1)c1ccc(C)c(C)c1 ZINC000217873514 EJ In-Stock Unstable TAAR1 19 46 CC[C@H](NC(=O)c1ccc(Cl)c([N+](=O)[O-])c1)c1ccc(C)c(C)c1 ZINC000217873514 EJ In-Stock Unstable UTS2 53 34 CCC[C@@H](O)CNCCCOC ZINC000217873521 AC For-Sale Unstable SPPS 43 38 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)Nc1nc(-c3ccncc3)cs1)C(=O)OC2 ZINC000217873529 JK In-Stock Unstable IMPDH1 0 57 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)Nc1nc(-c3ccncc3)cs1)C(=O)OC2 ZINC000217873529 JK In-Stock Unstable ROCK1 21 41 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)Nc1nc(-c3ccncc3)cs1)C(=O)OC2 ZINC000217873529 JK In-Stock Unstable IMPDH2 0 57 CC[C@H](C(=O)NCCn1nc(-c2cccs2)cc1C)c1ccccc1 ZINC000217873535 FI In-Stock Unstable KCNQ2 41 38 N#Cc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217873549 CG For-Sale Unstable MAOB 55 45 N#Cc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217873549 CG For-Sale Unstable PTGER2 36 50 N#Cc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217873549 CG For-Sale Unstable EDNRA 0 45 N#Cc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217873549 CG For-Sale Unstable PTGER4 25 50 N#Cc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217873549 CG For-Sale Unstable PTGER3 23 50 N#Cc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217873549 CG For-Sale Unstable FFAR1 42 55 N#Cc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217873549 CG For-Sale Unstable AKR1C3 33 45 CCC[C@H](O)CNCCCOC ZINC000217873602 AC For-Sale Unstable SPPS 43 38 CC[C@@H](C(=O)NCCn1nc(-c2cccs2)cc1C)c1ccccc1 ZINC000217873604 FI In-Stock Unstable KCNQ2 41 38 Cc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217873639 CH For-Sale Unstable OPRL1 0 41 Cc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217873639 CH For-Sale Unstable PTGER2 30 54 Cc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217873639 CH For-Sale Unstable PTGER4 46 49 Cc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217873639 CH For-Sale Unstable PTGER3 33 56 Cc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217873639 CH For-Sale Unstable PTGDR 0 56 Cc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217873639 CH For-Sale Unstable FFAR1 34 49 Cc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217873639 CH For-Sale Unstable FFAR4 51 49 O=C(O)/C=C\c1cccc(COC[C@@H]2CCCCO2)c1 ZINC000217873729 CF For-Sale Unstable PTGER2 0 40 CCN1CCC(Nc2nc(Cl)c(C(=O)OC)s2)CC1 ZINC000217873744 DE On-Demand Unstable HTR4 19 40 COc1ccccc1CCNC(=O)N/C=C/c1ccccc1Br ZINC000217873748 GH For-Sale Unstable MTNR1A 31 42 COc1ccccc1CCNC(=O)N/C=C/c1ccccc1Br ZINC000217873748 GH For-Sale Unstable MTNR1B 22 42 CC[C@@H](NC(=O)c1ccc(Cl)c([N+](=O)[O-])c1)c1ccc(OC)c(OC)c1 ZINC000217873801 GI In-Stock Unstable TAAR1 24 52 CC[C@@H](NC(=O)c1ccc(Cl)c([N+](=O)[O-])c1)c1ccc(OC)c(OC)c1 ZINC000217873801 GI In-Stock Unstable UTS2 56 35 CC[C@@H](NC(=O)c1ccc(Cl)c([N+](=O)[O-])c1)c1ccc(OC)c(OC)c1 ZINC000217873801 GI In-Stock Unstable APLNR 0 41 O=C(O)/C=C\c1cccc(COC[C@H]2CCCCO2)c1 ZINC000217873803 CF For-Sale Unstable PTGER2 0 40 C[C@@H]1CCC[C@@H](NCCN(C)[C@H](C)c2ccc(Cl)cc2)C1 ZINC000217873826 DJ For-Sale Unstable UTS2 42 33 CC[C@H](NC(=O)c1ccc(Cl)c([N+](=O)[O-])c1)c1ccc(OC)c(OC)c1 ZINC000217873870 GI In-Stock Unstable TAAR1 24 52 CC[C@H](NC(=O)c1ccc(Cl)c([N+](=O)[O-])c1)c1ccc(OC)c(OC)c1 ZINC000217873870 GI In-Stock Unstable UTS2 56 35 CC[C@H](NC(=O)c1ccc(Cl)c([N+](=O)[O-])c1)c1ccc(OC)c(OC)c1 ZINC000217873870 GI In-Stock Unstable APLNR 0 41 CC[C@@H](c1ccc(O)cc1)N1C[C@@H](C)Cc2ccccc21 ZINC000217873907 CJ For-Sale Unstable TPP2 43 32 CC[C@H](c1ccc(O)cc1)N1C[C@@H](C)Cc2ccccc21 ZINC000217873986 CJ For-Sale Unstable TPP2 43 32 CC(F)(F)COc1ccc(N2CCNCC2)cc1 ZINC000217874000 CE For-Sale Unstable ACVR1 51 39 CC[C@@H](NC(=O)c1ccc(Cl)c([N+](=O)[O-])c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217874001 GH In-Stock Unstable COLA 50 34 CC[C@@H](NC(=O)c1ccc(Cl)c([N+](=O)[O-])c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217874001 GH In-Stock Unstable CA4 15 41 CC[C@@H](NC(=O)c1ccc(Cl)c([N+](=O)[O-])c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217874001 GH In-Stock Unstable UTS2 47 34 COc1cccc(N2C[C@H](C(=O)NCCn3nc(-c4cccs4)cc3C)CC2=O)c1 ZINC000217874025 HG In-Stock Unstable DRD4 43 33 C[C@H]1Cc2ccccc2N([C@H](C)c2cc(Cl)ccc2O)C1 ZINC000217874069 DJ For-Sale Unstable DRD4 16 40 CC[C@H](NC(=O)c1ccc(Cl)c([N+](=O)[O-])c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217874077 GH In-Stock Unstable COLA 50 34 CC[C@H](NC(=O)c1ccc(Cl)c([N+](=O)[O-])c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217874077 GH In-Stock Unstable CA4 15 41 CC[C@H](NC(=O)c1ccc(Cl)c([N+](=O)[O-])c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217874077 GH In-Stock Unstable UTS2 47 34 COc1ccccc1[C@@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc3c21 ZINC000217874104 II In-Stock Unstable AKR1B1 23 48 COc1ccccc1[C@@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc3c21 ZINC000217874104 II In-Stock Unstable CYP1B1 74 39 COc1ccccc1[C@@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc3c21 ZINC000217874104 II In-Stock Unstable CYP1A1 59 42 COc1ccccc1[C@@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc3c21 ZINC000217874104 II In-Stock Unstable CYP1A2 47 47 O=C(N/C=C/c1ccccc1Br)NCCc1ccccc1Br ZINC000217874108 HJ For-Sale Unstable CA9 15 40 COc1cccc(N2C[C@@H](C(=O)NCCn3nc(-c4cccs4)cc3C)CC2=O)c1 ZINC000217874113 HG In-Stock Unstable DRD4 43 33 COc1ccccc1[C@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc3c21 ZINC000217874148 II In-Stock Unstable AKR1B1 23 48 COc1ccccc1[C@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc3c21 ZINC000217874148 II In-Stock Unstable CYP1B1 74 39 COc1ccccc1[C@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc3c21 ZINC000217874148 II In-Stock Unstable CYP1A1 59 42 COc1ccccc1[C@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc3c21 ZINC000217874148 II In-Stock Unstable CYP1A2 47 47 CN1CCO[C@@H]([C@@H](N)Cc2cc(Br)ccc2F)C1 ZINC000217874178 DD For-Sale Unstable DPP4 18 42 Cc1cc(-c2cccs2)nn1CCNC(=O)c1ccc(F)cc1Cl ZINC000217874197 FI In-Stock Unstable P2RX7 50 39 Cc1cc(-c2cccs2)nn1CCNC(=O)c1ccc(F)cc1Cl ZINC000217874197 FI In-Stock Unstable PYGL 0 40 COc1cccc(-c2noc(CNC(=O)c3ccc(Cl)c([N+](=O)[O-])c3)n2)c1 ZINC000217874202 GG In-Stock Unstable DRD4 44 35 COc1cccc(-c2noc(CNC(=O)c3ccc(Cl)c([N+](=O)[O-])c3)n2)c1 ZINC000217874202 GG In-Stock Unstable TAAR1 31 57 COc1cccc(-c2noc(CNC(=O)c3ccc(Cl)c([N+](=O)[O-])c3)n2)c1 ZINC000217874202 GG In-Stock Unstable APLNR 0 40 CCN(C)C(=O)CNC(=O)c1cc(OC)ccc1N ZINC000217874205 CC For-Sale Unstable MTNR1A 49 36 CCN(C)C(=O)CNC(=O)c1cc(OC)ccc1N ZINC000217874205 CC For-Sale Unstable MTNR1B 41 36 CN1CCO[C@H]([C@@H](N)Cc2cc(Br)ccc2F)C1 ZINC000217874244 DD For-Sale Unstable DPP4 18 42 COc1cccc(CCNC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217874261 GH For-Sale Unstable DRD4 41 32 COc1cccc(CCNC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217874261 GH For-Sale Unstable MTNR1A 84 51 COc1cccc(CCNC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217874261 GH For-Sale Unstable MTNR1B 78 51 COc1cccc(CCNC(=O)N/C=C/c2ccccc2Br)c1 ZINC000217874261 GH For-Sale Unstable CRTM 47 38 O=C(O)/C=C\c1ccccc1COCC(F)(F)C(F)F ZINC000217874264 CG For-Sale Unstable PTGER2 15 44 O=C(O)/C=C\c1ccccc1COCC(F)(F)C(F)F ZINC000217874264 CG For-Sale Unstable PTGER3 18 49 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc(OCc3ccccn3)c2)CC(=O)O4)cc1O ZINC000217874268 KK In-Stock Unstable AKR1B1 0 40 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc(OCc3ccccn3)c2)CC(=O)O4)cc1O ZINC000217874268 KK In-Stock Unstable CYP1A1 32 42 COc1ccc(-c2noc(CNC(=O)c3ccc(Cl)c([N+](=O)[O-])c3)n2)c(OC)c1 ZINC000217874301 HG In-Stock Unstable TAAR1 25 51 COc1ccc(-c2noc(CNC(=O)c3ccc(Cl)c([N+](=O)[O-])c3)n2)c(OC)c1 ZINC000217874301 HG In-Stock Unstable APLNR 0 43 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc(OCc3ccccn3)c2)CC(=O)O4)cc1O ZINC000217874317 KK In-Stock Unstable AKR1B1 0 40 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc(OCc3ccccn3)c2)CC(=O)O4)cc1O ZINC000217874317 KK In-Stock Unstable CYP1A1 32 42 O=C(NCc1nc(-c2ccccc2Cl)no1)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217874411 GH In-Stock Unstable TAAR1 16 42 CCCCCCOCc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217874449 CH For-Sale Unstable PTGER2 36 45 CCCCCCOCc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217874449 CH For-Sale Unstable INHA 66 34 CCCCCCOCc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217874449 CH For-Sale Unstable PTGER4 22 45 CCCCCCOCc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217874449 CH For-Sale Unstable PTGER3 17 45 CCCCCCOCc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217874449 CH For-Sale Unstable LTB4R 42 43 CCCCCCOCc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217874449 CH For-Sale Unstable PLA2G4B 81 41 CCCCCCOCc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217874449 CH For-Sale Unstable S1PR2 41 32 CCCCCCOCc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217874449 CH For-Sale Unstable AKR1B10 31 42 COc1ccccc1CCNCC(=O)NC1CC1 ZINC000217874462 BD For-Sale Unstable NPY2R 0 40 COc1ccccc1CCNCC(=O)NC1CC1 ZINC000217874462 BD For-Sale Unstable KCNA3 28 43 COc1ccccc1CCNCC(=O)NC1CC1 ZINC000217874462 BD For-Sale Unstable GPM3 0 43 COc1ccccc1CCNCC(=O)NC1CC1 ZINC000217874462 BD For-Sale Unstable MBTPS1 46 37 C[C@H]1CCCC[C@H]1NCCN(C)[C@H](C)c1ccccc1Cl ZINC000217874468 DJ For-Sale Unstable PDE7A 0 48 CCCCCCOCc1ccc(/C=C\C(=O)O)cc1F ZINC000217874515 CI For-Sale Unstable PLA2G4B 69 34 CCCCCCOCc1ccc(/C=C\C(=O)O)cc1F ZINC000217874515 CI For-Sale Unstable AKR1C3 29 41 C=C(C)COc1ccccc1[C@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccc(OC)c(O)c4)oc3c21 ZINC000217874543 KK In-Stock Unstable AKR1B1 0 42 C=C(C)COc1ccccc1[C@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccc(OC)c(O)c4)oc3c21 ZINC000217874543 KK In-Stock Unstable CYP1B1 48 36 C=C(C)COc1ccccc1[C@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccc(OC)c(O)c4)oc3c21 ZINC000217874543 KK In-Stock Unstable CYP1A1 39 42 Cc1noc(C)c1CC(=O)NCCn1nc(-c2cccs2)cc1C ZINC000217874545 EF In-Stock Unstable P2RX7 31 47 Clc1cncc(NCCCC2CCCC2)n1 ZINC000217874557 BH On-Demand Unstable P2RX7 15 44 COc1ccccc1CCNCC(=O)Nc1ccccc1 ZINC000217874589 CE For-Sale Unstable ADRB1 20 46 COc1ccccc1CCNCC(=O)Nc1ccccc1 ZINC000217874589 CE For-Sale Unstable TSHR 67 33 COc1ccccc1CCNCC(=O)Nc1ccccc1 ZINC000217874589 CE For-Sale Unstable ADRB3 26 46 COc1ccccc1CCNCC(=O)Nc1ccccc1 ZINC000217874589 CE For-Sale Unstable LPL 44 33 COc1ccccc1CCNCC(=O)Nc1ccccc1 ZINC000217874589 CE For-Sale Unstable LTA4H 21 40 COc1ccccc1CCNCC(=O)Nc1ccccc1 ZINC000217874589 CE For-Sale Unstable CPT1A 43 30 COc1ccccc1CCNCC(=O)Nc1ccccc1 ZINC000217874589 CE For-Sale Unstable MTNR1B 29 43 COc1ccccc1CCNCC(=O)Nc1ccccc1 ZINC000217874589 CE For-Sale Unstable ACR 18 41 COc1ccccc1CCNCC(=O)Nc1ccccc1 ZINC000217874589 CE For-Sale Unstable ENPP1 45 32 COc1ccccc1CCNCC(=O)Nc1ccccc1 ZINC000217874589 CE For-Sale Unstable MBTPS1 49 33 COc1ccccc1CCNCC(=O)Nc1ccccc1 ZINC000217874589 CE For-Sale Unstable KCNK3 45 40 COc1ccccc1CCNCC(=O)Nc1ccccc1 ZINC000217874589 CE For-Sale Unstable KCNK9 34 40 C=C(C)COc1ccccc1[C@@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccc(OC)c(O)c4)oc3c21 ZINC000217874604 KK In-Stock Unstable AKR1B1 0 42 C=C(C)COc1ccccc1[C@@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccc(OC)c(O)c4)oc3c21 ZINC000217874604 KK In-Stock Unstable CYP1B1 48 36 C=C(C)COc1ccccc1[C@@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccc(OC)c(O)c4)oc3c21 ZINC000217874604 KK In-Stock Unstable CYP1A1 39 42 O=C(O)/C=C\c1ccccc1COc1ccc(F)c(F)c1 ZINC000217874616 CH For-Sale Unstable PTGER2 22 45 O=C(O)/C=C\c1ccccc1COc1ccc(F)c(F)c1 ZINC000217874616 CH For-Sale Unstable PTGER4 31 50 O=C(O)/C=C\c1ccccc1COc1ccc(F)c(F)c1 ZINC000217874616 CH For-Sale Unstable PTGER3 36 60 O=C(O)/C=C\c1ccccc1COc1ccc(F)c(F)c1 ZINC000217874616 CH For-Sale Unstable CDC25B 27 48 O=C(O)/C=C\c1ccccc1COc1ccc(F)c(F)c1 ZINC000217874616 CH For-Sale Unstable GYS1 50 33 O=C(O)/C=C\c1ccccc1COc1ccc(F)c(F)c1 ZINC000217874616 CH For-Sale Unstable PTGDR 0 60 O=C(O)/C=C\c1ccccc1COc1ccc(F)c(F)c1 ZINC000217874616 CH For-Sale Unstable AKR1C3 26 42 O=C(O)/C=C\c1ccccc1COc1ccc(F)c(F)c1 ZINC000217874616 CH For-Sale Unstable FFAR4 43 36 COc1cccc(-c2noc(CN(C)C(=O)c3ccc(Cl)c([N+](=O)[O-])c3)n2)c1 ZINC000217874647 HH In-Stock Unstable HSD17B2 22 45 COc1cccc(-c2noc(CN(C)C(=O)c3ccc(Cl)c([N+](=O)[O-])c3)n2)c1 ZINC000217874647 HH In-Stock Unstable TAAR1 23 49 COc1cccc(-c2noc(CN(C)C(=O)c3ccc(Cl)c([N+](=O)[O-])c3)n2)c1 ZINC000217874647 HH In-Stock Unstable APLNR 0 40 CC(=O)Nc1cccc([C@@H](C)Nc2cncc(Cl)n2)c1 ZINC000217874699 CG For-Sale Unstable CSF1R 19 78 CC(=O)Nc1cccc([C@@H](C)Nc2cncc(Cl)n2)c1 ZINC000217874699 CG For-Sale Unstable IMDH_CRYPV 26 40 O=C(O)/C=C\c1ccc(COc2ccc(F)c(F)c2)cc1 ZINC000217874700 CH For-Sale Unstable MAOB 39 40 O=C(O)/C=C\c1ccc(COc2ccc(F)c(F)c2)cc1 ZINC000217874700 CH For-Sale Unstable PTGER2 33 45 O=C(O)/C=C\c1ccc(COc2ccc(F)c(F)c2)cc1 ZINC000217874700 CH For-Sale Unstable PTGER4 23 45 O=C(O)/C=C\c1ccc(COc2ccc(F)c(F)c2)cc1 ZINC000217874700 CH For-Sale Unstable PTPN2 0 45 O=C(O)/C=C\c1ccc(COc2ccc(F)c(F)c2)cc1 ZINC000217874700 CH For-Sale Unstable PTGER3 16 52 O=C(O)/C=C\c1ccc(COc2ccc(F)c(F)c2)cc1 ZINC000217874700 CH For-Sale Unstable CDC25B 24 45 O=C(O)/C=C\c1ccc(COc2ccc(F)c(F)c2)cc1 ZINC000217874700 CH For-Sale Unstable GYS1 50 31 O=C(O)/C=C\c1ccc(COc2ccc(F)c(F)c2)cc1 ZINC000217874700 CH For-Sale Unstable PTGDR 0 52 O=C(O)/C=C\c1ccc(COc2ccc(F)c(F)c2)cc1 ZINC000217874700 CH For-Sale Unstable FFAR1 44 38 O=C(O)/C=C\c1ccc(COc2ccc(F)c(F)c2)cc1 ZINC000217874700 CH For-Sale Unstable AKR1C3 34 46 O=C(CCc1nnc(-c2ccccc2)o1)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217874708 FG In-Stock Unstable HCRTR1 19 42 COc1ccccc1CCNCC(=O)NC1CCCC1 ZINC000217874709 CD For-Sale Unstable HTR1A 28 52 COc1ccccc1CCNCC(=O)NC1CCCC1 ZINC000217874709 CD For-Sale Unstable DRD2 30 40 COc1ccccc1CCNCC(=O)NC1CCCC1 ZINC000217874709 CD For-Sale Unstable CNR1 19 42 COc1ccccc1CCNCC(=O)NC1CCCC1 ZINC000217874709 CD For-Sale Unstable SLC18A2 15 44 COc1ccccc1CCNCC(=O)NC1CCCC1 ZINC000217874709 CD For-Sale Unstable HTR4 22 40 COc1ccccc1CCNCC(=O)NC1CCCC1 ZINC000217874709 CD For-Sale Unstable CNR2 24 43 COc1ccccc1CCNCC(=O)NC1CCCC1 ZINC000217874709 CD For-Sale Unstable SIGMAR1 22 54 COc1ccccc1CCNCC(=O)NC1CCCC1 ZINC000217874709 CD For-Sale Unstable CCR3 15 44 COc1ccccc1CCNCC(=O)NC1CCCC1 ZINC000217874709 CD For-Sale Unstable KCNA3 31 41 COc1ccccc1CCNCC(=O)NC1CCCC1 ZINC000217874709 CD For-Sale Unstable EPHX2 24 42 COc1ccccc1CCNCC(=O)NC1CCCC1 ZINC000217874709 CD For-Sale Unstable CCR8 15 43 COc1ccccc1CCNCC(=O)NC1CCCC1 ZINC000217874709 CD For-Sale Unstable TYRO3 19 46 COc1ccccc1CCNCC(=O)NC1CCCC1 ZINC000217874709 CD For-Sale Unstable BIRC2 20 44 COc1ccccc1CCNCC(=O)NC1CCCC1 ZINC000217874709 CD For-Sale Unstable MBTPS1 57 38 COc1ccc(-c2noc(CN(C)C(=O)c3ccc(Cl)c([N+](=O)[O-])c3)n2)c(OC)c1 ZINC000217874777 IH In-Stock Unstable TAAR1 20 44 COc1ccc(-c2noc(CN(C)C(=O)c3ccc(Cl)c([N+](=O)[O-])c3)n2)c(OC)c1 ZINC000217874777 IH In-Stock Unstable APLNR 0 42 CC(=O)Nc1cccc([C@H](C)Nc2cncc(Cl)n2)c1 ZINC000217874780 CG For-Sale Unstable CSF1R 19 78 CC(=O)Nc1cccc([C@H](C)Nc2cncc(Cl)n2)c1 ZINC000217874780 CG For-Sale Unstable IMDH_CRYPV 26 40 Cc1cc(-c2cccs2)nn1CCNC(=O)c1ccccc1SC(F)F ZINC000217874781 GJ In-Stock Unstable GPR142 40 31 O=C(O)/C=C\c1cccc(COc2ccc(F)c(F)c2)c1 ZINC000217874791 CH For-Sale Unstable ALOX5 15 43 O=C(O)/C=C\c1cccc(COc2ccc(F)c(F)c2)c1 ZINC000217874791 CH For-Sale Unstable MAOB 71 47 O=C(O)/C=C\c1cccc(COc2ccc(F)c(F)c2)c1 ZINC000217874791 CH For-Sale Unstable PTGER2 40 49 O=C(O)/C=C\c1cccc(COc2ccc(F)c(F)c2)c1 ZINC000217874791 CH For-Sale Unstable PTGER4 28 49 O=C(O)/C=C\c1cccc(COc2ccc(F)c(F)c2)c1 ZINC000217874791 CH For-Sale Unstable PTGER3 22 50 O=C(O)/C=C\c1cccc(COc2ccc(F)c(F)c2)c1 ZINC000217874791 CH For-Sale Unstable LTB4R 18 42 O=C(O)/C=C\c1cccc(COc2ccc(F)c(F)c2)c1 ZINC000217874791 CH For-Sale Unstable CDC25B 23 43 O=C(O)/C=C\c1cccc(COc2ccc(F)c(F)c2)c1 ZINC000217874791 CH For-Sale Unstable NR1H4 41 35 O=C(O)/C=C\c1cccc(COc2ccc(F)c(F)c2)c1 ZINC000217874791 CH For-Sale Unstable GYS1 56 38 O=C(O)/C=C\c1cccc(COc2ccc(F)c(F)c2)c1 ZINC000217874791 CH For-Sale Unstable PTGDR 0 50 O=C(O)/C=C\c1cccc(COc2ccc(F)c(F)c2)c1 ZINC000217874791 CH For-Sale Unstable HCAR2 0 44 O=C(O)/C=C\c1cccc(COc2ccc(F)c(F)c2)c1 ZINC000217874791 CH For-Sale Unstable FFAR1 70 44 O=C(O)/C=C\c1cccc(COc2ccc(F)c(F)c2)c1 ZINC000217874791 CH For-Sale Unstable AKR1C3 36 49 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)N1CCOCC1)C(=O)OC2 ZINC000217874806 HF In-Stock Unstable IMPDH1 0 67 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)N1CCOCC1)C(=O)OC2 ZINC000217874806 HF In-Stock Unstable IMPDH2 0 67 COc1ccccc1CCNCC(=O)NC1CCCCC1 ZINC000217874811 CE For-Sale Unstable HTR1A 26 51 COc1ccccc1CCNCC(=O)NC1CCCCC1 ZINC000217874811 CE For-Sale Unstable DRD2 26 40 COc1ccccc1CCNCC(=O)NC1CCCCC1 ZINC000217874811 CE For-Sale Unstable CNR1 23 44 COc1ccccc1CCNCC(=O)NC1CCCCC1 ZINC000217874811 CE For-Sale Unstable CNR2 27 42 COc1ccccc1CCNCC(=O)NC1CCCCC1 ZINC000217874811 CE For-Sale Unstable SIGMAR1 23 53 COc1ccccc1CCNCC(=O)NC1CCCCC1 ZINC000217874811 CE For-Sale Unstable KCNA3 30 41 COc1ccccc1CCNCC(=O)NC1CCCCC1 ZINC000217874811 CE For-Sale Unstable FAAH 19 40 COc1ccccc1CCNCC(=O)NC1CCCCC1 ZINC000217874811 CE For-Sale Unstable EPHX2 27 44 COc1ccccc1CCNCC(=O)NC1CCCCC1 ZINC000217874811 CE For-Sale Unstable BIRC2 22 43 COc1ccccc1CCNCC(=O)NC1CCCCC1 ZINC000217874811 CE For-Sale Unstable MBTPS1 57 39 Cc1cc(C=O)cc(C(=O)O)c1N ZINC000217874813 AD For-Sale Unstable HAAO 40 33 CN(Cc1nc(-c2ccccc2Cl)no1)C(=O)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217874867 HI In-Stock Unstable GPBAR1 28 40 Cc1cc(-c2cccs2)nn1CCNC(=O)c1ccccc1S(=O)(=O)C(F)F ZINC000217874893 IG In-Stock Unstable GPR142 47 30 O=C(N/C=C/c1ccccc1Br)NCCc1ccc(Br)cc1 ZINC000217874910 HJ For-Sale Unstable LIG1 0 42 COc1ccccc1CCNCC(=O)NC(C)C ZINC000217874930 CD For-Sale Unstable GPM3 0 45 COc1ccccc1CCNCC(=O)NC(C)C ZINC000217874930 CD For-Sale Unstable MBTPS1 51 34 CCOc1ccccc1/C=C/C(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217874953 CE On-Demand Unstable HCN4 41 32 O=C(O)/C=C\c1ccc(OCCSc2cccs2)cc1 ZINC000217874962 DI For-Sale Unstable HCAR2 0 44 CC(C)c1ccc(CCCNC(=O)c2ccc(Cl)c([N+](=O)[O-])c2)cc1 ZINC000217874992 FJ In-Stock Unstable PTAFR 17 44 Cc1cc(-c2cccs2)nn1CCNC(=O)c1noc2c1CCCC2 ZINC000217875030 FG In-Stock Unstable PANC 48 32 COCCNC(=O)CNCCc1ccccc1OC ZINC000217875043 CC For-Sale Unstable HTR1A 15 40 COCCNC(=O)CNCCc1ccccc1OC ZINC000217875043 CC For-Sale Unstable DRD2 23 40 COCCNC(=O)CNCCc1ccccc1OC ZINC000217875043 CC For-Sale Unstable MTNR1A 50 38 COCCNC(=O)CNCCc1ccccc1OC ZINC000217875043 CC For-Sale Unstable MTNR1B 41 38 COCCNC(=O)CNCCc1ccccc1OC ZINC000217875043 CC For-Sale Unstable MBTPS1 52 35 COc1ccc(CSc2ccccc2)cc1/C=C\C(=O)O ZINC000217875070 DI For-Sale Unstable PTGER2 54 49 COc1ccc(CSc2ccccc2)cc1/C=C\C(=O)O ZINC000217875070 DI For-Sale Unstable PTGER4 29 49 COc1ccc(CSc2ccccc2)cc1/C=C\C(=O)O ZINC000217875070 DI For-Sale Unstable PTGER3 24 49 COc1ccc(CSc2ccccc2)cc1/C=C\C(=O)O ZINC000217875070 DI For-Sale Unstable LTB4R 44 52 COc1ccc(CSc2ccccc2)cc1/C=C\C(=O)O ZINC000217875070 DI For-Sale Unstable PTGDR 0 43 COc1ccc(CSc2ccccc2)cc1/C=C\C(=O)O ZINC000217875070 DI For-Sale Unstable AKR1B10 30 41 COc1ccc(CSc2ccccc2)cc1/C=C\C(=O)O ZINC000217875070 DI For-Sale Unstable CYSP_PLAFA 47 37 O=C(NCCCN1CCCc2ccccc21)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217875085 FH In-Stock Unstable DRD2 26 40 O=C(NCCCN1CCCc2ccccc21)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217875085 FH In-Stock Unstable HTR2C 18 43 O=C(NCCCN1CCCc2ccccc21)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217875085 FH In-Stock Unstable AVPR2 31 44 O=C(NCCCN1CCCc2ccccc21)c1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217875085 FH In-Stock Unstable DRD3 51 43 COCCCNC(=O)CNCCc1ccccc1OC ZINC000217875152 CC For-Sale Unstable HTR1A 21 41 COCCCNC(=O)CNCCc1ccccc1OC ZINC000217875152 CC For-Sale Unstable DRD2 27 43 COCCCNC(=O)CNCCc1ccccc1OC ZINC000217875152 CC For-Sale Unstable ADRA1D 20 40 COCCCNC(=O)CNCCc1ccccc1OC ZINC000217875152 CC For-Sale Unstable ADRA1A 16 40 COCCCNC(=O)CNCCc1ccccc1OC ZINC000217875152 CC For-Sale Unstable DRD3 37 41 COCCCNC(=O)CNCCc1ccccc1OC ZINC000217875152 CC For-Sale Unstable MTNR1A 56 37 COCCCNC(=O)CNCCc1ccccc1OC ZINC000217875152 CC For-Sale Unstable MTNR1B 49 39 COCCCNC(=O)CNCCc1ccccc1OC ZINC000217875152 CC For-Sale Unstable MBTPS1 54 36 O=C(O)/C=C\c1ccc(CSc2ccccc2F)c(F)c1 ZINC000217875161 DI For-Sale Unstable AKR1C3 31 46 COc1ccc(CNC(=O)c2cccc([N+](=O)[O-])c2C)c(OC)c1OC ZINC000217875234 FF In-Stock Unstable SLC9A1 22 43 CCC[C@@H](O)CNCC(=O)OC(C)(C)C ZINC000217875242 BD For-Sale Unstable CTSK 0 44 O=C(O)/C=C\c1cccc(CSc2ccccc2F)c1 ZINC000217875247 CI For-Sale Unstable PTGER2 28 42 O=C(O)/C=C\c1cccc(CSc2ccccc2F)c1 ZINC000217875247 CI For-Sale Unstable AKR1C3 33 47 O=C(O)/C=C\c1cccc(CSc2ccccc2F)c1 ZINC000217875247 CI For-Sale Unstable HD1B 0 43 COc1ccccc1CCNCC(=O)NCC(C)C ZINC000217875254 CD For-Sale Unstable ANPEP 17 44 COc1ccccc1CCNCC(=O)NCC(C)C ZINC000217875254 CD For-Sale Unstable MTNR1A 43 38 COc1ccccc1CCNCC(=O)NCC(C)C ZINC000217875254 CD For-Sale Unstable MBTPS1 51 35 C[C@H](C(=O)O)c1ccc(CN2C(=O)[C@@H](C)[C@@H](C)C2=O)cc1 ZINC000217875279 CE For-Sale Unstable PTGS1 33 53 C[C@H](C(=O)O)c1ccc(CN2C(=O)[C@@H](C)[C@@H](C)C2=O)cc1 ZINC000217875279 CE For-Sale Unstable PTGS2 27 53 O=C(O)/C=C\c1cc(F)ccc1CSc1ccccc1F ZINC000217875333 DI For-Sale Unstable PTGER2 32 44 O=C(O)/C=C\c1cc(F)ccc1CSc1ccccc1F ZINC000217875333 DI For-Sale Unstable PTGER4 0 40 O=C(O)/C=C\c1cc(F)ccc1CSc1ccccc1F ZINC000217875333 DI For-Sale Unstable PTGER3 17 42 O=C(O)/C=C\c1cc(F)ccc1CSc1ccccc1F ZINC000217875333 DI For-Sale Unstable PTGDR 0 42 CCC[C@H](O)CNCC(=O)OC(C)(C)C ZINC000217875334 BD For-Sale Unstable CTSK 0 44 CCOc1ccc(CNC(=O)c2cccc([N+](=O)[O-])c2C)cc1OCC ZINC000217875339 FH In-Stock Unstable CACNA1D 40 33 CCOc1ccc(CNC(=O)c2cccc([N+](=O)[O-])c2C)cc1OCC ZINC000217875339 FH In-Stock Unstable CCR3 0 40 C[C@H](C(=O)O)c1ccc(CN2C(=O)[C@H](C)[C@@H](C)C2=O)cc1 ZINC000217875359 CE For-Sale Unstable PTGS1 33 53 C[C@H](C(=O)O)c1ccc(CN2C(=O)[C@H](C)[C@@H](C)C2=O)cc1 ZINC000217875359 CE For-Sale Unstable PTGS2 27 53 Cc1cccc(N2CCN(CCC(=O)NCCc3ccncc3)CC2)c1 ZINC000217875373 FE In-Stock Unstable HTR1A 52 52 Cc1cccc(N2CCN(CCC(=O)NCCc3ccncc3)CC2)c1 ZINC000217875373 FE In-Stock Unstable DRD2 35 52 Cc1cccc(N2CCN(CCC(=O)NCCc3ccncc3)CC2)c1 ZINC000217875373 FE In-Stock Unstable DRD4 45 39 Cc1cccc(N2CCN(CCC(=O)NCCc3ccncc3)CC2)c1 ZINC000217875373 FE In-Stock Unstable HTR2A 52 52 Cc1cccc(N2CCN(CCC(=O)NCCc3ccncc3)CC2)c1 ZINC000217875373 FE In-Stock Unstable HTR2C 39 49 Cc1cccc(N2CCN(CCC(=O)NCCc3ccncc3)CC2)c1 ZINC000217875373 FE In-Stock Unstable DRD3 39 49 Cc1cccc(N2CCN(CCC(=O)NCCc3ccncc3)CC2)c1 ZINC000217875373 FE In-Stock Unstable HTR7 58 43 CC[C@@H](C)[C@H](N)C(=O)N1CC[C@@H](C)[C@@H]2CCCC[C@H]21 ZINC000217875391 CF For-Sale Unstable TPP2 41 46 CC[C@H](C)[C@H](N)C(=O)N1CC[C@@H](C)[C@@H]2CCCC[C@H]21 ZINC000217875460 CF For-Sale Unstable TPP2 41 46 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCc1ccccc1 ZINC000217875490 FF For-Sale Unstable AGTR2 41 33 O=C(N/C=C/c1ccccc1Br)Nc1ccc(Cl)cn1 ZINC000217875492 FI For-Sale Anodyne LUCI_LUCLA 32 42 CCC[C@@H](O)CNC[C@@H](O)COCC(C)C ZINC000217875494 BC On-Demand Unstable ADRB2 0 56 COc1ccccc1CCCNC(=O)c1cccc([N+](=O)[O-])c1C ZINC000217875499 EG In-Stock Unstable COLA 82 34 COc1ccccc1CCCNC(=O)c1cccc([N+](=O)[O-])c1C ZINC000217875499 EG In-Stock Unstable MTNR1B 38 40 COc1ccccc1CCCNC(=O)c1cccc([N+](=O)[O-])c1C ZINC000217875499 EG In-Stock Unstable KCNMA1 24 41 CCC[C@H](O)CNC[C@@H](O)COCC(C)C ZINC000217875557 BC On-Demand Unstable ADRB2 0 56 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCc1ccccc1 ZINC000217875567 FF For-Sale Unstable AGTR2 41 33 Cc1c(C(=O)Nc2ccccc2C(=O)c2ccccc2)cccc1[N+](=O)[O-] ZINC000217875593 FI In-Stock Unstable NR1H4 0 44 Cc1c(C(=O)Nc2ccccc2C(=O)c2ccccc2)cccc1[N+](=O)[O-] ZINC000217875593 FI In-Stock Unstable KCNMA1 32 49 Cc1c(C(=O)Nc2ccccc2C(=O)c2ccccc2)cccc1[N+](=O)[O-] ZINC000217875593 FI In-Stock Unstable AKR1C3 21 44 Cc1c(C(=O)Nc2ccccc2C(=O)c2ccccc2)cccc1[N+](=O)[O-] ZINC000217875593 FI In-Stock Unstable AKR1C2 33 40 Cc1c(C(=O)Nc2ccccc2C(=O)c2ccccc2)cccc1[N+](=O)[O-] ZINC000217875593 FI In-Stock Unstable KCNK3 43 36 Cc1c(C(=O)Nc2ccccc2C(=O)c2ccccc2)cccc1[N+](=O)[O-] ZINC000217875593 FI In-Stock Unstable KCNK9 40 34 CC[C@H](C)[C@H](N)C(=O)N1CC[C@H](C)[C@@H]2CCCC[C@H]21 ZINC000217875620 CF For-Sale Unstable TPP2 41 46 CCC[C@@H](O)CNC[C@H](O)COCC(C)C ZINC000217875633 BC On-Demand Unstable ADRB2 0 56 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCc1ccccc1 ZINC000217875640 FF For-Sale Unstable AGTR2 41 33 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCc1cccc(O)c1 ZINC000217875675 CH On-Demand Unstable SLC6A13 0 42 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCc1cccc(O)c1 ZINC000217875675 CH On-Demand Unstable TRPM8 18 47 CCC[C@H](O)CNC[C@H](O)COCC(C)C ZINC000217875695 BC On-Demand Unstable ADRB2 0 56 CCOc1ccc(CCCNC(=O)c2cccc([N+](=O)[O-])c2C)cc1 ZINC000217875708 EH In-Stock Unstable SCN2A 21 41 CCOc1ccc(CCCNC(=O)c2cccc([N+](=O)[O-])c2C)cc1 ZINC000217875708 EH In-Stock Unstable SLC6A5 18 41 CN(c1cc(Cl)ccc1CBr)C1CCC1 ZINC000217875709 CI For-Sale Unstable NOS2 19 40 CN(c1cc(Cl)ccc1CBr)C1CCC1 ZINC000217875709 CI For-Sale Unstable NOS3 18 40 COc1ccc2c(c1OC)C(=O)O[C@@H]2CC(=O)Nc1ccc2occc(=O)c2c1 ZINC000217875715 GG In-Stock Unstable ENPP1 40 32 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCc1ccccc1 ZINC000217875747 FF For-Sale Unstable AGTR2 41 33 COc1cccc(NC(=O)NCCn2nc(-c3cccs3)cc2C)c1 ZINC000217875761 FH In-Stock Unstable DRD4 42 33 COc1cccc(NC(=O)NCCn2nc(-c3cccs3)cc2C)c1 ZINC000217875761 FH In-Stock Unstable HRH2 19 42 COc1cccc(NC(=O)NCCn2nc(-c3cccs3)cc2C)c1 ZINC000217875761 FH In-Stock Unstable CCR3 24 43 COc1cccc(NC(=O)NCCn2nc(-c3cccs3)cc2C)c1 ZINC000217875761 FH In-Stock Unstable ROCK1 17 40 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCc1cccc(O)c1 ZINC000217875779 CH On-Demand Unstable SLC6A13 0 42 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCc1cccc(O)c1 ZINC000217875779 CH On-Demand Unstable TRPM8 18 47 COc1ccc2c(c1OC)C(=O)O[C@H]2CC(=O)Nc1ccc2occc(=O)c2c1 ZINC000217875790 GG In-Stock Unstable ENPP1 40 32 CCCOc1ccccc1CCCNC(=O)c1cccc([N+](=O)[O-])c1C ZINC000217875806 FI In-Stock Unstable COLA 52 30 CCCOc1ccccc1CCCNC(=O)c1cccc([N+](=O)[O-])c1C ZINC000217875806 FI In-Stock Unstable ACAT 0 41 O=C(N/C=C/c1ccccc1Br)NCCCc1ccccc1 ZINC000217875807 FI For-Sale Unstable HDAC8 15 42 O=C(N/C=C/c1ccccc1Br)NCCCc1ccccc1 ZINC000217875807 FI For-Sale Unstable MTNR1B 27 41 O=C(N/C=C/c1ccccc1Br)NCCCc1ccccc1 ZINC000217875807 FI For-Sale Unstable AMP1_PLAFQ 32 45 O=C(N/C=C/c1ccccc1Br)NCCCc1ccccc1 ZINC000217875807 FI For-Sale Unstable HDA106 0 41 CN(c1ccc(Cl)cc1CBr)C1CCC1 ZINC000217875820 CI For-Sale Unstable NOS2 20 43 CN(c1ccc(Cl)cc1CBr)C1CCC1 ZINC000217875820 CI For-Sale Unstable NOS3 20 43 COc1ccc(CNC(=O)NCCn2nc(-c3cccs3)cc2C)cc1 ZINC000217875864 FG In-Stock Unstable PROKR1 51 31 NC(=O)c1cccc(NCC(=O)NC2CC2)c1 ZINC000217875870 BC For-Sale Unstable CCR2 38 41 NC(=O)c1cccc(NCC(=O)NC2CC2)c1 ZINC000217875870 BC For-Sale Unstable FAAH2 0 43 NC(=O)c1cccc(NCC(=O)NC2CC2)c1 ZINC000217875870 BC For-Sale Unstable PARP14 0 40 NC(=O)c1cccc(NCC(=O)NC2CC2)c1 ZINC000217875870 BC For-Sale Unstable PARP15 0 42 NC(=O)c1cccc(NCC(=O)NC2CC2)c1 ZINC000217875870 BC For-Sale Unstable MVFR 0 43 NC(=O)c1cccc(NCC(=O)NC2CC2)c1 ZINC000217875870 BC For-Sale Unstable PARP10 0 48 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCc1cccc(O)c1 ZINC000217875889 CH For-Sale Unstable TRPM8 17 47 O=C(N/C=C/c1ccccc1Br)NCCCCc1ccccc1 ZINC000217875907 FJ For-Sale Unstable MTNR1B 23 40 O=C(N/C=C/c1ccccc1Br)NCCCCc1ccccc1 ZINC000217875907 FJ For-Sale Unstable FAAH 32 41 O=C(N/C=C/c1ccccc1Br)NCCCCc1ccccc1 ZINC000217875907 FJ For-Sale Unstable SCN5A 0 40 O=C(N/C=C/c1ccccc1Br)NCCCCc1ccccc1 ZINC000217875907 FJ For-Sale Unstable CES1 40 35 O=C(N/C=C/c1ccccc1Br)NCCCCc1ccccc1 ZINC000217875907 FJ For-Sale Unstable AMP1_PLAFQ 28 41 O=C(N/C=C/c1ccccc1Br)NCCCCc1ccccc1 ZINC000217875907 FJ For-Sale Unstable HDA106 0 40 CCN(C)C(=O)CNC(=O)c1cc(N)n[nH]1 ZINC000217875925 BB For-Sale Unstable PYGL 26 41 CCN(C)C(=O)CNC(=O)c1cc(N)n[nH]1 ZINC000217875925 BB For-Sale Unstable ALPL 54 32 CCCOc1ccc(CN2CCN(C)[C@@H](CC)C2)c(O)c1 ZINC000217875930 CF For-Sale Unstable CHRNA10 50 34 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCc1cccc(O)c1 ZINC000217875963 CH For-Sale Unstable TRPM8 17 47 CCNC(=O)NCCn1nc(-c2cccs2)cc1C ZINC000217875968 CE In-Stock Unstable GPR142 49 32 CCC[C@@H](O)CNCCCO ZINC000217876009 AC For-Sale Unstable SPPS 42 37 CC[C@@H](C)[C@H](N)C(=O)N1CCO[C@@H]2CCCC[C@H]21 ZINC000217876071 CD For-Sale Unstable TPP2 41 46 CCC[C@H](O)CNCCCO ZINC000217876099 AC For-Sale Unstable SPPS 42 37 O=C(O)/C=C\c1ccccc1CSc1ccc(F)c(F)c1 ZINC000217876141 DI For-Sale Unstable PTGER2 39 51 O=C(O)/C=C\c1ccccc1CSc1ccc(F)c(F)c1 ZINC000217876141 DI For-Sale Unstable PTGER4 0 47 O=C(O)/C=C\c1ccccc1CSc1ccc(F)c(F)c1 ZINC000217876141 DI For-Sale Unstable PTGER3 22 54 O=C(O)/C=C\c1ccccc1CSc1ccc(F)c(F)c1 ZINC000217876141 DI For-Sale Unstable PTGDR 0 54 CN1C(=O)N(C)C2(CCN(C(=O)c3cc4sccc4[nH]3)CC2)C1=O ZINC000217876172 ED In-Stock Unstable HRH4 30 63 CC[C@@H](C)[C@H](N)C(=O)N1CCO[C@H]2CCCC[C@H]21 ZINC000217876177 CD For-Sale Unstable TPP2 41 46 CC(C)CNC(=O)CNc1cccc(C(N)=O)c1 ZINC000217876203 BC For-Sale Unstable F3 71 35 CC(C)CNC(=O)CNc1cccc(C(N)=O)c1 ZINC000217876203 BC For-Sale Unstable PARP14 0 40 CC(C)CNC(=O)CNc1cccc(C(N)=O)c1 ZINC000217876203 BC For-Sale Unstable PARP15 0 40 CC(C)CNC(=O)CNc1cccc(C(N)=O)c1 ZINC000217876203 BC For-Sale Unstable MVFR 0 41 CC(C)CNC(=O)CNc1cccc(C(N)=O)c1 ZINC000217876203 BC For-Sale Unstable PARP10 0 48 C[C@H]1C[C@@H](C)CN(Cc2ccc([C@H](C)C(=O)O)cc2)C1 ZINC000217876213 CG For-Sale Unstable PTGS1 33 50 C[C@H]1C[C@@H](C)CN(Cc2ccc([C@H](C)C(=O)O)cc2)C1 ZINC000217876213 CG For-Sale Unstable PTGS2 22 50 C[C@H]1C[C@@H](C)CN(Cc2ccc([C@H](C)C(=O)O)cc2)C1 ZINC000217876213 CG For-Sale Unstable MLNR 23 42 C[C@H]1C[C@@H](C)CN(Cc2ccc([C@H](C)C(=O)O)cc2)C1 ZINC000217876213 CG For-Sale Unstable SLC22A20 0 50 Cn1cc(SCc2ccc(F)cc2/C=C\C(=O)O)cn1 ZINC000217876224 CF For-Sale Unstable PLA2G7 66 38 C[C@H](C(=O)O)c1ccc(CN2C[C@H](C)C[C@@H](C)C2)cc1 ZINC000217876291 CG For-Sale Unstable PTGS1 33 50 C[C@H](C(=O)O)c1ccc(CN2C[C@H](C)C[C@@H](C)C2)cc1 ZINC000217876291 CG For-Sale Unstable PTGS2 22 50 C[C@H](C(=O)O)c1ccc(CN2C[C@H](C)C[C@@H](C)C2)cc1 ZINC000217876291 CG For-Sale Unstable MLNR 23 42 C[C@H](C(=O)O)c1ccc(CN2C[C@H](C)C[C@@H](C)C2)cc1 ZINC000217876291 CG For-Sale Unstable SLC22A20 0 50 Cn1cc(SCc2ccc(F)c(/C=C\C(=O)O)c2)cn1 ZINC000217876326 CF For-Sale Unstable PLA2G7 63 37 O=C(N/C=C/c1ccccc1Br)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217876347 JG For-Sale Unstable TGM2 69 37 O=C(N/C=C/c1ccccc1Br)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217876347 JG For-Sale Unstable F13A1 85 40 O=C(N/C=C/c1ccccc1Br)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000217876347 JG For-Sale Unstable AKR1C3 37 40 COc1ccc(/C=C/C(=O)N[C@@H]2CCC[C@@H]2CO)cc1 ZINC000217876382 CD On-Demand Unstable HDAC1 24 45 COc1ccc(/C=C/C(=O)N[C@@H]2CCC[C@@H]2CO)cc1 ZINC000217876382 CD On-Demand Unstable GPR183 0 42 O=C(O)/C=C\c1cc(F)ccc1COc1cccc(Cl)c1 ZINC000217876403 DI For-Sale Unstable MAOB 29 42 O=C(O)/C=C\c1cc(F)ccc1COc1cccc(Cl)c1 ZINC000217876403 DI For-Sale Unstable PTGER2 45 46 O=C(O)/C=C\c1cc(F)ccc1COc1cccc(Cl)c1 ZINC000217876403 DI For-Sale Unstable PTGER1 26 41 O=C(O)/C=C\c1cc(F)ccc1COc1cccc(Cl)c1 ZINC000217876403 DI For-Sale Unstable PTGER4 27 46 O=C(O)/C=C\c1cc(F)ccc1COc1cccc(Cl)c1 ZINC000217876403 DI For-Sale Unstable PTGER3 28 46 O=C(O)/C=C\c1cc(F)ccc1COc1cccc(Cl)c1 ZINC000217876403 DI For-Sale Unstable CDC25B 22 40 O=C(O)/C=C\c1cc(F)ccc1COc1cccc(Cl)c1 ZINC000217876403 DI For-Sale Unstable PTGDR 0 42 C[C@@H](C(=O)O)c1ccc(CN2CCC[C@@H](C(N)=O)C2)cc1 ZINC000217876407 CD For-Sale Unstable PTGS1 22 50 C[C@@H](C(=O)O)c1ccc(CN2CCC[C@@H](C(N)=O)C2)cc1 ZINC000217876407 CD For-Sale Unstable SLC6A1 132 38 C[C@@H](C(=O)O)c1ccc(CN2CCC[C@@H](C(N)=O)C2)cc1 ZINC000217876407 CD For-Sale Unstable HRH3 19 42 C[C@@H](C(=O)O)c1ccc(CN2CCC[C@@H](C(N)=O)C2)cc1 ZINC000217876407 CD For-Sale Unstable MBTPS1 21 42 COc1cc2c(c(OC)c1OC)-c1ccc(NCCCCCC(=O)Nc3nc(-c4c[nH]c5ccccc45)cs3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217876437 KK In-Stock Unstable TUBA1A 15 53 Cc1ccc(S(=O)(=O)N2CCN(C(=O)N/C=C/c3ccccc3Br)CC2)cc1 ZINC000217876461 JG For-Sale Unstable TGM2 67 38 Cc1ccc(S(=O)(=O)N2CCN(C(=O)N/C=C/c3ccccc3Br)CC2)cc1 ZINC000217876461 JG For-Sale Unstable F13A1 84 38 Cc1ccc(S(=O)(=O)N2CCN(C(=O)N/C=C/c3ccccc3Br)CC2)cc1 ZINC000217876461 JG For-Sale Unstable GPR183 0 40 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](C(N)=O)C2)cc1 ZINC000217876484 CD For-Sale Unstable SLC6A1 132 38 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](C(N)=O)C2)cc1 ZINC000217876484 CD For-Sale Unstable HRH3 19 42 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](C(N)=O)C2)cc1 ZINC000217876484 CD For-Sale Unstable SLC22A20 0 43 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](C(N)=O)C2)cc1 ZINC000217876484 CD For-Sale Unstable MBTPS1 21 42 O=C(O)/C=C\c1cc(COc2cccc(Cl)c2)ccc1F ZINC000217876493 DI For-Sale Unstable MAOB 46 39 O=C(O)/C=C\c1cc(COc2cccc(Cl)c2)ccc1F ZINC000217876493 DI For-Sale Unstable PTGER2 51 52 O=C(O)/C=C\c1cc(COc2cccc(Cl)c2)ccc1F ZINC000217876493 DI For-Sale Unstable PTGER1 47 38 O=C(O)/C=C\c1cc(COc2cccc(Cl)c2)ccc1F ZINC000217876493 DI For-Sale Unstable PTGER4 30 52 O=C(O)/C=C\c1cc(COc2cccc(Cl)c2)ccc1F ZINC000217876493 DI For-Sale Unstable PTGER3 38 52 O=C(O)/C=C\c1cc(COc2cccc(Cl)c2)ccc1F ZINC000217876493 DI For-Sale Unstable CDC25B 23 42 O=C(O)/C=C\c1cc(COc2cccc(Cl)c2)ccc1F ZINC000217876493 DI For-Sale Unstable PTGDR 0 47 O=C(O)/C=C\c1cc(COc2cccc(Cl)c2)ccc1F ZINC000217876493 DI For-Sale Unstable FFAR1 50 40 O=C(O)/C=C\c1cc(COc2cccc(Cl)c2)ccc1F ZINC000217876493 DI For-Sale Unstable AKR1C3 30 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccccc1 ZINC000217876535 FE For-Sale Unstable COLA 136 42 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccccc1 ZINC000217876535 FE For-Sale Unstable CPT1A 121 42 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccccc1 ZINC000217876535 FE For-Sale Unstable CPT2 48 42 COc1cc(NC(=O)CC[C@@H]2NC(=O)c3ccccc3NC2=O)ccc1N1CCCCS1(=O)=O ZINC000217876550 JE In-Stock Unstable CASP2 19 40 COc1cc(NC(=O)CC[C@@H]2NC(=O)c3ccccc3NC2=O)ccc1N1CCCCS1(=O)=O ZINC000217876550 JE In-Stock Unstable CASP6 18 40 COc1ccccc1OCc1ccccc1/C=C\C(=O)O ZINC000217876576 CG For-Sale Unstable PTGER2 27 60 COc1ccccc1OCc1ccccc1/C=C\C(=O)O ZINC000217876576 CG For-Sale Unstable PTGER4 49 60 COc1ccccc1OCc1ccccc1/C=C\C(=O)O ZINC000217876576 CG For-Sale Unstable PTGER3 36 61 COc1ccccc1OCc1ccccc1/C=C\C(=O)O ZINC000217876576 CG For-Sale Unstable AKR1B10 37 44 COc1ccccc1OCc1ccccc1/C=C\C(=O)O ZINC000217876576 CG For-Sale Unstable CYSP_PLAFA 45 33 COC(=O)c1ccnc(NCCS(C)(=O)=O)c1 ZINC000217876579 CC On-Demand Unstable KDM3A 0 48 COC(=O)c1ccnc(NCCS(C)(=O)=O)c1 ZINC000217876579 CC On-Demand Unstable KDM5C 0 48 O=C(NCCN1CCC(O)CC1)c1ccc(Cl)cc1O ZINC000217876615 CD In-Stock Unstable CACNA1H 24 40 O=C(NCCN1CCC(O)CC1)c1ccc(Cl)cc1O ZINC000217876615 CD In-Stock Unstable DRD2 21 41 O=C(NCCN1CCC(O)CC1)c1ccc(Cl)cc1O ZINC000217876615 CD In-Stock Unstable DRD4 48 41 O=C(NCCN1CCC(O)CC1)c1ccc(Cl)cc1O ZINC000217876615 CD In-Stock Unstable HTR2A 19 40 O=C(NCCN1CCC(O)CC1)c1ccc(Cl)cc1O ZINC000217876615 CD In-Stock Unstable HTR2C 16 41 O=C(NCCN1CCC(O)CC1)c1ccc(Cl)cc1O ZINC000217876615 CD In-Stock Unstable PLD1 62 44 O=C(NCCN1CCC(O)CC1)c1ccc(Cl)cc1O ZINC000217876615 CD In-Stock Unstable PLD2 89 44 O=C(NCCN1CCC(O)CC1)c1ccc(Cl)cc1O ZINC000217876615 CD In-Stock Unstable CACNA1I 54 36 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccccc1 ZINC000217876622 FE For-Sale Unstable COLA 136 42 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccccc1 ZINC000217876622 FE For-Sale Unstable CPT1A 121 42 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccccc1 ZINC000217876622 FE For-Sale Unstable CPT2 48 42 COCCCN(C)S(=O)(=O)N1CCC[C@@H](C(=O)O)C1 ZINC000217876626 CB On-Demand Unstable SLC6A1 77 35 Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217876655 CH For-Sale Unstable MAOB 26 55 Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217876655 CH For-Sale Unstable PPARG 17 42 Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217876655 CH For-Sale Unstable PTGER2 23 44 Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217876655 CH For-Sale Unstable PTGER4 27 42 Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217876655 CH For-Sale Unstable PTGER3 22 46 Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217876655 CH For-Sale Unstable PTGDR 0 46 Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217876655 CH For-Sale Unstable ADAMTS4 43 36 Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217876655 CH For-Sale Unstable FFAR1 48 49 Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217876655 CH For-Sale Unstable AKR1C3 36 54 Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217876655 CH For-Sale Unstable FFAR4 47 42 Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217876655 CH For-Sale Unstable HPGD 22 50 CCOC(=O)/C=C/B(O)OC(C)(C)C(C)(C)O ZINC000217876667 BC For-Sale Unstable HCAR2 15 43 C[C@H](C(=O)O)c1ccc(CN2CCCC[C@@H]2C)cc1 ZINC000217876669 CG For-Sale Unstable PTGS1 28 51 C[C@H](C(=O)O)c1ccc(CN2CCCC[C@@H]2C)cc1 ZINC000217876669 CG For-Sale Unstable PTGS2 0 51 C[C@H](C(=O)O)c1ccc(CN2CCCC[C@@H]2C)cc1 ZINC000217876669 CG For-Sale Unstable HRH3 55 52 C[C@H](C(=O)O)c1ccc(CN2CCCC[C@@H]2C)cc1 ZINC000217876669 CG For-Sale Unstable SLC22A20 0 47 COC(=O)c1ccc(COc2ccc3occ(-c4ccc(OC)cc4)c3c2)o1 ZINC000217876678 GK In-Stock Unstable ALDH2 95 40 COC(=O)c1ccc(COc2ccc3occ(-c4ccc(OC)cc4)c3c2)o1 ZINC000217876678 GK In-Stock Unstable MTNR1A 33 40 COC(=O)c1ccc(COc2ccc3occ(-c4ccc(OC)cc4)c3c2)o1 ZINC000217876678 GK In-Stock Unstable MTNR1B 25 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccccc1 ZINC000217876705 FE For-Sale Unstable COLA 136 42 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccccc1 ZINC000217876705 FE For-Sale Unstable CPT1A 121 42 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccccc1 ZINC000217876705 FE For-Sale Unstable CPT2 48 42 O=C(N[C@@H]1CCC[C@@H]1CO)c1ccc(Cl)nc1 ZINC000217876713 CD For-Sale Unstable SSTR3 29 40 COc1ccc2c(c1)[C@@H](NC(=O)c1cccc([N+](=O)[O-])c1C)CC(C)(C)O2 ZINC000217876743 FH In-Stock Unstable CACNA1D 41 34 Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2F)cc1 ZINC000217876747 CH For-Sale Unstable PTGER4 15 40 Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2F)cc1 ZINC000217876747 CH For-Sale Unstable CDC25B 23 40 Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2F)cc1 ZINC000217876747 CH For-Sale Unstable GYS1 60 36 Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2F)cc1 ZINC000217876747 CH For-Sale Unstable FFAR1 30 40 Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2F)cc1 ZINC000217876747 CH For-Sale Unstable AKR1C3 33 47 Cc1ccc(OCc2ccc(/C=C\C(=O)O)cc2F)cc1 ZINC000217876747 CH For-Sale Unstable FFAR4 50 42 Cc1cc(-c2cccs2)nn1CCNS(=O)(=O)c1ccc(Cl)s1 ZINC000217876765 GH In-Stock Unstable CCR4 62 35 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccccc1 ZINC000217876777 FE For-Sale Unstable COLA 136 42 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccccc1 ZINC000217876777 FE For-Sale Unstable CPT1A 121 42 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccccc1 ZINC000217876777 FE For-Sale Unstable CPT2 48 42 O=C(N[C@H]1CCC[C@@H]1CO)c1ccc(Cl)nc1 ZINC000217876794 CD For-Sale Unstable SSTR3 29 40 COc1ccc2c(c1)[C@H](NC(=O)c1cccc([N+](=O)[O-])c1C)CC(C)(C)O2 ZINC000217876820 FH In-Stock Unstable CACNA1D 41 34 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217876837 CH For-Sale Unstable ALOX5 23 51 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217876837 CH For-Sale Unstable MAOB 76 49 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217876837 CH For-Sale Unstable PPARG 18 42 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217876837 CH For-Sale Unstable PTGER2 28 54 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217876837 CH For-Sale Unstable PTGER4 40 48 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217876837 CH For-Sale Unstable PTGER3 37 48 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217876837 CH For-Sale Unstable LTB4R 26 46 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217876837 CH For-Sale Unstable KCNA3 0 42 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217876837 CH For-Sale Unstable NR1H4 62 39 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217876837 CH For-Sale Unstable GYS1 56 36 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217876837 CH For-Sale Unstable PTGDR 0 46 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217876837 CH For-Sale Unstable ADAMTS4 43 39 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217876837 CH For-Sale Unstable HCAR2 0 40 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217876837 CH For-Sale Unstable FFAR1 94 54 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217876837 CH For-Sale Unstable AKR1C3 45 54 Cc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217876837 CH For-Sale Unstable FFAR4 47 43 COc1cccc(C(=O)N2CCC(C(=O)N(C)Cc3cnccn3)CC2)c1 ZINC000217876858 FD In-Stock Unstable DRD4 43 33 COc1cccc(C(=O)N2CCC(C(=O)N(C)Cc3cnccn3)CC2)c1 ZINC000217876858 FD In-Stock Unstable SLC18A3 23 43 COc1cccc(C(=O)N2CCC(C(=O)N(C)Cc3cnccn3)CC2)c1 ZINC000217876858 FD In-Stock Unstable PTR1 48 36 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccccc1OC ZINC000217876872 FF For-Sale Unstable HCRTR1 50 38 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccccc1OC ZINC000217876872 FF For-Sale Unstable HCRTR2 55 38 O=C(N[C@@H]1CCC[C@H]1CO)c1ccc(Cl)nc1 ZINC000217876888 CD For-Sale Unstable SSTR3 29 40 CCC[C@@H]1C[C@@H](O)CN1CCC(C)C ZINC000217876906 AE In-Stock Unstable P0504H10.9 49 31 CC(C)OCCOCCOc1cccc(/C=C\C(=O)O)c1 ZINC000217876909 CF For-Sale Unstable AKR1C3 39 40 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1cccc([N+](=O)[O-])c1C ZINC000217876923 FH In-Stock Unstable CACNA1D 44 35 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](C)C2)cc1 ZINC000217876924 CG For-Sale Unstable PTGS1 28 50 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](C)C2)cc1 ZINC000217876924 CG For-Sale Unstable SLC6A1 61 33 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](C)C2)cc1 ZINC000217876924 CG For-Sale Unstable PTGS2 0 50 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](C)C2)cc1 ZINC000217876924 CG For-Sale Unstable HRH3 22 43 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](C)C2)cc1 ZINC000217876924 CG For-Sale Unstable SIGMAR1 28 46 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](C)C2)cc1 ZINC000217876924 CG For-Sale Unstable MLNR 43 42 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](C)C2)cc1 ZINC000217876924 CG For-Sale Unstable BIRC2 40 35 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](C)C2)cc1 ZINC000217876924 CG For-Sale Unstable SLC22A20 0 45 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccccc1OC ZINC000217876956 FF For-Sale Unstable HCRTR1 50 38 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccccc1OC ZINC000217876956 FF For-Sale Unstable HCRTR2 55 38 O=C(N[C@H]1CCC[C@H]1CO)c1ccc(Cl)nc1 ZINC000217876970 CD On-Demand Unstable SSTR3 29 40 CC(C)(C)OC(=O)NCCNC(=O)N/C=C/c1ccccc1Br ZINC000217876995 GG For-Sale Unstable PAPA1_CARPA 32 41 CCC[C@H]1C[C@@H](O)CN1CCC(C)C ZINC000217876996 AE In-Stock Unstable P0504H10.9 49 31 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1cccc([N+](=O)[O-])c1C ZINC000217877015 FH In-Stock Unstable CACNA1D 44 35 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccccc1OC ZINC000217877045 FF For-Sale Unstable HCRTR1 50 38 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccccc1OC ZINC000217877045 FF For-Sale Unstable HCRTR2 55 38 C[C@H]1CN(Cc2ccc([C@H](C)C(=O)O)cc2)CCO1 ZINC000217877060 CE For-Sale Unstable DRD4 19 41 C[C@H]1CN(Cc2ccc([C@H](C)C(=O)O)cc2)CCO1 ZINC000217877060 CE For-Sale Unstable PTGS1 24 44 C[C@H]1CN(Cc2ccc([C@H](C)C(=O)O)cc2)CCO1 ZINC000217877060 CE For-Sale Unstable PTGS2 15 44 O=C(N[C@@H]1CCC[C@@H]1CO)c1c(Cl)cccc1Cl ZINC000217877078 CF For-Sale Unstable SSTR3 32 41 O=C(N[C@@H]1CCC[C@@H]1CO)c1c(Cl)cccc1Cl ZINC000217877078 CF For-Sale Unstable TYK2 40 37 CCC[C@@H]1C[C@H](O)CN1CCC(C)C ZINC000217877089 AE In-Stock Unstable P0504H10.9 49 31 COc1ccc([C@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2oc(C)cc(=O)c2O)cc1OC ZINC000217877110 JI In-Stock Unstable RORC 43 33 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccccc1OC ZINC000217877136 FF For-Sale Unstable HCRTR1 50 38 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccccc1OC ZINC000217877136 FF For-Sale Unstable HCRTR2 55 38 CC(C)(C)OC(=O)N1CCN(C(=O)N/C=C/c2ccccc2Br)CC1 ZINC000217877146 HH For-Sale Unstable GPR119 33 44 CC(C)(C)OC(=O)N1CCN(C(=O)N/C=C/c2ccccc2Br)CC1 ZINC000217877146 HH For-Sale Unstable Q6PRC7_IXORI 19 40 CCC[C@H]1C[C@H](O)CN1CCC(C)C ZINC000217877159 AE In-Stock Unstable P0504H10.9 49 31 O=C(N[C@H]1CCC[C@@H]1CO)c1c(Cl)cccc1Cl ZINC000217877181 CF For-Sale Unstable SSTR3 32 41 O=C(N[C@H]1CCC[C@@H]1CO)c1c(Cl)cccc1Cl ZINC000217877181 CF For-Sale Unstable TYK2 40 37 COc1ccc([C@@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2oc(C)cc(=O)c2O)cc1OC ZINC000217877186 JI In-Stock Unstable RORC 43 33 COc1cc(F)cc(C[C@H](N)C(=O)O)c1Cl ZINC000217877205 BD For-Sale Unstable CACNA2D1 38 41 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc(OC)c1 ZINC000217877219 FF For-Sale Unstable DRD4 44 34 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc(OC)c1 ZINC000217877219 FF For-Sale Unstable CFTR 46 41 O=C(N[C@@H]1CCC[C@H]1CO)c1c(Cl)cccc1Cl ZINC000217877248 CF For-Sale Unstable SSTR3 32 41 O=C(N[C@@H]1CCC[C@H]1CO)c1c(Cl)cccc1Cl ZINC000217877248 CF For-Sale Unstable TYK2 40 37 COc1cc(F)cc(C[C@@H](N)C(=O)O)c1Cl ZINC000217877268 BD For-Sale Unstable CACNA2D1 38 41 O=C(O)/C=C\c1cccc(COCC(F)(F)C(F)F)c1 ZINC000217877278 CG For-Sale Unstable AKR1C3 25 44 CC(C)(C)OC(=O)N1CCC(NC(=O)N/C=C/c2ccccc2Br)CC1 ZINC000217877284 HI For-Sale Unstable CCR8 19 42 CC(C)(C)OC(=O)N1CCC(NC(=O)N/C=C/c2ccccc2Br)CC1 ZINC000217877284 HI For-Sale Unstable GPR119 38 41 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc(OC)c1 ZINC000217877305 FF For-Sale Unstable DRD4 44 34 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc(OC)c1 ZINC000217877305 FF For-Sale Unstable CFTR 46 41 O=C(N[C@H]1CCC[C@H]1CO)c1c(Cl)cccc1Cl ZINC000217877319 CF For-Sale Unstable SSTR3 32 41 O=C(N[C@H]1CCC[C@H]1CO)c1c(Cl)cccc1Cl ZINC000217877319 CF For-Sale Unstable TYK2 40 37 CC[C@@H](NC(=O)c1cccc([N+](=O)[O-])c1C)c1ccc(C)cc1C ZINC000217877355 EI In-Stock Unstable CCR3 0 48 O=C(NCCn1nc(-c2ccsc2)cc1C1CC1)c1ccccc1C(F)(F)F ZINC000217877378 HJ In-Stock Unstable RBP4 40 32 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc(OC)c1 ZINC000217877383 FF For-Sale Unstable DRD4 44 34 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc(OC)c1 ZINC000217877383 FF For-Sale Unstable CFTR 46 41 C[C@H](C(=O)O)c1ccc(CN2[C@@H](C)CCC[C@@H]2C)cc1 ZINC000217877392 CH For-Sale Unstable PTGS1 37 58 C[C@H](C(=O)O)c1ccc(CN2[C@@H](C)CCC[C@@H]2C)cc1 ZINC000217877392 CH For-Sale Unstable PTGS2 24 58 COc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1OC ZINC000217877394 DH For-Sale Unstable KIT 18 40 COc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1OC ZINC000217877394 DH For-Sale Unstable KDR 21 42 COc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1OC ZINC000217877394 DH For-Sale Unstable CYP1A1 15 40 COc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1OC ZINC000217877394 DH For-Sale Unstable PDGFRA 32 42 COc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1OC ZINC000217877394 DH For-Sale Unstable ENPP1 70 33 COc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1OC ZINC000217877394 DH For-Sale Unstable KCNK3 69 42 COc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1OC ZINC000217877394 DH For-Sale Unstable KCNK9 61 40 O=C(N[C@@H]1CCC[C@@H]1CO)c1cc(F)c(F)cc1Cl ZINC000217877424 CF For-Sale Unstable SSTR3 32 46 CC[C@H](NC(=O)c1cccc([N+](=O)[O-])c1C)c1ccc(C)cc1C ZINC000217877429 EI In-Stock Unstable CCR3 0 48 CC(C)[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217877455 GD In-Stock Unstable EDNRA 31 40 CC(C)[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217877455 GD In-Stock Unstable TACR2 48 39 CC(C)[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217877455 GD In-Stock Unstable CCKAR 44 36 CC(C)[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217877455 GD In-Stock Unstable MMP14 47 35 CC(C)[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217877455 GD In-Stock Unstable GRPR 45 31 CC(C)[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217877455 GD In-Stock Unstable ECE1 40 37 CC(C)[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217877455 GD In-Stock Unstable CCKBR 41 36 CC(C)[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217877455 GD In-Stock Unstable GHSR 63 41 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc(OC)c1 ZINC000217877460 FF For-Sale Unstable DRD4 44 34 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc(OC)c1 ZINC000217877460 FF For-Sale Unstable CFTR 46 41 CCCCCCOCc1ccc(F)cc1/C=C\C(=O)O ZINC000217877462 CI For-Sale Unstable PLA2G4B 84 35 O=C(/C=C/c1ccccc1)NCCn1nc(-c2ccsc2)cc1C1CC1 ZINC000217877476 FI In-Stock Unstable HDAC8 42 32 O=C(N[C@H]1CCC[C@@H]1CO)c1cc(F)c(F)cc1Cl ZINC000217877509 CF For-Sale Unstable SSTR3 32 46 CCCCCCOCc1ccc(F)c(/C=C\C(=O)O)c1 ZINC000217877523 CI For-Sale Unstable PLA2G4B 76 41 CC[C@@H](NC(=O)c1cccc([N+](=O)[O-])c1C)c1ccc(OC)c(OC)c1 ZINC000217877543 FH In-Stock Unstable PTGER3 15 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccn(C)c1=O ZINC000217877545 FD In-Stock Unstable HCRTR2 44 35 C[C@@H]1CCC[C@H](OCc2ccccc2/C=C\C(=O)O)C1 ZINC000217877597 CH For-Sale Unstable PTGER2 44 42 C[C@@H]1CCC[C@H](OCc2ccccc2/C=C\C(=O)O)C1 ZINC000217877597 CH For-Sale Unstable PTGER4 0 42 C[C@@H]1CCC[C@H](OCc2ccccc2/C=C\C(=O)O)C1 ZINC000217877597 CH For-Sale Unstable PTGER3 16 44 C[C@@H]1CCC[C@H](OCc2ccccc2/C=C\C(=O)O)C1 ZINC000217877597 CH For-Sale Unstable PTGDR 0 44 O=C(N[C@@H]1CCC[C@H]1CO)c1cc(F)c(F)cc1Cl ZINC000217877600 CF For-Sale Unstable SSTR3 32 46 CC[C@H](NC(=O)c1cccc([N+](=O)[O-])c1C)c1ccc(OC)c(OC)c1 ZINC000217877620 FH In-Stock Unstable PTGER3 15 40 Cc1cccc(/C=C/NC(=O)Nc2ccc(Br)cc2)c1 ZINC000217877627 EJ For-Sale Unstable MMP1 15 46 Cc1cccc(/C=C/NC(=O)Nc2ccc(Br)cc2)c1 ZINC000217877627 EJ For-Sale Unstable IDO1 20 42 Cc1cccc(/C=C/NC(=O)Nc2ccc(Br)cc2)c1 ZINC000217877627 EJ For-Sale Unstable KCNK3 40 35 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccn(C)c1=O ZINC000217877637 FD In-Stock Unstable HCRTR2 44 35 O=C(N[C@H]1CCC[C@H]1CO)c1cc(F)c(F)cc1Cl ZINC000217877686 CF On-Demand Unstable SSTR3 20 46 C[C@H]1CCC[C@H](OCc2ccccc2/C=C\C(=O)O)C1 ZINC000217877690 CH For-Sale Unstable PTGER2 44 42 C[C@H]1CCC[C@H](OCc2ccccc2/C=C\C(=O)O)C1 ZINC000217877690 CH For-Sale Unstable PTGER4 0 42 C[C@H]1CCC[C@H](OCc2ccccc2/C=C\C(=O)O)C1 ZINC000217877690 CH For-Sale Unstable PTGER3 16 44 C[C@H]1CCC[C@H](OCc2ccccc2/C=C\C(=O)O)C1 ZINC000217877690 CH For-Sale Unstable PTGDR 0 44 CO[C@@H]1O[C@H](CO)[C@@H](O)[C@H]2O[C@@H]12 ZINC000217877709 AA For-Sale Unstable FIMH 47 41 CC[C@H]1C(=O)NC(=O)CN1C(=O)/C=C\c1ccc(C)cc1 ZINC000217877716 CD For-Sale Unstable GPR183 0 41 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccn(C)c1=O ZINC000217877729 FD In-Stock Unstable HCRTR2 44 35 Cc1cccc(/C=C/NC(=O)Nc2cccc(C(=O)O)c2)c1 ZINC000217877743 CG For-Sale Unstable CCKAR 23 48 Cc1cccc(/C=C/NC(=O)Nc2cccc(C(=O)O)c2)c1 ZINC000217877743 CG For-Sale Unstable AKR1C3 40 52 Cc1cccc(/C=C/NC(=O)Nc2cccc(C(=O)O)c2)c1 ZINC000217877743 CG For-Sale Unstable IMDH_CRYPV 48 32 Cc1cccc(/C=C/NC(=O)Nc2cccc(C(=O)O)c2)c1 ZINC000217877743 CG For-Sale Unstable PARP15 0 40 Cc1cccc(/C=C/NC(=O)Nc2cccc(C(=O)O)c2)c1 ZINC000217877743 CG For-Sale Unstable KCNK3 103 46 Cc1cccc(/C=C/NC(=O)Nc2cccc(C(=O)O)c2)c1 ZINC000217877743 CG For-Sale Unstable KCNK9 55 46 CC[C@@H](NC(=O)c1cccc([N+](=O)[O-])c1C)c1ccc(S(C)(=O)=O)cc1 ZINC000217877747 GG In-Stock Unstable COLA 94 35 COc1ccc(/C=C\C(=O)O)cc1CSc1cccs1 ZINC000217877769 DI For-Sale Unstable PTGER2 24 40 COc1ccc(/C=C\C(=O)O)cc1CSc1cccs1 ZINC000217877769 DI For-Sale Unstable PTGER4 17 40 COc1ccc(/C=C\C(=O)O)cc1CSc1cccs1 ZINC000217877769 DI For-Sale Unstable AKR1C3 23 43 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccn(C)c1=O ZINC000217877813 FD In-Stock Unstable HCRTR2 44 35 CC[C@H](NC(=O)c1cccc([N+](=O)[O-])c1C)c1ccc(S(C)(=O)=O)cc1 ZINC000217877821 GG In-Stock Unstable COLA 94 35 Oc1ccc2c(c1)CCC[C@@H]2N1CCC[C@@H]2CCC[C@@H]21 ZINC000217877832 CI For-Sale Unstable DRD5 16 45 Oc1ccc2c(c1)CCC[C@@H]2N1CCC[C@@H]2CCC[C@@H]21 ZINC000217877832 CI For-Sale Unstable HSD17B1 53 37 Cc1cccc(/C=C/NC(=O)Nc2ccccc2[N+](=O)[O-])c1 ZINC000217877842 CH For-Sale Unstable COLA 40 33 COc1ccc(CSc2cccs2)cc1/C=C\C(=O)O ZINC000217877850 DI For-Sale Unstable PTGER2 43 43 COc1ccc(CSc2cccs2)cc1/C=C\C(=O)O ZINC000217877850 DI For-Sale Unstable PTGER4 26 43 COc1ccc(CSc2cccs2)cc1/C=C\C(=O)O ZINC000217877850 DI For-Sale Unstable PTGER3 23 40 COc1ccc(CSc2cccs2)cc1/C=C\C(=O)O ZINC000217877850 DI For-Sale Unstable TNFRSF1A 33 43 c1ccc(CCN2CCN(c3ccc4ccccc4n3)CC2)cc1 ZINC000217877914 DH On-Demand Unstable HTR1A 53 58 c1ccc(CCN2CCN(c3ccc4ccccc4n3)CC2)cc1 ZINC000217877914 DH On-Demand Unstable DRD2 32 63 c1ccc(CCN2CCN(c3ccc4ccccc4n3)CC2)cc1 ZINC000217877914 DH On-Demand Unstable DRD4 42 58 c1ccc(CCN2CCN(c3ccc4ccccc4n3)CC2)cc1 ZINC000217877914 DH On-Demand Unstable HTR1D 49 42 c1ccc(CCN2CCN(c3ccc4ccccc4n3)CC2)cc1 ZINC000217877914 DH On-Demand Unstable HTR1B 41 42 c1ccc(CCN2CCN(c3ccc4ccccc4n3)CC2)cc1 ZINC000217877914 DH On-Demand Unstable HTR2A 29 54 c1ccc(CCN2CCN(c3ccc4ccccc4n3)CC2)cc1 ZINC000217877914 DH On-Demand Unstable SLC6A4 20 54 c1ccc(CCN2CCN(c3ccc4ccccc4n3)CC2)cc1 ZINC000217877914 DH On-Demand Unstable DRD3 24 46 c1ccc(CCN2CCN(c3ccc4ccccc4n3)CC2)cc1 ZINC000217877914 DH On-Demand Unstable HTR3A 55 63 c1ccc(CCN2CCN(c3ccc4ccccc4n3)CC2)cc1 ZINC000217877914 DH On-Demand Unstable SLC6A3 21 47 c1ccc(CCN2CCN(c3ccc4ccccc4n3)CC2)cc1 ZINC000217877914 DH On-Demand Unstable HTR7 34 48 c1ccc(CCN2CCN(c3ccc4ccccc4n3)CC2)cc1 ZINC000217877914 DH On-Demand Unstable SIGMAR1 41 53 c1ccc(CCN2CCN(c3ccc4ccccc4n3)CC2)cc1 ZINC000217877914 DH On-Demand Unstable SORD 36 56 COC(=O)c1ccnc(N[C@@H]2CCN(C)C2)c1 ZINC000217877926 BC For-Sale Unstable HRH4 23 43 COC(=O)c1ccnc(N[C@@H]2CCN(C)C2)c1 ZINC000217877926 BC For-Sale Unstable PRKD1 76 42 COC(=O)c1ccnc(N[C@@H]2CCN(C)C2)c1 ZINC000217877926 BC For-Sale Unstable PKD2 0 42 COC(=O)c1ccnc(N[C@@H]2CCN(C)C2)c1 ZINC000217877926 BC For-Sale Unstable KDM4C 0 48 COC(=O)c1ccnc(N[C@@H]2CCN(C)C2)c1 ZINC000217877926 BC For-Sale Unstable KDM3A 0 48 COC(=O)c1ccnc(N[C@@H]2CCN(C)C2)c1 ZINC000217877926 BC For-Sale Unstable KDM5C 0 48 O=C(O)/C=C\c1ccc(CSc2ccccc2)c(F)c1 ZINC000217877939 CI For-Sale Unstable AKR1C3 29 40 O=C(O)/C=C\c1ccc(CSc2ccccc2)c(F)c1 ZINC000217877939 CI For-Sale Unstable GPR183 0 40 Cc1cccc(/C=C/NC(=O)Nc2cccc(O)c2)c1 ZINC000217877962 CG For-Sale Unstable CCKAR 0 42 Cc1cccc(/C=C/NC(=O)Nc2cccc(O)c2)c1 ZINC000217877962 CG For-Sale Unstable MMP2 0 62 Cc1cccc(/C=C/NC(=O)Nc2cccc(O)c2)c1 ZINC000217877962 CG For-Sale Unstable MMP9 0 62 Cc1cccc(/C=C/NC(=O)Nc2cccc(O)c2)c1 ZINC000217877962 CG For-Sale Unstable MMP1 0 62 Cc1cccc(/C=C/NC(=O)Nc2cccc(O)c2)c1 ZINC000217877962 CG For-Sale Unstable KCNK3 62 41 Cc1cccc(/C=C/NC(=O)Nc2cccc(O)c2)c1 ZINC000217877962 CG For-Sale Unstable KCNK9 49 41 C[C@H](C(=O)O)c1ccc(CN2CCOC[C@@H]2C)cc1 ZINC000217877986 CE For-Sale Unstable PTGS1 25 46 C[C@H](C(=O)O)c1ccc(CN2CCOC[C@@H]2C)cc1 ZINC000217877986 CE For-Sale Unstable PTGS2 15 46 COC(=O)c1ccnc(N[C@H]2CCN(C)C2)c1 ZINC000217878005 BC For-Sale Unstable HRH4 23 43 COC(=O)c1ccnc(N[C@H]2CCN(C)C2)c1 ZINC000217878005 BC For-Sale Unstable PRKD1 76 42 COC(=O)c1ccnc(N[C@H]2CCN(C)C2)c1 ZINC000217878005 BC For-Sale Unstable PKD2 0 42 COC(=O)c1ccnc(N[C@H]2CCN(C)C2)c1 ZINC000217878005 BC For-Sale Unstable KDM4C 0 48 COC(=O)c1ccnc(N[C@H]2CCN(C)C2)c1 ZINC000217878005 BC For-Sale Unstable KDM3A 0 48 COC(=O)c1ccnc(N[C@H]2CCN(C)C2)c1 ZINC000217878005 BC For-Sale Unstable KDM5C 0 48 O=C(O)/C=C\c1cc(F)ccc1CSc1ccccc1 ZINC000217878040 CI For-Sale Unstable PTGER2 34 41 O=C(O)/C=C\c1cc(F)ccc1CSc1ccccc1 ZINC000217878040 CI For-Sale Unstable PTGER4 0 42 O=C(O)/C=C\c1cc(F)ccc1CSc1ccccc1 ZINC000217878040 CI For-Sale Unstable PTGER3 15 44 O=C(O)/C=C\c1cc(F)ccc1CSc1ccccc1 ZINC000217878040 CI For-Sale Unstable PTGDR 0 44 Cc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217878084 CI For-Sale Unstable KIT 30 40 Cc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217878084 CI For-Sale Unstable KDR 25 41 Cc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217878084 CI For-Sale Unstable MMP2 0 47 Cc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217878084 CI For-Sale Unstable MMP9 0 56 Cc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217878084 CI For-Sale Unstable FLT3 15 40 Cc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217878084 CI For-Sale Unstable MMP1 0 47 Cc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217878084 CI For-Sale Unstable TRPM8 0 42 Cc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217878084 CI For-Sale Unstable KCNK3 49 38 C[C@H]1CO[C@H](C)CN1Cc1ccc([C@@H](C)C(=O)O)cc1 ZINC000217878104 CE For-Sale Unstable PTGS1 24 46 C[C@H]1CO[C@H](C)CN1Cc1ccc([C@@H](C)C(=O)O)cc1 ZINC000217878104 CE For-Sale Unstable PTGS2 17 46 O=C(O)/C=C\c1cc(CSc2ccccc2F)ccc1F ZINC000217878112 DI For-Sale Unstable PTGER2 33 42 O=C(O)/C=C\c1cc(CSc2ccccc2F)ccc1F ZINC000217878112 DI For-Sale Unstable PTGER4 0 42 O=C(O)/C=C\c1cc(CSc2ccccc2F)ccc1F ZINC000217878112 DI For-Sale Unstable PTGER3 18 44 O=C(O)/C=C\c1cc(CSc2ccccc2F)ccc1F ZINC000217878112 DI For-Sale Unstable PTGDR 0 44 O=C(O)/C=C\c1cc(CSc2ccccc2F)ccc1F ZINC000217878112 DI For-Sale Unstable PTPRG 0 40 C[C@H]1Cc2ccccc2N(CCN[C@H](C)c2ccco2)C1 ZINC000217878147 CH For-Sale Unstable TPP2 42 29 O=C(N[C@@H]1CCC[C@@H]1CO)Oc1ccccc1 ZINC000217878160 BD For-Sale Unstable SSTR3 28 41 O=C(N[C@@H]1CCC[C@@H]1CO)Oc1ccccc1 ZINC000217878160 BD For-Sale Unstable FAAH 31 49 O=C(N[C@@H]1CCC[C@@H]1CO)Oc1ccccc1 ZINC000217878160 BD For-Sale Unstable FAAH2 0 41 NS(=O)(=O)c1ccc(C(=O)NCc2ccccc2-n2cncn2)cc1 ZINC000217878161 FC In-Stock Unstable CA2 66 50 NS(=O)(=O)c1ccc(C(=O)NCc2ccccc2-n2cncn2)cc1 ZINC000217878161 FC In-Stock Unstable CA1 44 50 NS(=O)(=O)c1ccc(C(=O)NCc2ccccc2-n2cncn2)cc1 ZINC000217878161 FC In-Stock Unstable CA5B 56 42 NS(=O)(=O)c1ccc(C(=O)NCc2ccccc2-n2cncn2)cc1 ZINC000217878161 FC In-Stock Unstable CA4 40 44 NS(=O)(=O)c1ccc(C(=O)NCc2ccccc2-n2cncn2)cc1 ZINC000217878161 FC In-Stock Unstable CA5A 59 42 NS(=O)(=O)c1ccc(C(=O)NCc2ccccc2-n2cncn2)cc1 ZINC000217878161 FC In-Stock Unstable CA14 36 46 NS(=O)(=O)c1ccc(C(=O)NCc2ccccc2-n2cncn2)cc1 ZINC000217878161 FC In-Stock Unstable CA12 31 43 NS(=O)(=O)c1ccc(C(=O)NCc2ccccc2-n2cncn2)cc1 ZINC000217878161 FC In-Stock Unstable CA9 38 42 NS(=O)(=O)c1ccc(C(=O)NCc2ccccc2-n2cncn2)cc1 ZINC000217878161 FC In-Stock Unstable TTK 15 43 NS(=O)(=O)c1ccc(C(=O)NCc2ccccc2-n2cncn2)cc1 ZINC000217878161 FC In-Stock Unstable CYNT 21 45 Cc1cccc(/C=C/NC(=O)NCCC(=O)O)c1 ZINC000217878169 BD For-Sale Unstable FBP1 15 41 O=C(NCCn1nc(-c2ccsc2)cc1C1CC1)c1ccc(F)cc1Cl ZINC000217878179 GJ In-Stock Unstable P2RX7 46 35 COc1cccc(SCc2ccccc2/C=C\C(=O)O)c1 ZINC000217878189 DI For-Sale Unstable PTGER2 63 53 COc1cccc(SCc2ccccc2/C=C\C(=O)O)c1 ZINC000217878189 DI For-Sale Unstable PTGER4 32 44 COc1cccc(SCc2ccccc2/C=C\C(=O)O)c1 ZINC000217878189 DI For-Sale Unstable PTGER3 29 53 COc1cccc(SCc2ccccc2/C=C\C(=O)O)c1 ZINC000217878189 DI For-Sale Unstable LTB4R 33 49 COc1cccc(SCc2ccccc2/C=C\C(=O)O)c1 ZINC000217878189 DI For-Sale Unstable MTNR1A 30 45 COc1cccc(SCc2ccccc2/C=C\C(=O)O)c1 ZINC000217878189 DI For-Sale Unstable MTNR1B 31 45 COc1cccc(SCc2ccccc2/C=C\C(=O)O)c1 ZINC000217878189 DI For-Sale Unstable PTGDR 0 47 COc1cccc(SCc2ccccc2/C=C\C(=O)O)c1 ZINC000217878189 DI For-Sale Unstable AKR1C3 23 40 C[C@H](C(=O)O)c1ccc(CN2C[C@@H](C)OC[C@@H]2C)cc1 ZINC000217878192 CE For-Sale Unstable PTGS1 24 46 C[C@H](C(=O)O)c1ccc(CN2C[C@@H](C)OC[C@@H]2C)cc1 ZINC000217878192 CE For-Sale Unstable PTGS2 17 46 O=C(CCCCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCCc1ccccc1 ZINC000217878211 JJ In-Stock Unstable TOP1 0 41 O=C(N[C@H]1CCC[C@@H]1CO)Oc1ccccc1 ZINC000217878226 BD For-Sale Unstable SSTR3 28 41 O=C(N[C@H]1CCC[C@@H]1CO)Oc1ccccc1 ZINC000217878226 BD For-Sale Unstable FAAH 31 49 O=C(N[C@H]1CCC[C@@H]1CO)Oc1ccccc1 ZINC000217878226 BD For-Sale Unstable FAAH2 0 41 CCCCC[C@@H](C)NCCN1C[C@@H](C)Cc2ccccc21 ZINC000217878258 CI For-Sale Unstable TPP2 45 35 Cc1cccc(/C=C/NC(=O)Nc2ccc(N)cc2)c1 ZINC000217878266 CG For-Sale Unstable KIT 34 40 Cc1cccc(/C=C/NC(=O)Nc2ccc(N)cc2)c1 ZINC000217878266 CG For-Sale Unstable KDR 25 40 Cc1cccc(/C=C/NC(=O)Nc2ccc(N)cc2)c1 ZINC000217878266 CG For-Sale Unstable FLT3 15 40 Cc1cccc(/C=C/NC(=O)Nc2ccc(N)cc2)c1 ZINC000217878266 CG For-Sale Unstable MMP1 0 43 Cc1cccc(/C=C/NC(=O)Nc2ccc(N)cc2)c1 ZINC000217878266 CG For-Sale Unstable KCNK3 40 35 COc1cccc(SCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217878270 DI For-Sale Unstable PTGER2 36 45 COc1cccc(SCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217878270 DI For-Sale Unstable PTGER4 0 45 COc1cccc(SCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217878270 DI For-Sale Unstable CYP1B1 32 42 COc1cccc(SCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217878270 DI For-Sale Unstable PTGER3 17 45 COc1cccc(SCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217878270 DI For-Sale Unstable LTB4R 40 55 COc1cccc(SCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217878270 DI For-Sale Unstable MTNR1A 22 46 COc1cccc(SCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217878270 DI For-Sale Unstable MTNR1B 28 46 COc1cccc(SCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217878270 DI For-Sale Unstable AKR1C3 40 48 COc1cccc(SCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217878270 DI For-Sale Unstable ABCG2 15 41 COc1cccc(SCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217878270 DI For-Sale Unstable GPR183 0 40 O=C(N[C@@H]1CCC[C@H]1CO)Oc1ccccc1 ZINC000217878296 BD For-Sale Unstable SSTR3 28 41 O=C(N[C@@H]1CCC[C@H]1CO)Oc1ccccc1 ZINC000217878296 BD For-Sale Unstable FAAH 31 49 O=C(N[C@@H]1CCC[C@H]1CO)Oc1ccccc1 ZINC000217878296 BD For-Sale Unstable FAAH2 0 41 O=C(CCCCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCCc1ccccc1 ZINC000217878297 JJ In-Stock Unstable TOP1 0 41 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cn(C)nc1OC ZINC000217878313 GD For-Sale Unstable HCRTR2 40 34 CCCCC[C@H](C)NCCN1C[C@@H](C)Cc2ccccc21 ZINC000217878339 CI For-Sale Unstable TPP2 45 35 CC(C)C[C@@H]1C[C@H](NC(=O)OC(C)(C)C)CCN1 ZINC000217878350 CF For-Sale Unstable CTSK 16 40 O=C(N[C@H]1CCC[C@H]1CO)Oc1ccccc1 ZINC000217878382 BD For-Sale Unstable SSTR3 28 41 O=C(N[C@H]1CCC[C@H]1CO)Oc1ccccc1 ZINC000217878382 BD For-Sale Unstable FAAH 31 49 O=C(N[C@H]1CCC[C@H]1CO)Oc1ccccc1 ZINC000217878382 BD For-Sale Unstable FAAH2 0 41 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cn(C)nc1OC ZINC000217878384 GD For-Sale Unstable HCRTR2 40 34 COc1cccc(-c2noc(CN(C)C(=O)c3cccc([N+](=O)[O-])c3C)n2)c1 ZINC000217878401 GG In-Stock Unstable HSD17B2 21 42 COc1ccc2[nH]c3c(c2c1)CCC[C@@H]3NC(=O)CC(C)C ZINC000217878430 DH In-Stock Unstable MAPKAPK2 26 49 COc1ccc2[nH]c3c(c2c1)CCC[C@@H]3NC(=O)CC(C)C ZINC000217878430 DH In-Stock Unstable MTNR1A 44 39 COc1ccc2[nH]c3c(c2c1)CCC[C@@H]3NC(=O)CC(C)C ZINC000217878430 DH In-Stock Unstable MTNR1B 47 39 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cn(C)nc1OC ZINC000217878446 GD For-Sale Unstable HCRTR2 40 34 CC(C)C[C@H]1C[C@H](NC(=O)OC(C)(C)C)CCN1 ZINC000217878448 CF For-Sale Unstable CTSK 16 40 COc1ccc2[nH]c3c(c2c1)CCC[C@H]3NC(=O)CC(C)C ZINC000217878509 DH In-Stock Unstable MAPKAPK2 26 49 COc1ccc2[nH]c3c(c2c1)CCC[C@H]3NC(=O)CC(C)C ZINC000217878509 DH In-Stock Unstable MTNR1A 44 39 COc1ccc2[nH]c3c(c2c1)CCC[C@H]3NC(=O)CC(C)C ZINC000217878509 DH In-Stock Unstable MTNR1B 47 39 CC(=O)Nc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217878530 DH For-Sale Unstable MMP2 15 46 CC(=O)Nc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217878530 DH For-Sale Unstable MMP9 16 49 CC(=O)Nc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217878530 DH For-Sale Unstable MMP1 18 46 CC(=O)Nc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217878530 DH For-Sale Unstable IDO1 31 48 CC(=O)Nc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217878530 DH For-Sale Unstable KCNK3 49 38 CC(C)C[C@@H]1C[C@@H](NC(=O)OC(C)(C)C)CCN1 ZINC000217878546 CF For-Sale Unstable CTSK 16 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cn(C)nc1OC ZINC000217878551 GD For-Sale Unstable HCRTR2 40 34 Cc1c(C(=O)N(C)Cc2nc(-c3ccccc3Cl)no2)cccc1[N+](=O)[O-] ZINC000217878566 GH In-Stock Unstable COLA 40 35 O=C(O)/C=C\c1cccc(CSc2ccc(F)c(F)c2)c1 ZINC000217878599 DI For-Sale Unstable LTB4R 18 42 O=C(O)/C=C\c1cccc(CSc2ccc(F)c(F)c2)c1 ZINC000217878599 DI For-Sale Unstable AKR1C3 32 42 CC(C)C[C@H]1C[C@@H](NC(=O)OC(C)(C)C)CCN1 ZINC000217878601 CF For-Sale Unstable CTSK 16 40 Cc1cccc(/C=C/NC(=O)Nc2ccc(S(=O)(=O)O)cc2)c1 ZINC000217878647 EG For-Sale Unstable LPL 43 34 Cc1cccc(/C=C/NC(=O)Nc2ccc(S(=O)(=O)O)cc2)c1 ZINC000217878647 EG For-Sale Unstable CA12 21 41 Cc1cccc(/C=C/NC(=O)Nc2ccc(S(=O)(=O)O)cc2)c1 ZINC000217878647 EG For-Sale Unstable CA9 17 41 Cc1cccc(/C=C/NC(=O)Nc2ccc(S(=O)(=O)O)cc2)c1 ZINC000217878647 EG For-Sale Unstable IDO1 34 48 Cc1cccc(/C=C/NC(=O)Nc2ccc(S(=O)(=O)O)cc2)c1 ZINC000217878647 EG For-Sale Unstable MTCA1 42 41 Cc1cccc(/C=C/NC(=O)Nc2ccc(S(=O)(=O)O)cc2)c1 ZINC000217878647 EG For-Sale Unstable P96878_MYCTU 53 41 CC[C@@H](C)NCCN1C[C@@H](C)Cc2ccccc21 ZINC000217878671 BG For-Sale Unstable TPP2 52 34 O=C(O)/C=C\c1ccccc1CSc1ccc(F)cc1F ZINC000217878701 DI For-Sale Unstable PTGER2 45 47 O=C(O)/C=C\c1ccccc1CSc1ccc(F)cc1F ZINC000217878701 DI For-Sale Unstable PTGER4 23 46 O=C(O)/C=C\c1ccccc1CSc1ccc(F)cc1F ZINC000217878701 DI For-Sale Unstable PTGER3 22 47 O=C(O)/C=C\c1ccccc1CSc1ccc(F)cc1F ZINC000217878701 DI For-Sale Unstable PTGDR 0 47 CC[C@H](C)NCCN1C[C@@H](C)Cc2ccccc21 ZINC000217878735 BG For-Sale Unstable TPP2 52 34 C[C@@H]1CCN(c2ccc(CBr)cc2C(F)(F)F)C[C@@H]1C ZINC000217878737 FK For-Sale Unstable LIPG 40 35 COC(=O)c1ccnc(N[C@@H](C)c2ccc(C)s2)c1 ZINC000217878742 CG On-Demand Unstable KDM3A 0 47 COC(=O)c1ccnc(N[C@@H](C)c2ccc(C)s2)c1 ZINC000217878742 CG On-Demand Unstable KDM5C 0 47 CCCC[C@@H]1C[C@@H](O)CN1C ZINC000217878745 AD In-Stock Unstable GBA2 42 33 C[C@@H](C(=O)O)c1ccc(CN2CCC[C@@H](CO)C2)cc1 ZINC000217878747 CE For-Sale Unstable SLC6A1 42 32 C[C@@H](C(=O)O)c1ccc(CN2CCC[C@@H](CO)C2)cc1 ZINC000217878747 CE For-Sale Unstable SIGMAR1 24 46 CCOC(=O)CSCCOc1cccc(/C=C\C(=O)O)c1 ZINC000217878752 DE For-Sale Unstable PLA2G4B 32 40 CCOC(=O)CSCCOc1cccc(/C=C\C(=O)O)c1 ZINC000217878752 DE For-Sale Unstable AKR1C3 29 40 Cc1ccc2c(c1)CCCN2S(=O)(=O)C[C@@]12CC[C@@H](CC1=O)C2(C)C ZINC000217878780 FG On-Demand Unstable CA5B 25 42 Cc1ccc2c(c1)CCCN2S(=O)(=O)C[C@@]12CC[C@@H](CC1=O)C2(C)C ZINC000217878780 FG On-Demand Unstable CA5A 28 42 Cc1ccc2c(c1)CCCN2S(=O)(=O)C[C@@]12CC[C@@H](CC1=O)C2(C)C ZINC000217878780 FG On-Demand Unstable CXCR3 47 47 Cc1cccc(/C=C/NC(=O)Nc2cccc(S(=O)(=O)O)c2)c1 ZINC000217878786 EG For-Sale Unstable FBP1 0 41 Cc1cccc(/C=C/NC(=O)Nc2cccc(S(=O)(=O)O)c2)c1 ZINC000217878786 EG For-Sale Unstable IDO1 17 42 Cc1cccc(/C=C/NC(=O)Nc2cccc(S(=O)(=O)O)c2)c1 ZINC000217878786 EG For-Sale Unstable KCNK3 53 38 Cc1cccc(/C=C/NC(=O)Nc2cccc(S(=O)(=O)O)c2)c1 ZINC000217878786 EG For-Sale Unstable KCNK9 42 38 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](CO)C2)cc1 ZINC000217878808 CE For-Sale Unstable SLC6A1 42 32 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](CO)C2)cc1 ZINC000217878808 CE For-Sale Unstable SIGMAR1 24 46 CCOC(=O)CSCCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217878831 DE For-Sale Unstable PLA2G4B 47 39 COC(=O)c1ccnc(N[C@H](C)c2ccc(C)s2)c1 ZINC000217878833 CG On-Demand Unstable KDM3A 0 47 COC(=O)c1ccnc(N[C@H](C)c2ccc(C)s2)c1 ZINC000217878833 CG On-Demand Unstable KDM5C 0 47 CCCC[C@H]1C[C@@H](O)CN1C ZINC000217878836 AD In-Stock Unstable GBA2 42 33 C[C@H]1CCN(c2ccc(CBr)cc2C(F)(F)F)C[C@@H]1C ZINC000217878847 FK For-Sale Unstable LIPG 40 35 Cc1c(C(=O)NCCCN2CCCc3ccccc32)cccc1[N+](=O)[O-] ZINC000217878886 FG In-Stock Unstable HTR1A 15 40 Cc1c(C(=O)NCCCN2CCCc3ccccc32)cccc1[N+](=O)[O-] ZINC000217878886 FG In-Stock Unstable DRD2 19 40 Cc1c(C(=O)NCCCN2CCCc3ccccc32)cccc1[N+](=O)[O-] ZINC000217878886 FG In-Stock Unstable AVPR2 30 46 Cc1c(C(=O)NCCCN2CCCc3ccccc32)cccc1[N+](=O)[O-] ZINC000217878886 FG In-Stock Unstable ADRA1B 22 42 CCCC[C@@H]1C[C@H](O)CN1C ZINC000217878913 AD In-Stock Unstable GBA2 42 33 Cc1cnc(SCc2ccccc2/C=C\C(=O)O)nc1 ZINC000217878916 CG For-Sale Unstable PTGER2 49 46 Cc1cnc(SCc2ccccc2/C=C\C(=O)O)nc1 ZINC000217878916 CG For-Sale Unstable PTGER4 23 46 Cc1cnc(SCc2ccccc2/C=C\C(=O)O)nc1 ZINC000217878916 CG For-Sale Unstable PTGER3 18 47 CCCC[C@H]1C[C@H](O)CN1C ZINC000217878968 AD In-Stock Unstable GBA2 42 33 Cc1cnc(SCc2ccc(/C=C\C(=O)O)cc2)nc1 ZINC000217878984 CG For-Sale Unstable PTGER2 0 40 COc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217878996 EG In-Stock Unstable HTR1A 19 47 COc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217878996 EG In-Stock Unstable DRD2 32 47 COc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217878996 EG In-Stock Unstable DRD1 0 47 COc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217878996 EG In-Stock Unstable DRD4 43 34 COc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217878996 EG In-Stock Unstable ACHE 15 47 COc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217878996 EG In-Stock Unstable ADRA1D 17 43 COc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217878996 EG In-Stock Unstable DRD3 45 47 COc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217878996 EG In-Stock Unstable CYSLTR1 47 37 COc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217878996 EG In-Stock Unstable PTAFR 15 51 COc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217878996 EG In-Stock Unstable PDE4D 17 44 COc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217878996 EG In-Stock Unstable PPARD 15 40 COc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217878996 EG In-Stock Unstable MTNR1A 55 41 COc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217878996 EG In-Stock Unstable MTNR1B 66 51 COc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217878996 EG In-Stock Unstable ABCB1 25 44 COc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217878996 EG In-Stock Unstable SCN5A 0 44 COc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217878996 EG In-Stock Unstable PTGDR 21 40 COc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217878996 EG In-Stock Unstable MT-ND1 24 40 COc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217878996 EG In-Stock Unstable MCHR1 15 41 COc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217878996 EG In-Stock Unstable PTGDR2 19 40 COc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217878996 EG In-Stock Unstable ABCG2 36 44 COc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217878996 EG In-Stock Unstable MBTPS1 42 36 COc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217878996 EG In-Stock Unstable AP2S1 0 44 COc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217878996 EG In-Stock Unstable ALPHA-1A 0 42 COc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217878996 EG In-Stock Unstable KCNK3 43 36 O=c1cc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)oc(CN2CCN(c3ccc(F)cc3)CC2)c1O ZINC000217879016 KF In-Stock Unstable CHRNA4 30 55 CCCC[C@@H]1C[C@@H](O)CN1CC ZINC000217879079 AD In-Stock Unstable GBA2 41 32 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H]2C)cc1 ZINC000217879105 BF For-Sale Unstable PTGS1 30 52 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H]2C)cc1 ZINC000217879105 BF For-Sale Unstable PTGS2 0 52 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H]2C)cc1 ZINC000217879105 BF For-Sale Unstable HRH3 70 52 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H]2C)cc1 ZINC000217879105 BF For-Sale Unstable SLC22A20 0 48 CC(C)C[C@H]1NCCC[C@H]1NC(=O)OC(C)(C)C ZINC000217879108 CF For-Sale Unstable CTSK 18 40 Cc1cccc(/C=C/NC(=O)Nc2ccc(C(C)C)cc2)c1 ZINC000217879112 CJ For-Sale Unstable CA1 15 40 Cc1cccc(/C=C/NC(=O)Nc2ccc(C(C)C)cc2)c1 ZINC000217879112 CJ For-Sale Unstable MMP1 0 42 COc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1OC ZINC000217879114 FI In-Stock Unstable EPHX1 0 41 COc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1OC ZINC000217879114 FI In-Stock Unstable PPARA 0 42 COc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1OC ZINC000217879114 FI In-Stock Unstable F10 0 48 COc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1OC ZINC000217879114 FI In-Stock Unstable MAPK14 17 49 COc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1OC ZINC000217879114 FI In-Stock Unstable ECR 24 40 COc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1OC ZINC000217879114 FI In-Stock Unstable COLA 51 38 COc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1OC ZINC000217879114 FI In-Stock Unstable CPT1A 51 38 COc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1OC ZINC000217879114 FI In-Stock Unstable PYGL 21 45 COc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1OC ZINC000217879114 FI In-Stock Unstable SYK 20 41 COc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1OC ZINC000217879114 FI In-Stock Unstable PPARD 28 44 COc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1OC ZINC000217879114 FI In-Stock Unstable KDR 42 36 COc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1OC ZINC000217879114 FI In-Stock Unstable ABCB1B 26 44 COc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1OC ZINC000217879114 FI In-Stock Unstable SLC9A1 47 34 COc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1OC ZINC000217879114 FI In-Stock Unstable NR1H4 26 59 COc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1OC ZINC000217879114 FI In-Stock Unstable HDAC1 26 49 COc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1OC ZINC000217879114 FI In-Stock Unstable HDAC2 19 49 COc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1OC ZINC000217879114 FI In-Stock Unstable PTK2 21 42 COc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1OC ZINC000217879114 FI In-Stock Unstable ABCB1 35 49 COc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1OC ZINC000217879114 FI In-Stock Unstable KCNMA1 30 42 COc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1OC ZINC000217879114 FI In-Stock Unstable FABH 0 50 COc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1OC ZINC000217879114 FI In-Stock Unstable AKR1C3 29 40 COc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1OC ZINC000217879114 FI In-Stock Unstable ABCG2 65 49 COc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1OC ZINC000217879114 FI In-Stock Unstable PAGA 0 49 COc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1OC ZINC000217879114 FI In-Stock Unstable AKR1C2 46 38 COc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1OC ZINC000217879114 FI In-Stock Unstable SMO 32 41 COc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1OC ZINC000217879114 FI In-Stock Unstable GPR35 39 46 COc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1OC ZINC000217879114 FI In-Stock Unstable GLMU 0 43 COc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1OC ZINC000217879114 FI In-Stock Unstable KCNK3 109 49 COc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1OC ZINC000217879114 FI In-Stock Unstable KCNK9 75 45 COc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1OC ZINC000217879114 FI In-Stock Unstable BRPF1 0 43 CCCC[C@H]1C[C@@H](O)CN1CC ZINC000217879154 AD In-Stock Unstable GBA2 41 32 CC(C)C[C@@H]1NCCC[C@H]1NC(=O)OC(C)(C)C ZINC000217879194 CF For-Sale Unstable CTSK 18 40 COc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217879203 CG For-Sale Unstable PTGER2 27 59 COc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217879203 CG For-Sale Unstable PPIA 41 32 COc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217879203 CG For-Sale Unstable PTGER4 47 59 COc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217879203 CG For-Sale Unstable CYP1B1 30 42 COc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217879203 CG For-Sale Unstable PTGER3 33 59 COc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217879203 CG For-Sale Unstable KCNA3 27 44 COc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217879203 CG For-Sale Unstable TNFRSF1A 28 44 COc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217879203 CG For-Sale Unstable CA14 0 50 COc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217879203 CG For-Sale Unstable CYP1A1 27 42 COc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217879203 CG For-Sale Unstable 17HSDCL 0 45 COc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217879203 CG For-Sale Unstable AKR1C3 38 52 COc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217879203 CG For-Sale Unstable ABCG2 22 47 COc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217879203 CG For-Sale Unstable AKR1B10 39 43 COc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217879203 CG For-Sale Unstable GPR183 0 41 C[C@H](CCc1ccc(O)cc1)N1CCC[C@@H]2CCC[C@@H]21 ZINC000217879217 CH For-Sale Unstable BIRC2 50 38 CCCC[C@@H]1C[C@H](O)CN1CC ZINC000217879230 AD In-Stock Unstable GBA2 41 32 CCOc1ccc(CCCNC(=O)c2ccc(OC)c(OC)c2)cc1 ZINC000217879236 EG In-Stock Unstable DRD2 15 40 CCOc1ccc(CCCNC(=O)c2ccc(OC)c(OC)c2)cc1 ZINC000217879236 EG In-Stock Unstable DRD4 41 31 CCOc1ccc(CCCNC(=O)c2ccc(OC)c(OC)c2)cc1 ZINC000217879236 EG In-Stock Unstable DRD3 22 40 CCOc1ccc(CCCNC(=O)c2ccc(OC)c(OC)c2)cc1 ZINC000217879236 EG In-Stock Unstable PPARA 17 44 CCOc1ccc(CCCNC(=O)c2ccc(OC)c(OC)c2)cc1 ZINC000217879236 EG In-Stock Unstable PTAFR 19 51 CCOc1ccc(CCCNC(=O)c2ccc(OC)c(OC)c2)cc1 ZINC000217879236 EG In-Stock Unstable CNR2 45 39 CCOc1ccc(CCCNC(=O)c2ccc(OC)c(OC)c2)cc1 ZINC000217879236 EG In-Stock Unstable KCNQ1 0 40 CCOc1ccc(CCCNC(=O)c2ccc(OC)c(OC)c2)cc1 ZINC000217879236 EG In-Stock Unstable TRPV1 0 47 CCOc1ccc(CCCNC(=O)c2ccc(OC)c(OC)c2)cc1 ZINC000217879236 EG In-Stock Unstable SCN2A 24 53 CCOc1ccc(CCCNC(=O)c2ccc(OC)c(OC)c2)cc1 ZINC000217879236 EG In-Stock Unstable MTNR1A 33 41 CCOc1ccc(CCCNC(=O)c2ccc(OC)c(OC)c2)cc1 ZINC000217879236 EG In-Stock Unstable MTNR1B 27 47 CCOc1ccc(CCCNC(=O)c2ccc(OC)c(OC)c2)cc1 ZINC000217879236 EG In-Stock Unstable PLA2G4B 45 41 CCOc1ccc(CCCNC(=O)c2ccc(OC)c(OC)c2)cc1 ZINC000217879236 EG In-Stock Unstable SCN5A 0 44 CCOc1ccc(CCCNC(=O)c2ccc(OC)c(OC)c2)cc1 ZINC000217879236 EG In-Stock Unstable PTGDR 27 42 CCOc1ccc(CCCNC(=O)c2ccc(OC)c(OC)c2)cc1 ZINC000217879236 EG In-Stock Unstable MT-ND1 30 48 CCOc1ccc(CCCNC(=O)c2ccc(OC)c(OC)c2)cc1 ZINC000217879236 EG In-Stock Unstable MCHR1 16 44 CCOc1ccc(CCCNC(=O)c2ccc(OC)c(OC)c2)cc1 ZINC000217879236 EG In-Stock Unstable PTGDR2 20 42 CCOc1ccc(CCCNC(=O)c2ccc(OC)c(OC)c2)cc1 ZINC000217879236 EG In-Stock Unstable ABCG2 31 45 CCOc1ccc(CCCNC(=O)c2ccc(OC)c(OC)c2)cc1 ZINC000217879236 EG In-Stock Unstable AP2S1 0 40 CCOc1ccc(CCCNC(=O)c2ccc(OC)c(OC)c2)cc1 ZINC000217879236 EG In-Stock Unstable CAN2 0 41 COc1ccccc1NC(=O)N/C=C/c1cccc(C)c1 ZINC000217879237 CH For-Sale Unstable KCNK3 43 40 COc1ccccc1NC(=O)N/C=C/c1cccc(C)c1 ZINC000217879237 CH For-Sale Unstable KCNK9 47 40 CC(C)(C)OC(=O)NCCC1CCN(C(=O)OCc2cc(Cl)cc(Cl)c2)CC1 ZINC000217879247 IK For-Sale Unstable GRIN2B 21 44 CC(C)(C)OC(=O)NCCC1CCN(C(=O)OCc2cc(Cl)cc(Cl)c2)CC1 ZINC000217879247 IK For-Sale Unstable CACNA1I 78 41 CC(C)(C)OC(=O)NCCC1CCN(C(=O)OCc2cc(Cl)cc(Cl)c2)CC1 ZINC000217879247 IK For-Sale Unstable SIRT3 34 44 CC(C)(C)OC(=O)NCCC1CCN(C(=O)OCc2cc(Cl)cc(Cl)c2)CC1 ZINC000217879247 IK For-Sale Unstable SIRT2 34 44 CC(C)(C)OC(=O)NCCC1CCN(C(=O)OCc2cc(Cl)cc(Cl)c2)CC1 ZINC000217879247 IK For-Sale Unstable SIRT1 34 44 CC(C)(C)OC(=O)NCCC1CCN(C(=O)OCc2cc(Cl)cc(Cl)c2)CC1 ZINC000217879247 IK For-Sale Unstable GPR119 36 43 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](C)C2)cc1 ZINC000217879260 BF For-Sale Unstable ACHE 16 48 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](C)C2)cc1 ZINC000217879260 BF For-Sale Unstable PTGS1 34 49 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](C)C2)cc1 ZINC000217879260 BF For-Sale Unstable PTGS2 23 49 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](C)C2)cc1 ZINC000217879260 BF For-Sale Unstable VACHT_TETCF 0 41 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](C)C2)cc1 ZINC000217879260 BF For-Sale Unstable SIGMAR1 43 39 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](C)C2)cc1 ZINC000217879260 BF For-Sale Unstable SLC18A3 27 40 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](C)C2)cc1 ZINC000217879260 BF For-Sale Unstable MLNR 57 43 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](C)C2)cc1 ZINC000217879260 BF For-Sale Unstable SLC22A20 0 48 COc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217879287 CG For-Sale Unstable ALOX5 18 42 COc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217879287 CG For-Sale Unstable MAOB 25 45 COc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217879287 CG For-Sale Unstable PTGER2 29 58 COc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217879287 CG For-Sale Unstable PPIA 42 34 COc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217879287 CG For-Sale Unstable PTGER1 52 40 COc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217879287 CG For-Sale Unstable PTGER4 47 58 COc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217879287 CG For-Sale Unstable CYP1B1 30 43 COc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217879287 CG For-Sale Unstable PTGER3 36 58 COc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217879287 CG For-Sale Unstable LTB4R 41 48 COc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217879287 CG For-Sale Unstable KCNA3 20 45 COc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217879287 CG For-Sale Unstable TNFRSF1A 28 40 COc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217879287 CG For-Sale Unstable CA14 0 51 COc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217879287 CG For-Sale Unstable MTNR1B 17 45 COc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217879287 CG For-Sale Unstable MMP2 0 49 COc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217879287 CG For-Sale Unstable CYP1A1 25 43 COc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217879287 CG For-Sale Unstable NR1H4 42 39 COc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217879287 CG For-Sale Unstable ABCB1 18 51 COc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217879287 CG For-Sale Unstable 17HSDCL 0 43 COc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217879287 CG For-Sale Unstable FFAR1 36 43 COc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217879287 CG For-Sale Unstable AKR1C3 44 58 COc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217879287 CG For-Sale Unstable PTPA 0 43 COc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217879287 CG For-Sale Unstable ABCG2 25 43 COc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217879287 CG For-Sale Unstable ADCYAP1R1 46 38 COc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217879287 CG For-Sale Unstable TRPM8 0 41 COc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217879287 CG For-Sale Unstable AKR1B10 39 43 CC(C)[C@@H]1COC(=O)N1c1ccnc(N[C@@H](C)c2ccc(CN3CCC(F)(F)CC3)cc2)n1 ZINC000217879290 JJ For-Sale Anodyne IDH1 18 45 CC(C)C[C@H]1NCCC[C@@H]1NC(=O)OC(C)(C)C ZINC000217879294 CF For-Sale Unstable CTSK 18 40 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cc(OC)c(OC(C)=O)c(OC)c2)CC(=O)O4)cc1O ZINC000217879305 KI In-Stock Unstable ALOX5 0 49 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cc(OC)c(OC(C)=O)c(OC)c2)CC(=O)O4)cc1O ZINC000217879305 KI In-Stock Unstable AKR1B1 0 49 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cc(OC)c(OC(C)=O)c(OC)c2)CC(=O)O4)cc1O ZINC000217879305 KI In-Stock Unstable CYP1B1 67 37 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cc(OC)c(OC(C)=O)c(OC)c2)CC(=O)O4)cc1O ZINC000217879305 KI In-Stock Unstable CYP1A1 43 45 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cc(OC)c(OC(C)=O)c(OC)c2)CC(=O)O4)cc1O ZINC000217879305 KI In-Stock Unstable CYP1A2 36 41 CCCC[C@H]1C[C@H](O)CN1CC ZINC000217879319 AD In-Stock Unstable GBA2 41 32 CC[C@@H](C)N(C)CCNCCCc1ccccc1 ZINC000217879343 BF For-Sale Unstable SIGMAR1 21 58 CCCOc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217879348 FH In-Stock Unstable HTR1A 15 42 CCCOc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217879348 FH In-Stock Unstable DRD2 26 48 CCCOc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217879348 FH In-Stock Unstable DRD1 0 44 CCCOc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217879348 FH In-Stock Unstable DRD3 34 44 CCCOc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217879348 FH In-Stock Unstable PPARG 20 42 CCCOc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217879348 FH In-Stock Unstable PTAFR 17 46 CCCOc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217879348 FH In-Stock Unstable CNR2 39 41 CCCOc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217879348 FH In-Stock Unstable PDE4D 15 40 CCCOc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217879348 FH In-Stock Unstable MTNR1A 43 42 CCCOc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217879348 FH In-Stock Unstable MTNR1B 57 48 CCCOc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217879348 FH In-Stock Unstable REN 20 41 CCCOc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217879348 FH In-Stock Unstable ABCB1 22 42 CCCOc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217879348 FH In-Stock Unstable PTGDR 20 40 CCCOc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217879348 FH In-Stock Unstable PTGDR2 18 40 CCCOc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217879348 FH In-Stock Unstable ABCG2 17 44 CCCOc1ccccc1CCCNC(=O)c1ccc(OC)c(OC)c1 ZINC000217879348 FH In-Stock Unstable ALPHA-1A 0 41 CN(CCC1CCN(C(=O)OCc2cc(Cl)cc(Cl)c2)CC1)C(=O)OC(C)(C)C ZINC000217879349 IK For-Sale Unstable GRIN2B 18 41 CN(CCC1CCN(C(=O)OCc2cc(Cl)cc(Cl)c2)CC1)C(=O)OC(C)(C)C ZINC000217879349 IK For-Sale Unstable CACNA1I 48 36 CN(CCC1CCN(C(=O)OCc2cc(Cl)cc(Cl)c2)CC1)C(=O)OC(C)(C)C ZINC000217879349 IK For-Sale Unstable GPR119 30 40 N#Cc1cccc(C(=O)NCCn2nc(-c3ccsc3)cc2C2CC2)c1 ZINC000217879354 FH In-Stock Unstable DRD4 40 31 Cc1cccc(/C=C/NC(=O)Nc2ccccc2C)c1 ZINC000217879358 CI For-Sale Unstable MMP1 0 55 Cc1cccc(/C=C/NC(=O)Nc2ccccc2C)c1 ZINC000217879358 CI For-Sale Unstable DDX3X 0 46 Cc1cccc(/C=C/NC(=O)Nc2ccccc2C)c1 ZINC000217879358 CI For-Sale Unstable KCNK3 44 36 CC(C)[C@@H]1COC(=O)N1c1ccnc(N[C@H](C)c2ccc(CN3CCC(F)(F)CC3)cc2)n1 ZINC000217879364 JJ In-Stock Unstable IDH1 18 45 O=C(O)/C=C\c1ccccc1COc1cccc(F)c1 ZINC000217879369 CH For-Sale Unstable PTGER2 22 46 O=C(O)/C=C\c1ccccc1COc1cccc(F)c1 ZINC000217879369 CH For-Sale Unstable PTGER4 35 55 O=C(O)/C=C\c1ccccc1COc1cccc(F)c1 ZINC000217879369 CH For-Sale Unstable PTGER3 29 56 O=C(O)/C=C\c1ccccc1COc1cccc(F)c1 ZINC000217879369 CH For-Sale Unstable CDC25B 24 43 O=C(O)/C=C\c1ccccc1COc1cccc(F)c1 ZINC000217879369 CH For-Sale Unstable PTGDR 0 56 O=C(O)/C=C\c1ccccc1COc1cccc(F)c1 ZINC000217879369 CH For-Sale Unstable HCAR2 0 44 O=C(O)/C=C\c1ccccc1COc1cccc(F)c1 ZINC000217879369 CH For-Sale Unstable AKR1C3 28 41 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cc(OC)c(OC(C)=O)c(OC)c2)CC(=O)O4)cc1O ZINC000217879370 KI In-Stock Unstable ALOX5 0 49 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cc(OC)c(OC(C)=O)c(OC)c2)CC(=O)O4)cc1O ZINC000217879370 KI In-Stock Unstable AKR1B1 0 49 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cc(OC)c(OC(C)=O)c(OC)c2)CC(=O)O4)cc1O ZINC000217879370 KI In-Stock Unstable CYP1B1 67 37 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cc(OC)c(OC(C)=O)c(OC)c2)CC(=O)O4)cc1O ZINC000217879370 KI In-Stock Unstable CYP1A1 43 45 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cc(OC)c(OC(C)=O)c(OC)c2)CC(=O)O4)cc1O ZINC000217879370 KI In-Stock Unstable CYP1A2 36 41 CC(C)C[C@@H]1NCCC[C@@H]1NC(=O)OC(C)(C)C ZINC000217879380 CF For-Sale Unstable CTSK 18 40 C[C@@H](C(=O)O)c1ccc(CN2CCC[C@@H](N)C2)cc1 ZINC000217879401 CD For-Sale Unstable SLC6A1 50 33 C[C@@H](C(=O)O)c1ccc(CN2CCC[C@@H](N)C2)cc1 ZINC000217879401 CD For-Sale Unstable SIGMAR1 27 41 C[C@@H](C(=O)O)c1ccc(CN2CCC[C@@H](N)C2)cc1 ZINC000217879401 CD For-Sale Unstable SLC22A20 0 44 CC[C@H](C)N(C)CCNCCCc1ccccc1 ZINC000217879433 BF For-Sale Unstable SIGMAR1 21 58 CCCC[C@@H]1C[C@@H](O)CN1CCC ZINC000217879438 AE In-Stock Unstable GBA2 44 34 CCCC[C@@H]1C[C@@H](O)CN1CCC ZINC000217879438 AE In-Stock Unstable P0504H10.9 57 36 CCCC[C@@H]1C[C@@H](O)CN1CCC ZINC000217879438 AE In-Stock Unstable SIS 66 34 CNCCC1CCN(C(=O)OCc2cc(Cl)cc(Cl)c2)CC1 ZINC000217879444 EH For-Sale Unstable GRIN2B 25 44 CNCCC1CCN(C(=O)OCc2cc(Cl)cc(Cl)c2)CC1 ZINC000217879444 EH For-Sale Unstable ST14 52 34 CNCCC1CCN(C(=O)OCc2cc(Cl)cc(Cl)c2)CC1 ZINC000217879444 EH For-Sale Unstable CACNA1I 72 42 CNCCC1CCN(C(=O)OCc2cc(Cl)cc(Cl)c2)CC1 ZINC000217879444 EH For-Sale Unstable TMPRSS6 51 32 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](N)C2)cc1 ZINC000217879461 CD For-Sale Unstable SLC6A1 50 33 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](N)C2)cc1 ZINC000217879461 CD For-Sale Unstable SIGMAR1 27 41 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](N)C2)cc1 ZINC000217879461 CD For-Sale Unstable SLC22A20 0 44 Cc1ccc(OCc2ccc(F)cc2/C=C\C(=O)O)cc1 ZINC000217879463 CH For-Sale Unstable PTGER2 51 43 Cc1ccc(OCc2ccc(F)cc2/C=C\C(=O)O)cc1 ZINC000217879463 CH For-Sale Unstable PTGER4 19 40 Cc1ccc(OCc2ccc(F)cc2/C=C\C(=O)O)cc1 ZINC000217879463 CH For-Sale Unstable PTGER3 23 43 Cc1ccc(OCc2ccc(F)cc2/C=C\C(=O)O)cc1 ZINC000217879463 CH For-Sale Unstable PTGDR 0 42 Cc1ccc(OCc2ccc(F)cc2/C=C\C(=O)O)cc1 ZINC000217879463 CH For-Sale Unstable FFAR1 24 40 Cc1ccc(OCc2ccc(F)cc2/C=C\C(=O)O)cc1 ZINC000217879463 CH For-Sale Unstable AKR1C3 27 43 Cc1ccc(OCc2ccc(F)cc2/C=C\C(=O)O)cc1 ZINC000217879463 CH For-Sale Unstable FFAR4 41 51 CC(C)[C@H]1COC(=O)N1c1ccnc(N[C@H](C)c2ccc(CN3CCC(F)(F)CC3)cc2)n1 ZINC000217879471 JJ For-Sale Anodyne IDH1 18 45 Cc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c(Cl)c2)c1 ZINC000217879501 DK For-Sale Unstable KIT 21 40 Cc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c(Cl)c2)c1 ZINC000217879501 DK For-Sale Unstable KDR 20 41 Cc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c(Cl)c2)c1 ZINC000217879501 DK For-Sale Unstable CSF1R 17 40 Cc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c(Cl)c2)c1 ZINC000217879501 DK For-Sale Unstable IDO1 15 40 Cc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c(Cl)c2)c1 ZINC000217879501 DK For-Sale Unstable IMDH_CRYPV 39 43 Cc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c(Cl)c2)c1 ZINC000217879501 DK For-Sale Unstable KCNK3 52 38 CCCC[C@H]1C[C@@H](O)CN1CCC ZINC000217879531 AE In-Stock Unstable GBA2 44 34 CCCC[C@H]1C[C@@H](O)CN1CCC ZINC000217879531 AE In-Stock Unstable P0504H10.9 57 36 CCCC[C@H]1C[C@@H](O)CN1CCC ZINC000217879531 AE In-Stock Unstable SIS 66 34 NCCC1CCN(C(=O)OCc2cc(Cl)cc(Cl)c2)CC1 ZINC000217879548 EH For-Sale Unstable PLG 15 43 NCCC1CCN(C(=O)OCc2cc(Cl)cc(Cl)c2)CC1 ZINC000217879548 EH For-Sale Unstable GRIN2B 22 45 NCCC1CCN(C(=O)OCc2cc(Cl)cc(Cl)c2)CC1 ZINC000217879548 EH For-Sale Unstable ST14 55 41 NCCC1CCN(C(=O)OCc2cc(Cl)cc(Cl)c2)CC1 ZINC000217879548 EH For-Sale Unstable CACNA1I 62 43 Cc1ccc(OCc2ccc(F)c(/C=C\C(=O)O)c2)cc1 ZINC000217879580 CH For-Sale Unstable PTGER2 16 45 Cc1ccc(OCc2ccc(F)c(/C=C\C(=O)O)c2)cc1 ZINC000217879580 CH For-Sale Unstable PTGER4 39 43 Cc1ccc(OCc2ccc(F)c(/C=C\C(=O)O)c2)cc1 ZINC000217879580 CH For-Sale Unstable PTGER3 41 36 Cc1ccc(OCc2ccc(F)c(/C=C\C(=O)O)c2)cc1 ZINC000217879580 CH For-Sale Unstable PPARD 17 42 Cc1ccc(OCc2ccc(F)c(/C=C\C(=O)O)c2)cc1 ZINC000217879580 CH For-Sale Unstable GYS1 61 37 Cc1ccc(OCc2ccc(F)c(/C=C\C(=O)O)c2)cc1 ZINC000217879580 CH For-Sale Unstable PTGDR 0 46 Cc1ccc(OCc2ccc(F)c(/C=C\C(=O)O)c2)cc1 ZINC000217879580 CH For-Sale Unstable FFAR1 69 45 Cc1ccc(OCc2ccc(F)c(/C=C\C(=O)O)c2)cc1 ZINC000217879580 CH For-Sale Unstable AKR1C3 27 45 Cc1ccc(OCc2ccc(F)c(/C=C\C(=O)O)c2)cc1 ZINC000217879580 CH For-Sale Unstable FFAR4 47 42 O=C(O)COc1ccccc1[C@@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc3c21 ZINC000217879582 JH In-Stock Unstable AKR1B1 0 43 O=C(O)COc1ccccc1[C@@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc3c21 ZINC000217879582 JH In-Stock Unstable CYP1A1 28 40 O=C(O)COc1ccccc1[C@@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc3c21 ZINC000217879582 JH In-Stock Unstable CYP1A2 20 40 Cc1cccc(/C=C/NC(=O)Nc2ccc(C)c(Cl)c2)c1 ZINC000217879595 DJ For-Sale Unstable KIT 15 43 Cc1cccc(/C=C/NC(=O)Nc2ccc(C)c(Cl)c2)c1 ZINC000217879595 DJ For-Sale Unstable MMP1 0 43 Cc1cccc(/C=C/NC(=O)Nc2ccc(C)c(Cl)c2)c1 ZINC000217879595 DJ For-Sale Unstable KCNK3 51 38 CCCC[C@@H]1C[C@H](O)CN1CCC ZINC000217879603 AE In-Stock Unstable GBA2 44 34 CCCC[C@@H]1C[C@H](O)CN1CCC ZINC000217879603 AE In-Stock Unstable P0504H10.9 57 36 CCCC[C@@H]1C[C@H](O)CN1CCC ZINC000217879603 AE In-Stock Unstable SIS 66 34 CNC[C@@H]1CCCN(Cc2ccc([C@@H](C)C(=O)O)cc2)C1 ZINC000217879629 CE For-Sale Unstable HTR4 15 43 CNC[C@@H]1CCCN(Cc2ccc([C@@H](C)C(=O)O)cc2)C1 ZINC000217879629 CE For-Sale Unstable SIGMAR1 21 43 CNC[C@@H]1CCCN(Cc2ccc([C@@H](C)C(=O)O)cc2)C1 ZINC000217879629 CE For-Sale Unstable CCR3 44 36 CNC[C@@H]1CCCN(Cc2ccc([C@@H](C)C(=O)O)cc2)C1 ZINC000217879629 CE For-Sale Unstable BIRC2 43 36 N[C@H](CCC(=O)O)c1c(Cl)ccc(F)c1O ZINC000217879644 BE For-Sale Unstable CACNA2D1 15 41 CC[C@@H]1CCCC[C@@H]1OCc1ccccc1/C=C\C(=O)O ZINC000217879650 CI For-Sale Unstable PTGER2 45 42 CC[C@@H]1CCCC[C@@H]1OCc1ccccc1/C=C\C(=O)O ZINC000217879650 CI For-Sale Unstable PTGER4 0 42 CC[C@@H]1CCCC[C@@H]1OCc1ccccc1/C=C\C(=O)O ZINC000217879650 CI For-Sale Unstable PTGER3 16 42 CC[C@@H]1CCCC[C@@H]1OCc1ccccc1/C=C\C(=O)O ZINC000217879650 CI For-Sale Unstable PTGDR 0 41 O=C(O)COc1ccccc1[C@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc3c21 ZINC000217879674 JH In-Stock Unstable AKR1B1 0 43 O=C(O)COc1ccccc1[C@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc3c21 ZINC000217879674 JH In-Stock Unstable CYP1A1 28 40 O=C(O)COc1ccccc1[C@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc3c21 ZINC000217879674 JH In-Stock Unstable CYP1A2 20 40 CCCC[C@H]1C[C@H](O)CN1CCC ZINC000217879676 AE In-Stock Unstable GBA2 44 34 CCCC[C@H]1C[C@H](O)CN1CCC ZINC000217879676 AE In-Stock Unstable P0504H10.9 57 36 CCCC[C@H]1C[C@H](O)CN1CCC ZINC000217879676 AE In-Stock Unstable SIS 66 34 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc(F)c(F)c1 ZINC000217879719 GF For-Sale Unstable CHRM5 24 40 COc1ccc(C(=O)N[C@@H](C)c2ccc(N3CCC[C@@H](C)C3)cc2)cc1OC ZINC000217879727 GI In-Stock Unstable ELANE 15 45 COc1ccc(C(=O)N[C@@H](C)c2ccc(N3CCC[C@@H](C)C3)cc2)cc1OC ZINC000217879727 GI In-Stock Unstable RORC 41 40 Cc1cccc(/C=C/NC(=O)Nc2c(C)cccc2C(C)C)c1 ZINC000217879732 DK For-Sale Unstable SOAT1 42 39 N[C@@H](CCC(=O)O)c1c(Cl)ccc(F)c1O ZINC000217879736 BE For-Sale Unstable CACNA2D1 15 41 CC[C@H]1CCCC[C@@H]1OCc1ccccc1/C=C\C(=O)O ZINC000217879758 CI For-Sale Unstable PTGER2 45 42 CC[C@H]1CCCC[C@@H]1OCc1ccccc1/C=C\C(=O)O ZINC000217879758 CI For-Sale Unstable PTGER4 0 42 CC[C@H]1CCCC[C@@H]1OCc1ccccc1/C=C\C(=O)O ZINC000217879758 CI For-Sale Unstable PTGER3 16 42 CC[C@H]1CCCC[C@@H]1OCc1ccccc1/C=C\C(=O)O ZINC000217879758 CI For-Sale Unstable PTGDR 0 41 CCCC[C@@H]1C[C@@H](O)CN1CCCC ZINC000217879777 AE In-Stock Unstable GAA 18 41 CCCC[C@@H]1C[C@@H](O)CN1CCCC ZINC000217879777 AE In-Stock Unstable GBA2 50 41 CCCC[C@@H]1C[C@@H](O)CN1CCCC ZINC000217879777 AE In-Stock Unstable P0504H10.9 0 41 CCCC[C@@H]1C[C@@H](O)CN1CCCC ZINC000217879777 AE In-Stock Unstable AGL 0 41 CCCC[C@@H]1C[C@@H](O)CN1CCCC ZINC000217879777 AE In-Stock Unstable SIS 0 41 COc1ccc(C(=O)N[C@H](C)c2ccc(N3CCC[C@@H](C)C3)cc2)cc1OC ZINC000217879800 GI In-Stock Unstable ELANE 15 45 COc1ccc(C(=O)N[C@H](C)c2ccc(N3CCC[C@@H](C)C3)cc2)cc1OC ZINC000217879800 GI In-Stock Unstable RORC 41 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc(F)c(F)c1 ZINC000217879801 GF For-Sale Unstable CHRM5 24 40 Cc1cccc(/C=C/NC(=O)Nc2ccccc2C(F)(F)F)c1 ZINC000217879833 DJ For-Sale Unstable KCNK3 32 42 CCCC[C@H]1C[C@@H](O)CN1CCCC ZINC000217879862 AE In-Stock Unstable GAA 18 41 CCCC[C@H]1C[C@@H](O)CN1CCCC ZINC000217879862 AE In-Stock Unstable GBA2 50 41 CCCC[C@H]1C[C@@H](O)CN1CCCC ZINC000217879862 AE In-Stock Unstable P0504H10.9 0 41 CCCC[C@H]1C[C@@H](O)CN1CCCC ZINC000217879862 AE In-Stock Unstable AGL 0 41 CCCC[C@H]1C[C@@H](O)CN1CCCC ZINC000217879862 AE In-Stock Unstable SIS 0 41 COc1ccc(/C=C\C(=O)O)cc1COCCOC(C)C ZINC000217879872 CF For-Sale Unstable PTGER2 0 42 COc1ccc(/C=C\C(=O)O)cc1COCCOC(C)C ZINC000217879872 CF For-Sale Unstable AKR1C3 41 43 O=C(CCn1ccc(=O)[nH]c1=O)N1CCCn2nc(CO)cc2C1 ZINC000217879886 EB In-Stock Unstable DUT 54 37 Fc1ccc(CNc2nccs2)c(Br)c1 ZINC000217879888 CH On-Demand Unstable MAP1 27 42 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc(F)c(F)c1 ZINC000217879893 GF For-Sale Unstable CHRM5 24 40 C[C@@H]1C[C@H](CNC(=O)OC(C)(C)C)CCN1C(=O)OCc1cc(Cl)cc(Cl)c1 ZINC000217879935 IK For-Sale Unstable CACNA1H 18 40 C[C@@H]1C[C@H](CNC(=O)OC(C)(C)C)CCN1C(=O)OCc1cc(Cl)cc(Cl)c1 ZINC000217879935 IK For-Sale Unstable CACNA1I 81 43 Cc1cccc(/C=C/NC(=O)Nc2ccc(C(=O)O)cc2)c1 ZINC000217879938 CG For-Sale Unstable MMP1 0 42 Cc1cccc(/C=C/NC(=O)Nc2ccc(C(=O)O)cc2)c1 ZINC000217879938 CG For-Sale Unstable AKR1C3 41 42 Cc1cccc(/C=C/NC(=O)Nc2ccc(C(=O)O)cc2)c1 ZINC000217879938 CG For-Sale Unstable KCNK3 59 38 Cc1cccc(/C=C/NC(=O)Nc2ccc(C(=O)O)cc2)c1 ZINC000217879938 CG For-Sale Unstable KCNK9 42 38 C[C@H]1C[C@H](CNC(=O)OC(C)(C)C)CCN1C(=O)OCc1cc(Cl)cc(Cl)c1 ZINC000217879951 IK For-Sale Unstable CACNA1H 18 40 C[C@H]1C[C@H](CNC(=O)OC(C)(C)C)CCN1C(=O)OCc1cc(Cl)cc(Cl)c1 ZINC000217879951 IK For-Sale Unstable CACNA1I 81 43 CCCC[C@@H]1C[C@H](O)CN1CCCC ZINC000217879956 AE In-Stock Unstable GAA 18 41 CCCC[C@@H]1C[C@H](O)CN1CCCC ZINC000217879956 AE In-Stock Unstable GBA2 50 41 CCCC[C@@H]1C[C@H](O)CN1CCCC ZINC000217879956 AE In-Stock Unstable P0504H10.9 0 41 CCCC[C@@H]1C[C@H](O)CN1CCCC ZINC000217879956 AE In-Stock Unstable AGL 0 41 CCCC[C@@H]1C[C@H](O)CN1CCCC ZINC000217879956 AE In-Stock Unstable SIS 0 41 Cc1noc(C)c1CC(=O)NCCn1nc(-c2ccsc2)cc1C1CC1 ZINC000217879960 FG In-Stock Unstable P2RX7 21 44 CC(=O)N1c2ccc(S(=O)(=O)N[C@@H](C)c3cc(F)c(Cl)cc3Cl)cc2C[C@@H]1C ZINC000217879968 II On-Demand Unstable NOD2 18 41 COc1ccc(COCCOC(C)C)cc1/C=C\C(=O)O ZINC000217879972 CF For-Sale Unstable PTGER2 35 44 COc1ccc(COCCOC(C)C)cc1/C=C\C(=O)O ZINC000217879972 CF For-Sale Unstable PTGER4 22 44 COc1ccc(COCCOC(C)C)cc1/C=C\C(=O)O ZINC000217879972 CF For-Sale Unstable PTGER3 17 44 COc1ccc(COCCOC(C)C)cc1/C=C\C(=O)O ZINC000217879972 CF For-Sale Unstable AKR1B10 30 41 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc(F)c(F)c1 ZINC000217879986 GF For-Sale Unstable CHRM5 24 40 CC(C)C[C@@H](NC(=O)OC1CCCCC1)C(=O)O ZINC000217880029 CF On-Demand Unstable EDNRA 25 41 CC(C)C[C@@H](NC(=O)OC1CCCCC1)C(=O)O ZINC000217880029 CF On-Demand Unstable CTSB 18 42 CC(C)C[C@@H](NC(=O)OC1CCCCC1)C(=O)O ZINC000217880029 CF On-Demand Unstable RIR1_HHV11 79 34 CC(C)C[C@@H](NC(=O)OC1CCCCC1)C(=O)O ZINC000217880029 CF On-Demand Unstable CTSK 24 44 CC(C)C[C@@H](NC(=O)OC1CCCCC1)C(=O)O ZINC000217880029 CF On-Demand Unstable CAPNS1 54 36 CC(C)C[C@@H](NC(=O)OC1CCCCC1)C(=O)O ZINC000217880029 CF On-Demand Unstable CAPN1 50 46 CC(C)C[C@@H](NC(=O)OC1CCCCC1)C(=O)O ZINC000217880029 CF On-Demand Unstable CAPN2 68 39 CC(C)C[C@@H](NC(=O)OC1CCCCC1)C(=O)O ZINC000217880029 CF On-Demand Unstable FPR1 51 43 CC(C)C[C@@H](NC(=O)OC1CCCCC1)C(=O)O ZINC000217880029 CF On-Demand Unstable NPR 42 36 C[C@@H]1C[C@@H](CNC(=O)OC(C)(C)C)CCN1C(=O)OCc1cc(Cl)cc(Cl)c1 ZINC000217880035 IK For-Sale Unstable CACNA1H 18 40 C[C@@H]1C[C@@H](CNC(=O)OC(C)(C)C)CCN1C(=O)OCc1cc(Cl)cc(Cl)c1 ZINC000217880035 IK For-Sale Unstable CACNA1I 81 43 CCCC[C@H]1C[C@H](O)CN1CCCC ZINC000217880041 AE In-Stock Unstable GAA 18 41 CCCC[C@H]1C[C@H](O)CN1CCCC ZINC000217880041 AE In-Stock Unstable GBA2 50 41 CCCC[C@H]1C[C@H](O)CN1CCCC ZINC000217880041 AE In-Stock Unstable P0504H10.9 0 41 CCCC[C@H]1C[C@H](O)CN1CCCC ZINC000217880041 AE In-Stock Unstable AGL 0 41 CCCC[C@H]1C[C@H](O)CN1CCCC ZINC000217880041 AE In-Stock Unstable SIS 0 41 CC(=O)N1c2ccc(S(=O)(=O)N[C@H](C)c3cc(F)c(Cl)cc3Cl)cc2C[C@@H]1C ZINC000217880045 II On-Demand Unstable NOD2 18 41 CC(C)[C@@H](NC(=O)OCC1CCCC1)C(=O)O ZINC000217880069 BE For-Sale Unstable CASP3 16 63 CC(C)[C@@H](NC(=O)OCC1CCCC1)C(=O)O ZINC000217880069 BE For-Sale Unstable DLG4 44 42 CC(=O)N1c2ccc(S(=O)(=O)N[C@@H](C)c3cc(F)c(Cl)cc3Cl)cc2C[C@H]1C ZINC000217880098 II On-Demand Unstable NOD2 18 41 COc1ccc(C(=O)N[C@@H]2CC(C)(C)Oc3cc(C)ccc32)cc1OC ZINC000217880115 FI In-Stock Unstable EZH2 41 35 C[C@H]1C[C@@H](CNC(=O)OC(C)(C)C)CCN1C(=O)OCc1cc(Cl)cc(Cl)c1 ZINC000217880124 IK For-Sale Unstable CACNA1H 18 40 C[C@H]1C[C@@H](CNC(=O)OC(C)(C)C)CCN1C(=O)OCc1cc(Cl)cc(Cl)c1 ZINC000217880124 IK For-Sale Unstable CACNA1I 81 43 CCOC(=O)c1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217880131 DH For-Sale Unstable CA1 17 45 CCOC(=O)c1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217880131 DH For-Sale Unstable ACR 64 37 CCOC(=O)c1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217880131 DH For-Sale Unstable KCNK3 45 34 CC(=O)N1c2ccc(S(=O)(=O)N[C@H](C)c3cc(F)c(Cl)cc3Cl)cc2C[C@H]1C ZINC000217880184 II On-Demand Unstable NOD2 18 41 O=C(CCCOc1ccccc1)N[C@H]1CCC[C@H]1CO ZINC000217880191 CE On-Demand Unstable CVIR 0 41 CCCCOCCOCc1ccccc1/C=C\C(=O)O ZINC000217880206 CG For-Sale Unstable PTGER2 56 48 CCCCOCCOCc1ccccc1/C=C\C(=O)O ZINC000217880206 CG For-Sale Unstable PTGER4 23 43 CCCCOCCOCc1ccccc1/C=C\C(=O)O ZINC000217880206 CG For-Sale Unstable PTGER3 21 48 CCCCOCCOCc1ccccc1/C=C\C(=O)O ZINC000217880206 CG For-Sale Unstable PLA2G4B 49 32 COc1ccc(C(=O)N[C@H]2CC(C)(C)Oc3cc(C)ccc32)cc1OC ZINC000217880213 FI In-Stock Unstable EZH2 41 35 Cc1cccc(/C=C/NC(=O)Nc2ccccc2Cl)c1 ZINC000217880223 CI For-Sale Unstable LPL 31 41 Cc1cccc(/C=C/NC(=O)Nc2ccccc2Cl)c1 ZINC000217880223 CI For-Sale Unstable CXCL8 43 35 Cc1cccc(/C=C/NC(=O)Nc2ccccc2Cl)c1 ZINC000217880223 CI For-Sale Unstable MMP1 0 53 Cc1cccc(/C=C/NC(=O)Nc2ccccc2Cl)c1 ZINC000217880223 CI For-Sale Unstable EPHB3 40 40 Cc1cccc(/C=C/NC(=O)Nc2ccccc2Cl)c1 ZINC000217880223 CI For-Sale Unstable LIPG 15 41 C[C@@H]1C[C@H](CN)CCN1C(=O)OCc1cc(Cl)cc(Cl)c1 ZINC000217880237 EH For-Sale Unstable CACNA1I 49 35 CN1CCCC[C@@H]1CNC(=O)c1ccc(SCCO)cc1 ZINC000217880244 DD In-Stock Unstable CACNA1I 41 35 COc1cccc([C@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c1 ZINC000217880249 KH In-Stock Unstable CYP1B1 45 36 COc1cccc([C@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c1 ZINC000217880249 KH In-Stock Unstable ABCB1 15 43 COc1cccc([C@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c1 ZINC000217880249 KH In-Stock Unstable RORC 0 45 CO[C@H]1CN[C@@H](C(=O)N[C@@H](C)Cc2ccc(F)cc2)C1 ZINC000217880254 CD For-Sale Unstable CTSC 25 42 C[C@@H](C(=O)O)c1ccc(CN2CCC[C@@H](O)C2)cc1 ZINC000217880270 CD For-Sale Unstable SLC6A1 68 34 C[C@@H](C(=O)O)c1ccc(CN2CCC[C@@H](O)C2)cc1 ZINC000217880270 CD For-Sale Unstable HRH3 21 41 C[C@@H](C(=O)O)c1ccc(CN2CCC[C@@H](O)C2)cc1 ZINC000217880270 CD For-Sale Unstable SIGMAR1 30 40 C[C@@H](C(=O)O)c1ccc(CN2CCC[C@@H](O)C2)cc1 ZINC000217880270 CD For-Sale Unstable CCR5 15 41 C[C@@H](C(=O)O)c1ccc(CN2CCC[C@@H](O)C2)cc1 ZINC000217880270 CD For-Sale Unstable MLNR 35 42 C[C@@H](C(=O)O)c1ccc(CN2CCC[C@@H](O)C2)cc1 ZINC000217880270 CD For-Sale Unstable SLC22A20 0 47 CCCCOCCOCc1ccc(/C=C\C(=O)O)cc1 ZINC000217880294 CG For-Sale Unstable PTGER2 26 40 CCCCOCCOCc1ccc(/C=C\C(=O)O)cc1 ZINC000217880294 CG For-Sale Unstable PLA2G4B 46 40 CCCCOCCOCc1ccc(/C=C\C(=O)O)cc1 ZINC000217880294 CG For-Sale Unstable AKR1C3 29 46 CCCCOCCOCc1ccc(/C=C\C(=O)O)cc1 ZINC000217880294 CG For-Sale Unstable AKR1B10 22 41 CCCCOCCOCc1ccc(/C=C\C(=O)O)cc1 ZINC000217880294 CG For-Sale Unstable TRPM2 0 41 COc1ccc2c(c1)[C@@H](NC(=O)c1ccc(OC)c(OC)c1)CC(C)(C)O2 ZINC000217880314 FH In-Stock Unstable MT-ND4 40 31 COc1ccc2c(c1)[C@@H](NC(=O)c1ccc(OC)c(OC)c1)CC(C)(C)O2 ZINC000217880314 FH In-Stock Unstable NAAA 18 46 C[C@@H](NS(=O)(=O)C[C@@]12CC[C@@H](CC1=O)C2(C)C)c1cc(F)c(Cl)cc1Cl ZINC000217880317 HJ On-Demand Unstable CA5B 27 46 C[C@@H](NS(=O)(=O)C[C@@]12CC[C@@H](CC1=O)C2(C)C)c1cc(F)c(Cl)cc1Cl ZINC000217880317 HJ On-Demand Unstable CA5A 30 46 Cc1cccc(/C=C/NC(=O)Nc2ccccc2C(C)C)c1 ZINC000217880328 CJ For-Sale Unstable TRPM8 22 52 Cc1cccc(/C=C/NC(=O)Nc2ccccc2C(C)C)c1 ZINC000217880328 CJ For-Sale Unstable ACAT 0 41 Cc1cccc(/C=C/NC(=O)Nc2ccccc2C(C)C)c1 ZINC000217880328 CJ For-Sale Unstable KCNK3 46 34 Cc1cccc(/C=C/NC(=O)Nc2ccccc2C(C)C)c1 ZINC000217880328 CJ For-Sale Unstable KCNK9 44 34 COc1cccc([C@@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c1 ZINC000217880332 KH In-Stock Unstable CYP1B1 45 36 COc1cccc([C@@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c1 ZINC000217880332 KH In-Stock Unstable ABCB1 15 43 COc1cccc([C@@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)c1 ZINC000217880332 KH In-Stock Unstable RORC 51 45 CO[C@H]1CN[C@H](C(=O)N[C@@H](C)Cc2ccc(F)cc2)C1 ZINC000217880336 CD For-Sale Unstable CTSC 25 42 C[C@H]1C[C@H](CN)CCN1C(=O)OCc1cc(Cl)cc(Cl)c1 ZINC000217880346 EH For-Sale Unstable CACNA1I 49 35 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](O)C2)cc1 ZINC000217880354 CD For-Sale Unstable SLC6A1 68 34 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](O)C2)cc1 ZINC000217880354 CD For-Sale Unstable HRH3 21 41 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](O)C2)cc1 ZINC000217880354 CD For-Sale Unstable SIGMAR1 30 40 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](O)C2)cc1 ZINC000217880354 CD For-Sale Unstable CCR5 15 41 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](O)C2)cc1 ZINC000217880354 CD For-Sale Unstable MLNR 35 42 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](O)C2)cc1 ZINC000217880354 CD For-Sale Unstable SLC22A20 0 47 CN1CCCC[C@H]1CNC(=O)c1ccc(SCCO)cc1 ZINC000217880356 DD In-Stock Unstable CACNA1I 41 35 C[C@H](NS(=O)(=O)C[C@@]12CC[C@@H](CC1=O)C2(C)C)c1cc(F)c(Cl)cc1Cl ZINC000217880357 HJ On-Demand Unstable CA5B 27 46 C[C@H](NS(=O)(=O)C[C@@]12CC[C@@H](CC1=O)C2(C)C)c1cc(F)c(Cl)cc1Cl ZINC000217880357 HJ On-Demand Unstable CA5A 30 46 COc1ccc2c(c1)[C@H](NC(=O)c1ccc(OC)c(OC)c1)CC(C)(C)O2 ZINC000217880404 FH In-Stock Unstable MT-ND4 40 31 COc1ccc2c(c1)[C@H](NC(=O)c1ccc(OC)c(OC)c1)CC(C)(C)O2 ZINC000217880404 FH In-Stock Unstable NAAA 18 46 CCN(C)C(=O)CNC(=O)c1ccc(Cl)cc1N ZINC000217880426 CD For-Sale Unstable PYGL 54 45 C[C@@H]1C[C@@H](CN)CCN1C(=O)OCc1cc(Cl)cc(Cl)c1 ZINC000217880435 EH For-Sale Unstable CACNA1I 49 35 COC(=O)c1ccnc(NCc2cnn(C)c2)c1 ZINC000217880464 BD On-Demand Unstable BDKRB1 26 41 COC(=O)c1ccnc(NCc2cnn(C)c2)c1 ZINC000217880464 BD On-Demand Unstable KDM3A 0 46 COC(=O)c1ccnc(NCc2cnn(C)c2)c1 ZINC000217880464 BD On-Demand Unstable KDM5C 0 46 C[C@H]1C[C@@H](CN)CCN1C(=O)OCc1cc(Cl)cc(Cl)c1 ZINC000217880525 EH For-Sale Unstable CACNA1I 49 35 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1ccc(OC)c(OC)c1 ZINC000217880550 FH In-Stock Unstable NAAA 22 46 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1ccc(OC)c(OC)c1 ZINC000217880550 FH In-Stock Unstable EZH2 40 35 CCCC[C@@H]1C[C@@H](O)CN1CC(C)C ZINC000217880554 AE In-Stock Unstable GBA2 41 32 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1N[C@@H](C)C1(C)CC1 ZINC000217880597 BI For-Sale Unstable TRPM8 0 42 COc1ccc(CCNC(=O)Cn2c(C)nc3cc(OC)c(OC)cc3c2=O)cc1OC ZINC000217880598 IE In-Stock Unstable F2 17 41 COc1ccc(CCNC(=O)Cn2c(C)nc3cc(OC)c(OC)cc3c2=O)cc1OC ZINC000217880598 IE In-Stock Unstable AVPR1B 43 36 COc1ccc(CCNC(=O)Cn2c(C)nc3cc(OC)c(OC)cc3c2=O)cc1OC ZINC000217880598 IE In-Stock Unstable ENPP1 55 31 CCCC[C@H]1C[C@@H](O)CN1CC(C)C ZINC000217880612 AE In-Stock Unstable GBA2 41 32 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1ccc(OC)c(OC)c1 ZINC000217880622 FH In-Stock Unstable NAAA 22 46 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1ccc(OC)c(OC)c1 ZINC000217880622 FH In-Stock Unstable EZH2 40 35 CCN1CCN(c2ccccc2NS(=O)(=O)c2ccc3c(c2)CC(=O)N3C)CC1 ZINC000217880649 HE On-Demand Unstable HTR1A 20 41 CCN1CCN(c2ccccc2NS(=O)(=O)c2ccc3c(c2)CC(=O)N3C)CC1 ZINC000217880649 HE On-Demand Unstable KCNQ2 57 31 CCN1CCN(c2ccccc2NS(=O)(=O)c2ccc3c(c2)CC(=O)N3C)CC1 ZINC000217880649 HE On-Demand Unstable HTR6 20 46 COc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1Cl ZINC000217880653 DI For-Sale Unstable KIT 16 45 COc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1Cl ZINC000217880653 DI For-Sale Unstable KDR 18 45 COc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1Cl ZINC000217880653 DI For-Sale Unstable IMPDH2 0 47 COc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1Cl ZINC000217880653 DI For-Sale Unstable KCNK3 63 40 COc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1Cl ZINC000217880653 DI For-Sale Unstable KCNK9 58 38 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1N[C@@H](C)C1(C)CC1 ZINC000217880672 BI For-Sale Unstable TRPM8 0 42 CCCC[C@@H]1C[C@H](O)CN1CC(C)C ZINC000217880690 AE In-Stock Unstable GBA2 41 32 CC[C@@H](NC(=O)c1ccc(OC)c(OC)c1)c1ccc(C)c(C)c1 ZINC000217880738 EI In-Stock Unstable PTGER3 23 42 CC[C@@H](NC(=O)c1ccc(OC)c(OC)c1)c1ccc(C)c(C)c1 ZINC000217880738 EI In-Stock Unstable ENPP1 48 34 CC[C@@H](NC(=O)c1ccc(OC)c(OC)c1)c1ccc(C)c(C)c1 ZINC000217880738 EI In-Stock Unstable UTS2 60 38 Cc1cccc(/C=C/NC(=O)Nc2cccc(C(F)(F)F)c2)c1 ZINC000217880741 DJ For-Sale Unstable KIT 27 42 Cc1cccc(/C=C/NC(=O)Nc2cccc(C(F)(F)F)c2)c1 ZINC000217880741 DJ For-Sale Unstable UL80 17 40 Cc1cccc(/C=C/NC(=O)Nc2cccc(C(F)(F)F)c2)c1 ZINC000217880741 DJ For-Sale Unstable KDR 25 42 Cc1cccc(/C=C/NC(=O)Nc2cccc(C(F)(F)F)c2)c1 ZINC000217880741 DJ For-Sale Unstable EPHX2 15 47 Cc1cccc(/C=C/NC(=O)Nc2cccc(C(F)(F)F)c2)c1 ZINC000217880741 DJ For-Sale Unstable TEK 31 42 Cc1cccc(/C=C/NC(=O)Nc2cccc(C(F)(F)F)c2)c1 ZINC000217880741 DJ For-Sale Unstable BTK 19 41 Cc1cccc(/C=C/NC(=O)Nc2cccc(C(F)(F)F)c2)c1 ZINC000217880741 DJ For-Sale Unstable RIPK1 47 39 Cc1cccc(/C=C/NC(=O)Nc2cccc(C(F)(F)F)c2)c1 ZINC000217880741 DJ For-Sale Unstable IMDH_CRYPV 46 36 Cc1cccc(/C=C/NC(=O)Nc2cccc(C(F)(F)F)c2)c1 ZINC000217880741 DJ For-Sale Unstable TRPM4 0 41 Cc1cccc(/C=C/NC(=O)Nc2cccc(C(F)(F)F)c2)c1 ZINC000217880741 DJ For-Sale Unstable KCNK3 69 53 Cc1cccc(/C=C/NC(=O)Nc2cccc(C(F)(F)F)c2)c1 ZINC000217880741 DJ For-Sale Unstable KCNK9 60 38 C[C@H](C(=O)O)c1ccc(CN(C)[C@@H]2CCC[C@@H](C)C2)cc1 ZINC000217880756 CH For-Sale Unstable PTGS1 28 53 CCN1CCN(c2ccccc2NS(=O)(=O)C[C@@]23CC[C@@H](CC2=O)C3(C)C)CC1 ZINC000217880767 HF On-Demand Unstable CA5B 31 54 CCN1CCN(c2ccccc2NS(=O)(=O)C[C@@]23CC[C@@H](CC2=O)C3(C)C)CC1 ZINC000217880767 HF On-Demand Unstable CA5A 33 54 CCN1CCN(c2ccccc2NS(=O)(=O)C[C@@]23CC[C@@H](CC2=O)C3(C)C)CC1 ZINC000217880767 HF On-Demand Unstable CXCR3 0 45 C[C@@H]1CCC[C@H](OCc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217880768 CH For-Sale Unstable PTGER2 22 41 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1N[C@@H](C)C1(C)CC1 ZINC000217880773 BI For-Sale Unstable TRPM8 0 42 CCCC[C@H]1C[C@H](O)CN1CC(C)C ZINC000217880780 AE In-Stock Unstable GBA2 41 32 CCC[C@@H](C)NC[C@@H](C)N1C[C@@H](C)Cc2ccccc21 ZINC000217880786 CH For-Sale Unstable TPP2 45 33 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)N1CCN(c3ccc(F)cc3)CC1)C(=O)OC2 ZINC000217880817 JI In-Stock Unstable IMPDH1 0 56 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)N1CCN(c3ccc(F)cc3)CC1)C(=O)OC2 ZINC000217880817 JI In-Stock Unstable IMPDH2 0 56 CC(C)[C@H]1CC[C@H](C)C[C@@H]1N[C@@H](C)C1(C)CC1 ZINC000217880837 BI For-Sale Unstable TRPM8 0 42 C[C@@H](Cc1ccc(F)cc1)NC(=O)[C@@H]1C[C@@H](O)CN1 ZINC000217880838 CC For-Sale Unstable CTSC 31 42 CCC[C@H](C)NC[C@@H](C)N1C[C@@H](C)Cc2ccccc21 ZINC000217880840 CH For-Sale Unstable TPP2 45 33 C[C@H]1CCC[C@H](OCc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217880848 CH For-Sale Unstable PTGER2 22 41 CC[C@H](NC(=O)c1ccc(OC)c(OC)c1)c1ccc(C)c(C)c1 ZINC000217880856 EI In-Stock Unstable PTGER3 23 42 CC[C@H](NC(=O)c1ccc(OC)c(OC)c1)c1ccc(C)c(C)c1 ZINC000217880856 EI In-Stock Unstable UTS2 60 38 CCCC[C@@H]1C[C@@H](O)CN1CCC(C)C ZINC000217880902 BF In-Stock Unstable GBA2 44 34 CCOC(=O)Cc1csc(NC(=O)[C@H](C)Nc2ccc3c(cc2=O)[C@@H](NC(C)=O)CCc2cc(OC)c(OC)c(OC)c2-3)n1 ZINC000217880925 KH In-Stock Unstable TUBA1A 16 58 CCOC(=O)Cc1csc(NC(=O)[C@H](C)Nc2ccc3c(cc2=O)[C@@H](NC(C)=O)CCc2cc(OC)c(OC)c(OC)c2-3)n1 ZINC000217880925 KH In-Stock Unstable TPPP 0 55 C[C@H](Cc1ccc(F)cc1)NC(=O)[C@@H]1C[C@@H](O)CN1 ZINC000217880936 CC For-Sale Unstable CTSC 31 42 O=C(O)/C=C\c1cc(CSc2ccccc2)ccc1F ZINC000217880941 CI For-Sale Unstable PTGER2 31 41 O=C(O)/C=C\c1cc(CSc2ccccc2)ccc1F ZINC000217880941 CI For-Sale Unstable PTGER4 0 44 O=C(O)/C=C\c1cc(CSc2ccccc2)ccc1F ZINC000217880941 CI For-Sale Unstable PTGER3 17 46 O=C(O)/C=C\c1cc(CSc2ccccc2)ccc1F ZINC000217880941 CI For-Sale Unstable PTGDR 0 46 CCC[C@@H](C)NC[C@H](C)N1C[C@@H](C)Cc2ccccc21 ZINC000217880942 CH For-Sale Unstable TPP2 45 33 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCc1ccc(Br)cc1F ZINC000217880950 EK For-Sale Unstable TRPM8 16 44 COC(=O)c1ccnc(NC[C@@H](C)CO)c1 ZINC000217880953 BC On-Demand Unstable KDM3A 0 48 COC(=O)c1ccnc(NC[C@@H](C)CO)c1 ZINC000217880953 BC On-Demand Unstable KDM5C 0 48 CCCC[C@H]1C[C@@H](O)CN1CCC(C)C ZINC000217880967 BF In-Stock Unstable GBA2 44 34 COc1ccccc1-c1ncc(CN2C[C@H]3[C@@H](C2)[C@@H]3C(=O)O)cn1 ZINC000217880984 ED In-Stock Unstable DRD4 25 41 COc1ccccc1-c1ncc(CN2C[C@H]3[C@@H](C2)[C@@H]3C(=O)O)cn1 ZINC000217880984 ED In-Stock Unstable DRD3 23 41 COc1ccccc1-c1ncc(CN2C[C@H]3[C@@H](C2)[C@@H]3C(=O)O)cn1 ZINC000217880984 ED In-Stock Unstable AGTR2 40 34 COc1ccccc1-c1ncc(CN2C[C@H]3[C@@H](C2)[C@@H]3C(=O)O)cn1 ZINC000217880984 ED In-Stock Unstable S1PR1 31 40 COc1ccccc1-c1ncc(CN2C[C@H]3[C@@H](C2)[C@@H]3C(=O)O)cn1 ZINC000217880984 ED In-Stock Unstable S1PR5 31 40 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)NC(C)C)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217881009 JF In-Stock Unstable TUBA1A 20 74 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)NC(C)C)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217881009 JF In-Stock Unstable SLC22A3 0 70 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)NC(C)C)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217881009 JF In-Stock Unstable TPPP 0 70 CCC[C@H](C)NC[C@H](C)N1C[C@@H](C)Cc2ccccc21 ZINC000217881019 CH For-Sale Unstable TPP2 45 33 C[C@@H](Cc1ccc(F)cc1)NC(=O)[C@H]1C[C@@H](O)CN1 ZINC000217881032 CC For-Sale Unstable CTSC 31 42 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCc1ccc(Br)cc1F ZINC000217881036 EK For-Sale Unstable TRPM8 15 44 COC(=O)c1ccnc(NC[C@H](C)CO)c1 ZINC000217881040 BC On-Demand Unstable KDM3A 0 48 COC(=O)c1ccnc(NC[C@H](C)CO)c1 ZINC000217881040 BC On-Demand Unstable KDM5C 0 48 CCCC[C@@H]1C[C@H](O)CN1CCC(C)C ZINC000217881046 BF In-Stock Unstable GBA2 44 34 COc1ccc(CNC(=O)NCCn2nc(-c3ccsc3)cc2C2CC2)cc1 ZINC000217881092 GH In-Stock Unstable NPBWR1 52 30 C[C@H](Cc1ccc(F)cc1)NC(=O)[C@H]1C[C@@H](O)CN1 ZINC000217881107 CC For-Sale Unstable CTSC 31 42 COc1ccc2ncc(C(=O)N3CCc4cc(OC)c(OC)cc4C3)c(O)c2c1 ZINC000217881114 GG In-Stock Unstable ABCB1B 59 35 COc1ccc2ncc(C(=O)N3CCc4cc(OC)c(OC)cc4C3)c(O)c2c1 ZINC000217881114 GG In-Stock Unstable ABCB1 24 51 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCc1ccc(Br)cc1F ZINC000217881117 EK For-Sale Unstable TRPM8 15 44 CCCC[C@H]1C[C@H](O)CN1CCC(C)C ZINC000217881134 BF In-Stock Unstable GBA2 44 34 CC[C@@H](NC(=O)CCCn1cncn1)c1nc(C)c[nH]1 ZINC000217881139 CD In-Stock Unstable HIS3 84 45 CC[C@@H]1COCCN1C[C@@H](O)COc1ccccc1C#N ZINC000217881140 CD On-Demand Unstable ADRB2 29 49 CC[C@@H]1COCCN1C[C@@H](O)COc1ccccc1C#N ZINC000217881140 CD On-Demand Unstable ADRB1 55 38 CC[C@@H]1COCCN1C[C@@H](O)COc1ccccc1C#N ZINC000217881140 CD On-Demand Unstable ADRB3 27 44 CC[C@@H]1COCCN1C[C@@H](O)COc1ccccc1C#N ZINC000217881140 CD On-Demand Unstable CASR 38 40 CC[C@@H]1COCCN1C[C@@H](O)COc1ccccc1C#N ZINC000217881140 CD On-Demand Unstable CYP2D6 15 40 CC[C@@H]1COCCN1C[C@@H](O)COc1ccccc1C#N ZINC000217881140 CD On-Demand Unstable ABCB1 41 38 CCOC(=O)CCCCC(=O)NC1CCN(C(=O)OCc2cc(Cl)cc(Cl)c2)CC1 ZINC000217881141 JI For-Sale Unstable EPHX2 24 47 CNC(=O)[C@@H]1CCCN1Cc1ccc([C@@H](C)C(=O)O)cc1 ZINC000217881149 CD For-Sale Unstable PTGS1 0 47 CNC(=O)[C@@H]1CCCN1Cc1ccc([C@@H](C)C(=O)O)cc1 ZINC000217881149 CD For-Sale Unstable HSD11B1 37 44 CNC(=O)[C@@H]1CCCN1Cc1ccc([C@@H](C)C(=O)O)cc1 ZINC000217881149 CD For-Sale Unstable LGMN 50 36 CNC(=O)[C@@H]1CCCN1Cc1ccc([C@@H](C)C(=O)O)cc1 ZINC000217881149 CD For-Sale Unstable XIAP 43 37 CNC(=O)[C@@H]1CCCN1Cc1ccc([C@@H](C)C(=O)O)cc1 ZINC000217881149 CD For-Sale Unstable BIRC8 40 32 Cc1cccc(/C=C/NC(=O)Nc2ccc(O)cc2)c1 ZINC000217881150 CG For-Sale Unstable MMP2 0 53 Cc1cccc(/C=C/NC(=O)Nc2ccc(O)cc2)c1 ZINC000217881150 CG For-Sale Unstable MMP9 0 53 Cc1cccc(/C=C/NC(=O)Nc2ccc(O)cc2)c1 ZINC000217881150 CG For-Sale Unstable MMP1 23 53 Cc1cccc(/C=C/NC(=O)Nc2ccc(O)cc2)c1 ZINC000217881150 CG For-Sale Unstable KCNK3 43 36 CC[C@@H](NC(=O)c1ccc(OC)c(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217881154 FH In-Stock Unstable PTGER3 16 43 CC[C@@H](NC(=O)c1ccc(OC)c(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217881154 FH In-Stock Unstable TACR3 41 38 CC[C@@H](NC(=O)c1ccc(OC)c(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217881154 FH In-Stock Unstable ABCG2 18 41 CC[C@@H](NC(=O)c1ccc(OC)c(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217881154 FH In-Stock Unstable ENPP1 57 34 CC[C@@H](NC(=O)c1ccc(OC)c(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217881154 FH In-Stock Unstable UTS2 67 41 CC(C)[C@@H](NC(=O)OCc1ccccc1F)C(=O)O ZINC000217881188 CE For-Sale Unstable ACE 31 45 CC(C)[C@@H](NC(=O)OCc1ccccc1F)C(=O)O ZINC000217881188 CE For-Sale Unstable CELA1 19 41 CC(C)[C@@H](NC(=O)OCc1ccccc1F)C(=O)O ZINC000217881188 CE For-Sale Unstable MME 63 45 CC(C)[C@@H](NC(=O)OCc1ccccc1F)C(=O)O ZINC000217881188 CE For-Sale Unstable CTRA_BOVIN 15 47 CC(C)[C@@H](NC(=O)OCc1ccccc1F)C(=O)O ZINC000217881188 CE For-Sale Unstable CASP3 38 68 CC(C)[C@@H](NC(=O)OCc1ccccc1F)C(=O)O ZINC000217881188 CE For-Sale Unstable BMP1 64 43 CC(C)[C@@H](NC(=O)OCc1ccccc1F)C(=O)O ZINC000217881188 CE For-Sale Unstable CASP8 16 50 CC(C)[C@@H](NC(=O)OCc1ccccc1F)C(=O)O ZINC000217881188 CE For-Sale Unstable KLK3 76 36 CC(C)[C@@H](NC(=O)OCc1ccccc1F)C(=O)O ZINC000217881188 CE For-Sale Unstable CTSB 58 49 CC(C)[C@@H](NC(=O)OCc1ccccc1F)C(=O)O ZINC000217881188 CE For-Sale Unstable PAPA1_CARPA 87 45 CC(C)[C@@H](NC(=O)OCc1ccccc1F)C(=O)O ZINC000217881188 CE For-Sale Unstable CYSP_TRYCR 56 37 CC(C)[C@@H](NC(=O)OCc1ccccc1F)C(=O)O ZINC000217881188 CE For-Sale Unstable CTSK 37 47 CC(C)[C@@H](NC(=O)OCc1ccccc1F)C(=O)O ZINC000217881188 CE For-Sale Unstable CTSL 39 47 CC(C)[C@@H](NC(=O)OCc1ccccc1F)C(=O)O ZINC000217881188 CE For-Sale Unstable CPA1 15 40 CC(C)[C@@H](NC(=O)OCc1ccccc1F)C(=O)O ZINC000217881188 CE For-Sale Unstable PGA 32 46 CC(C)[C@@H](NC(=O)OCc1ccccc1F)C(=O)O ZINC000217881188 CE For-Sale Unstable CAPNS1 64 38 CC(C)[C@@H](NC(=O)OCc1ccccc1F)C(=O)O ZINC000217881188 CE For-Sale Unstable ECE1 20 43 CC(C)[C@@H](NC(=O)OCc1ccccc1F)C(=O)O ZINC000217881188 CE For-Sale Unstable HLA-DRB1 74 37 CC(C)[C@@H](NC(=O)OCc1ccccc1F)C(=O)O ZINC000217881188 CE For-Sale Unstable CTSS 20 42 CC(C)[C@@H](NC(=O)OCc1ccccc1F)C(=O)O ZINC000217881188 CE For-Sale Unstable CAPN1 83 49 CC(C)[C@@H](NC(=O)OCc1ccccc1F)C(=O)O ZINC000217881188 CE For-Sale Unstable CASP1 36 50 CC(C)[C@@H](NC(=O)OCc1ccccc1F)C(=O)O ZINC000217881188 CE For-Sale Unstable CAPN2 116 49 CC(C)[C@@H](NC(=O)OCc1ccccc1F)C(=O)O ZINC000217881188 CE For-Sale Unstable ACE2 57 33 CC(C)[C@@H](NC(=O)OCc1ccccc1F)C(=O)O ZINC000217881188 CE For-Sale Unstable CASP6 38 50 CC(C)[C@@H](NC(=O)OCc1ccccc1F)C(=O)O ZINC000217881188 CE For-Sale Unstable CASP9 52 50 CC(C)[C@@H](NC(=O)OCc1ccccc1F)C(=O)O ZINC000217881188 CE For-Sale Unstable ADAMTS4 51 34 CC(C)[C@@H](NC(=O)OCc1ccccc1F)C(=O)O ZINC000217881188 CE For-Sale Unstable NPR 81 45 CC(C)[C@@H](NC(=O)OCc1ccccc1F)C(=O)O ZINC000217881188 CE For-Sale Unstable ADAM12 15 44 COc1cccc(SCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217881207 DI For-Sale Unstable PTGER2 28 40 COc1cccc(SCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217881207 DI For-Sale Unstable PTGER4 0 40 COc1cccc(SCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217881207 DI For-Sale Unstable CYP1B1 16 42 COc1cccc(SCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217881207 DI For-Sale Unstable LTB4R 36 52 COc1cccc(SCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217881207 DI For-Sale Unstable MTNR1A 32 49 COc1cccc(SCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217881207 DI For-Sale Unstable MTNR1B 39 49 COc1cccc(SCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217881207 DI For-Sale Unstable AKR1C3 42 50 COc1cccc(SCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217881207 DI For-Sale Unstable ABCG2 15 43 CC[C@H]1COCCN1C[C@@H](O)COc1ccccc1C#N ZINC000217881211 CD On-Demand Unstable ADRB2 29 49 CC[C@H]1COCCN1C[C@@H](O)COc1ccccc1C#N ZINC000217881211 CD On-Demand Unstable ADRB1 55 38 CC[C@H]1COCCN1C[C@@H](O)COc1ccccc1C#N ZINC000217881211 CD On-Demand Unstable ADRB3 27 44 CC[C@H]1COCCN1C[C@@H](O)COc1ccccc1C#N ZINC000217881211 CD On-Demand Unstable CASR 38 40 CC[C@H]1COCCN1C[C@@H](O)COc1ccccc1C#N ZINC000217881211 CD On-Demand Unstable CYP2D6 15 40 CC[C@H]1COCCN1C[C@@H](O)COc1ccccc1C#N ZINC000217881211 CD On-Demand Unstable ABCB1 41 38 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCc1ccc(Br)cc1F ZINC000217881217 EK For-Sale Unstable TRPM8 15 44 CC[C@H](NC(=O)CCCn1cncn1)c1nc(C)c[nH]1 ZINC000217881220 CD In-Stock Unstable HIS3 84 45 CC[C@H](NC(=O)c1ccc(OC)c(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217881230 FH In-Stock Unstable PTGER3 16 43 CC[C@H](NC(=O)c1ccc(OC)c(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217881230 FH In-Stock Unstable TACR3 41 38 CC[C@H](NC(=O)c1ccc(OC)c(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217881230 FH In-Stock Unstable ABCG2 18 41 CC[C@H](NC(=O)c1ccc(OC)c(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217881230 FH In-Stock Unstable ENPP1 57 34 CC[C@H](NC(=O)c1ccc(OC)c(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217881230 FH In-Stock Unstable UTS2 67 41 CCCC[C@@H]1C[C@@H](O)CN1CCOCC ZINC000217881235 BD In-Stock Unstable GBA2 44 33 COc1ccc(Cl)cc1NC(=O)N/C=C/c1cccc(C)c1 ZINC000217881246 DI For-Sale Unstable NR1H4 19 41 COc1ccc(Cl)cc1NC(=O)N/C=C/c1cccc(C)c1 ZINC000217881246 DI For-Sale Unstable KCNMA1 27 43 COc1ccc(Cl)cc1NC(=O)N/C=C/c1cccc(C)c1 ZINC000217881246 DI For-Sale Unstable RBP4 23 41 O=C(O)/C=C\c1ccccc1CSc1ccc(F)cc1 ZINC000217881282 CI For-Sale Unstable PTGER2 47 49 O=C(O)/C=C\c1ccccc1CSc1ccc(F)cc1 ZINC000217881282 CI For-Sale Unstable PTGER4 25 49 O=C(O)/C=C\c1ccccc1CSc1ccc(F)cc1 ZINC000217881282 CI For-Sale Unstable PTGER3 22 57 O=C(O)/C=C\c1ccccc1CSc1ccc(F)cc1 ZINC000217881282 CI For-Sale Unstable PTGDR 0 57 CCC[C@@H](C)NCCN1C[C@@H](C)Cc2ccccc21 ZINC000217881292 CG For-Sale Unstable TPP2 55 34 CS(=O)(=O)Nc1cccc2c1ccn2CC(=O)N1CCc2[nH]c3ccccc3c2C1 ZINC000217881301 HG In-Stock Unstable FABI 45 34 CCCC[C@H]1C[C@@H](O)CN1CCOCC ZINC000217881320 BD In-Stock Unstable GBA2 44 33 CC[C@@H](NC(=O)c1ccc(OC)c(OC)c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217881347 GF In-Stock Unstable PTGS2 16 40 CC[C@@H](NC(=O)c1ccc(OC)c(OC)c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217881347 GF In-Stock Unstable LOX1.1 44 41 CC[C@@H](NC(=O)c1ccc(OC)c(OC)c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217881347 GF In-Stock Unstable O49150_SOLTU 40 51 CC[C@@H](NC(=O)c1ccc(OC)c(OC)c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217881347 GF In-Stock Unstable UTS2 65 37 O=C(O)/C=C\c1ccc(CSc2ccc(F)cc2)cc1 ZINC000217881353 CI For-Sale Unstable AKR1C3 26 41 CCC[C@H](C)NCCN1C[C@@H](C)Cc2ccccc21 ZINC000217881356 CG For-Sale Unstable TPP2 55 34 COc1ccc([C@@H](C)N2CCCCC[C@@H]2C)c(O)c1 ZINC000217881375 CH For-Sale Unstable CHRM2 15 42 CCCC[C@@H]1C[C@H](O)CN1CCOCC ZINC000217881387 BD In-Stock Unstable GBA2 44 33 O=C(CC[C@@H]1NC(=O)c2ccccc2NC1=O)Nc1cccc(N2CCCCC2)c1 ZINC000217881417 HG In-Stock Unstable CASP3 0 40 O=C(CC[C@@H]1NC(=O)c2ccccc2NC1=O)Nc1cccc(N2CCCCC2)c1 ZINC000217881417 HG In-Stock Unstable CASP2 20 40 O=C(CC[C@@H]1NC(=O)c2ccccc2NC1=O)Nc1cccc(N2CCCCC2)c1 ZINC000217881417 HG In-Stock Unstable CASP8 0 40 O=C(CC[C@@H]1NC(=O)c2ccccc2NC1=O)Nc1cccc(N2CCCCC2)c1 ZINC000217881417 HG In-Stock Unstable CASP6 18 40 O=C(CC[C@@H]1NC(=O)c2ccccc2NC1=O)Nc1cccc(N2CCCCC2)c1 ZINC000217881417 HG In-Stock Unstable CASP7 0 40 CC[C@H](NC(=O)c1ccc(OC)c(OC)c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217881424 GF In-Stock Unstable PTGS2 16 40 CC[C@H](NC(=O)c1ccc(OC)c(OC)c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217881424 GF In-Stock Unstable LOX1.1 44 41 CC[C@H](NC(=O)c1ccc(OC)c(OC)c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217881424 GF In-Stock Unstable O49150_SOLTU 40 51 CC[C@H](NC(=O)c1ccc(OC)c(OC)c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217881424 GF In-Stock Unstable UTS2 65 37 COc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217881444 CH For-Sale Unstable KDR 29 41 COc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217881444 CH For-Sale Unstable MTNR1A 29 45 COc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217881444 CH For-Sale Unstable MTNR1B 30 45 COc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217881444 CH For-Sale Unstable CA12 18 42 COc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217881444 CH For-Sale Unstable PDGFRA 38 41 COc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217881444 CH For-Sale Unstable CA9 18 42 COc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217881444 CH For-Sale Unstable Q8MMZ8_EIMTE 23 43 COc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217881444 CH For-Sale Unstable AKR1C3 18 43 COc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217881444 CH For-Sale Unstable AKR1C2 47 43 COc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217881444 CH For-Sale Unstable IMDH_CRYPV 15 43 COc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217881444 CH For-Sale Unstable KCNK3 53 42 CCCC[C@H]1C[C@H](O)CN1CCOCC ZINC000217881473 BD In-Stock Unstable GBA2 44 33 O=C(O)/C=C\c1ccc(CSc2ccc(F)cc2F)cc1 ZINC000217881496 DI For-Sale Unstable AKR1C3 33 44 COC(=O)COc1ccccc1[C@@H](CC(=O)OC)c1c(O)c2ccccc2oc1=O ZINC000217881522 HF In-Stock Unstable NQO1 45 50 COC[C@H](O)CN(C)Cc1ccc([C@@H](C)C(=O)O)cc1 ZINC000217881530 CD For-Sale Unstable PTGS1 27 47 COC[C@H](O)CN(C)Cc1ccc([C@@H](C)C(=O)O)cc1 ZINC000217881530 CD For-Sale Unstable PTGS2 0 47 COc1ccc(-c2noc(CNC(=O)c3ccc(OC)c(OC)c3)n2)c(OC)c1 ZINC000217881536 GF In-Stock Unstable HRH3 15 44 COc1ccc(-c2noc(CNC(=O)c3ccc(OC)c(OC)c3)n2)c(OC)c1 ZINC000217881536 GF In-Stock Unstable SLC5A7 34 41 COc1ccc(-c2noc(CNC(=O)c3ccc(OC)c(OC)c3)n2)c(OC)c1 ZINC000217881536 GF In-Stock Unstable MT-ND1 25 44 COc1ccc(-c2noc(CNC(=O)c3ccc(OC)c(OC)c3)n2)c(OC)c1 ZINC000217881536 GF In-Stock Unstable ABCG2 27 44 C[C@H]1CCCCCN1[C@H](C)c1ccc(O)cc1 ZINC000217881560 BH For-Sale Unstable CHRM2 25 43 CCCC[C@@H]1C[C@@H](O)CN1CCOC ZINC000217881581 BD In-Stock Unstable GBA2 43 33 COC(=O)COc1ccccc1[C@H](CC(=O)OC)c1c(O)c2ccccc2oc1=O ZINC000217881600 HF In-Stock Unstable NQO1 45 50 O=C(O)/C=C\c1cccc(CSc2ccc(F)cc2F)c1 ZINC000217881612 DI For-Sale Unstable LTB4R 15 42 O=C(O)/C=C\c1cccc(CSc2ccc(F)cc2F)c1 ZINC000217881612 DI For-Sale Unstable HCAR2 0 41 O=C(O)/C=C\c1cccc(CSc2ccc(F)cc2F)c1 ZINC000217881612 DI For-Sale Unstable AKR1C3 35 48 C/C=C\C(=O)c1c(C(C)C)cc(C(C)C)cc1C(C)C ZINC000217881647 CK For-Sale Unstable FABP3 17 58 COc1cccc(-c2noc(CN(C)C(=O)c3ccc(OC)c(OC)c3)n2)c1 ZINC000217881649 GG In-Stock Unstable MT-ND1 24 42 COc1cccc(-c2noc(CN(C)C(=O)c3ccc(OC)c(OC)c3)n2)c1 ZINC000217881649 GG In-Stock Unstable HSD17B2 31 52 COc1cccc(-c2noc(CN(C)C(=O)c3ccc(OC)c(OC)c3)n2)c1 ZINC000217881649 GG In-Stock Unstable WNT3A 18 40 COc1cccc(-c2noc(CN(C)C(=O)c3ccc(OC)c(OC)c3)n2)c1 ZINC000217881649 GG In-Stock Unstable AXIN2 0 40 CN1CCO[C@@H]([C@@H](N)Cc2ccc(Cl)c(Cl)c2)C1 ZINC000217881651 CE For-Sale Unstable SIGMAR1 15 44 Cc1cccc(/C=C/NC(=O)NCCc2ccc(O)cc2)c1 ZINC000217881663 CG For-Sale Unstable STAT6 27 42 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC1C[C@@H]2CC[C@@H](C1)N2C ZINC000217881678 CH For-Sale Unstable TRPM8 0 41 CCCC[C@H]1C[C@@H](O)CN1CCOC ZINC000217881683 BD In-Stock Unstable GBA2 43 33 CCOC(=O)CSCc1cc(/C=C\C(=O)O)ccc1OC ZINC000217881690 DF For-Sale Unstable PTGER2 15 40 CCOC(=O)CSCc1cc(/C=C\C(=O)O)ccc1OC ZINC000217881690 DF For-Sale Unstable AKR1C3 41 43 Cc1cccc([C@@H]2CCCN(C(=O)c3cc(C)nc(N)n3)C2)c1 ZINC000217881694 DF In-Stock Unstable HPGD 15 40 CN1CCO[C@H]([C@@H](N)Cc2ccc(Cl)c(Cl)c2)C1 ZINC000217881719 CE For-Sale Unstable SIGMAR1 15 44 C[C@H]1CCCCCN1[C@H](C)Cc1ccc(O)cc1 ZINC000217881723 BH For-Sale Unstable OPRM1 21 42 C[C@H]1CCCCCN1[C@H](C)Cc1ccc(O)cc1 ZINC000217881723 BH For-Sale Unstable YARS 51 32 CC[C@@H]1COCCN1C[C@@H](O)COc1ccc(C#N)cc1 ZINC000217881727 CD On-Demand Unstable ABCB1 0 40 C/C=C/C(=O)c1c(C(C)C)cc(C(C)C)cc1C(C)C ZINC000217881728 CK For-Sale Unstable FABP3 17 58 COc1ccc(-c2noc(CN(C)C(=O)c3ccc(OC)c(OC)c3)n2)c(OC)c1 ZINC000217881748 HG In-Stock Unstable MT-ND1 25 44 Cc1cccc(/C=C/NC(=O)NC(C)C)c1 ZINC000217881759 BF For-Sale Unstable NR1H4 25 42 CCCC[C@@H]1C[C@H](O)CN1CCOC ZINC000217881772 BD In-Stock Unstable GBA2 43 33 CCOC(=O)CSCc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217881773 DF For-Sale Unstable PTGER2 34 42 CCOC(=O)CSCc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217881773 DF For-Sale Unstable PTGER4 19 42 CCOC(=O)CSCc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217881773 DF For-Sale Unstable PTGER3 15 42 CCOC(=O)CSCc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217881773 DF For-Sale Unstable LTB4R 38 42 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC1C[C@@H]2CC[C@@H](C1)N2C ZINC000217881776 CH For-Sale Unstable TRPM8 0 41 Cc1cccc([C@H]2CCCN(C(=O)c3cc(C)nc(N)n3)C2)c1 ZINC000217881777 DF In-Stock Unstable HPGD 15 40 Cc1c(Cl)cc(F)c(O)c1C[C@H](N)C(=O)O ZINC000217881787 BD For-Sale Unstable CACNA2D1 29 40 CC[C@H]1COCCN1C[C@@H](O)COc1ccc(C#N)cc1 ZINC000217881788 CD On-Demand Unstable ABCB1 0 40 C[C@H](C(=O)O)c1ccc(CN(C)[C@@H]2CCCC[C@@H]2C)cc1 ZINC000217881847 CH For-Sale Unstable PTGS1 28 51 Cc1cnc(SCc2cccc(/C=C\C(=O)O)c2)nc1 ZINC000217881848 CG For-Sale Unstable PTGER2 24 43 Cc1cnc(SCc2cccc(/C=C\C(=O)O)c2)nc1 ZINC000217881848 CG For-Sale Unstable LTB4R 19 44 Cc1cnc(SCc2cccc(/C=C\C(=O)O)c2)nc1 ZINC000217881848 CG For-Sale Unstable AKR1C3 32 40 CCCC[C@H]1C[C@H](O)CN1CCOC ZINC000217881850 BD In-Stock Unstable GBA2 43 33 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC1C[C@@H]2CC[C@@H](C1)N2C ZINC000217881852 CH For-Sale Unstable TRPM8 0 41 Cc1cccc(/C=C/NC(=O)N(Cc2ccccc2)C(C)C)c1 ZINC000217881863 DJ For-Sale Unstable NR1H4 36 40 Cc1cccc(/C=C/NC(=O)N(Cc2ccccc2)C(C)C)c1 ZINC000217881863 DJ For-Sale Unstable PTGES 23 46 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1OC ZINC000217881868 EI In-Stock Unstable DRD4 40 30 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1OC ZINC000217881868 EI In-Stock Unstable DRD3 26 42 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1OC ZINC000217881868 EI In-Stock Unstable SCNN1A 48 36 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1OC ZINC000217881868 EI In-Stock Unstable GCGR 21 46 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1OC ZINC000217881868 EI In-Stock Unstable TRPV1 22 51 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1OC ZINC000217881868 EI In-Stock Unstable SCN5A 0 44 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1OC ZINC000217881868 EI In-Stock Unstable MT-ND1 27 43 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1OC ZINC000217881868 EI In-Stock Unstable ABCG2 22 42 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1OC ZINC000217881868 EI In-Stock Unstable ADCYAP1R1 38 43 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1OC ZINC000217881868 EI In-Stock Unstable AP2S1 0 42 COc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1OC ZINC000217881868 EI In-Stock Unstable CAN2 0 43 Cc1c(Cl)cc(F)c(O)c1C[C@@H](N)C(=O)O ZINC000217881889 BD For-Sale Unstable CACNA2D1 29 40 CC[C@@H]1COCCN1C[C@@H](O)COc1cccc(C#N)c1 ZINC000217881893 CD For-Sale Unstable ABCB1 0 42 CC[C@@H]1COCCN1C[C@@H](O)COc1cccc(C#N)c1 ZINC000217881893 CD For-Sale Unstable CHRNA10 29 44 CSCC[C@@H](CO)NC(=O)[C@H](Cc1ccccc1)N1Cc2ccccc2C1=O ZINC000217881905 GE In-Stock Unstable ACE 22 43 CSCC[C@@H](CO)NC(=O)[C@H](Cc1ccccc1)N1Cc2ccccc2C1=O ZINC000217881905 GE In-Stock Unstable MME 45 43 CSCC[C@@H](CO)NC(=O)[C@H](Cc1ccccc1)N1Cc2ccccc2C1=O ZINC000217881905 GE In-Stock Unstable TACR2 31 40 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC1C[C@@H]2CC[C@@H](C1)N2C ZINC000217881922 CH For-Sale Unstable TRPM8 0 41 C[C@H]1CCCCCN1[C@H](C)CCc1ccc(O)cc1 ZINC000217881941 CH For-Sale Unstable HRH3 24 42 CC[C@H]1COCCN1C[C@@H](O)COc1cccc(C#N)c1 ZINC000217881957 CD For-Sale Unstable CHRNA10 29 44 CNC1CCN(C(=O)OCc2cc(Cl)cc(Cl)c2)CC1 ZINC000217881991 DG For-Sale Unstable GRIN2B 20 42 CNC1CCN(C(=O)OCc2cc(Cl)cc(Cl)c2)CC1 ZINC000217881991 DG For-Sale Unstable EPHX2 16 46 CNC1CCN(C(=O)OCc2cc(Cl)cc(Cl)c2)CC1 ZINC000217881991 DG For-Sale Unstable CACNA1I 52 36 CNC1CCN(C(=O)OCc2cc(Cl)cc(Cl)c2)CC1 ZINC000217881991 DG For-Sale Unstable F13A1 40 41 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1OC ZINC000217881993 FG In-Stock Unstable HTR1A 50 52 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1OC ZINC000217881993 FG In-Stock Unstable ADRA2A 16 52 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1OC ZINC000217881993 FG In-Stock Unstable DRD2 58 50 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1OC ZINC000217881993 FG In-Stock Unstable DRD1 31 50 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1OC ZINC000217881993 FG In-Stock Unstable DRD4 51 42 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1OC ZINC000217881993 FG In-Stock Unstable ADRA1D 39 49 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1OC ZINC000217881993 FG In-Stock Unstable HTR2A 40 50 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1OC ZINC000217881993 FG In-Stock Unstable HTR2C 30 50 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1OC ZINC000217881993 FG In-Stock Unstable AVPR2 37 43 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1OC ZINC000217881993 FG In-Stock Unstable ADRA1A 39 41 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1OC ZINC000217881993 FG In-Stock Unstable ADRA1B 23 49 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1OC ZINC000217881993 FG In-Stock Unstable DRD3 75 50 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1OC ZINC000217881993 FG In-Stock Unstable CPT1A 45 32 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1OC ZINC000217881993 FG In-Stock Unstable SLC9A1 53 33 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1OC ZINC000217881993 FG In-Stock Unstable ABCB1 15 40 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1OC ZINC000217881993 FG In-Stock Unstable PLD2 30 40 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1OC ZINC000217881993 FG In-Stock Unstable TYRO3 30 44 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1OC ZINC000217881993 FG In-Stock Unstable ABCG2 35 40 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1OC ZINC000217881993 FG In-Stock Unstable AP2S1 0 45 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1OC ZINC000217881993 FG In-Stock Unstable ALPHA-1A 0 47 COc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1OC ZINC000217881993 FG In-Stock Unstable ACKR3 56 37 C#CCOc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OC ZINC000217881994 KH In-Stock Unstable ALOX5 0 42 C#CCOc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OC ZINC000217881994 KH In-Stock Unstable CYP1B1 46 39 C#CCOc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OC ZINC000217881994 KH In-Stock Unstable CYP1A1 46 39 C#CCOc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OC ZINC000217881994 KH In-Stock Unstable ABCB1A 22 41 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1N[C@@H](C)c1cc(O)ccc1O ZINC000217882037 CI For-Sale Unstable TRPM8 17 47 C#CCOc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OC ZINC000217882074 KH In-Stock Unstable ALOX5 0 42 C#CCOc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OC ZINC000217882074 KH In-Stock Unstable CYP1B1 46 39 C#CCOc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OC ZINC000217882074 KH In-Stock Unstable CYP1A1 46 39 C#CCOc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)ccc1OC ZINC000217882074 KH In-Stock Unstable ABCB1A 22 41 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1N[C@@H](C)c1cc(O)ccc1O ZINC000217882123 CI For-Sale Unstable TRPM8 17 47 O=C(O)/C=C\c1ccc(COc2cccc(F)c2)cc1 ZINC000217882126 CH For-Sale Unstable MAOB 33 54 O=C(O)/C=C\c1ccc(COc2cccc(F)c2)cc1 ZINC000217882126 CH For-Sale Unstable PTGER2 16 53 O=C(O)/C=C\c1ccc(COc2cccc(F)c2)cc1 ZINC000217882126 CH For-Sale Unstable F10 0 44 O=C(O)/C=C\c1ccc(COc2cccc(F)c2)cc1 ZINC000217882126 CH For-Sale Unstable PTGER4 23 53 O=C(O)/C=C\c1ccc(COc2cccc(F)c2)cc1 ZINC000217882126 CH For-Sale Unstable PTPN2 0 43 O=C(O)/C=C\c1ccc(COc2cccc(F)c2)cc1 ZINC000217882126 CH For-Sale Unstable PTGER3 25 53 O=C(O)/C=C\c1ccc(COc2cccc(F)c2)cc1 ZINC000217882126 CH For-Sale Unstable LTB4R 18 40 O=C(O)/C=C\c1ccc(COc2cccc(F)c2)cc1 ZINC000217882126 CH For-Sale Unstable CDC25B 23 43 O=C(O)/C=C\c1ccc(COc2cccc(F)c2)cc1 ZINC000217882126 CH For-Sale Unstable PTGDR 0 48 O=C(O)/C=C\c1ccc(COc2cccc(F)c2)cc1 ZINC000217882126 CH For-Sale Unstable HCAR2 0 48 O=C(O)/C=C\c1ccc(COc2cccc(F)c2)cc1 ZINC000217882126 CH For-Sale Unstable FFAR1 39 43 O=C(O)/C=C\c1ccc(COc2cccc(F)c2)cc1 ZINC000217882126 CH For-Sale Unstable AKR1C3 38 53 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccccc2)c1 ZINC000217882127 CH In-Stock Unstable ANPEP 29 47 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccccc2)c1 ZINC000217882127 CH In-Stock Unstable HDAC8 65 38 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccccc2)c1 ZINC000217882127 CH In-Stock Unstable MMP2 23 64 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccccc2)c1 ZINC000217882127 CH In-Stock Unstable HDAC1 31 40 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccccc2)c1 ZINC000217882127 CH In-Stock Unstable HDAC2 21 43 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccccc2)c1 ZINC000217882127 CH In-Stock Unstable HDAC6 50 43 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccccc2)c1 ZINC000217882127 CH In-Stock Unstable MMP9 21 64 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccccc2)c1 ZINC000217882127 CH In-Stock Unstable MMP1 0 40 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccccc2)c1 ZINC000217882127 CH In-Stock Unstable AMP1_PLAFQ 60 42 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccccc2)c1 ZINC000217882127 CH In-Stock Unstable 17HSDCL 0 41 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccccc2)c1 ZINC000217882127 CH In-Stock Unstable AKR1C3 0 42 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccccc2)c1 ZINC000217882127 CH In-Stock Unstable PDS 70 38 COc1ccc2[nH]cc(CCNC(=O)[C@@H](NC(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)C(C)C)c2c1 ZINC000217882200 KF In-Stock Unstable NQO2 24 46 COc1ccc2[nH]cc(CCNC(=O)[C@@H](NC(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)C(C)C)c2c1 ZINC000217882200 KF In-Stock Unstable MTNR1A 57 47 COc1ccc2[nH]cc(CCNC(=O)[C@@H](NC(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)C(C)C)c2c1 ZINC000217882200 KF In-Stock Unstable MTNR1B 40 46 COc1ccc2[nH]cc(CCNC(=O)[C@@H](NC(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)C(C)C)c2c1 ZINC000217882200 KF In-Stock Unstable ABCG2 25 41 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1N[C@@H](C)c1cc(O)ccc1O ZINC000217882208 CI For-Sale Unstable TRPM8 17 47 O=C(O)/C=C\c1ccc(COc2cccc(F)c2)c(F)c1 ZINC000217882218 CH For-Sale Unstable PTGER2 35 42 O=C(O)/C=C\c1ccc(COc2cccc(F)c2)c(F)c1 ZINC000217882218 CH For-Sale Unstable PTGER4 22 42 O=C(O)/C=C\c1ccc(COc2cccc(F)c2)c(F)c1 ZINC000217882218 CH For-Sale Unstable PTGER3 15 42 O=C(O)/C=C\c1ccc(COc2cccc(F)c2)c(F)c1 ZINC000217882218 CH For-Sale Unstable CDC25B 24 48 O=C(O)/C=C\c1ccc(COc2cccc(F)c2)c(F)c1 ZINC000217882218 CH For-Sale Unstable HCAR2 0 42 O=C(O)/C=C\c1ccc(COc2cccc(F)c2)c(F)c1 ZINC000217882218 CH For-Sale Unstable AKR1C3 34 48 CCOc1ccc(CNC(=O)/C=C/c2ccccc2)cc1OCC ZINC000217882233 EH In-Stock Unstable BDKRB2 45 33 CCOc1ccc(CNC(=O)/C=C/c2ccccc2)cc1OCC ZINC000217882233 EH In-Stock Unstable HDAC8 52 39 CCOc1ccc(CNC(=O)/C=C/c2ccccc2)cc1OCC ZINC000217882233 EH In-Stock Unstable MMP2 20 60 CCOc1ccc(CNC(=O)/C=C/c2ccccc2)cc1OCC ZINC000217882233 EH In-Stock Unstable HDAC2 16 43 CCOc1ccc(CNC(=O)/C=C/c2ccccc2)cc1OCC ZINC000217882233 EH In-Stock Unstable HDAC6 42 43 CCOc1ccc(CNC(=O)/C=C/c2ccccc2)cc1OCC ZINC000217882233 EH In-Stock Unstable MMP9 17 60 CCOc1ccc(CNC(=O)/C=C/c2ccccc2)cc1OCC ZINC000217882233 EH In-Stock Unstable AKR1C3 28 47 CCOc1ccc(CNC(=O)/C=C/c2ccccc2)cc1OCC ZINC000217882233 EH In-Stock Unstable PDS 42 34 Cc1ccc2c(c1)c(=O)c(C(=O)N(C)Cc1nnc(C)o1)cn2C ZINC000217882234 ED In-Stock Unstable UL54 57 30 COc1cc([C@@H](C)N2CCCCC[C@@H]2C)ccc1O ZINC000217882259 CH For-Sale Unstable CHRM2 16 42 C[C@H](C(=O)O)c1ccc(CN2CCO[C@@H]3CCC[C@@H]32)cc1 ZINC000217882289 CF For-Sale Unstable PTGS1 23 50 CC(C)[C@H]1CC[C@H](C)C[C@@H]1N[C@@H](C)c1cc(O)ccc1O ZINC000217882291 CI For-Sale Unstable TRPM8 17 47 O=C(O)/C=C\c1cccc(COc2cccc(F)c2)c1 ZINC000217882300 CH For-Sale Unstable MAOA 15 42 O=C(O)/C=C\c1cccc(COc2cccc(F)c2)c1 ZINC000217882300 CH For-Sale Unstable MAOB 58 49 O=C(O)/C=C\c1cccc(COc2cccc(F)c2)c1 ZINC000217882300 CH For-Sale Unstable PTGER2 16 53 O=C(O)/C=C\c1cccc(COc2cccc(F)c2)c1 ZINC000217882300 CH For-Sale Unstable PTGER4 23 53 O=C(O)/C=C\c1cccc(COc2cccc(F)c2)c1 ZINC000217882300 CH For-Sale Unstable PTGER3 24 53 O=C(O)/C=C\c1cccc(COc2cccc(F)c2)c1 ZINC000217882300 CH For-Sale Unstable LTB4R 15 43 O=C(O)/C=C\c1cccc(COc2cccc(F)c2)c1 ZINC000217882300 CH For-Sale Unstable CDC25B 0 45 O=C(O)/C=C\c1cccc(COc2cccc(F)c2)c1 ZINC000217882300 CH For-Sale Unstable NR1H4 41 36 O=C(O)/C=C\c1cccc(COc2cccc(F)c2)c1 ZINC000217882300 CH For-Sale Unstable GYS1 44 32 O=C(O)/C=C\c1cccc(COc2cccc(F)c2)c1 ZINC000217882300 CH For-Sale Unstable PTGDR 0 45 O=C(O)/C=C\c1cccc(COc2cccc(F)c2)c1 ZINC000217882300 CH For-Sale Unstable HCAR2 0 54 O=C(O)/C=C\c1cccc(COc2cccc(F)c2)c1 ZINC000217882300 CH For-Sale Unstable FFAR1 52 43 O=C(O)/C=C\c1cccc(COc2cccc(F)c2)c1 ZINC000217882300 CH For-Sale Unstable AKR1C3 39 58 O=C(O)/C=C\c1cccc(COc2cccc(F)c2)c1 ZINC000217882300 CH For-Sale Unstable PDS 33 41 CCCC[C@@H]1C[C@@H](O)CN1CCF ZINC000217882330 AD In-Stock Unstable GBA2 41 32 COc1cc(CNC(=O)/C=C/c2ccccc2)ccc1OC(C)C ZINC000217882337 EH In-Stock Unstable TRPV1 23 45 COc1cc(CNC(=O)/C=C/c2ccccc2)ccc1OC(C)C ZINC000217882337 EH In-Stock Unstable HDAC8 46 45 COc1cc(CNC(=O)/C=C/c2ccccc2)ccc1OC(C)C ZINC000217882337 EH In-Stock Unstable MMP2 18 55 COc1cc(CNC(=O)/C=C/c2ccccc2)ccc1OC(C)C ZINC000217882337 EH In-Stock Unstable HDAC6 33 40 COc1cc(CNC(=O)/C=C/c2ccccc2)ccc1OC(C)C ZINC000217882337 EH In-Stock Unstable MMP9 15 55 COc1cc(CNC(=O)/C=C/c2ccccc2)ccc1OC(C)C ZINC000217882337 EH In-Stock Unstable AKR1C3 25 44 CCOc1ccccc1C(=O)N1C[C@H](Oc2ccccc2F)C[C@@H]1C(=O)OC ZINC000217882347 GG For-Sale Unstable HCRTR1 58 39 CCOc1ccccc1C(=O)N1C[C@H](Oc2ccccc2F)C[C@@H]1C(=O)OC ZINC000217882347 GG For-Sale Unstable HCRTR2 64 39 CCOc1ccccc1C(=O)N1C[C@H](Oc2ccccc2F)C[C@@H]1C(=O)OC ZINC000217882347 GG For-Sale Unstable HCN1 51 33 CCOc1ccccc1C(=O)N1C[C@H](Oc2ccccc2F)C[C@@H]1C(=O)OC ZINC000217882347 GG For-Sale Unstable HCN4 43 33 C[C@H]1CCCCCN1[C@H](C)c1ccc2ccccc2c1O ZINC000217882370 CJ For-Sale Unstable HRH3 16 40 CCCC[C@H]1C[C@@H](O)CN1CCF ZINC000217882381 AD In-Stock Unstable GBA2 41 32 CCOc1ccccc1C(=O)N1C[C@@H](Oc2ccccc2F)C[C@@H]1C(=O)OC ZINC000217882421 GG For-Sale Unstable HCRTR1 58 39 CCOc1ccccc1C(=O)N1C[C@@H](Oc2ccccc2F)C[C@@H]1C(=O)OC ZINC000217882421 GG For-Sale Unstable HCRTR2 64 39 CCOc1ccccc1C(=O)N1C[C@@H](Oc2ccccc2F)C[C@@H]1C(=O)OC ZINC000217882421 GG For-Sale Unstable HCN1 51 33 CCOc1ccccc1C(=O)N1C[C@@H](Oc2ccccc2F)C[C@@H]1C(=O)OC ZINC000217882421 GG For-Sale Unstable HCN4 43 33 Cc1cccc(/C=C/NC(=O)NC2CCCCC2)c1 ZINC000217882431 CH For-Sale Unstable FAAH 20 52 Cc1cccc(/C=C/NC(=O)NC2CCCCC2)c1 ZINC000217882431 CH For-Sale Unstable EPHX2 29 45 O=C(/C=C/c1ccccc1)NCCCc1ccccc1Cl ZINC000217882433 CI In-Stock Unstable DRD3 15 43 O=C(/C=C/c1ccccc1)NCCCc1ccccc1Cl ZINC000217882433 CI In-Stock Unstable PYGL 28 53 O=C(/C=C/c1ccccc1)NCCCc1ccccc1Cl ZINC000217882433 CI In-Stock Unstable HDAC8 41 35 O=C(/C=C/c1ccccc1)NCCCc1ccccc1Cl ZINC000217882433 CI In-Stock Unstable MMP2 21 60 O=C(/C=C/c1ccccc1)NCCCc1ccccc1Cl ZINC000217882433 CI In-Stock Unstable HDAC1 29 45 O=C(/C=C/c1ccccc1)NCCCc1ccccc1Cl ZINC000217882433 CI In-Stock Unstable HDAC2 24 45 O=C(/C=C/c1ccccc1)NCCCc1ccccc1Cl ZINC000217882433 CI In-Stock Unstable HDAC3 15 45 O=C(/C=C/c1ccccc1)NCCCc1ccccc1Cl ZINC000217882433 CI In-Stock Unstable HDAC4 22 45 O=C(/C=C/c1ccccc1)NCCCc1ccccc1Cl ZINC000217882433 CI In-Stock Unstable HDAC6 32 48 O=C(/C=C/c1ccccc1)NCCCc1ccccc1Cl ZINC000217882433 CI In-Stock Unstable MMP9 18 60 O=C(/C=C/c1ccccc1)NCCCc1ccccc1Cl ZINC000217882433 CI In-Stock Unstable HDAC9 43 45 O=C(/C=C/c1ccccc1)NCCCc1ccccc1Cl ZINC000217882433 CI In-Stock Unstable HDAC7 54 45 O=C(/C=C/c1ccccc1)NCCCc1ccccc1Cl ZINC000217882433 CI In-Stock Unstable MMP1 0 52 O=C(/C=C/c1ccccc1)NCCCc1ccccc1Cl ZINC000217882433 CI In-Stock Unstable IMA1 0 41 CCOC(=O)Cc1csc(NC(=O)CNc2ccc3c(cc2=O)[C@@H](NC(C)=O)CCc2cc(OC)c(OC)c(OC)c2-3)n1 ZINC000217882441 KG In-Stock Unstable TUBA1A 16 59 CCOC(=O)Cc1csc(NC(=O)CNc2ccc3c(cc2=O)[C@@H](NC(C)=O)CCc2cc(OC)c(OC)c(OC)c2-3)n1 ZINC000217882441 KG In-Stock Unstable TPPP 0 56 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCc1ccc(F)c(Br)c1 ZINC000217882450 EK For-Sale Unstable TRPM8 16 44 CNCCCN1CCN(C(=O)OCc2cc(Cl)cc(Cl)c2)CC1 ZINC000217882458 FF For-Sale Unstable HRP1_PLAFA 45 37 CCCC[C@@H]1C[C@H](O)CN1CCF ZINC000217882484 AD In-Stock Unstable GBA2 41 32 COc1ccc(CC[C@@H](C)N[C@@H]2CCC[C@@H](C)[C@@H]2C)cc1 ZINC000217882495 CI For-Sale Unstable SLC18A2 27 42 CCOc1ccccc1C(=O)N1C[C@H](Oc2ccccc2F)C[C@H]1C(=O)OC ZINC000217882503 GG For-Sale Unstable HCRTR1 58 39 CCOc1ccccc1C(=O)N1C[C@H](Oc2ccccc2F)C[C@H]1C(=O)OC ZINC000217882503 GG For-Sale Unstable HCRTR2 64 39 CCOc1ccccc1C(=O)N1C[C@H](Oc2ccccc2F)C[C@H]1C(=O)OC ZINC000217882503 GG For-Sale Unstable HCN1 51 33 CCOc1ccccc1C(=O)N1C[C@H](Oc2ccccc2F)C[C@H]1C(=O)OC ZINC000217882503 GG For-Sale Unstable HCN4 43 33 O=C(/C=C/c1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217882527 CI In-Stock Unstable MAOB 0 46 O=C(/C=C/c1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217882527 CI In-Stock Unstable SDH1 0 47 O=C(/C=C/c1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217882527 CI In-Stock Unstable PYGL 26 50 O=C(/C=C/c1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217882527 CI In-Stock Unstable HDAC8 46 39 O=C(/C=C/c1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217882527 CI In-Stock Unstable HDAC1 38 45 O=C(/C=C/c1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217882527 CI In-Stock Unstable HDAC2 25 45 O=C(/C=C/c1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217882527 CI In-Stock Unstable HDAC3 19 45 O=C(/C=C/c1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217882527 CI In-Stock Unstable HDAC4 28 45 O=C(/C=C/c1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217882527 CI In-Stock Unstable HDAC6 34 48 O=C(/C=C/c1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217882527 CI In-Stock Unstable SCN5A 0 45 O=C(/C=C/c1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217882527 CI In-Stock Unstable SLC6A5 28 41 O=C(/C=C/c1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217882527 CI In-Stock Unstable MMP9 19 68 O=C(/C=C/c1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217882527 CI In-Stock Unstable HDAC9 45 45 O=C(/C=C/c1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217882527 CI In-Stock Unstable HDAC7 57 45 O=C(/C=C/c1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217882527 CI In-Stock Unstable MMP1 25 56 O=C(/C=C/c1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217882527 CI In-Stock Unstable AMP1_PLAFQ 39 42 O=C(/C=C/c1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217882527 CI In-Stock Unstable CRTM 43 41 O=C(/C=C/c1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217882527 CI In-Stock Unstable IMA1 0 41 O=C(/C=C/c1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217882527 CI In-Stock Unstable TRPM2 0 45 C[C@H](C(=O)O)c1ccc(CN2C[C@@H](C)OC(C)(C)C2)cc1 ZINC000217882533 CF For-Sale Unstable PTGS1 22 43 C[C@H](C(=O)O)c1ccc(CN2C[C@@H](C)OC(C)(C)C2)cc1 ZINC000217882533 CF For-Sale Unstable PTGS2 0 43 CCCC[C@H]1C[C@H](O)CN1CCF ZINC000217882545 AD In-Stock Unstable GBA2 41 32 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCc1ccc(F)c(Br)c1 ZINC000217882551 EK For-Sale Unstable TRPM8 16 44 COc1ccc(CC[C@H](C)N[C@@H]2CCC[C@@H](C)[C@@H]2C)cc1 ZINC000217882559 CI For-Sale Unstable SLC18A2 27 42 Clc1cccc2[nH]cc(C3=CCN(Cc4ccccc4)CC3)c12 ZINC000217882586 DK For-Sale Unstable DRD2 18 51 Clc1cccc2[nH]cc(C3=CCN(Cc4ccccc4)CC3)c12 ZINC000217882586 DK For-Sale Unstable DRD4 16 51 Clc1cccc2[nH]cc(C3=CCN(Cc4ccccc4)CC3)c12 ZINC000217882586 DK For-Sale Unstable SLC6A4 16 46 CCOc1ccccc1C(=O)N1C[C@@H](Oc2ccccc2F)C[C@H]1C(=O)OC ZINC000217882594 GG For-Sale Unstable HCRTR1 58 39 CCOc1ccccc1C(=O)N1C[C@@H](Oc2ccccc2F)C[C@H]1C(=O)OC ZINC000217882594 GG For-Sale Unstable HCRTR2 64 39 CCOc1ccccc1C(=O)N1C[C@@H](Oc2ccccc2F)C[C@H]1C(=O)OC ZINC000217882594 GG For-Sale Unstable HCN1 51 33 CCOc1ccccc1C(=O)N1C[C@@H](Oc2ccccc2F)C[C@H]1C(=O)OC ZINC000217882594 GG For-Sale Unstable HCN4 43 33 CC[C@@H]1CCCC[C@@H]1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217882599 CI For-Sale Unstable PTGER2 23 41 CC[C@@H]1CCCC[C@@H]1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217882599 CI For-Sale Unstable HCAR2 0 40 C[C@H]1CCCCCN1[C@H](C)c1cccc(O)c1 ZINC000217882605 BH For-Sale Unstable OPRM1 15 43 Cc1cccc(/C=C/NC(=O)N2CCC(C(=O)O)CC2)c1 ZINC000217882633 CE For-Sale Unstable EPHX2 21 41 O=C(/C=C/c1ccccc1)NCCCc1ccc(F)cc1 ZINC000217882634 CH In-Stock Unstable NA 0 43 O=C(/C=C/c1ccccc1)NCCCc1ccc(F)cc1 ZINC000217882634 CH In-Stock Unstable DRD3 15 48 O=C(/C=C/c1ccccc1)NCCCc1ccc(F)cc1 ZINC000217882634 CH In-Stock Unstable F2R 22 42 O=C(/C=C/c1ccccc1)NCCCc1ccc(F)cc1 ZINC000217882634 CH In-Stock Unstable PYGL 22 44 O=C(/C=C/c1ccccc1)NCCCc1ccc(F)cc1 ZINC000217882634 CH In-Stock Unstable HDAC8 45 39 O=C(/C=C/c1ccccc1)NCCCc1ccc(F)cc1 ZINC000217882634 CH In-Stock Unstable MMP2 22 68 O=C(/C=C/c1ccccc1)NCCCc1ccc(F)cc1 ZINC000217882634 CH In-Stock Unstable HDAC1 26 45 O=C(/C=C/c1ccccc1)NCCCc1ccc(F)cc1 ZINC000217882634 CH In-Stock Unstable HDAC2 22 45 O=C(/C=C/c1ccccc1)NCCCc1ccc(F)cc1 ZINC000217882634 CH In-Stock Unstable HDAC3 17 45 O=C(/C=C/c1ccccc1)NCCCc1ccc(F)cc1 ZINC000217882634 CH In-Stock Unstable HDAC4 28 45 O=C(/C=C/c1ccccc1)NCCCc1ccc(F)cc1 ZINC000217882634 CH In-Stock Unstable HDAC6 35 48 O=C(/C=C/c1ccccc1)NCCCc1ccc(F)cc1 ZINC000217882634 CH In-Stock Unstable MMP9 19 68 O=C(/C=C/c1ccccc1)NCCCc1ccc(F)cc1 ZINC000217882634 CH In-Stock Unstable HDAC9 45 45 O=C(/C=C/c1ccccc1)NCCCc1ccc(F)cc1 ZINC000217882634 CH In-Stock Unstable HDAC7 57 45 O=C(/C=C/c1ccccc1)NCCCc1ccc(F)cc1 ZINC000217882634 CH In-Stock Unstable MMP1 0 56 O=C(/C=C/c1ccccc1)NCCCc1ccc(F)cc1 ZINC000217882634 CH In-Stock Unstable AMP1_PLAFQ 29 45 O=C(/C=C/c1ccccc1)NCCCc1ccc(F)cc1 ZINC000217882634 CH In-Stock Unstable CRTM 31 41 COc1ccc(CC[C@@H](C)N[C@H]2CCC[C@@H](C)[C@@H]2C)cc1 ZINC000217882644 CI For-Sale Unstable SLC18A2 27 42 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCc1ccc(F)c(Br)c1 ZINC000217882657 EK For-Sale Unstable TRPM8 16 44 CC[C@H]1CCCC[C@@H]1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217882706 CI For-Sale Unstable PTGER2 23 41 CC[C@H]1CCCC[C@@H]1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217882706 CI For-Sale Unstable HCAR2 0 40 Cc1ccc2[nH]cc(C3=CCN(Cc4ccccc4)CC3)c2c1 ZINC000217882707 DJ For-Sale Unstable HTR1A 22 53 Cc1ccc2[nH]cc(C3=CCN(Cc4ccccc4)CC3)c2c1 ZINC000217882707 DJ For-Sale Unstable DRD2 21 54 Cc1ccc2[nH]cc(C3=CCN(Cc4ccccc4)CC3)c2c1 ZINC000217882707 DJ For-Sale Unstable DRD4 18 48 Cc1ccc2[nH]cc(C3=CCN(Cc4ccccc4)CC3)c2c1 ZINC000217882707 DJ For-Sale Unstable HTR1D 57 42 Cc1ccc2[nH]cc(C3=CCN(Cc4ccccc4)CC3)c2c1 ZINC000217882707 DJ For-Sale Unstable HTR1B 46 38 Cc1ccc2[nH]cc(C3=CCN(Cc4ccccc4)CC3)c2c1 ZINC000217882707 DJ For-Sale Unstable SLC6A4 26 63 COc1ccc(CC[C@H](C)N[C@H]2CCC[C@@H](C)[C@@H]2C)cc1 ZINC000217882720 CI For-Sale Unstable SLC18A2 27 42 Cc1cccc(S(=O)(=O)Nc2ccc3nc(N4CCCC4)sc3c2)c1 ZINC000217882727 FI On-Demand Unstable NR1I2 44 39 COc1ccccc1CCCNC(=O)/C=C/c1ccccc1 ZINC000217882732 CG In-Stock Unstable DRD2 18 59 COc1ccccc1CCCNC(=O)/C=C/c1ccccc1 ZINC000217882732 CG In-Stock Unstable ACHE 0 40 COc1ccccc1CCCNC(=O)/C=C/c1ccccc1 ZINC000217882732 CG In-Stock Unstable DRD3 32 59 COc1ccccc1CCCNC(=O)/C=C/c1ccccc1 ZINC000217882732 CG In-Stock Unstable PTGER2 0 41 COc1ccccc1CCCNC(=O)/C=C/c1ccccc1 ZINC000217882732 CG In-Stock Unstable PTGER4 0 41 COc1ccccc1CCCNC(=O)/C=C/c1ccccc1 ZINC000217882732 CG In-Stock Unstable BCHE 15 41 COc1ccccc1CCCNC(=O)/C=C/c1ccccc1 ZINC000217882732 CG In-Stock Unstable KCNA3 15 43 COc1ccccc1CCCNC(=O)/C=C/c1ccccc1 ZINC000217882732 CG In-Stock Unstable PYGL 0 41 COc1ccccc1CCCNC(=O)/C=C/c1ccccc1 ZINC000217882732 CG In-Stock Unstable MTNR1A 33 40 COc1ccccc1CCCNC(=O)/C=C/c1ccccc1 ZINC000217882732 CG In-Stock Unstable MTNR1B 44 44 COc1ccccc1CCCNC(=O)/C=C/c1ccccc1 ZINC000217882732 CG In-Stock Unstable F3 17 40 COc1ccccc1CCCNC(=O)/C=C/c1ccccc1 ZINC000217882732 CG In-Stock Unstable MMP2 22 56 COc1ccccc1CCCNC(=O)/C=C/c1ccccc1 ZINC000217882732 CG In-Stock Unstable HDAC2 20 45 COc1ccccc1CCCNC(=O)/C=C/c1ccccc1 ZINC000217882732 CG In-Stock Unstable HDAC4 16 45 COc1ccccc1CCCNC(=O)/C=C/c1ccccc1 ZINC000217882732 CG In-Stock Unstable HDAC6 28 44 COc1ccccc1CCCNC(=O)/C=C/c1ccccc1 ZINC000217882732 CG In-Stock Unstable MMP9 18 56 COc1ccccc1CCCNC(=O)/C=C/c1ccccc1 ZINC000217882732 CG In-Stock Unstable HDAC9 41 45 COc1ccccc1CCCNC(=O)/C=C/c1ccccc1 ZINC000217882732 CG In-Stock Unstable HDAC7 51 45 COc1ccccc1CCCNC(=O)/C=C/c1ccccc1 ZINC000217882732 CG In-Stock Unstable MMP1 0 40 COc1ccccc1CCCNC(=O)/C=C/c1ccccc1 ZINC000217882732 CG In-Stock Unstable MBTPS1 40 31 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCc1ccc(F)c(Br)c1 ZINC000217882735 EK For-Sale Unstable TRPM8 16 44 Cc1cccc(/C=C/NC(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)c1 ZINC000217882758 HK For-Sale Unstable OPRD1 0 45 Cc1cccc(/C=C/NC(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)c1 ZINC000217882758 HK For-Sale Unstable NMUR2 0 46 Cc1cccc(/C=C/NC(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)c1 ZINC000217882758 HK For-Sale Unstable NMUR1 0 46 C[C@@H]1CCCC[C@@H]1OCc1ccccc1/C=C\C(=O)O ZINC000217882772 CH For-Sale Unstable PTGER2 49 45 C[C@@H]1CCCC[C@@H]1OCc1ccccc1/C=C\C(=O)O ZINC000217882772 CH For-Sale Unstable PTGER4 22 45 C[C@@H]1CCCC[C@@H]1OCc1ccccc1/C=C\C(=O)O ZINC000217882772 CH For-Sale Unstable PTGER3 18 45 C[C@@H]1CCCC[C@@H]1OCc1ccccc1/C=C\C(=O)O ZINC000217882772 CH For-Sale Unstable PTGDR 0 43 C[C@@H](C(=O)O)c1ccc(CN2CC[C@@H](N)C2)cc1 ZINC000217882806 BD For-Sale Unstable PTGS1 31 48 C[C@@H](C(=O)O)c1ccc(CN2CC[C@@H](N)C2)cc1 ZINC000217882806 BD For-Sale Unstable PTGS2 23 48 C[C@@H](C(=O)O)c1ccc(CN2CC[C@@H](N)C2)cc1 ZINC000217882806 BD For-Sale Unstable SIGMAR1 42 39 C[C@@H](C(=O)O)c1ccc(CN2CC[C@@H](N)C2)cc1 ZINC000217882806 BD For-Sale Unstable MLNR 33 40 C[C@@H](C(=O)O)c1ccc(CN2CC[C@@H](N)C2)cc1 ZINC000217882806 BD For-Sale Unstable SLC22A20 0 47 CN1CCO[C@@H]([C@@H](N)Cc2cc(F)ccc2Br)C1 ZINC000217882812 DD For-Sale Unstable DPP4 15 40 COc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217882845 CG In-Stock Unstable DRD4 41 32 COc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217882845 CG In-Stock Unstable ACHE 0 46 COc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217882845 CG In-Stock Unstable DRD3 20 48 COc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217882845 CG In-Stock Unstable PTAFR 23 46 COc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217882845 CG In-Stock Unstable FDFT1 15 47 COc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217882845 CG In-Stock Unstable SCN2A 15 41 COc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217882845 CG In-Stock Unstable PYGL 0 42 COc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217882845 CG In-Stock Unstable HDAC8 64 41 COc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217882845 CG In-Stock Unstable MTNR1A 80 64 COc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217882845 CG In-Stock Unstable MTNR1B 66 47 COc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217882845 CG In-Stock Unstable MMP2 23 59 COc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217882845 CG In-Stock Unstable NR1H4 33 40 COc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217882845 CG In-Stock Unstable HDAC1 30 42 COc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217882845 CG In-Stock Unstable HDAC2 22 41 COc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217882845 CG In-Stock Unstable HDAC3 17 43 COc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217882845 CG In-Stock Unstable HDAC4 21 43 COc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217882845 CG In-Stock Unstable HDAC6 47 41 COc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217882845 CG In-Stock Unstable MMP9 22 59 COc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217882845 CG In-Stock Unstable HDAC9 34 43 COc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217882845 CG In-Stock Unstable HDAC7 43 43 COc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217882845 CG In-Stock Unstable MMP1 0 41 COc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217882845 CG In-Stock Unstable AMP1_PLAFQ 36 47 COc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217882845 CG In-Stock Unstable AKR1C3 27 44 COc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217882845 CG In-Stock Unstable CRTM 79 56 COc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217882845 CG In-Stock Unstable PDS 44 38 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1N[C@@H](C)c1ccc(O)cc1 ZINC000217882851 CJ For-Sale Unstable TRPM8 17 47 O=C(N[C@@H]1CCC[C@@H]1CO)c1ccc(Br)c(F)c1 ZINC000217882852 DE For-Sale Unstable SSTR3 28 45 COc1ccccc1S(=O)(=O)Nc1ccc2nc(N3CCCC3)sc2c1 ZINC000217882857 GH On-Demand Unstable GHSR 23 41 COc1ccccc1S(=O)(=O)Nc1ccc2nc(N3CCCC3)sc2c1 ZINC000217882857 GH On-Demand Unstable NR1I2 49 36 COc1ccccc1S(=O)(=O)Nc1ccc2nc(N3CCCC3)sc2c1 ZINC000217882857 GH On-Demand Unstable ALPL 20 41 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](N)C2)cc1 ZINC000217882866 BD For-Sale Unstable PTGS1 31 48 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](N)C2)cc1 ZINC000217882866 BD For-Sale Unstable PTGS2 23 48 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](N)C2)cc1 ZINC000217882866 BD For-Sale Unstable SIGMAR1 42 39 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](N)C2)cc1 ZINC000217882866 BD For-Sale Unstable MLNR 33 40 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](N)C2)cc1 ZINC000217882866 BD For-Sale Unstable SLC22A20 0 47 C[C@H]1CCCC[C@@H]1OCc1ccccc1/C=C\C(=O)O ZINC000217882888 CH For-Sale Unstable PTGER2 49 45 C[C@H]1CCCC[C@@H]1OCc1ccccc1/C=C\C(=O)O ZINC000217882888 CH For-Sale Unstable PTGER4 22 45 C[C@H]1CCCC[C@@H]1OCc1ccccc1/C=C\C(=O)O ZINC000217882888 CH For-Sale Unstable PTGER3 18 45 C[C@H]1CCCC[C@@H]1OCc1ccccc1/C=C\C(=O)O ZINC000217882888 CH For-Sale Unstable PTGDR 0 43 CN1CCO[C@H]([C@@H](N)Cc2cc(F)ccc2Br)C1 ZINC000217882890 DD For-Sale Unstable DPP4 15 40 Cn1cccc(C(=O)NCCn2ccc(-c3ccsc3)n2)c1=O ZINC000217882897 ED In-Stock Unstable POLR1A 48 35 O=C(N[C@H]1CCC[C@@H]1CO)c1ccc(Br)c(F)c1 ZINC000217882920 DE For-Sale Unstable SSTR3 28 45 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1N[C@@H](C)c1ccc(O)cc1 ZINC000217882931 CJ For-Sale Unstable TRPM8 17 47 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217882954 DG In-Stock Unstable PTAFR 15 46 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217882954 DG In-Stock Unstable SDH1 0 47 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217882954 DG In-Stock Unstable MMP13 24 40 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217882954 DG In-Stock Unstable HDAC8 54 49 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217882954 DG In-Stock Unstable CDC25B 22 40 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217882954 DG In-Stock Unstable MMP2 37 59 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217882954 DG In-Stock Unstable HDAC1 22 44 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217882954 DG In-Stock Unstable HDAC2 25 47 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217882954 DG In-Stock Unstable HDAC6 35 49 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217882954 DG In-Stock Unstable MMP9 31 59 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217882954 DG In-Stock Unstable MMP1 22 40 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217882954 DG In-Stock Unstable GPR183 0 43 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217882954 DG In-Stock Unstable GPR88 0 40 CC(C)OCCOCc1ccc(/C=C\C(=O)O)cc1F ZINC000217882971 CF For-Sale Unstable AKR1C3 30 42 O=C(N[C@@H]1CCC[C@H]1CO)c1ccc(Br)c(F)c1 ZINC000217882997 DE For-Sale Unstable SSTR3 28 45 C[C@@H](C(=O)O)c1ccc(CN2CC[C@@H](CN)C2)cc1 ZINC000217883003 CD For-Sale Unstable SLC6A3 15 42 C[C@@H](C(=O)O)c1ccc(CN2CC[C@@H](CN)C2)cc1 ZINC000217883003 CD For-Sale Unstable SIGMAR1 38 40 C[C@@H](C(=O)O)c1ccc(CN2CC[C@@H](CN)C2)cc1 ZINC000217883003 CD For-Sale Unstable SLC22A20 0 44 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1N[C@@H](C)c1ccc(O)cc1 ZINC000217883005 CJ For-Sale Unstable TRPM8 17 47 CC[C@H]1COCCN1C(=O)[C@H](N)[C@H](C)CC ZINC000217883008 BC For-Sale Unstable TPP2 29 44 CC(C)(C)OC(=O)N1CCC(CNC(=O)CCc2cc(=O)[nH]o2)CC1 ZINC000217883015 FD For-Sale Unstable CACNA1I 49 34 CC(C)(C)OC(=O)N1CCC(CNC(=O)CCc2cc(=O)[nH]o2)CC1 ZINC000217883015 FD For-Sale Unstable GPR119 39 44 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)Nc1nc2c(s1)CCC2 ZINC000217883019 JI In-Stock Unstable SLC27A1 31 43 CN(Cc1ccccc1N1CCOCC1)S(=O)(=O)C[C@@]12CC[C@@H](CC1=O)C2(C)C ZINC000217883022 HF On-Demand Unstable CA5B 24 40 CN(Cc1ccccc1N1CCOCC1)S(=O)(=O)C[C@@]12CC[C@@H](CC1=O)C2(C)C ZINC000217883022 HF On-Demand Unstable CA5A 26 40 CN(Cc1ccccc1N1CCOCC1)S(=O)(=O)C[C@@]12CC[C@@H](CC1=O)C2(C)C ZINC000217883022 HF On-Demand Unstable CXCR3 0 42 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217883030 DG In-Stock Unstable PTAFR 15 46 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217883030 DG In-Stock Unstable SDH1 0 47 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217883030 DG In-Stock Unstable MMP13 24 40 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217883030 DG In-Stock Unstable HDAC8 54 49 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217883030 DG In-Stock Unstable CDC25B 22 40 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217883030 DG In-Stock Unstable MMP2 37 59 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217883030 DG In-Stock Unstable HDAC1 22 44 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217883030 DG In-Stock Unstable HDAC2 25 47 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217883030 DG In-Stock Unstable HDAC6 35 49 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217883030 DG In-Stock Unstable MMP9 31 59 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217883030 DG In-Stock Unstable MMP1 22 40 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217883030 DG In-Stock Unstable GPR183 0 43 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217883030 DG In-Stock Unstable GPR88 0 40 c1cncc(-c2ccc(N3CCOCC3)cc2)c1 ZINC000217883047 BF Annotated Unstable PRKAB1 30 42 c1cncc(-c2ccc(N3CCOCC3)cc2)c1 ZINC000217883047 BF Annotated Unstable PIK3CA 35 49 c1cncc(-c2ccc(N3CCOCC3)cc2)c1 ZINC000217883047 BF Annotated Unstable CHRNA4 22 41 c1cncc(-c2ccc(N3CCOCC3)cc2)c1 ZINC000217883047 BF Annotated Unstable CYP11B2 57 38 c1cncc(-c2ccc(N3CCOCC3)cc2)c1 ZINC000217883047 BF Annotated Unstable PRNP 27 47 c1cncc(-c2ccc(N3CCOCC3)cc2)c1 ZINC000217883047 BF Annotated Unstable JAK2 15 46 c1cncc(-c2ccc(N3CCOCC3)cc2)c1 ZINC000217883047 BF Annotated Unstable MAPKAPK5 43 34 c1cncc(-c2ccc(N3CCOCC3)cc2)c1 ZINC000217883047 BF Annotated Unstable MTOR 24 43 c1cncc(-c2ccc(N3CCOCC3)cc2)c1 ZINC000217883047 BF Annotated Unstable MAPK10 21 47 c1cncc(-c2ccc(N3CCOCC3)cc2)c1 ZINC000217883047 BF Annotated Unstable PIK3CG 19 43 c1cncc(-c2ccc(N3CCOCC3)cc2)c1 ZINC000217883047 BF Annotated Unstable CYP2E1 47 34 c1cncc(-c2ccc(N3CCOCC3)cc2)c1 ZINC000217883047 BF Annotated Unstable CYP2A6 52 38 c1cncc(-c2ccc(N3CCOCC3)cc2)c1 ZINC000217883047 BF Annotated Unstable TGFBR2 43 44 c1cncc(-c2ccc(N3CCOCC3)cc2)c1 ZINC000217883047 BF Annotated Unstable ACVR1B 20 44 c1cncc(-c2ccc(N3CCOCC3)cc2)c1 ZINC000217883047 BF Annotated Unstable BMPR2 21 42 c1cncc(-c2ccc(N3CCOCC3)cc2)c1 ZINC000217883047 BF Annotated Unstable BMP4 45 44 c1cncc(-c2ccc(N3CCOCC3)cc2)c1 ZINC000217883047 BF Annotated Unstable STAT6 41 34 c1cncc(-c2ccc(N3CCOCC3)cc2)c1 ZINC000217883047 BF Annotated Unstable BMPR1B 34 44 c1cncc(-c2ccc(N3CCOCC3)cc2)c1 ZINC000217883047 BF Annotated Unstable ACVR1 36 44 c1cncc(-c2ccc(N3CCOCC3)cc2)c1 ZINC000217883047 BF Annotated Unstable SMG1 40 32 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)Cc1cccc(OC)c1 ZINC000217883055 GF In-Stock Unstable DRD4 41 32 O=C(N[C@H]1CCC[C@H]1CO)c1ccc(Br)c(F)c1 ZINC000217883080 DE On-Demand Unstable SSTR3 26 43 CCCCNC(=O)N/C=C/c1cccc(C)c1 ZINC000217883085 BG For-Sale Unstable ACAT 0 44 CCCCN1C[C@@H](O)C[C@@H]1C(C)C ZINC000217883094 AD In-Stock Unstable GBA2 43 35 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](CN)C2)cc1 ZINC000217883106 CD For-Sale Unstable SLC6A3 15 42 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](CN)C2)cc1 ZINC000217883106 CD For-Sale Unstable SIGMAR1 38 40 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](CN)C2)cc1 ZINC000217883106 CD For-Sale Unstable SLC22A20 0 44 CC(C)[C@H]1CC[C@H](C)C[C@@H]1N[C@@H](C)c1ccc(O)cc1 ZINC000217883107 CJ For-Sale Unstable TRPM8 17 47 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)Nc1nc2c(s1)CCC2 ZINC000217883118 JI In-Stock Unstable SLC27A1 31 43 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)Cc1cccc(OC)c1 ZINC000217883137 GF In-Stock Unstable DRD4 41 32 CC[C@@H](C)[C@H](NS(=O)(=O)N1C[C@H](C)O[C@@H](C)C1)C(=O)O ZINC000217883150 DC For-Sale Unstable ENPEP 50 36 CCCCOCCOCc1ccc(/C=C\C(=O)O)cc1F ZINC000217883155 CG For-Sale Unstable AKR1C3 29 44 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217883162 DI In-Stock Unstable ANPEP 17 42 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217883162 DI In-Stock Unstable PTAFR 23 41 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217883162 DI In-Stock Unstable FDFT1 23 46 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217883162 DI In-Stock Unstable PYGL 0 40 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217883162 DI In-Stock Unstable HDAC8 59 40 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217883162 DI In-Stock Unstable MTNR1A 31 49 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217883162 DI In-Stock Unstable MTNR1B 35 41 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217883162 DI In-Stock Unstable MMP2 24 56 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217883162 DI In-Stock Unstable HDAC1 34 44 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217883162 DI In-Stock Unstable HDAC2 21 44 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217883162 DI In-Stock Unstable HDAC3 18 44 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217883162 DI In-Stock Unstable HDAC4 26 44 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217883162 DI In-Stock Unstable HDAC6 42 40 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217883162 DI In-Stock Unstable FAAH 15 43 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217883162 DI In-Stock Unstable MMP9 18 56 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217883162 DI In-Stock Unstable HDAC9 40 44 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217883162 DI In-Stock Unstable HDAC7 42 44 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217883162 DI In-Stock Unstable TSPAN17 0 40 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217883162 DI In-Stock Unstable AMP1_PLAFQ 48 48 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217883162 DI In-Stock Unstable HDA106 0 40 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217883162 DI In-Stock Unstable CRTM 77 56 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccccc2)c1 ZINC000217883162 DI In-Stock Unstable PDS 51 39 CCCCN1C[C@H](O)C[C@@H]1C(C)C ZINC000217883205 AD In-Stock Unstable GBA2 43 35 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)Cc1cccc(OC)c1 ZINC000217883224 GF In-Stock Unstable DRD4 41 32 CC(C)Oc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883246 DI In-Stock Unstable ANPEP 15 44 CC(C)Oc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883246 DI In-Stock Unstable SDH1 0 42 CC(C)Oc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883246 DI In-Stock Unstable MMP2 28 59 CC(C)Oc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883246 DI In-Stock Unstable NR1H4 20 40 CC(C)Oc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883246 DI In-Stock Unstable HDAC1 29 48 CC(C)Oc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883246 DI In-Stock Unstable HDAC2 21 48 CC(C)Oc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883246 DI In-Stock Unstable HDAC3 16 48 CC(C)Oc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883246 DI In-Stock Unstable HDAC4 28 48 CC(C)Oc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883246 DI In-Stock Unstable HDAC6 29 41 CC(C)Oc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883246 DI In-Stock Unstable MMP9 18 59 CC(C)Oc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883246 DI In-Stock Unstable HDAC9 47 48 CC(C)Oc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883246 DI In-Stock Unstable HDAC7 52 48 CC(C)Oc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883246 DI In-Stock Unstable AMP1_PLAFQ 33 44 CC(C)Oc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883246 DI In-Stock Unstable AKR1C3 0 40 CC(C)Oc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883246 DI In-Stock Unstable CRTM 42 42 CC(C)Oc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883246 DI In-Stock Unstable TRPM2 0 43 CC(=O)N1c2ccc(S(=O)(=O)N3CCN([C@@H](C#N)c4ccccc4)CC3)cc2C[C@@H]1C ZINC000217883253 IF On-Demand Unstable NOD1 15 49 CC(=O)N1c2ccc(S(=O)(=O)N3CCN([C@@H](C#N)c4ccccc4)CC3)cc2C[C@@H]1C ZINC000217883253 IF On-Demand Unstable NOD2 23 49 COC(=O)C[C@@H]1CCCCN1C[C@@H](O)c1ccccc1 ZINC000217883254 CE On-Demand Unstable SLC6A3 52 51 COC(=O)C[C@@H]1CCCCN1C[C@@H](O)c1ccccc1 ZINC000217883254 CE On-Demand Unstable SLC18A2 56 45 COC(=O)C[C@@H]1CCCCN1C[C@@H](O)c1ccccc1 ZINC000217883254 CE On-Demand Unstable SIGMAR1 17 43 COC(=O)C[C@@H]1CCCCN1C[C@@H](O)c1ccccc1 ZINC000217883254 CE On-Demand Unstable BIRC8 40 31 COC(=O)C[C@@H]1CCCCN1C[C@@H](O)c1ccccc1 ZINC000217883254 CE On-Demand Unstable ACHP_LYMST 17 45 COC(=O)C[C@@H]1CCCCN1C[C@@H](O)c1ccccc1 ZINC000217883254 CE On-Demand Unstable Q8WSF8_APLCA 34 45 CC[C@@H](C)[C@H](NS(=O)(=O)N1C[C@H](C)C[C@@H](C)C1)C(=O)O ZINC000217883265 DD For-Sale Unstable ENPEP 50 36 CCCCOCCOCc1cccc(/C=C\C(=O)O)c1 ZINC000217883276 CG For-Sale Unstable PTGER2 30 44 CCCCOCCOCc1cccc(/C=C\C(=O)O)c1 ZINC000217883276 CG For-Sale Unstable LTB4R 27 44 CCCCOCCOCc1cccc(/C=C\C(=O)O)c1 ZINC000217883276 CG For-Sale Unstable PLA2G4B 54 43 CCCCOCCOCc1cccc(/C=C\C(=O)O)c1 ZINC000217883276 CG For-Sale Unstable 17HSDCL 0 40 CCCCOCCOCc1cccc(/C=C\C(=O)O)c1 ZINC000217883276 CG For-Sale Unstable AKR1C3 32 51 COC(=O)C[C@H]1CCCCN1C[C@@H](O)c1ccccc1 ZINC000217883309 CE On-Demand Unstable SLC6A3 52 51 COC(=O)C[C@H]1CCCCN1C[C@@H](O)c1ccccc1 ZINC000217883309 CE On-Demand Unstable SLC18A2 56 45 COC(=O)C[C@H]1CCCCN1C[C@@H](O)c1ccccc1 ZINC000217883309 CE On-Demand Unstable SIGMAR1 17 43 COC(=O)C[C@H]1CCCCN1C[C@@H](O)c1ccccc1 ZINC000217883309 CE On-Demand Unstable BIRC8 40 31 COC(=O)C[C@H]1CCCCN1C[C@@H](O)c1ccccc1 ZINC000217883309 CE On-Demand Unstable ACHP_LYMST 17 45 COC(=O)C[C@H]1CCCCN1C[C@@H](O)c1ccccc1 ZINC000217883309 CE On-Demand Unstable Q8WSF8_APLCA 34 45 CC(=O)N1c2ccc(S(=O)(=O)N3CCN([C@H](C#N)c4ccccc4)CC3)cc2C[C@@H]1C ZINC000217883318 IF On-Demand Unstable NOD1 15 49 CC(=O)N1c2ccc(S(=O)(=O)N3CCN([C@H](C#N)c4ccccc4)CC3)cc2C[C@@H]1C ZINC000217883318 IF On-Demand Unstable NOD2 23 49 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](C)[C@@H]2C)cc1 ZINC000217883320 CG For-Sale Unstable PTGS1 25 50 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](C)[C@@H]2C)cc1 ZINC000217883320 CG For-Sale Unstable PTGS2 0 50 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](C)[C@@H]2C)cc1 ZINC000217883320 CG For-Sale Unstable HRH3 23 43 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](C)[C@@H]2C)cc1 ZINC000217883320 CG For-Sale Unstable SLC22A20 0 45 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)Cc1cccc(OC)c1 ZINC000217883321 GF In-Stock Unstable DRD4 41 32 Cc1cccc(=O)n1CCCNC(=O)CN1CC[C@@H](c2ccccc2)C1 ZINC000217883364 FE In-Stock Unstable DRD4 22 52 Cc1cccc(=O)n1CCCNC(=O)CN1CC[C@@H](c2ccccc2)C1 ZINC000217883364 FE In-Stock Unstable ADRA1D 42 54 Cc1cccc(=O)n1CCCNC(=O)CN1CC[C@@H](c2ccccc2)C1 ZINC000217883364 FE In-Stock Unstable ADRA1A 33 40 Cc1cccc(=O)n1CCCNC(=O)CN1CC[C@@H](c2ccccc2)C1 ZINC000217883364 FE In-Stock Unstable ADRA1B 28 54 Cc1cccc(=O)n1CCCNC(=O)CN1CC[C@@H](c2ccccc2)C1 ZINC000217883364 FE In-Stock Unstable PRCP 23 40 Cc1cccc(=O)n1CCCNC(=O)CN1CC[C@@H](c2ccccc2)C1 ZINC000217883364 FE In-Stock Unstable MCHR1 25 44 O=C(/C=C/c1ccccc1)Nc1ccc(OC2CCCC2)cc1 ZINC000217883365 DJ In-Stock Unstable HDAC8 40 47 O=C(/C=C/c1ccccc1)Nc1ccc(OC2CCCC2)cc1 ZINC000217883365 DJ In-Stock Unstable MMP2 27 64 O=C(/C=C/c1ccccc1)Nc1ccc(OC2CCCC2)cc1 ZINC000217883365 DJ In-Stock Unstable HDAC1 34 40 O=C(/C=C/c1ccccc1)Nc1ccc(OC2CCCC2)cc1 ZINC000217883365 DJ In-Stock Unstable HDAC2 22 45 O=C(/C=C/c1ccccc1)Nc1ccc(OC2CCCC2)cc1 ZINC000217883365 DJ In-Stock Unstable HDAC6 29 47 O=C(/C=C/c1ccccc1)Nc1ccc(OC2CCCC2)cc1 ZINC000217883365 DJ In-Stock Unstable MMP9 22 64 O=C(/C=C/c1ccccc1)Nc1ccc(OC2CCCC2)cc1 ZINC000217883365 DJ In-Stock Unstable EPHX2 21 40 O=C(/C=C/c1ccccc1)Nc1ccc(OC2CCCC2)cc1 ZINC000217883365 DJ In-Stock Unstable MMP1 29 58 O=C(/C=C/c1ccccc1)Nc1ccc(OC2CCCC2)cc1 ZINC000217883365 DJ In-Stock Unstable MCHR1 17 40 O=C(/C=C/c1ccccc1)Nc1ccc(OC2CCCC2)cc1 ZINC000217883365 DJ In-Stock Unstable METAP2 0 45 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1cccc(C)c1 ZINC000217883416 GF For-Sale Unstable COLA 70 38 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1cccc(C)c1 ZINC000217883416 GF For-Sale Unstable CPT1A 62 38 CC(=O)N1c2ccc(S(=O)(=O)N3CCN([C@@H](C#N)c4ccccc4)CC3)cc2C[C@H]1C ZINC000217883419 IF On-Demand Unstable NOD1 15 49 CC(=O)N1c2ccc(S(=O)(=O)N3CCN([C@@H](C#N)c4ccccc4)CC3)cc2C[C@H]1C ZINC000217883419 IF On-Demand Unstable NOD2 23 49 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)Nc1cccc(C(C)=O)c1)C(=O)OC2 ZINC000217883424 JJ In-Stock Unstable IMPDH1 0 63 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)Nc1cccc(C(C)=O)c1)C(=O)OC2 ZINC000217883424 JJ In-Stock Unstable IMPDH2 0 63 Cc1cccc(=O)n1CCCNC(=O)CN1CC[C@H](c2ccccc2)C1 ZINC000217883451 FE In-Stock Unstable DRD4 22 52 Cc1cccc(=O)n1CCCNC(=O)CN1CC[C@H](c2ccccc2)C1 ZINC000217883451 FE In-Stock Unstable ADRA1D 42 54 Cc1cccc(=O)n1CCCNC(=O)CN1CC[C@H](c2ccccc2)C1 ZINC000217883451 FE In-Stock Unstable ADRA1A 33 40 Cc1cccc(=O)n1CCCNC(=O)CN1CC[C@H](c2ccccc2)C1 ZINC000217883451 FE In-Stock Unstable ADRA1B 28 54 Cc1cccc(=O)n1CCCNC(=O)CN1CC[C@H](c2ccccc2)C1 ZINC000217883451 FE In-Stock Unstable PRCP 23 40 Cc1cccc(=O)n1CCCNC(=O)CN1CC[C@H](c2ccccc2)C1 ZINC000217883451 FE In-Stock Unstable MCHR1 25 44 COc1ccc(F)cc1-c1c(Cl)cnc2[nH]c(I)cc12 ZINC000217883461 HJ For-Sale Unstable KIT 18 45 Cc1cccc(/C=C/NC(=O)N2CCCc3ccccc32)c1 ZINC000217883465 CI For-Sale Unstable AVPR2 46 52 C[C@H]1C[C@H](C)CCN1Cc1ccc([C@@H](C)C(=O)O)cc1 ZINC000217883472 CG For-Sale Unstable PTGS1 25 47 C[C@H]1C[C@H](C)CCN1Cc1ccc([C@@H](C)C(=O)O)cc1 ZINC000217883472 CG For-Sale Unstable PTGS2 0 47 C[C@H]1C[C@H](C)CCN1Cc1ccc([C@@H](C)C(=O)O)cc1 ZINC000217883472 CG For-Sale Unstable SLC22A20 0 45 CC1(C)C[C@@H](NC(=O)/C=C/c2ccccc2)c2ccccc2O1 ZINC000217883480 DI In-Stock Unstable MMP2 16 40 CC1(C)C[C@@H](NC(=O)/C=C/c2ccccc2)c2ccccc2O1 ZINC000217883480 DI In-Stock Unstable HDAC6 19 43 CC[C@@H](c1ccccc1O)N1CCC[C@@H](C(C)(C)C)CC1 ZINC000217883487 CJ For-Sale Unstable AMY2 44 31 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1cccc(C)c1 ZINC000217883497 GF For-Sale Unstable COLA 70 38 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1cccc(C)c1 ZINC000217883497 GF For-Sale Unstable CPT1A 62 38 CC(=O)N1c2ccc(S(=O)(=O)N3CCN([C@H](C#N)c4ccccc4)CC3)cc2C[C@H]1C ZINC000217883508 IF On-Demand Unstable NOD1 15 49 CC(=O)N1c2ccc(S(=O)(=O)N3CCN([C@H](C#N)c4ccccc4)CC3)cc2C[C@H]1C ZINC000217883508 IF On-Demand Unstable NOD2 23 49 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cnn(C)c2C)CC(=O)O4)cc1O ZINC000217883519 IG In-Stock Unstable CYP1A1 30 44 CC1(C)C[C@H](NC(=O)/C=C/c2ccccc2)c2ccccc2O1 ZINC000217883546 DI In-Stock Unstable MMP2 16 40 CC1(C)C[C@H](NC(=O)/C=C/c2ccccc2)c2ccccc2O1 ZINC000217883546 DI In-Stock Unstable HDAC6 19 43 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](C)C[C@@H]2C)cc1 ZINC000217883552 CG For-Sale Unstable PTGS1 25 47 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](C)C[C@@H]2C)cc1 ZINC000217883552 CG For-Sale Unstable PTGS2 0 47 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](C)C[C@@H]2C)cc1 ZINC000217883552 CG For-Sale Unstable SLC22A20 0 45 Cc1cccc(/C=C/NC(=O)NCCc2ccccc2)c1 ZINC000217883566 CH For-Sale Unstable HDAC8 37 40 Cc1cccc(/C=C/NC(=O)NCCc2ccccc2)c1 ZINC000217883566 CH For-Sale Unstable MMP2 17 55 Cc1cccc(/C=C/NC(=O)NCCc2ccccc2)c1 ZINC000217883566 CH For-Sale Unstable HDAC1 17 40 Cc1cccc(/C=C/NC(=O)NCCc2ccccc2)c1 ZINC000217883566 CH For-Sale Unstable HDAC6 30 42 Cc1cccc(/C=C/NC(=O)NCCc2ccccc2)c1 ZINC000217883566 CH For-Sale Unstable FBP1 15 40 Cc1cccc(/C=C/NC(=O)NCCc2ccccc2)c1 ZINC000217883566 CH For-Sale Unstable SCN5A 0 43 Cc1cccc(/C=C/NC(=O)NCCc2ccccc2)c1 ZINC000217883566 CH For-Sale Unstable AKR1C3 30 41 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1cccc(C)c1 ZINC000217883574 GF For-Sale Unstable COLA 70 38 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1cccc(C)c1 ZINC000217883574 GF For-Sale Unstable CPT1A 62 38 CC[C@H](c1ccccc1O)N1CCC[C@@H](C(C)(C)C)CC1 ZINC000217883582 CJ For-Sale Unstable AMY2 44 31 Nc1cccc(-c2nnc(-c3ccc(-c4ccccc4)cc3)o2)c1 ZINC000217883593 DJ In-Stock Unstable CYP73A16 31 47 Nc1cccc(-c2nnc(-c3ccc(-c4ccccc4)cc3)o2)c1 ZINC000217883593 DJ In-Stock Unstable MVFR 0 47 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cnn(C)c2C)CC(=O)O4)cc1O ZINC000217883598 IG In-Stock Unstable CYP1A1 30 44 COc1cccc(CN[C@H]2C[C@@H](C)CC[C@@H]2C(C)C)c1O ZINC000217883607 CH For-Sale Unstable TRPM8 16 44 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1cccc(C)c1 ZINC000217883644 GF For-Sale Unstable COLA 70 38 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1cccc(C)c1 ZINC000217883644 GF For-Sale Unstable CPT1A 62 38 CCOc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883652 DH In-Stock Unstable ALOX5 15 42 CCOc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883652 DH In-Stock Unstable PPARG 24 48 CCOc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883652 DH In-Stock Unstable PPARA 18 43 CCOc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883652 DH In-Stock Unstable LTA4H 23 40 CCOc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883652 DH In-Stock Unstable SDH1 0 45 CCOc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883652 DH In-Stock Unstable LTB4R 25 40 CCOc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883652 DH In-Stock Unstable SCN2A 23 50 CCOc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883652 DH In-Stock Unstable PYGL 0 40 CCOc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883652 DH In-Stock Unstable HDAC8 41 38 CCOc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883652 DH In-Stock Unstable MTNR1B 30 40 CCOc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883652 DH In-Stock Unstable MMP2 26 60 CCOc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883652 DH In-Stock Unstable HDAC1 31 46 CCOc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883652 DH In-Stock Unstable HDAC2 22 46 CCOc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883652 DH In-Stock Unstable HDAC3 19 46 CCOc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883652 DH In-Stock Unstable HDAC4 26 46 CCOc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883652 DH In-Stock Unstable HDAC6 31 42 CCOc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883652 DH In-Stock Unstable FAAH 27 45 CCOc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883652 DH In-Stock Unstable MMP9 20 60 CCOc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883652 DH In-Stock Unstable HDAC9 41 46 CCOc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883652 DH In-Stock Unstable HDAC7 53 46 CCOc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883652 DH In-Stock Unstable AMP1_PLAFQ 27 41 CCOc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883652 DH In-Stock Unstable CRTM 43 43 CCOc1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217883652 DH In-Stock Unstable TRPM2 0 47 Cc1cccc(/C=C/NC(=O)NC2CCCC2)c1 ZINC000217883661 BG For-Sale Unstable EPHX2 26 43 C[C@H]1C[C@H](C)CCN1Cc1ccc(CC(=O)O)cc1 ZINC000217883667 CF For-Sale Unstable SIGMAR1 29 41 CCC[C@@H](O)CNCCCCOC ZINC000217883669 AD For-Sale Unstable SPPS 45 38 CCN(C)C(=O)CNC(=O)c1ccc(N)cc1OC ZINC000217883671 CC For-Sale Unstable HTR4 33 47 CC1(C)[C@H]2CC[C@@]1(CS(=O)(=O)N1CCN([C@@H](C#N)c3ccccc3)CC1)C(=O)C2 ZINC000217883681 HF On-Demand Unstable AVPR2 98 36 CC1(C)[C@H]2CC[C@@]1(CS(=O)(=O)N1CCN([C@@H](C#N)c3ccccc3)CC1)C(=O)C2 ZINC000217883681 HF On-Demand Unstable OXTR 72 44 CC1(C)[C@H]2CC[C@@]1(CS(=O)(=O)N1CCN([C@@H](C#N)c3ccccc3)CC1)C(=O)C2 ZINC000217883681 HF On-Demand Unstable CA5B 24 41 CC1(C)[C@H]2CC[C@@]1(CS(=O)(=O)N1CCN([C@@H](C#N)c3ccccc3)CC1)C(=O)C2 ZINC000217883681 HF On-Demand Unstable CA5A 27 41 CC1(C)[C@H]2CC[C@@]1(CS(=O)(=O)N1CCN([C@@H](C#N)c3ccccc3)CC1)C(=O)C2 ZINC000217883681 HF On-Demand Unstable CXCR3 50 54 COc1cccc(CN[C@H]2C[C@H](C)CC[C@@H]2C(C)C)c1O ZINC000217883700 CH For-Sale Unstable TRPM8 16 44 CCC[C@H](O)CNCCCCOC ZINC000217883725 AD For-Sale Unstable SPPS 45 38 C[C@H]1CCN(Cc2ccc(CC(=O)O)cc2)[C@@H](C)C1 ZINC000217883754 CF For-Sale Unstable SIGMAR1 29 41 Cc1cccc(/C=C/NC(=O)NCc2ccccc2Cl)c1 ZINC000217883758 DI For-Sale Unstable P2RX7 49 43 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccccc1 ZINC000217883759 DI In-Stock Unstable DRD3 15 48 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccccc1 ZINC000217883759 DI In-Stock Unstable MTNR1A 41 47 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccccc1 ZINC000217883759 DI In-Stock Unstable MTNR1B 46 41 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccccc1 ZINC000217883759 DI In-Stock Unstable MMP2 17 51 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccccc1 ZINC000217883759 DI In-Stock Unstable HDAC1 19 42 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccccc1 ZINC000217883759 DI In-Stock Unstable HDAC2 18 42 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccccc1 ZINC000217883759 DI In-Stock Unstable HDAC3 15 42 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccccc1 ZINC000217883759 DI In-Stock Unstable HDAC4 20 42 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccccc1 ZINC000217883759 DI In-Stock Unstable HDAC6 18 42 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccccc1 ZINC000217883759 DI In-Stock Unstable HDAC9 39 42 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccccc1 ZINC000217883759 DI In-Stock Unstable HDAC7 41 42 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccccc1 ZINC000217883759 DI In-Stock Unstable IMA1 0 41 O=C(CCc1ccccc1Cl)N[C@H]1CCC[C@H]1CO ZINC000217883786 CF On-Demand Unstable PDE7A 15 41 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccccc1SC ZINC000217883788 GG For-Sale Unstable HCRTR1 44 36 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccccc1SC ZINC000217883788 GG For-Sale Unstable HCRTR2 46 36 COc1ccc([C@@H](C)N[C@H]2C[C@@H](C)CC[C@@H]2C(C)C)cc1 ZINC000217883810 CJ For-Sale Unstable TRPM8 17 48 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccccc1SC ZINC000217883849 GG For-Sale Unstable HCRTR1 44 36 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccccc1SC ZINC000217883849 GG For-Sale Unstable HCRTR2 46 36 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccccc1 ZINC000217883851 CH In-Stock Unstable HDAC8 51 35 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccccc1 ZINC000217883851 CH In-Stock Unstable MMP2 20 50 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccccc1 ZINC000217883851 CH In-Stock Unstable HDAC2 17 45 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccccc1 ZINC000217883851 CH In-Stock Unstable HDAC6 32 45 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccccc1 ZINC000217883851 CH In-Stock Unstable MMP9 18 50 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccccc1 ZINC000217883851 CH In-Stock Unstable UL26 36 41 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccccc1 ZINC000217883851 CH In-Stock Unstable MMP1 0 42 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccccc1 ZINC000217883851 CH In-Stock Unstable SCAF_EBVB9 25 41 COc1ccc(CCNC(=O)N/C=C/c2cccc(C)c2)cc1OC ZINC000217883860 EH For-Sale Unstable MTNR1A 26 42 COc1ccc(CCNC(=O)N/C=C/c2cccc(C)c2)cc1OC ZINC000217883860 EH For-Sale Unstable MTNR1B 28 44 COc1ccc(CCNC(=O)N/C=C/c2cccc(C)c2)cc1OC ZINC000217883860 EH For-Sale Unstable ABCG2 18 43 COc1ccc(CCNC(=O)N/C=C/c2cccc(C)c2)cc1OC ZINC000217883860 EH For-Sale Unstable STAT6 24 40 Nc1nccc(C2CCN(C(=O)c3ccc4cc[nH]c4c3)CC2)n1 ZINC000217883876 DF In-Stock Unstable L3MBTL1 0 40 Nc1nccc(C2CCN(C(=O)c3ccc4cc[nH]c4c3)CC2)n1 ZINC000217883876 DF In-Stock Unstable L3MBTL3 46 33 Cc1ccccc1C(=O)NCCn1ccc(-c2ccsc2)n1 ZINC000217883879 DG In-Stock Unstable POLR1A 47 35 COc1ccc([C@H](C)N[C@H]2C[C@@H](C)CC[C@@H]2C(C)C)cc1 ZINC000217883899 CJ For-Sale Unstable TRPM8 17 48 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccccc1SC ZINC000217883933 GG For-Sale Unstable HCRTR1 44 36 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccccc1SC ZINC000217883933 GG For-Sale Unstable HCRTR2 46 36 O=C(O)/C=C\c1cccc(CSc2ccc(F)cc2)c1 ZINC000217883953 CI For-Sale Unstable LTB4R 19 43 O=C(O)/C=C\c1cccc(CSc2ccc(F)cc2)c1 ZINC000217883953 CI For-Sale Unstable TDO2 0 41 O=C(O)/C=C\c1cccc(CSc2ccc(F)cc2)c1 ZINC000217883953 CI For-Sale Unstable HCAR2 0 43 O=C(O)/C=C\c1cccc(CSc2ccc(F)cc2)c1 ZINC000217883953 CI For-Sale Unstable AKR1C3 32 46 Clc1ccc2c(C3=CCN(Cc4ccccc4)CC3)c[nH]c2c1 ZINC000217883966 DK For-Sale Unstable HTR1A 18 48 Clc1ccc2c(C3=CCN(Cc4ccccc4)CC3)c[nH]c2c1 ZINC000217883966 DK For-Sale Unstable DRD2 24 56 Clc1ccc2c(C3=CCN(Cc4ccccc4)CC3)c[nH]c2c1 ZINC000217883966 DK For-Sale Unstable DRD4 21 56 Clc1ccc2c(C3=CCN(Cc4ccccc4)CC3)c[nH]c2c1 ZINC000217883966 DK For-Sale Unstable HTR1B 15 42 Clc1ccc2c(C3=CCN(Cc4ccccc4)CC3)c[nH]c2c1 ZINC000217883966 DK For-Sale Unstable SLC6A4 23 57 Clc1ccc2c(C3=CCN(Cc4ccccc4)CC3)c[nH]c2c1 ZINC000217883966 DK For-Sale Unstable DRD3 15 56 O=C(NCCn1ccc(-c2ccsc2)n1)c1ccc2c(c1)OCO2 ZINC000217883968 EF In-Stock Unstable DYRK2 49 37 C[C@@H](C(=O)O)c1ccc(CN2CC[C@@H](O)C2)cc1 ZINC000217883983 BD For-Sale Unstable PTGS1 35 50 C[C@@H](C(=O)O)c1ccc(CN2CC[C@@H](O)C2)cc1 ZINC000217883983 BD For-Sale Unstable PTGS2 25 50 C[C@@H](C(=O)O)c1ccc(CN2CC[C@@H](O)C2)cc1 ZINC000217883983 BD For-Sale Unstable OPRK1 25 45 C[C@@H](C(=O)O)c1ccc(CN2CC[C@@H](O)C2)cc1 ZINC000217883983 BD For-Sale Unstable MCHR1 30 41 C[C@@H](C(=O)O)c1ccc(CN2CC[C@@H](O)C2)cc1 ZINC000217883983 BD For-Sale Unstable SLC22A20 0 49 Cc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217883986 CH In-Stock Unstable HDAC8 50 40 Cc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217883986 CH In-Stock Unstable MMP2 24 52 Cc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217883986 CH In-Stock Unstable HDAC1 22 43 Cc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217883986 CH In-Stock Unstable HDAC2 20 44 Cc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217883986 CH In-Stock Unstable HDAC6 29 44 Cc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217883986 CH In-Stock Unstable MMP9 21 52 CC(C)[C@@H](NC(=O)OCc1cccc(F)c1)C(=O)O ZINC000217883991 CE For-Sale Unstable CELA1 19 42 CC(C)[C@@H](NC(=O)OCc1cccc(F)c1)C(=O)O ZINC000217883991 CE For-Sale Unstable ELANE 46 47 CC(C)[C@@H](NC(=O)OCc1cccc(F)c1)C(=O)O ZINC000217883991 CE For-Sale Unstable MME 46 40 CC(C)[C@@H](NC(=O)OCc1cccc(F)c1)C(=O)O ZINC000217883991 CE For-Sale Unstable CTRA_BOVIN 19 48 CC(C)[C@@H](NC(=O)OCc1cccc(F)c1)C(=O)O ZINC000217883991 CE For-Sale Unstable CASP3 34 68 CC(C)[C@@H](NC(=O)OCc1cccc(F)c1)C(=O)O ZINC000217883991 CE For-Sale Unstable BMP1 68 42 CC(C)[C@@H](NC(=O)OCc1cccc(F)c1)C(=O)O ZINC000217883991 CE For-Sale Unstable MMP13 15 54 CC(C)[C@@H](NC(=O)OCc1cccc(F)c1)C(=O)O ZINC000217883991 CE For-Sale Unstable KLK3 74 37 CC(C)[C@@H](NC(=O)OCc1cccc(F)c1)C(=O)O ZINC000217883991 CE For-Sale Unstable CTSB 70 51 CC(C)[C@@H](NC(=O)OCc1cccc(F)c1)C(=O)O ZINC000217883991 CE For-Sale Unstable PAPA1_CARPA 85 43 CC(C)[C@@H](NC(=O)OCc1cccc(F)c1)C(=O)O ZINC000217883991 CE For-Sale Unstable CYSP_TRYCR 58 38 CC(C)[C@@H](NC(=O)OCc1cccc(F)c1)C(=O)O ZINC000217883991 CE For-Sale Unstable CTSK 39 51 CC(C)[C@@H](NC(=O)OCc1cccc(F)c1)C(=O)O ZINC000217883991 CE For-Sale Unstable CTSL 42 51 CC(C)[C@@H](NC(=O)OCc1cccc(F)c1)C(=O)O ZINC000217883991 CE For-Sale Unstable CPA1 21 43 CC(C)[C@@H](NC(=O)OCc1cccc(F)c1)C(=O)O ZINC000217883991 CE For-Sale Unstable PGA 32 47 CC(C)[C@@H](NC(=O)OCc1cccc(F)c1)C(=O)O ZINC000217883991 CE For-Sale Unstable CAPNS1 67 39 CC(C)[C@@H](NC(=O)OCc1cccc(F)c1)C(=O)O ZINC000217883991 CE For-Sale Unstable HLA-DRB1 47 36 CC(C)[C@@H](NC(=O)OCc1cccc(F)c1)C(=O)O ZINC000217883991 CE For-Sale Unstable CTSS 19 43 CC(C)[C@@H](NC(=O)OCc1cccc(F)c1)C(=O)O ZINC000217883991 CE For-Sale Unstable CAPN1 82 50 CC(C)[C@@H](NC(=O)OCc1cccc(F)c1)C(=O)O ZINC000217883991 CE For-Sale Unstable CASP1 32 51 CC(C)[C@@H](NC(=O)OCc1cccc(F)c1)C(=O)O ZINC000217883991 CE For-Sale Unstable CTRC 17 40 CC(C)[C@@H](NC(=O)OCc1cccc(F)c1)C(=O)O ZINC000217883991 CE For-Sale Unstable CAPN2 119 50 CC(C)[C@@H](NC(=O)OCc1cccc(F)c1)C(=O)O ZINC000217883991 CE For-Sale Unstable CASP6 37 51 CC(C)[C@@H](NC(=O)OCc1cccc(F)c1)C(=O)O ZINC000217883991 CE For-Sale Unstable CASP9 50 51 CC(C)[C@@H](NC(=O)OCc1cccc(F)c1)C(=O)O ZINC000217883991 CE For-Sale Unstable ADAMTS4 57 40 CC(C)[C@@H](NC(=O)OCc1cccc(F)c1)C(=O)O ZINC000217883991 CE For-Sale Unstable HCAR2 17 50 CC(C)[C@@H](NC(=O)OCc1cccc(F)c1)C(=O)O ZINC000217883991 CE For-Sale Unstable NPR 73 46 CC(C)[C@@H](NC(=O)OCc1cccc(F)c1)C(=O)O ZINC000217883991 CE For-Sale Unstable PSMB5 38 40 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCc1c(F)cccc1Cl ZINC000217884020 CK For-Sale Unstable TRPM8 16 46 Cc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217884036 CH In-Stock Unstable HDAC8 50 40 Cc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217884036 CH In-Stock Unstable MMP2 24 52 Cc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217884036 CH In-Stock Unstable HDAC1 22 43 Cc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217884036 CH In-Stock Unstable HDAC2 20 44 Cc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217884036 CH In-Stock Unstable HDAC6 29 44 Cc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2)cc1 ZINC000217884036 CH In-Stock Unstable MMP9 21 52 O=C(O)/C=C\c1cc(F)ccc1CSc1ccc(F)cc1 ZINC000217884039 DI For-Sale Unstable PTGDR 0 42 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccccc1SC ZINC000217884048 GG For-Sale Unstable HCRTR1 44 36 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccccc1SC ZINC000217884048 GG For-Sale Unstable HCRTR2 46 36 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](O)C2)cc1 ZINC000217884056 BD For-Sale Unstable PTGS1 35 50 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](O)C2)cc1 ZINC000217884056 BD For-Sale Unstable PTGS2 25 50 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](O)C2)cc1 ZINC000217884056 BD For-Sale Unstable OPRK1 25 45 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](O)C2)cc1 ZINC000217884056 BD For-Sale Unstable MCHR1 30 41 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](O)C2)cc1 ZINC000217884056 BD For-Sale Unstable SLC22A20 0 49 N#Cc1cc(C(=O)N2CCOCC2)ccc1Cl ZINC000217884057 CD On-Demand Unstable AKR1C3 33 53 C=C(CNC[C@@H](O)CCC)c1ccccc1 ZINC000217884073 BE For-Sale Unstable AOC3 40 46 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCc1c(F)cccc1Cl ZINC000217884082 CK For-Sale Unstable TRPM8 16 46 COc1ccc(CSc2nc(C)cs2)cc1/C=C\C(=O)O ZINC000217884132 DH For-Sale Unstable PTGER4 23 42 COc1ccc(CSc2nc(C)cs2)cc1/C=C\C(=O)O ZINC000217884132 DH For-Sale Unstable PTGER3 17 42 CC1CCN(c2ccc([C@@H](C)NC(=O)/C=C/c3ccccc3)cc2)CC1 ZINC000217884136 EJ In-Stock Unstable KCNQ2 51 39 CC1CCN(c2ccc([C@@H](C)NC(=O)/C=C/c3ccccc3)cc2)CC1 ZINC000217884136 EJ In-Stock Unstable HDAC8 45 37 CC1CCN(c2ccc([C@@H](C)NC(=O)/C=C/c3ccccc3)cc2)CC1 ZINC000217884136 EJ In-Stock Unstable MMP2 15 40 CC1CCN(c2ccc([C@@H](C)NC(=O)/C=C/c3ccccc3)cc2)CC1 ZINC000217884136 EJ In-Stock Unstable HDAC6 35 43 Cc1c(CC(=O)N[C@H](CO)C(C)C)c(=O)oc2cc(O)ccc12 ZINC000217884142 DD In-Stock Unstable HSD17B3 47 54 Cc1c(CC(=O)N[C@H](CO)C(C)C)c(=O)oc2cc(O)ccc12 ZINC000217884142 DD In-Stock Unstable NQO1 52 37 C=C(CNC[C@H](O)CCC)c1ccccc1 ZINC000217884154 BE For-Sale Unstable AOC3 40 46 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCc1c(F)cccc1Cl ZINC000217884162 CK For-Sale Unstable TRPM8 16 46 Cc1cccc(/C=C/NC(=O)NCc2cccnc2)c1 ZINC000217884178 CF For-Sale Unstable TBXAS1 23 40 Cc1cccc(/C=C/NC(=O)NCc2cccnc2)c1 ZINC000217884178 CF For-Sale Unstable PTAFR 31 45 Cc1cccc(/C=C/NC(=O)NCc2cccnc2)c1 ZINC000217884178 CF For-Sale Unstable NAMPT 71 45 C[C@H]1CN(Cc2ccc([C@H](C)C(=O)O)cc2)CCCO1 ZINC000217884197 CE For-Sale Unstable DRD4 18 42 C[C@H]1CN(Cc2ccc([C@H](C)C(=O)O)cc2)CCCO1 ZINC000217884197 CE For-Sale Unstable PTGS1 22 44 C[C@H]1CN(Cc2ccc([C@H](C)C(=O)O)cc2)CCCO1 ZINC000217884197 CE For-Sale Unstable PTGS2 15 44 CC1CCN(c2ccc([C@H](C)NC(=O)/C=C/c3ccccc3)cc2)CC1 ZINC000217884232 EJ In-Stock Unstable KCNQ2 51 39 CC1CCN(c2ccc([C@H](C)NC(=O)/C=C/c3ccccc3)cc2)CC1 ZINC000217884232 EJ In-Stock Unstable HDAC8 45 37 CC1CCN(c2ccc([C@H](C)NC(=O)/C=C/c3ccccc3)cc2)CC1 ZINC000217884232 EJ In-Stock Unstable MMP2 15 40 CC1CCN(c2ccc([C@H](C)NC(=O)/C=C/c3ccccc3)cc2)CC1 ZINC000217884232 EJ In-Stock Unstable HDAC6 35 43 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCc1c(F)cccc1Cl ZINC000217884251 CK For-Sale Unstable TRPM8 16 46 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)/C=C/c3ccccc3)cc2)C1 ZINC000217884331 EJ In-Stock Unstable KCNQ2 50 39 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)/C=C/c3ccccc3)cc2)C1 ZINC000217884331 EJ In-Stock Unstable HDAC8 48 41 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)/C=C/c3ccccc3)cc2)C1 ZINC000217884331 EJ In-Stock Unstable HDAC1 23 41 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)/C=C/c3ccccc3)cc2)C1 ZINC000217884331 EJ In-Stock Unstable HDAC6 36 41 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)/C=C/c3ccccc3)cc2)C1 ZINC000217884331 EJ In-Stock Unstable BIRC8 49 31 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1N[C@@H](C)c1ccc(O)cc1O ZINC000217884394 CI For-Sale Unstable TRPM8 16 46 CC[C@@H]1CC[C@@H](O)[C@@H](N2CCC(CN3CCCC3)CC2)C1 ZINC000217884395 CF For-Sale Unstable SLC18A3 20 42 O=C(NCCn1ccc(-c2ccsc2)n1)c1ccc(F)c(F)c1 ZINC000217884414 EG In-Stock Unstable PLD2 40 40 C[C@H](NC(=O)/C=C/c1ccccc1)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217884416 EJ In-Stock Unstable KCNQ2 50 39 C[C@H](NC(=O)/C=C/c1ccccc1)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217884416 EJ In-Stock Unstable HDAC8 48 41 C[C@H](NC(=O)/C=C/c1ccccc1)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217884416 EJ In-Stock Unstable HDAC1 23 41 C[C@H](NC(=O)/C=C/c1ccccc1)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217884416 EJ In-Stock Unstable HDAC6 36 41 C[C@H](NC(=O)/C=C/c1ccccc1)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217884416 EJ In-Stock Unstable BIRC8 49 31 Cc1cccc(/C=C/NC(=O)N2CCC(Cc3ccccc3)CC2)c1 ZINC000217884422 EJ For-Sale Unstable GRIN2B 84 50 Cc1cccc(/C=C/NC(=O)N2CCC(Cc3ccccc3)CC2)c1 ZINC000217884422 EJ For-Sale Unstable SIGMAR1 21 52 Cc1cccc(/C=C/NC(=O)N2CCC(Cc3ccccc3)CC2)c1 ZINC000217884422 EJ For-Sale Unstable CCR3 59 41 C[C@@H](C(=O)O)c1ccc(CN2CC[C@@H](N(C)C)C2)cc1 ZINC000217884434 CE For-Sale Unstable HRH3 15 40 C[C@@H](C(=O)O)c1ccc(CN2CC[C@@H](N(C)C)C2)cc1 ZINC000217884434 CE For-Sale Unstable SIGMAR1 33 42 C[C@@H](C(=O)O)c1ccc(CN2CC[C@@H](N(C)C)C2)cc1 ZINC000217884434 CE For-Sale Unstable CCR5 47 42 C[C@@H](C(=O)O)c1ccc(CN2CC[C@@H](N(C)C)C2)cc1 ZINC000217884434 CE For-Sale Unstable MLNR 50 39 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1N[C@@H](C)c1ccc(O)cc1O ZINC000217884481 CI For-Sale Unstable TRPM8 16 46 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccc(F)cc1 ZINC000217884496 GF For-Sale Unstable COLA 88 38 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccc(F)cc1 ZINC000217884496 GF For-Sale Unstable CPT1A 76 38 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](N(C)C)C2)cc1 ZINC000217884519 CE For-Sale Unstable HRH3 15 40 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](N(C)C)C2)cc1 ZINC000217884519 CE For-Sale Unstable SIGMAR1 33 42 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](N(C)C)C2)cc1 ZINC000217884519 CE For-Sale Unstable CCR5 47 42 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](N(C)C)C2)cc1 ZINC000217884519 CE For-Sale Unstable MLNR 50 39 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccc(F)cc1 ZINC000217884557 GF For-Sale Unstable COLA 88 38 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccc(F)cc1 ZINC000217884557 GF For-Sale Unstable CPT1A 76 38 CC[C@@H]1CC[C@H](O)[C@@H](N2CCC(CN3CCCC3)CC2)C1 ZINC000217884561 CF For-Sale Unstable SLC18A3 20 42 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1N[C@@H](C)c1ccc(O)cc1O ZINC000217884577 CI For-Sale Unstable TRPM8 16 46 NCC1CCN(C(=O)OCc2cc(Cl)cc(Cl)c2)CC1 ZINC000217884589 DG For-Sale Unstable GRIN2B 24 45 NCC1CCN(C(=O)OCc2cc(Cl)cc(Cl)c2)CC1 ZINC000217884589 DG For-Sale Unstable CACNA1I 47 39 O=C(Cn1cncn1)N[C@@H]1CCC[C@@H]1CO ZINC000217884611 BB For-Sale Unstable HIS3 44 36 COc1ccc(CCNC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217884643 DH For-Sale Unstable NQO2 36 40 COc1ccc(CCNC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217884643 DH For-Sale Unstable CTSL 24 40 COc1ccc(CCNC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217884643 DH For-Sale Unstable MTNR1A 110 44 COc1ccc(CCNC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217884643 DH For-Sale Unstable MTNR1B 90 44 COc1ccc(CCNC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217884643 DH For-Sale Unstable NR1H4 31 40 COc1ccc(CCNC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217884643 DH For-Sale Unstable PTGDR 23 40 COc1ccc(CCNC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217884643 DH For-Sale Unstable ABCG2 16 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccc(F)cc1 ZINC000217884653 GF For-Sale Unstable COLA 88 38 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccc(F)cc1 ZINC000217884653 GF For-Sale Unstable CPT1A 76 38 CC(C)[C@H]1CC[C@H](C)C[C@@H]1N[C@@H](C)c1ccc(O)cc1O ZINC000217884656 CI For-Sale Unstable TRPM8 16 46 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccccc2OC)CC(=O)O4)cc1O ZINC000217884667 JI In-Stock Unstable AKR1B1 0 48 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccccc2OC)CC(=O)O4)cc1O ZINC000217884667 JI In-Stock Unstable CYP1B1 68 39 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccccc2OC)CC(=O)O4)cc1O ZINC000217884667 JI In-Stock Unstable CYP1A1 52 48 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccccc2OC)CC(=O)O4)cc1O ZINC000217884667 JI In-Stock Unstable CYP1A2 45 40 O=C(O)/C=C\c1cc(F)ccc1COc1cccc(F)c1 ZINC000217884680 CH For-Sale Unstable PTGER2 49 50 O=C(O)/C=C\c1cc(F)ccc1COc1cccc(F)c1 ZINC000217884680 CH For-Sale Unstable PTGER4 26 50 O=C(O)/C=C\c1cc(F)ccc1COc1cccc(F)c1 ZINC000217884680 CH For-Sale Unstable PTGER3 24 50 O=C(O)/C=C\c1cc(F)ccc1COc1cccc(F)c1 ZINC000217884680 CH For-Sale Unstable PTGDR 0 45 O=C(O)/C=C\c1cc(F)ccc1COc1cccc(F)c1 ZINC000217884680 CH For-Sale Unstable HCAR2 0 45 O=C(O)/C=C\c1cc(F)ccc1COc1cccc(F)c1 ZINC000217884680 CH For-Sale Unstable AKR1C3 24 41 Cc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)/C=C/c1ccccc1 ZINC000217884686 DI In-Stock Unstable HDAC8 49 35 Cc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)/C=C/c1ccccc1 ZINC000217884686 DI In-Stock Unstable MMP2 15 43 O=C(Cn1cncn1)N[C@H]1CCC[C@@H]1CO ZINC000217884696 BB For-Sale Unstable HIS3 44 36 C[C@H](C(=O)O)c1ccc(CN(C)[C@@H](C)CC#N)cc1 ZINC000217884711 CF For-Sale Unstable PTGS1 27 49 C[C@H](C(=O)O)c1ccc(CN(C)[C@@H](C)CC#N)cc1 ZINC000217884711 CF For-Sale Unstable PTGS2 0 49 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccccc2OC)CC(=O)O4)cc1O ZINC000217884730 JI In-Stock Unstable AKR1B1 0 48 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccccc2OC)CC(=O)O4)cc1O ZINC000217884730 JI In-Stock Unstable CYP1B1 68 39 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccccc2OC)CC(=O)O4)cc1O ZINC000217884730 JI In-Stock Unstable CYP1A1 52 48 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccccc2OC)CC(=O)O4)cc1O ZINC000217884730 JI In-Stock Unstable CYP1A2 45 40 CC1(C)[C@H]2CC[C@@]1(CS(=O)(=O)N1CCN(CCCc3nc(-c4cccs4)no3)CC1)C(=O)C2 ZINC000217884733 JG On-Demand Unstable CXCR3 19 47 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccc(F)cc1 ZINC000217884744 GF For-Sale Unstable COLA 88 38 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccc(F)cc1 ZINC000217884744 GF For-Sale Unstable CPT1A 76 38 Cc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)/C=C/c1ccccc1 ZINC000217884754 DI In-Stock Unstable HDAC8 49 35 Cc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)/C=C/c1ccccc1 ZINC000217884754 DI In-Stock Unstable MMP2 15 43 O=C(Cn1cncn1)N[C@@H]1CCC[C@H]1CO ZINC000217884757 BB For-Sale Unstable HIS3 44 36 C[C@@H]1CC[C@@H](O)[C@@H](N2CCC(CN3CCCC3)CC2)C1 ZINC000217884769 CE For-Sale Unstable SLC18A3 19 40 O=C(NCCn1ccc(-c2ccsc2)n1)c1cccc2ccccc12 ZINC000217884772 EI In-Stock Unstable POLR1A 62 37 O=C(O)/C=C\c1cc(COc2cccc(F)c2)ccc1F ZINC000217884783 CH For-Sale Unstable MAOB 31 40 O=C(O)/C=C\c1cc(COc2cccc(F)c2)ccc1F ZINC000217884783 CH For-Sale Unstable PTGER2 48 53 O=C(O)/C=C\c1cc(COc2cccc(F)c2)ccc1F ZINC000217884783 CH For-Sale Unstable PTGER4 28 53 O=C(O)/C=C\c1cc(COc2cccc(F)c2)ccc1F ZINC000217884783 CH For-Sale Unstable PTGER3 35 53 O=C(O)/C=C\c1cc(COc2cccc(F)c2)ccc1F ZINC000217884783 CH For-Sale Unstable CDC25B 22 40 O=C(O)/C=C\c1cc(COc2cccc(F)c2)ccc1F ZINC000217884783 CH For-Sale Unstable PTGDR 0 48 O=C(O)/C=C\c1cc(COc2cccc(F)c2)ccc1F ZINC000217884783 CH For-Sale Unstable HCAR2 0 48 O=C(O)/C=C\c1cc(COc2cccc(F)c2)ccc1F ZINC000217884783 CH For-Sale Unstable FFAR1 47 41 O=C(O)/C=C\c1cc(COc2cccc(F)c2)ccc1F ZINC000217884783 CH For-Sale Unstable AKR1C3 27 45 O=C(Cn1cncn1)N[C@H]1CCC[C@H]1CO ZINC000217884833 BB For-Sale Unstable HIS3 44 36 CC(C)S(=O)(=O)N[C@@H]1CCC[C@@H](C)[C@@H]1C ZINC000217884834 BE For-Sale Unstable GRIA4 34 46 COc1ccc2[nH]c3c(c2c1)CN(C(=O)c1csc(NCCC(C)C)n1)CC3 ZINC000217884848 GI In-Stock Unstable TRPC6 60 46 COc1ccc2[nH]c3c(c2c1)CN(C(=O)c1csc(NCCC(C)C)n1)CC3 ZINC000217884848 GI In-Stock Unstable TRPC3 28 41 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCc1cc(Cl)ccc1O ZINC000217884854 CJ For-Sale Unstable TRPM8 19 53 C[C@H](C(=O)O)c1ccc(CN2CCNC(=O)[C@@H]2C)cc1 ZINC000217884874 CD For-Sale Unstable SLC22A20 0 43 Cc1ccc2c(c1)nc(N)n2[C@H]1CCC[C@@H](C)[C@H]1C ZINC000217884877 CH For-Sale Unstable RPS6KB1 18 48 COc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217884879 CG For-Sale Unstable TSHR 55 33 COc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217884879 CG For-Sale Unstable PTGS2 0 45 COc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217884879 CG For-Sale Unstable OPRL1 0 41 COc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217884879 CG For-Sale Unstable PTGER2 24 49 COc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217884879 CG For-Sale Unstable PTGER4 45 49 COc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217884879 CG For-Sale Unstable PTGER3 34 67 COc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217884879 CG For-Sale Unstable LTB4R 35 40 COc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217884879 CG For-Sale Unstable CDC25B 22 41 COc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217884879 CG For-Sale Unstable GYS1 44 35 COc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217884879 CG For-Sale Unstable FFAR1 34 40 COc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217884879 CG For-Sale Unstable FFAR4 48 48 COc1ccc(OCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217884879 CG For-Sale Unstable GPR183 0 41 CC(C)S(=O)(=O)N[C@H]1CCC[C@@H](C)[C@@H]1C ZINC000217884922 BE For-Sale Unstable GRIA4 34 46 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCc1cc(Cl)ccc1O ZINC000217884943 CJ For-Sale Unstable TRPM8 19 53 COc1c(Cl)cc(F)cc1C[C@H](N)C(=O)O ZINC000217884944 BD For-Sale Unstable CACNA2D1 53 40 O=C(N[C@@H](CCn1cncn1)c1ccccc1)c1c[nH]c2ncnn2c1=O ZINC000217884950 FC In-Stock Unstable HIS3 48 35 O=C(N[C@@H](CCn1cncn1)c1ccccc1)c1c[nH]c2ncnn2c1=O ZINC000217884950 FC In-Stock Unstable CYP51 0 42 Cc1cccc(CCC(=O)N[C@@H]2CCC[C@@H]2CO)c1 ZINC000217884957 CE On-Demand Unstable LUXR 33 40 Cc1ccc2c(c1)nc(N)n2[C@H]1CCC[C@H](C)[C@H]1C ZINC000217884958 CH For-Sale Unstable RPS6KB1 18 48 C[C@@H]1CC[C@H](O)[C@@H](N2CCC(CN3CCCC3)CC2)C1 ZINC000217884961 CE For-Sale Unstable SLC18A3 19 40 CC(C)S(=O)(=O)N[C@@H]1CCC[C@H](C)[C@@H]1C ZINC000217885008 BE For-Sale Unstable GRIA4 34 46 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCc1cc(Cl)ccc1O ZINC000217885024 CJ For-Sale Unstable TRPM8 0 53 O=[N+]([O-])c1cccc(S(=O)(=O)N2CCCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217885026 HG On-Demand Unstable DRD4 18 40 O=[N+]([O-])c1cccc(S(=O)(=O)N2CCCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217885026 HG On-Demand Unstable ADORA2B 45 39 O=[N+]([O-])c1cccc(S(=O)(=O)N2CCCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217885026 HG On-Demand Unstable LSS 18 52 O=[N+]([O-])c1cccc(S(=O)(=O)N2CCCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217885026 HG On-Demand Unstable PKM 39 40 O=[N+]([O-])c1cccc(S(=O)(=O)N2CCCN(Cc3ccc(Cl)cc3)CC2)c1 ZINC000217885026 HG On-Demand Unstable CASP7 15 40 O=C(N[C@H](CCn1cncn1)c1ccccc1)c1c[nH]c2ncnn2c1=O ZINC000217885038 FC In-Stock Unstable HIS3 48 35 O=C(N[C@H](CCn1cncn1)c1ccccc1)c1c[nH]c2ncnn2c1=O ZINC000217885038 FC In-Stock Unstable CYP51 0 42 COc1c(Cl)cc(F)cc1C[C@@H](N)C(=O)O ZINC000217885040 BD For-Sale Unstable CACNA2D1 53 40 C[C@H](C(=O)O)c1ccc(CN2CCN(C)[C@@H](C)C2)cc1 ZINC000217885041 CE For-Sale Unstable DRD4 26 41 C[C@H](C(=O)O)c1ccc(CN2CCN(C)[C@@H](C)C2)cc1 ZINC000217885041 CE For-Sale Unstable PTGS1 23 45 C[C@H](C(=O)O)c1ccc(CN2CCN(C)[C@@H](C)C2)cc1 ZINC000217885041 CE For-Sale Unstable PTGS2 16 45 C[C@H](C(=O)O)c1ccc(CN2CCN(C)[C@@H](C)C2)cc1 ZINC000217885041 CE For-Sale Unstable MLNR 33 42 Cc1cccc(CCC(=O)N[C@H]2CCC[C@@H]2CO)c1 ZINC000217885042 CE For-Sale Unstable VIPR1 18 45 Cc1cccc(CCC(=O)N[C@H]2CCC[C@@H]2CO)c1 ZINC000217885042 CE For-Sale Unstable LUXR 33 40 Cc1ccc2c(c1)nc(N)n2[C@@H]1CCC[C@H](C)[C@H]1C ZINC000217885049 CH For-Sale Unstable RPS6KB1 18 48 Cc1cccc(/C=C/NC(=O)N[C@H](C)c2ccccc2)c1 ZINC000217885068 CI For-Sale Unstable KCNQ2 22 41 Cc1cccc(/C=C/NC(=O)N[C@H](C)c2ccccc2)c1 ZINC000217885068 CI For-Sale Unstable ACACA 27 41 CC(C)S(=O)(=O)N[C@H]1CCC[C@H](C)[C@@H]1C ZINC000217885100 BE For-Sale Unstable GRIA4 34 46 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCc1cc(Cl)ccc1O ZINC000217885105 CJ For-Sale Unstable TRPM8 19 53 Cc1cccc(CCC(=O)N[C@@H]2CCC[C@H]2CO)c1 ZINC000217885119 CE For-Sale Unstable VIPR1 18 45 Cc1cccc(CCC(=O)N[C@@H]2CCC[C@H]2CO)c1 ZINC000217885119 CE For-Sale Unstable LUXR 33 40 Cc1cccc(/C=C/NC(=O)N[C@@H](C)c2ccccc2)c1 ZINC000217885149 CI For-Sale Unstable ACACA 27 41 COc1ccc2cc(CNS(=O)(=O)c3cccc([N+](=O)[O-])c3)ccc2c1 ZINC000217885159 FG On-Demand Unstable CACNA1C 39 43 COc1ccc2cc(CNS(=O)(=O)c3cccc([N+](=O)[O-])c3)ccc2c1 ZINC000217885159 FG On-Demand Unstable MMP13 17 41 COc1ccc2cc(CNS(=O)(=O)c3cccc([N+](=O)[O-])c3)ccc2c1 ZINC000217885159 FG On-Demand Unstable NPY1R 19 41 COc1ccc2cc(CNS(=O)(=O)c3cccc([N+](=O)[O-])c3)ccc2c1 ZINC000217885159 FG On-Demand Unstable NPY2R 28 43 COc1ccc2cc(CNS(=O)(=O)c3cccc([N+](=O)[O-])c3)ccc2c1 ZINC000217885159 FG On-Demand Unstable CACNA1D 72 43 COc1ccc2cc(CNS(=O)(=O)c3cccc([N+](=O)[O-])c3)ccc2c1 ZINC000217885159 FG On-Demand Unstable MMP2 15 40 COc1ccc2cc(CNS(=O)(=O)c3cccc([N+](=O)[O-])c3)ccc2c1 ZINC000217885159 FG On-Demand Unstable MMP8 18 40 COc1ccc2cc(CNS(=O)(=O)c3cccc([N+](=O)[O-])c3)ccc2c1 ZINC000217885159 FG On-Demand Unstable ALOX15 21 45 COc1ccc2cc(CNS(=O)(=O)c3cccc([N+](=O)[O-])c3)ccc2c1 ZINC000217885159 FG On-Demand Unstable MMP9 21 40 COc1ccc2cc(CNS(=O)(=O)c3cccc([N+](=O)[O-])c3)ccc2c1 ZINC000217885159 FG On-Demand Unstable MMP1 19 40 COC(=O)C[C@H](c1cc2cc3c(cc2[nH]c1=O)OCCO3)c1c(O)c2ccccc2oc1=O ZINC000217885181 IF In-Stock Unstable NQO1 24 44 Cc1cccc(CCC(=O)N[C@H]2CCC[C@H]2CO)c1 ZINC000217885187 CE For-Sale Unstable VIPR1 18 45 Cc1cccc(CCC(=O)N[C@H]2CCC[C@H]2CO)c1 ZINC000217885187 CE For-Sale Unstable LUXR 33 40 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](C)CC2)cc1 ZINC000217885206 CG For-Sale Unstable ACHE 26 52 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](C)CC2)cc1 ZINC000217885206 CG For-Sale Unstable PTGS1 32 50 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](C)CC2)cc1 ZINC000217885206 CG For-Sale Unstable PTGS2 0 50 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](C)CC2)cc1 ZINC000217885206 CG For-Sale Unstable HRH3 28 55 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](C)CC2)cc1 ZINC000217885206 CG For-Sale Unstable SIGMAR1 45 39 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](C)CC2)cc1 ZINC000217885206 CG For-Sale Unstable MCHR1 23 40 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](C)CC2)cc1 ZINC000217885206 CG For-Sale Unstable SLC22A20 0 45 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1N[C@@H](C)c1cccc(O)c1 ZINC000217885211 CJ For-Sale Unstable TRPM8 17 45 C[C@]12CCC[C@@H]1[C@@H]2C=O ZINC000217885241 AD For-Sale Unstable UGT2B7 81 38 COC(=O)C[C@@H](c1cc2cc3c(cc2[nH]c1=O)OCCO3)c1c(O)c2ccccc2oc1=O ZINC000217885262 IF In-Stock Unstable NQO1 24 44 CO[C@@H](C(=O)NCc1ccc2nc(C)[nH]c2c1)c1ccccc1 ZINC000217885271 DF In-Stock Unstable TYMS 41 36 CC[C@@H](NC(=O)/C=C/c1ccccc1)c1ccc(C)c(C)c1 ZINC000217885283 CJ In-Stock Unstable KCNQ2 44 33 CC[C@@H](NC(=O)/C=C/c1ccccc1)c1ccc(C)c(C)c1 ZINC000217885283 CJ In-Stock Unstable HDAC8 59 36 CC[C@@H](NC(=O)/C=C/c1ccccc1)c1ccc(C)c(C)c1 ZINC000217885283 CJ In-Stock Unstable MMP2 19 46 CC[C@@H](NC(=O)/C=C/c1ccccc1)c1ccc(C)c(C)c1 ZINC000217885283 CJ In-Stock Unstable HDAC6 38 44 CC[C@@H](NC(=O)/C=C/c1ccccc1)c1ccc(C)c(C)c1 ZINC000217885283 CJ In-Stock Unstable MMP9 16 46 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1N[C@@H](C)c1cccc(O)c1 ZINC000217885293 CJ For-Sale Unstable TRPM8 17 45 C[C@@H]1CCCC[C@@H]1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217885295 CH For-Sale Unstable PTGER2 25 43 C[C@@H]1CCCC[C@@H]1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217885295 CH For-Sale Unstable HCAR2 0 40 C[C@@H]1CCCC[C@@H]1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217885295 CH For-Sale Unstable AKR1C3 31 40 COc1ccc(CNC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217885326 CG For-Sale Unstable MTNR1A 59 45 COc1ccc(CNC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217885326 CG For-Sale Unstable MTNR1B 56 45 COc1ccc(CNC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217885326 CG For-Sale Unstable NR1H4 37 41 COc1ccc(CNC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217885326 CG For-Sale Unstable U38 0 40 CO[C@H](C(=O)NCc1ccc2nc(C)[nH]c2c1)c1ccccc1 ZINC000217885350 DF In-Stock Unstable TYMS 41 36 CC[C@H](NC(=O)/C=C/c1ccccc1)c1ccc(C)c(C)c1 ZINC000217885358 CJ In-Stock Unstable KCNQ2 44 33 CC[C@H](NC(=O)/C=C/c1ccccc1)c1ccc(C)c(C)c1 ZINC000217885358 CJ In-Stock Unstable HDAC8 59 36 CC[C@H](NC(=O)/C=C/c1ccccc1)c1ccc(C)c(C)c1 ZINC000217885358 CJ In-Stock Unstable MMP2 19 46 CC[C@H](NC(=O)/C=C/c1ccccc1)c1ccc(C)c(C)c1 ZINC000217885358 CJ In-Stock Unstable HDAC6 38 44 CC[C@H](NC(=O)/C=C/c1ccccc1)c1ccc(C)c(C)c1 ZINC000217885358 CJ In-Stock Unstable MMP9 16 46 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1N[C@@H](C)c1cccc(O)c1 ZINC000217885385 CJ For-Sale Unstable TRPM8 17 45 C[C@H]1CCCC[C@@H]1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217885398 CH For-Sale Unstable PTGER2 25 43 C[C@H]1CCCC[C@@H]1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217885398 CH For-Sale Unstable HCAR2 0 40 C[C@H]1CCCC[C@@H]1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217885398 CH For-Sale Unstable AKR1C3 31 40 C[C@]12CCC[C@H]1[C@@H]2C=O ZINC000217885409 AD For-Sale Unstable UGT2B7 81 38 CC[C@@H](NC(=O)/C=C/c1ccccc1)c1ccc(C)cc1C ZINC000217885446 CJ In-Stock Unstable HDAC8 54 36 CC[C@@H](NC(=O)/C=C/c1ccccc1)c1ccc(C)cc1C ZINC000217885446 CJ In-Stock Unstable MMP2 18 48 CC[C@@H](NC(=O)/C=C/c1ccccc1)c1ccc(C)cc1C ZINC000217885446 CJ In-Stock Unstable HDAC6 36 43 CC[C@@H](NC(=O)/C=C/c1ccccc1)c1ccc(C)cc1C ZINC000217885446 CJ In-Stock Unstable MMP9 15 48 CC[C@@H](NC(=O)/C=C/c1ccccc1)c1ccc(C)cc1C ZINC000217885446 CJ In-Stock Unstable UL26 32 40 CC[C@@H](NC(=O)/C=C/c1ccccc1)c1ccc(C)cc1C ZINC000217885446 CJ In-Stock Unstable U53 0 40 CC[C@@H](NC(=O)/C=C/c1ccccc1)c1ccc(C)cc1C ZINC000217885446 CJ In-Stock Unstable SCAF_EBVB9 24 40 CC(C)[C@H]1CC[C@H](C)C[C@@H]1N[C@@H](C)c1cccc(O)c1 ZINC000217885475 CJ For-Sale Unstable TRPM8 17 45 C[C@H](C(=O)O)c1ccc(CN(C)C[C@@H]2C[C@@H]2C)cc1 ZINC000217885491 CF For-Sale Unstable PTGS1 29 49 C[C@H](C(=O)O)c1ccc(CN(C)C[C@@H]2C[C@@H]2C)cc1 ZINC000217885491 CF For-Sale Unstable PTGS2 0 49 CC[C@H](NC(=O)/C=C/c1ccccc1)c1ccc(C)cc1C ZINC000217885509 CJ In-Stock Unstable HDAC8 54 36 CC[C@H](NC(=O)/C=C/c1ccccc1)c1ccc(C)cc1C ZINC000217885509 CJ In-Stock Unstable MMP2 18 48 CC[C@H](NC(=O)/C=C/c1ccccc1)c1ccc(C)cc1C ZINC000217885509 CJ In-Stock Unstable HDAC6 36 43 CC[C@H](NC(=O)/C=C/c1ccccc1)c1ccc(C)cc1C ZINC000217885509 CJ In-Stock Unstable MMP9 15 48 CC[C@H](NC(=O)/C=C/c1ccccc1)c1ccc(C)cc1C ZINC000217885509 CJ In-Stock Unstable UL26 32 40 CC[C@H](NC(=O)/C=C/c1ccccc1)c1ccc(C)cc1C ZINC000217885509 CJ In-Stock Unstable U53 0 40 CC[C@H](NC(=O)/C=C/c1ccccc1)c1ccc(C)cc1C ZINC000217885509 CJ In-Stock Unstable SCAF_EBVB9 24 40 Cc1cccc(/C=C/NC(=O)NCc2ccc3c(c2)OCO3)c1 ZINC000217885521 DG For-Sale Unstable BMP1 33 44 Cc1cccc(/C=C/NC(=O)NCc2ccc3c(c2)OCO3)c1 ZINC000217885521 DG For-Sale Unstable NOS2 84 35 Cc1cccc(/C=C/NC(=O)NCc2ccc3c(c2)OCO3)c1 ZINC000217885521 DG For-Sale Unstable NR1H4 19 42 Cc1cccc(/C=C/NC(=O)NCc2ccc3c(c2)OCO3)c1 ZINC000217885521 DG For-Sale Unstable DYRK2 45 34 CC(=O)Nc1ccc(NC(=O)CCCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@H]23)cc1 ZINC000217885539 JI In-Stock Unstable TOP1 0 42 CC[C@@H](N[C@@H]1C[C@@H](C)CC[C@@H]1C(C)C)c1ccc(F)cc1 ZINC000217885591 CK For-Sale Unstable TRPM8 15 41 CC(=O)Nc1ccc(NC(=O)CCCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@@H]23)cc1 ZINC000217885608 JI In-Stock Unstable TOP1 0 42 CC[C@@H](NC(=O)/C=C/c1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217885616 EH In-Stock Unstable CYP1B1 19 46 CC[C@@H](NC(=O)/C=C/c1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217885616 EH In-Stock Unstable LTB4R 0 41 CC[C@@H](NC(=O)/C=C/c1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217885616 EH In-Stock Unstable HDAC8 44 43 CC[C@@H](NC(=O)/C=C/c1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217885616 EH In-Stock Unstable MMP2 20 50 CC[C@@H](NC(=O)/C=C/c1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217885616 EH In-Stock Unstable CYP1A1 19 46 CC[C@@H](NC(=O)/C=C/c1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217885616 EH In-Stock Unstable HDAC1 18 45 CC[C@@H](NC(=O)/C=C/c1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217885616 EH In-Stock Unstable HDAC2 16 42 CC[C@@H](NC(=O)/C=C/c1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217885616 EH In-Stock Unstable HDAC6 32 42 CC[C@@H](NC(=O)/C=C/c1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217885616 EH In-Stock Unstable MMP9 16 50 CC[C@@H](NC(=O)/C=C/c1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217885616 EH In-Stock Unstable ABCG2 19 44 Cc1cccc(/C=C/NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217885618 EE For-Sale Unstable CA2 100 50 Cc1cccc(/C=C/NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217885618 EE For-Sale Unstable CA6 15 41 Cc1cccc(/C=C/NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217885618 EE For-Sale Unstable CA1 96 50 Cc1cccc(/C=C/NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217885618 EE For-Sale Unstable CA7 42 41 Cc1cccc(/C=C/NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217885618 EE For-Sale Unstable CA5B 41 40 Cc1cccc(/C=C/NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217885618 EE For-Sale Unstable CA4 80 50 Cc1cccc(/C=C/NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217885618 EE For-Sale Unstable CA5A 47 40 Cc1cccc(/C=C/NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217885618 EE For-Sale Unstable CA14 36 43 Cc1cccc(/C=C/NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217885618 EE For-Sale Unstable CA12 77 55 Cc1cccc(/C=C/NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217885618 EE For-Sale Unstable CA9 84 55 Cc1cccc(/C=C/NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217885618 EE For-Sale Unstable UREA_CANEN 28 51 Cc1cccc(/C=C/NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217885618 EE For-Sale Unstable IDO1 34 47 Cc1cccc(/C=C/NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217885618 EE For-Sale Unstable CYNT 31 40 Cc1cccc(/C=C/NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217885618 EE For-Sale Unstable NCE103 54 42 Cc1cccc(/C=C/NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217885618 EE For-Sale Unstable MTCA1 60 55 Cc1cccc(/C=C/NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217885618 EE For-Sale Unstable P96878_MYCTU 75 55 CCN(C)C(=O)CNC(=O)c1cccc(OC)c1N ZINC000217885624 CC For-Sale Unstable KCNA3 40 38 CCN(C)C(=O)CNC(=O)c1cccc(OC)c1N ZINC000217885624 CC For-Sale Unstable HCN1 47 33 CCN(C)C(=O)CNC(=O)c1cccc(OC)c1N ZINC000217885624 CC For-Sale Unstable KCNK3 45 40 CCN(C)C(=O)CNC(=O)c1cccc(OC)c1N ZINC000217885624 CC For-Sale Unstable KCNK9 34 40 CCCCN1C[C@@H](O)C[C@@H]1CC(C)C ZINC000217885632 AE In-Stock Unstable GBA2 51 41 CCCCN1C[C@@H](O)C[C@@H]1CC(C)C ZINC000217885632 AE In-Stock Unstable P0504H10.9 0 41 CCCCN1C[C@@H](O)C[C@@H]1CC(C)C ZINC000217885632 AE In-Stock Unstable AGL 0 41 CCCCN1C[C@@H](O)C[C@@H]1CC(C)C ZINC000217885632 AE In-Stock Unstable SIS 0 41 C[C@H](C(=O)O)c1ccc(CN2CCSC[C@@H]2C)cc1 ZINC000217885667 CF For-Sale Unstable PTGS1 25 45 C[C@H](C(=O)O)c1ccc(CN2CCSC[C@@H]2C)cc1 ZINC000217885667 CF For-Sale Unstable PTGS2 0 45 CC[C@H](N[C@@H]1C[C@@H](C)CC[C@@H]1C(C)C)c1ccc(F)cc1 ZINC000217885684 CK For-Sale Unstable TRPM8 15 41 CC[C@H](NC(=O)/C=C/c1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217885700 EH In-Stock Unstable CYP1B1 19 46 CC[C@H](NC(=O)/C=C/c1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217885700 EH In-Stock Unstable LTB4R 0 41 CC[C@H](NC(=O)/C=C/c1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217885700 EH In-Stock Unstable HDAC8 44 43 CC[C@H](NC(=O)/C=C/c1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217885700 EH In-Stock Unstable MMP2 20 50 CC[C@H](NC(=O)/C=C/c1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217885700 EH In-Stock Unstable CYP1A1 19 46 CC[C@H](NC(=O)/C=C/c1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217885700 EH In-Stock Unstable HDAC1 18 45 CC[C@H](NC(=O)/C=C/c1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217885700 EH In-Stock Unstable HDAC2 16 42 CC[C@H](NC(=O)/C=C/c1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217885700 EH In-Stock Unstable HDAC6 32 42 CC[C@H](NC(=O)/C=C/c1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217885700 EH In-Stock Unstable MMP9 16 50 CC[C@H](NC(=O)/C=C/c1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217885700 EH In-Stock Unstable ABCG2 19 44 CCCCN1C[C@H](O)C[C@@H]1CC(C)C ZINC000217885702 AE In-Stock Unstable GBA2 51 41 CCCCN1C[C@H](O)C[C@@H]1CC(C)C ZINC000217885702 AE In-Stock Unstable P0504H10.9 0 41 CCCCN1C[C@H](O)C[C@@H]1CC(C)C ZINC000217885702 AE In-Stock Unstable AGL 0 41 CCCCN1C[C@H](O)C[C@@H]1CC(C)C ZINC000217885702 AE In-Stock Unstable SIS 0 41 COc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)NCCSc1ccccc1)C(=O)OC2 ZINC000217885728 JJ In-Stock Unstable IMPDH1 0 72 COc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)NCCSc1ccccc1)C(=O)OC2 ZINC000217885728 JJ In-Stock Unstable IMPDH2 0 72 Cc1cccc(/C=C/NC(=O)NCc2ccccc2)c1 ZINC000217885739 CG For-Sale Unstable ANPEP 28 46 Cc1cccc(/C=C/NC(=O)NCc2ccccc2)c1 ZINC000217885739 CG For-Sale Unstable HDAC6 32 40 Cc1cccc(/C=C/NC(=O)NCc2ccccc2)c1 ZINC000217885739 CG For-Sale Unstable AMP1_PLAFQ 41 35 Cc1cccc(/C=C/NC(=O)NCc2ccccc2)c1 ZINC000217885739 CG For-Sale Unstable PDS 44 43 CC[C@@H](N[C@H]1C[C@@H](C)CC[C@@H]1C(C)C)c1ccc(F)cc1 ZINC000217885749 CK For-Sale Unstable TRPM8 15 41 C[C@H]1CN(Cc2ccc([C@H](C)C(=O)O)cc2)C[C@@H](C)S1 ZINC000217885793 CG For-Sale Unstable PTGS1 32 50 C[C@H]1CN(Cc2ccc([C@H](C)C(=O)O)cc2)C[C@@H](C)S1 ZINC000217885793 CG For-Sale Unstable PTGS2 0 50 C[C@H]1CN(Cc2ccc([C@H](C)C(=O)O)cc2)C[C@@H](C)S1 ZINC000217885793 CG For-Sale Unstable MLNR 16 41 C[C@H]1CN(Cc2ccc([C@H](C)C(=O)O)cc2)C[C@@H](C)S1 ZINC000217885793 CG For-Sale Unstable SLC22A20 0 49 CC[C@@H](NC(=O)/C=C/c1ccccc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217885807 EG In-Stock Unstable PTGS2 21 40 CC[C@@H](NC(=O)/C=C/c1ccccc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217885807 EG In-Stock Unstable CTSF 49 35 CC[C@@H](NC(=O)/C=C/c1ccccc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217885807 EG In-Stock Unstable TACR3 43 39 CC[C@@H](NC(=O)/C=C/c1ccccc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217885807 EG In-Stock Unstable MMP2 18 41 CC[C@@H](NC(=O)/C=C/c1ccccc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217885807 EG In-Stock Unstable HDAC6 20 43 CC[C@H](N[C@H]1C[C@@H](C)CC[C@@H]1C(C)C)c1ccc(F)cc1 ZINC000217885820 CK For-Sale Unstable TRPM8 15 41 CC(C)[C@@H]1CN(c2cnc3cc(Cl)c(Cl)cc3n2)CCN1 ZINC000217885892 EG For-Sale Unstable PRKCQ 19 42 CC[C@H](NC(=O)/C=C/c1ccccc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217885898 EG In-Stock Unstable PTGS2 21 40 CC[C@H](NC(=O)/C=C/c1ccccc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217885898 EG In-Stock Unstable CTSF 49 35 CC[C@H](NC(=O)/C=C/c1ccccc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217885898 EG In-Stock Unstable TACR3 43 39 CC[C@H](NC(=O)/C=C/c1ccccc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217885898 EG In-Stock Unstable MMP2 18 41 CC[C@H](NC(=O)/C=C/c1ccccc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217885898 EG In-Stock Unstable HDAC6 20 43 CC(C)(C)OC(=O)N[C@@H]1CCN(C(=O)OCc2cc(Cl)cc(Cl)c2)C1 ZINC000217885944 GI For-Sale Unstable CACNA1I 48 35 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1N[C@@H]1COc2cc(O)ccc21 ZINC000217885953 CH For-Sale Unstable TRPM8 15 41 CC(C)[C@H]1CN(c2cnc3cc(Cl)c(Cl)cc3n2)CCN1 ZINC000217885966 EG For-Sale Unstable PRKCQ 19 42 O=C(O)/C=C\c1ccccc1COC1CCCCCC1 ZINC000217885982 CI For-Sale Unstable PTGER2 50 48 O=C(O)/C=C\c1ccccc1COC1CCCCCC1 ZINC000217885982 CI For-Sale Unstable PTGER4 24 48 O=C(O)/C=C\c1ccccc1COC1CCCCCC1 ZINC000217885982 CI For-Sale Unstable PTGER3 18 48 O=C(O)/C=C\c1ccccc1COC1CCCCCC1 ZINC000217885982 CI For-Sale Unstable PTGDR 0 44 CC[C@@H](NS(=O)(=O)c1ccccc1C(=O)OC)c1ccc(Cl)cc1 ZINC000217885987 FH On-Demand Unstable UTS2 42 33 COc1cc([C@@H](C)N2CCC[C@@H](C(C)C)CC2)ccc1O ZINC000217885997 CI For-Sale Unstable PNLIP 0 46 COc1cc([C@@H](C)N2CCC[C@@H](C(C)C)CC2)ccc1O ZINC000217885997 CI For-Sale Unstable N1L 0 47 COc1cc([C@@H](C)N2CCC[C@@H](C(C)C)CC2)ccc1O ZINC000217885997 CI For-Sale Unstable SLC22A3 0 43 C[C@H](C(=O)O)c1ccc(CN2CCCCC[C@@H]2C)cc1 ZINC000217886000 CH For-Sale Unstable PTGS1 26 50 C[C@H](C(=O)O)c1ccc(CN2CCCCC[C@@H]2C)cc1 ZINC000217886000 CH For-Sale Unstable PTGS2 0 50 C[C@H](C(=O)O)c1ccc(CN2CCCCC[C@@H]2C)cc1 ZINC000217886000 CH For-Sale Unstable HRH3 53 54 COC(=O)C[C@H](C1=C(O)C(=O)c2ccccc2C1=O)c1coc2ccccc2c1=O ZINC000217886011 HG In-Stock Unstable ALDH2 47 32 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccccc3)n2)c(OC)c1 ZINC000217886015 FG In-Stock Unstable HDAC8 40 38 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccccc3)n2)c(OC)c1 ZINC000217886015 FG In-Stock Unstable IMPDH2 0 44 CC[C@@H](O)c1cc2n(n1)CCCN(C(=O)Cc1ccc3c(c1)OCO3)C2 ZINC000217886031 FE In-Stock Unstable NOS2 48 35 CC[C@@H](O)c1cc2n(n1)CCCN(C(=O)Cc1ccc3c(c1)OCO3)C2 ZINC000217886031 FE In-Stock Unstable SSTR3 90 30 CC(C)(C)OC(=O)N[C@H]1CCN(C(=O)OCc2cc(Cl)cc(Cl)c2)C1 ZINC000217886035 GI For-Sale Unstable CACNA1I 48 35 Cc1cccc(/C=C/NC(=O)Nc2cccc3c(O)cccc23)c1 ZINC000217886036 DJ For-Sale Unstable MMP9 0 42 Cc1cccc(/C=C/NC(=O)Nc2cccc3c(O)cccc23)c1 ZINC000217886036 DJ For-Sale Unstable MMP1 0 42 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1N[C@@H]1COc2cc(O)ccc21 ZINC000217886039 CH For-Sale Unstable TRPM8 15 41 O=C(NCCn1ccc(-c2ccsc2)n1)c1cc(=O)c2ccccc2o1 ZINC000217886058 FG In-Stock Unstable BCHE 25 42 O=C(O)/C=C\c1ccc(COC2CCCCCC2)cc1 ZINC000217886063 CI For-Sale Unstable NR1H4 20 40 O=C(O)/C=C\c1ccc(COC2CCCCCC2)cc1 ZINC000217886063 CI For-Sale Unstable 17HSDCL 0 43 CC[C@H](NS(=O)(=O)c1ccccc1C(=O)OC)c1ccc(Cl)cc1 ZINC000217886070 FH On-Demand Unstable UTS2 42 33 COC(=O)C[C@@H](C1=C(O)C(=O)c2ccccc2C1=O)c1coc2ccccc2c1=O ZINC000217886084 HG In-Stock Unstable ALDH2 47 32 CC[C@H](O)c1cc2n(n1)CCCN(C(=O)Cc1ccc3c(c1)OCO3)C2 ZINC000217886115 FE In-Stock Unstable NOS2 48 35 CC[C@H](O)c1cc2n(n1)CCCN(C(=O)Cc1ccc3c(c1)OCO3)C2 ZINC000217886115 FE In-Stock Unstable SSTR3 90 30 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1N[C@@H]1COc2cc(O)ccc21 ZINC000217886118 CH For-Sale Unstable TRPM8 15 41 COc1ccc(CSc2nccn2C)cc1/C=C\C(=O)O ZINC000217886149 DF For-Sale Unstable PTGER2 26 41 COc1ccc(CSc2nccn2C)cc1/C=C\C(=O)O ZINC000217886149 DF For-Sale Unstable PTGER4 17 41 COc1ccc(CSc2nccn2C)cc1/C=C\C(=O)O ZINC000217886149 DF For-Sale Unstable LTB4R 34 41 Cc1cccc(/C=C/NC(=O)Nc2ccc(O)cc2C)c1 ZINC000217886153 CH For-Sale Unstable MMP2 0 49 Cc1cccc(/C=C/NC(=O)Nc2ccc(O)cc2C)c1 ZINC000217886153 CH For-Sale Unstable MMP9 0 49 Cc1cccc(/C=C/NC(=O)Nc2ccc(O)cc2C)c1 ZINC000217886153 CH For-Sale Unstable MMP1 0 49 O=C(/C=C/c1ccccc1)NCc1nc(-c2cccc(Br)c2)no1 ZINC000217886155 GH In-Stock Unstable HDAC8 62 39 O=C(/C=C/c1ccccc1)NCc1nc(-c2cccc(Br)c2)no1 ZINC000217886155 GH In-Stock Unstable HDAC2 16 40 O=C(/C=C/c1ccccc1)NCc1nc(-c2cccc(Br)c2)no1 ZINC000217886155 GH In-Stock Unstable HDAC6 52 40 O=C(/C=C/c1ccccc1)NCc1nc(-c2cccc(Br)c2)no1 ZINC000217886155 GH In-Stock Unstable HPSE 26 40 CC(C)[C@H]1CC[C@H](C)C[C@@H]1N[C@@H]1COc2cc(O)ccc21 ZINC000217886183 CH For-Sale Unstable TRPM8 15 41 COC(=O)C[C@@H](C1=C(O)C(=O)c2ccccc2C1=O)C(C)C ZINC000217886196 DF In-Stock Unstable KCNA5 33 45 COC[C@@H]1CCN(Cc2ccc([C@@H](C)C(=O)O)cc2)C1 ZINC000217886201 CE For-Sale Unstable DRD4 33 41 COC[C@@H]1CCN(Cc2ccc([C@@H](C)C(=O)O)cc2)C1 ZINC000217886201 CE For-Sale Unstable SLC6A3 19 46 COC[C@@H]1CCN(Cc2ccc([C@@H](C)C(=O)O)cc2)C1 ZINC000217886201 CE For-Sale Unstable HTR4 31 49 COC[C@@H]1CCN(Cc2ccc([C@@H](C)C(=O)O)cc2)C1 ZINC000217886201 CE For-Sale Unstable SIGMAR1 46 43 COc1ccc(CN2CCCN(S(=O)(=O)c3cccc([N+](=O)[O-])c3)CC2)cc1 ZINC000217886207 HF On-Demand Unstable AVPR1B 40 34 COc1ccc(CN2CCCN(S(=O)(=O)c3cccc([N+](=O)[O-])c3)CC2)cc1 ZINC000217886207 HF On-Demand Unstable ADORA2B 46 42 COc1ccc(CN2CCCN(S(=O)(=O)c3cccc([N+](=O)[O-])c3)CC2)cc1 ZINC000217886207 HF On-Demand Unstable CASP3 0 46 COc1ccc(CN2CCCN(S(=O)(=O)c3cccc([N+](=O)[O-])c3)CC2)cc1 ZINC000217886207 HF On-Demand Unstable SIGMAR1 20 45 COc1ccc(CN2CCCN(S(=O)(=O)c3cccc([N+](=O)[O-])c3)CC2)cc1 ZINC000217886207 HF On-Demand Unstable MMP13 27 40 COc1ccc(CN2CCCN(S(=O)(=O)c3cccc([N+](=O)[O-])c3)CC2)cc1 ZINC000217886207 HF On-Demand Unstable ADAM17 20 40 COc1ccc(CN2CCCN(S(=O)(=O)c3cccc([N+](=O)[O-])c3)CC2)cc1 ZINC000217886207 HF On-Demand Unstable MMP9 28 40 COc1ccc(CN2CCCN(S(=O)(=O)c3cccc([N+](=O)[O-])c3)CC2)cc1 ZINC000217886207 HF On-Demand Unstable PKM 33 46 COc1ccc(CN2CCCN(S(=O)(=O)c3cccc([N+](=O)[O-])c3)CC2)cc1 ZINC000217886207 HF On-Demand Unstable CASP7 24 46 COc1ccc(CN2CCCN(S(=O)(=O)c3cccc([N+](=O)[O-])c3)CC2)cc1 ZINC000217886207 HF On-Demand Unstable MMP1 26 42 COc1ccc(CN2CCCN(S(=O)(=O)c3cccc([N+](=O)[O-])c3)CC2)cc1 ZINC000217886207 HF On-Demand Unstable MGLL 0 52 COc1ccc(CN2CCCN(S(=O)(=O)c3cccc([N+](=O)[O-])c3)CC2)cc1 ZINC000217886207 HF On-Demand Unstable ABHD6 0 52 O[C@H]1CN(c2ccc3ccccc3n2)CCN(C2CCOCC2)C1 ZINC000217886234 ED In-Stock Unstable HTR3A 22 42 O[C@H]1CN(c2ccc3ccccc3n2)CCN(C2CCOCC2)C1 ZINC000217886234 ED In-Stock Unstable PDE1B 0 40 O[C@H]1CN(c2ccc3ccccc3n2)CCN(C2CCOCC2)C1 ZINC000217886234 ED In-Stock Unstable SORD 17 42 COc1ccc(-c2noc(CN(C)C(=O)/C=C/c3ccccc3)n2)c(OC)c1 ZINC000217886262 GG In-Stock Unstable ABCG2 17 41 COC(=O)C[C@H](C1=C(O)C(=O)c2ccccc2C1=O)C(C)C ZINC000217886289 DF In-Stock Unstable KCNA5 33 45 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc(F)cc1Cl ZINC000217886313 GG For-Sale Unstable HCRTR2 42 34 CCc1ccccc1NC(=O)Cl ZINC000217886318 AG For-Sale Unstable CXCL8 56 41 CCc1ccccc1NC(=O)Cl ZINC000217886318 AG For-Sale Unstable KCNQ2 54 36 O=C(O)/C=C\c1cc(CSc2ccc(F)cc2)ccc1F ZINC000217886333 DI For-Sale Unstable PTGDR 0 42 Cc1ccc(S(=O)(=O)N2CCC(NS(=O)(=O)c3cccc(C)c3)CC2)cc1 ZINC000217886354 HE On-Demand Unstable ADRA1D 23 40 Cc1ccc(S(=O)(=O)N2CCC(NS(=O)(=O)c3cccc(C)c3)CC2)cc1 ZINC000217886354 HE On-Demand Unstable ADRA1A 16 40 Cc1ccc(S(=O)(=O)N2CCC(NS(=O)(=O)c3cccc(C)c3)CC2)cc1 ZINC000217886354 HE On-Demand Unstable ADRA1B 30 40 Cc1ccc(S(=O)(=O)N2CCC(NS(=O)(=O)c3cccc(C)c3)CC2)cc1 ZINC000217886354 HE On-Demand Unstable DCK 19 42 Cc1ccc(S(=O)(=O)N2CCC(NS(=O)(=O)c3cccc(C)c3)CC2)cc1 ZINC000217886354 HE On-Demand Unstable EPHX2 30 49 Cc1ccc(S(=O)(=O)N2CCC(NS(=O)(=O)c3cccc(C)c3)CC2)cc1 ZINC000217886354 HE On-Demand Unstable TGM2 47 36 Cc1ccc(S(=O)(=O)N2CCC(NS(=O)(=O)c3cccc(C)c3)CC2)cc1 ZINC000217886354 HE On-Demand Unstable CCR8 54 37 Cc1ccc(S(=O)(=O)N2CCC(NS(=O)(=O)c3cccc(C)c3)CC2)cc1 ZINC000217886354 HE On-Demand Unstable SFRP1 131 51 Cc1ccc(S(=O)(=O)N2CCC(NS(=O)(=O)c3cccc(C)c3)CC2)cc1 ZINC000217886354 HE On-Demand Unstable WNT3 84 35 CN(Cc1nc(-c2cccc(Br)c2)no1)C(=O)/C=C/c1ccccc1 ZINC000217886368 GI In-Stock Unstable FABI 42 32 CN(Cc1nc(-c2cccc(Br)c2)no1)C(=O)/C=C/c1ccccc1 ZINC000217886368 GI In-Stock Unstable HDAC8 46 35 CCC[C@H](O)CNCC(=O)N[C@H](C)CCC ZINC000217886382 BD For-Sale Unstable NOD1 42 35 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc(F)cc1Cl ZINC000217886393 GG For-Sale Unstable HCRTR2 42 34 CCN(C)C(=O)CNC(=O)c1cc2cccc(N)c2[nH]1 ZINC000217886417 CC For-Sale Unstable PYGL 52 46 COc1ccc(SCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217886422 DI For-Sale Unstable PTGER2 61 63 COc1ccc(SCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217886422 DI For-Sale Unstable PTGER4 29 43 COc1ccc(SCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217886422 DI For-Sale Unstable PTGER3 28 63 COc1ccc(SCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217886422 DI For-Sale Unstable LTB4R 27 48 COc1ccc(SCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217886422 DI For-Sale Unstable PTGDR 0 53 COc1ccc(SCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217886422 DI For-Sale Unstable GPR88 0 41 Cc1cc(C)cc(COC(=O)N2CCC(NC(=O)OC(C)(C)C)CC2)c1 ZINC000217886444 FH For-Sale Unstable GRIN2B 17 47 Cc1cc(C)cc(COC(=O)N2CCC(NC(=O)OC(C)(C)C)CC2)c1 ZINC000217886444 FH For-Sale Unstable F13A1 40 38 Cc1cc(C)cc(COC(=O)N2CCC(NC(=O)OC(C)(C)C)CC2)c1 ZINC000217886444 FH For-Sale Unstable GPR119 37 43 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H]3CCC[C@@H]32)cc1 ZINC000217886449 CH For-Sale Unstable PTGS1 28 53 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H]3CCC[C@@H]32)cc1 ZINC000217886449 CH For-Sale Unstable PTGS2 0 53 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H]3CCC[C@@H]32)cc1 ZINC000217886449 CH For-Sale Unstable SLC18A3 20 41 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H]3CCC[C@@H]32)cc1 ZINC000217886449 CH For-Sale Unstable FAAH 0 40 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H]3CCC[C@@H]32)cc1 ZINC000217886449 CH For-Sale Unstable BIRC2 41 32 CCC[C@H](O)CNCC(=O)N[C@@H](C)CCC ZINC000217886462 BD For-Sale Unstable NOD1 42 35 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc(F)cc1Cl ZINC000217886479 GG For-Sale Unstable HCRTR2 42 34 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217886495 DJ In-Stock Unstable DRD3 15 46 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217886495 DJ In-Stock Unstable SDH1 0 44 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217886495 DJ In-Stock Unstable PYGL 0 44 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217886495 DJ In-Stock Unstable HDAC8 54 37 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217886495 DJ In-Stock Unstable MMP2 26 63 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217886495 DJ In-Stock Unstable NR1H4 15 42 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217886495 DJ In-Stock Unstable HDAC1 35 45 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217886495 DJ In-Stock Unstable HDAC2 22 45 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217886495 DJ In-Stock Unstable HDAC3 18 45 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217886495 DJ In-Stock Unstable HDAC4 32 45 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217886495 DJ In-Stock Unstable HDAC6 36 44 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217886495 DJ In-Stock Unstable MMP9 20 63 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217886495 DJ In-Stock Unstable HDAC9 48 45 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217886495 DJ In-Stock Unstable HDAC7 54 45 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217886495 DJ In-Stock Unstable MMP1 0 40 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217886495 DJ In-Stock Unstable AMP1_PLAFQ 36 46 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217886495 DJ In-Stock Unstable HDA106 0 41 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccccc2)cc1 ZINC000217886495 DJ In-Stock Unstable TRPM2 0 46 COc1ccc(SCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217886501 DI For-Sale Unstable PTGS2 0 47 COc1ccc(SCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217886501 DI For-Sale Unstable PTGER2 26 52 COc1ccc(SCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217886501 DI For-Sale Unstable PTGER4 0 52 COc1ccc(SCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217886501 DI For-Sale Unstable PTGER3 15 52 COc1ccc(SCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217886501 DI For-Sale Unstable LTB4R 33 49 COc1ccc(SCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217886501 DI For-Sale Unstable GPR183 0 45 CC(C)NC(=O)COc1ccc2c(c1)O/C(=C/c1cn(C)c3ccccc13)C2=O ZINC000217886526 GH In-Stock Unstable MTOR 0 49 CC(C)NC(=O)COc1ccc2c(c1)O/C(=C/c1cn(C)c3ccccc13)C2=O ZINC000217886526 GH In-Stock Unstable RASGRP3 0 42 CCC[C@@H](O)CNCC(=O)N[C@H](C)CCC ZINC000217886548 BD For-Sale Unstable NOD1 42 35 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc(F)cc1Cl ZINC000217886561 GG For-Sale Unstable HCRTR2 42 34 CC(C)(C)OC(=O)N1CCC(NC(=O)OCc2cc(Cl)cc(Cl)c2)CC1 ZINC000217886566 HJ For-Sale Unstable EPHX2 26 45 CC(C)(C)OC(=O)N1CCC(NC(=O)OCc2cc(Cl)cc(Cl)c2)CC1 ZINC000217886566 HJ For-Sale Unstable CACNA1I 56 36 CC(C)(C)OC(=O)N1CCC(NC(=O)OCc2cc(Cl)cc(Cl)c2)CC1 ZINC000217886566 HJ For-Sale Unstable GPR119 49 44 CN(CCCNC(=O)/C=C/c1ccccc1)c1ccccc1 ZINC000217886609 CG In-Stock Unstable DRD3 15 47 CN(CCCNC(=O)/C=C/c1ccccc1)c1ccccc1 ZINC000217886609 CG In-Stock Unstable PYGL 24 45 CN(CCCNC(=O)/C=C/c1ccccc1)c1ccccc1 ZINC000217886609 CG In-Stock Unstable HDAC8 44 36 CN(CCCNC(=O)/C=C/c1ccccc1)c1ccccc1 ZINC000217886609 CG In-Stock Unstable MMP2 21 57 CN(CCCNC(=O)/C=C/c1ccccc1)c1ccccc1 ZINC000217886609 CG In-Stock Unstable NR1H4 17 45 CN(CCCNC(=O)/C=C/c1ccccc1)c1ccccc1 ZINC000217886609 CG In-Stock Unstable HDAC1 24 43 CN(CCCNC(=O)/C=C/c1ccccc1)c1ccccc1 ZINC000217886609 CG In-Stock Unstable HDAC2 25 49 CN(CCCNC(=O)/C=C/c1ccccc1)c1ccccc1 ZINC000217886609 CG In-Stock Unstable HDAC3 16 49 CN(CCCNC(=O)/C=C/c1ccccc1)c1ccccc1 ZINC000217886609 CG In-Stock Unstable HDAC4 25 49 CN(CCCNC(=O)/C=C/c1ccccc1)c1ccccc1 ZINC000217886609 CG In-Stock Unstable HDAC6 35 49 CN(CCCNC(=O)/C=C/c1ccccc1)c1ccccc1 ZINC000217886609 CG In-Stock Unstable MMP9 18 57 CN(CCCNC(=O)/C=C/c1ccccc1)c1ccccc1 ZINC000217886609 CG In-Stock Unstable HDAC9 43 49 CN(CCCNC(=O)/C=C/c1ccccc1)c1ccccc1 ZINC000217886609 CG In-Stock Unstable HDAC7 55 49 CN(CCCNC(=O)/C=C/c1ccccc1)c1ccccc1 ZINC000217886609 CG In-Stock Unstable MMP1 0 42 CCC[C@H](C)NC(=O)CNC[C@H](O)CCC ZINC000217886626 BD For-Sale Unstable NOD1 42 35 O=C(CNC(=O)c1ccccc1)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217886632 ED In-Stock Unstable SLC6A1 77 37 O=C(CNC(=O)c1ccccc1)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217886632 ED In-Stock Unstable VACHT_TETCF 0 48 O=C(CNC(=O)c1ccccc1)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217886632 ED In-Stock Unstable SLC18A3 45 35 O=C(CNC(=O)c1ccccc1)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217886632 ED In-Stock Unstable PREP 28 50 O=C(CNC(=O)c1ccccc1)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217886632 ED In-Stock Unstable CCR2 32 46 O=C(CNC(=O)c1ccccc1)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217886632 ED In-Stock Unstable FAP 0 50 Cc1cccc(/C=C/NC(=O)NCCCCCC(=O)O)c1 ZINC000217886678 CF For-Sale Unstable FBP1 24 49 Cc1cccc(/C=C/NC(=O)NCCCCCC(=O)O)c1 ZINC000217886678 CF For-Sale Unstable EPHX2 0 41 Cc1cccc(/C=C/NC(=O)NCCCCCC(=O)O)c1 ZINC000217886678 CF For-Sale Unstable HDAC9 35 45 Cc1cccc(/C=C/NC(=O)NCCCCCC(=O)O)c1 ZINC000217886678 CF For-Sale Unstable HDAC7 33 45 CC(C)(C)OC(=O)NC1CCN(C(=O)COc2cc(Cl)cc(Cl)c2)CC1 ZINC000217886684 HH On-Demand Unstable EPHX2 24 47 CC(C)(C)OC(=O)NC1CCN(C(=O)COc2cc(Cl)cc(Cl)c2)CC1 ZINC000217886684 HH On-Demand Unstable CACNA1I 60 38 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1N[C@@H](C)c1ccccc1O ZINC000217886686 CJ For-Sale Unstable TRPM8 20 50 CN(C)CCNC(=O)c1cc(-c2ccccc2)nc2c1cnn2Cc1ccccc1 ZINC000217886710 GG On-Demand Unstable ACACB 20 41 CN(C)CCNC(=O)c1cc(-c2ccccc2)nc2c1cnn2Cc1ccccc1 ZINC000217886710 GG On-Demand Unstable TACR3 21 47 CN(C)CCNC(=O)c1cc(-c2ccccc2)nc2c1cnn2Cc1ccccc1 ZINC000217886710 GG On-Demand Unstable POLR1A 40 42 O=C(/C=C/c1ccccc1)NCCCN1CCCc2ccccc21 ZINC000217886723 DH In-Stock Unstable DRD3 23 52 O=C(/C=C/c1ccccc1)NCCCN1CCCc2ccccc21 ZINC000217886723 DH In-Stock Unstable PYGL 24 44 O=C(/C=C/c1ccccc1)NCCCN1CCCc2ccccc21 ZINC000217886723 DH In-Stock Unstable HDAC6 28 40 CCC[C@@H](O)CNC[C@@H](O)c1ccccc1 ZINC000217886727 BD On-Demand Unstable ADRB2 19 44 CCC[C@@H](O)CNC[C@@H](O)c1ccccc1 ZINC000217886727 BD On-Demand Unstable AOC3 20 50 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1N[C@@H](C)c1ccccc1O ZINC000217886755 CJ For-Sale Unstable TRPM8 20 50 CCOC(=O)c1csc(NC(=O)CNc2ccc3c(cc2=O)[C@@H](NC(C)=O)CCc2cc(OC)c(OC)c(OC)c2-3)n1 ZINC000217886762 KH In-Stock Unstable TUBA1A 17 60 CCOC(=O)c1csc(NC(=O)CNc2ccc3c(cc2=O)[C@@H](NC(C)=O)CCc2cc(OC)c(OC)c(OC)c2-3)n1 ZINC000217886762 KH In-Stock Unstable TPPP 0 57 C[C@@H](C(=O)O)c1ccc(CN2CCC[C@@H](N(C)C)C2)cc1 ZINC000217886766 CE For-Sale Unstable SLC6A1 42 32 C[C@@H](C(=O)O)c1ccc(CN2CCC[C@@H](N(C)C)C2)cc1 ZINC000217886766 CE For-Sale Unstable HRH3 18 41 C[C@@H](C(=O)O)c1ccc(CN2CCC[C@@H](N(C)C)C2)cc1 ZINC000217886766 CE For-Sale Unstable SIGMAR1 23 40 CCC[C@H](O)CNC[C@@H](O)c1ccccc1 ZINC000217886813 BD On-Demand Unstable ADRB2 19 44 CCC[C@H](O)CNC[C@@H](O)c1ccccc1 ZINC000217886813 BD On-Demand Unstable AOC3 20 50 CN(C)CCNC(=O)[C@@H]1CCCN(S(=O)(=O)c2ccc(Br)cc2)C1 ZINC000217886821 HD On-Demand Unstable MMP13 29 41 CN(C)CCNC(=O)[C@@H]1CCCN(S(=O)(=O)c2ccc(Br)cc2)C1 ZINC000217886821 HD On-Demand Unstable EPHX2 17 47 CN(C)CCNC(=O)[C@@H]1CCCN(S(=O)(=O)c2ccc(Br)cc2)C1 ZINC000217886821 HD On-Demand Unstable MMP7 41 36 CN(C)CCNC(=O)[C@@H]1CCCN(S(=O)(=O)c2ccc(Br)cc2)C1 ZINC000217886821 HD On-Demand Unstable MMP1 31 41 CN(C)CCNC(=O)[C@@H]1CCCN(S(=O)(=O)c2ccc(Br)cc2)C1 ZINC000217886821 HD On-Demand Unstable GPBAR1 16 43 CN(C)CCNC(=O)[C@@H]1CCCN(S(=O)(=O)c2ccc(Br)cc2)C1 ZINC000217886821 HD On-Demand Unstable AKR1C1 22 44 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1N[C@@H](C)c1ccccc1O ZINC000217886834 CJ For-Sale Unstable TRPM8 20 50 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](N(C)C)C2)cc1 ZINC000217886850 CE For-Sale Unstable SLC6A1 42 32 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](N(C)C)C2)cc1 ZINC000217886850 CE For-Sale Unstable HRH3 18 41 C[C@H](C(=O)O)c1ccc(CN2CCC[C@@H](N(C)C)C2)cc1 ZINC000217886850 CE For-Sale Unstable SIGMAR1 23 40 COc1ccc(CNC(=O)/C=C/c2cccc([N+](=O)[O-])c2)c(OC)c1OC ZINC000217886852 FF In-Stock Unstable TRPM8 20 59 CCC[C@@H](O)CNC[C@H](O)c1ccccc1 ZINC000217886883 BD On-Demand Unstable ADRB2 19 44 CCC[C@@H](O)CNC[C@H](O)c1ccccc1 ZINC000217886883 BD On-Demand Unstable AOC3 20 50 COc1ccc(/C=C\C(=O)O)cc1CSc1nccs1 ZINC000217886901 DH For-Sale Unstable AKR1C3 40 40 CN(C)CCNC(=O)[C@H]1CCCN(S(=O)(=O)c2ccc(Br)cc2)C1 ZINC000217886906 HD On-Demand Unstable MMP13 29 41 CN(C)CCNC(=O)[C@H]1CCCN(S(=O)(=O)c2ccc(Br)cc2)C1 ZINC000217886906 HD On-Demand Unstable EPHX2 17 47 CN(C)CCNC(=O)[C@H]1CCCN(S(=O)(=O)c2ccc(Br)cc2)C1 ZINC000217886906 HD On-Demand Unstable MMP7 41 36 CN(C)CCNC(=O)[C@H]1CCCN(S(=O)(=O)c2ccc(Br)cc2)C1 ZINC000217886906 HD On-Demand Unstable MMP1 31 41 CN(C)CCNC(=O)[C@H]1CCCN(S(=O)(=O)c2ccc(Br)cc2)C1 ZINC000217886906 HD On-Demand Unstable GPBAR1 16 43 CN(C)CCNC(=O)[C@H]1CCCN(S(=O)(=O)c2ccc(Br)cc2)C1 ZINC000217886906 HD On-Demand Unstable AKR1C1 22 44 CC(C)[C@H]1CC[C@H](C)C[C@@H]1N[C@@H](C)c1ccccc1O ZINC000217886917 CJ For-Sale Unstable TRPM8 20 50 CCC[C@H](O)CNC[C@H](O)c1ccccc1 ZINC000217886947 BD On-Demand Unstable ADRB2 19 44 CCC[C@H](O)CNC[C@H](O)c1ccccc1 ZINC000217886947 BD On-Demand Unstable AOC3 20 50 O=C(NCCn1ccc(-c2ccsc2)n1)c1cnc2ccccc2n1 ZINC000217886971 EF In-Stock Unstable CCR1 40 34 CCOc1ccc(CNC(=O)/C=C/c2cccc([N+](=O)[O-])c2)cc1OCC ZINC000217886974 FH In-Stock Unstable CACNA1C 46 36 CCOc1ccc(CNC(=O)/C=C/c2cccc([N+](=O)[O-])c2)cc1OCC ZINC000217886974 FH In-Stock Unstable CACNA1D 80 36 CCOc1ccc(CNC(=O)/C=C/c2cccc([N+](=O)[O-])c2)cc1OCC ZINC000217886974 FH In-Stock Unstable TRPM8 0 52 Cc1cccc(/C=C/NC(=O)NCCCC(=O)O)c1 ZINC000217886981 CE For-Sale Unstable FBP1 16 45 CC[C@@H](C)N(C)CCNCc1cc(OC)c(O)c(OC)c1 ZINC000217886982 CE On-Demand Unstable SLC6A13 0 41 C[C@H](C(=O)O)c1ccc(CN2CC(=O)NC(=O)[C@@H]2C)cc1 ZINC000217886986 CC For-Sale Unstable PTGS1 0 43 C[C@H](C(=O)O)c1ccc(CN2CC(=O)NC(=O)[C@@H]2C)cc1 ZINC000217886986 CC For-Sale Unstable SLC22A20 0 43 COc1ccc(CSc2nccs2)cc1/C=C\C(=O)O ZINC000217887006 DH For-Sale Unstable PTGER2 32 42 COc1ccc(CSc2nccs2)cc1/C=C\C(=O)O ZINC000217887006 DH For-Sale Unstable PTGER4 0 42 COc1ccc(CSc2nccs2)cc1/C=C\C(=O)O ZINC000217887006 DH For-Sale Unstable PTGER3 16 42 COc1ccc(CSc2nccs2)cc1/C=C\C(=O)O ZINC000217887006 DH For-Sale Unstable LTB4R 34 40 COc1ccc(CSc2nccs2)cc1/C=C\C(=O)O ZINC000217887006 DH For-Sale Unstable TNFRSF1A 32 41 Cc1nc(CN[C@H]2C[C@H](C)CC[C@H]2C(C)C)cs1 ZINC000217887016 CI For-Sale Unstable TRPM8 0 41 O=C(O)CCC1CCN(C(=O)OCc2cc(Cl)cc(Cl)c2)CC1 ZINC000217887021 FI For-Sale Unstable GRIN2B 29 46 O=C(O)CCC1CCN(C(=O)OCc2cc(Cl)cc(Cl)c2)CC1 ZINC000217887021 FI For-Sale Unstable CACNA1I 57 41 CC[C@H](C)N(C)CCNCc1cc(OC)c(O)c(OC)c1 ZINC000217887028 CE On-Demand Unstable SLC6A13 0 41 COc1cc(CNC(=O)/C=C/c2cccc([N+](=O)[O-])c2)ccc1OC(C)C ZINC000217887060 FH In-Stock Unstable CACNA1C 40 35 COc1cc(CNC(=O)/C=C/c2cccc([N+](=O)[O-])c2)ccc1OC(C)C ZINC000217887060 FH In-Stock Unstable CACNA1D 76 35 COc1cc(CNC(=O)/C=C/c2cccc([N+](=O)[O-])c2)ccc1OC(C)C ZINC000217887060 FH In-Stock Unstable TRPM8 0 56 Cc1cccc(/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O)c1 ZINC000217887066 CF For-Sale Unstable FOLH1 57 40 Cc1cccc(/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O)c1 ZINC000217887066 CF For-Sale Unstable MME 20 43 Cc1cccc(/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O)c1 ZINC000217887066 CF For-Sale Unstable ANPEP 33 50 Cc1cccc(/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O)c1 ZINC000217887066 CF For-Sale Unstable FPR1 72 48 COc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217887091 CG For-Sale Unstable ALOX5 19 58 COc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217887091 CG For-Sale Unstable MAOB 24 70 COc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217887091 CG For-Sale Unstable PTGS2 0 54 COc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217887091 CG For-Sale Unstable PPARG 15 42 COc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217887091 CG For-Sale Unstable PTGER2 50 52 COc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217887091 CG For-Sale Unstable LTA4H 19 41 COc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217887091 CG For-Sale Unstable PTGER4 25 44 COc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217887091 CG For-Sale Unstable CYP1B1 32 45 COc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217887091 CG For-Sale Unstable PTPN2 0 46 COc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217887091 CG For-Sale Unstable PTGER3 21 52 COc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217887091 CG For-Sale Unstable LTB4R 33 42 COc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217887091 CG For-Sale Unstable AHR 32 41 COc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217887091 CG For-Sale Unstable HDAC8 15 49 COc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217887091 CG For-Sale Unstable PPARD 16 41 COc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217887091 CG For-Sale Unstable CA14 0 45 COc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217887091 CG For-Sale Unstable MMP2 20 48 COc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217887091 CG For-Sale Unstable CYP1A1 15 45 COc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217887091 CG For-Sale Unstable MMP9 26 48 COc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217887091 CG For-Sale Unstable 17HSDCL 0 41 COc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217887091 CG For-Sale Unstable FFAR1 47 52 COc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217887091 CG For-Sale Unstable AKR1C3 36 46 COc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217887091 CG For-Sale Unstable ACP1 0 40 COc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217887091 CG For-Sale Unstable FFAR4 44 42 COc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217887091 CG For-Sale Unstable ABCG2 15 44 COc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217887091 CG For-Sale Unstable AKR1B10 25 41 COc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217887091 CG For-Sale Unstable HPGD 22 50 COc1ccc(OCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217887091 CG For-Sale Unstable GPR183 0 48 Cc1nc(CN[C@H]2C[C@@H](C)CC[C@H]2C(C)C)cs1 ZINC000217887100 CI For-Sale Unstable TRPM8 0 41 Cc1cccc(/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O)c1 ZINC000217887133 CF For-Sale Unstable FOLH1 57 40 Cc1cccc(/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O)c1 ZINC000217887133 CF For-Sale Unstable MME 20 43 Cc1cccc(/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O)c1 ZINC000217887133 CF For-Sale Unstable ANPEP 39 50 Cc1cccc(/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O)c1 ZINC000217887133 CF For-Sale Unstable FPR1 72 48 O=C(O)CC1CCN(C(=O)OCc2cc(Cl)cc(Cl)c2)CC1 ZINC000217887143 EH For-Sale Unstable GRIN2B 34 47 O=C(O)CC1CCN(C(=O)OCc2cc(Cl)cc(Cl)c2)CC1 ZINC000217887143 EH For-Sale Unstable TGM2 22 40 O=C(O)CC1CCN(C(=O)OCc2cc(Cl)cc(Cl)c2)CC1 ZINC000217887143 EH For-Sale Unstable CACNA1I 50 38 O=C(O)CC1CCN(C(=O)OCc2cc(Cl)cc(Cl)c2)CC1 ZINC000217887143 EH For-Sale Unstable F13A1 37 40 C[C@H](C(=O)O)c1ccc(CN2C[C@@H](C)[C@@H](C)C2)cc1 ZINC000217887158 CF For-Sale Unstable PTGS1 36 53 C[C@H](C(=O)O)c1ccc(CN2C[C@@H](C)[C@@H](C)C2)cc1 ZINC000217887158 CF For-Sale Unstable PTGS2 26 53 C[C@H](C(=O)O)c1ccc(CN2C[C@@H](C)[C@@H](C)C2)cc1 ZINC000217887158 CF For-Sale Unstable MLNR 34 43 COc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217887170 CG For-Sale Unstable ALOX5 32 51 COc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217887170 CG For-Sale Unstable TSHR 50 36 COc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217887170 CG For-Sale Unstable MAOA 21 41 COc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217887170 CG For-Sale Unstable MAOB 76 62 COc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217887170 CG For-Sale Unstable PTGS2 0 48 COc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217887170 CG For-Sale Unstable PPARG 19 42 COc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217887170 CG For-Sale Unstable PTGER2 23 51 COc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217887170 CG For-Sale Unstable PPARA 22 42 COc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217887170 CG For-Sale Unstable LTA4H 19 42 COc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217887170 CG For-Sale Unstable PTGER4 39 48 COc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217887170 CG For-Sale Unstable CA7 0 46 COc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217887170 CG For-Sale Unstable PTGER3 37 49 COc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217887170 CG For-Sale Unstable LTB4R 46 46 COc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217887170 CG For-Sale Unstable KCNA3 26 40 COc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217887170 CG For-Sale Unstable ADAM17 15 41 COc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217887170 CG For-Sale Unstable HDAC8 38 40 COc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217887170 CG For-Sale Unstable PPARD 24 42 COc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217887170 CG For-Sale Unstable CA14 0 46 COc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217887170 CG For-Sale Unstable MTNR1A 49 41 COc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217887170 CG For-Sale Unstable MTNR1B 50 40 COc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217887170 CG For-Sale Unstable MMP2 17 51 COc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217887170 CG For-Sale Unstable NR1H4 71 42 COc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217887170 CG For-Sale Unstable GYS1 57 38 COc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217887170 CG For-Sale Unstable HDAC6 25 40 COc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217887170 CG For-Sale Unstable MMP9 19 51 COc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217887170 CG For-Sale Unstable 17HSDCL 0 41 COc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217887170 CG For-Sale Unstable FFAR1 89 47 COc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217887170 CG For-Sale Unstable AKR1C3 50 56 COc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217887170 CG For-Sale Unstable PTPA 0 43 COc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217887170 CG For-Sale Unstable FFAR4 36 43 COc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217887170 CG For-Sale Unstable ABCG2 19 43 COc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217887170 CG For-Sale Unstable ADCYAP1R1 41 37 COc1ccc(OCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217887170 CG For-Sale Unstable GPR183 0 45 O=C(/C=C/c1cccc([N+](=O)[O-])c1)NCCCc1ccccc1Cl ZINC000217887189 EI In-Stock Unstable PYGL 26 48 O=C(/C=C/c1cccc([N+](=O)[O-])c1)NCCCc1ccccc1Cl ZINC000217887189 EI In-Stock Unstable TRPM8 21 62 C[C@H](C(=O)O)c1ccc(CN2C[C@H](C)[C@@H](C)C2)cc1 ZINC000217887237 CF For-Sale Unstable PTGS1 36 53 C[C@H](C(=O)O)c1ccc(CN2C[C@H](C)[C@@H](C)C2)cc1 ZINC000217887237 CF For-Sale Unstable PTGS2 26 53 C[C@H](C(=O)O)c1ccc(CN2C[C@H](C)[C@@H](C)C2)cc1 ZINC000217887237 CF For-Sale Unstable MLNR 34 43 CSCC[C@@H](NC(=O)N/C=C/c1cccc(C)c1)C(=O)O ZINC000217887239 DE For-Sale Unstable FOLH1 19 41 CSCC[C@@H](NC(=O)N/C=C/c1cccc(C)c1)C(=O)O ZINC000217887239 DE For-Sale Unstable NAALAD2 42 33 CSCC[C@@H](NC(=O)N/C=C/c1cccc(C)c1)C(=O)O ZINC000217887239 DE For-Sale Unstable PAM 0 41 CSCC[C@@H](NC(=O)N/C=C/c1cccc(C)c1)C(=O)O ZINC000217887239 DE For-Sale Unstable FPR1 41 41 CSCC[C@@H](NC(=O)N/C=C/c1cccc(C)c1)C(=O)O ZINC000217887239 DE For-Sale Unstable SLC15A2 0 40 CCOCCOCCOc1cccc(/C=C\C(=O)O)c1 ZINC000217887254 CE For-Sale Unstable LTB4R 22 43 CCOCCOCCOc1cccc(/C=C\C(=O)O)c1 ZINC000217887254 CE For-Sale Unstable AKR1C3 29 41 O=C(/C=C/c1cccc([N+](=O)[O-])c1)NCCCc1ccc(Cl)cc1 ZINC000217887295 EI In-Stock Unstable CACNA1D 42 40 O=C(/C=C/c1cccc([N+](=O)[O-])c1)NCCCc1ccc(Cl)cc1 ZINC000217887295 EI In-Stock Unstable PYGL 25 46 O=C(/C=C/c1cccc([N+](=O)[O-])c1)NCCCc1ccc(Cl)cc1 ZINC000217887295 EI In-Stock Unstable TRPM8 0 57 COc1c([C@@H]2CCNC2)cc(F)c(Cl)c1F ZINC000217887305 BF For-Sale Unstable SLC6A2 28 41 Cn1c(CO)nnc1C1CCN(C(=O)CCC(F)(F)F)CC1 ZINC000217887312 DD In-Stock Unstable ETHR 81 50 CSCC[C@H](NC(=O)N/C=C/c1cccc(C)c1)C(=O)O ZINC000217887331 DE For-Sale Unstable FOLH1 19 41 CSCC[C@H](NC(=O)N/C=C/c1cccc(C)c1)C(=O)O ZINC000217887331 DE For-Sale Unstable NAALAD2 42 33 CSCC[C@H](NC(=O)N/C=C/c1cccc(C)c1)C(=O)O ZINC000217887331 DE For-Sale Unstable PAM 0 41 CSCC[C@H](NC(=O)N/C=C/c1cccc(C)c1)C(=O)O ZINC000217887331 DE For-Sale Unstable FPR1 41 41 CSCC[C@H](NC(=O)N/C=C/c1cccc(C)c1)C(=O)O ZINC000217887331 DE For-Sale Unstable SLC15A2 0 40 COc1c([C@H]2CCNC2)cc(F)c(Cl)c1F ZINC000217887386 BF For-Sale Unstable SLC6A2 28 41 O=C(/C=C/c1cccc([N+](=O)[O-])c1)NCCCc1ccc(F)cc1 ZINC000217887419 EG In-Stock Unstable CACNA1D 62 35 O=C(/C=C/c1cccc([N+](=O)[O-])c1)NCCCc1ccc(F)cc1 ZINC000217887419 EG In-Stock Unstable PYGL 25 41 O=C(/C=C/c1cccc([N+](=O)[O-])c1)NCCCc1ccc(F)cc1 ZINC000217887419 EG In-Stock Unstable TRPM8 0 53 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC1CC(c2ccccc2)C1 ZINC000217887427 CJ For-Sale Unstable TRPM8 17 46 Cc1nc(C2CCN(C(=O)Cc3ccc(N(C)C)cc3)CC2)no1 ZINC000217887436 EE In-Stock Unstable ETHR 69 41 C[C@@H](C(=O)O)c1ccc(CN2CCO[C@@H](C#N)C2)cc1 ZINC000217887504 CD For-Sale Unstable PTGS1 0 41 C[C@@H](C(=O)O)c1ccc(CN2CCO[C@@H](C#N)C2)cc1 ZINC000217887504 CD For-Sale Unstable SLC22A20 0 41 COc1ccccc1CCCNC(=O)/C=C/c1cccc([N+](=O)[O-])c1 ZINC000217887522 EG In-Stock Unstable DRD3 20 52 COc1ccccc1CCCNC(=O)/C=C/c1cccc([N+](=O)[O-])c1 ZINC000217887522 EG In-Stock Unstable CACNA1C 43 37 COc1ccccc1CCCNC(=O)/C=C/c1cccc([N+](=O)[O-])c1 ZINC000217887522 EG In-Stock Unstable CACNA1D 78 37 COc1ccccc1CCCNC(=O)/C=C/c1cccc([N+](=O)[O-])c1 ZINC000217887522 EG In-Stock Unstable MTNR1B 36 41 COc1ccccc1CCCNC(=O)/C=C/c1cccc([N+](=O)[O-])c1 ZINC000217887522 EG In-Stock Unstable TRPM8 0 64 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC1CC(c2ccccc2)C1 ZINC000217887542 CJ For-Sale Unstable TRPM8 17 46 C[C@H](C(=O)O)c1ccc(CN2CCO[C@@H](C#N)C2)cc1 ZINC000217887588 CD For-Sale Unstable PTGS1 0 41 C[C@H](C(=O)O)c1ccc(CN2CCO[C@@H](C#N)C2)cc1 ZINC000217887588 CD For-Sale Unstable SLC22A20 0 41 COc1ccc([C@@H](C)NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217887601 DI For-Sale Unstable ACACA 23 42 COc1ccc([C@@H](C)NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217887601 DI For-Sale Unstable ACACB 26 48 COc1ccc([C@@H](C)NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217887601 DI For-Sale Unstable MTNR1A 23 41 COc1ccc([C@@H](C)NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217887601 DI For-Sale Unstable MTNR1B 22 41 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC1CC(c2ccccc2)C1 ZINC000217887623 CJ For-Sale Unstable TRPM8 17 46 N#Cc1cccc(C(=O)NCCn2ccc(-c3ccsc3)n2)c1 ZINC000217887630 DF In-Stock Unstable DRD4 40 30 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2cccc([N+](=O)[O-])c2)cc1 ZINC000217887637 FG In-Stock Unstable CACNA1D 70 38 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2cccc([N+](=O)[O-])c2)cc1 ZINC000217887637 FG In-Stock Unstable TRPM8 0 59 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2cccc([N+](=O)[O-])c2)cc1 ZINC000217887637 FG In-Stock Unstable AKR1C2 15 42 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2cccc([N+](=O)[O-])c2)cc1 ZINC000217887637 FG In-Stock Unstable EXSA 0 41 CN1CCO[C@@H]([C@@H](N)c2cccc(Cl)c2)C1 ZINC000217887676 BD For-Sale Unstable OPRL1 0 47 COc1ccc([C@H](C)NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217887677 DI For-Sale Unstable ACACA 23 42 COc1ccc([C@H](C)NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217887677 DI For-Sale Unstable ACACB 26 48 COc1ccc([C@H](C)NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217887677 DI For-Sale Unstable MTNR1A 23 41 COc1ccc([C@H](C)NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217887677 DI For-Sale Unstable MTNR1B 22 41 CC(C)C[C@@H]1CNC[C@@H]1CNC(=O)OC(C)(C)C ZINC000217887693 CE For-Sale Unstable CTSK 17 40 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2cccc([N+](=O)[O-])c2)cc1 ZINC000217887695 FG In-Stock Unstable CACNA1D 70 38 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2cccc([N+](=O)[O-])c2)cc1 ZINC000217887695 FG In-Stock Unstable TRPM8 0 59 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2cccc([N+](=O)[O-])c2)cc1 ZINC000217887695 FG In-Stock Unstable AKR1C2 15 42 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2cccc([N+](=O)[O-])c2)cc1 ZINC000217887695 FG In-Stock Unstable EXSA 0 41 CSc1ccc(Cl)c(C(=O)ON2C(=O)CCC2=O)c1 ZINC000217887707 CE In-Stock Unstable Q9FYV8_MAIZE 46 38 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC1CC(c2ccccc2)C1 ZINC000217887731 CJ For-Sale Unstable TRPM8 17 46 CN1CCO[C@H]([C@@H](N)c2cccc(Cl)c2)C1 ZINC000217887742 BD For-Sale Unstable OPRL1 0 47 CC(C)C[C@H]1CNC[C@@H]1CNC(=O)OC(C)(C)C ZINC000217887765 CE For-Sale Unstable CTSK 17 40 O=C(/C=C/c1cccc([N+](=O)[O-])c1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217887777 FI In-Stock Bother LTB4R 0 46 O=C(/C=C/c1cccc([N+](=O)[O-])c1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217887777 FI In-Stock Bother PYGL 25 43 O=C(/C=C/c1cccc([N+](=O)[O-])c1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217887777 FI In-Stock Bother HDAC8 24 45 O=C(/C=C/c1cccc([N+](=O)[O-])c1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217887777 FI In-Stock Bother MMP2 21 50 O=C(/C=C/c1cccc([N+](=O)[O-])c1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217887777 FI In-Stock Bother MMP9 19 50 O=C(/C=C/c1cccc([N+](=O)[O-])c1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217887777 FI In-Stock Bother MMP1 24 50 O=C(/C=C/c1cccc([N+](=O)[O-])c1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217887777 FI In-Stock Bother AKR1C3 18 48 O=C(/C=C/c1cccc([N+](=O)[O-])c1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217887777 FI In-Stock Bother TRPM8 24 71 O=C(/C=C/c1cccc([N+](=O)[O-])c1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217887777 FI In-Stock Bother AKR1C2 23 48 O=C(/C=C/c1cccc([N+](=O)[O-])c1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217887777 FI In-Stock Bother TRPM2 0 40 CCOC(=O)c1cc(F)c(F)[nH]1 ZINC000217887784 AD For-Sale Unstable CACNA1C 19 42 CCOC(=O)c1cc(F)c(F)[nH]1 ZINC000217887784 AD For-Sale Unstable CACNA1D 23 42 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1N[C@@H]1CCc2c(O)cccc21 ZINC000217887826 CI For-Sale Unstable TRPM8 16 45 CCOc1ccccc1C(=O)ON1C(=O)CCC1=O ZINC000217887835 CD In-Stock Unstable HCN1 52 40 CCOc1ccccc1C(=O)ON1C(=O)CCC1=O ZINC000217887835 CD In-Stock Unstable HCN4 49 38 CC(C)C[C@@H]1CNC[C@H]1CNC(=O)OC(C)(C)C ZINC000217887859 CE For-Sale Unstable CTSK 17 40 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2cccc([N+](=O)[O-])c2)c1 ZINC000217887880 FI In-Stock Unstable CACNA1D 47 34 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2cccc([N+](=O)[O-])c2)c1 ZINC000217887880 FI In-Stock Unstable CRTM 39 45 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2cccc([N+](=O)[O-])c2)c1 ZINC000217887880 FI In-Stock Unstable TRPM8 0 52 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1N[C@@H]1CCc2c(O)cccc21 ZINC000217887895 CI For-Sale Unstable TRPM8 16 45 O=C(O)/C=C\c1ccc(COC2CCCCCC2)c(F)c1 ZINC000217887902 CI For-Sale Unstable AKR1C3 28 40 O=S(=O)(c1ccccc1)N(CCF)Cc1cccnc1 ZINC000217887910 CE For-Sale Unstable TBXAS1 27 43 O=S(=O)(c1ccccc1)N(CCF)Cc1cccnc1 ZINC000217887910 CE For-Sale Unstable NAMPT 27 42 O=S(=O)(c1ccccc1)N(CCF)Cc1cccnc1 ZINC000217887910 CE For-Sale Unstable NR1D1 41 33 C[C@@H](C(=O)O)c1ccc(CN2CCO[C@@H](CO)C2)cc1 ZINC000217887912 CD For-Sale Unstable DRD4 18 47 C[C@@H](C(=O)O)c1ccc(CN2CCO[C@@H](CO)C2)cc1 ZINC000217887912 CD For-Sale Unstable PTGS1 0 43 C[C@@H](C(=O)O)c1ccc(CN2CCO[C@@H](CO)C2)cc1 ZINC000217887912 CD For-Sale Unstable PTGS2 0 43 CC(C)C[C@H]1CNC[C@H]1CNC(=O)OC(C)(C)C ZINC000217887934 CE For-Sale Unstable CTSK 17 40 COC[C@@H]1CCN([C@@H](C)c2ccc(O)c(OC)c2)C1 ZINC000217887952 CE For-Sale Unstable RORC 48 35 CC(C)Oc1ccc(CCCNC(=O)/C=C/c2cccc([N+](=O)[O-])c2)cc1 ZINC000217887956 FI In-Stock Unstable CACNA1D 50 38 CC(C)Oc1ccc(CCCNC(=O)/C=C/c2cccc([N+](=O)[O-])c2)cc1 ZINC000217887956 FI In-Stock Unstable TRPM8 0 49 O=C(O)/C=C\c1cccc(COC2CCCCCC2)c1 ZINC000217887971 CI For-Sale Unstable PTGER2 24 42 O=C(O)/C=C\c1cccc(COC2CCCCCC2)c1 ZINC000217887971 CI For-Sale Unstable NR1H4 39 42 O=C(O)/C=C\c1cccc(COC2CCCCCC2)c1 ZINC000217887971 CI For-Sale Unstable HCAR2 0 42 O=C(O)/C=C\c1cccc(COC2CCCCCC2)c1 ZINC000217887971 CI For-Sale Unstable 17HSDCL 0 43 O=C(O)/C=C\c1cccc(COC2CCCCCC2)c1 ZINC000217887971 CI For-Sale Unstable AKR1C3 31 40 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1N[C@@H]1CCc2c(O)cccc21 ZINC000217887982 CI For-Sale Unstable TRPM8 16 45 C[C@H](C(=O)O)c1ccc(CN2CCO[C@@H](CO)C2)cc1 ZINC000217888008 CD For-Sale Unstable DRD4 18 47 C[C@H](C(=O)O)c1ccc(CN2CCO[C@@H](CO)C2)cc1 ZINC000217888008 CD For-Sale Unstable PTGS1 0 43 C[C@H](C(=O)O)c1ccc(CN2CCO[C@@H](CO)C2)cc1 ZINC000217888008 CD For-Sale Unstable PTGS2 0 43 COc1ccc(CCN2C(=O)N[C@@H](CCC(=O)N3CCCC3)C2=O)cc1OC ZINC000217888056 GD In-Stock Unstable FKBP1A 43 41 COc1ccc(CCN2C(=O)N[C@@H](CCC(=O)N3CCCC3)C2=O)cc1OC ZINC000217888056 GD In-Stock Unstable ACKR3 40 34 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCc1ccc(OC)cc1 ZINC000217888060 HF For-Sale Unstable MMP1 25 40 CC1(C)C[C@@H](NC(=O)/C=C/c2cccc([N+](=O)[O-])c2)c2ccccc2O1 ZINC000217888062 FI In-Stock Unstable CACNA1D 67 37 CC1(C)C[C@@H](NC(=O)/C=C/c2cccc([N+](=O)[O-])c2)c2ccccc2O1 ZINC000217888062 FI In-Stock Unstable TRPM8 0 51 CC(C)[C@H]1CC[C@H](C)C[C@@H]1N[C@@H]1CCc2c(O)cccc21 ZINC000217888092 CI For-Sale Unstable TRPM8 16 45 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCc1ccc(OC)cc1 ZINC000217888136 HF For-Sale Unstable MMP1 25 40 CC1(C)C[C@H](NC(=O)/C=C/c2cccc([N+](=O)[O-])c2)c2ccccc2O1 ZINC000217888140 FI In-Stock Unstable CACNA1C 40 37 CC1(C)C[C@H](NC(=O)/C=C/c2cccc([N+](=O)[O-])c2)c2ccccc2O1 ZINC000217888140 FI In-Stock Unstable CACNA1D 68 37 CC1(C)C[C@H](NC(=O)/C=C/c2cccc([N+](=O)[O-])c2)c2ccccc2O1 ZINC000217888140 FI In-Stock Unstable TRPM8 0 51 CCc1ccc([C@@H](C)NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217888141 DJ For-Sale Unstable ACACA 44 37 C[C@H](C(=O)O)c1ccc(CN2C[C@@H](CO)OC[C@@H]2C)cc1 ZINC000217888169 CD For-Sale Unstable PTGS1 0 43 O=C(NCCn1ccc(-c2ccsc2)n1)c1ccc(Cl)s1 ZINC000217888189 EH In-Stock Unstable F10 23 43 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCc1ccc(OC)cc1 ZINC000217888201 HF For-Sale Unstable MMP1 25 40 CCc1ccc([C@H](C)NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217888206 DJ For-Sale Unstable ACACA 44 37 CCOc1ccc(CCCNC(=O)/C=C/c2cccc([N+](=O)[O-])c2)cc1 ZINC000217888226 FH In-Stock Unstable CACNA1D 67 38 CCOc1ccc(CCCNC(=O)/C=C/c2cccc([N+](=O)[O-])c2)cc1 ZINC000217888226 FH In-Stock Unstable TRPM8 0 50 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCc1ccc(OC)cc1 ZINC000217888258 HF For-Sale Unstable MMP1 25 40 C[C@H](C(=O)O)c1ccc(CN2C[C@@H](C)[C@@H](N(C)C)C2)cc1 ZINC000217888284 CE For-Sale Unstable PTGS1 27 46 C[C@H](C(=O)O)c1ccc(CN2C[C@@H](C)[C@@H](N(C)C)C2)cc1 ZINC000217888284 CE For-Sale Unstable PTGS2 16 46 CCCOc1ccccc1CCCNC(=O)/C=C/c1cccc([N+](=O)[O-])c1 ZINC000217888328 FI In-Stock Unstable CACNA1D 53 35 CCCOc1ccccc1CCCNC(=O)/C=C/c1cccc([N+](=O)[O-])c1 ZINC000217888328 FI In-Stock Unstable MTNR1A 34 43 CCCOc1ccccc1CCCNC(=O)/C=C/c1cccc([N+](=O)[O-])c1 ZINC000217888328 FI In-Stock Unstable MTNR1B 34 43 CCCOc1ccccc1CCCNC(=O)/C=C/c1cccc([N+](=O)[O-])c1 ZINC000217888328 FI In-Stock Unstable TRPM8 0 52 CCOc1ccc(CC(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217888368 HF For-Sale Unstable ITGA4 47 38 COc1ccc(SCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217888387 DI For-Sale Unstable PTGER2 32 46 COc1ccc(SCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217888387 DI For-Sale Unstable PTGER4 0 46 COc1ccc(SCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217888387 DI For-Sale Unstable CYP1B1 19 40 COc1ccc(SCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217888387 DI For-Sale Unstable PTGER3 17 46 COc1ccc(SCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217888387 DI For-Sale Unstable LTB4R 38 47 COc1ccc(SCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217888387 DI For-Sale Unstable NR1H4 30 40 COc1ccc(SCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217888387 DI For-Sale Unstable AKR1C3 43 44 COc1ccc(SCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217888387 DI For-Sale Unstable PTPA 0 44 COc1ccc(SCc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000217888387 DI For-Sale Unstable GPR183 0 43 Brc1cccc(N2C[C@H]3CNC[C@@H](C3)C2)c1 ZINC000217888408 CE For-Sale Unstable CHRNA4 34 42 O=C(O)COc1ccn(-c2ccccc2)n1 ZINC000217888414 BD In-Stock Unstable PTGDR2 15 45 C[C@H](C(=O)O)c1ccc(CN(C)[C@@H]2CCO[C@@H]2C)cc1 ZINC000217888416 CE For-Sale Unstable PTGS1 25 46 O=C(CCc1ccc(O)cc1)NCc1ccc2ccccc2n1 ZINC000217888418 DG In-Stock Unstable CYSLTR1 68 48 O=C(CCc1ccc(O)cc1)NCc1ccc2ccccc2n1 ZINC000217888418 DG In-Stock Unstable HCAR2 32 42 O=C(CCc1ccc(O)cc1)NCc1ccc2ccccc2n1 ZINC000217888418 DG In-Stock Unstable SUCNR1 51 42 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1N[C@@H]1C[C@@H](C)N(C)C[C@@H]1C ZINC000217888420 CH For-Sale Unstable TRPM8 0 40 Cc1ccccc1OC[C@H](C)NC(=O)/C=C/c1cccc([N+](=O)[O-])c1 ZINC000217888425 EH In-Stock Unstable CACNA1C 44 37 Cc1ccccc1OC[C@H](C)NC(=O)/C=C/c1cccc([N+](=O)[O-])c1 ZINC000217888425 EH In-Stock Unstable CACNA1D 75 37 Cc1ccccc1OC[C@H](C)NC(=O)/C=C/c1cccc([N+](=O)[O-])c1 ZINC000217888425 EH In-Stock Unstable TRPM8 0 60 CCOc1ccc(CC(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217888450 HF For-Sale Unstable ITGA4 47 38 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1N[C@@H]1C[C@@H](C)N(C)C[C@@H]1C ZINC000217888481 CH For-Sale Unstable TRPM8 0 40 O=CCCCc1cn(Cc2ccccc2)nn1 ZINC000217888512 BD For-Sale Unstable HDAC1 15 55 CC1CCN(c2ccc([C@@H](C)NC(=O)/C=C/c3cccc([N+](=O)[O-])c3)cc2)CC1 ZINC000217888514 GJ In-Stock Unstable KCNQ2 47 36 CCOc1ccc(CC(=O)N2C[C@H](Oc3ccccc3F)C[C@H]2C(=O)OC)cc1 ZINC000217888541 HF For-Sale Unstable ITGA4 47 38 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1N[C@@H]1C[C@@H](C)N(C)C[C@@H]1C ZINC000217888579 CH For-Sale Unstable TRPM8 0 40 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H]3CCCC[C@@H]32)cc1 ZINC000217888621 CH For-Sale Unstable PTGS1 27 50 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H]3CCCC[C@@H]32)cc1 ZINC000217888621 CH For-Sale Unstable PTGS2 0 50 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H]3CCCC[C@@H]32)cc1 ZINC000217888621 CH For-Sale Unstable FAAH 0 40 CCOc1ccc(CC(=O)N2C[C@@H](Oc3ccccc3F)C[C@H]2C(=O)OC)cc1 ZINC000217888622 HF For-Sale Unstable ITGA4 47 38 CC1CCN(c2ccc([C@H](C)NC(=O)/C=C/c3cccc([N+](=O)[O-])c3)cc2)CC1 ZINC000217888629 GJ In-Stock Unstable KCNQ2 47 36 Cc1cccc(/C=C/NC(=O)Nc2ccc(Oc3ccccc3)cc2)c1 ZINC000217888646 EK For-Sale Unstable LPL 41 32 Cc1cccc(/C=C/NC(=O)Nc2ccc(Oc3ccccc3)cc2)c1 ZINC000217888646 EK For-Sale Unstable LTA4H 31 43 Cc1cccc(/C=C/NC(=O)Nc2ccc(Oc3ccccc3)cc2)c1 ZINC000217888646 EK For-Sale Unstable CA1 48 45 Cc1cccc(/C=C/NC(=O)Nc2ccc(Oc3ccccc3)cc2)c1 ZINC000217888646 EK For-Sale Unstable RAF1 30 47 Cc1cccc(/C=C/NC(=O)Nc2ccc(Oc3ccccc3)cc2)c1 ZINC000217888646 EK For-Sale Unstable KDR 25 40 Cc1cccc(/C=C/NC(=O)Nc2ccc(Oc3ccccc3)cc2)c1 ZINC000217888646 EK For-Sale Unstable MTNR1B 17 46 Cc1cccc(/C=C/NC(=O)Nc2ccc(Oc3ccccc3)cc2)c1 ZINC000217888646 EK For-Sale Unstable CA12 17 45 Cc1cccc(/C=C/NC(=O)Nc2ccc(Oc3ccccc3)cc2)c1 ZINC000217888646 EK For-Sale Unstable PDGFRA 34 40 Cc1cccc(/C=C/NC(=O)Nc2ccc(Oc3ccccc3)cc2)c1 ZINC000217888646 EK For-Sale Unstable CA9 18 45 Cc1cccc(/C=C/NC(=O)Nc2ccc(Oc3ccccc3)cc2)c1 ZINC000217888646 EK For-Sale Unstable MMP1 0 43 Cc1cccc(/C=C/NC(=O)Nc2ccc(Oc3ccccc3)cc2)c1 ZINC000217888646 EK For-Sale Unstable Q8MMZ8_EIMTE 51 47 Cc1cccc(/C=C/NC(=O)Nc2ccc(Oc3ccccc3)cc2)c1 ZINC000217888646 EK For-Sale Unstable KCNK3 42 36 CC(C)[C@H]1CC[C@H](C)C[C@@H]1N[C@@H]1C[C@@H](C)N(C)C[C@@H]1C ZINC000217888664 CH For-Sale Unstable TRPM8 0 40 Brc1ccc(N2C[C@H]3CNC[C@@H](C3)C2)cc1 ZINC000217888669 CE For-Sale Unstable CHRNA4 33 43 CC[C@@H]1CCN(C(=O)OC(C)(C)C)CC[C@@H]1CN ZINC000217888671 CF For-Sale Unstable GPR119 42 44 COc1cc(CCC(=O)N[C@H](CO)c2ccccc2)on1 ZINC000217888716 CD In-Stock Unstable GPR88 0 45 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)C12CC3CC(CC(C3)C1)C2 ZINC000217888730 HH For-Sale Unstable GRM1 16 43 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)/C=C/c3cccc([N+](=O)[O-])c3)cc2)C1 ZINC000217888732 GJ In-Stock Unstable KCNQ2 47 36 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)/C=C/c3cccc([N+](=O)[O-])c3)cc2)C1 ZINC000217888732 GJ In-Stock Unstable TRPM8 0 48 CC[C@H]1CCN(C(=O)OC(C)(C)C)CC[C@@H]1CN ZINC000217888738 CF For-Sale Unstable GPR119 42 44 CN1CCO[C@@H]([C@@H](N)c2cccc(F)c2)C1 ZINC000217888745 BD For-Sale Unstable OPRL1 0 45 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NCc1cc[nH]n1 ZINC000217888763 BF On-Demand Unstable TRPM8 15 41 CCOCCOCCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217888806 CE For-Sale Unstable PPARA 15 47 CCOCCOCCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217888806 CE For-Sale Unstable PLA2G4B 74 34 CCOCCOCCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217888806 CE For-Sale Unstable AKR1C3 24 40 CC[C@@H]1CCN(C(=O)OC(C)(C)C)CC[C@H]1CN ZINC000217888820 CF For-Sale Unstable GPR119 42 44 CN1CCO[C@H]([C@@H](N)c2cccc(F)c2)C1 ZINC000217888828 BD For-Sale Unstable OPRL1 0 45 C[C@H](NC(=O)/C=C/c1cccc([N+](=O)[O-])c1)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217888829 GJ In-Stock Unstable KCNQ2 47 36 C[C@H](NC(=O)/C=C/c1cccc([N+](=O)[O-])c1)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217888829 GJ In-Stock Unstable TRPM8 0 48 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)C12CC3CC(CC(C3)C1)C2 ZINC000217888830 HH For-Sale Unstable GRM1 16 43 C[C@@H](C(=O)O)c1ccc(CN2CC[C@@H](CO)C2)cc1 ZINC000217888839 CD For-Sale Unstable ACHE 33 40 C[C@@H](C(=O)O)c1ccc(CN2CC[C@@H](CO)C2)cc1 ZINC000217888839 CD For-Sale Unstable PTGS1 31 47 C[C@@H](C(=O)O)c1ccc(CN2CC[C@@H](CO)C2)cc1 ZINC000217888839 CD For-Sale Unstable PTGS2 0 47 C[C@@H](C(=O)O)c1ccc(CN2CC[C@@H](CO)C2)cc1 ZINC000217888839 CD For-Sale Unstable SLC6A3 17 43 C[C@@H](C(=O)O)c1ccc(CN2CC[C@@H](CO)C2)cc1 ZINC000217888839 CD For-Sale Unstable SIGMAR1 46 40 C[C@@H](C(=O)O)c1ccc(CN2CC[C@@H](CO)C2)cc1 ZINC000217888839 CD For-Sale Unstable S1PR5 16 42 C[C@@H](C(=O)O)c1ccc(CN2CC[C@@H](CO)C2)cc1 ZINC000217888839 CD For-Sale Unstable SLC22A20 0 45 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NCc1cc[nH]n1 ZINC000217888842 BF On-Demand Unstable TRPM8 15 41 COc1ccc(OC)c(NC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217888867 DH For-Sale Unstable CYP1B1 52 36 COc1ccc(OC)c(NC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217888867 DH For-Sale Unstable MTNR1A 31 45 COc1ccc(OC)c(NC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217888867 DH For-Sale Unstable MTNR1B 31 45 COc1ccc(OC)c(NC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217888867 DH For-Sale Unstable CYP1A1 34 40 COc1ccc(OC)c(NC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217888867 DH For-Sale Unstable AKR1C3 18 45 COc1ccc(OC)c(NC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217888867 DH For-Sale Unstable ABCG2 21 41 COc1ccc(OC)c(NC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217888867 DH For-Sale Unstable AKR1C2 50 45 COc1ccc(OC)c(NC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217888867 DH For-Sale Unstable KCNK3 19 46 COc1ccc(OC)c(NC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217888867 DH For-Sale Unstable CYSP_PLAFA 41 37 COc1cccc(-c2cc(C(=O)NCCn3ccc(-c4ccsc4)n3)n(C)n2)c1 ZINC000217888870 HG In-Stock Unstable DRD4 44 33 COCCOCCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217888881 CD For-Sale Unstable PTGER2 24 44 COCCOCCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217888881 CD For-Sale Unstable AHR 23 40 COCCOCCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217888881 CD For-Sale Unstable PLA2G4B 57 32 CC[C@H]1CCN(C(=O)OC(C)(C)C)CC[C@H]1CN ZINC000217888904 CF For-Sale Unstable GPR119 42 44 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)C12CC3CC(CC(C3)C1)C2 ZINC000217888910 HH For-Sale Unstable GRM1 16 43 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NCc1cc[nH]n1 ZINC000217888914 BF For-Sale Unstable TRPM8 15 41 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](CO)C2)cc1 ZINC000217888921 CD For-Sale Unstable ACHE 33 40 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](CO)C2)cc1 ZINC000217888921 CD For-Sale Unstable PTGS1 31 47 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](CO)C2)cc1 ZINC000217888921 CD For-Sale Unstable PTGS2 0 47 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](CO)C2)cc1 ZINC000217888921 CD For-Sale Unstable SLC6A3 17 43 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](CO)C2)cc1 ZINC000217888921 CD For-Sale Unstable SIGMAR1 46 40 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](CO)C2)cc1 ZINC000217888921 CD For-Sale Unstable S1PR5 16 42 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](CO)C2)cc1 ZINC000217888921 CD For-Sale Unstable SLC22A20 0 45 Cc1ccc2c(c1)[C@@H](NC(=O)/C=C/c1cccc([N+](=O)[O-])c1)CC(C)(C)O2 ZINC000217888927 FI In-Stock Unstable CACNA1D 64 35 Cc1ccc2c(c1)[C@@H](NC(=O)/C=C/c1cccc([N+](=O)[O-])c1)CC(C)(C)O2 ZINC000217888927 FI In-Stock Unstable TRPM8 0 53 COc1ccc(COC[C@@H]2CCCO2)cc1/C=C\C(=O)O ZINC000217888965 CE For-Sale Unstable PTGER2 29 40 CN1CCO[C@@H]([C@@H](N)Cc2cc(F)ccc2F)C1 ZINC000217888975 CD For-Sale Unstable DPP4 40 52 COc1ccc2[nH]c3c(c2c1)CN(C(=O)[C@@H]1CCc2ccccc2O1)CC3 ZINC000217888980 FG In-Stock Unstable DRD5 30 48 COc1ccc2[nH]c3c(c2c1)CN(C(=O)[C@@H]1CCc2ccccc2O1)CC3 ZINC000217888980 FG In-Stock Unstable MAPKAPK2 0 42 CCC[C@@H](O)CNCCc1ccccn1 ZINC000217888991 BD For-Sale Unstable ADRB1 22 41 CCC[C@@H](O)CNCCc1ccccn1 ZINC000217888991 BD For-Sale Unstable ADRB3 32 41 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)C12CC3CC(CC(C3)C1)C2 ZINC000217889002 HH For-Sale Unstable GRM1 16 43 C[C@H](Cc1ccc(F)cc1)NC(=O)[C@@H]1CCC[C@@H](C)N1 ZINC000217889007 CE For-Sale Unstable MC4R 19 41 C[C@H](Cc1ccc(F)cc1)NC(=O)[C@@H]1CCC[C@@H](C)N1 ZINC000217889007 CE For-Sale Unstable MC5R 24 41 Cc1ccc2c(c1)[C@H](NC(=O)/C=C/c1cccc([N+](=O)[O-])c1)CC(C)(C)O2 ZINC000217889008 FI In-Stock Unstable CACNA1D 64 35 Cc1ccc2c(c1)[C@H](NC(=O)/C=C/c1cccc([N+](=O)[O-])c1)CC(C)(C)O2 ZINC000217889008 FI In-Stock Unstable TRPM8 0 53 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NCc1cc[nH]n1 ZINC000217889010 BF For-Sale Unstable TRPM8 15 41 CC(C)[C@@H]1CCN(C(=O)OC(C)(C)C)CC[C@@H]1N ZINC000217889032 CF For-Sale Unstable GPR119 36 43 CCN(C)C(=O)CNC(=O)c1cc2cc(N)ccc2[nH]1 ZINC000217889035 CC For-Sale Unstable PYGL 83 60 COc1ccc2[nH]c3c(c2c1)CN(C(=O)[C@H]1CCc2ccccc2O1)CC3 ZINC000217889066 FG In-Stock Unstable MAPKAPK2 0 42 CN1CCO[C@H]([C@@H](N)Cc2cc(F)ccc2F)C1 ZINC000217889067 CD For-Sale Unstable DPP4 40 52 O=C(NCCn1ccc(-c2ccsc2)n1)c1noc2c1CCCC2 ZINC000217889073 EF In-Stock Unstable PANC 41 32 C[C@H](Cc1ccc(F)cc1)NC(=O)[C@H]1CCC[C@@H](C)N1 ZINC000217889082 CE For-Sale Unstable MC4R 19 41 C[C@H](Cc1ccc(F)cc1)NC(=O)[C@H]1CCC[C@@H](C)N1 ZINC000217889082 CE For-Sale Unstable MC5R 24 41 CCC[C@H](O)CNCCc1ccccn1 ZINC000217889092 BD For-Sale Unstable ADRB1 22 41 CCC[C@H](O)CNCCc1ccccn1 ZINC000217889092 BD For-Sale Unstable ADRB3 32 41 CC(C)[C@H]1CCN(C(=O)OC(C)(C)C)CC[C@@H]1N ZINC000217889094 CF For-Sale Unstable GPR119 36 43 Cc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)/C=C/c1cccc([N+](=O)[O-])c1 ZINC000217889114 FI In-Stock Unstable CACNA1C 44 36 Cc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)/C=C/c1cccc([N+](=O)[O-])c1 ZINC000217889114 FI In-Stock Unstable CACNA1D 75 36 Cc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)/C=C/c1cccc([N+](=O)[O-])c1 ZINC000217889114 FI In-Stock Unstable TRPM8 0 55 COc1ccc(COC[C@H]2CCCO2)cc1/C=C\C(=O)O ZINC000217889119 CE For-Sale Unstable PTGER2 29 40 NC(=O)[C@@H]1CCCCN1C(=O)c1cc(-c2ccccc2)nc2c1cnn2Cc1ccco1 ZINC000217889130 IG On-Demand Unstable COLA 40 34 Cc1nc([C@H](C)N[C@H]2C[C@H](C)CC[C@H]2C(C)C)cs1 ZINC000217889147 CJ For-Sale Unstable TRPM8 0 42 CC(C)[C@@H]1CCN(C(=O)OC(C)(C)C)CC[C@H]1N ZINC000217889173 CF For-Sale Unstable GPR119 36 43 Cc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)/C=C/c1cccc([N+](=O)[O-])c1 ZINC000217889185 FI In-Stock Unstable CACNA1C 44 36 Cc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)/C=C/c1cccc([N+](=O)[O-])c1 ZINC000217889185 FI In-Stock Unstable CACNA1D 75 36 Cc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)/C=C/c1cccc([N+](=O)[O-])c1 ZINC000217889185 FI In-Stock Unstable TRPM8 0 55 NC(=O)[C@H]1CCCCN1C(=O)c1cc(-c2ccccc2)nc2c1cnn2Cc1ccco1 ZINC000217889211 IG On-Demand Unstable COLA 40 34 COC(=O)c1ccccc1NC(=O)N/C=C/c1cccc(C)c1 ZINC000217889216 DH For-Sale Unstable AKR1C2 18 40 CC(C)S(=O)(=O)N[C@@H]1C[C@@H]2C[C@@H]1[C@@H]1CCC[C@@H]21 ZINC000217889221 CE For-Sale Unstable GRIA4 29 40 Cc1nc([C@H](C)N[C@H]2C[C@@H](C)CC[C@H]2C(C)C)cs1 ZINC000217889231 CJ For-Sale Unstable TRPM8 0 42 CC(C)[C@H]1CCN(C(=O)OC(C)(C)C)CC[C@H]1N ZINC000217889260 CF For-Sale Unstable GPR119 36 43 COc1ccc2c(c1)[C@@H](NC(=O)/C=C/c1cccc([N+](=O)[O-])c1)CC(C)(C)O2 ZINC000217889292 GI In-Stock Unstable CACNA1C 40 36 COc1ccc2c(c1)[C@@H](NC(=O)/C=C/c1cccc([N+](=O)[O-])c1)CC(C)(C)O2 ZINC000217889292 GI In-Stock Unstable CACNA1D 73 36 COc1ccc2c(c1)[C@@H](NC(=O)/C=C/c1cccc([N+](=O)[O-])c1)CC(C)(C)O2 ZINC000217889292 GI In-Stock Unstable TRPM8 0 55 CC(C)S(=O)(=O)N[C@H]1C[C@@H]2C[C@@H]1[C@@H]1CCC[C@@H]21 ZINC000217889311 CE For-Sale Unstable GRIA4 29 40 Cc1nc([C@H](C)N[C@H]2C[C@@H](C)CC[C@@H]2C(C)C)cs1 ZINC000217889315 CJ For-Sale Unstable TRPM8 0 42 Cc1cccc(/C=C/NC(=O)Nc2ccc(F)cc2)c1 ZINC000217889337 CH For-Sale Unstable MMP2 0 52 Cc1cccc(/C=C/NC(=O)Nc2ccc(F)cc2)c1 ZINC000217889337 CH For-Sale Unstable MMP9 0 52 Cc1cccc(/C=C/NC(=O)Nc2ccc(F)cc2)c1 ZINC000217889337 CH For-Sale Unstable MMP1 0 52 Cc1cccc(/C=C/NC(=O)Nc2ccc(F)cc2)c1 ZINC000217889337 CH For-Sale Unstable IDO1 16 40 Cc1cccc(/C=C/NC(=O)Nc2ccc(F)cc2)c1 ZINC000217889337 CH For-Sale Unstable KCNK3 55 39 Cc1cccc(/C=C/NC(=O)Nc2ccc(F)cc2)c1 ZINC000217889337 CH For-Sale Unstable KCNK9 41 39 CCC[C@@H]1CCN(C(=O)OC(C)(C)C)CC[C@@H]1N ZINC000217889370 CF For-Sale Unstable GPR119 39 45 COC(=O)C[C@H](c1ccccc1OC)c1c(O)c2ccccc2oc1=O ZINC000217889383 FG In-Stock Unstable NQO1 67 54 CC(C)S(=O)(=O)N[C@@H]1C[C@H]2C[C@@H]1[C@@H]1CCC[C@@H]21 ZINC000217889389 CE For-Sale Unstable GRIA4 29 40 COc1ccc2c(c1)[C@H](NC(=O)/C=C/c1cccc([N+](=O)[O-])c1)CC(C)(C)O2 ZINC000217889393 GI In-Stock Unstable CACNA1D 73 36 COc1ccc2c(c1)[C@H](NC(=O)/C=C/c1cccc([N+](=O)[O-])c1)CC(C)(C)O2 ZINC000217889393 GI In-Stock Unstable TRPM8 0 55 O=C(N[C@H]1CCC[C@H]1CO)c1cccc(-n2cccc2)c1 ZINC000217889394 CE On-Demand Unstable AOC2 0 56 CCc1ccccc1OCc1ccccc1/C=C\C(=O)O ZINC000217889397 CH For-Sale Unstable PTGER2 27 61 CCc1ccccc1OCc1ccccc1/C=C\C(=O)O ZINC000217889397 CH For-Sale Unstable PTGER4 46 61 CCc1ccccc1OCc1ccccc1/C=C\C(=O)O ZINC000217889397 CH For-Sale Unstable PTGER3 34 61 CCc1ccccc1OCc1ccccc1/C=C\C(=O)O ZINC000217889397 CH For-Sale Unstable PTGDR 0 48 O=C(NCCn1ccc(-c2ccsc2)n1)c1cccc(OC(F)(F)F)c1 ZINC000217889400 GH In-Stock Unstable DRD4 45 34 O=C(NCCn1ccc(-c2ccsc2)n1)c1cccc(OC(F)(F)F)c1 ZINC000217889400 GH In-Stock Unstable GCGR 17 42 CCC[C@H]1CCN(C(=O)OC(C)(C)C)CC[C@@H]1N ZINC000217889450 CF For-Sale Unstable GPR119 39 45 C[C@H](C(=O)O)c1ccc(CN2C[C@H]3[C@H](O)CC[C@H]3C2)cc1 ZINC000217889455 CE For-Sale Unstable PTGS1 24 47 C[C@H](C(=O)O)c1ccc(CN2C[C@H]3[C@H](O)CC[C@H]3C2)cc1 ZINC000217889455 CE For-Sale Unstable PTGS2 17 47 COC(=O)C[C@@H](c1ccccc1OC)c1c(O)c2ccccc2oc1=O ZINC000217889457 FG In-Stock Unstable NQO1 67 54 CC(C)S(=O)(=O)N[C@H]1C[C@H]2C[C@@H]1[C@@H]1CCC[C@@H]21 ZINC000217889461 CE For-Sale Unstable GRIA4 29 40 CCc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217889471 CH For-Sale Unstable PTGER2 32 58 CCc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217889471 CH For-Sale Unstable PPIA 41 33 CCc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217889471 CH For-Sale Unstable PTGER1 43 46 CCc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217889471 CH For-Sale Unstable PTGER4 47 58 CCc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217889471 CH For-Sale Unstable PTGER3 34 58 CCc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217889471 CH For-Sale Unstable PTGDR 0 46 CCc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217889471 CH For-Sale Unstable AKR1C3 38 51 CCc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217889471 CH For-Sale Unstable AKR1B10 26 42 Cc1ccc(O)c([C@H](C)N[C@H]2C[C@H](C)CC[C@H]2C(C)C)c1 ZINC000217889484 CJ For-Sale Unstable TRPM8 19 53 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc(OC)c1OC ZINC000217889486 HF For-Sale Unstable HCRTR1 46 39 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc(OC)c1OC ZINC000217889486 HF For-Sale Unstable AGTR2 47 33 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc(OC)c1OC ZINC000217889486 HF For-Sale Unstable HCRTR2 52 39 Cc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c([N+](=O)[O-])c2)c1 ZINC000217889488 EI For-Sale Unstable TRPM8 0 47 Cc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c([N+](=O)[O-])c2)c1 ZINC000217889488 EI For-Sale Unstable IMDH_CRYPV 37 48 Cc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c([N+](=O)[O-])c2)c1 ZINC000217889488 EI For-Sale Unstable BLM 0 45 Cc1cc(C(=O)N(C)Cc2cc(-c3ccccc3)on2)cc(=O)[nH]1 ZINC000217889490 DF In-Stock Unstable GRM7 56 32 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)/C=C/c1cccc([N+](=O)[O-])c1 ZINC000217889491 GI In-Stock Unstable CACNA1C 44 37 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)/C=C/c1cccc([N+](=O)[O-])c1 ZINC000217889491 GI In-Stock Unstable CACNA1D 74 37 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)/C=C/c1cccc([N+](=O)[O-])c1 ZINC000217889491 GI In-Stock Unstable TRPM8 0 56 CCC[C@@H]1CCN(C(=O)OC(C)(C)C)CC[C@H]1N ZINC000217889512 CF For-Sale Unstable GPR119 39 45 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc(OC)c1OC ZINC000217889579 HF For-Sale Unstable HCRTR1 46 39 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc(OC)c1OC ZINC000217889579 HF For-Sale Unstable AGTR2 47 33 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc(OC)c1OC ZINC000217889579 HF For-Sale Unstable HCRTR2 52 39 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)/C=C/c1cccc([N+](=O)[O-])c1 ZINC000217889584 GI In-Stock Unstable CACNA1D 74 37 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)/C=C/c1cccc([N+](=O)[O-])c1 ZINC000217889584 GI In-Stock Unstable TRPM8 0 56 Cc1ccc(O)c([C@H](C)N[C@H]2C[C@@H](C)CC[C@H]2C(C)C)c1 ZINC000217889585 CJ For-Sale Unstable TRPM8 19 53 COc1cc([N+](=O)[O-])ccc1NC(=O)N/C=C/c1cccc(C)c1 ZINC000217889591 EH For-Sale Unstable EPHX1 0 53 COc1cc([N+](=O)[O-])ccc1NC(=O)N/C=C/c1cccc(C)c1 ZINC000217889591 EH For-Sale Unstable CACNA1C 45 36 COc1cc([N+](=O)[O-])ccc1NC(=O)N/C=C/c1cccc(C)c1 ZINC000217889591 EH For-Sale Unstable CACNA1D 75 36 COc1cc([N+](=O)[O-])ccc1NC(=O)N/C=C/c1cccc(C)c1 ZINC000217889591 EH For-Sale Unstable PYGL 22 40 COc1cc([N+](=O)[O-])ccc1NC(=O)N/C=C/c1cccc(C)c1 ZINC000217889591 EH For-Sale Unstable KCNMA1 23 51 COc1cc([N+](=O)[O-])ccc1NC(=O)N/C=C/c1cccc(C)c1 ZINC000217889591 EH For-Sale Unstable TRPM8 0 55 CCC[C@H]1CCN(C(=O)OC(C)(C)C)CC[C@H]1N ZINC000217889607 CF For-Sale Unstable GPR119 39 45 O=C(O)Cc1ccc(CN2C[C@H]3[C@H](O)CC[C@H]3C2)cc1 ZINC000217889611 CD For-Sale Unstable SIGMAR1 24 41 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc(OC)c1OC ZINC000217889657 HF For-Sale Unstable HCRTR1 46 39 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc(OC)c1OC ZINC000217889657 HF For-Sale Unstable AGTR2 47 33 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc(OC)c1OC ZINC000217889657 HF For-Sale Unstable HCRTR2 52 39 COc1ccc(Cn2cc(CCCC=O)nn2)cc1 ZINC000217889662 CD For-Sale Unstable HSP90AB1 25 43 O=C(O)/C=C\c1ccccc1COc1ccc(CO)cc1 ZINC000217889674 CF For-Sale Unstable PTGER2 72 49 O=C(O)/C=C\c1ccccc1COc1ccc(CO)cc1 ZINC000217889674 CF For-Sale Unstable PTGER4 58 53 O=C(O)/C=C\c1ccccc1COc1ccc(CO)cc1 ZINC000217889674 CF For-Sale Unstable PTPN2 0 40 O=C(O)/C=C\c1ccccc1COc1ccc(CO)cc1 ZINC000217889674 CF For-Sale Unstable PTGER3 34 61 O=C(O)/C=C\c1ccccc1COc1ccc(CO)cc1 ZINC000217889674 CF For-Sale Unstable CDC25B 23 42 O=C(O)/C=C\c1ccccc1COc1ccc(CO)cc1 ZINC000217889674 CF For-Sale Unstable FFAR1 35 45 O=C(O)/C=C\c1ccccc1COc1ccc(CO)cc1 ZINC000217889674 CF For-Sale Unstable FFAR4 54 46 Cc1ccc(O)c([C@H](C)N[C@H]2C[C@@H](C)CC[C@@H]2C(C)C)c1 ZINC000217889676 CJ For-Sale Unstable TRPM8 19 53 CC[C@@H](NC(=O)/C=C/c1cccc([N+](=O)[O-])c1)c1ccc(C)c(C)c1 ZINC000217889691 EI In-Stock Unstable CACNA1D 49 34 CC[C@@H](NC(=O)/C=C/c1cccc([N+](=O)[O-])c1)c1ccc(C)c(C)c1 ZINC000217889691 EI In-Stock Unstable TRPM8 0 55 Cc1cccc(/C=C/NC(=O)Nc2ccc([N+](=O)[O-])cc2)c1 ZINC000217889698 CH For-Sale Unstable MMP9 0 43 Cc1cccc(/C=C/NC(=O)Nc2ccc([N+](=O)[O-])cc2)c1 ZINC000217889698 CH For-Sale Unstable MMP1 0 40 Cc1cccc(/C=C/NC(=O)Nc2ccc([N+](=O)[O-])cc2)c1 ZINC000217889698 CH For-Sale Unstable TRPM8 0 55 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc(OC)c1OC ZINC000217889762 HF For-Sale Unstable HCRTR1 46 39 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc(OC)c1OC ZINC000217889762 HF For-Sale Unstable AGTR2 47 33 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc(OC)c1OC ZINC000217889762 HF For-Sale Unstable HCRTR2 52 39 O=C(O)/C=C\c1ccc(COc2ccc(CO)cc2)cc1 ZINC000217889767 CF For-Sale Unstable MAOB 15 53 O=C(O)/C=C\c1ccc(COc2ccc(CO)cc2)cc1 ZINC000217889767 CF For-Sale Unstable PTGER2 34 45 O=C(O)/C=C\c1ccc(COc2ccc(CO)cc2)cc1 ZINC000217889767 CF For-Sale Unstable PTGER4 26 43 O=C(O)/C=C\c1ccc(COc2ccc(CO)cc2)cc1 ZINC000217889767 CF For-Sale Unstable PTGER3 15 47 O=C(O)/C=C\c1ccc(COc2ccc(CO)cc2)cc1 ZINC000217889767 CF For-Sale Unstable FFAR1 34 44 O=C(O)/C=C\c1ccc(COc2ccc(CO)cc2)cc1 ZINC000217889767 CF For-Sale Unstable AKR1C3 41 43 O=C(O)/C=C\c1ccc(COc2ccc(CO)cc2)cc1 ZINC000217889767 CF For-Sale Unstable FFAR4 45 35 O=C(O)/C=C\c1ccc(COc2ccc(CO)cc2)cc1 ZINC000217889767 CF For-Sale Unstable AKR1B10 15 45 COc1ccc(Cn2cc(CCCCO)nn2)cc1 ZINC000217889776 CD For-Sale Unstable FIMH 23 51 COc1ccc(Cn2cc(CCCCO)nn2)cc1 ZINC000217889776 CD For-Sale Unstable PROKR1 52 32 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc(OCc3cccnc3)c2)CC(=O)O4)cc1O ZINC000217889783 KK In-Stock Unstable CYP1A1 30 41 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc(OCc3cccnc3)c2)CC(=O)O4)cc1O ZINC000217889783 KK In-Stock Unstable CYP1A2 25 40 CC[C@H](NC(=O)/C=C/c1cccc([N+](=O)[O-])c1)c1ccc(C)c(C)c1 ZINC000217889787 EI In-Stock Unstable CACNA1D 49 34 CC[C@H](NC(=O)/C=C/c1cccc([N+](=O)[O-])c1)c1ccc(C)c(C)c1 ZINC000217889787 EI In-Stock Unstable TRPM8 0 55 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC1CCSCC1 ZINC000217889800 CH On-Demand Unstable TRPM8 17 43 Cc1cccc(/C=C/NC(=O)Nc2cccc([N+](=O)[O-])c2)c1 ZINC000217889821 CH For-Sale Unstable CACNA1D 48 35 Cc1cccc(/C=C/NC(=O)Nc2cccc([N+](=O)[O-])c2)c1 ZINC000217889821 CH For-Sale Unstable TRPM8 0 66 Cc1cccc(/C=C/NC(=O)Nc2cccc([N+](=O)[O-])c2)c1 ZINC000217889821 CH For-Sale Unstable KCNK3 51 37 Cc1cccc(/C=C/NC(=O)Nc2cccc([N+](=O)[O-])c2)c1 ZINC000217889821 CH For-Sale Unstable KCNK9 41 37 O=C(O)C[C@H](NC(=O)c1cc(O)ccc1O)C(=O)O ZINC000217889833 CB For-Sale Unstable FOLH1 27 43 CC(=O)N[C@@H]1CCN(Cc2ccc([C@@H](C)C(=O)O)cc2)C1 ZINC000217889836 CD For-Sale Unstable CHRM2 16 41 CC(=O)N[C@@H]1CCN(Cc2ccc([C@@H](C)C(=O)O)cc2)C1 ZINC000217889836 CD For-Sale Unstable DRD4 35 49 CC(=O)N[C@@H]1CCN(Cc2ccc([C@@H](C)C(=O)O)cc2)C1 ZINC000217889836 CD For-Sale Unstable CHRM3 24 41 CC(=O)N[C@@H]1CCN(Cc2ccc([C@@H](C)C(=O)O)cc2)C1 ZINC000217889836 CD For-Sale Unstable LTA4H 18 43 CC(=O)N[C@@H]1CCN(Cc2ccc([C@@H](C)C(=O)O)cc2)C1 ZINC000217889836 CD For-Sale Unstable SIGMAR1 33 45 CC(=O)N[C@@H]1CCN(Cc2ccc([C@@H](C)C(=O)O)cc2)C1 ZINC000217889836 CD For-Sale Unstable CCR3 29 45 CC(=O)N[C@@H]1CCN(Cc2ccc([C@@H](C)C(=O)O)cc2)C1 ZINC000217889836 CD For-Sale Unstable CCR5 26 40 CC(=O)N[C@@H]1CCN(Cc2ccc([C@@H](C)C(=O)O)cc2)C1 ZINC000217889836 CD For-Sale Unstable UTS2R 23 41 CC(=O)N[C@@H]1CCN(Cc2ccc([C@@H](C)C(=O)O)cc2)C1 ZINC000217889836 CD For-Sale Unstable MLNR 36 44 CC(=O)N[C@@H]1CCN(Cc2ccc([C@@H](C)C(=O)O)cc2)C1 ZINC000217889836 CD For-Sale Unstable CCR2 16 42 CC(=O)N[C@@H]1CCN(Cc2ccc([C@@H](C)C(=O)O)cc2)C1 ZINC000217889836 CD For-Sale Unstable MCHR1 44 49 CC(=O)N[C@@H]1CCN(Cc2ccc([C@@H](C)C(=O)O)cc2)C1 ZINC000217889836 CD For-Sale Unstable BIRC2 62 37 CC(=O)N[C@@H]1CCN(Cc2ccc([C@@H](C)C(=O)O)cc2)C1 ZINC000217889836 CD For-Sale Unstable SLC22A20 0 43 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc(OCc3cccnc3)c2)CC(=O)O4)cc1O ZINC000217889863 KK In-Stock Unstable CYP1A1 30 41 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc(OCc3cccnc3)c2)CC(=O)O4)cc1O ZINC000217889863 KK In-Stock Unstable CYP1A2 25 40 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC1CCSCC1 ZINC000217889884 CH On-Demand Unstable TRPM8 17 43 CC[C@@H](NC(=O)/C=C/c1cccc([N+](=O)[O-])c1)c1ccc(C)cc1C ZINC000217889885 EI In-Stock Unstable CACNA1D 42 34 CC[C@@H](NC(=O)/C=C/c1cccc([N+](=O)[O-])c1)c1ccc(C)cc1C ZINC000217889885 EI In-Stock Unstable TRPM8 0 58 CS(=O)(=O)N1CCC(C(=O)Nc2ccc(-c3nc4ccccc4s3)cn2)CC1 ZINC000217889893 HF On-Demand Unstable FAAH 0 47 CS(=O)(=O)N1CCC(C(=O)Nc2ccc(-c3nc4ccccc4s3)cn2)CC1 ZINC000217889893 HF On-Demand Unstable EPHX2 24 41 CS(=O)(=O)N1CCC(C(=O)Nc2ccc(-c3nc4ccccc4s3)cn2)CC1 ZINC000217889893 HF On-Demand Unstable APEX1 0 42 CN(C[C@@H]1COCCO1)C(=O)c1cccc(O)c1 ZINC000217889915 CC In-Stock Unstable HSD17B2 25 43 O=C(O)C[C@@H](NC(=O)c1cc(O)ccc1O)C(=O)O ZINC000217889920 CB For-Sale Unstable FOLH1 27 43 CC(C)[C@@H](NC(=O)OCc1ccc(Cl)cc1)C(=O)O ZINC000217889926 CF For-Sale Unstable ELANE 38 46 CC(C)[C@@H](NC(=O)OCc1ccc(Cl)cc1)C(=O)O ZINC000217889926 CF For-Sale Unstable MME 44 43 CC(C)[C@@H](NC(=O)OCc1ccc(Cl)cc1)C(=O)O ZINC000217889926 CF For-Sale Unstable CASP3 26 64 CC(C)[C@@H](NC(=O)OCc1ccc(Cl)cc1)C(=O)O ZINC000217889926 CF For-Sale Unstable BMP1 70 42 CC(C)[C@@H](NC(=O)OCc1ccc(Cl)cc1)C(=O)O ZINC000217889926 CF For-Sale Unstable KLK3 79 37 CC(C)[C@@H](NC(=O)OCc1ccc(Cl)cc1)C(=O)O ZINC000217889926 CF For-Sale Unstable CTSB 60 52 CC(C)[C@@H](NC(=O)OCc1ccc(Cl)cc1)C(=O)O ZINC000217889926 CF For-Sale Unstable PAPA1_CARPA 80 44 CC(C)[C@@H](NC(=O)OCc1ccc(Cl)cc1)C(=O)O ZINC000217889926 CF For-Sale Unstable CYSP_TRYCR 49 39 CC(C)[C@@H](NC(=O)OCc1ccc(Cl)cc1)C(=O)O ZINC000217889926 CF For-Sale Unstable CTSK 35 52 CC(C)[C@@H](NC(=O)OCc1ccc(Cl)cc1)C(=O)O ZINC000217889926 CF For-Sale Unstable CTSL 37 52 CC(C)[C@@H](NC(=O)OCc1ccc(Cl)cc1)C(=O)O ZINC000217889926 CF For-Sale Unstable CCR1 44 37 CC(C)[C@@H](NC(=O)OCc1ccc(Cl)cc1)C(=O)O ZINC000217889926 CF For-Sale Unstable PGA 24 47 CC(C)[C@@H](NC(=O)OCc1ccc(Cl)cc1)C(=O)O ZINC000217889926 CF For-Sale Unstable CAPNS1 67 40 CC(C)[C@@H](NC(=O)OCc1ccc(Cl)cc1)C(=O)O ZINC000217889926 CF For-Sale Unstable HLA-DRB1 44 41 CC(C)[C@@H](NC(=O)OCc1ccc(Cl)cc1)C(=O)O ZINC000217889926 CF For-Sale Unstable CTSS 15 43 CC(C)[C@@H](NC(=O)OCc1ccc(Cl)cc1)C(=O)O ZINC000217889926 CF For-Sale Unstable CAPN1 82 51 CC(C)[C@@H](NC(=O)OCc1ccc(Cl)cc1)C(=O)O ZINC000217889926 CF For-Sale Unstable CASP1 29 52 CC(C)[C@@H](NC(=O)OCc1ccc(Cl)cc1)C(=O)O ZINC000217889926 CF For-Sale Unstable CTRC 15 42 CC(C)[C@@H](NC(=O)OCc1ccc(Cl)cc1)C(=O)O ZINC000217889926 CF For-Sale Unstable CAPN2 122 51 CC(C)[C@@H](NC(=O)OCc1ccc(Cl)cc1)C(=O)O ZINC000217889926 CF For-Sale Unstable ACE2 41 34 CC(C)[C@@H](NC(=O)OCc1ccc(Cl)cc1)C(=O)O ZINC000217889926 CF For-Sale Unstable CASP6 28 49 CC(C)[C@@H](NC(=O)OCc1ccc(Cl)cc1)C(=O)O ZINC000217889926 CF For-Sale Unstable CASP9 45 49 CC(C)[C@@H](NC(=O)OCc1ccc(Cl)cc1)C(=O)O ZINC000217889926 CF For-Sale Unstable TPSAB1 44 45 CC(C)[C@@H](NC(=O)OCc1ccc(Cl)cc1)C(=O)O ZINC000217889926 CF For-Sale Unstable ADAMTS4 55 38 CC(C)[C@@H](NC(=O)OCc1ccc(Cl)cc1)C(=O)O ZINC000217889926 CF For-Sale Unstable FPR1 24 41 CC(C)[C@@H](NC(=O)OCc1ccc(Cl)cc1)C(=O)O ZINC000217889926 CF For-Sale Unstable NPR 69 47 CC(C)[C@@H](NC(=O)OCc1ccc(Cl)cc1)C(=O)O ZINC000217889926 CF For-Sale Unstable PSMB5 34 41 Cc1cccc(/C=C/NC(=O)Nc2cc([N+](=O)[O-])ccc2Cl)c1 ZINC000217889932 EI For-Sale Unstable DDX3X 0 40 Cc1cccc(/C=C/NC(=O)Nc2cc([N+](=O)[O-])ccc2Cl)c1 ZINC000217889932 EI For-Sale Unstable TRPM8 0 52 COc1ccc(/C=C\C(=O)O)cc1CSc1ccccn1 ZINC000217889938 DG For-Sale Unstable PTGER2 30 44 COc1ccc(/C=C\C(=O)O)cc1CSc1ccccn1 ZINC000217889938 DG For-Sale Unstable PTGER4 0 44 COc1ccc(/C=C\C(=O)O)cc1CSc1ccccn1 ZINC000217889938 DG For-Sale Unstable AKR1C3 32 43 COc1ccc(/C=C\C(=O)O)cc1CSc1ccccn1 ZINC000217889938 DG For-Sale Unstable PTPA 0 40 CC[C@H](NC(=O)/C=C/c1cccc([N+](=O)[O-])c1)c1ccc(C)cc1C ZINC000217889956 EI In-Stock Unstable CACNA1D 42 34 CC[C@H](NC(=O)/C=C/c1cccc([N+](=O)[O-])c1)c1ccc(C)cc1C ZINC000217889956 EI In-Stock Unstable TRPM8 0 58 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC1CCSCC1 ZINC000217889965 CH For-Sale Unstable TRPM8 0 43 C[C@@H](C(=O)O)c1ccc(CN2CC[C@@H](C(C)(C)C)C2)cc1 ZINC000217889977 CH For-Sale Unstable PTGS1 28 49 C[C@@H](C(=O)O)c1ccc(CN2CC[C@@H](C(C)(C)C)C2)cc1 ZINC000217889977 CH For-Sale Unstable PTGS2 0 49 C[C@@H](C(=O)O)c1ccc(CN2CC[C@@H](C(C)(C)C)C2)cc1 ZINC000217889977 CH For-Sale Unstable CYP2J2 48 34 COC(=O)[C@H](CC(C)C)NC(=O)CC[C@H]1NC(=O)c2ccccc2NC1=O ZINC000217889982 GD In-Stock Unstable NPR 43 36 CN(C[C@H]1COCCO1)C(=O)c1cccc(O)c1 ZINC000217889998 CC In-Stock Unstable HSD17B2 25 43 COc1ccc(/C=C\C(=O)O)cc1CSc1ncccn1 ZINC000217890011 DF For-Sale Unstable PTGER2 23 44 COc1ccc(/C=C\C(=O)O)cc1CSc1ncccn1 ZINC000217890011 DF For-Sale Unstable TUBB1 52 41 COc1ccc(/C=C\C(=O)O)cc1CSc1ncccn1 ZINC000217890011 DF For-Sale Unstable AKR1C3 41 42 COc1ccc(/C=C\C(=O)O)cc1CSc1ncccn1 ZINC000217890011 DF For-Sale Unstable ABCG2 16 40 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC1CCSCC1 ZINC000217890035 CH For-Sale Unstable TRPM8 0 43 COc1ccccc1NC(=O)NCCn1ccc(-c2ccsc2)n1 ZINC000217890037 EG In-Stock Unstable ACAT 0 42 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](C(C)(C)C)C2)cc1 ZINC000217890058 CH For-Sale Unstable PTGS1 28 49 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](C(C)(C)C)C2)cc1 ZINC000217890058 CH For-Sale Unstable PTGS2 0 49 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](C(C)(C)C)C2)cc1 ZINC000217890058 CH For-Sale Unstable CYP2J2 48 34 CC[C@@H](NC(=O)/C=C/c1cccc([N+](=O)[O-])c1)c1ccc(OC)c(OC)c1 ZINC000217890068 FH In-Stock Unstable CACNA1C 41 35 CC[C@@H](NC(=O)/C=C/c1cccc([N+](=O)[O-])c1)c1ccc(OC)c(OC)c1 ZINC000217890068 FH In-Stock Unstable CACNA1D 76 35 CC[C@@H](NC(=O)/C=C/c1cccc([N+](=O)[O-])c1)c1ccc(OC)c(OC)c1 ZINC000217890068 FH In-Stock Unstable TRPM8 0 58 COc1ccc(CSc2ncccn2)cc1/C=C\C(=O)O ZINC000217890093 DF For-Sale Unstable PTGER3 20 47 COc1ccc(CSc2ncccn2)cc1/C=C\C(=O)O ZINC000217890093 DF For-Sale Unstable LTB4R 43 44 COc1ccc(CSc2ncccn2)cc1/C=C\C(=O)O ZINC000217890093 DF For-Sale Unstable TNFRSF1A 34 40 COc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)Nc1ccccc1O)C(=O)OC2 ZINC000217890095 HH In-Stock Unstable IMPDH1 0 85 COc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)Nc1ccccc1O)C(=O)OC2 ZINC000217890095 HH In-Stock Unstable IMPDH2 0 85 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC1Cc2ccccc2C1 ZINC000217890143 CI For-Sale Unstable TRPM8 17 49 O=C(NCCn1ccc(-c2ccsc2)n1)Nc1ccc2c(c1)OCO2 ZINC000217890145 FG In-Stock Unstable DYRK2 44 34 CC[C@H](NC(=O)/C=C/c1cccc([N+](=O)[O-])c1)c1ccc(OC)c(OC)c1 ZINC000217890146 FH In-Stock Unstable CACNA1C 41 35 CC[C@H](NC(=O)/C=C/c1cccc([N+](=O)[O-])c1)c1ccc(OC)c(OC)c1 ZINC000217890146 FH In-Stock Unstable CACNA1D 76 35 CC[C@H](NC(=O)/C=C/c1cccc([N+](=O)[O-])c1)c1ccc(OC)c(OC)c1 ZINC000217890146 FH In-Stock Unstable TRPM8 0 58 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc(OC)c(OC)c1 ZINC000217890222 HF For-Sale Unstable PDE4D 15 44 C[C@H](C(=O)O)c1ccc(CN(C)[C@@H](C)CO)cc1 ZINC000217890224 CD For-Sale Unstable PTGS1 33 54 C[C@H](C(=O)O)c1ccc(CN(C)[C@@H](C)CO)cc1 ZINC000217890224 CD For-Sale Unstable PTGS2 24 54 C[C@H](C(=O)O)c1ccc(CN(C)[C@@H](C)CO)cc1 ZINC000217890224 CD For-Sale Unstable SLC22A20 0 54 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC1Cc2ccccc2C1 ZINC000217890231 CI For-Sale Unstable TRPM8 17 49 O=C(O)/C=C\c1ccccc1CSc1cc(F)ccc1F ZINC000217890250 DI For-Sale Unstable PTGER2 40 50 O=C(O)/C=C\c1ccccc1CSc1cc(F)ccc1F ZINC000217890250 DI For-Sale Unstable PTGER4 18 41 O=C(O)/C=C\c1ccccc1CSc1cc(F)ccc1F ZINC000217890250 DI For-Sale Unstable PTGER3 19 47 O=C(O)/C=C\c1ccccc1CSc1cc(F)ccc1F ZINC000217890250 DI For-Sale Unstable PTGDR 0 47 CC[C@@H](NC(=O)/C=C/c1cccc([N+](=O)[O-])c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217890290 GG In-Stock Unstable TRPM8 0 52 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc(OC)c(OC)c1 ZINC000217890306 HF For-Sale Unstable PDE4D 15 44 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC1Cc2ccccc2C1 ZINC000217890317 CI For-Sale Unstable TRPM8 17 49 O=C(O)/C=C\c1ccc(CSc2cc(F)ccc2F)cc1 ZINC000217890351 DI For-Sale Unstable AKR1C3 31 41 CC[C@H](NC(=O)/C=C/c1cccc([N+](=O)[O-])c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217890370 GG In-Stock Unstable TRPM8 0 52 COC(=O)c1nc(NC(=O)CC/C(C)=C/Cc2c(O)c3c(c(C)c2OC)COC3=O)sc1CC(C)C ZINC000217890376 KJ In-Stock Unstable IMPDH2 81 53 Oc1cccc2c1CC[C@@H]2N1CCC[C@@H](C(F)(F)F)C1 ZINC000217890379 CH For-Sale Unstable SLC6A1 0 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc(OC)c(OC)c1 ZINC000217890396 HF For-Sale Unstable PDE4D 15 44 Cc1cccc(/C=C/NC(=O)Nc2ccccc2O)c1 ZINC000217890400 CG For-Sale Unstable MMP2 0 52 Cc1cccc(/C=C/NC(=O)Nc2ccccc2O)c1 ZINC000217890400 CG For-Sale Unstable MMP9 0 52 Cc1cccc(/C=C/NC(=O)Nc2ccccc2O)c1 ZINC000217890400 CG For-Sale Unstable MMP1 22 52 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC1Cc2ccccc2C1 ZINC000217890420 CI For-Sale Unstable TRPM8 17 49 O=C(O)/C=C\c1cccc(CSc2cc(F)ccc2F)c1 ZINC000217890431 DI For-Sale Unstable HCAR2 0 41 O=C(O)/C=C\c1cccc(CSc2cc(F)ccc2F)c1 ZINC000217890431 DI For-Sale Unstable AKR1C3 33 44 Oc1cccc2c1CC[C@H]2N1CCC[C@@H](C(F)(F)F)C1 ZINC000217890459 CH For-Sale Unstable SLC6A1 0 40 C[C@H]1CN(Cc2ccc([C@H](C)C(=O)O)cc2)CCS1 ZINC000217890467 CF For-Sale Unstable PTGS1 22 44 C[C@H]1CN(Cc2ccc([C@H](C)C(=O)O)cc2)CCS1 ZINC000217890467 CF For-Sale Unstable PTGS2 0 44 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc(OC)c(OC)c1 ZINC000217890477 HF For-Sale Unstable PDE4D 15 44 COc1cc2c(cc1OC)CN(C(=O)CCn1c3c(c4ccccc41)CCCC3)CC2 ZINC000217890508 HJ In-Stock Unstable FABI 65 42 COc1cc2c(cc1OC)CN(C(=O)CCn1c3c(c4ccccc41)CCCC3)CC2 ZINC000217890508 HJ In-Stock Unstable HTR7 17 44 COc1cc2c(cc1OC)CN(C(=O)CCn1c3c(c4ccccc41)CCCC3)CC2 ZINC000217890508 HJ In-Stock Unstable FABP4 62 43 COc1cc2c(cc1OC)CN(C(=O)CCn1c3c(c4ccccc41)CCCC3)CC2 ZINC000217890508 HJ In-Stock Unstable ABCB1B 65 38 COc1cc2c(cc1OC)CN(C(=O)CCn1c3c(c4ccccc41)CCCC3)CC2 ZINC000217890508 HJ In-Stock Unstable ABCB1 26 48 COc1cc2c(cc1OC)CN(C(=O)CCn1c3c(c4ccccc41)CCCC3)CC2 ZINC000217890508 HJ In-Stock Unstable HCRTR2 15 43 COc1cc2c(cc1OC)CN(C(=O)CCn1c3c(c4ccccc41)CCCC3)CC2 ZINC000217890508 HJ In-Stock Unstable SCARB1 46 36 Cc1cccc(-c2noc(CNC(=O)/C=C/c3cccc([N+](=O)[O-])c3)n2)c1 ZINC000217890513 FG In-Stock Unstable CACNA1D 56 33 Cc1cccc(-c2noc(CNC(=O)/C=C/c3cccc([N+](=O)[O-])c3)n2)c1 ZINC000217890513 FG In-Stock Unstable HDAC8 49 34 Cc1cccc(-c2noc(CNC(=O)/C=C/c3cccc([N+](=O)[O-])c3)n2)c1 ZINC000217890513 FG In-Stock Unstable TRPM8 0 53 Cc1cc(CN[C@H]2C[C@H](C)CC[C@H]2C(C)C)cc(C)c1O ZINC000217890528 CJ For-Sale Unstable TRPM8 17 44 CCOc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217890529 CI For-Sale Unstable SCN2A 24 42 Cc1cccc(SCc2ccccc2/C=C\C(=O)O)c1 ZINC000217890532 CI For-Sale Unstable PTGER2 16 49 Cc1cccc(SCc2ccccc2/C=C\C(=O)O)c1 ZINC000217890532 CI For-Sale Unstable PTGER4 26 48 Cc1cccc(SCc2ccccc2/C=C\C(=O)O)c1 ZINC000217890532 CI For-Sale Unstable PTGER3 20 51 Cc1cccc(SCc2ccccc2/C=C\C(=O)O)c1 ZINC000217890532 CI For-Sale Unstable PTGDR 0 51 Cc1cc(CN[C@H]2C[C@@H](C)CC[C@H]2C(C)C)cc(C)c1O ZINC000217890579 CJ For-Sale Unstable TRPM8 17 44 Cc1cccc(SCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217890584 CI For-Sale Unstable PTGER2 29 42 Cc1cccc(SCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217890584 CI For-Sale Unstable LTB4R 23 40 Cc1cccc(SCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217890584 CI For-Sale Unstable AKR1C3 34 42 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1cccc(OC)c1 ZINC000217890602 HE For-Sale Unstable DRD4 40 31 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1cccc(OC)c1 ZINC000217890602 HE For-Sale Unstable COLA 81 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1cccc(OC)c1 ZINC000217890602 HE For-Sale Unstable CPT1A 70 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1cccc(OC)c1 ZINC000217890602 HE For-Sale Unstable CPT2 36 40 Cc1ccc(-c2noc(CNC(=O)/C=C/c3cccc([N+](=O)[O-])c3)n2)cc1 ZINC000217890629 FG In-Stock Unstable CACNA1D 61 34 Cc1ccc(-c2noc(CNC(=O)/C=C/c3cccc([N+](=O)[O-])c3)n2)cc1 ZINC000217890629 FG In-Stock Unstable HDAC8 46 33 Cc1ccc(-c2noc(CNC(=O)/C=C/c3cccc([N+](=O)[O-])c3)n2)cc1 ZINC000217890629 FG In-Stock Unstable TRPM8 0 52 COC(=O)COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)ccc1OC ZINC000217890630 KH In-Stock Unstable AKR1B1 0 45 COC(=O)COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)ccc1OC ZINC000217890630 KH In-Stock Unstable CYP1B1 47 34 COC(=O)COc1cc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)ccc1OC ZINC000217890630 KH In-Stock Unstable CYP1A1 33 43 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](C)[C@@H](C)C2)cc1 ZINC000217890637 CG For-Sale Unstable ACHE 18 40 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](C)[C@@H](C)C2)cc1 ZINC000217890637 CG For-Sale Unstable PTGS1 31 48 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](C)[C@@H](C)C2)cc1 ZINC000217890637 CG For-Sale Unstable PTGS2 22 48 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](C)[C@@H](C)C2)cc1 ZINC000217890637 CG For-Sale Unstable SIGMAR1 40 38 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](C)[C@@H](C)C2)cc1 ZINC000217890637 CG For-Sale Unstable MLNR 50 42 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](C)[C@@H](C)C2)cc1 ZINC000217890637 CG For-Sale Unstable SLC22A20 0 47 CCOCCOCc1cc(/C=C\C(=O)O)ccc1OC ZINC000217890668 CE For-Sale Unstable TUBB1 47 38 CCOCCOCc1cc(/C=C\C(=O)O)ccc1OC ZINC000217890668 CE For-Sale Unstable AKR1C3 31 42 CCOCCOCc1cc(/C=C\C(=O)O)ccc1OC ZINC000217890668 CE For-Sale Unstable ABCG2 16 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1cccc(OC)c1 ZINC000217890677 HE For-Sale Unstable DRD4 40 31 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1cccc(OC)c1 ZINC000217890677 HE For-Sale Unstable COLA 81 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1cccc(OC)c1 ZINC000217890677 HE For-Sale Unstable CPT1A 70 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1cccc(OC)c1 ZINC000217890677 HE For-Sale Unstable CPT2 36 40 CC(=O)c1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217890712 CH For-Sale Unstable MMP1 0 43 CC(=O)c1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217890712 CH For-Sale Unstable AKR1C3 15 42 CC(=O)c1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217890712 CH For-Sale Unstable KCNK3 53 38 CC(=O)c1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217890712 CH For-Sale Unstable KCNK9 42 38 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1cccc(OC)c1 ZINC000217890728 HE For-Sale Unstable DRD4 40 31 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1cccc(OC)c1 ZINC000217890728 HE For-Sale Unstable COLA 81 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1cccc(OC)c1 ZINC000217890728 HE For-Sale Unstable CPT1A 70 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1cccc(OC)c1 ZINC000217890728 HE For-Sale Unstable CPT2 36 40 COC(=O)COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)ccc1OC ZINC000217890738 KH In-Stock Unstable AKR1B1 0 45 COC(=O)COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)ccc1OC ZINC000217890738 KH In-Stock Unstable CYP1B1 47 34 COC(=O)COc1cc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(OC)c(O)c5)oc4c32)ccc1OC ZINC000217890738 KH In-Stock Unstable CYP1A1 33 43 COc1cccc(-c2noc(CNC(=O)/C=C/c3cccc([N+](=O)[O-])c3)n2)c1 ZINC000217890740 GF In-Stock Unstable CACNA1D 60 34 COc1cccc(-c2noc(CNC(=O)/C=C/c3cccc([N+](=O)[O-])c3)n2)c1 ZINC000217890740 GF In-Stock Unstable TRPM8 0 57 CC(C)(C)OC(=O)N1CC[C@H](N)[C@H](C(C)(C)C)C1 ZINC000217890752 CF For-Sale Unstable GPR119 42 44 COc1ccc(CNC(=O)NCCn2ccc(-c3ccsc3)n2)cc1 ZINC000217890756 FG In-Stock Unstable PROKR1 51 32 CCOCCOCc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217890762 CE For-Sale Unstable PTGER3 18 47 CCOCCOCc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217890762 CE For-Sale Unstable AKR1B10 32 43 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NS(=O)(=O)C(C)C ZINC000217890789 CF For-Sale Unstable TRPM8 15 44 C[C@H](C(=O)O)c1ccc(CN2CCS[C@@H](C)[C@@H]2C)cc1 ZINC000217890792 CG For-Sale Unstable PTGS1 24 45 C[C@H](C(=O)O)c1ccc(CN2CCS[C@@H](C)[C@@H]2C)cc1 ZINC000217890792 CG For-Sale Unstable PTGS2 0 45 C[C@H](C(=O)O)c1ccc(CN2CCS[C@@H](C)[C@@H]2C)cc1 ZINC000217890792 CG For-Sale Unstable SLC22A20 0 45 CC(=O)c1cccc(NC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217890804 CH For-Sale Unstable CCKAR 0 47 CC(=O)c1cccc(NC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217890804 CH For-Sale Unstable CCR3 17 41 CC(=O)c1cccc(NC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217890804 CH For-Sale Unstable AKR1C3 30 48 CC(=O)c1cccc(NC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217890804 CH For-Sale Unstable KCNK3 107 48 CC(=O)c1cccc(NC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217890804 CH For-Sale Unstable KCNK9 60 48 CC(C)(C)OC(=O)N1CC[C@H](N)[C@@H](C(C)(C)C)C1 ZINC000217890830 CF For-Sale Unstable GPR119 42 44 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1cccc(OC)c1 ZINC000217890834 HE For-Sale Unstable DRD4 40 31 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1cccc(OC)c1 ZINC000217890834 HE For-Sale Unstable COLA 81 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1cccc(OC)c1 ZINC000217890834 HE For-Sale Unstable CPT1A 70 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1cccc(OC)c1 ZINC000217890834 HE For-Sale Unstable CPT2 36 40 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NS(=O)(=O)C(C)C ZINC000217890852 CF For-Sale Unstable TRPM8 15 44 O=C(NCCn1ccc(-c2ccsc2)n1)Nc1cccc(C(F)(F)F)c1 ZINC000217890871 GI In-Stock Unstable BRAF 23 42 COc1ccc(-c2noc(CNC(=O)/C=C/c3cccc([N+](=O)[O-])c3)n2)cc1 ZINC000217890883 GF In-Stock Unstable CACNA1D 61 36 COc1ccc(-c2noc(CNC(=O)/C=C/c3cccc([N+](=O)[O-])c3)n2)cc1 ZINC000217890883 GF In-Stock Unstable TRPM8 0 53 COc1ccc(-c2noc(CNC(=O)/C=C/c3cccc([N+](=O)[O-])c3)n2)cc1 ZINC000217890883 GF In-Stock Unstable EXSA 0 43 C[C@H](CCCC(N)=O)c1ccccc1 ZINC000217890891 AE For-Sale Unstable C3AR1 55 39 C[C@H](CCCC(N)=O)c1ccccc1 ZINC000217890891 AE For-Sale Unstable AOC3 17 43 CC(C)(C)OC(=O)N1CC[C@@H](N)[C@H](C(C)(C)C)C1 ZINC000217890912 CF For-Sale Unstable GPR119 42 44 CCSc1ccccc1C(=O)N1C[C@H](Oc2ccccc2F)C[C@@H]1C(=O)OC ZINC000217890921 HH For-Sale Unstable HCRTR1 40 35 CCSc1ccccc1C(=O)N1C[C@H](Oc2ccccc2F)C[C@@H]1C(=O)OC ZINC000217890921 HH For-Sale Unstable HCRTR2 43 35 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NS(=O)(=O)C(C)C ZINC000217890939 CF For-Sale Unstable TRPM8 15 44 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)Nc3ccc4cc[nH]c4c3)[C@H]21 ZINC000217890977 JI In-Stock Unstable TSHR 50 34 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)Nc3ccc4cc[nH]c4c3)[C@H]21 ZINC000217890977 JI In-Stock Unstable ENPP1 70 36 COc1ccc(-c2noc(CNC(=O)/C=C/c3cccc([N+](=O)[O-])c3)n2)c(OC)c1 ZINC000217890983 HF In-Stock Unstable TRPM8 0 51 CC(C)(C)OC(=O)N1CC[C@@H](N)[C@@H](C(C)(C)C)C1 ZINC000217890988 CF For-Sale Unstable GPR119 42 44 CCSc1ccccc1C(=O)N1C[C@@H](Oc2ccccc2F)C[C@@H]1C(=O)OC ZINC000217890998 HH For-Sale Unstable HCRTR1 40 35 CCSc1ccccc1C(=O)N1C[C@@H](Oc2ccccc2F)C[C@@H]1C(=O)OC ZINC000217890998 HH For-Sale Unstable HCRTR2 43 35 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)Nc3ccc4cc[nH]c4c3)[C@@H]21 ZINC000217891025 JI In-Stock Unstable TSHR 50 34 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)Nc3ccc4cc[nH]c4c3)[C@@H]21 ZINC000217891025 JI In-Stock Unstable ENPP1 70 36 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NS(=O)(=O)C(C)C ZINC000217891038 CF For-Sale Unstable TRPM8 15 44 CCSc1ccccc1C(=O)N1C[C@H](Oc2ccccc2F)C[C@H]1C(=O)OC ZINC000217891060 HH For-Sale Unstable HCRTR1 40 35 CCSc1ccccc1C(=O)N1C[C@H](Oc2ccccc2F)C[C@H]1C(=O)OC ZINC000217891060 HH For-Sale Unstable HCRTR2 43 35 O=C(/C=C/c1cccc([N+](=O)[O-])c1)NCc1nc(-c2ccccc2Cl)no1 ZINC000217891080 GH In-Stock Unstable TRPM8 0 56 Cc1ccc(Cn2nccc2NC(=O)c2ccc(-c3cccs3)nc2C)cc1 ZINC000217891096 GJ On-Demand Unstable GPR142 40 32 CCSc1ccccc1C(=O)N1C[C@@H](Oc2ccccc2F)C[C@H]1C(=O)OC ZINC000217891174 HH For-Sale Unstable HCRTR1 40 35 CCSc1ccccc1C(=O)N1C[C@@H](Oc2ccccc2F)C[C@H]1C(=O)OC ZINC000217891174 HH For-Sale Unstable HCRTR2 43 35 O=C([C@@H]1CCCN(S(=O)(=O)c2ccc(Br)cc2)C1)N1CCC[C@@H](O)C1 ZINC000217891182 ID On-Demand Unstable TGM2 15 41 O=C([C@@H]1CCCN(S(=O)(=O)c2ccc(Br)cc2)C1)N1CCC[C@@H](O)C1 ZINC000217891182 ID On-Demand Unstable F13A1 23 41 O=C([C@@H]1CCCN(S(=O)(=O)c2ccc(Br)cc2)C1)N1CCC[C@@H](O)C1 ZINC000217891182 ID On-Demand Unstable AKR1C1 24 47 O=C([C@@H]1CCCN(S(=O)(=O)c2ccc(Br)cc2)C1)N1CCC[C@@H](O)C1 ZINC000217891182 ID On-Demand Unstable NAMPT 22 45 CN(C(=O)c1c(F)cccc1Cl)c1ccc(-c2cc(C(N)=O)ccc2Cl)cc1 ZINC000217891191 HK Annotated Unstable GPBAR1 40 46 O=C(/C=C/c1cccc([N+](=O)[O-])c1)NCc1nc(-c2ccc(Cl)cc2)no1 ZINC000217891197 GH In-Stock Unstable TRPM8 0 50 CCCCOc1ccc(NC(=O)NCCn2ccc(-c3ccsc3)n2)cc1 ZINC000217891207 GJ In-Stock Unstable PLA2G4B 46 32 C[C@H]1CN(Cc2ccc([C@H](C)C(=O)O)cc2)CCC1=O ZINC000217891209 CE For-Sale Unstable PTGS1 24 52 C[C@H]1CN(Cc2ccc([C@H](C)C(=O)O)cc2)CCC1=O ZINC000217891209 CE For-Sale Unstable PTGS2 15 52 CC(C)C[C@@H](C)OCCOc1cccc(/C=C\C(=O)O)c1 ZINC000217891239 CH For-Sale Unstable AKR1C3 30 43 O=C([C@H]1CCCN(S(=O)(=O)c2ccc(Br)cc2)C1)N1CCC[C@@H](O)C1 ZINC000217891258 ID On-Demand Unstable TGM2 15 41 O=C([C@H]1CCCN(S(=O)(=O)c2ccc(Br)cc2)C1)N1CCC[C@@H](O)C1 ZINC000217891258 ID On-Demand Unstable F13A1 23 41 O=C([C@H]1CCCN(S(=O)(=O)c2ccc(Br)cc2)C1)N1CCC[C@@H](O)C1 ZINC000217891258 ID On-Demand Unstable AKR1C1 24 47 O=C([C@H]1CCCN(S(=O)(=O)c2ccc(Br)cc2)C1)N1CCC[C@@H](O)C1 ZINC000217891258 ID On-Demand Unstable NAMPT 22 45 C[C@H](C(=O)O)c1ccc(CN2C[C@H](C)N(C)[C@H](C)C2)cc1 ZINC000217891312 CE For-Sale Unstable PTGS1 15 41 C[C@H](C(=O)O)c1ccc(CN2C[C@H](C)N(C)[C@H](C)C2)cc1 ZINC000217891312 CE For-Sale Unstable MLNR 24 42 COc1ccc(C)cc1NC(=O)N/C=C/c1cccc(C)c1 ZINC000217891316 CI For-Sale Unstable KCNK3 31 41 COc1ccc(/C=C2\Oc3c(ccc4c3[C@H](c3ccc5c(c3)OCO5)CC(=O)O4)C2=O)cc1 ZINC000217891322 II In-Stock Unstable EDNRB 58 38 COc1ccc(/C=C2\Oc3c(ccc4c3[C@H](c3ccc5c(c3)OCO5)CC(=O)O4)C2=O)cc1 ZINC000217891322 II In-Stock Unstable EDNRA 52 38 O=C(/C=C/c1cccc([N+](=O)[O-])c1)NCc1nc(-c2cccc(Br)c2)no1 ZINC000217891327 IH In-Stock Unstable HDAC8 48 32 O=C(/C=C/c1cccc([N+](=O)[O-])c1)NCc1nc(-c2cccc(Br)c2)no1 ZINC000217891327 IH In-Stock Unstable TRPM8 0 54 CC(C)C[C@H](C)OCCOc1cccc(/C=C\C(=O)O)c1 ZINC000217891330 CH For-Sale Unstable AKR1C3 30 43 COc1ccc(/C=C2\Oc3c(ccc4c3[C@@H](c3ccc5c(c3)OCO5)CC(=O)O4)C2=O)cc1 ZINC000217891402 II In-Stock Unstable EDNRB 58 38 COc1ccc(/C=C2\Oc3c(ccc4c3[C@@H](c3ccc5c(c3)OCO5)CC(=O)O4)C2=O)cc1 ZINC000217891402 II In-Stock Unstable EDNRA 52 38 C[C@H](C(=O)O)c1ccc(CN2C[C@H](C)N(C)[C@@H](C)C2)cc1 ZINC000217891407 CE For-Sale Unstable PTGS1 15 41 C[C@H](C(=O)O)c1ccc(CN2C[C@H](C)N(C)[C@@H](C)C2)cc1 ZINC000217891407 CE For-Sale Unstable MLNR 24 42 CC(C)CCCOCCOc1cccc(/C=C\C(=O)O)c1 ZINC000217891416 CH For-Sale Unstable AKR1C3 29 41 Cc1cccc(/C=C/NC(=O)Nc2cccc(C)c2)c1 ZINC000217891448 CI For-Sale Unstable KIT 23 40 Cc1cccc(/C=C/NC(=O)Nc2cccc(C)c2)c1 ZINC000217891448 CI For-Sale Unstable CCKAR 23 48 Cc1cccc(/C=C/NC(=O)Nc2cccc(C)c2)c1 ZINC000217891448 CI For-Sale Unstable KDR 19 42 Cc1cccc(/C=C/NC(=O)Nc2cccc(C)c2)c1 ZINC000217891448 CI For-Sale Unstable MMP2 0 57 Cc1cccc(/C=C/NC(=O)Nc2cccc(C)c2)c1 ZINC000217891448 CI For-Sale Unstable MMP9 0 57 Cc1cccc(/C=C/NC(=O)Nc2cccc(C)c2)c1 ZINC000217891448 CI For-Sale Unstable IMPDH2 0 46 Cc1cccc(/C=C/NC(=O)Nc2cccc(C)c2)c1 ZINC000217891448 CI For-Sale Unstable MMP1 0 57 Cc1cccc(/C=C/NC(=O)Nc2cccc(C)c2)c1 ZINC000217891448 CI For-Sale Unstable PSBA 0 49 Cc1cccc(/C=C/NC(=O)Nc2cccc(C)c2)c1 ZINC000217891448 CI For-Sale Unstable KCNK3 76 45 Cc1cccc(/C=C/NC(=O)Nc2cccc(C)c2)c1 ZINC000217891448 CI For-Sale Unstable KCNK9 53 45 O=C(/C=C/c1cccc([N+](=O)[O-])c1)NCc1nc(-c2cccs2)no1 ZINC000217891451 FG In-Stock Unstable TRPM8 0 44 CCc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217891508 CH For-Sale Unstable ALOX5 16 42 CCc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217891508 CH For-Sale Unstable PTGER2 33 57 CCc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217891508 CH For-Sale Unstable PPIA 42 33 CCc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217891508 CH For-Sale Unstable PTGER1 57 42 CCc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217891508 CH For-Sale Unstable PTGER4 50 56 CCc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217891508 CH For-Sale Unstable PTGER3 37 56 CCc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217891508 CH For-Sale Unstable LTB4R 33 50 CCc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217891508 CH For-Sale Unstable ABCB1 15 42 CCc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217891508 CH For-Sale Unstable PTGDR 0 45 CCc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217891508 CH For-Sale Unstable AKR1C3 40 52 CN(Cc1nc(-c2ccccc2)no1)C(=O)/C=C/c1cccc([N+](=O)[O-])c1 ZINC000217891555 FG In-Stock Unstable FABI 40 30 CN(Cc1nc(-c2ccccc2)no1)C(=O)/C=C/c1cccc([N+](=O)[O-])c1 ZINC000217891555 FG In-Stock Unstable TRPM8 0 42 Cc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)c1 ZINC000217891566 FK For-Sale Unstable GUAB 0 49 Cc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)c1 ZINC000217891566 FK For-Sale Unstable RAF1 32 46 Cc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)c1 ZINC000217891566 FK For-Sale Unstable Q8MMZ8_EIMTE 52 46 Cc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)c1 ZINC000217891566 FK For-Sale Unstable BRAF 17 40 Cc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)c1 ZINC000217891566 FK For-Sale Unstable IMDH_CRYPV 39 52 Cc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)c1 ZINC000217891566 FK For-Sale Unstable BLM 0 44 Cc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)c1 ZINC000217891566 FK For-Sale Unstable KCNK3 42 39 O=C(O)/C=C\c1cccc(COc2ccc(CO)cc2)c1 ZINC000217891592 CF For-Sale Unstable ALOX5 16 48 O=C(O)/C=C\c1cccc(COc2ccc(CO)cc2)c1 ZINC000217891592 CF For-Sale Unstable MAOB 60 46 O=C(O)/C=C\c1cccc(COc2ccc(CO)cc2)c1 ZINC000217891592 CF For-Sale Unstable PTGER2 50 48 O=C(O)/C=C\c1cccc(COc2ccc(CO)cc2)c1 ZINC000217891592 CF For-Sale Unstable LTA4H 19 40 O=C(O)/C=C\c1cccc(COc2ccc(CO)cc2)c1 ZINC000217891592 CF For-Sale Unstable PTGER4 41 48 O=C(O)/C=C\c1cccc(COc2ccc(CO)cc2)c1 ZINC000217891592 CF For-Sale Unstable PTPN2 0 40 O=C(O)/C=C\c1cccc(COc2ccc(CO)cc2)c1 ZINC000217891592 CF For-Sale Unstable PTGER3 28 49 O=C(O)/C=C\c1cccc(COc2ccc(CO)cc2)c1 ZINC000217891592 CF For-Sale Unstable LTB4R 25 43 O=C(O)/C=C\c1cccc(COc2ccc(CO)cc2)c1 ZINC000217891592 CF For-Sale Unstable NR1H4 55 35 O=C(O)/C=C\c1cccc(COc2ccc(CO)cc2)c1 ZINC000217891592 CF For-Sale Unstable GYS1 47 34 O=C(O)/C=C\c1cccc(COc2ccc(CO)cc2)c1 ZINC000217891592 CF For-Sale Unstable FFAR1 70 47 O=C(O)/C=C\c1cccc(COc2ccc(CO)cc2)c1 ZINC000217891592 CF For-Sale Unstable AKR1C3 46 47 O=C(O)/C=C\c1cccc(COc2ccc(CO)cc2)c1 ZINC000217891592 CF For-Sale Unstable FFAR4 48 46 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc(C(F)(F)F)c1 ZINC000217891645 HH For-Sale Unstable CACNA1B 40 33 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc(C(F)(F)F)c1 ZINC000217891645 HH For-Sale Unstable CCR2 61 37 Cc1cccc(-c2noc(CN(C)C(=O)/C=C/c3cccc([N+](=O)[O-])c3)n2)c1 ZINC000217891649 GH In-Stock Unstable TRPM8 0 45 CCOc1ccccc1CCC(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217891650 CE On-Demand Unstable HCN1 41 33 CCOc1ccccc1CCC(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217891650 CE On-Demand Unstable HCN4 41 33 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc(C(F)(F)F)c1 ZINC000217891712 HH For-Sale Unstable CACNA1B 40 33 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc(C(F)(F)F)c1 ZINC000217891712 HH For-Sale Unstable CCR2 61 37 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc(C(F)(F)F)c1 ZINC000217891768 HH For-Sale Unstable CACNA1B 40 33 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc(C(F)(F)F)c1 ZINC000217891768 HH For-Sale Unstable CCR2 61 37 Cc1cccc(/C=C/NC(=O)Nc2ccc(N)c(Cl)c2)c1 ZINC000217891794 DI For-Sale Unstable KIT 24 40 Cc1cccc(/C=C/NC(=O)Nc2ccc(N)c(Cl)c2)c1 ZINC000217891794 DI For-Sale Unstable KDR 19 40 Cc1cccc(/C=C/NC(=O)Nc2ccc(N)c(Cl)c2)c1 ZINC000217891794 DI For-Sale Unstable KCNK3 41 36 O=C(O)/C=C\c1ccc(OCCOC2CCOCC2)cc1 ZINC000217891814 CE For-Sale Unstable HPGD 17 42 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)N1CCC(O)(c3ccc(Cl)cc3)CC1)C(=O)OC2 ZINC000217891839 KK In-Stock Unstable IMPDH1 0 56 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)N1CCC(O)(c3ccc(Cl)cc3)CC1)C(=O)OC2 ZINC000217891839 KK In-Stock Unstable IMPDH2 0 56 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc(C(F)(F)F)c1 ZINC000217891870 HH For-Sale Unstable CACNA1B 40 33 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc(C(F)(F)F)c1 ZINC000217891870 HH For-Sale Unstable CCR2 61 37 CCC[C@@H](O)CN[C@@H](C)C(=O)OC(C)(C)C ZINC000217891883 BD For-Sale Unstable ADRB2 0 40 CCC[C@@H](O)CN[C@@H](C)C(=O)OC(C)(C)C ZINC000217891883 BD For-Sale Unstable CTSK 0 40 CC(C)S(=O)(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000217891972 BC For-Sale Unstable GRIA4 21 41 CCC[C@H](O)CN[C@@H](C)C(=O)OC(C)(C)C ZINC000217892001 BD For-Sale Unstable ADRB2 0 40 CCC[C@H](O)CN[C@@H](C)C(=O)OC(C)(C)C ZINC000217892001 BD For-Sale Unstable CTSK 0 40 Cc1cccc(/C=C/NC(=O)Nc2cccc(Cl)c2)c1 ZINC000217892015 CI For-Sale Unstable CCKAR 15 41 Cc1cccc(/C=C/NC(=O)Nc2cccc(Cl)c2)c1 ZINC000217892015 CI For-Sale Unstable MMP1 0 53 Cc1cccc(/C=C/NC(=O)Nc2cccc(Cl)c2)c1 ZINC000217892015 CI For-Sale Unstable IMDH_CRYPV 15 42 Cc1cccc(/C=C/NC(=O)Nc2cccc(Cl)c2)c1 ZINC000217892015 CI For-Sale Unstable PSBA 0 46 Cc1cccc(/C=C/NC(=O)Nc2cccc(Cl)c2)c1 ZINC000217892015 CI For-Sale Unstable KCNK3 64 50 Cc1cccc(/C=C/NC(=O)Nc2cccc(Cl)c2)c1 ZINC000217892015 CI For-Sale Unstable KCNK9 46 50 CC(C)S(=O)(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000217892064 BC For-Sale Unstable GRIA4 21 41 CCC[C@@H](O)CN[C@H](C)C(=O)OC(C)(C)C ZINC000217892095 BD For-Sale Unstable ADRB2 0 40 CCC[C@@H](O)CN[C@H](C)C(=O)OC(C)(C)C ZINC000217892095 BD For-Sale Unstable CTSK 0 40 Cc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cc2)c1 ZINC000217892119 CI For-Sale Unstable GUAB 0 43 Cc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cc2)c1 ZINC000217892119 CI For-Sale Unstable MMP2 0 52 Cc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cc2)c1 ZINC000217892119 CI For-Sale Unstable MMP9 0 52 Cc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cc2)c1 ZINC000217892119 CI For-Sale Unstable MMP1 0 52 Cc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cc2)c1 ZINC000217892119 CI For-Sale Unstable IDO1 16 40 Cc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cc2)c1 ZINC000217892119 CI For-Sale Unstable IMDH_CRYPV 25 43 Cc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cc2)c1 ZINC000217892119 CI For-Sale Unstable P95276_MYCTO 0 42 Cc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cc2)c1 ZINC000217892119 CI For-Sale Unstable KCNK3 44 44 CSCC[C@@H](CO)NC(=O)Cc1c(C)c2ccc(O)cc2oc1=O ZINC000217892132 FD In-Stock Unstable HSD17B3 44 49 CSCC[C@@H](CO)NC(=O)Cc1c(C)c2ccc(O)cc2oc1=O ZINC000217892132 FD In-Stock Unstable NQO1 44 34 COc1ccc(CSc2ccccn2)cc1/C=C\C(=O)O ZINC000217892145 DG For-Sale Unstable PTGER2 48 47 COc1ccc(CSc2ccccn2)cc1/C=C\C(=O)O ZINC000217892145 DG For-Sale Unstable PTGER4 24 47 COc1ccc(CSc2ccccn2)cc1/C=C\C(=O)O ZINC000217892145 DG For-Sale Unstable PTGER3 22 42 COc1ccc(CSc2ccccn2)cc1/C=C\C(=O)O ZINC000217892145 DG For-Sale Unstable LTB4R 43 45 COc1ccc(CSc2ccccn2)cc1/C=C\C(=O)O ZINC000217892145 DG For-Sale Unstable AKR1B10 29 40 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](O)[C@@H](C)C2)cc1 ZINC000217892156 CE For-Sale Unstable ACHE 15 40 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](O)[C@@H](C)C2)cc1 ZINC000217892156 CE For-Sale Unstable SIGMAR1 40 37 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](O)[C@@H](C)C2)cc1 ZINC000217892156 CE For-Sale Unstable SLC18A3 25 40 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](O)[C@@H](C)C2)cc1 ZINC000217892156 CE For-Sale Unstable MLNR 50 42 CCC[C@H](O)CN[C@H](C)C(=O)OC(C)(C)C ZINC000217892165 BD For-Sale Unstable ADRB2 0 40 CCC[C@H](O)CN[C@H](C)C(=O)OC(C)(C)C ZINC000217892165 BD For-Sale Unstable CTSK 0 40 Cc1cn2c(CN(C)C(=O)c3ccc(S(=O)(=O)N(C)C(C)C)cc3)c(C)nc2s1 ZINC000217892207 IG On-Demand Unstable LIMK2 35 40 CC[C@@H](C)[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(CCc2ccccc2)C1=O ZINC000217892217 FD In-Stock Unstable GALR1 47 34 O=C(O)/C=C\c1ccc(CSc2ccccn2)c(F)c1 ZINC000217892228 CH For-Sale Unstable AKR1C3 30 41 O=C(c1cc2c([nH]c1=O)CCC2)N1CCC[C@@H]1c1nc2cc(F)ccc2[nH]1 ZINC000217892269 FF In-Stock Unstable PRCP 48 39 C[C@@H](C(=O)O)c1ccc(CN2CC[C@@H](CCO)C2)cc1 ZINC000217892282 CE For-Sale Unstable ACHE 38 41 C[C@@H](C(=O)O)c1ccc(CN2CC[C@@H](CCO)C2)cc1 ZINC000217892282 CE For-Sale Unstable SLC6A3 17 45 C[C@@H](C(=O)O)c1ccc(CN2CC[C@@H](CCO)C2)cc1 ZINC000217892282 CE For-Sale Unstable SIGMAR1 42 39 Cc1cccc(/C=C/NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000217892322 EG For-Sale Unstable DRD2 27 44 Cc1cccc(/C=C/NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000217892322 EG For-Sale Unstable DRD4 58 44 Cc1cccc(/C=C/NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000217892322 EG For-Sale Unstable ACHE 29 44 Cc1cccc(/C=C/NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000217892322 EG For-Sale Unstable CHRM3 17 50 Cc1cccc(/C=C/NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000217892322 EG For-Sale Unstable SIGMAR1 48 49 Cc1cccc(/C=C/NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000217892322 EG For-Sale Unstable HDAC8 40 37 Cc1cccc(/C=C/NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000217892322 EG For-Sale Unstable HDAC1 16 42 Cc1cccc(/C=C/NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000217892322 EG For-Sale Unstable FAAH 33 52 Cc1cccc(/C=C/NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000217892322 EG For-Sale Unstable MGLL 0 40 Cc1cccc(/C=C/NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000217892322 EG For-Sale Unstable GPR183 0 41 O=C(c1cc2c([nH]c1=O)CCC2)N1CCC[C@H]1c1nc2cc(F)ccc2[nH]1 ZINC000217892325 FF In-Stock Unstable PRCP 48 39 CN1CCN(CCNC(=O)[C@@H]2CCCN(S(=O)(=O)c3ccc(Br)cc3)C2)CC1 ZINC000217892344 JD On-Demand Unstable EPHX2 16 46 CN1CCN(CCNC(=O)[C@@H]2CCCN(S(=O)(=O)c3ccc(Br)cc3)C2)CC1 ZINC000217892344 JD On-Demand Unstable GPBAR1 18 42 CN1CCN(CCNC(=O)[C@@H]2CCCN(S(=O)(=O)c3ccc(Br)cc3)C2)CC1 ZINC000217892344 JD On-Demand Unstable AKR1C1 21 43 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](CCO)C2)cc1 ZINC000217892349 CE For-Sale Unstable ACHE 38 41 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](CCO)C2)cc1 ZINC000217892349 CE For-Sale Unstable SLC6A3 17 45 C[C@H](C(=O)O)c1ccc(CN2CC[C@@H](CCO)C2)cc1 ZINC000217892349 CE For-Sale Unstable SIGMAR1 42 39 CN1CCN(CCNC(=O)[C@H]2CCCN(S(=O)(=O)c3ccc(Br)cc3)C2)CC1 ZINC000217892436 JD On-Demand Unstable EPHX2 16 46 CN1CCN(CCNC(=O)[C@H]2CCCN(S(=O)(=O)c3ccc(Br)cc3)C2)CC1 ZINC000217892436 JD On-Demand Unstable GPBAR1 18 42 CN1CCN(CCNC(=O)[C@H]2CCCN(S(=O)(=O)c3ccc(Br)cc3)C2)CC1 ZINC000217892436 JD On-Demand Unstable AKR1C1 21 43 CSCC[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217892485 HD In-Stock Unstable EDNRA 16 41 CSCC[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O ZINC000217892485 HD In-Stock Unstable GHSR 40 37 Cc1cccc(SCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217892607 CI For-Sale Unstable PTGER2 26 43 Cc1cccc(SCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217892607 CI For-Sale Unstable LTB4R 20 46 Cc1cccc(SCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217892607 CI For-Sale Unstable AKR1C3 35 42 Cc1cccc(/C=C/NC(=O)NC2CCCCCCCCCCC2)c1 ZINC000217892662 EK For-Sale Unstable FAAH 20 52 Cc1cccc(/C=C/NC(=O)NC2CCCCCCCCCCC2)c1 ZINC000217892662 EK For-Sale Unstable EPHX2 29 45 CC(C)c1ccc(CCCNC(=O)/C=C/c2cccc([N+](=O)[O-])c2)cc1 ZINC000217892693 FI In-Stock Unstable CACNA1D 46 34 CC(C)c1ccc(CCCNC(=O)/C=C/c2cccc([N+](=O)[O-])c2)cc1 ZINC000217892693 FI In-Stock Unstable PYGL 0 41 CC(C)c1ccc(CCCNC(=O)/C=C/c2cccc([N+](=O)[O-])c2)cc1 ZINC000217892693 FI In-Stock Unstable TRPM8 0 59 COc1ccccc1SCc1ccccc1/C=C\C(=O)O ZINC000217892721 DI For-Sale Unstable PTGER2 59 53 COc1ccccc1SCc1ccccc1/C=C\C(=O)O ZINC000217892721 DI For-Sale Unstable PTGER4 30 47 COc1ccccc1SCc1ccccc1/C=C\C(=O)O ZINC000217892721 DI For-Sale Unstable PTGER3 24 53 COc1ccccc1SCc1ccccc1/C=C\C(=O)O ZINC000217892721 DI For-Sale Unstable PTGDR 0 48 COc1ccccc1SCc1ccccc1/C=C\C(=O)O ZINC000217892721 DI For-Sale Unstable AKR1B10 28 40 COc1ccccc1SCc1ccc(/C=C\C(=O)O)cc1 ZINC000217892769 DI For-Sale Unstable PTGER2 43 47 COc1ccccc1SCc1ccc(/C=C\C(=O)O)cc1 ZINC000217892769 DI For-Sale Unstable PTGER4 22 44 COc1ccccc1SCc1ccc(/C=C\C(=O)O)cc1 ZINC000217892769 DI For-Sale Unstable PTGER3 19 47 COc1ccccc1SCc1ccc(/C=C\C(=O)O)cc1 ZINC000217892769 DI For-Sale Unstable NPY2R 0 47 COc1ccccc1SCc1ccc(/C=C\C(=O)O)cc1 ZINC000217892769 DI For-Sale Unstable LTB4R 0 42 COc1ccccc1SCc1ccc(/C=C\C(=O)O)cc1 ZINC000217892769 DI For-Sale Unstable AKR1C3 32 41 Oc1cccc2c1CCC[C@@H]2N1CCC[C@@H](C(F)(F)F)C1 ZINC000217892787 CI For-Sale Unstable SLC6A1 0 42 CC(C)c1cc(C(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)n(C)n1 ZINC000217892797 ED In-Stock Unstable CHRNA4 29 48 Cc1cccc(/C=C/NC(=O)NCCN2CCOCC2)c1 ZINC000217892799 CD For-Sale Unstable CNR1 0 45 Cc1cccc(/C=C/NC(=O)NCCN2CCOCC2)c1 ZINC000217892799 CD For-Sale Unstable DRD4 44 37 Cc1cccc(/C=C/NC(=O)NCCN2CCOCC2)c1 ZINC000217892799 CD For-Sale Unstable CASR 44 37 Cc1cccc(/C=C/NC(=O)NCCN2CCOCC2)c1 ZINC000217892799 CD For-Sale Unstable HDAC8 15 46 Cc1cccc(/C=C/NC(=O)NCCN2CCOCC2)c1 ZINC000217892799 CD For-Sale Unstable PTGDS 42 37 Cc1cccc(/C=C/NC(=O)NCCN2CCOCC2)c1 ZINC000217892799 CD For-Sale Unstable EPHX2 21 43 Cc1cccc(/C=C/NC(=O)NCCN2CCOCC2)c1 ZINC000217892799 CD For-Sale Unstable HPGDS 23 41 O=C(/C=C/c1cccc([N+](=O)[O-])c1)NCCCN1CCCc2ccccc21 ZINC000217892810 FH In-Stock Unstable DRD3 17 47 O=C(/C=C/c1cccc([N+](=O)[O-])c1)NCCCN1CCCc2ccccc21 ZINC000217892810 FH In-Stock Unstable TRPM8 0 46 Cc1ccc(NCCO[C@H]2C[C@H](C)CC[C@H]2C(C)C)cc1 ZINC000217892831 CJ For-Sale Unstable TRPM8 0 43 Oc1cccc2c1CCC[C@H]2N1CCC[C@@H](C(F)(F)F)C1 ZINC000217892851 CI For-Sale Unstable SLC6A1 0 42 COc1ccc(NC(=O)COc2coc(CN3CCc4cc(OC)c(OC)cc4C3)cc2=O)c(OC)c1 ZINC000217892892 KG In-Stock Unstable ABCB1B 54 37 COc1ccc(NC(=O)COc2coc(CN3CCc4cc(OC)c(OC)cc4C3)cc2=O)c(OC)c1 ZINC000217892892 KG In-Stock Unstable ABCB1 26 49 Cc1ccc(NCCO[C@H]2C[C@@H](C)CC[C@H]2C(C)C)cc1 ZINC000217892912 CJ For-Sale Unstable TRPM8 0 43 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1OCCNc1ccc(Cl)cc1 ZINC000217892981 DK For-Sale Unstable TRPM8 0 44 Cc1cc(-c2ccccc2)c(N)nn1 ZINC000217893059 AE For-Sale Unstable DRTS_PLAFK 18 40 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1OCCNc1ccc(Cl)cc1 ZINC000217893062 DK For-Sale Unstable TRPM8 0 44 COc1ccc(/C=C\C(=O)O)cc1COC1CCOCC1 ZINC000217893077 CE For-Sale Unstable PDE4D 15 40 COc1cc(CNC(=O)/C=C/c2ccc([N+](=O)[O-])cc2)ccc1OC(C)C ZINC000217893097 FH In-Stock Unstable U38 0 41 Cc1cccc(/C=C/NC(=O)NCCN2CCNCC2)c1 ZINC000217893125 CD For-Sale Unstable DRD4 43 35 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1OCCNc1ccc(Cl)cc1 ZINC000217893151 DK For-Sale Unstable TRPM8 0 44 CC(C)[C@H]1CC[C@H](C)C[C@@H]1OCCNc1ccc(Cl)cc1 ZINC000217893229 DK For-Sale Unstable TRPM8 0 44 O=C(/C=C/c1ccc([N+](=O)[O-])cc1)NCCCc1ccccc1Cl ZINC000217893242 EI In-Stock Unstable PYGL 26 48 O=C(/C=C/c1ccc([N+](=O)[O-])cc1)NCCCc1ccccc1Cl ZINC000217893242 EI In-Stock Unstable HDAC7 40 37 Cc1ccc(CNC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217893243 CH For-Sale Unstable ANPEP 15 43 Cc1ccc(CNC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217893243 CH For-Sale Unstable FBP1 18 40 CC(C)Nc1nc(-c2ccc(I)cc2)cs1 ZINC000217893351 EI For-Sale Unstable MAOA 22 44 CC(C)Nc1nc(-c2ccc(I)cc2)cs1 ZINC000217893351 EI For-Sale Unstable MAOB 39 44 CC(C)Nc1nc(-c2ccc(I)cc2)cs1 ZINC000217893351 EI For-Sale Unstable SREBF2 0 42 O=C(/C=C/c1ccc([N+](=O)[O-])cc1)NCCCc1ccc(Cl)cc1 ZINC000217893354 EI In-Stock Unstable PYGL 25 47 O=C(/C=C/c1ccc([N+](=O)[O-])cc1)NCCCc1ccc(Cl)cc1 ZINC000217893354 EI In-Stock Unstable HDAC7 41 39 O=C(/C=C/c1ccc([N+](=O)[O-])cc1)NCCCc1ccc(F)cc1 ZINC000217893460 EG In-Stock Unstable PYGL 0 42 O=C(/C=C/c1ccc([N+](=O)[O-])cc1)NCCCc1ccc(F)cc1 ZINC000217893460 EG In-Stock Unstable MMP2 17 46 O=C(/C=C/c1ccc([N+](=O)[O-])cc1)NCCCc1ccc(F)cc1 ZINC000217893460 EG In-Stock Unstable MMP8 21 43 O=C(/C=C/c1ccc([N+](=O)[O-])cc1)NCCCc1ccc(F)cc1 ZINC000217893460 EG In-Stock Unstable MMP9 16 46 O=C(/C=C/c1ccc([N+](=O)[O-])cc1)NCCCc1ccc(F)cc1 ZINC000217893460 EG In-Stock Unstable HDAC7 49 36 O=C(/C=C/c1ccc([N+](=O)[O-])cc1)NCCCc1ccc(F)cc1 ZINC000217893460 EG In-Stock Unstable MMP1 21 43 O=C(/C=C/c1ccc([N+](=O)[O-])cc1)NCCCc1ccc(F)cc1 ZINC000217893460 EG In-Stock Unstable EXSA 0 42 Brc1ccc(-c2nc(-c3ccc(I)cc3)cs2)cc1 ZINC000217893563 IK For-Sale Anodyne CDC25C 0 43 Brc1ccc(-c2nc(-c3ccc(I)cc3)cs2)cc1 ZINC000217893563 IK For-Sale Anodyne SREBF2 0 52 COc1ccccc1CCCNC(=O)/C=C/c1ccc([N+](=O)[O-])cc1 ZINC000217893581 EG In-Stock Unstable DRD3 19 64 Cc1cccc(/C=C/NC(=O)NCCCN2CCOCC2)c1 ZINC000217893615 DD For-Sale Unstable DRD2 18 40 Cc1cccc(/C=C/NC(=O)NCCCN2CCOCC2)c1 ZINC000217893615 DD For-Sale Unstable CNR1 0 42 Cc1cccc(/C=C/NC(=O)NCCCN2CCOCC2)c1 ZINC000217893615 DD For-Sale Unstable DRD3 37 40 Cc1cccc(/C=C/NC(=O)NCCCN2CCOCC2)c1 ZINC000217893615 DD For-Sale Unstable CASR 44 36 Cc1cccc(/C=C/NC(=O)NCCCN2CCOCC2)c1 ZINC000217893615 DD For-Sale Unstable TACR2 28 41 Cc1cccc(/C=C/NC(=O)NCCCN2CCOCC2)c1 ZINC000217893615 DD For-Sale Unstable EPHX2 22 43 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1OCCNc1cccc(Cl)c1 ZINC000217893635 DK For-Sale Unstable TRPM8 0 45 CCC[C@@H](O)CN[C@@H]1CCCCNC1=O ZINC000217893639 BC For-Sale Unstable MMP1 0 44 CCCNc1nc(-c2ccc(I)cc2)cs1 ZINC000217893688 EI For-Sale Unstable MAOA 0 40 CCCNc1nc(-c2ccc(I)cc2)cs1 ZINC000217893688 EI For-Sale Unstable MAOB 34 40 CCCNc1nc(-c2ccc(I)cc2)cs1 ZINC000217893688 EI For-Sale Unstable ROCK2 16 46 COc1ccc(CCCNC(=O)/C=C/c2ccc([N+](=O)[O-])cc2)cc1 ZINC000217893689 EG In-Stock Unstable PTGS2 0 50 COc1ccc(CCCNC(=O)/C=C/c2ccc([N+](=O)[O-])cc2)cc1 ZINC000217893689 EG In-Stock Unstable CACNA1D 21 41 COc1ccc(CCCNC(=O)/C=C/c2ccc([N+](=O)[O-])cc2)cc1 ZINC000217893689 EG In-Stock Unstable HDAC8 20 49 COc1ccc(CCCNC(=O)/C=C/c2ccc([N+](=O)[O-])cc2)cc1 ZINC000217893689 EG In-Stock Unstable MMP2 15 43 COc1ccc(CCCNC(=O)/C=C/c2ccc([N+](=O)[O-])cc2)cc1 ZINC000217893689 EG In-Stock Unstable MMP8 25 44 COc1ccc(CCCNC(=O)/C=C/c2ccc([N+](=O)[O-])cc2)cc1 ZINC000217893689 EG In-Stock Unstable HDAC1 0 49 COc1ccc(CCCNC(=O)/C=C/c2ccc([N+](=O)[O-])cc2)cc1 ZINC000217893689 EG In-Stock Unstable MMP9 17 44 COc1ccc(CCCNC(=O)/C=C/c2ccc([N+](=O)[O-])cc2)cc1 ZINC000217893689 EG In-Stock Unstable MMP1 25 44 COc1ccc(CCCNC(=O)/C=C/c2ccc([N+](=O)[O-])cc2)cc1 ZINC000217893689 EG In-Stock Unstable U38 0 46 COc1ccc(CCCNC(=O)/C=C/c2ccc([N+](=O)[O-])cc2)cc1 ZINC000217893689 EG In-Stock Unstable ABHD6 0 41 COc1ccc(CCCNC(=O)/C=C/c2ccc([N+](=O)[O-])cc2)cc1 ZINC000217893689 EG In-Stock Unstable EXSA 0 45 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1OCCNc1cccc(Cl)c1 ZINC000217893712 DK For-Sale Unstable TRPM8 0 45 CCN(C(=O)N/C=C/c1cccc(C)c1)c1ccccc1 ZINC000217893716 CI For-Sale Unstable NR1H4 40 38 CCC[C@H](O)CN[C@@H]1CCCCNC1=O ZINC000217893722 BC For-Sale Unstable MMP1 0 44 COc1ccccc1SCc1cccc(/C=C\C(=O)O)c1 ZINC000217893744 DI For-Sale Unstable PTGER2 44 45 COc1ccccc1SCc1cccc(/C=C\C(=O)O)c1 ZINC000217893744 DI For-Sale Unstable PTGER4 23 45 COc1ccccc1SCc1cccc(/C=C\C(=O)O)c1 ZINC000217893744 DI For-Sale Unstable PTGER3 19 45 COc1ccccc1SCc1cccc(/C=C\C(=O)O)c1 ZINC000217893744 DI For-Sale Unstable NPY2R 0 45 COc1ccccc1SCc1cccc(/C=C\C(=O)O)c1 ZINC000217893744 DI For-Sale Unstable LTB4R 31 45 COc1ccccc1SCc1cccc(/C=C\C(=O)O)c1 ZINC000217893744 DI For-Sale Unstable MTNR1B 18 45 COc1ccccc1SCc1cccc(/C=C\C(=O)O)c1 ZINC000217893744 DI For-Sale Unstable ALS 43 36 COc1ccccc1SCc1cccc(/C=C\C(=O)O)c1 ZINC000217893744 DI For-Sale Unstable AKR1C3 36 45 O=C1N[C@@H](CC(=O)N2CCN(Cc3nc4ccccc4c(=O)[nH]3)CC2)C(=O)Nc2ccccc21 ZINC000217893754 JC In-Stock Unstable PARP1 21 47 CCCCOc1ccc(C(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217893767 HH For-Sale Unstable PLA2G4B 71 34 CCCCOc1ccc(C(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217893767 HH For-Sale Unstable FAAH 18 45 CCC[C@@H](O)CN[C@H]1CCCCNC1=O ZINC000217893793 BC For-Sale Unstable MMP1 0 44 O=C(/C=C/c1ccc([N+](=O)[O-])cc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217893799 FI In-Stock Bother LTB4R 0 55 O=C(/C=C/c1ccc([N+](=O)[O-])cc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217893799 FI In-Stock Bother MMP2 24 50 O=C(/C=C/c1ccc([N+](=O)[O-])cc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217893799 FI In-Stock Bother HDAC1 16 45 O=C(/C=C/c1ccc([N+](=O)[O-])cc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217893799 FI In-Stock Bother HDAC2 16 41 O=C(/C=C/c1ccc([N+](=O)[O-])cc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217893799 FI In-Stock Bother MMP9 21 50 O=C(/C=C/c1ccc([N+](=O)[O-])cc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217893799 FI In-Stock Bother MMP1 24 50 O=C(/C=C/c1ccc([N+](=O)[O-])cc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217893799 FI In-Stock Bother HDA106 0 43 O=C(/C=C/c1ccc([N+](=O)[O-])cc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217893799 FI In-Stock Bother TRPM8 0 53 O=C(/C=C/c1ccc([N+](=O)[O-])cc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217893799 FI In-Stock Bother AKR1C2 15 45 O=C(/C=C/c1ccc([N+](=O)[O-])cc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217893799 FI In-Stock Bother TRPM2 0 47 O=C(/C=C/c1ccc([N+](=O)[O-])cc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217893799 FI In-Stock Bother H9B8T9_CAPHI 15 50 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1OCCNc1cccc(Cl)c1 ZINC000217893801 DK For-Sale Unstable TRPM8 0 45 C[C@@]1(C#N)CCCN(C(=O)c2cccc(-c3ccco3)c2)C1 ZINC000217893807 CH In-Stock Unstable RHOA 0 47 CC(C)CNc1nc(-c2ccc(I)cc2)cs1 ZINC000217893811 FI For-Sale Unstable MAOB 21 43 CC(C)CNc1nc(-c2ccc(I)cc2)cs1 ZINC000217893811 FI For-Sale Unstable ROCK2 16 43 Nc1cc(N)nc(SCc2ccccc2/C=C\C(=O)O)n1 ZINC000217893812 DE For-Sale Unstable PTGER2 42 47 Nc1cc(N)nc(SCc2ccccc2/C=C\C(=O)O)n1 ZINC000217893812 DE For-Sale Unstable PTGER4 22 49 Nc1cc(N)nc(SCc2ccccc2/C=C\C(=O)O)n1 ZINC000217893812 DE For-Sale Unstable PTGER3 22 49 Nc1cc(N)nc(SCc2ccccc2/C=C\C(=O)O)n1 ZINC000217893812 DE For-Sale Unstable PTGDR 0 49 Cc1cccc(/C=C/NC(=O)N(C)Cc2ccccc2)c1 ZINC000217893835 CH For-Sale Unstable HSP90AB1 24 40 Cc1cccc(/C=C/NC(=O)N(C)Cc2ccccc2)c1 ZINC000217893835 CH For-Sale Unstable PTGES 19 43 Cc1cccc(/C=C/NC(=O)N(C)Cc2ccccc2)c1 ZINC000217893835 CH For-Sale Unstable LIMK2 29 47 CCCCOc1ccc(C(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217893851 HH For-Sale Unstable PLA2G4B 71 34 CCCCOc1ccc(C(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217893851 HH For-Sale Unstable FAAH 18 45 COc1ccc(CCOc2cc([C@@H]3CC(=O)Oc4ccc(C(C)=O)c(O)c43)ccc2OC)cc1 ZINC000217893860 JJ In-Stock Unstable PDEB1 0 42 CCC[C@H](O)CN[C@H]1CCCCNC1=O ZINC000217893878 BC For-Sale Unstable MMP1 0 44 C[C@]1(C#N)CCCN(C(=O)c2cccc(-c3ccco3)c2)C1 ZINC000217893888 CH In-Stock Unstable RHOA 0 47 CC(C)[C@H]1CC[C@H](C)C[C@@H]1OCCNc1cccc(Cl)c1 ZINC000217893889 DK For-Sale Unstable TRPM8 0 45 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccc([N+](=O)[O-])cc2)c1 ZINC000217893906 FI In-Stock Unstable HDAC8 20 42 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccc([N+](=O)[O-])cc2)c1 ZINC000217893906 FI In-Stock Unstable CRTM 45 45 COc1ccc(CCOc2cc([C@H]3CC(=O)Oc4ccc(C(C)=O)c(O)c43)ccc2OC)cc1 ZINC000217893927 JJ In-Stock Unstable PDEB1 0 42 CCCCOc1ccc(C(=O)N2C[C@H](Oc3ccccc3F)C[C@H]2C(=O)OC)cc1 ZINC000217893929 HH For-Sale Unstable PLA2G4B 71 34 CCCCOc1ccc(C(=O)N2C[C@H](Oc3ccccc3F)C[C@H]2C(=O)OC)cc1 ZINC000217893929 HH For-Sale Unstable FAAH 18 45 CS(=O)(=O)c1ccc(C(=O)CN)cc1Cl ZINC000217893936 BC For-Sale Unstable CA2 16 46 CS(=O)(=O)c1ccc(C(=O)CN)cc1Cl ZINC000217893936 BC For-Sale Unstable CA6 27 40 CS(=O)(=O)c1ccc(C(=O)CN)cc1Cl ZINC000217893936 BC For-Sale Unstable CA1 18 44 CS(=O)(=O)c1ccc(C(=O)CN)cc1Cl ZINC000217893936 BC For-Sale Unstable CA7 25 46 CS(=O)(=O)c1ccc(C(=O)CN)cc1Cl ZINC000217893936 BC For-Sale Unstable CA13 37 45 CC(C)(C)Nc1nc(-c2ccc(I)cc2)cs1 ZINC000217893959 FJ For-Sale Unstable MAOA 0 41 CC(C)(C)Nc1nc(-c2ccc(I)cc2)cs1 ZINC000217893959 FJ For-Sale Unstable MAOB 36 41 Cc1ncsc1CCOCc1ccccc1/C=C\C(=O)O ZINC000217893985 DG For-Sale Unstable PTGER2 55 45 Cc1ncsc1CCOCc1ccccc1/C=C\C(=O)O ZINC000217893985 DG For-Sale Unstable PTGER4 27 42 Cc1ncsc1CCOCc1ccccc1/C=C\C(=O)O ZINC000217893985 DG For-Sale Unstable PTGER3 21 45 Cc1ncsc1CCOCc1ccccc1/C=C\C(=O)O ZINC000217893985 DG For-Sale Unstable PTGDR 0 40 CCCCOc1ccc(C(=O)N2C[C@@H](Oc3ccccc3F)C[C@H]2C(=O)OC)cc1 ZINC000217894001 HH For-Sale Unstable PLA2G4B 71 34 CCCCOc1ccc(C(=O)N2C[C@@H](Oc3ccccc3F)C[C@H]2C(=O)OC)cc1 ZINC000217894001 HH For-Sale Unstable FAAH 18 45 Cc1ncsc1CCOCc1ccc(/C=C\C(=O)O)cc1 ZINC000217894072 DG For-Sale Unstable PTGER2 22 40 Brc1cccc(-c2nc(-c3ccc(I)cc3)cs2)c1 ZINC000217894076 IK For-Sale Anodyne SREBF2 0 47 Cc1cccc(/C=C/NC(=O)Nc2nc(C)cs2)c1 ZINC000217894079 CH For-Sale Unstable ROCK1 15 44 Cc1cccc(/C=C/NC(=O)Nc2nc(C)cs2)c1 ZINC000217894079 CH For-Sale Unstable GCK 19 43 O=C(/C=C/c1ccc([N+](=O)[O-])cc1)Nc1ccc(OC2CCCC2)cc1 ZINC000217894132 FJ In-Stock Unstable MMP2 17 46 O=C(/C=C/c1ccc([N+](=O)[O-])cc1)Nc1ccc(OC2CCCC2)cc1 ZINC000217894132 FJ In-Stock Unstable EXSA 0 48 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccc(C(C)C)cc1 ZINC000217894133 HH For-Sale Unstable COLA 43 36 CN1CCO[C@@H]([C@@H](N)Cc2ccc(F)cc2Cl)C1 ZINC000217894145 CD For-Sale Unstable P2RX7 44 39 Cc1ncc(C(=O)N[C@@H]2CCC[C@@H]2CO)s1 ZINC000217894162 BD On-Demand Unstable GYRB 24 41 Cc1ncsc1CCOCc1cccc(/C=C\C(=O)O)c1 ZINC000217894168 DG For-Sale Unstable PTGER2 30 43 Cc1ncsc1CCOCc1cccc(/C=C\C(=O)O)c1 ZINC000217894168 DG For-Sale Unstable LTB4R 16 41 Cc1ncsc1CCOCc1cccc(/C=C\C(=O)O)c1 ZINC000217894168 DG For-Sale Unstable AKR1C3 24 40 O=C(N[C@H](CO)Cc1ccccc1)[C@@H]1CC(=O)N(Cc2ccc3c(c2)OCO3)C1 ZINC000217894212 GD In-Stock Unstable BACE2 0 41 O=C(N[C@H](CO)Cc1ccccc1)[C@@H]1CC(=O)N(Cc2ccc3c(c2)OCO3)C1 ZINC000217894212 GD In-Stock Unstable NOS2 50 33 O=C(N[C@H](CO)Cc1ccccc1)[C@@H]1CC(=O)N(Cc2ccc3c(c2)OCO3)C1 ZINC000217894212 GD In-Stock Unstable SSTR3 47 32 O=C(N[C@H](CO)Cc1ccccc1)[C@@H]1CC(=O)N(Cc2ccc3c(c2)OCO3)C1 ZINC000217894212 GD In-Stock Unstable MCHR1 16 40 O=C(N[C@H](CO)Cc1ccccc1)[C@@H]1CC(=O)N(Cc2ccc3c(c2)OCO3)C1 ZINC000217894212 GD In-Stock Unstable SAP2 31 42 Cc1cccc(/C=C/NC(=O)Nc2ccc(C#N)cc2)c1 ZINC000217894214 CH For-Sale Unstable IDO1 17 43 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccc(C(C)C)cc1 ZINC000217894216 HH For-Sale Unstable COLA 43 36 CN1CCO[C@H]([C@@H](N)Cc2ccc(F)cc2Cl)C1 ZINC000217894224 CD For-Sale Unstable P2RX7 44 39 Cc1ncc(C(=O)N[C@H]2CCC[C@@H]2CO)s1 ZINC000217894239 BD For-Sale Unstable GYRB 24 41 COc1ccc(/C=C\C(=O)O)cc1CO[C@H](C)CC(C)C ZINC000217894258 CH For-Sale Unstable PTGER2 0 43 COc1ccc(/C=C\C(=O)O)cc1CO[C@H](C)CC(C)C ZINC000217894258 CH For-Sale Unstable AKR1C3 32 43 CS(=O)(=O)c1cc(Cl)cc(C(=O)CN)c1 ZINC000217894273 BC For-Sale Unstable O49150_SOLTU 41 33 O=C(N[C@H](CO)Cc1ccccc1)[C@H]1CC(=O)N(Cc2ccc3c(c2)OCO3)C1 ZINC000217894295 GD In-Stock Unstable BACE2 0 41 O=C(N[C@H](CO)Cc1ccccc1)[C@H]1CC(=O)N(Cc2ccc3c(c2)OCO3)C1 ZINC000217894295 GD In-Stock Unstable NOS2 50 33 O=C(N[C@H](CO)Cc1ccccc1)[C@H]1CC(=O)N(Cc2ccc3c(c2)OCO3)C1 ZINC000217894295 GD In-Stock Unstable SSTR3 47 32 O=C(N[C@H](CO)Cc1ccccc1)[C@H]1CC(=O)N(Cc2ccc3c(c2)OCO3)C1 ZINC000217894295 GD In-Stock Unstable MCHR1 16 40 O=C(N[C@H](CO)Cc1ccccc1)[C@H]1CC(=O)N(Cc2ccc3c(c2)OCO3)C1 ZINC000217894295 GD In-Stock Unstable SAP2 31 42 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccc(C(C)C)cc1 ZINC000217894300 HH For-Sale Unstable COLA 43 36 COc1cccc(NC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217894323 CH For-Sale Unstable KIT 15 41 COc1cccc(NC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217894323 CH For-Sale Unstable CCKAR 0 42 COc1cccc(NC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217894323 CH For-Sale Unstable KDR 16 41 COc1cccc(NC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217894323 CH For-Sale Unstable MTNR1A 28 50 COc1cccc(NC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217894323 CH For-Sale Unstable MTNR1B 32 50 COc1cccc(NC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217894323 CH For-Sale Unstable CCKBR 17 42 COc1cccc(NC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217894323 CH For-Sale Unstable TAAR1 33 43 COc1cccc(NC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217894323 CH For-Sale Unstable AKR1C3 15 44 COc1cccc(NC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217894323 CH For-Sale Unstable AKR1C2 29 44 COc1cccc(NC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217894323 CH For-Sale Unstable KCNK3 78 52 COc1cccc(NC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217894323 CH For-Sale Unstable KCNK9 65 40 Cc1ncc(C(=O)N[C@@H]2CCC[C@H]2CO)s1 ZINC000217894329 BD For-Sale Unstable GYRB 24 41 COc1ccc(/C=C\C(=O)O)cc1CO[C@@H](C)CC(C)C ZINC000217894332 CH For-Sale Unstable PTGER2 0 43 COc1ccc(/C=C\C(=O)O)cc1CO[C@@H](C)CC(C)C ZINC000217894332 CH For-Sale Unstable AKR1C3 32 43 CCC[C@@H](O)CNCCc1ccncc1 ZINC000217894370 BD For-Sale Unstable ADRB2 51 41 CCC[C@@H](O)CNCCc1ccncc1 ZINC000217894370 BD For-Sale Unstable ADRB3 66 44 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccc(C(C)C)cc1 ZINC000217894383 HH For-Sale Unstable COLA 43 36 CNCCc1ccc(CN2CCC[C@@H](C)[C@@H]2C)cc1 ZINC000217894404 CG For-Sale Unstable HRH3 29 42 COc1ccc(CO[C@H](C)CC(C)C)cc1/C=C\C(=O)O ZINC000217894406 CH For-Sale Unstable PTGER2 39 46 COc1ccc(CO[C@H](C)CC(C)C)cc1/C=C\C(=O)O ZINC000217894406 CH For-Sale Unstable PTGER4 22 46 COc1ccc(CO[C@H](C)CC(C)C)cc1/C=C\C(=O)O ZINC000217894406 CH For-Sale Unstable PTGER3 22 46 COc1ccc(CO[C@H](C)CC(C)C)cc1/C=C\C(=O)O ZINC000217894406 CH For-Sale Unstable AKR1B10 29 40 Cc1ncc(C(=O)N[C@H]2CCC[C@H]2CO)s1 ZINC000217894420 BD For-Sale Unstable GYRB 24 41 Cc1cccc(/C=C/NC(=O)Nc2cc(Cl)ccc2O)c1 ZINC000217894441 DI For-Sale Unstable MMP9 0 42 Cc1cccc(/C=C/NC(=O)Nc2cc(Cl)ccc2O)c1 ZINC000217894441 DI For-Sale Unstable KCNMA1 26 44 Cc1cccc(/C=C/NC(=O)Nc2cc(Cl)ccc2O)c1 ZINC000217894441 DI For-Sale Unstable MMP1 0 42 Cc1cccc(/C=C/NC(=O)Nc2cc(Cl)ccc2O)c1 ZINC000217894441 DI For-Sale Unstable TUBA4A 0 44 CCC[C@H](O)CNCCc1ccncc1 ZINC000217894457 BD For-Sale Unstable ADRB2 51 41 CCC[C@H](O)CNCCc1ccncc1 ZINC000217894457 BD For-Sale Unstable ADRB3 66 44 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)Cc1ccc(OC)c(OC)c1 ZINC000217894483 HF For-Sale Unstable ITGA4 30 40 COc1ccc(CO[C@@H](C)CC(C)C)cc1/C=C\C(=O)O ZINC000217894488 CH For-Sale Unstable PTGER2 39 46 COc1ccc(CO[C@@H](C)CC(C)C)cc1/C=C\C(=O)O ZINC000217894488 CH For-Sale Unstable PTGER4 22 46 COc1ccc(CO[C@@H](C)CC(C)C)cc1/C=C\C(=O)O ZINC000217894488 CH For-Sale Unstable PTGER3 22 46 COc1ccc(CO[C@@H](C)CC(C)C)cc1/C=C\C(=O)O ZINC000217894488 CH For-Sale Unstable AKR1B10 29 40 CNCCc1ccc(CN2CCC[C@H](C)[C@@H]2C)cc1 ZINC000217894493 CG For-Sale Unstable HRH3 29 42 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccc([N+](=O)[O-])cc1 ZINC000217894506 FI In-Stock Unstable DRD3 15 54 CCOc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1OCC ZINC000217894556 EJ For-Sale Unstable IMPDH2 0 43 CCOc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1OCC ZINC000217894556 EJ For-Sale Unstable KCNK3 53 43 CCOc1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1OCC ZINC000217894556 EJ For-Sale Unstable KCNK9 51 43 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)Cc1ccc(OC)c(OC)c1 ZINC000217894559 HF For-Sale Unstable ITGA4 30 40 CC(C)C[C@@H](C)OCc1ccc(/C=C\C(=O)O)cc1F ZINC000217894562 CH For-Sale Unstable AKR1C3 31 43 C[C@@H]1C[C@](C)(C(=O)O)C[C@@]1(N)C(=O)O ZINC000217894565 BC In-Stock Unstable GRM3 41 41 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)NCc3ccccc3)[C@H]21 ZINC000217894584 JH In-Stock Unstable TSHR 51 34 Cn1nc(CN(Cc2ccco2)C(=O)c2cccc(C(F)(F)F)c2)cc1C1CC1 ZINC000217894603 HJ In-Stock Unstable CCR2 49 36 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)Cc1ccc(OC)c(OC)c1 ZINC000217894618 HF For-Sale Unstable ITGA4 30 40 Cc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc([N+](=O)[O-])cc2)cc1 ZINC000217894622 EH In-Stock Unstable EXSA 0 41 Cc1cccc(/C=C/NC(=O)Nc2nccs2)c1 ZINC000217894641 CG For-Sale Unstable MAP 0 42 Cc1cccc(/C=C/NC(=O)Nc2nccs2)c1 ZINC000217894641 CG For-Sale Unstable MAP1 116 40 CC(C)C[C@H](C)OCc1ccc(/C=C\C(=O)O)cc1F ZINC000217894653 CH For-Sale Unstable AKR1C3 31 43 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)NCc3ccccc3)[C@@H]21 ZINC000217894655 JH In-Stock Unstable TSHR 51 34 C[C@H]1C[C@](C)(C(=O)O)C[C@@]1(N)C(=O)O ZINC000217894660 BC In-Stock Unstable GRM3 41 41 O=C(O)c1oc2cc(O)ccc2c1Br ZINC000217894664 CF For-Sale Anodyne ESR1 20 46 O=C(O)c1oc2cc(O)ccc2c1Br ZINC000217894664 CF For-Sale Anodyne ESR2 16 46 O=C(O)c1oc2cc(O)ccc2c1Br ZINC000217894664 CF For-Sale Anodyne HSD17B3 37 45 O=C(O)c1oc2cc(O)ccc2c1Br ZINC000217894664 CF For-Sale Anodyne SLC22A12 20 42 Cc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc([N+](=O)[O-])cc2)cc1 ZINC000217894706 EH In-Stock Unstable EXSA 0 41 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)Cc1ccc(OC)c(OC)c1 ZINC000217894716 HF For-Sale Unstable ITGA4 30 40 C[C@@H]1C[C@@](C)(C(=O)O)C[C@@]1(N)C(=O)O ZINC000217894741 BC In-Stock Unstable GRM3 41 41 COc1ccc(/C=C\C(=O)O)cc1COCCCC(C)C ZINC000217894757 CH For-Sale Unstable PTGER2 0 41 COc1ccc(/C=C\C(=O)O)cc1COCCCC(C)C ZINC000217894757 CH For-Sale Unstable AKR1C3 31 41 CSc1cccc(NC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217894759 CJ For-Sale Unstable KCNK3 55 39 CSc1cccc(NC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217894759 CJ For-Sale Unstable KCNK9 43 39 COC(=O)[C@@H](N[C@@H]1CCC[C@@H](C)[C@@H]1C)c1ccccc1 ZINC000217894760 CG For-Sale Unstable SLC6A3 15 45 O=C(O)c1oc2ccc(O)cc2c1Br ZINC000217894761 CF For-Sale Anodyne SLC22A12 38 42 CC(C)NCCc1ccc(CN2CCC[C@@H](C)[C@@H]2C)cc1 ZINC000217894801 CH For-Sale Unstable HRH3 31 40 CC1CCN(c2ccc([C@@H](C)NC(=O)/C=C/c3ccc([N+](=O)[O-])cc3)cc2)CC1 ZINC000217894813 GJ In-Stock Unstable SSTR2 28 41 CCOc1ccc(OCC(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217894819 HF For-Sale Unstable CPT1A 59 38 C[C@H]1C[C@@](C)(C(=O)O)C[C@@]1(N)C(=O)O ZINC000217894824 BC In-Stock Unstable GRM3 41 41 COc1ccc(COCCCC(C)C)cc1/C=C\C(=O)O ZINC000217894828 CH For-Sale Unstable PTGER2 36 44 COc1ccc(COCCCC(C)C)cc1/C=C\C(=O)O ZINC000217894828 CH For-Sale Unstable PTGER4 0 44 COc1ccc(COCCCC(C)C)cc1/C=C\C(=O)O ZINC000217894828 CH For-Sale Unstable PTGER3 19 44 COc1ccc(COCCCC(C)C)cc1/C=C\C(=O)O ZINC000217894828 CH For-Sale Unstable AKR1B10 32 43 Cc1cccc(/C=C/NC(=O)Nc2cc(S(=O)(=O)N3CCOCC3)ccc2Cl)c1 ZINC000217894853 IG For-Sale Unstable LPL 49 43 Cc1cccc(/C=C/NC(=O)Nc2cc(S(=O)(=O)N3CCOCC3)ccc2Cl)c1 ZINC000217894853 IG For-Sale Unstable LIPG 20 43 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC1CCS(=O)(=O)CC1 ZINC000217894871 CF For-Sale Unstable TRPM8 17 42 COc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)N1CCSCC1)C(=O)OC2 ZINC000217894879 HG In-Stock Unstable IMPDH1 0 74 COc1c(C)c2c(c(O)c1C/C=C(\C)CCC(=O)N1CCSCC1)C(=O)OC2 ZINC000217894879 HG In-Stock Unstable IMPDH2 0 74 CC(C)NCCc1ccc(CN2CCC[C@H](C)[C@@H]2C)cc1 ZINC000217894895 CH For-Sale Unstable HRH3 31 40 CC1CCN(c2ccc([C@H](C)NC(=O)/C=C/c3ccc([N+](=O)[O-])cc3)cc2)CC1 ZINC000217894897 GJ In-Stock Unstable SSTR2 28 41 CCOc1ccc(OCC(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217894902 HF For-Sale Unstable CPT1A 59 38 CC(C)CCCOCc1ccc(/C=C\C(=O)O)cc1F ZINC000217894910 CH For-Sale Unstable AKR1C3 30 41 COC(=O)[C@@H](N[C@H]1CCC[C@@H](C)[C@@H]1C)c1ccccc1 ZINC000217894941 CG For-Sale Unstable SLC6A3 15 45 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC1CCS(=O)(=O)CC1 ZINC000217894964 CF For-Sale Unstable TRPM8 17 42 Cc1cccc(/C=C/NC(=O)NCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217894972 EE For-Sale Unstable CA2 112 51 Cc1cccc(/C=C/NC(=O)NCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217894972 EE For-Sale Unstable CA1 92 50 Cc1cccc(/C=C/NC(=O)NCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217894972 EE For-Sale Unstable CA7 53 48 Cc1cccc(/C=C/NC(=O)NCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217894972 EE For-Sale Unstable CA5B 51 46 Cc1cccc(/C=C/NC(=O)NCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217894972 EE For-Sale Unstable CA4 77 51 Cc1cccc(/C=C/NC(=O)NCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217894972 EE For-Sale Unstable CA5A 53 46 Cc1cccc(/C=C/NC(=O)NCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217894972 EE For-Sale Unstable CA14 45 48 Cc1cccc(/C=C/NC(=O)NCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217894972 EE For-Sale Unstable FBP1 20 43 Cc1cccc(/C=C/NC(=O)NCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217894972 EE For-Sale Unstable CA12 69 47 Cc1cccc(/C=C/NC(=O)NCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217894972 EE For-Sale Unstable ALPL 15 46 Cc1cccc(/C=C/NC(=O)NCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217894972 EE For-Sale Unstable CA9 78 47 Cc1cccc(/C=C/NC(=O)NCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217894972 EE For-Sale Unstable CYNT 30 44 Cc1cccc(/C=C/NC(=O)NCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217894972 EE For-Sale Unstable MTCA1 47 47 Cc1cccc(/C=C/NC(=O)NCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217894972 EE For-Sale Unstable P96878_MYCTU 60 47 CCOc1ccc(OCC(=O)N2C[C@H](Oc3ccccc3F)C[C@H]2C(=O)OC)cc1 ZINC000217894988 HF For-Sale Unstable CPT1A 59 38 O=C(C[C@@H]1NC(=O)N(Cc2ccc(Cl)cc2)C1=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217894992 JD In-Stock Unstable CHRNA4 29 50 COc1ccc(COC2CCOCC2)cc1/C=C\C(=O)O ZINC000217895000 CE For-Sale Unstable PTGER2 29 43 COc1ccc(COC2CCOCC2)cc1/C=C\C(=O)O ZINC000217895000 CE For-Sale Unstable PTGER4 17 43 COC(=O)[C@H](N[C@H]1CCC[C@@H](C)[C@@H]1C)c1ccccc1 ZINC000217895031 CG For-Sale Unstable SLC6A3 15 45 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC1CCS(=O)(=O)CC1 ZINC000217895041 CF For-Sale Unstable TRPM8 15 41 CN1CCO[C@@H]([C@@H](N)Cc2ccc(F)cc2F)C1 ZINC000217895060 CD For-Sale Unstable DPP4 20 41 CCOc1ccc(OCC(=O)N2C[C@@H](Oc3ccccc3F)C[C@H]2C(=O)OC)cc1 ZINC000217895072 HF For-Sale Unstable CPT1A 59 38 COc1nc(Br)nc2ccc(F)cc12 ZINC000217895084 CF For-Sale Unstable DHODH 35 40 Cc1cccc(/C=C/NC(=O)Nc2cccnc2Cl)c1 ZINC000217895092 CH For-Sale Unstable G2YM83_BOTF4 69 35 COc1cc2oc(=O)cc(-c3ccccc3)c2cc1CCC(=O)N[C@@H](C)CO ZINC000217895109 GF In-Stock Unstable CMA1 15 44 CN1CCO[C@H]([C@@H](N)Cc2ccc(F)cc2F)C1 ZINC000217895123 CD For-Sale Unstable DPP4 20 41 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC1CCS(=O)(=O)CC1 ZINC000217895126 CF For-Sale Unstable TRPM8 15 41 O=C(O)/C=C\c1ccccc1CSCc1ccccc1 ZINC000217895180 CI For-Sale Unstable PTGER2 25 51 O=C(O)/C=C\c1ccccc1CSCc1ccccc1 ZINC000217895180 CI For-Sale Unstable CACNA2D1 24 41 O=C(O)/C=C\c1ccccc1CSCc1ccccc1 ZINC000217895180 CI For-Sale Unstable PTGER4 30 51 O=C(O)/C=C\c1ccccc1CSCc1ccccc1 ZINC000217895180 CI For-Sale Unstable PTGER3 27 58 O=C(O)/C=C\c1ccccc1CSCc1ccccc1 ZINC000217895180 CI For-Sale Unstable PTGDR 0 55 O=C(O)/C=C\c1ccccc1CSCc1ccccc1 ZINC000217895180 CI For-Sale Unstable HCAR2 0 40 Cc1ccc2c(c1)[C@@H](NC(=O)/C=C/c1ccc([N+](=O)[O-])cc1)CC(C)(C)O2 ZINC000217895203 FI In-Stock Unstable SLC27A4 42 30 O=S(=O)(Cl)Cc1cc2ccncc2s1 ZINC000217895257 BE For-Sale Unstable CYP2A6 21 48 O=C(O)/C=C\c1ccc(CSCc2ccccc2)cc1 ZINC000217895265 CI For-Sale Unstable NA 0 44 O=C(O)/C=C\c1ccc(CSCc2ccccc2)cc1 ZINC000217895265 CI For-Sale Unstable PTGER2 40 50 O=C(O)/C=C\c1ccc(CSCc2ccccc2)cc1 ZINC000217895265 CI For-Sale Unstable CACNA2D1 23 45 O=C(O)/C=C\c1ccc(CSCc2ccccc2)cc1 ZINC000217895265 CI For-Sale Unstable PTGER4 0 50 O=C(O)/C=C\c1ccc(CSCc2ccccc2)cc1 ZINC000217895265 CI For-Sale Unstable PTGER3 16 50 O=C(O)/C=C\c1ccc(CSCc2ccccc2)cc1 ZINC000217895265 CI For-Sale Unstable LTB4R 21 42 O=C(O)/C=C\c1ccc(CSCc2ccccc2)cc1 ZINC000217895265 CI For-Sale Unstable F3 26 45 O=C(O)/C=C\c1ccc(CSCc2ccccc2)cc1 ZINC000217895265 CI For-Sale Unstable HDAC1 19 41 O=C(O)/C=C\c1ccc(CSCc2ccccc2)cc1 ZINC000217895265 CI For-Sale Unstable HDAC6 22 42 O=C(O)/C=C\c1ccc(CSCc2ccccc2)cc1 ZINC000217895265 CI For-Sale Unstable PTGDR 0 41 O=C(O)/C=C\c1ccc(CSCc2ccccc2)cc1 ZINC000217895265 CI For-Sale Unstable HCAR2 0 44 O=C(O)/C=C\c1ccc(CSCc2ccccc2)cc1 ZINC000217895265 CI For-Sale Unstable 17HSDCL 0 46 O=C(O)/C=C\c1ccc(CSCc2ccccc2)cc1 ZINC000217895265 CI For-Sale Unstable HDA106 0 41 O=C(O)/C=C\c1ccc(CSCc2ccccc2)cc1 ZINC000217895265 CI For-Sale Unstable AKR1C3 31 41 O=C(O)/C=C\c1ccc(CSCc2ccccc2)cc1 ZINC000217895265 CI For-Sale Unstable AKR1B10 18 47 O=C(O)/C=C\c1ccc(CSCc2ccccc2)cc1 ZINC000217895265 CI For-Sale Unstable GPR183 0 40 Cc1ccc2c(c1)[C@H](NC(=O)/C=C/c1ccc([N+](=O)[O-])cc1)CC(C)(C)O2 ZINC000217895285 FI In-Stock Unstable SLC27A4 42 30 O=C(O)/C=C\c1ccc(CSCc2ccccc2)c(F)c1 ZINC000217895357 DI For-Sale Unstable PTGER2 32 40 O=C(O)/C=C\c1ccc(CSCc2ccccc2)c(F)c1 ZINC000217895357 DI For-Sale Unstable PTGER3 16 40 O=C(O)/C=C\c1ccc(CSCc2ccccc2)c(F)c1 ZINC000217895357 DI For-Sale Unstable AKR1C3 32 44 O=C(O)/C=C\c1ccc(CSCc2ccccc2)c(F)c1 ZINC000217895357 DI For-Sale Unstable GPR183 0 45 Cc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)/C=C/c1ccc([N+](=O)[O-])cc1 ZINC000217895405 FI In-Stock Unstable CACNA1D 50 33 Cc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)/C=C/c1ccc([N+](=O)[O-])cc1 ZINC000217895405 FI In-Stock Unstable SLC27A4 42 30 O=C(N[C@H]1CCC[C@H]1CO)c1cnn2ccccc12 ZINC000217895437 CD On-Demand Unstable JAK1 0 45 O=C(N[C@H]1CCC[C@H]1CO)c1cnn2ccccc12 ZINC000217895437 CD On-Demand Unstable TYK2 36 45 COc1ccc2[nH]c3c(c2c1)CN(C(=O)CCn1sc2ccccc2c1=O)CC3 ZINC000217895448 HH In-Stock Unstable DRD5 22 46 COc1ccc2[nH]c3c(c2c1)CN(C(=O)CCn1sc2ccccc2c1=O)CC3 ZINC000217895448 HH In-Stock Unstable CASP3 22 40 COc1ccc2[nH]c3c(c2c1)CN(C(=O)CCn1sc2ccccc2c1=O)CC3 ZINC000217895448 HH In-Stock Unstable MAPKAPK2 0 40 COc1ccc2[nH]c3c(c2c1)CN(C(=O)CCn1sc2ccccc2c1=O)CC3 ZINC000217895448 HH In-Stock Unstable CASP7 39 40 COc1ccc2[nH]c3c(c2c1)CN(C(=O)CCn1sc2ccccc2c1=O)CC3 ZINC000217895448 HH In-Stock Unstable SRTA 0 40 NC(=O)NCC(=O)NCc1cccc2[nH]ccc12 ZINC000217895452 BC In-Stock Unstable KISS1R 40 32 Cc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)/C=C/c1ccc([N+](=O)[O-])cc1 ZINC000217895473 FI In-Stock Unstable CACNA1D 50 33 Cc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)/C=C/c1ccc([N+](=O)[O-])cc1 ZINC000217895473 FI In-Stock Unstable SLC27A4 42 30 COc1ccc(-c2n[nH]cc2C(=O)NC[C@@H]2CCCN3CCCC[C@H]23)cc1OC ZINC000217895541 GG In-Stock Unstable STK17B 44 38 Cc1cccc(/C=C/NC(=O)Nc2ccccc2F)c1 ZINC000217895551 CH For-Sale Unstable MMP1 0 53 COc1ccc2c(c1)[C@@H](NC(=O)/C=C/c1ccc([N+](=O)[O-])cc1)CC(C)(C)O2 ZINC000217895598 GI In-Stock Unstable EXSA 0 40 COc1cc2c(cc1OC)CN(C(=O)c1cnc3c(OC)cccc3c1O)CC2 ZINC000217895648 GG In-Stock Unstable ABCB1B 63 40 COc1cc2c(cc1OC)CN(C(=O)c1cnc3c(OC)cccc3c1O)CC2 ZINC000217895648 GG In-Stock Unstable ABCB1 25 47 COc1cc2c(cc1OC)CN(C(=O)c1cnc3c(OC)cccc3c1O)CC2 ZINC000217895648 GG In-Stock Unstable ABCG2 35 40 O=C(O)c1cc(Br)ccc1C1(O)CC1 ZINC000217895669 CE For-Sale Unstable RARA 43 34 O=C(O)c1cc(Br)ccc1C1(O)CC1 ZINC000217895669 CE For-Sale Unstable PRS 60 37 COc1ccc2c(c1)[C@H](NC(=O)/C=C/c1ccc([N+](=O)[O-])cc1)CC(C)(C)O2 ZINC000217895674 GI In-Stock Unstable EXSA 0 40 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)OCC(F)(F)F ZINC000217895684 CH For-Sale Unstable TRPM8 20 62 CC(C)CNC[C@@H](C)c1ccc(CN2CCC[C@@H]2C)cc1 ZINC000217895707 CI For-Sale Unstable HRH3 49 50 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1OCCNCc1ccccc1 ZINC000217895758 CI For-Sale Unstable TRPM8 15 42 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)OCC(F)(F)F ZINC000217895765 CH For-Sale Unstable TRPM8 20 62 COCCCN(C)C[C@@H](C)[C@@H](O)c1ccccc1 ZINC000217895777 CE For-Sale Unstable AOC3 24 42 O=C(O)c1ccc(C2(O)CC2)c(Br)c1 ZINC000217895798 CE For-Sale Unstable RARA 69 43 O=C(O)c1ccc(C2(O)CC2)c(Br)c1 ZINC000217895798 CE For-Sale Unstable SRD5A2 21 40 O=C(O)c1ccc(C2(O)CC2)c(Br)c1 ZINC000217895798 CE For-Sale Unstable RARG 90 43 O=C(O)c1ccc(C2(O)CC2)c(Br)c1 ZINC000217895798 CE For-Sale Unstable RXRG 55 44 O=C(O)c1ccc(C2(O)CC2)c(Br)c1 ZINC000217895798 CE For-Sale Unstable RARB 83 43 O=C(O)c1ccc(C2(O)CC2)c(Br)c1 ZINC000217895798 CE For-Sale Unstable RXRA 50 44 O=C(O)c1ccc(C2(O)CC2)c(Br)c1 ZINC000217895798 CE For-Sale Unstable RXRB 56 44 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)/C=C/c1ccc([N+](=O)[O-])cc1 ZINC000217895801 GI In-Stock Unstable CACNA1D 63 35 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)/C=C/c1ccc([N+](=O)[O-])cc1 ZINC000217895801 GI In-Stock Unstable EXSA 0 40 Nc1cc(N)nc(SCc2cccc(/C=C\C(=O)O)c2)n1 ZINC000217895812 DE For-Sale Unstable LTB4R 23 43 Nc1cc(N)nc(SCc2cccc(/C=C\C(=O)O)c2)n1 ZINC000217895812 DE For-Sale Unstable RHOA 0 40 C[C@H](CNC1CC1)c1ccc(CN2CCC[C@@H]2C)cc1 ZINC000217895822 CH For-Sale Unstable HRH3 54 51 O=C(Nc1cnn(C[C@@H]2CCCO2)c1)[C@@H]1C[C@@H](O)CN1 ZINC000217895824 CB For-Sale Unstable PANC 44 31 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1OCCNCc1ccccc1 ZINC000217895844 CI For-Sale Unstable TRPM8 15 42 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)OCC(F)(F)F ZINC000217895853 CH For-Sale Unstable TRPM8 20 62 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)/C=C/c1ccc([N+](=O)[O-])cc1 ZINC000217895873 GI In-Stock Unstable CACNA1D 63 35 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)/C=C/c1ccc([N+](=O)[O-])cc1 ZINC000217895873 GI In-Stock Unstable EXSA 0 40 Cn1nc(CN(Cc2ccco2)C(=O)Cn2c(=O)oc3ccccc32)cc1C1CC1 ZINC000217895884 HG In-Stock Unstable TSPO 19 45 COCCCN(C)C[C@H](C)[C@@H](O)c1ccccc1 ZINC000217895893 CE For-Sale Unstable AOC3 24 42 O=C(Nc1cnn(C[C@@H]2CCCO2)c1)[C@H]1C[C@@H](O)CN1 ZINC000217895901 CB For-Sale Unstable PANC 44 31 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1OCCNCc1ccccc1 ZINC000217895923 CI For-Sale Unstable TRPM8 15 42 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)OCC(F)(F)F ZINC000217895924 CH For-Sale Unstable TRPM8 20 62 CC(C)NC[C@@H](C)c1ccc(CN2CCC[C@@H]2C)cc1 ZINC000217895927 CH For-Sale Unstable HRH3 55 52 COc1ccccc1-c1noc(CCC(=O)NC[C@@H]2CCCN3CCCC[C@H]23)n1 ZINC000217895941 GG In-Stock Unstable MBTPS1 40 33 Cn1cc(C(=O)N2CCn3nc([C@@H](O)CO)cc3C2)c2ccccc21 ZINC000217895946 ED In-Stock Unstable TPSAB1 29 42 CC(C)[C@H]1CC[C@H](C)C[C@@H]1OCCNCc1ccccc1 ZINC000217895993 CI For-Sale Unstable TRPM8 15 42 Cn1cc(C(=O)N2CCn3nc([C@H](O)CO)cc3C2)c2ccccc21 ZINC000217896020 ED In-Stock Unstable TPSAB1 29 42 CNC[C@@H](C)c1ccc(CN2CCC[C@@H]2C)cc1 ZINC000217896060 BF For-Sale Unstable HRH3 56 52 COc1cc(CN2CC[C@H]3CC[C@@H](C2)N3C)cc(Cl)c1O ZINC000217896083 DF For-Sale Unstable HTR4 42 35 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NS(=O)(=O)CC(=O)O ZINC000217896118 CD For-Sale Unstable TRPM8 19 46 O=C(O)/C=C\c1ccccc1COCc1ccccc1Cl ZINC000217896154 DI For-Sale Unstable PTGER2 59 56 O=C(O)/C=C\c1ccccc1COCc1ccccc1Cl ZINC000217896154 DI For-Sale Unstable PTGER4 25 52 O=C(O)/C=C\c1ccccc1COCc1ccccc1Cl ZINC000217896154 DI For-Sale Unstable FABP4 20 43 O=C(O)/C=C\c1ccccc1COCc1ccccc1Cl ZINC000217896154 DI For-Sale Unstable PTGER3 24 56 O=C(O)/C=C\c1ccccc1COCc1ccccc1Cl ZINC000217896154 DI For-Sale Unstable PTGDR 0 47 O=C(O)/C=C\c1ccccc1COCc1ccccc1Cl ZINC000217896154 DI For-Sale Unstable FABP5 29 43 CC[C@@H](NC(=O)/C=C/c1ccc([N+](=O)[O-])cc1)c1ccc(C)cc1C ZINC000217896178 EI In-Stock Unstable U53 0 45 C[C@H](CNC(C)(C)C)c1ccc(CN2CCC[C@@H]2C)cc1 ZINC000217896198 CI For-Sale Unstable HRH3 49 49 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NS(=O)(=O)CC(=O)O ZINC000217896203 CD For-Sale Unstable TRPM8 19 46 O=C(O)/C=C\c1ccc(COCc2ccccc2Cl)cc1 ZINC000217896227 DI For-Sale Unstable PTGER2 49 47 O=C(O)/C=C\c1ccc(COCc2ccccc2Cl)cc1 ZINC000217896227 DI For-Sale Unstable PTGER4 21 41 O=C(O)/C=C\c1ccc(COCc2ccccc2Cl)cc1 ZINC000217896227 DI For-Sale Unstable FABP4 18 40 O=C(O)/C=C\c1ccc(COCc2ccccc2Cl)cc1 ZINC000217896227 DI For-Sale Unstable PTGER3 19 46 O=C(O)/C=C\c1ccc(COCc2ccccc2Cl)cc1 ZINC000217896227 DI For-Sale Unstable PTGDR 0 41 O=C(O)/C=C\c1ccc(COCc2ccccc2Cl)cc1 ZINC000217896227 DI For-Sale Unstable 17HSDCL 0 44 O=C(O)/C=C\c1ccc(COCc2ccccc2Cl)cc1 ZINC000217896227 DI For-Sale Unstable FABP5 28 40 O=C(O)/C=C\c1ccc(COCc2ccccc2Cl)cc1 ZINC000217896227 DI For-Sale Unstable AKR1C3 30 43 CC[C@H](NC(=O)/C=C/c1ccc([N+](=O)[O-])cc1)c1ccc(C)cc1C ZINC000217896266 EI In-Stock Unstable U53 0 45 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NS(=O)(=O)CC(=O)O ZINC000217896286 CD For-Sale Unstable TRPM8 17 45 C[C@H](CN)c1ccc(CN2CCC[C@@H]2C)cc1 ZINC000217896298 BF For-Sale Unstable HRH3 59 55 COc1cc(CN2CC[C@H]3CC[C@@H](C2)N3C)ccc1O ZINC000217896321 CE On-Demand Unstable SSTR5 62 39 COc1cc(CN2CC[C@H]3CC[C@@H](C2)N3C)ccc1O ZINC000217896321 CE On-Demand Unstable CAN2 0 45 O=C(O)/C=C\c1cccc(COCc2ccccc2Cl)c1 ZINC000217896324 DI For-Sale Unstable PTGER2 47 49 O=C(O)/C=C\c1cccc(COCc2ccccc2Cl)c1 ZINC000217896324 DI For-Sale Unstable PTGER4 22 44 O=C(O)/C=C\c1cccc(COCc2ccccc2Cl)c1 ZINC000217896324 DI For-Sale Unstable FABP4 18 41 O=C(O)/C=C\c1cccc(COCc2ccccc2Cl)c1 ZINC000217896324 DI For-Sale Unstable PTGER3 21 44 O=C(O)/C=C\c1cccc(COCc2ccccc2Cl)c1 ZINC000217896324 DI For-Sale Unstable PTGDR 0 40 O=C(O)/C=C\c1cccc(COCc2ccccc2Cl)c1 ZINC000217896324 DI For-Sale Unstable 17HSDCL 0 43 O=C(O)/C=C\c1cccc(COCc2ccccc2Cl)c1 ZINC000217896324 DI For-Sale Unstable FABP5 29 41 O=C(O)/C=C\c1cccc(COCc2ccccc2Cl)c1 ZINC000217896324 DI For-Sale Unstable AKR1C3 32 42 O=C(O)/C=C\c1cccc(COCc2ccccc2Cl)c1 ZINC000217896324 DI For-Sale Unstable GPR183 0 41 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NS(=O)(=O)CC(=O)O ZINC000217896371 CD For-Sale Unstable TRPM8 17 45 CC[C@@H](NC(=O)/C=C/c1ccc([N+](=O)[O-])cc1)c1ccc(OC)c(OC)c1 ZINC000217896376 FH In-Stock Unstable ABCG2 15 42 CCCCCNC(=O)N/C=C/c1cccc(C)c1 ZINC000217896377 BG For-Sale Unstable PA2A1_NAJMO 0 43 CCCCCNC(=O)N/C=C/c1cccc(C)c1 ZINC000217896377 BG For-Sale Unstable ASAH1 70 33 CCCCCNC(=O)N/C=C/c1cccc(C)c1 ZINC000217896377 BG For-Sale Unstable ACAT 0 49 COc1cc2c(cc1OC)CC(=O)N(CC(=O)N[C@H](CO)C(C)C)C=C2 ZINC000217896433 FD In-Stock Unstable HCN2 0 44 CC[C@H](NC(=O)/C=C/c1ccc([N+](=O)[O-])cc1)c1ccc(OC)c(OC)c1 ZINC000217896454 FH In-Stock Unstable ABCG2 15 42 Cc1cccc(/C=C/NC(=O)Nc2ccccc2)c1 ZINC000217896473 CH For-Sale Unstable LPL 42 38 Cc1cccc(/C=C/NC(=O)Nc2ccccc2)c1 ZINC000217896473 CH For-Sale Unstable CCKAR 23 50 Cc1cccc(/C=C/NC(=O)Nc2ccccc2)c1 ZINC000217896473 CH For-Sale Unstable HDAC8 34 45 Cc1cccc(/C=C/NC(=O)Nc2ccccc2)c1 ZINC000217896473 CH For-Sale Unstable MMP2 0 49 Cc1cccc(/C=C/NC(=O)Nc2ccccc2)c1 ZINC000217896473 CH For-Sale Unstable HDAC6 22 45 Cc1cccc(/C=C/NC(=O)Nc2ccccc2)c1 ZINC000217896473 CH For-Sale Unstable MMP9 0 49 Cc1cccc(/C=C/NC(=O)Nc2ccccc2)c1 ZINC000217896473 CH For-Sale Unstable MMP1 0 49 Cc1cccc(/C=C/NC(=O)Nc2ccccc2)c1 ZINC000217896473 CH For-Sale Unstable AKR1C3 15 43 Cc1cccc(/C=C/NC(=O)Nc2ccccc2)c1 ZINC000217896473 CH For-Sale Unstable IDO1 16 42 Cc1cccc(/C=C/NC(=O)Nc2ccccc2)c1 ZINC000217896473 CH For-Sale Unstable TRPM8 0 44 Cc1cccc(/C=C/NC(=O)Nc2ccccc2)c1 ZINC000217896473 CH For-Sale Unstable KCNK3 95 44 Cc1cccc(/C=C/NC(=O)Nc2ccccc2)c1 ZINC000217896473 CH For-Sale Unstable KCNK9 55 44 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NS(=O)(=O)CCCC(=O)O ZINC000217896482 DE On-Demand Unstable TRPM8 0 45 COc1ccc(CN2CC[C@H]3CC[C@@H](C2)N3C)cc1O ZINC000217896511 CE On-Demand Unstable SSTR5 44 37 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NS(=O)(=O)CCCC(=O)O ZINC000217896564 DE On-Demand Unstable TRPM8 0 45 O=C(NCCc1ccc(O)cc1)c1cc(Cl)ccc1Br ZINC000217896584 FH On-Demand Unstable SLC6A5 34 52 O=C(NCCc1ccc(O)cc1)c1cc(Cl)ccc1Br ZINC000217896584 FH On-Demand Unstable NCE103 28 41 O=C(NCCc1ccc(O)cc1)c1cc(Cl)ccc1Br ZINC000217896584 FH On-Demand Unstable P96878_MYCTU 18 41 O=C(N[C@@H]1CCC[C@@H]1CO)c1cccc(Cl)c1F ZINC000217896589 CE For-Sale Unstable SSTR3 32 41 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NS(=O)(=O)CCCC(=O)O ZINC000217896646 DE For-Sale Unstable TRPM8 15 45 O=C(N[C@H]1CCC[C@@H]1CO)c1cccc(Cl)c1F ZINC000217896680 CE For-Sale Unstable SSTR3 32 41 CC(C)Oc1ccc(CCC(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc1 ZINC000217896706 GG In-Stock Unstable CHRNA4 30 51 COc1ccc(O)c(CN2CC[C@H]3CC[C@@H](C2)N3C)c1 ZINC000217896708 CE On-Demand Unstable EBP 44 35 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NS(=O)(=O)CCCC(=O)O ZINC000217896730 DE For-Sale Unstable TRPM8 15 45 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1OCCNCC1CCCC1 ZINC000217896746 CI For-Sale Unstable TRPM8 0 40 O=C(N[C@@H]1CCC[C@H]1CO)c1cccc(Cl)c1F ZINC000217896758 CE For-Sale Unstable SSTR3 32 41 Cc1cccc(-c2noc(CNC(=O)/C=C/c3ccc([N+](=O)[O-])cc3)n2)c1 ZINC000217896804 FG In-Stock Unstable HDAC8 48 39 Cc1cccc(-c2noc(CNC(=O)/C=C/c3ccc([N+](=O)[O-])cc3)n2)c1 ZINC000217896804 FG In-Stock Unstable HDAC1 0 46 C[C@H](CNC1CC1)c1ccc(CN2CCCC[C@@H]2C)cc1 ZINC000217896820 CH For-Sale Unstable HRH3 36 50 O=C(NCCc1ccc(O)cc1)c1cc(I)ccc1O ZINC000217896827 GF On-Demand Unstable SLC6A5 30 43 O=C(NCCc1ccc(O)cc1)c1cc(I)ccc1O ZINC000217896827 GF On-Demand Unstable NCE103 31 43 O=C(NCCc1ccc(O)cc1)c1cc(I)ccc1O ZINC000217896827 GF On-Demand Unstable CAN2 0 43 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NS(=O)(=O)CCC(=O)O ZINC000217896830 CD For-Sale Unstable TRPM8 16 44 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1OCCNCC1CCCC1 ZINC000217896839 CI For-Sale Unstable TRPM8 0 40 O=C(N[C@H]1CCC[C@H]1CO)c1cccc(Cl)c1F ZINC000217896865 CE On-Demand Unstable SSTR3 30 41 O=C(NCc1cnc2cnccn12)c1ccccc1N1CCOCC1 ZINC000217896887 ED In-Stock Unstable STAT6 43 33 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1OCCNCC1CCCC1 ZINC000217896906 CI For-Sale Unstable TRPM8 0 40 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NS(=O)(=O)CCC(=O)O ZINC000217896907 CD For-Sale Unstable TRPM8 16 44 Cc1cccc(/C=C/NC(=O)NCc2ccc(C(=O)O)cc2)c1 ZINC000217896929 DG For-Sale Unstable FBP1 18 40 CC(C)NC[C@@H](C)c1ccc(CN2CCCC[C@@H]2C)cc1 ZINC000217896957 CI For-Sale Unstable HRH3 38 51 Cc1ccc(-c2noc(CNC(=O)/C=C/c3ccc([N+](=O)[O-])cc3)n2)cc1 ZINC000217896959 FG In-Stock Unstable EXSA 0 41 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NS(=O)(=O)CCC(=O)O ZINC000217896984 CD For-Sale Unstable TRPM8 16 44 CC(C)[C@H]1CC[C@H](C)C[C@@H]1OCCNCC1CCCC1 ZINC000217896991 CI For-Sale Unstable TRPM8 0 40 COc1cccc(-c2noc(CNC(=O)/C=C/c3ccc([N+](=O)[O-])cc3)n2)c1 ZINC000217897054 GF In-Stock Unstable EXSA 0 43 CNC[C@@H](C)c1ccc(CN2CCCC[C@@H]2C)cc1 ZINC000217897058 CG For-Sale Unstable HRH3 37 51 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NS(=O)(=O)CCC(=O)O ZINC000217897094 CD For-Sale Unstable TRPM8 16 44 O=C(O)/C=C\c1cccc(OCCOCc2cccs2)c1 ZINC000217897117 DG For-Sale Unstable PTGER2 0 41 Cn1nc(CN(Cc2ccco2)C(=O)NCc2ccc(Cl)cc2)cc1C1CC1 ZINC000217897143 GI In-Stock Unstable IL2RA 49 31 Cn1nc(CN(Cc2ccco2)C(=O)NCc2ccc(Cl)cc2)cc1C1CC1 ZINC000217897143 GI In-Stock Unstable UL54 52 34 COc1cc2oc(=O)cc(C)c2cc1CCC(=O)N[C@@H](CC(C)C)c1nnc2ccccn12 ZINC000217897145 IH In-Stock Unstable PTGER3 44 36 CN1CC[C@@H](NC(=O)c2cc(Cl)ccc2Br)C1 ZINC000217897176 DF For-Sale Unstable DRD2 17 46 CN1CC[C@@H](NC(=O)c2cc(Cl)ccc2Br)C1 ZINC000217897176 DF For-Sale Unstable DRD4 21 42 CN1CC[C@@H](NC(=O)c2cc(Cl)ccc2Br)C1 ZINC000217897176 DF For-Sale Unstable SLC6A1 50 45 CN1CC[C@@H](NC(=O)c2cc(Cl)ccc2Br)C1 ZINC000217897176 DF For-Sale Unstable DRD3 16 42 CN1CC[C@@H](NC(=O)c2cc(Cl)ccc2Br)C1 ZINC000217897176 DF For-Sale Unstable SLC6A3 20 45 CN1CC[C@@H](NC(=O)c2cc(Cl)ccc2Br)C1 ZINC000217897176 DF For-Sale Unstable HTR4 46 47 CN1CC[C@@H](NC(=O)c2cc(Cl)ccc2Br)C1 ZINC000217897176 DF For-Sale Unstable UTS2R 34 43 CN1CC[C@@H](NC(=O)c2cc(Cl)ccc2Br)C1 ZINC000217897176 DF For-Sale Unstable SLC6A5 17 43 C[C@H](CN)c1ccc(CN2CCCC[C@@H]2C)cc1 ZINC000217897179 BG For-Sale Unstable HRH3 40 53 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccc([N+](=O)[O-])cc3)n2)cc1 ZINC000217897185 GF In-Stock Unstable HDAC2 16 43 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccc([N+](=O)[O-])cc3)n2)cc1 ZINC000217897185 GF In-Stock Unstable EXSA 0 47 O=C(O)/C=C\c1cccc(CSCc2ccccc2)c1 ZINC000217897218 CI For-Sale Unstable NA 0 42 O=C(O)/C=C\c1cccc(CSCc2ccccc2)c1 ZINC000217897218 CI For-Sale Unstable PTGER2 38 48 O=C(O)/C=C\c1cccc(CSCc2ccccc2)c1 ZINC000217897218 CI For-Sale Unstable CACNA2D1 30 43 O=C(O)/C=C\c1cccc(CSCc2ccccc2)c1 ZINC000217897218 CI For-Sale Unstable PTGER4 0 48 O=C(O)/C=C\c1cccc(CSCc2ccccc2)c1 ZINC000217897218 CI For-Sale Unstable PTGER3 15 48 O=C(O)/C=C\c1cccc(CSCc2ccccc2)c1 ZINC000217897218 CI For-Sale Unstable LTB4R 21 52 O=C(O)/C=C\c1cccc(CSCc2ccccc2)c1 ZINC000217897218 CI For-Sale Unstable MMP1 0 45 O=C(O)/C=C\c1cccc(CSCc2ccccc2)c1 ZINC000217897218 CI For-Sale Unstable HCAR2 0 41 O=C(O)/C=C\c1cccc(CSCc2ccccc2)c1 ZINC000217897218 CI For-Sale Unstable 17HSDCL 0 44 O=C(O)/C=C\c1cccc(CSCc2ccccc2)c1 ZINC000217897218 CI For-Sale Unstable AKR1C3 32 43 CN1CC[C@H](NC(=O)c2cc(Cl)ccc2Br)C1 ZINC000217897258 DF For-Sale Unstable DRD2 17 46 CN1CC[C@H](NC(=O)c2cc(Cl)ccc2Br)C1 ZINC000217897258 DF For-Sale Unstable DRD4 21 42 CN1CC[C@H](NC(=O)c2cc(Cl)ccc2Br)C1 ZINC000217897258 DF For-Sale Unstable SLC6A1 50 45 CN1CC[C@H](NC(=O)c2cc(Cl)ccc2Br)C1 ZINC000217897258 DF For-Sale Unstable DRD3 16 42 CN1CC[C@H](NC(=O)c2cc(Cl)ccc2Br)C1 ZINC000217897258 DF For-Sale Unstable SLC6A3 20 45 CN1CC[C@H](NC(=O)c2cc(Cl)ccc2Br)C1 ZINC000217897258 DF For-Sale Unstable HTR4 46 47 CN1CC[C@H](NC(=O)c2cc(Cl)ccc2Br)C1 ZINC000217897258 DF For-Sale Unstable UTS2R 34 43 CN1CC[C@H](NC(=O)c2cc(Cl)ccc2Br)C1 ZINC000217897258 DF For-Sale Unstable SLC6A5 17 43 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccc([N+](=O)[O-])cc3)n2)c(OC)c1 ZINC000217897273 HF In-Stock Unstable EXSA 0 41 O=C(Cc1cccc([N+](=O)[O-])c1)N[C@H]1CCC[C@H]1CO ZINC000217897281 CD On-Demand Unstable CACNA1D 80 36 O=C(Cc1cccc([N+](=O)[O-])c1)N[C@H]1CCC[C@H]1CO ZINC000217897281 CD On-Demand Unstable LUXR 24 56 O=C(O)/C=C\c1cc(F)ccc1CSCc1ccccc1 ZINC000217897290 DI For-Sale Unstable PTGER2 42 48 O=C(O)/C=C\c1cc(F)ccc1CSCc1ccccc1 ZINC000217897290 DI For-Sale Unstable PTGER4 17 43 O=C(O)/C=C\c1cc(F)ccc1CSCc1ccccc1 ZINC000217897290 DI For-Sale Unstable PTGER3 20 48 O=C(O)/C=C\c1cc(F)ccc1CSCc1ccccc1 ZINC000217897290 DI For-Sale Unstable PTGDR 0 43 O=C(O)/C=C\c1cc(F)ccc1CSCc1ccccc1 ZINC000217897290 DI For-Sale Unstable HCAR2 0 43 O=C(O)/C=C\c1cc(CSCc2ccccc2)ccc1F ZINC000217897395 DI For-Sale Unstable PTGER2 42 49 O=C(O)/C=C\c1cc(CSCc2ccccc2)ccc1F ZINC000217897395 DI For-Sale Unstable PTGER4 22 49 O=C(O)/C=C\c1cc(CSCc2ccccc2)ccc1F ZINC000217897395 DI For-Sale Unstable PTGER3 24 49 O=C(O)/C=C\c1cc(CSCc2ccccc2)ccc1F ZINC000217897395 DI For-Sale Unstable LTB4R 17 41 O=C(O)/C=C\c1cc(CSCc2ccccc2)ccc1F ZINC000217897395 DI For-Sale Unstable PTGDR 0 44 COc1ccc(F)cc1C(=O)N[C@@H](C)Cc1cccnc1 ZINC000217897416 CF In-Stock Unstable GRIN2B 25 40 COc1ccc(F)cc1C(=O)N[C@@H](C)Cc1cccnc1 ZINC000217897416 CF In-Stock Unstable PTAFR 27 46 COc1ccc(F)cc1C(=O)N[C@@H](C)Cc1cccnc1 ZINC000217897416 CF In-Stock Unstable SDH1 0 44 CN1CC[C@@H](NC(=O)c2ccc([N+](=O)[O-])c(O)c2)C1 ZINC000217897420 CC For-Sale Unstable UTS2R 22 43 Cc1cccc(/C=C/NC(=O)NC2CC(C)(C)NC(C)(C)C2)c1 ZINC000217897455 DH For-Sale Unstable EZH2 52 37 COc1ccc(CN2CC[C@H]3CC[C@@H](C2)N3C)c(O)c1 ZINC000217897467 CE For-Sale Unstable EBP 42 35 CN1CC[C@H](NC(=O)c2ccc([N+](=O)[O-])c(O)c2)C1 ZINC000217897487 CC For-Sale Unstable UTS2R 22 43 COc1ccc(F)cc1C(=O)N[C@H](C)Cc1cccnc1 ZINC000217897496 CF In-Stock Unstable GRIN2B 25 40 COc1ccc(F)cc1C(=O)N[C@H](C)Cc1cccnc1 ZINC000217897496 CF In-Stock Unstable PTAFR 27 46 COc1ccc(F)cc1C(=O)N[C@H](C)Cc1cccnc1 ZINC000217897496 CF In-Stock Unstable SDH1 0 44 COc1ccc(C(=O)NC[C@@H]2CCCN3CCCC[C@H]23)cc1-n1nc(C)cc1C ZINC000217897511 GG In-Stock Unstable ACKR3 53 34 COC(CN1CCC(CNC(C)=O)CC1)OC ZINC000217897537 BC On-Demand Unstable HTR4 43 38 COC(CN1CCC(CNC(C)=O)CC1)OC ZINC000217897537 BC On-Demand Unstable CACNA1I 67 42 O=C(/C=C/c1ccc([N+](=O)[O-])cc1)NCc1nc(-c2cccc(Br)c2)no1 ZINC000217897539 IH In-Stock Unstable HDAC8 40 41 O=C(/C=C/c1ccc([N+](=O)[O-])cc1)NCc1nc(-c2cccc(Br)c2)no1 ZINC000217897539 IH In-Stock Unstable HDAC1 15 41 Cc1cccc(/C=C/NC(=O)Nc2cc(C)ccc2O)c1 ZINC000217897548 CH For-Sale Unstable MMP2 0 45 Cc1cccc(/C=C/NC(=O)Nc2cc(C)ccc2O)c1 ZINC000217897548 CH For-Sale Unstable MMP9 0 45 Cc1cccc(/C=C/NC(=O)Nc2cc(C)ccc2O)c1 ZINC000217897548 CH For-Sale Unstable MMP1 0 45 CN1CCO[C@@H]([C@@H](N)CCCc2ccccc2)C1 ZINC000217897553 BD For-Sale Unstable SLC18A2 22 41 CN1CCO[C@@H]([C@@H](N)CCCc2ccccc2)C1 ZINC000217897553 BD For-Sale Unstable SIGMAR1 28 40 CN1CCO[C@H]([C@@H](N)CCCc2ccccc2)C1 ZINC000217897616 BD For-Sale Unstable SLC18A2 22 41 CN1CCO[C@H]([C@@H](N)CCCc2ccccc2)C1 ZINC000217897616 BD For-Sale Unstable SIGMAR1 28 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1c(-c2ccccc2Cl)noc1C ZINC000217897627 JI For-Sale Unstable GPBAR1 32 44 CN1CC[C@@H](NC(=O)c2cc(I)ccc2O)C1 ZINC000217897638 ED For-Sale Unstable SLC6A1 22 43 CN1CC[C@@H](NC(=O)c2cc(I)ccc2O)C1 ZINC000217897638 ED For-Sale Unstable HTR4 22 42 CN1CC[C@H](NC(=O)c2cc(I)ccc2O)C1 ZINC000217897704 ED For-Sale Unstable SLC6A1 22 43 CN1CC[C@H](NC(=O)c2cc(I)ccc2O)C1 ZINC000217897704 ED For-Sale Unstable HTR4 22 42 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1c(-c2ccccc2Cl)noc1C ZINC000217897705 JI For-Sale Unstable GPBAR1 32 44 O=C(Cc1ccccn1)NCc1nc2c(s1)CCCC2 ZINC000217897741 CE In-Stock Unstable SLC27A1 28 48 COC(=O)CCSCCOc1cccc(/C=C\C(=O)O)c1 ZINC000217897768 DE For-Sale Unstable AKR1C3 32 43 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1c(-c2ccccc2Cl)noc1C ZINC000217897783 JI For-Sale Unstable GPBAR1 32 44 CCCC(=O)[C@H](N)C(=O)OCc1ccccc1 ZINC000217897828 BD For-Sale Unstable LTA4H 19 40 CCCC(=O)[C@H](N)C(=O)OCc1ccccc1 ZINC000217897828 BD For-Sale Unstable KLK3 41 31 CCCC(=O)[C@H](N)C(=O)OCc1ccccc1 ZINC000217897828 BD For-Sale Unstable CTSB 40 36 CCCC(=O)[C@H](N)C(=O)OCc1ccccc1 ZINC000217897828 BD For-Sale Unstable PAPA1_CARPA 54 35 CCCC(=O)[C@H](N)C(=O)OCc1ccccc1 ZINC000217897828 BD For-Sale Unstable CYSP_TRYCR 41 37 CCCC(=O)[C@H](N)C(=O)OCc1ccccc1 ZINC000217897828 BD For-Sale Unstable CAPNS1 49 36 CCCC(=O)[C@H](N)C(=O)OCc1ccccc1 ZINC000217897828 BD For-Sale Unstable CAPN1 56 37 CCCC(=O)[C@H](N)C(=O)OCc1ccccc1 ZINC000217897828 BD For-Sale Unstable CAPN2 87 39 CCCC(=O)[C@H](N)C(=O)OCc1ccccc1 ZINC000217897828 BD For-Sale Unstable NPR 56 38 CCCC(=O)[C@H](N)C(=O)OCc1ccccc1 ZINC000217897828 BD For-Sale Unstable SLC12A5 62 34 COC(=O)CCSCCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217897852 DE For-Sale Unstable AKR1C3 29 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1c(-c2ccccc2Cl)noc1C ZINC000217897884 JI For-Sale Unstable GPBAR1 32 44 CCCC(=O)[C@@H](N)C(=O)OCc1ccccc1 ZINC000217897891 BD For-Sale Unstable LTA4H 19 40 CCCC(=O)[C@@H](N)C(=O)OCc1ccccc1 ZINC000217897891 BD For-Sale Unstable KLK3 41 31 CCCC(=O)[C@@H](N)C(=O)OCc1ccccc1 ZINC000217897891 BD For-Sale Unstable CTSB 40 36 CCCC(=O)[C@@H](N)C(=O)OCc1ccccc1 ZINC000217897891 BD For-Sale Unstable PAPA1_CARPA 54 35 CCCC(=O)[C@@H](N)C(=O)OCc1ccccc1 ZINC000217897891 BD For-Sale Unstable CYSP_TRYCR 41 37 CCCC(=O)[C@@H](N)C(=O)OCc1ccccc1 ZINC000217897891 BD For-Sale Unstable CAPNS1 49 36 CCCC(=O)[C@@H](N)C(=O)OCc1ccccc1 ZINC000217897891 BD For-Sale Unstable CAPN1 56 37 CCCC(=O)[C@@H](N)C(=O)OCc1ccccc1 ZINC000217897891 BD For-Sale Unstable CAPN2 87 39 CCCC(=O)[C@@H](N)C(=O)OCc1ccccc1 ZINC000217897891 BD For-Sale Unstable NPR 56 38 CCCC(=O)[C@@H](N)C(=O)OCc1ccccc1 ZINC000217897891 BD For-Sale Unstable SLC12A5 62 34 Cc1cccc(/C=C/NC(=O)Nc2ccc(C)c(C)c2)c1 ZINC000217897931 CI For-Sale Unstable IMPDH2 0 43 Cc1cccc(/C=C/NC(=O)Nc2ccc(C)c(C)c2)c1 ZINC000217897931 CI For-Sale Unstable MMP1 0 46 Cc1cccc(/C=C/NC(=O)Nc2ccc(C)c(C)c2)c1 ZINC000217897931 CI For-Sale Unstable KCNK3 59 38 Cc1cccc(/C=C/NC(=O)Nc2ccc(C)c(C)c2)c1 ZINC000217897931 CI For-Sale Unstable KCNK9 47 38 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)Cc1ccc(S(=O)(=O)C(C)C)cc1 ZINC000217897970 JF For-Sale Unstable MMP2 17 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)Cc1ccc(S(=O)(=O)C(C)C)cc1 ZINC000217898031 JF For-Sale Unstable MMP2 17 40 COc1ccc(CCNC(=O)CCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@H]23)cc1 ZINC000217898044 JH In-Stock Unstable SCN9A 0 47 COc1ccc(CCNC(=O)CCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@H]23)cc1 ZINC000217898044 JH In-Stock Unstable MTNR1A 44 36 COc1ccc(-c2noc(CN(C)C(=O)/C=C/c3ccc([N+](=O)[O-])cc3)n2)cc1 ZINC000217898046 GG In-Stock Unstable EXSA 0 41 CC(C)OC(=O)[C@@H](NC(=O)c1ccccc1)[C@@H](O)C(C)C ZINC000217898050 CD For-Sale Unstable CTSB 16 42 CC(C)OC(=O)[C@@H](NC(=O)c1ccccc1)[C@@H](O)C(C)C ZINC000217898050 CD For-Sale Unstable CCR1 19 41 CC(C)OC(=O)[C@@H](NC(=O)c1ccccc1)[C@@H](O)C(C)C ZINC000217898050 CD For-Sale Unstable CTRB1 42 39 CC(C)OC(=O)[C@@H](NC(=O)c1ccccc1)[C@@H](O)C(C)C ZINC000217898050 CD For-Sale Unstable KCNK3 47 34 CCN(Cc1ccccc1)C(=O)N/C=C/c1cccc(C)c1 ZINC000217898057 CI For-Sale Unstable PTGES 22 45 CC(C)(C)OC(=O)NC1C2CCC1CC2 ZINC000217898059 BF In-Stock Unstable CTSK 0 43 CC(C)(C)OC(=O)NC1C2CCC1CC2 ZINC000217898059 BF In-Stock Unstable NAAA 15 47 O=C1CN(C(=O)c2cccc(=O)[nH]2)CCN1Cc1ccc(F)cc1 ZINC000217898060 EC In-Stock Unstable P2RX7 20 42 O=C(/C=C\c1ccccc1)N1CCN(Cc2cccnc2)CC1 ZINC000217898082 DE On-Demand Unstable DRD4 19 43 O=C(/C=C\c1ccccc1)N1CCN(Cc2cccnc2)CC1 ZINC000217898082 DE On-Demand Unstable TBXAS1 26 40 O=C(/C=C\c1ccccc1)N1CCN(Cc2cccnc2)CC1 ZINC000217898082 DE On-Demand Unstable SIGMAR1 28 46 O=C(/C=C\c1ccccc1)N1CCN(Cc2cccnc2)CC1 ZINC000217898082 DE On-Demand Unstable CHRNA7 30 48 O=C(/C=C\c1ccccc1)N1CCN(Cc2cccnc2)CC1 ZINC000217898082 DE On-Demand Unstable C3AR1 43 48 O=C(/C=C\c1ccccc1)N1CCN(Cc2cccnc2)CC1 ZINC000217898082 DE On-Demand Unstable FAAH 28 42 CC(C)OC(=O)[C@@H](NC(=O)c1ccccc1)[C@H](O)C(C)C ZINC000217898110 CD For-Sale Unstable CTSB 16 42 CC(C)OC(=O)[C@@H](NC(=O)c1ccccc1)[C@H](O)C(C)C ZINC000217898110 CD For-Sale Unstable CCR1 19 41 CC(C)OC(=O)[C@@H](NC(=O)c1ccccc1)[C@H](O)C(C)C ZINC000217898110 CD For-Sale Unstable CTRB1 42 39 CC(C)OC(=O)[C@@H](NC(=O)c1ccccc1)[C@H](O)C(C)C ZINC000217898110 CD For-Sale Unstable KCNK3 47 34 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)Cc1ccc(S(=O)(=O)C(C)C)cc1 ZINC000217898124 JF For-Sale Unstable MMP2 17 40 COc1ccc(CCNC(=O)CCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@@H]23)cc1 ZINC000217898130 JH In-Stock Unstable SCN9A 0 47 COc1ccc(CCNC(=O)CCN2C(=O)c3ccccc3N3C(=O)c4ccccc4[C@@H]23)cc1 ZINC000217898130 JH In-Stock Unstable MTNR1A 44 36 CCCCCCCCC(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217898157 CG On-Demand Unstable FAAH 0 44 CCCCCCCCC(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217898157 CG On-Demand Unstable GBA2 44 31 CCCCCCCCC(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217898157 CG On-Demand Unstable LUXR 35 46 CCCCCCCCC(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217898157 CG On-Demand Unstable TRAR 15 46 CCCCCCCCC(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217898157 CG On-Demand Unstable LASR 64 46 CCCCCCCCC(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217898157 CG On-Demand Unstable PHZR 0 46 CCCCCCCCC(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217898157 CG On-Demand Unstable CQSS 52 32 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)Cc1ccc(S(=O)(=O)C(C)C)cc1 ZINC000217898204 JF For-Sale Unstable MMP2 17 40 COc1ccc(/C=C\C(=O)O)cc1COCCC(C)C ZINC000217898208 CG For-Sale Unstable PTGER2 0 42 COc1ccc(/C=C\C(=O)O)cc1COCCC(C)C ZINC000217898208 CG For-Sale Unstable AKR1C3 32 42 CCCCCCCCC(=O)N[C@H]1CCC[C@@H]1CO ZINC000217898231 CG For-Sale Unstable FAAH 0 44 CCCCCCCCC(=O)N[C@H]1CCC[C@@H]1CO ZINC000217898231 CG For-Sale Unstable GBA2 44 31 CCCCCCCCC(=O)N[C@H]1CCC[C@@H]1CO ZINC000217898231 CG For-Sale Unstable LUXR 35 46 CCCCCCCCC(=O)N[C@H]1CCC[C@@H]1CO ZINC000217898231 CG For-Sale Unstable TRAR 15 46 CCCCCCCCC(=O)N[C@H]1CCC[C@@H]1CO ZINC000217898231 CG For-Sale Unstable LASR 64 46 CCCCCCCCC(=O)N[C@H]1CCC[C@@H]1CO ZINC000217898231 CG For-Sale Unstable PHZR 0 46 CCCCCCCCC(=O)N[C@H]1CCC[C@@H]1CO ZINC000217898231 CG For-Sale Unstable CQSS 52 32 CCNC[C@H](C)c1ccc(CN2C[C@H](C)O[C@@H](C)C2)cc1 ZINC000217898236 CG For-Sale Unstable ERG2 17 40 CCNC[C@H](C)c1ccc(CN2C[C@H](C)O[C@@H](C)C2)cc1 ZINC000217898236 CG For-Sale Unstable ZM.86993 0 40 CCNC[C@H](C)c1ccc(CN2C[C@H](C)O[C@@H](C)C2)cc1 ZINC000217898236 CG For-Sale Unstable Q2TU57_MAIZE 19 40 Cc1ccc(CNC(=O)CCN2CCCCC2)c2cccnc12 ZINC000217898275 DG In-Stock Unstable HNMT 79 37 N#Cc1ccccc1OCc1ccccc1/C=C\C(=O)O ZINC000217898288 CG For-Sale Unstable ADRB1 41 37 N#Cc1ccccc1OCc1ccccc1/C=C\C(=O)O ZINC000217898288 CG For-Sale Unstable PTGER2 23 53 N#Cc1ccccc1OCc1ccccc1/C=C\C(=O)O ZINC000217898288 CG For-Sale Unstable PTGER4 29 53 N#Cc1ccccc1OCc1ccccc1/C=C\C(=O)O ZINC000217898288 CG For-Sale Unstable PTGER3 27 53 CCCCCCCCC(=O)N[C@@H]1CCC[C@H]1CO ZINC000217898290 CG For-Sale Unstable FAAH 0 44 CCCCCCCCC(=O)N[C@@H]1CCC[C@H]1CO ZINC000217898290 CG For-Sale Unstable GBA2 44 31 CCCCCCCCC(=O)N[C@@H]1CCC[C@H]1CO ZINC000217898290 CG For-Sale Unstable LUXR 35 46 CCCCCCCCC(=O)N[C@@H]1CCC[C@H]1CO ZINC000217898290 CG For-Sale Unstable TRAR 15 46 CCCCCCCCC(=O)N[C@@H]1CCC[C@H]1CO ZINC000217898290 CG For-Sale Unstable LASR 64 46 CCCCCCCCC(=O)N[C@@H]1CCC[C@H]1CO ZINC000217898290 CG For-Sale Unstable PHZR 0 46 CCCCCCCCC(=O)N[C@@H]1CCC[C@H]1CO ZINC000217898290 CG For-Sale Unstable CQSS 52 32 Cn1cc(CNC(=O)c2cc(Cl)ccc2Br)cn1 ZINC000217898320 EF On-Demand Unstable UL54 83 39 Cn1cc(CNC(=O)c2cc(Cl)ccc2Br)cn1 ZINC000217898320 EF On-Demand Unstable U38 0 40 Cn1cc(CNC(=O)c2cc(Cl)ccc2Br)cn1 ZINC000217898320 EF On-Demand Unstable DPOL_VZVD 43 39 CCCCCCCCC(=O)N[C@H]1CCC[C@H]1CO ZINC000217898346 CG For-Sale Unstable FAAH 0 44 CCCCCCCCC(=O)N[C@H]1CCC[C@H]1CO ZINC000217898346 CG For-Sale Unstable GBA2 44 31 CCCCCCCCC(=O)N[C@H]1CCC[C@H]1CO ZINC000217898346 CG For-Sale Unstable LUXR 35 46 CCCCCCCCC(=O)N[C@H]1CCC[C@H]1CO ZINC000217898346 CG For-Sale Unstable TRAR 15 46 CCCCCCCCC(=O)N[C@H]1CCC[C@H]1CO ZINC000217898346 CG For-Sale Unstable LASR 64 46 CCCCCCCCC(=O)N[C@H]1CCC[C@H]1CO ZINC000217898346 CG For-Sale Unstable PHZR 0 46 CCCCCCCCC(=O)N[C@H]1CCC[C@H]1CO ZINC000217898346 CG For-Sale Unstable CQSS 52 32 N#Cc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217898386 CG For-Sale Unstable ADRB1 42 33 N#Cc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217898386 CG For-Sale Unstable PTGER2 23 47 N#Cc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217898386 CG For-Sale Unstable PPIA 41 33 N#Cc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217898386 CG For-Sale Unstable PTGER4 30 47 N#Cc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217898386 CG For-Sale Unstable PTGER3 26 47 N#Cc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217898386 CG For-Sale Unstable 17HSDCL 0 43 N#Cc1ccccc1OCc1ccc(/C=C\C(=O)O)cc1 ZINC000217898386 CG For-Sale Unstable AKR1C3 35 49 CCOc1ccccc1C(=O)N(Cc1cc(C2CC2)n(C)n1)C1CCCC1 ZINC000217898406 FI In-Stock Unstable TRPM8 31 43 CCOc1ccccc1C(=O)N(Cc1cc(C2CC2)n(C)n1)C1CCCC1 ZINC000217898406 FI In-Stock Unstable HCN1 47 37 CCOc1ccccc1C(=O)N(Cc1cc(C2CC2)n(C)n1)C1CCCC1 ZINC000217898406 FI In-Stock Unstable HCN4 47 37 N#Cc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217898460 CG For-Sale Unstable ADRB1 44 34 N#Cc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217898460 CG For-Sale Unstable MAOB 15 40 N#Cc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217898460 CG For-Sale Unstable PTGER2 23 49 N#Cc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217898460 CG For-Sale Unstable PTGER4 32 45 N#Cc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217898460 CG For-Sale Unstable PTGER3 27 49 N#Cc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217898460 CG For-Sale Unstable 17HSDCL 0 41 N#Cc1ccccc1OCc1cccc(/C=C\C(=O)O)c1 ZINC000217898460 CG For-Sale Unstable AKR1C3 38 50 Cc1cccc(/C=C/NC(=O)N(Cc2ccccc2)Cc2ccccc2)c1 ZINC000217898512 FK For-Sale Unstable NR1H4 42 39 Cc1cccc(/C=C/NC(=O)N(Cc2ccccc2)Cc2ccccc2)c1 ZINC000217898512 FK For-Sale Unstable PTGES 27 50 Cc1cccc(/C=C/NC(=O)N(Cc2ccccc2)Cc2ccccc2)c1 ZINC000217898512 FK For-Sale Unstable LIMK2 26 43 CCC(C)(C)OCCOc1cccc(/C=C\C(=O)O)c1 ZINC000217898581 CG For-Sale Unstable PTGER2 25 40 CCC(C)(C)OCCOc1cccc(/C=C\C(=O)O)c1 ZINC000217898581 CG For-Sale Unstable AKR1C3 30 40 Cn1nc(CN(C(=O)c2ccccc2Cl)C2CCCC2)cc1C1CC1 ZINC000217898596 FJ In-Stock Unstable ACE 44 39 Cc1cccc(/C=C/NC(=O)N(CCO)Cc2ccccc2)c1 ZINC000217898601 DG For-Sale Unstable PTGES 20 43 CCC(C)(C)OCCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217898654 CG For-Sale Unstable PLA2G4B 65 35 CCC(C)(C)OCCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217898654 CG For-Sale Unstable AKR1C3 27 40 COc1ccc(NC(=O)N/C=C/c2cccc(C)c2)c(OC)c1 ZINC000217898691 DH For-Sale Unstable CYP1B1 51 46 COc1ccc(NC(=O)N/C=C/c2cccc(C)c2)c(OC)c1 ZINC000217898691 DH For-Sale Unstable MTNR1A 29 42 COc1ccc(NC(=O)N/C=C/c2cccc(C)c2)c(OC)c1 ZINC000217898691 DH For-Sale Unstable MTNR1B 28 42 COc1ccc(NC(=O)N/C=C/c2cccc(C)c2)c(OC)c1 ZINC000217898691 DH For-Sale Unstable ABCG2 19 43 COc1ccc(NC(=O)N/C=C/c2cccc(C)c2)c(OC)c1 ZINC000217898691 DH For-Sale Unstable AKR1C2 31 42 COc1ccc(NC(=O)N/C=C/c2cccc(C)c2)c(OC)c1 ZINC000217898691 DH For-Sale Unstable KCNK3 19 43 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccc([N+](=O)[O-])cc2)cc1 ZINC000217898710 FI In-Stock Unstable PYGL 0 42 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccc([N+](=O)[O-])cc2)cc1 ZINC000217898710 FI In-Stock Unstable HDAC8 16 47 O=C(O)/C=C\c1ccc(OCCOCc2cccs2)cc1 ZINC000217898742 DG For-Sale Unstable PTGER2 0 41 O=C(c1ccccc1Br)N1C[C@H]2CNC[C@@H](C2)C1 ZINC000217898746 DE For-Sale Unstable CHRNA7 25 55 C[C@H](CN)c1ccc(CN2CCC[C@@H](C)C2)cc1 ZINC000217898765 BF For-Sale Unstable HRH3 18 45 Cc1cccc(/C=C/NC(=O)Nc2cc(C)on2)c1 ZINC000217898815 CG For-Sale Unstable Q8MMZ8_EIMTE 0 41 O=C(/C=C/c1ccc([N+](=O)[O-])cc1)NCCCN1CCCc2ccccc21 ZINC000217898853 FH In-Stock Unstable DRD3 17 57 Clc1ccc(/C=C\CN2CCN(Cc3cccnc3)CC2)cc1 ZINC000217898953 EH On-Demand Unstable DRD4 32 50 Clc1ccc(/C=C\CN2CCN(Cc3cccnc3)CC2)cc1 ZINC000217898953 EH On-Demand Unstable FAAH 16 41 Cc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cc2C)c1 ZINC000217898965 DJ For-Sale Unstable KCNK3 32 40 Cc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cc2C)c1 ZINC000217898965 DJ For-Sale Unstable KCNK9 23 40 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccccc2Cl)c1 ZINC000217898967 EI In-Stock Unstable KCNQ2 52 44 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccccc2Cl)c1 ZINC000217898967 EI In-Stock Unstable PDS 66 38 Clc1ccc(/C=C/CN2CCN(Cc3cccnc3)CC2)cc1 ZINC000217899021 EH On-Demand Unstable DRD4 32 50 Clc1ccc(/C=C/CN2CCN(Cc3cccnc3)CC2)cc1 ZINC000217899021 EH On-Demand Unstable FAAH 16 41 O=C(c1cccc(Br)c1)N1C[C@H]2CNC[C@@H](C2)C1 ZINC000217899051 DE For-Sale Unstable CHRNA7 26 54 CCOc1ccc(CNC(=O)/C=C/c2ccccc2Cl)cc1OCC ZINC000217899081 FI In-Stock Unstable PDE6A 42 32 Cc1cc(Cl)ccc1OCC(=O)N[C@H]1CCC[C@@H]1CO ZINC000217899166 CE For-Sale Unstable PTGDR2 27 40 O=C(Nc1ccccc1)[C@H]1[C@@H]2C=C[C@@H]([C@H]3C[C@@H]23)[C@H]1C(=O)O ZINC000217899211 CE In-Stock Unstable P95276_MYCTO 0 40 COc1cc(CNC(=O)/C=C/c2ccccc2Cl)ccc1OC(C)C ZINC000217899212 FI In-Stock Unstable PTGER2 22 40 COc1cc(CNC(=O)/C=C/c2ccccc2Cl)ccc1OC(C)C ZINC000217899212 FI In-Stock Unstable PTGER4 19 40 COc1cc(CNC(=O)/C=C/c2ccccc2Cl)ccc1OC(C)C ZINC000217899212 FI In-Stock Unstable KCNQ2 29 41 COc1cc(CNC(=O)/C=C/c2ccccc2Cl)ccc1OC(C)C ZINC000217899212 FI In-Stock Unstable PDE6A 41 31 COc1cc(CNC(=O)/C=C/c2ccccc2Cl)ccc1OC(C)C ZINC000217899212 FI In-Stock Unstable CYSP_PLAFA 42 36 O=C(CCc1cc(Cl)no1)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217899234 EE In-Stock Unstable CHRNA4 31 46 Cc1cc(Cl)ccc1OCC(=O)N[C@@H]1CCC[C@H]1CO ZINC000217899254 CE For-Sale Unstable PTGDR2 27 40 O=C(c1ccc(Br)cc1)N1C[C@H]2CNC[C@@H](C2)C1 ZINC000217899265 DE For-Sale Unstable CHRNA7 33 66 CN(C)S(=O)(=O)c1ccc(C(=O)N(Cc2cc(C3CC3)n(C)n2)C2CCCC2)cc1 ZINC000217899293 IG In-Stock Unstable AVPR1B 17 43 CN1CCO[C@H]([C@@H](N)C[C@@H]2CCCc3ccccc32)C1 ZINC000217899324 CE For-Sale Unstable EBP 19 40 O=C(/C=C/c1ccccc1Cl)NCCCc1ccccc1Cl ZINC000217899327 EJ In-Stock Unstable PYGL 23 47 O=C(/C=C/c1ccccc1Cl)NCCCc1ccccc1Cl ZINC000217899327 EJ In-Stock Unstable HDAC9 27 41 O=C(/C=C/c1ccccc1Cl)NCCCc1ccccc1Cl ZINC000217899327 EJ In-Stock Unstable HDAC7 32 41 Cc1cc(Cl)ccc1OCC(=O)N[C@H]1CCC[C@H]1CO ZINC000217899357 CE For-Sale Unstable PTGDR2 27 40 COc1cc([C@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)ccc1O ZINC000217899384 KH In-Stock Unstable AKR1B1 0 46 COc1cc([C@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)ccc1O ZINC000217899384 KH In-Stock Unstable CYP1B1 47 37 COc1cc([C@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)ccc1O ZINC000217899384 KH In-Stock Unstable CYP1A1 42 37 COc1cc([C@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)ccc1O ZINC000217899384 KH In-Stock Unstable RORC 55 40 COC(=O)CCSCc1cc(/C=C\C(=O)O)ccc1OC ZINC000217899406 DF For-Sale Unstable TUBB1 41 36 COC(=O)CCSCc1cc(/C=C\C(=O)O)ccc1OC ZINC000217899406 DF For-Sale Unstable AKR1C3 25 47 O=S(=O)(c1ccccc1)N(CCF)Cc1ccncc1 ZINC000217899442 CE For-Sale Unstable CXCR3 20 41 O=C(/C=C/c1ccccc1Cl)NCCCc1ccc(Cl)cc1 ZINC000217899443 EJ In-Stock Unstable PYGL 23 45 O=C(/C=C/c1ccccc1Cl)NCCCc1ccc(Cl)cc1 ZINC000217899443 EJ In-Stock Unstable HDAC9 27 45 O=C(/C=C/c1ccccc1Cl)NCCCc1ccc(Cl)cc1 ZINC000217899443 EJ In-Stock Unstable HDAC7 32 45 O=C(/C=C/c1ccccc1Cl)NCCCc1ccc(Cl)cc1 ZINC000217899443 EJ In-Stock Unstable BOTA 24 42 O=C(CCc1ccc(F)c(F)c1)N[C@@H]1CCC[C@@H]1CO ZINC000217899451 CE For-Sale Unstable SSTR3 18 41 COc1cc([C@@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)ccc1O ZINC000217899475 KH In-Stock Unstable AKR1B1 0 46 COc1cc([C@@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)ccc1O ZINC000217899475 KH In-Stock Unstable CYP1B1 47 37 COc1cc([C@@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)ccc1O ZINC000217899475 KH In-Stock Unstable CYP1A1 42 37 COc1cc([C@@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)ccc1O ZINC000217899475 KH In-Stock Unstable RORC 55 40 Cc1ccccc1SCc1ccccc1/C=C\C(=O)O ZINC000217899483 CI For-Sale Unstable PTGER2 22 49 Cc1ccccc1SCc1ccccc1/C=C\C(=O)O ZINC000217899483 CI For-Sale Unstable PTGER4 0 50 Cc1ccccc1SCc1ccccc1/C=C\C(=O)O ZINC000217899483 CI For-Sale Unstable PTGER3 22 54 Cc1ccccc1SCc1ccccc1/C=C\C(=O)O ZINC000217899483 CI For-Sale Unstable PTGDR 0 54 O=C(CCc1ccc(F)c(F)c1)N[C@H]1CCC[C@@H]1CO ZINC000217899521 CE For-Sale Unstable SSTR3 18 41 COc1ccccc1CCCNC(=O)/C=C/c1ccccc1Cl ZINC000217899543 EI In-Stock Unstable DRD3 26 62 COc1ccccc1CCCNC(=O)/C=C/c1ccccc1Cl ZINC000217899543 EI In-Stock Unstable PTGER2 31 43 COc1ccccc1CCCNC(=O)/C=C/c1ccccc1Cl ZINC000217899543 EI In-Stock Unstable PYGL 0 41 COc1ccccc1CCCNC(=O)/C=C/c1ccccc1Cl ZINC000217899543 EI In-Stock Unstable MTNR1B 36 41 Cc1ccccc1SCc1ccc(/C=C\C(=O)O)cc1 ZINC000217899563 CI For-Sale Unstable PTGER2 41 51 Cc1ccccc1SCc1ccc(/C=C\C(=O)O)cc1 ZINC000217899563 CI For-Sale Unstable PTGER4 0 43 Cc1ccccc1SCc1ccc(/C=C\C(=O)O)cc1 ZINC000217899563 CI For-Sale Unstable PTGER3 15 44 Cc1ccccc1SCc1ccc(/C=C\C(=O)O)cc1 ZINC000217899563 CI For-Sale Unstable NPY2R 0 46 Cc1ccccc1SCc1ccc(/C=C\C(=O)O)cc1 ZINC000217899563 CI For-Sale Unstable PTGDR 0 44 Cc1ccccc1SCc1ccc(/C=C\C(=O)O)cc1 ZINC000217899563 CI For-Sale Unstable AKR1C3 23 40 O=C(CCc1ccc(F)c(F)c1)N[C@@H]1CCC[C@H]1CO ZINC000217899598 CE For-Sale Unstable SSTR3 18 41 Cc1ccc(N2CCN(Cc3oc(CN4C[C@@H]5C[C@H](C4)c4cccc(=O)n4C5)cc(=O)c3O)CC2)c(C)c1 ZINC000217899615 KG In-Stock Unstable CHRNA4 27 45 Cc1ccccc1SCc1cccc(/C=C\C(=O)O)c1 ZINC000217899644 CI For-Sale Unstable PTGER2 22 53 Cc1ccccc1SCc1cccc(/C=C\C(=O)O)c1 ZINC000217899644 CI For-Sale Unstable PTGER3 15 41 Cc1ccccc1SCc1cccc(/C=C\C(=O)O)c1 ZINC000217899644 CI For-Sale Unstable NPY2R 0 45 Cc1ccccc1SCc1cccc(/C=C\C(=O)O)c1 ZINC000217899644 CI For-Sale Unstable PTGDR 0 40 Cc1ccccc1SCc1cccc(/C=C\C(=O)O)c1 ZINC000217899644 CI For-Sale Unstable HDA106 0 43 Cc1ccccc1SCc1cccc(/C=C\C(=O)O)c1 ZINC000217899644 CI For-Sale Unstable AKR1C3 32 42 C[C@@H](CCc1ccc(O)cc1)NC(=O)[C@@H]1C[C@@H](O)CN1 ZINC000217899645 CC For-Sale Unstable YARS 68 34 O=C(CCc1ccc(F)c(F)c1)N[C@H]1CCC[C@H]1CO ZINC000217899666 CE For-Sale Unstable SSTR3 18 41 COc1cccc(CCCNC(=O)/C=C/c2ccccc2Cl)c1 ZINC000217899676 EI In-Stock Unstable DRD4 47 40 COc1cccc(CCCNC(=O)/C=C/c2ccccc2Cl)c1 ZINC000217899676 EI In-Stock Unstable PTAFR 22 45 COc1cccc(CCCNC(=O)/C=C/c2ccccc2Cl)c1 ZINC000217899676 EI In-Stock Unstable PYGL 21 41 COc1cccc(CCCNC(=O)/C=C/c2ccccc2Cl)c1 ZINC000217899676 EI In-Stock Unstable MTNR1B 49 59 COc1cccc(CCCNC(=O)/C=C/c2ccccc2Cl)c1 ZINC000217899676 EI In-Stock Unstable CRTM 74 49 COc1cccc(CCCNC(=O)/C=C/c2ccccc2Cl)c1 ZINC000217899676 EI In-Stock Unstable CAN2 0 48 COc1cccc(CCCNC(=O)/C=C/c2ccccc2Cl)c1 ZINC000217899676 EI In-Stock Unstable CYSP_PLAFA 27 42 C[C@H](CCc1ccc(O)cc1)NC(=O)[C@@H]1C[C@@H](O)CN1 ZINC000217899709 CC For-Sale Unstable YARS 68 34 CCCCCCC(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217899743 BE On-Demand Unstable FAAH 0 44 CCCCCCC(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217899743 BE On-Demand Unstable LUXR 35 46 CCCCCCC(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217899743 BE On-Demand Unstable TRAR 15 46 CCCCCCC(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217899743 BE On-Demand Unstable LASR 64 46 CCCCCCC(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217899743 BE On-Demand Unstable PHZR 0 46 CCCCCCC(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217899743 BE On-Demand Unstable CQSS 52 32 Cc1ccccc1-c1nc(N)nc2c1CN(C(=O)OC(C)(C)C)CC2 ZINC000217899753 EG For-Sale Unstable P2RY14 57 45 C[C@@H](CCc1ccc(O)cc1)NC(=O)[C@H]1C[C@@H](O)CN1 ZINC000217899783 CC For-Sale Unstable YARS 68 34 FC(F)[C@H]1CNc2cc(Br)ccc21 ZINC000217899811 BG For-Sale Unstable PNMT 15 40 COc1ccc(CCCNC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217899814 EI In-Stock Unstable SCNN1A 55 40 COc1ccc(CCCNC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217899814 EI In-Stock Unstable PTGER2 22 45 COc1ccc(CCCNC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217899814 EI In-Stock Unstable PTGER4 0 45 COc1ccc(CCCNC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217899814 EI In-Stock Unstable PYGL 0 41 COc1ccc(CCCNC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217899814 EI In-Stock Unstable CDC25B 0 42 COc1ccc(CCCNC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217899814 EI In-Stock Unstable MTNR1A 40 34 COc1ccc(CCCNC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217899814 EI In-Stock Unstable MTNR1B 40 38 COc1ccc(CCCNC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217899814 EI In-Stock Unstable CRTM 41 37 CCCCCCC(=O)N[C@H]1CCC[C@@H]1CO ZINC000217899846 BE For-Sale Unstable FAAH 0 44 CCCCCCC(=O)N[C@H]1CCC[C@@H]1CO ZINC000217899846 BE For-Sale Unstable LUXR 35 46 CCCCCCC(=O)N[C@H]1CCC[C@@H]1CO ZINC000217899846 BE For-Sale Unstable TRAR 15 46 CCCCCCC(=O)N[C@H]1CCC[C@@H]1CO ZINC000217899846 BE For-Sale Unstable LASR 64 46 CCCCCCC(=O)N[C@H]1CCC[C@@H]1CO ZINC000217899846 BE For-Sale Unstable PHZR 0 46 CCCCCCC(=O)N[C@H]1CCC[C@@H]1CO ZINC000217899846 BE For-Sale Unstable CQSS 52 32 C[C@H](CCc1ccc(O)cc1)NC(=O)[C@H]1C[C@@H](O)CN1 ZINC000217899870 CC For-Sale Unstable YARS 68 34 FC(F)[C@@H]1CNc2cc(Br)ccc21 ZINC000217899885 BG For-Sale Unstable PNMT 15 40 CCCCCCC(=O)N[C@@H]1CCC[C@H]1CO ZINC000217899913 BE For-Sale Unstable FAAH 0 44 CCCCCCC(=O)N[C@@H]1CCC[C@H]1CO ZINC000217899913 BE For-Sale Unstable LUXR 35 46 CCCCCCC(=O)N[C@@H]1CCC[C@H]1CO ZINC000217899913 BE For-Sale Unstable TRAR 15 46 CCCCCCC(=O)N[C@@H]1CCC[C@H]1CO ZINC000217899913 BE For-Sale Unstable LASR 64 46 CCCCCCC(=O)N[C@@H]1CCC[C@H]1CO ZINC000217899913 BE For-Sale Unstable PHZR 0 46 CCCCCCC(=O)N[C@@H]1CCC[C@H]1CO ZINC000217899913 BE For-Sale Unstable CQSS 52 32 COc1ccc(COCCC(C)C)cc1/C=C\C(=O)O ZINC000217899916 CG For-Sale Unstable PTGER2 36 45 COc1ccc(COCCC(C)C)cc1/C=C\C(=O)O ZINC000217899916 CG For-Sale Unstable PTGER4 23 45 COc1ccc(COCCC(C)C)cc1/C=C\C(=O)O ZINC000217899916 CG For-Sale Unstable PTGER3 19 45 COc1ccc(COCCC(C)C)cc1/C=C\C(=O)O ZINC000217899916 CG For-Sale Unstable AKR1B10 31 41 Cc1cc(C(=O)N(Cc2cc(C3CC3)n(C)n2)C2CCCC2)no1 ZINC000217899943 EG In-Stock Unstable S1PR3 24 57 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217899944 EH In-Stock Unstable PTGER2 0 41 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217899944 EH In-Stock Unstable SDH1 0 42 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217899944 EH In-Stock Unstable KCNQ2 51 45 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217899944 EH In-Stock Unstable CDC25B 0 45 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217899944 EH In-Stock Unstable UL26 30 41 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217899944 EH In-Stock Unstable U53 0 41 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217899944 EH In-Stock Unstable SCAF_EBVB9 15 41 CCCc1nc2ccccc2n1CCC(C)=O ZINC000217899988 BF For-Sale Unstable AGTR1 30 45 CCCc1nc2ccccc2n1CCC(C)=O ZINC000217899988 BF For-Sale Unstable HRH1 17 40 CCCc1nc2ccccc2n1CCC(C)=O ZINC000217899988 BF For-Sale Unstable AGTR1B 25 45 CCCc1nc2ccccc2n1CCC(C)=O ZINC000217899988 BF For-Sale Unstable HDAC1 16 43 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217900011 EH In-Stock Unstable PTGER2 0 41 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217900011 EH In-Stock Unstable SDH1 0 42 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217900011 EH In-Stock Unstable KCNQ2 51 45 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217900011 EH In-Stock Unstable CDC25B 0 45 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217900011 EH In-Stock Unstable UL26 30 41 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217900011 EH In-Stock Unstable U53 0 41 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217900011 EH In-Stock Unstable SCAF_EBVB9 15 41 C[C@H](OCc1ccccc1/C=C\C(=O)O)c1ccccc1 ZINC000217900015 CI For-Sale Unstable PTGER2 55 49 C[C@H](OCc1ccccc1/C=C\C(=O)O)c1ccccc1 ZINC000217900015 CI For-Sale Unstable PTGER4 25 44 C[C@H](OCc1ccccc1/C=C\C(=O)O)c1ccccc1 ZINC000217900015 CI For-Sale Unstable PTGER3 21 49 C[C@H](OCc1ccccc1/C=C\C(=O)O)c1ccccc1 ZINC000217900015 CI For-Sale Unstable PTGDR 0 47 CCCCCCC(=O)N[C@H]1CCC[C@H]1CO ZINC000217900033 BE For-Sale Unstable FAAH 0 44 CCCCCCC(=O)N[C@H]1CCC[C@H]1CO ZINC000217900033 BE For-Sale Unstable LUXR 35 46 CCCCCCC(=O)N[C@H]1CCC[C@H]1CO ZINC000217900033 BE For-Sale Unstable TRAR 15 46 CCCCCCC(=O)N[C@H]1CCC[C@H]1CO ZINC000217900033 BE For-Sale Unstable LASR 64 46 CCCCCCC(=O)N[C@H]1CCC[C@H]1CO ZINC000217900033 BE For-Sale Unstable PHZR 0 46 CCCCCCC(=O)N[C@H]1CCC[C@H]1CO ZINC000217900033 BE For-Sale Unstable CQSS 52 32 CCc1cc(Br)cc([C@@H](C)C(=O)O)c1 ZINC000217900042 CG For-Sale Unstable PTGS1 27 48 CCc1cc(Br)cc([C@@H](C)C(=O)O)c1 ZINC000217900042 CG For-Sale Unstable PTGS2 19 48 CCCc1nc2ccccc2n1C[C@@H](C)C(=O)OC ZINC000217900089 CF For-Sale Unstable AGTR1 56 44 CCCc1nc2ccccc2n1C[C@@H](C)C(=O)OC ZINC000217900089 CF For-Sale Unstable AGTR2 41 36 CCCc1nc2ccccc2n1C[C@@H](C)C(=O)OC ZINC000217900089 CF For-Sale Unstable AGTR1B 53 44 CCCc1nc2ccccc2n1C[C@@H](C)C(=O)OC ZINC000217900089 CF For-Sale Unstable PDE6D 48 34 C[C@@H](OCc1ccccc1/C=C\C(=O)O)c1ccccc1 ZINC000217900097 CI For-Sale Unstable PTGER2 55 49 C[C@@H](OCc1ccccc1/C=C\C(=O)O)c1ccccc1 ZINC000217900097 CI For-Sale Unstable PTGER4 25 44 C[C@@H](OCc1ccccc1/C=C\C(=O)O)c1ccccc1 ZINC000217900097 CI For-Sale Unstable PTGER3 21 49 C[C@@H](OCc1ccccc1/C=C\C(=O)O)c1ccccc1 ZINC000217900097 CI For-Sale Unstable PTGDR 0 47 CCc1cc(Br)cc([C@H](C)C(=O)O)c1 ZINC000217900106 CG For-Sale Unstable PTGS1 27 48 CCc1cc(Br)cc([C@H](C)C(=O)O)c1 ZINC000217900106 CG For-Sale Unstable PTGS2 19 48 CC(C)COc1ccc(C(=O)N[C@@H]2CCC[C@@H]2CO)cc1 ZINC000217900115 CF On-Demand Unstable SSTR3 25 42 O=C(/C=C/c1ccccc1Cl)Nc1ccccc1C(=O)c1ccccc1 ZINC000217900135 FK In-Stock Anodyne MMP2 19 56 O=C(/C=C/c1ccccc1Cl)Nc1ccccc1C(=O)c1ccccc1 ZINC000217900135 FK In-Stock Anodyne MMP9 16 52 O=C(/C=C/c1ccccc1Cl)Nc1ccccc1C(=O)c1ccccc1 ZINC000217900135 FK In-Stock Anodyne MMP1 0 56 O=C(/C=C/c1ccccc1Cl)Nc1ccccc1C(=O)c1ccccc1 ZINC000217900135 FK In-Stock Anodyne SMO 19 41 O=C(/C=C/c1ccccc1Cl)Nc1ccccc1C(=O)c1ccccc1 ZINC000217900135 FK In-Stock Anodyne TRPM2 0 40 CCCc1nc2ccccc2n1C[C@H](C)C(=O)OC ZINC000217900170 CF For-Sale Unstable AGTR1 56 44 CCCc1nc2ccccc2n1C[C@H](C)C(=O)OC ZINC000217900170 CF For-Sale Unstable AGTR2 41 36 CCCc1nc2ccccc2n1C[C@H](C)C(=O)OC ZINC000217900170 CF For-Sale Unstable AGTR1B 53 44 CCCc1nc2ccccc2n1C[C@H](C)C(=O)OC ZINC000217900170 CF For-Sale Unstable PDE6D 48 34 C[C@H](OCc1ccc(/C=C\C(=O)O)cc1)c1ccccc1 ZINC000217900184 CI For-Sale Unstable PTGER2 39 45 C[C@H](OCc1ccc(/C=C\C(=O)O)cc1)c1ccccc1 ZINC000217900184 CI For-Sale Unstable PTGER4 0 41 C[C@H](OCc1ccc(/C=C\C(=O)O)cc1)c1ccccc1 ZINC000217900184 CI For-Sale Unstable 17HSDCL 0 45 C[C@H](OCc1ccc(/C=C\C(=O)O)cc1)c1ccccc1 ZINC000217900184 CI For-Sale Unstable AKR1C3 33 44 C[C@H](OCc1ccc(/C=C\C(=O)O)cc1)c1ccccc1 ZINC000217900184 CI For-Sale Unstable AKR1B10 18 46 O[C@H](CN1CCO[C@@H]2CCC[C@@H]21)c1ccc2c(c1)OCO2 ZINC000217900193 CD For-Sale Unstable SSTR3 46 30 FC(F)[C@H]1Cc2cc(Br)ccc2N1 ZINC000217900196 BG For-Sale Unstable PNMT 27 41 CCc1ccc(Br)cc1[C@@H](C)C(=O)O ZINC000217900204 CG For-Sale Unstable PTGS1 30 46 CCc1ccc(Br)cc1[C@@H](C)C(=O)O ZINC000217900204 CG For-Sale Unstable PTGS2 22 44 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccccc2Cl)c1 ZINC000217900217 FJ In-Stock Unstable KCNQ2 41 41 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccccc2Cl)c1 ZINC000217900217 FJ In-Stock Unstable PYGL 0 40 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccccc2Cl)c1 ZINC000217900217 FJ In-Stock Unstable AMP1_PLAFQ 23 41 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccccc2Cl)c1 ZINC000217900217 FJ In-Stock Unstable CRTM 67 50 CCc1ccc(Br)cc1[C@H](C)C(=O)O ZINC000217900257 CG For-Sale Unstable PTGS1 30 46 CCc1ccc(Br)cc1[C@H](C)C(=O)O ZINC000217900257 CG For-Sale Unstable PTGS2 22 44 C[C@@H](OCc1ccc(/C=C\C(=O)O)cc1)c1ccccc1 ZINC000217900262 CI For-Sale Unstable PTGER2 39 45 C[C@@H](OCc1ccc(/C=C\C(=O)O)cc1)c1ccccc1 ZINC000217900262 CI For-Sale Unstable PTGER4 0 41 C[C@@H](OCc1ccc(/C=C\C(=O)O)cc1)c1ccccc1 ZINC000217900262 CI For-Sale Unstable 17HSDCL 0 45 C[C@@H](OCc1ccc(/C=C\C(=O)O)cc1)c1ccccc1 ZINC000217900262 CI For-Sale Unstable AKR1C3 33 44 C[C@@H](OCc1ccc(/C=C\C(=O)O)cc1)c1ccccc1 ZINC000217900262 CI For-Sale Unstable AKR1B10 18 46 CCCc1nc2ccccc2n1CCC(=O)OCC ZINC000217900280 CF For-Sale Unstable AGTR1 38 42 CCCc1nc2ccccc2n1CCC(=O)OCC ZINC000217900280 CF For-Sale Unstable AGTR1B 31 43 CCCc1nc2ccccc2n1CCC(=O)OCC ZINC000217900280 CF For-Sale Unstable HDAC1 15 40 FC(F)[C@@H]1Cc2cc(Br)ccc2N1 ZINC000217900308 BG For-Sale Unstable PNMT 27 41 CC(C)Oc1ccc(CCCNC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217900327 FJ In-Stock Unstable KCNQ2 21 40 CCc1cccc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217900358 CH For-Sale Unstable PTGER2 33 52 CCc1cccc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217900358 CH For-Sale Unstable PTGER4 44 62 CCc1cccc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217900358 CH For-Sale Unstable PTGER3 42 62 CCc1cccc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217900358 CH For-Sale Unstable LTB4R 24 40 CCc1cccc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217900358 CH For-Sale Unstable CDC25B 22 40 CCc1cccc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217900358 CH For-Sale Unstable ACE2 17 40 CCc1cccc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217900358 CH For-Sale Unstable PTGDR 0 60 CCc1cccc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217900358 CH For-Sale Unstable FFAR1 38 41 CCc1cccc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217900358 CH For-Sale Unstable AKR1C3 29 41 CCc1cccc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217900358 CH For-Sale Unstable CRTM 43 32 CCc1cccc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217900358 CH For-Sale Unstable PDS 64 36 Cc1cc([C@@H](C)C(=O)O)cc(Br)c1C ZINC000217900364 CG For-Sale Unstable PTGS1 21 49 CCCc1nc2ccccc2n1CCC(=O)OC ZINC000217900368 BF For-Sale Unstable AGTR1 49 43 CCCc1nc2ccccc2n1CCC(=O)OC ZINC000217900368 BF For-Sale Unstable HRH1 19 41 CCCc1nc2ccccc2n1CCC(=O)OC ZINC000217900368 BF For-Sale Unstable AGTR1B 31 43 Cn1nc(CN(C(=O)c2ccc(OC(F)(F)F)cc2)C2CCCC2)cc1C1CC1 ZINC000217900370 HJ In-Stock Unstable GCGR 26 40 Cn1nc(CN(C(=O)c2ccc(OC(F)(F)F)cc2)C2CCCC2)cc1C1CC1 ZINC000217900370 HJ In-Stock Unstable SLC6A9 15 46 CCC[C@@H](O)CNCCCC(=O)O ZINC000217900404 AC For-Sale Unstable FABP2 0 41 CCC[C@@H](O)CNCCCC(=O)O ZINC000217900404 AC For-Sale Unstable SLC22A20 0 42 CCC[C@@H](O)CNCCCC(=O)O ZINC000217900404 AC For-Sale Unstable SPPS 42 37 CCC[C@@H](O)CNCCCC(=O)O ZINC000217900404 AC For-Sale Unstable CQSS 40 34 FC(F)[C@@H]1Cc2ccc(Br)cc2N1 ZINC000217900405 BG For-Sale Unstable PNMT 38 47 O=C(O)CNC(=O)c1ccc2c(ccn2Cc2ccccc2)c1 ZINC000217900411 DF In-Stock Unstable GLO1 19 41 O=C(O)CNC(=O)c1ccc2c(ccn2Cc2ccccc2)c1 ZINC000217900411 DF In-Stock Unstable EGLN1 0 48 O=C(O)CNC(=O)c1ccc2c(ccn2Cc2ccccc2)c1 ZINC000217900411 DF In-Stock Unstable EGLN3 0 51 CCc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217900432 CH For-Sale Unstable ALOX5 23 52 CCc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217900432 CH For-Sale Unstable MAOB 49 50 CCc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217900432 CH For-Sale Unstable PTGER2 27 47 CCc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217900432 CH For-Sale Unstable PTGER4 37 58 CCc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217900432 CH For-Sale Unstable PTGER3 31 58 CCc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217900432 CH For-Sale Unstable DRTS_LEIMA 35 42 CCc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217900432 CH For-Sale Unstable DYR_PNECA 16 42 CCc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217900432 CH For-Sale Unstable LTB4R 35 41 CCc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217900432 CH For-Sale Unstable ACE2 15 42 CCc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217900432 CH For-Sale Unstable PTGDR 0 50 CCc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217900432 CH For-Sale Unstable FFAR1 59 48 CCc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217900432 CH For-Sale Unstable AKR1C3 37 49 CCc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217900432 CH For-Sale Unstable AKR1B10 22 40 CCc1cccc(OCc2ccc(/C=C\C(=O)O)cc2)c1 ZINC000217900432 CH For-Sale Unstable PDS 54 34 Cc1cc([C@H](C)C(=O)O)cc(Br)c1C ZINC000217900439 CG For-Sale Unstable PTGS1 21 49 O[C@@H](CN1CCO[C@@H]2CCC[C@@H]21)c1ccccc1 ZINC000217900449 BD On-Demand Unstable SLC18A3 24 41 COc1cccc(NC(=O)N(Cc2cc(C3CC3)n(C)n2)C2CCCC2)c1OC ZINC000217900470 GI In-Stock Unstable ACAT 40 40 CCC[C@H](O)CNCCCC(=O)O ZINC000217900475 AC For-Sale Unstable FABP2 0 41 CCC[C@H](O)CNCCCC(=O)O ZINC000217900475 AC For-Sale Unstable SLC22A20 0 42 CCC[C@H](O)CNCCCC(=O)O ZINC000217900475 AC For-Sale Unstable SPPS 42 37 CCC[C@H](O)CNCCCC(=O)O ZINC000217900475 AC For-Sale Unstable CQSS 40 34 FC(F)[C@H]1Cc2ccc(Br)cc2N1 ZINC000217900477 BG For-Sale Unstable PNMT 38 47 O=C(/C=C/c1ccccc1Cl)Nc1ccc(OC2CCCC2)cc1 ZINC000217900501 EK In-Stock Unstable EPHX2 22 40 O=C(C[C@@H]1NC(=O)N(CCc2ccccc2)C1=O)NCCc1ccc(O)cc1 ZINC000217900511 GD In-Stock Unstable SLC6A5 27 40 O=C(C[C@@H]1NC(=O)N(CCc2ccccc2)C1=O)NCCc1ccc(O)cc1 ZINC000217900511 GD In-Stock Unstable NCE103 21 43 O=C(C[C@@H]1NC(=O)N(CCc2ccccc2)C1=O)NCCc1ccc(O)cc1 ZINC000217900511 GD In-Stock Unstable P96878_MYCTU 16 43 O=C(C[C@@H]1NC(=O)N(CCc2ccccc2)C1=O)NCCc1ccc(O)cc1 ZINC000217900511 GD In-Stock Unstable CAN2 0 43 O[C@H](CN1CCO[C@@H]2CCC[C@@H]21)c1ccccc1 ZINC000217900526 BD On-Demand Unstable SLC18A3 24 41 CCc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217900536 CH For-Sale Unstable ALOX5 22 44 CCc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217900536 CH For-Sale Unstable MAOB 63 43 CCc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217900536 CH For-Sale Unstable PTGER2 23 50 CCc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217900536 CH For-Sale Unstable CYSLTR1 16 40 CCc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217900536 CH For-Sale Unstable PTGER4 30 56 CCc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217900536 CH For-Sale Unstable PTGER3 28 56 CCc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217900536 CH For-Sale Unstable DRTS_LEIMA 27 40 CCc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217900536 CH For-Sale Unstable LTB4R 27 45 CCc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217900536 CH For-Sale Unstable NR1H4 48 36 CCc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217900536 CH For-Sale Unstable PTGDR 0 45 CCc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217900536 CH For-Sale Unstable FFAR1 65 46 CCc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217900536 CH For-Sale Unstable AKR1C3 37 53 CCc1cccc(OCc2cccc(/C=C\C(=O)O)c2)c1 ZINC000217900536 CH For-Sale Unstable PDS 58 35 COc1ccc(CCCCCc2ccccc2)cc1 ZINC000217900587 CJ For-Sale Unstable ALOX5 17 58 COc1ccc(CCCCCc2ccccc2)cc1 ZINC000217900587 CJ For-Sale Unstable DRTS_PLAFK 22 40 COc1ccc(CCCCCc2ccccc2)cc1 ZINC000217900587 CJ For-Sale Unstable HTR2A 15 53 COc1ccc(CCCCCc2ccccc2)cc1 ZINC000217900587 CJ For-Sale Unstable HTR2C 16 53 COc1ccc(CCCCCc2ccccc2)cc1 ZINC000217900587 CJ For-Sale Unstable INHA 64 41 COc1ccc(CCCCCc2ccccc2)cc1 ZINC000217900587 CJ For-Sale Unstable SLC18A2 50 46 COc1ccc(CCCCCc2ccccc2)cc1 ZINC000217900587 CJ For-Sale Unstable SIGMAR1 53 63 COc1ccc(CCCCCc2ccccc2)cc1 ZINC000217900587 CJ For-Sale Unstable G6PC 26 44 COc1ccc(CCCCCc2ccccc2)cc1 ZINC000217900587 CJ For-Sale Unstable P2RX1 15 40 COc1ccc(CCCCCc2ccccc2)cc1 ZINC000217900587 CJ For-Sale Unstable LTB4R 43 38 COc1ccc(CCCCCc2ccccc2)cc1 ZINC000217900587 CJ For-Sale Unstable KCNA3 15 44 COc1ccc(CCCCCc2ccccc2)cc1 ZINC000217900587 CJ For-Sale Unstable SCN2A 26 49 COc1ccc(CCCCCc2ccccc2)cc1 ZINC000217900587 CJ For-Sale Unstable MTNR1B 19 41 COc1ccc(CCCCCc2ccccc2)cc1 ZINC000217900587 CJ For-Sale Unstable MMP3 18 47 COc1ccc(CCCCCc2ccccc2)cc1 ZINC000217900587 CJ For-Sale Unstable EBP 18 42 COc1ccc(CCCCCc2ccccc2)cc1 ZINC000217900587 CJ For-Sale Unstable SLC2A1 17 42 COc1ccc(CCCCCc2ccccc2)cc1 ZINC000217900587 CJ For-Sale Unstable PLA2G4B 17 43 COc1ccc(CCCCCc2ccccc2)cc1 ZINC000217900587 CJ For-Sale Unstable FAAH 69 44 COc1ccc(CCCCCc2ccccc2)cc1 ZINC000217900587 CJ For-Sale Unstable ABCB1 17 54 COc1ccc(CCCCCc2ccccc2)cc1 ZINC000217900587 CJ For-Sale Unstable ALOX15 32 44 COc1ccc(CCCCCc2ccccc2)cc1 ZINC000217900587 CJ For-Sale Unstable CES1 71 41 COc1ccc(CCCCCc2ccccc2)cc1 ZINC000217900587 CJ For-Sale Unstable PTGDR 24 43 COc1ccc(CCCCCc2ccccc2)cc1 ZINC000217900587 CJ For-Sale Unstable AOC3 25 48 COc1ccc(CCCCCc2ccccc2)cc1 ZINC000217900587 CJ For-Sale Unstable MGLL 17 48 COc1ccc(CCCCCc2ccccc2)cc1 ZINC000217900587 CJ For-Sale Unstable TAAR1 33 53 COc1ccc(CCCCCc2ccccc2)cc1 ZINC000217900587 CJ For-Sale Unstable HT1 15 42 COc1ccc(CCCCCc2ccccc2)cc1 ZINC000217900587 CJ For-Sale Unstable FFAR4 19 41 COc1ccc(CCCCCc2ccccc2)cc1 ZINC000217900587 CJ For-Sale Unstable LUCI_PHOPY 36 40 COc1ccc(CCCCCc2ccccc2)cc1 ZINC000217900587 CJ For-Sale Unstable LMGT2 17 42 Cc1cccc(/C=C/NC(=O)Nc2ccc(Nc3ccccc3)cc2)c1 ZINC000217900610 EK For-Sale Unstable CCKAR 0 46 Cc1cccc(/C=C/NC(=O)Nc2ccc(Nc3ccccc3)cc2)c1 ZINC000217900610 EK For-Sale Unstable HDAC8 19 42 Cc1cccc(/C=C/NC(=O)Nc2ccc(Nc3ccccc3)cc2)c1 ZINC000217900610 EK For-Sale Unstable MMP2 0 45 Cc1cccc(/C=C/NC(=O)Nc2ccc(Nc3ccccc3)cc2)c1 ZINC000217900610 EK For-Sale Unstable MMP9 0 45 Cc1cccc(/C=C/NC(=O)Nc2ccc(Nc3ccccc3)cc2)c1 ZINC000217900610 EK For-Sale Unstable MMP1 0 45 Cc1cccc(/C=C/NC(=O)Nc2ccc(Nc3ccccc3)cc2)c1 ZINC000217900610 EK For-Sale Unstable AKR1C3 29 45 Cc1cccc(/C=C/NC(=O)Nc2ccc(Nc3ccccc3)cc2)c1 ZINC000217900610 EK For-Sale Unstable TRPM8 0 41 Cc1cccc(/C=C/NC(=O)Nc2ccc(Nc3ccccc3)cc2)c1 ZINC000217900610 EK For-Sale Unstable AKR1C2 20 43 Cc1cccc(/C=C/NC(=O)Nc2ccc(Nc3ccccc3)cc2)c1 ZINC000217900610 EK For-Sale Unstable P95276_MYCTO 0 40 Cc1cccc(/C=C/NC(=O)Nc2ccc(Nc3ccccc3)cc2)c1 ZINC000217900610 EK For-Sale Unstable KCNK3 64 41 Cc1cccc(/C=C/NC(=O)Nc2ccc(Nc3ccccc3)cc2)c1 ZINC000217900610 EK For-Sale Unstable KCNK9 44 41 CCC(C)(C)OCc1cc(/C=C\C(=O)O)ccc1OC ZINC000217900613 CG For-Sale Unstable PTGER2 0 43 CCC(C)(C)OCc1cc(/C=C\C(=O)O)ccc1OC ZINC000217900613 CG For-Sale Unstable TUBB1 49 40 CCC(C)(C)OCc1cc(/C=C\C(=O)O)ccc1OC ZINC000217900613 CG For-Sale Unstable AKR1C3 23 41 CCC(C)(C)OCc1cc(/C=C\C(=O)O)ccc1OC ZINC000217900613 CG For-Sale Unstable ABCG2 15 42 CC1(C)C[C@@H](NC(=O)/C=C/c2ccccc2Cl)c2ccccc2O1 ZINC000217900617 EJ In-Stock Unstable KCNQ2 21 44 CC[C@@H](C(=O)NC[C@@H]1CC[C@@H](C)NC1)c1ccccc1 ZINC000217900654 CF For-Sale Unstable KCNQ2 42 40 Cn1nc(CN(C(=O)NCc2ccc(Cl)cc2)C2CCCC2)cc1C1CC1 ZINC000217900683 GJ In-Stock Unstable IL2RA 50 32 Cn1nc(CN(C(=O)NCc2ccc(Cl)cc2)C2CCCC2)cc1C1CC1 ZINC000217900683 GJ In-Stock Unstable UL54 56 32 CC1(C)C[C@H](NC(=O)/C=C/c2ccccc2Cl)c2ccccc2O1 ZINC000217900706 EJ In-Stock Unstable KCNQ2 21 44 CCC(C)(C)OCc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217900712 CG For-Sale Unstable PTGER2 39 46 CCC(C)(C)OCc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217900712 CG For-Sale Unstable PTGER4 22 46 CCC(C)(C)OCc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217900712 CG For-Sale Unstable PTGER3 17 46 CCC(C)(C)OCc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217900712 CG For-Sale Unstable AKR1B10 29 40 CC[C@H](C(=O)NC[C@@H]1CC[C@@H](C)NC1)c1ccccc1 ZINC000217900726 CF For-Sale Unstable KCNQ2 42 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1c2ccccc2nc2ccccc12 ZINC000217900751 II For-Sale Unstable HCRTR2 40 37 Cc1cccc(/C=C/NC(=O)N2CCc3ccccc3C2)c1 ZINC000217900754 CH For-Sale Unstable HDAC6 32 44 Cc1cccc(/C=C/NC(=O)N2CCc3ccccc3C2)c1 ZINC000217900754 CH For-Sale Unstable BCL2 0 41 CCCCCOCCOc1cccc(/C=C\C(=O)O)c1 ZINC000217900767 CG For-Sale Unstable THRA 48 43 CCCCCOCCOc1cccc(/C=C\C(=O)O)c1 ZINC000217900767 CG For-Sale Unstable THRB 29 43 CCCCCOCCOc1cccc(/C=C\C(=O)O)c1 ZINC000217900767 CG For-Sale Unstable CYSLTR2 15 55 CCCCCOCCOc1cccc(/C=C\C(=O)O)c1 ZINC000217900767 CG For-Sale Unstable LTB4R 35 46 CCCCCOCCOc1cccc(/C=C\C(=O)O)c1 ZINC000217900767 CG For-Sale Unstable PLA2G4B 97 47 CCCCCOCCOc1cccc(/C=C\C(=O)O)c1 ZINC000217900767 CG For-Sale Unstable FAAH 22 42 CCCCCOCCOc1cccc(/C=C\C(=O)O)c1 ZINC000217900767 CG For-Sale Unstable AKR1C3 28 44 CCOc1ccc(CCCNC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217900808 EJ In-Stock Unstable SCN2A 19 44 CCOc1ccc(CCCNC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217900808 EJ In-Stock Unstable CRTM 40 38 NC1C[C@@H]2CC[C@H](C1)N2CCc1ccc(Br)cc1 ZINC000217900809 DF For-Sale Unstable Q8WSF8_APLCA 17 42 CC[C@@H](C(=O)NC[C@H]1CC[C@@H](C)NC1)c1ccccc1 ZINC000217900821 CF For-Sale Unstable KCNQ2 42 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1c2ccccc2nc2ccccc12 ZINC000217900829 II For-Sale Unstable HCRTR2 40 37 COc1ccc(/C=C\C(=O)O)cc1COCc1cccs1 ZINC000217900845 DH For-Sale Unstable AKR1C3 32 41 Cn1nc(CN(C(=O)NCc2ccc(F)cc2)C2CCCC2)cc1C1CC1 ZINC000217900857 FI In-Stock Unstable CCR5 54 35 Cn1nc(CN(C(=O)NCc2ccc(F)cc2)C2CCCC2)cc1C1CC1 ZINC000217900857 FI In-Stock Unstable ACAT 42 41 O=C(O)[C@@H]1CC[C@](O)(c2ccccc2)C1 ZINC000217900864 BD In-Stock Unstable OPRL1 18 43 Cc1cccc(/C=C/NC(=O)Nc2cccc(C)n2)c1 ZINC000217900874 CG For-Sale Unstable GRM5 19 48 Cc1cccc(/C=C/NC(=O)Nc2cccc(C)n2)c1 ZINC000217900874 CG For-Sale Unstable SORT1 17 42 CC[C@H](C(=O)NC[C@H]1CC[C@@H](C)NC1)c1ccccc1 ZINC000217900898 CF For-Sale Unstable KCNQ2 42 40 Cc1c(Br)ccc([C@@H](C)C(=O)O)c1C ZINC000217900907 CG For-Sale Unstable PTGS1 26 42 Cc1c(Br)ccc([C@@H](C)C(=O)O)c1C ZINC000217900907 CG For-Sale Unstable PTGS2 19 42 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccccc1Cl ZINC000217900919 FJ In-Stock Unstable MTNR1A 28 44 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccccc1Cl ZINC000217900919 FJ In-Stock Unstable MTNR1B 27 44 COc1ccc(COCc2cccs2)cc1/C=C\C(=O)O ZINC000217900930 DH For-Sale Unstable PTGER4 31 45 COc1ccc(COCc2cccs2)cc1/C=C\C(=O)O ZINC000217900930 DH For-Sale Unstable PTGER3 26 45 COc1ccc(COCc2cccs2)cc1/C=C\C(=O)O ZINC000217900930 DH For-Sale Unstable TNFRSF1A 37 43 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1c2ccccc2nc2ccccc12 ZINC000217900940 II For-Sale Unstable HCRTR2 40 37 O=C(O)[C@H]1CC[C@](O)(c2ccccc2)C1 ZINC000217900945 BD In-Stock Unstable OPRL1 18 43 Cn1nc(CN(C(=O)NCc2ccc3c(c2)OCO3)C2CCCC2)cc1C1CC1 ZINC000217900956 GH In-Stock Unstable NOS2 100 40 Cn1nc(CN(C(=O)NCc2ccc3c(c2)OCO3)C2CCCC2)cc1C1CC1 ZINC000217900956 GH In-Stock Unstable SSTR3 58 29 Cc1c(Br)ccc([C@H](C)C(=O)O)c1C ZINC000217900963 CG For-Sale Unstable PTGS1 26 42 Cc1c(Br)ccc([C@H](C)C(=O)O)c1C ZINC000217900963 CG For-Sale Unstable PTGS2 19 42 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccccc1Cl ZINC000217901007 EI In-Stock Unstable PTGER2 24 40 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccccc1Cl ZINC000217901007 EI In-Stock Unstable SDH1 0 40 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccccc1Cl ZINC000217901007 EI In-Stock Unstable KCNQ2 51 45 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccccc1Cl ZINC000217901007 EI In-Stock Unstable UL26 32 43 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccccc1Cl ZINC000217901007 EI In-Stock Unstable U53 0 43 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccccc1Cl ZINC000217901007 EI In-Stock Unstable SCAF_EBVB9 26 43 O=C(O)/C=C\c1ccc(COCc2cccs2)c(F)c1 ZINC000217901013 CH For-Sale Unstable HCAR2 0 40 O=C(O)/C=C\c1ccc(COCc2cccs2)c(F)c1 ZINC000217901013 CH For-Sale Unstable AKR1C3 30 43 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1c2ccccc2nc2ccccc12 ZINC000217901018 II For-Sale Unstable HCRTR2 40 37 O=C(O)[C@@H]1CC[C@@](O)(c2ccccc2)C1 ZINC000217901019 BD In-Stock Unstable OPRL1 18 43 Cc1cc([C@@H](C)C(=O)O)c(C)cc1Br ZINC000217901075 CG For-Sale Unstable PTGS1 20 41 Cc1ccccc1OC[C@H](C)NC(=O)/C=C/c1ccccc1Cl ZINC000217901087 EI In-Stock Unstable PTGER2 24 40 Cc1ccccc1OC[C@H](C)NC(=O)/C=C/c1ccccc1Cl ZINC000217901087 EI In-Stock Unstable SDH1 0 40 Cc1ccccc1OC[C@H](C)NC(=O)/C=C/c1ccccc1Cl ZINC000217901087 EI In-Stock Unstable KCNQ2 51 45 Cc1ccccc1OC[C@H](C)NC(=O)/C=C/c1ccccc1Cl ZINC000217901087 EI In-Stock Unstable UL26 32 43 Cc1ccccc1OC[C@H](C)NC(=O)/C=C/c1ccccc1Cl ZINC000217901087 EI In-Stock Unstable U53 0 43 Cc1ccccc1OC[C@H](C)NC(=O)/C=C/c1ccccc1Cl ZINC000217901087 EI In-Stock Unstable SCAF_EBVB9 26 43 O=C(O)[C@H]1CC[C@@](O)(c2ccccc2)C1 ZINC000217901108 BD In-Stock Unstable OPRL1 18 43 Cc1cc([C@H](C)C(=O)O)c(C)cc1Br ZINC000217901141 CG For-Sale Unstable PTGS1 20 41 Cc1cccc(/C=C/NC(=O)Nc2cccnc2)c1 ZINC000217901181 CG For-Sale Unstable KCNK3 49 40 COc1ccc(CSc2ncn[nH]2)cc1/C=C\C(=O)O ZINC000217901183 CE For-Sale Unstable PTGER2 28 42 COc1ccc(CSc2ncn[nH]2)cc1/C=C\C(=O)O ZINC000217901183 CE For-Sale Unstable PTGER4 17 42 COc1ccc(S(=O)(=O)N(Cc2cc(C3CC3)n(C)n2)C2CCCC2)cc1 ZINC000217901184 GG In-Stock Unstable AVPR1B 35 55 Cc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217901213 EI In-Stock Unstable SDH1 0 42 Cc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217901213 EI In-Stock Unstable KCNQ2 52 45 Cc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217901213 EI In-Stock Unstable CDC25B 0 43 Cc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217901213 EI In-Stock Unstable UL26 24 41 Cc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217901213 EI In-Stock Unstable U53 0 41 O=C(O)/C=C\c1ccccc1CSc1nnnn1C1CC1 ZINC000217901251 DE For-Sale Unstable PTGER2 25 40 Cc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217901296 EI In-Stock Unstable SDH1 0 42 Cc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217901296 EI In-Stock Unstable KCNQ2 52 45 Cc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217901296 EI In-Stock Unstable CDC25B 0 43 Cc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217901296 EI In-Stock Unstable UL26 24 41 Cc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217901296 EI In-Stock Unstable U53 0 41 Cn1nc(CN(C2CCCC2)S(=O)(=O)c2cccs2)cc1C1CC1 ZINC000217901317 FG In-Stock Unstable AVPR1B 17 40 CC1CCN(c2ccc([C@@H](C)NC(=O)/C=C/c3ccccc3Cl)cc2)CC1 ZINC000217901405 GK In-Stock Unstable KCNQ2 60 56 CC1CCN(c2ccc([C@@H](C)NC(=O)/C=C/c3ccccc3Cl)cc2)CC1 ZINC000217901405 GK In-Stock Unstable UL26 18 40 CC1CCN(c2ccc([C@@H](C)NC(=O)/C=C/c3ccccc3Cl)cc2)CC1 ZINC000217901405 GK In-Stock Unstable U53 0 40 CC1CCN(c2ccc([C@@H](C)NC(=O)/C=C/c3ccccc3Cl)cc2)CC1 ZINC000217901405 GK In-Stock Unstable SCAF_EBVB9 15 40 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cc(OC)c(O)c(OC)c2)CC(=O)O4)cc1O ZINC000217901423 KI In-Stock Unstable AKR1B1 24 58 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cc(OC)c(O)c(OC)c2)CC(=O)O4)cc1O ZINC000217901423 KI In-Stock Unstable CYP1B1 74 42 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cc(OC)c(O)c(OC)c2)CC(=O)O4)cc1O ZINC000217901423 KI In-Stock Unstable CYP1A1 55 50 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cc(OC)c(O)c(OC)c2)CC(=O)O4)cc1O ZINC000217901423 KI In-Stock Unstable CYP1A2 44 43 CC1CCN(c2ccc([C@H](C)NC(=O)/C=C/c3ccccc3Cl)cc2)CC1 ZINC000217901468 GK In-Stock Unstable KCNQ2 60 56 CC1CCN(c2ccc([C@H](C)NC(=O)/C=C/c3ccccc3Cl)cc2)CC1 ZINC000217901468 GK In-Stock Unstable UL26 18 40 CC1CCN(c2ccc([C@H](C)NC(=O)/C=C/c3ccccc3Cl)cc2)CC1 ZINC000217901468 GK In-Stock Unstable U53 0 40 CC1CCN(c2ccc([C@H](C)NC(=O)/C=C/c3ccccc3Cl)cc2)CC1 ZINC000217901468 GK In-Stock Unstable SCAF_EBVB9 15 40 COc1ccc(/C=C\C(=O)O)cc1CSCc1ccco1 ZINC000217901478 DH For-Sale Unstable PTGER2 18 40 COc1ccc(/C=C\C(=O)O)cc1CSCc1ccco1 ZINC000217901478 DH For-Sale Unstable AKR1C3 38 41 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cc(OC)c(O)c(OC)c2)CC(=O)O4)cc1O ZINC000217901495 KI In-Stock Unstable AKR1B1 24 58 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cc(OC)c(O)c(OC)c2)CC(=O)O4)cc1O ZINC000217901495 KI In-Stock Unstable CYP1B1 74 42 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cc(OC)c(O)c(OC)c2)CC(=O)O4)cc1O ZINC000217901495 KI In-Stock Unstable CYP1A1 55 50 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cc(OC)c(O)c(OC)c2)CC(=O)O4)cc1O ZINC000217901495 KI In-Stock Unstable CYP1A2 44 43 COC(=O)CCSCc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217901545 DF For-Sale Unstable LTB4R 35 42 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)/C=C/c3ccccc3Cl)cc2)C1 ZINC000217901563 GK In-Stock Unstable KCNQ2 59 56 C[C@H](NC(=O)/C=C/c1ccccc1Cl)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217901645 GK In-Stock Unstable KCNQ2 59 56 COC(=O)CCSCc1ccc(/C=C\C(=O)O)cc1F ZINC000217901664 CF For-Sale Unstable AKR1C3 32 41 Cc1ccc2c(c1)[C@@H](NC(=O)/C=C/c1ccccc1Cl)CC(C)(C)O2 ZINC000217901749 FK In-Stock Unstable KCNQ2 22 44 O=C(CCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCc1ccccn1 ZINC000217901782 HF In-Stock Unstable SCN9A 0 46 Cc1cc([C@@H](C)C(=O)O)cc(C)c1Br ZINC000217901788 CG For-Sale Unstable PTGS1 26 45 Cc1cc([C@@H](C)C(=O)O)cc(C)c1Br ZINC000217901788 CG For-Sale Unstable PTGS2 15 42 Cc1ccc2c(c1)[C@H](NC(=O)/C=C/c1ccccc1Cl)CC(C)(C)O2 ZINC000217901829 FK In-Stock Unstable KCNQ2 22 44 O=C(CCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCc1ccccn1 ZINC000217901849 HF In-Stock Unstable SCN9A 0 46 Cc1cc([C@H](C)C(=O)O)cc(C)c1Br ZINC000217901865 CG For-Sale Unstable PTGS1 26 45 Cc1cc([C@H](C)C(=O)O)cc(C)c1Br ZINC000217901865 CG For-Sale Unstable PTGS2 15 42 CC(=O)Nc1cccc(NC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217901914 DH For-Sale Unstable IDO1 18 44 CC(=O)Nc1cccc(NC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217901914 DH For-Sale Unstable KCNK3 98 47 CC(=O)Nc1cccc(NC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217901914 DH For-Sale Unstable KCNK9 63 47 Cc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)/C=C/c1ccccc1Cl ZINC000217901924 FK In-Stock Unstable KCNQ2 21 42 COc1ccc(/C=C\C(=O)O)cc1CSC1CCCCC1 ZINC000217901934 DI For-Sale Unstable QRFPR 60 52 Cc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)/C=C/c1ccccc1Cl ZINC000217902001 FK In-Stock Unstable KCNQ2 21 42 C[C@@H]1CN([C@H]2CCCc3cc(O)ccc32)C[C@@H]1C ZINC000217902041 BG For-Sale Unstable DRD2 16 41 C[C@@H]1CN([C@H]2CCCc3cc(O)ccc32)C[C@@H]1C ZINC000217902041 BG For-Sale Unstable OPRK1 16 40 C[C@@H]1CN([C@H]2CCCc3cc(O)ccc32)C[C@@H]1C ZINC000217902041 BG For-Sale Unstable DRD5 26 48 C[C@@H]1CN([C@H]2CCCc3cc(O)ccc32)C[C@@H]1C ZINC000217902041 BG For-Sale Unstable HSD17B1 65 39 COc1ccc2c(c1)[C@@H](NC(=O)/C=C/c1ccccc1Cl)CC(C)(C)O2 ZINC000217902127 FJ In-Stock Unstable KCNQ2 21 42 COc1ccc2c(c1)[C@H](NC(=O)/C=C/c1ccccc1Cl)CC(C)(C)O2 ZINC000217902182 FJ In-Stock Unstable KCNQ2 21 42 C[C@@H]1CN([C@H]2CCc3c(O)cccc32)C[C@@H]1C ZINC000217902213 BF For-Sale Unstable DRD1 23 40 C[C@@H]1CN([C@H]2CCc3c(O)cccc32)C[C@@H]1C ZINC000217902213 BF For-Sale Unstable DRD5 26 40 O=C(Cc1csc2nc(-c3ccccc3)cn12)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217902271 IG In-Stock Unstable CHRNA4 26 43 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)/C=C/c1ccccc1Cl ZINC000217902278 FJ In-Stock Unstable KCNQ2 20 41 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)/C=C/c1ccccc1Cl ZINC000217902278 FJ In-Stock Unstable CYSP_PLAFA 38 40 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)/C=C/c1ccccc1Cl ZINC000217902346 FJ In-Stock Unstable KCNQ2 20 41 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)/C=C/c1ccccc1Cl ZINC000217902346 FJ In-Stock Unstable CYSP_PLAFA 38 40 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](CC(C)C)C(=O)NCCCN(C)C)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217902378 KH In-Stock Unstable TUBA1A 18 65 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](CC(C)C)C(=O)NCCCN(C)C)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217902378 KH In-Stock Unstable TPPP 0 62 Cn1nc(Br)nc1CCCC(=O)O ZINC000217902423 BC For-Sale Unstable CSNK2A2 25 40 CC[C@@H](NC(=O)/C=C/c1ccccc1Cl)c1ccc(C)c(C)c1 ZINC000217902463 EK In-Stock Unstable KCNQ2 53 50 CC[C@@H](NC(=O)/C=C/c1ccccc1Cl)c1ccc(C)c(C)c1 ZINC000217902463 EK In-Stock Unstable UL26 21 41 CC[C@@H](NC(=O)/C=C/c1ccccc1Cl)c1ccc(C)c(C)c1 ZINC000217902463 EK In-Stock Unstable U53 0 41 CC[C@@H](NC(=O)/C=C/c1ccccc1Cl)c1ccc(C)c(C)c1 ZINC000217902463 EK In-Stock Unstable SCAF_EBVB9 20 41 CC[C@H](NC(=O)/C=C/c1ccccc1Cl)c1ccc(C)c(C)c1 ZINC000217902522 EK In-Stock Unstable KCNQ2 53 50 CC[C@H](NC(=O)/C=C/c1ccccc1Cl)c1ccc(C)c(C)c1 ZINC000217902522 EK In-Stock Unstable UL26 21 41 CC[C@H](NC(=O)/C=C/c1ccccc1Cl)c1ccc(C)c(C)c1 ZINC000217902522 EK In-Stock Unstable U53 0 41 CC[C@H](NC(=O)/C=C/c1ccccc1Cl)c1ccc(C)c(C)c1 ZINC000217902522 EK In-Stock Unstable SCAF_EBVB9 20 41 CC1CCC(OCc2ccccc2/C=C\C(=O)O)CC1 ZINC000217902527 CH For-Sale Unstable PTGER2 49 46 CC1CCC(OCc2ccccc2/C=C\C(=O)O)CC1 ZINC000217902527 CH For-Sale Unstable PTGER4 0 46 CC1CCC(OCc2ccccc2/C=C\C(=O)O)CC1 ZINC000217902527 CH For-Sale Unstable PTGER3 18 46 CC1CCC(OCc2ccccc2/C=C\C(=O)O)CC1 ZINC000217902527 CH For-Sale Unstable PTGDR 0 44 CC[C@@H](NC(=O)/C=C/c1ccccc1Cl)c1ccc(C)cc1C ZINC000217902620 EK In-Stock Unstable KCNQ2 40 44 CC[C@@H](NC(=O)/C=C/c1ccccc1Cl)c1ccc(C)cc1C ZINC000217902620 EK In-Stock Unstable UL26 28 43 CC[C@@H](NC(=O)/C=C/c1ccccc1Cl)c1ccc(C)cc1C ZINC000217902620 EK In-Stock Unstable U53 0 43 CC[C@@H](NC(=O)/C=C/c1ccccc1Cl)c1ccc(C)cc1C ZINC000217902620 EK In-Stock Unstable SCAF_EBVB9 25 43 C[C@H](OCc1cccc(/C=C\C(=O)O)c1)c1ccccc1 ZINC000217902621 CI For-Sale Unstable PTGER2 41 47 C[C@H](OCc1cccc(/C=C\C(=O)O)c1)c1ccccc1 ZINC000217902621 CI For-Sale Unstable 17HSDCL 0 43 C[C@H](OCc1cccc(/C=C\C(=O)O)c1)c1ccccc1 ZINC000217902621 CI For-Sale Unstable AKR1C3 35 47 CC[C@H](NC(=O)/C=C/c1ccccc1Cl)c1ccc(C)cc1C ZINC000217902689 EK In-Stock Unstable KCNQ2 40 44 CC[C@H](NC(=O)/C=C/c1ccccc1Cl)c1ccc(C)cc1C ZINC000217902689 EK In-Stock Unstable UL26 28 43 CC[C@H](NC(=O)/C=C/c1ccccc1Cl)c1ccc(C)cc1C ZINC000217902689 EK In-Stock Unstable U53 0 43 CC[C@H](NC(=O)/C=C/c1ccccc1Cl)c1ccc(C)cc1C ZINC000217902689 EK In-Stock Unstable SCAF_EBVB9 25 43 C[C@@H](OCc1cccc(/C=C\C(=O)O)c1)c1ccccc1 ZINC000217902704 CI For-Sale Unstable PTGER2 41 47 C[C@@H](OCc1cccc(/C=C\C(=O)O)c1)c1ccccc1 ZINC000217902704 CI For-Sale Unstable 17HSDCL 0 43 C[C@@H](OCc1cccc(/C=C\C(=O)O)c1)c1ccccc1 ZINC000217902704 CI For-Sale Unstable AKR1C3 35 47 C[C@@H]1CN([C@H](C)Cc2ccc(O)cc2)C[C@@H]1C ZINC000217902749 BF For-Sale Unstable OPRM1 15 40 CCCCCOCCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217902771 CG For-Sale Unstable THRA 48 40 CCCCCOCCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217902771 CG For-Sale Unstable THRB 28 40 CCCCCOCCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217902771 CG For-Sale Unstable KCNQ1 0 42 CCCCCOCCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217902771 CG For-Sale Unstable LTB4R 30 40 CCCCCOCCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217902771 CG For-Sale Unstable PLA2G4B 111 48 CCCCCOCCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217902771 CG For-Sale Unstable FAAH 26 45 CCCCCOCCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217902771 CG For-Sale Unstable AKR1C3 27 45 CC[C@@H](NC(=O)/C=C/c1ccccc1Cl)c1ccc(OC)c(OC)c1 ZINC000217902787 FJ In-Stock Unstable KCNQ2 53 48 CC[C@@H](NC(=O)/C=C/c1ccccc1Cl)c1ccc(OC)c(OC)c1 ZINC000217902787 FJ In-Stock Unstable CYSP_PLAFA 45 39 O=C(O)/C=C\c1cc(F)ccc1COCc1cccs1 ZINC000217902860 CH For-Sale Unstable PTGER2 39 40 O=C(O)/C=C\c1cc(F)ccc1COCc1cccs1 ZINC000217902860 CH For-Sale Unstable PTGER4 0 40 O=C(O)/C=C\c1cc(F)ccc1COCc1cccs1 ZINC000217902860 CH For-Sale Unstable PTGER3 16 40 O=C(O)/C=C\c1cc(F)ccc1COCc1cccs1 ZINC000217902860 CH For-Sale Unstable HCAR2 0 40 CC[C@H](NC(=O)/C=C/c1ccccc1Cl)c1ccc(OC)c(OC)c1 ZINC000217902861 FJ In-Stock Unstable KCNQ2 53 48 CC[C@H](NC(=O)/C=C/c1ccccc1Cl)c1ccc(OC)c(OC)c1 ZINC000217902861 FJ In-Stock Unstable CYSP_PLAFA 45 39 O=C(O)/C=C\c1cc(COCc2cccs2)ccc1F ZINC000217902952 CH For-Sale Unstable PTGER2 36 44 O=C(O)/C=C\c1cc(COCc2cccs2)ccc1F ZINC000217902952 CH For-Sale Unstable PTGER4 0 44 O=C(O)/C=C\c1cc(COCc2cccs2)ccc1F ZINC000217902952 CH For-Sale Unstable PTGER3 17 44 O=C(O)/C=C\c1cc(COCc2cccs2)ccc1F ZINC000217902952 CH For-Sale Unstable HCAR2 0 40 Cc1ccc(CCC(=O)O)c(C)c1Br ZINC000217902955 CG For-Sale Unstable FFAR1 43 40 CC[C@@H](NC(=O)/C=C/c1ccccc1Cl)c1ccc(S(C)(=O)=O)cc1 ZINC000217902980 GI In-Stock Unstable KCNQ2 41 47 CC[C@@H](NC(=O)/C=C/c1ccccc1Cl)c1ccc(S(C)(=O)=O)cc1 ZINC000217902980 GI In-Stock Unstable CTSF 47 32 CC[C@H](NC(=O)/C=C/c1ccccc1Cl)c1ccc(S(C)(=O)=O)cc1 ZINC000217903056 GI In-Stock Unstable KCNQ2 41 47 CC[C@H](NC(=O)/C=C/c1ccccc1Cl)c1ccc(S(C)(=O)=O)cc1 ZINC000217903056 GI In-Stock Unstable CTSF 46 32 Cc1cccc(/C=C/NC(=O)Nc2ccccc2N2CCOCC2)c1 ZINC000217903085 EH For-Sale Unstable KCNQ2 83 45 Cc1cccc(/C=C/NC(=O)Nc2ccccc2N2CCOCC2)c1 ZINC000217903085 EH For-Sale Unstable CSF1R 0 44 Cc1n[nH]c([C@@H]2CCCN2C(=O)CN2CCOc3ccccc3C2)n1 ZINC000217903109 ED In-Stock Unstable COLA 115 43 Cc1n[nH]c([C@@H]2CCCN2C(=O)CN2CCOc3ccccc3C2)n1 ZINC000217903109 ED In-Stock Unstable CPT1A 100 43 O=C(N[C@@H]1CCC[C@@H]1CO)[C@@H]1CC(=O)N(C2CC2)C1 ZINC000217903122 CC For-Sale Unstable INHA 19 44 Cc1n[nH]c([C@H]2CCCN2C(=O)CN2CCOc3ccccc3C2)n1 ZINC000217903174 ED In-Stock Unstable COLA 115 43 Cc1n[nH]c([C@H]2CCCN2C(=O)CN2CCOc3ccccc3C2)n1 ZINC000217903174 ED In-Stock Unstable CPT1A 100 43 Cc1cccc(/C=C/NC(=O)Nc2ccc(N3CCN(C)CC3)cc2)c1 ZINC000217903185 FH For-Sale Unstable PRNP 38 45 Cc1cccc(/C=C/NC(=O)Nc2ccc(N3CCN(C)CC3)cc2)c1 ZINC000217903185 FH For-Sale Unstable FLT3 18 42 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1ccc(N(C)C)cc1 ZINC000217903193 CJ For-Sale Unstable TRPM8 16 44 Cc1cc(C)c(CCC(=O)O)c(Br)c1 ZINC000217903213 CG For-Sale Unstable THRA 15 45 Cc1cc(C)c(CCC(=O)O)c(Br)c1 ZINC000217903213 CG For-Sale Unstable FFAR1 35 40 Cc1cc(C)c(CCC(=O)O)c(Br)c1 ZINC000217903213 CG For-Sale Unstable GPR17 19 41 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1ccc(N(C)C)cc1 ZINC000217903256 CJ For-Sale Unstable TRPM8 16 44 O=C(N[C@@H]1CCC[C@H]1CO)[C@@H]1CC(=O)N(C2CC2)C1 ZINC000217903265 CC For-Sale Unstable INHA 19 44 O=C(N[C@H]1CCC[C@H]1CO)[C@@H]1CC(=O)N(C2CC2)C1 ZINC000217903319 CC On-Demand Unstable INHA 40 44 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1ccc(N(C)C)cc1 ZINC000217903320 CJ For-Sale Unstable TRPM8 16 44 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccccc3Cl)n2)c(OC)c1 ZINC000217903338 GH In-Stock Unstable CYSP_PLAFA 34 40 Cc1ccc(C)c(CCC(=O)O)c1Br ZINC000217903341 CG For-Sale Unstable FFAR1 44 39 Cc1cccc(/C=C/NC(=O)Nc2ccc(N3CCCCC3)cc2)c1 ZINC000217903345 EJ For-Sale Unstable LPL 44 35 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1ccc(N(C)C)cc1 ZINC000217903407 CJ For-Sale Unstable TRPM8 16 44 Cc1cc(C)c(CCC(=O)O)cc1Br ZINC000217903473 CG For-Sale Unstable THRA 16 40 CNC(=O)c1cccc(NC(=O)CC[C@@H]2NC(=O)c3ccccc3NC2=O)c1 ZINC000217903491 GD In-Stock Unstable KCNK3 48 32 CNC(=O)c1cccc(NC(=O)CC[C@@H]2NC(=O)c3ccccc3NC2=O)c1 ZINC000217903491 GD In-Stock Unstable PARP10 0 40 Cc1cc(CCC(=O)O)cc(C)c1Br ZINC000217903554 CG For-Sale Unstable THRA 25 47 Cc1cc(CCC(=O)O)cc(C)c1Br ZINC000217903554 CG For-Sale Unstable THRB 18 49 Cc1cc(CCC(=O)O)cc(C)c1Br ZINC000217903554 CG For-Sale Unstable FFAR1 78 44 Cc1cccc(/C=C/NC(=O)Nc2ccc(N(C)C)cc2)c1 ZINC000217903561 CH For-Sale Unstable KCNK3 41 46 O=C(N1CCOCC1)N1CCCS(=O)(=O)CC1 ZINC000217903593 CB On-Demand Unstable AKR1C3 33 42 O=C(N1CCCCC1)N1CCCS(=O)(=O)CC1 ZINC000217903680 CC On-Demand Unstable LIPE 17 41 CCC#CCN1CCN(c2ncnc3[nH]ccc23)C[C@@H](O)C1 ZINC000217903698 CC In-Stock Unstable AKT2 45 42 CCC#CCN1CCN(c2ncnc3[nH]ccc23)C[C@@H](O)C1 ZINC000217903698 CC In-Stock Unstable ROCK2 40 39 CCC#CCN1CCN(c2ncnc3[nH]ccc23)C[C@@H](O)C1 ZINC000217903698 CC In-Stock Unstable AKT1 22 40 COC(=O)[C@H](CC(C)C)NC(=O)CC[C@@H]1NC(=O)c2ccccc2NC1=O ZINC000217903704 GD In-Stock Unstable NPR 55 36 Cc1cccc(/C=C/NC(=O)Nc2cccc3ccccc23)c1 ZINC000217903770 DJ For-Sale Unstable TRPV1 45 47 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccccc2Cl)cc1 ZINC000217903854 EK In-Stock Unstable KCNQ2 41 47 COC(=O)c1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217903858 DH For-Sale Unstable ACR 43 40 COC(=O)c1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217903858 DH For-Sale Unstable KCNK3 52 36 COC(=O)c1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217903858 DH For-Sale Unstable KCNK9 41 36 N#Cc1ccc(Br)c(-n2ccnc2)c1 ZINC000217903873 BF For-Sale Mild CYP19A1 18 48 OC[C@@H](O)c1cc2n(n1)CCCN(C1CCN(c3ccccc3)CC1)C2 ZINC000217903955 FD In-Stock Unstable L3MBTL3 50 38 CC(C)c1cc(Br)cc(CC(=O)O)c1 ZINC000217903956 CG For-Sale Unstable THRA 32 42 CC(C)c1cc(Br)cc(CC(=O)O)c1 ZINC000217903956 CG For-Sale Unstable THRB 28 42 CN(CCCNC(=O)/C=C/c1ccccc1Cl)c1ccccc1 ZINC000217903966 EH In-Stock Unstable PYGL 24 43 Cc1cccc(/C=C/NC(=O)N(Cc2ccccc2)c2ccccc2)c1 ZINC000217903975 EK For-Sale Unstable NR1H4 55 48 Cc1cccc(/C=C/NC(=O)N(Cc2ccccc2)c2ccccc2)c1 ZINC000217903975 EK For-Sale Unstable PTGES 19 42 COC(=O)C[C@H](c1ccc2c(c1)OCCO2)c1c(O)cc(C)n(CCc2ccc(O)cc2)c1=O ZINC000217903989 JG In-Stock Unstable RORC 41 39 O=S(=O)(Nc1cccnc1Cl)N1CCOCC1 ZINC000217904021 CC For-Sale Unstable G2YM83_BOTF4 44 31 OC[C@H](O)c1cc2n(n1)CCCN(C1CCN(c3ccccc3)CC1)C2 ZINC000217904028 FD In-Stock Unstable L3MBTL3 50 38 COc1ccc(CSCc2ccco2)cc1/C=C\C(=O)O ZINC000217904037 DH For-Sale Unstable PTGER3 17 43 COc1ccc(CSCc2ccco2)cc1/C=C\C(=O)O ZINC000217904037 DH For-Sale Unstable LTB4R 39 46 O=C(/C=C/c1ccccc1Cl)NCCCN1CCCc2ccccc21 ZINC000217904054 FI In-Stock Unstable DRD3 35 55 COC(=O)C[C@@H](c1ccc2c(c1)OCCO2)c1c(O)cc(C)n(CCc2ccc(O)cc2)c1=O ZINC000217904059 JG In-Stock Unstable RORC 41 39 Cc1cccc(/C=C/NC(=O)Nc2ccc3ccccc3c2)c1 ZINC000217904073 DJ For-Sale Unstable CA1 15 42 Cc1cccc(/C=C/NC(=O)Nc2ccc3ccccc3c2)c1 ZINC000217904073 DJ For-Sale Unstable MMP1 0 44 Cc1cccc(/C=C/NC(=O)Nc2ccc3ccccc3c2)c1 ZINC000217904073 DJ For-Sale Unstable TRPM8 0 40 Cc1cccc(/C=C/NC(=O)Nc2ccc3ccccc3c2)c1 ZINC000217904073 DJ For-Sale Unstable IMDH_CRYPV 35 44 Cc1cccc(/C=C/NC(=O)Nc2ccc3ccccc3c2)c1 ZINC000217904073 DJ For-Sale Unstable KCNK3 56 37 Cc1cccc(/C=C/NC(=O)Nc2ccc3ccccc3c2)c1 ZINC000217904073 DJ For-Sale Unstable KCNK9 42 37 CC(C)(C)c1ccc(Br)cc1C(=O)O ZINC000217904074 CG For-Sale Unstable PRS 65 39 CC(C)(C)c1ccc(Br)cc1C(=O)O ZINC000217904074 CG For-Sale Unstable AKR1C2 21 41 CC(C)(C)c1ccc(Br)cc1C(=O)O ZINC000217904074 CG For-Sale Unstable AKR1C1 23 41 O=S(=O)(c1ccccc1)N(CCF)CCc1ccccc1 ZINC000217904088 DF For-Sale Unstable BMP1 17 51 O=S(=O)(c1ccccc1)N(CCF)CCc1ccccc1 ZINC000217904088 DF For-Sale Unstable RORC 19 50 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)cc1OCC(N)=O ZINC000217904163 KF In-Stock Unstable ALOX5 0 42 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)cc1OCC(N)=O ZINC000217904163 KF In-Stock Unstable AKR1B1 0 42 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)cc1OCC(N)=O ZINC000217904163 KF In-Stock Unstable CYP1B1 47 39 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)cc1OCC(N)=O ZINC000217904163 KF In-Stock Unstable CYP1A1 47 39 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)cc1OCC(N)=O ZINC000217904163 KF In-Stock Unstable ABCB1A 22 41 CC1(C)C(=O)NC(=O)CN1C(=O)/C=C\c1ccc(O)cc1 ZINC000217904222 CC For-Sale Unstable F3 19 41 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)cc1OCC(N)=O ZINC000217904247 KF In-Stock Unstable ALOX5 0 42 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)cc1OCC(N)=O ZINC000217904247 KF In-Stock Unstable AKR1B1 0 42 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)cc1OCC(N)=O ZINC000217904247 KF In-Stock Unstable CYP1B1 47 39 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)cc1OCC(N)=O ZINC000217904247 KF In-Stock Unstable CYP1A1 47 39 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)c(O)c(-c5ccc(O)c(O)c5)oc4c32)cc1OCC(N)=O ZINC000217904247 KF In-Stock Unstable ABCB1A 22 41 COc1cccc(C(=O)N2CCC(C(=O)N3CCc4n[nH]cc4C3)CC2)c1 ZINC000217904261 FD In-Stock Unstable DRD4 46 36 COc1cccc(C(=O)N2CCC(C(=O)N3CCc4n[nH]cc4C3)CC2)c1 ZINC000217904261 FD In-Stock Unstable SLC18A3 23 41 COc1cccc(C(=O)N2CCC(C(=O)N3CCc4n[nH]cc4C3)CC2)c1 ZINC000217904261 FD In-Stock Unstable ROCK2 40 34 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccc(Cl)cc2Cl)c1 ZINC000217904287 FK In-Stock Unstable KCNQ2 40 36 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccc(Cl)cc2Cl)c1 ZINC000217904287 FK In-Stock Unstable BOTA 29 49 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccc(Cl)cc2Cl)c1 ZINC000217904287 FK In-Stock Unstable PDS 65 38 O=C(/C=C/c1ccc(F)c(Cl)c1)N[C@H]1CCC[C@H]1CO ZINC000217904311 CF On-Demand Unstable HD1B 0 41 COc1cc([C@@H](C)N2C[C@@H](C)[C@@H](C)C2)ccc1O ZINC000217904360 BG For-Sale Unstable PNLIP 0 53 COc1cc([C@@H](C)N2C[C@@H](C)[C@@H](C)C2)ccc1O ZINC000217904360 BG For-Sale Unstable SHBG 17 40 COc1cc([C@@H](C)N2C[C@@H](C)[C@@H](C)C2)ccc1O ZINC000217904360 BG For-Sale Unstable N1L 0 54 COc1cc([C@@H](C)N2C[C@@H](C)[C@@H](C)C2)ccc1O ZINC000217904360 BG For-Sale Unstable CAN2 0 43 COc1cc([C@@H](C)N2C[C@@H](C)[C@@H](C)C2)ccc1O ZINC000217904360 BG For-Sale Unstable SLC22A3 0 46 COC(=O)CSCCOc1cccc(/C=C\C(=O)O)c1 ZINC000217904380 CE For-Sale Unstable AKR1C3 31 40 COc1ccc(CNC(=O)/C=C/c2ccc(Cl)cc2Cl)c(OC)c1OC ZINC000217904400 GI In-Stock Unstable P2RX7 26 40 COc1ccc(CNC(=O)/C=C/c2ccc(Cl)cc2Cl)c(OC)c1OC ZINC000217904400 GI In-Stock Unstable BOTA 32 50 COc1ccc(CNC(=O)/C=C/c2ccc(Cl)cc2Cl)c(OC)c1OC ZINC000217904400 GI In-Stock Unstable CYSP_PLAFA 61 56 COc1cc2c(c(OC)c1OC)-c1ccc(NCCCCCC(=O)NCc3cccn3C)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217904437 KI In-Stock Unstable TUBA1A 17 61 COc1cc2c(c(OC)c1OC)-c1ccc(NCCCCCC(=O)NCc3cccn3C)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217904437 KI In-Stock Unstable TPPP 0 58 COc1ccc(CSC2CCCCC2)cc1/C=C\C(=O)O ZINC000217904458 DI For-Sale Unstable PTGER2 24 41 COc1ccc(CSC2CCCCC2)cc1/C=C\C(=O)O ZINC000217904458 DI For-Sale Unstable QRFPR 49 44 CCOc1ccc(CNC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1OCC ZINC000217904509 GK In-Stock Unstable BOTA 30 50 CCC[C@@H](O)CNCCCC(C)C ZINC000217904536 AE On-Demand Unstable SPPS 41 36 O=C1C[C@@H](c2ccsc2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217904543 HI In-Stock Unstable AKR1B1 0 43 O=C1C[C@@H](c2ccsc2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217904543 HI In-Stock Unstable CYP1B1 20 41 O=C1C[C@@H](c2ccsc2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217904543 HI In-Stock Unstable CYP1A1 20 41 O=C(NCc1ccccc1)N1CCCS(=O)(=O)CC1 ZINC000217904552 CD On-Demand Unstable DPP7 33 40 O=C(NCc1ccccc1)N1CCCS(=O)(=O)CC1 ZINC000217904552 CD On-Demand Unstable TPSAB1 16 46 O=C(NCc1ccccc1)N1CCCS(=O)(=O)CC1 ZINC000217904552 CD On-Demand Unstable NPSR1 27 43 O=C(NCc1ccccc1)N1CCCS(=O)(=O)CC1 ZINC000217904552 CD On-Demand Unstable NAMPT 28 44 O=C(NCc1ccccc1)N1CCCS(=O)(=O)CC1 ZINC000217904552 CD On-Demand Unstable TMPRSS11D 40 31 O=C1C[C@H](c2ccsc2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217904607 HI In-Stock Unstable AKR1B1 0 43 O=C1C[C@H](c2ccsc2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217904607 HI In-Stock Unstable CYP1B1 20 41 O=C1C[C@H](c2ccsc2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217904607 HI In-Stock Unstable CYP1A1 20 41 CCC[C@H](O)CNCCCC(C)C ZINC000217904608 AE On-Demand Unstable SPPS 41 36 COc1cc(CNC(=O)/C=C/c2ccc(Cl)cc2Cl)ccc1OC(C)C ZINC000217904612 GK In-Stock Unstable BOTA 30 46 COc1cc(CNC(=O)/C=C/c2ccc(Cl)cc2Cl)ccc1OC(C)C ZINC000217904612 GK In-Stock Unstable CYSP_PLAFA 51 43 CC1(C)C(=O)NC(=O)CN1c1ccc(/C=C\C(=O)O)cc1 ZINC000217904662 CD For-Sale Unstable LGB 0 40 Cn1nc(CN(Cc2ccco2)C(=O)Cn2c(=O)oc3ccccc32)c2c1CCC2 ZINC000217904726 HF In-Stock Unstable TSPO 20 43 O=C(/C=C/c1ccc(Cl)cc1Cl)NCCCc1ccccc1Cl ZINC000217904727 FK In-Stock Unstable PYGL 0 45 O=C(/C=C/c1ccc(Cl)cc1Cl)NCCCc1ccccc1Cl ZINC000217904727 FK In-Stock Unstable HPSE 17 40 O=C(/C=C/c1ccc(Cl)cc1Cl)NCCCc1ccccc1Cl ZINC000217904727 FK In-Stock Unstable HDAC9 28 50 O=C(/C=C/c1ccc(Cl)cc1Cl)NCCCc1ccccc1Cl ZINC000217904727 FK In-Stock Unstable HDAC7 33 50 O=C(/C=C/c1ccc(Cl)cc1Cl)NCCCc1ccccc1Cl ZINC000217904727 FK In-Stock Unstable BOTA 32 54 Cc1nc(C2CCN(C(=O)CN3CCOc4ccccc4C3)CC2)no1 ZINC000217904801 FD In-Stock Unstable ETHR 50 38 O=C(/C=C/c1ccc(Cl)cc1Cl)NCCCc1ccc(Cl)cc1 ZINC000217904841 FK In-Stock Unstable PYGL 25 48 O=C(/C=C/c1ccc(Cl)cc1Cl)NCCCc1ccc(Cl)cc1 ZINC000217904841 FK In-Stock Unstable HPSE 21 43 O=C(/C=C/c1ccc(Cl)cc1Cl)NCCCc1ccc(Cl)cc1 ZINC000217904841 FK In-Stock Unstable HDAC9 17 53 O=C(/C=C/c1ccc(Cl)cc1Cl)NCCCc1ccc(Cl)cc1 ZINC000217904841 FK In-Stock Unstable HDAC7 25 53 O=C(/C=C/c1ccc(Cl)cc1Cl)NCCCc1ccc(Cl)cc1 ZINC000217904841 FK In-Stock Unstable BOTA 34 58 O=C(O)C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1cccs1 ZINC000217904897 CC For-Sale Unstable CTSC 21 40 CCC[C@@H](O)CNCCOc1ccccc1 ZINC000217904908 BD For-Sale Unstable ADRB2 22 43 CCC[C@@H](O)CNCCOc1ccccc1 ZINC000217904908 BD For-Sale Unstable DRD4 22 49 CCC[C@@H](O)CNCCOc1ccccc1 ZINC000217904908 BD For-Sale Unstable ADRA1D 0 43 CCC[C@@H](O)CNCCOc1ccccc1 ZINC000217904908 BD For-Sale Unstable ADRB3 59 58 O=C(/C=C/c1ccc(Cl)cc1Cl)NCCCc1ccc(F)cc1 ZINC000217904941 FJ In-Stock Unstable HPSE 27 43 O=C(/C=C/c1ccc(Cl)cc1Cl)NCCCc1ccc(F)cc1 ZINC000217904941 FJ In-Stock Unstable HDAC9 17 55 O=C(/C=C/c1ccc(Cl)cc1Cl)NCCCc1ccc(F)cc1 ZINC000217904941 FJ In-Stock Unstable HDAC7 25 55 O=C(/C=C/c1ccc(Cl)cc1Cl)NCCCc1ccc(F)cc1 ZINC000217904941 FJ In-Stock Unstable ALPL 51 37 O=C(/C=C/c1ccc(Cl)cc1Cl)NCCCc1ccc(F)cc1 ZINC000217904941 FJ In-Stock Unstable BOTA 35 53 O=C(O)C[C@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1cccs1 ZINC000217904969 CC For-Sale Unstable CTSC 21 40 CCC[C@H](O)CNCCOc1ccccc1 ZINC000217905007 BD For-Sale Unstable ADRB2 22 43 CCC[C@H](O)CNCCOc1ccccc1 ZINC000217905007 BD For-Sale Unstable DRD4 22 49 CCC[C@H](O)CNCCOc1ccccc1 ZINC000217905007 BD For-Sale Unstable ADRA1D 0 43 CCC[C@H](O)CNCCOc1ccccc1 ZINC000217905007 BD For-Sale Unstable ADRB3 59 58 Cc1cccc(/C=C/NC(=O)N2C[C@@]3(C)C[C@H]2CC(C)(C)C3)c1 ZINC000217905009 DJ For-Sale Unstable AVPR2 17 49 Cc1cccc(/C=C/NC(=O)N2C[C@@]3(C)C[C@H]2CC(C)(C)C3)c1 ZINC000217905009 DJ For-Sale Unstable AVPR1A 37 45 O=C(CCc1cccc(Br)c1)N[C@H]1CCC[C@H]1CO ZINC000217905018 EF On-Demand Unstable LUXR 38 56 COc1ccccc1CCCNC(=O)/C=C/c1ccc(Cl)cc1Cl ZINC000217905033 FJ In-Stock Unstable DRD3 23 51 COc1ccccc1CCCNC(=O)/C=C/c1ccc(Cl)cc1Cl ZINC000217905033 FJ In-Stock Unstable MTNR1B 34 41 COc1ccccc1CCCNC(=O)/C=C/c1ccc(Cl)cc1Cl ZINC000217905033 FJ In-Stock Unstable HDAC9 20 45 COc1ccccc1CCCNC(=O)/C=C/c1ccc(Cl)cc1Cl ZINC000217905033 FJ In-Stock Unstable HDAC7 31 45 COc1ccccc1CCCNC(=O)/C=C/c1ccc(Cl)cc1Cl ZINC000217905033 FJ In-Stock Unstable BOTA 32 48 COc1ccccc1CCCNC(=O)/C=C/c1ccc(Cl)cc1Cl ZINC000217905033 FJ In-Stock Unstable CYSP_PLAFA 54 42 CSCC[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(Cc2ccc3c(c2)OCO3)C1=O ZINC000217905037 HC In-Stock Unstable NOS2 60 34 CSCC[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(Cc2ccc3c(c2)OCO3)C1=O ZINC000217905037 HC In-Stock Unstable SSTR3 88 32 COc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)c1 ZINC000217905146 FJ In-Stock Unstable DRD4 45 37 COc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)c1 ZINC000217905146 FJ In-Stock Unstable DRD3 17 42 COc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)c1 ZINC000217905146 FJ In-Stock Unstable PTAFR 21 44 COc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)c1 ZINC000217905146 FJ In-Stock Unstable MTNR1A 40 57 COc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)c1 ZINC000217905146 FJ In-Stock Unstable MTNR1B 39 57 COc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)c1 ZINC000217905146 FJ In-Stock Unstable HDAC7 22 44 COc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)c1 ZINC000217905146 FJ In-Stock Unstable BOTA 29 47 COc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)c1 ZINC000217905146 FJ In-Stock Unstable CRTM 60 45 COc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)c1 ZINC000217905146 FJ In-Stock Unstable CYSP_PLAFA 53 44 CCC[C@@H](O)CNCCCCO ZINC000217905149 AC For-Sale Unstable SPPS 45 38 Cc1cccc(/C=C/NC(=O)Nc2cccc(N(C)C)c2)c1 ZINC000217905196 CH For-Sale Unstable CCKBR 16 41 Cc1cccc(/C=C/NC(=O)Nc2cccc(N(C)C)c2)c1 ZINC000217905196 CH For-Sale Unstable KCNK3 59 45 Cc1cccc(/C=C/NC(=O)Nc2cccc(N(C)C)c2)c1 ZINC000217905196 CH For-Sale Unstable KCNK9 43 39 CCC[C@H](O)CNCCCCO ZINC000217905206 AC For-Sale Unstable SPPS 45 38 COc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1 ZINC000217905239 FJ In-Stock Unstable DRD3 15 41 COc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1 ZINC000217905239 FJ In-Stock Unstable PTAFR 18 41 COc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1 ZINC000217905239 FJ In-Stock Unstable HPSE 22 41 COc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1 ZINC000217905239 FJ In-Stock Unstable HDAC9 21 47 COc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1 ZINC000217905239 FJ In-Stock Unstable HDAC7 31 47 COc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1 ZINC000217905239 FJ In-Stock Unstable U38 0 40 COc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1 ZINC000217905239 FJ In-Stock Unstable BOTA 32 50 COc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1 ZINC000217905239 FJ In-Stock Unstable CYSP_PLAFA 43 46 C[C@@H]1CN([C@H](C)c2cccc(O)c2)C[C@@H]1C ZINC000217905242 BG For-Sale Unstable OPRM1 16 52 Cc1cccc(/C=C/NC(=O)Nc2nc3c(s2)CN(C)CC3)c1 ZINC000217905277 EG For-Sale Unstable F10 26 43 CC1CCC(OCc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217905293 CH For-Sale Unstable PTGER2 23 40 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1 ZINC000217905321 GJ In-Stock Unstable PTGS2 0 45 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1 ZINC000217905321 GJ In-Stock Unstable KCNQ2 47 35 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1 ZINC000217905321 GJ In-Stock Unstable CDC25B 0 46 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1 ZINC000217905321 GJ In-Stock Unstable BOTA 33 51 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1 ZINC000217905321 GJ In-Stock Unstable CYSP_PLAFA 49 47 COc1cc2c(c(OC)c1OC)-c1ccc(NCCCCCC(=O)N3CCN(c4nc5ccccc5n4C)CC3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217905330 KK In-Stock Unstable TUBA1A 15 55 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Oc1cccc(F)c1[N+](=O)[O-] ZINC000217905354 CJ For-Sale Unstable SERPINE1 41 40 CCN(CCNC(=O)c1ccc(Cl)c(N)c1)C1CC1 ZINC000217905378 CE For-Sale Unstable HTR4 22 42 Cc1cccc(/C=C/NC(=O)Nc2ccc3nc[nH]c3c2)c1 ZINC000217905390 CH For-Sale Unstable KCNK3 43 35 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1 ZINC000217905405 GJ In-Stock Unstable PTGS2 0 45 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1 ZINC000217905405 GJ In-Stock Unstable KCNQ2 47 35 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1 ZINC000217905405 GJ In-Stock Unstable CDC25B 0 46 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1 ZINC000217905405 GJ In-Stock Unstable BOTA 33 51 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1 ZINC000217905405 GJ In-Stock Unstable CYSP_PLAFA 49 47 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Oc1cccc(F)c1[N+](=O)[O-] ZINC000217905453 CJ For-Sale Unstable SERPINE1 41 40 CC1CCC(OCc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217905456 CH For-Sale Unstable PTGER2 25 43 CC1CCC(OCc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217905456 CH For-Sale Unstable GRM2 19 40 CC1CCC(OCc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217905456 CH For-Sale Unstable AKR1C3 31 41 COc1ccc([C@H](C)N2C[C@@H]3CCCN3C[C@@H]2C)c(O)c1 ZINC000217905466 CF For-Sale Unstable CHRM2 18 45 O=C(/C=C/c1ccc(Cl)cc1Cl)Nc1ccccc1C(=O)c1ccccc1 ZINC000217905496 GK In-Stock Anodyne LTB4R 0 44 O=C(/C=C/c1ccc(Cl)cc1Cl)Nc1ccccc1C(=O)c1ccccc1 ZINC000217905496 GK In-Stock Anodyne MMP2 17 48 O=C(/C=C/c1ccc(Cl)cc1Cl)Nc1ccccc1C(=O)c1ccccc1 ZINC000217905496 GK In-Stock Anodyne MMP9 15 48 O=C(/C=C/c1ccc(Cl)cc1Cl)Nc1ccccc1C(=O)c1ccccc1 ZINC000217905496 GK In-Stock Anodyne HPSE 23 42 O=C(/C=C/c1ccc(Cl)cc1Cl)Nc1ccccc1C(=O)c1ccccc1 ZINC000217905496 GK In-Stock Anodyne MMP1 0 48 O=C(/C=C/c1ccc(Cl)cc1Cl)Nc1ccccc1C(=O)c1ccccc1 ZINC000217905496 GK In-Stock Anodyne BOTA 31 56 CCCCCCOCCOc1cccc(/C=C\C(=O)O)c1 ZINC000217905542 CH For-Sale Unstable THRA 61 45 CCCCCCOCCOc1cccc(/C=C\C(=O)O)c1 ZINC000217905542 CH For-Sale Unstable PTAFR 27 40 CCCCCCOCCOc1cccc(/C=C\C(=O)O)c1 ZINC000217905542 CH For-Sale Unstable THRB 40 45 CCCCCCOCCOc1cccc(/C=C\C(=O)O)c1 ZINC000217905542 CH For-Sale Unstable LTB4R 42 48 CCCCCCOCCOc1cccc(/C=C\C(=O)O)c1 ZINC000217905542 CH For-Sale Unstable MTNR1A 21 41 CCCCCCOCCOc1cccc(/C=C\C(=O)O)c1 ZINC000217905542 CH For-Sale Unstable PLA2G4B 101 49 CCCCCCOCCOc1cccc(/C=C\C(=O)O)c1 ZINC000217905542 CH For-Sale Unstable FAAH 25 43 CCCCCCOCCOc1cccc(/C=C\C(=O)O)c1 ZINC000217905542 CH For-Sale Unstable AKR1C3 27 44 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Oc1cccc(F)c1[N+](=O)[O-] ZINC000217905544 CJ For-Sale Unstable SERPINE1 41 40 Cc1cccc(/C=C/NC(=O)Nc2ccccc2C(N)=O)c1 ZINC000217905590 CF For-Sale Unstable MMP1 0 43 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)c1 ZINC000217905602 GK In-Stock Unstable PTAFR 15 42 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)c1 ZINC000217905602 GK In-Stock Unstable HDAC9 20 43 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)c1 ZINC000217905602 GK In-Stock Unstable HDAC7 30 43 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)c1 ZINC000217905602 GK In-Stock Unstable BOTA 27 45 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)c1 ZINC000217905602 GK In-Stock Unstable CRTM 54 46 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Oc1cccc(F)c1[N+](=O)[O-] ZINC000217905614 CJ For-Sale Unstable SERPINE1 41 40 COc1ccc2[nH]c3c(c2c1)CN(C(=O)CC[C@@H]1NC(=O)c2ccccc2NC1=O)CC3 ZINC000217905625 IF In-Stock Unstable PDGFRA 0 44 CCCCCCOCCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217905630 CH For-Sale Unstable THRA 61 42 CCCCCCOCCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217905630 CH For-Sale Unstable RARB 22 54 CCCCCCOCCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217905630 CH For-Sale Unstable THRB 40 42 CCCCCCOCCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217905630 CH For-Sale Unstable CYSLTR2 22 41 CCCCCCOCCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217905630 CH For-Sale Unstable LTB4R 34 41 CCCCCCOCCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217905630 CH For-Sale Unstable PLA2G4A 29 48 CCCCCCOCCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217905630 CH For-Sale Unstable PLA2G4B 116 50 CCCCCCOCCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217905630 CH For-Sale Unstable FAAH 27 46 CCCCCCOCCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217905630 CH For-Sale Unstable AKR1C3 0 44 CC(C)Oc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1 ZINC000217905688 GK In-Stock Unstable PYGL 0 40 CC(C)Oc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1 ZINC000217905688 GK In-Stock Unstable HDAC7 22 44 CC(C)Oc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1 ZINC000217905688 GK In-Stock Unstable BOTA 30 47 O=C(c1cccs1)N1CCC(N2CCn3nc([C@@H](O)CO)cc3C2)CC1 ZINC000217905707 GD In-Stock Unstable L3MBTL3 58 36 CCCCCOCc1cc(/C=C\C(=O)O)ccc1OC ZINC000217905725 CG For-Sale Unstable PTGER2 0 42 CCCCCOCc1cc(/C=C\C(=O)O)ccc1OC ZINC000217905725 CG For-Sale Unstable LTB4R 40 43 CCCCCOCc1cc(/C=C\C(=O)O)ccc1OC ZINC000217905725 CG For-Sale Unstable PLA2G4B 79 41 CCCCCOCc1cc(/C=C\C(=O)O)ccc1OC ZINC000217905725 CG For-Sale Unstable TUBB1 42 37 CCCCCOCc1cc(/C=C\C(=O)O)ccc1OC ZINC000217905725 CG For-Sale Unstable AKR1C3 30 46 CN(CCNC(=O)/C=C/c1ccc(Cl)cc1Cl)c1ccccc1 ZINC000217905781 EI In-Stock Unstable HDAC7 30 44 CN(CCNC(=O)/C=C/c1ccc(Cl)cc1Cl)c1ccccc1 ZINC000217905781 EI In-Stock Unstable BOTA 31 53 O=C(c1cccs1)N1CCC(N2CCn3nc([C@H](O)CO)cc3C2)CC1 ZINC000217905787 GD In-Stock Unstable L3MBTL3 58 36 CCCCC/C=C/C/C=C\C/C=C\CCCCC(=O)NCCO ZINC000217905789 DJ For-Sale Unstable CNR1 61 97 CCCCC/C=C/C/C=C\C/C=C\CCCCC(=O)NCCO ZINC000217905789 DJ For-Sale Unstable PPARA 28 88 CCCCC/C=C/C/C=C\C/C=C\CCCCC(=O)NCCO ZINC000217905789 DJ For-Sale Unstable CNR2 23 94 CCCCC/C=C/C/C=C\C/C=C\CCCCC(=O)NCCO ZINC000217905789 DJ For-Sale Unstable FABP4 21 58 CCCCC/C=C/C/C=C\C/C=C\CCCCC(=O)NCCO ZINC000217905789 DJ For-Sale Unstable TRPV1 22 97 CCCCC/C=C/C/C=C\C/C=C\CCCCC(=O)NCCO ZINC000217905789 DJ For-Sale Unstable PLA2G4A 29 50 CCCCC/C=C/C/C=C\C/C=C\CCCCC(=O)NCCO ZINC000217905789 DJ For-Sale Unstable LPAR1 31 59 CCCCC/C=C/C/C=C\C/C=C\CCCCC(=O)NCCO ZINC000217905789 DJ For-Sale Unstable SELP 15 57 CCCCC/C=C/C/C=C\C/C=C\CCCCC(=O)NCCO ZINC000217905789 DJ For-Sale Unstable FAAH 53 97 CCCCC/C=C/C/C=C\C/C=C\CCCCC(=O)NCCO ZINC000217905789 DJ For-Sale Unstable EPHX2 34 63 CCCCC/C=C/C/C=C\C/C=C\CCCCC(=O)NCCO ZINC000217905789 DJ For-Sale Unstable FABP3 46 58 CCCCC/C=C/C/C=C\C/C=C\CCCCC(=O)NCCO ZINC000217905789 DJ For-Sale Unstable FABP5 15 50 CCCCC/C=C/C/C=C\C/C=C\CCCCC(=O)NCCO ZINC000217905789 DJ For-Sale Unstable MGLL 16 50 CCCCC/C=C/C/C=C\C/C=C\CCCCC(=O)NCCO ZINC000217905789 DJ For-Sale Unstable FFAR1 26 58 CCCCC/C=C/C/C=C\C/C=C\CCCCC(=O)NCCO ZINC000217905789 DJ For-Sale Unstable FABP1 16 50 CCCCC/C=C/C/C=C\C/C=C\CCCCC(=O)NCCO ZINC000217905789 DJ For-Sale Unstable OXER1 23 48 CCCCC/C=C/C/C=C\C/C=C\CCCCC(=O)NCCO ZINC000217905789 DJ For-Sale Unstable CQSS 49 30 CCCCCOCc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217905801 CG For-Sale Unstable PTGER2 39 46 CCCCCOCc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217905801 CG For-Sale Unstable INHA 50 33 CCCCCOCc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217905801 CG For-Sale Unstable PTGER4 23 46 CCCCCOCc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217905801 CG For-Sale Unstable PTGER3 18 46 CCCCCOCc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217905801 CG For-Sale Unstable LTB4R 39 42 CCCCCOCc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217905801 CG For-Sale Unstable PLA2G4B 63 39 CCCCCOCc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217905801 CG For-Sale Unstable AKR1C3 26 40 CCCCCOCc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217905801 CG For-Sale Unstable AKR1B10 35 43 Cc1cccc(/C=C/NC(=O)Nc2cccc(Br)c2)c1 ZINC000217905804 EJ For-Sale Unstable EGFR 42 41 Cc1cccc(/C=C/NC(=O)Nc2cccc(Br)c2)c1 ZINC000217905804 EJ For-Sale Unstable CCKAR 15 43 Cc1cccc(/C=C/NC(=O)Nc2cccc(Br)c2)c1 ZINC000217905804 EJ For-Sale Unstable KCNK3 57 40 Cc1cccc(/C=C/NC(=O)Nc2cccc(Br)c2)c1 ZINC000217905804 EJ For-Sale Unstable KCNK9 44 40 O=C(O)/C=C\c1ccccc1COCCc1cccs1 ZINC000217905868 CH For-Sale Unstable PTGER2 64 48 O=C(O)/C=C\c1ccccc1COCCc1cccs1 ZINC000217905868 CH For-Sale Unstable PTGER4 31 43 O=C(O)/C=C\c1ccccc1COCCc1cccs1 ZINC000217905868 CH For-Sale Unstable PTGER3 26 48 O=C(O)/C=C\c1ccccc1COCCc1cccs1 ZINC000217905868 CH For-Sale Unstable PTGDR 0 43 O=C(O)/C=C\c1ccccc1COCCc1cccs1 ZINC000217905868 CH For-Sale Unstable HCAR2 0 41 O=C(/C=C/c1ccc(Cl)cc1Cl)Nc1ccc(OC2CCCC2)cc1 ZINC000217905891 GK In-Stock Unstable HPSE 18 41 O=C(/C=C/c1ccc(Cl)cc1Cl)Nc1ccc(OC2CCCC2)cc1 ZINC000217905891 GK In-Stock Unstable EPHX2 24 43 O=C(/C=C/c1ccc(Cl)cc1Cl)Nc1ccc(OC2CCCC2)cc1 ZINC000217905891 GK In-Stock Unstable BOTA 29 51 C[C@@H]1C(=O)NC(=O)CN1Cc1ccccc1/C=C\C(=O)O ZINC000217905895 CC For-Sale Unstable PTGER2 34 42 C[C@@H]1C(=O)NC(=O)CN1Cc1ccccc1/C=C\C(=O)O ZINC000217905895 CC For-Sale Unstable PTGER4 0 42 O=C(N[C@H](CO)Cc1ccccc1)[C@H](c1ccccc1)N1Cc2ccccc2C1=O ZINC000217905944 HG In-Stock Unstable MME 69 38 O=C(N[C@H](CO)Cc1ccccc1)[C@H](c1ccccc1)N1Cc2ccccc2C1=O ZINC000217905944 HG In-Stock Unstable SOAT1 26 40 CCCCC/C=C/C/C=C/C/C=C\CCCCC(=O)NCCO ZINC000217905962 DJ For-Sale Unstable CNR1 61 97 CCCCC/C=C/C/C=C/C/C=C\CCCCC(=O)NCCO ZINC000217905962 DJ For-Sale Unstable PPARA 28 88 CCCCC/C=C/C/C=C/C/C=C\CCCCC(=O)NCCO ZINC000217905962 DJ For-Sale Unstable CNR2 23 94 CCCCC/C=C/C/C=C/C/C=C\CCCCC(=O)NCCO ZINC000217905962 DJ For-Sale Unstable FABP4 21 58 CCCCC/C=C/C/C=C/C/C=C\CCCCC(=O)NCCO ZINC000217905962 DJ For-Sale Unstable TRPV1 22 97 CCCCC/C=C/C/C=C/C/C=C\CCCCC(=O)NCCO ZINC000217905962 DJ For-Sale Unstable PLA2G4A 29 50 CCCCC/C=C/C/C=C/C/C=C\CCCCC(=O)NCCO ZINC000217905962 DJ For-Sale Unstable LPAR1 31 59 CCCCC/C=C/C/C=C/C/C=C\CCCCC(=O)NCCO ZINC000217905962 DJ For-Sale Unstable SELP 15 57 CCCCC/C=C/C/C=C/C/C=C\CCCCC(=O)NCCO ZINC000217905962 DJ For-Sale Unstable FAAH 53 97 CCCCC/C=C/C/C=C/C/C=C\CCCCC(=O)NCCO ZINC000217905962 DJ For-Sale Unstable EPHX2 34 63 CCCCC/C=C/C/C=C/C/C=C\CCCCC(=O)NCCO ZINC000217905962 DJ For-Sale Unstable FABP3 46 58 CCCCC/C=C/C/C=C/C/C=C\CCCCC(=O)NCCO ZINC000217905962 DJ For-Sale Unstable FABP5 15 50 CCCCC/C=C/C/C=C/C/C=C\CCCCC(=O)NCCO ZINC000217905962 DJ For-Sale Unstable MGLL 16 50 CCCCC/C=C/C/C=C/C/C=C\CCCCC(=O)NCCO ZINC000217905962 DJ For-Sale Unstable FFAR1 26 58 CCCCC/C=C/C/C=C/C/C=C\CCCCC(=O)NCCO ZINC000217905962 DJ For-Sale Unstable FABP1 16 50 CCCCC/C=C/C/C=C/C/C=C\CCCCC(=O)NCCO ZINC000217905962 DJ For-Sale Unstable OXER1 23 48 CCCCC/C=C/C/C=C/C/C=C\CCCCC(=O)NCCO ZINC000217905962 DJ For-Sale Unstable CQSS 49 30 O=C(O)/C=C\c1ccc(COCCc2cccs2)cc1 ZINC000217905969 CH For-Sale Unstable PTGER2 36 46 O=C(O)/C=C\c1ccc(COCCc2cccs2)cc1 ZINC000217905969 CH For-Sale Unstable PTGER4 0 46 O=C(O)/C=C\c1ccc(COCCc2cccs2)cc1 ZINC000217905969 CH For-Sale Unstable PTGER3 16 46 O=C(O)/C=C\c1ccc(COCCc2cccs2)cc1 ZINC000217905969 CH For-Sale Unstable HCAR2 0 42 O=C(O)/C=C\c1ccc(COCCc2cccs2)cc1 ZINC000217905969 CH For-Sale Unstable AKR1C3 31 43 C[C@H]1C(=O)NC(=O)CN1Cc1ccccc1/C=C\C(=O)O ZINC000217906005 CC For-Sale Unstable PTGER2 34 42 C[C@H]1C(=O)NC(=O)CN1Cc1ccccc1/C=C\C(=O)O ZINC000217906005 CC For-Sale Unstable PTGER4 0 42 CC1(C)C[C@@H](NC(=O)/C=C/c2ccc(Cl)cc2Cl)c2ccccc2O1 ZINC000217906016 GK In-Stock Unstable BOTA 28 47 CCOc1ccc(CCNC(=O)N/C=C/c2cccc(C)c2)cc1OCC ZINC000217906040 FI For-Sale Unstable AKR1C3 25 40 O=C(O)/C=C\c1ccc(COCCc2cccs2)c(F)c1 ZINC000217906056 DH For-Sale Unstable AKR1C3 32 45 CC1(C)C(=O)NC(=O)CN1C(=O)/C=C\c1cccc(Cl)c1 ZINC000217906078 DD For-Sale Unstable TUBA4A 0 42 CC1(C)C[C@H](NC(=O)/C=C/c2ccc(Cl)cc2Cl)c2ccccc2O1 ZINC000217906096 GK In-Stock Unstable BOTA 28 47 Cc1ccc(SCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217906132 CI For-Sale Unstable PTGER2 50 49 Cc1ccc(SCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217906132 CI For-Sale Unstable PTGER4 0 49 Cc1ccc(SCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217906132 CI For-Sale Unstable PTGER3 19 57 Cc1ccc(SCc2ccccc2/C=C\C(=O)O)cc1 ZINC000217906132 CI For-Sale Unstable PTGDR 0 57 Cc1cccc(/C=C/NC(=O)Nc2ccc(C(C)(C)C)cc2)c1 ZINC000217906152 DK For-Sale Unstable TRPV1 21 45 Cc1cccc(/C=C/NC(=O)Nc2ccc(C(C)(C)C)cc2)c1 ZINC000217906152 DK For-Sale Unstable MMP1 0 42 Cc1cccc(/C=C/NC(=O)Nc2ccc(C(C)(C)C)cc2)c1 ZINC000217906152 DK For-Sale Unstable IMDH_CRYPV 54 36 Cc1cccc(/C=C/NC(=O)Nc2ccc(C(C)(C)C)cc2)c1 ZINC000217906152 DK For-Sale Unstable KCNK3 42 46 CSCC[C@@H](O)C(=O)N(C)Cc1ccc(-n2cccn2)cc1 ZINC000217906163 DD In-Stock Unstable AMP1_PLAFQ 50 34 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1 ZINC000217906202 GK In-Stock Unstable PYGL 0 40 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1 ZINC000217906202 GK In-Stock Unstable HDAC9 15 45 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1 ZINC000217906202 GK In-Stock Unstable HDAC7 22 45 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1 ZINC000217906202 GK In-Stock Unstable BOTA 31 48 Cc1ccc(SCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217906220 CI For-Sale Unstable AKR1C3 24 41 Cc1ccc(SCc2ccc(/C=C\C(=O)O)cc2)cc1 ZINC000217906220 CI For-Sale Unstable GPR183 0 42 CSCC[C@H](O)C(=O)N(C)Cc1ccc(-n2cccn2)cc1 ZINC000217906237 DD In-Stock Unstable AMP1_PLAFQ 50 34 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccc(Cl)cc1Cl ZINC000217906314 GK In-Stock Unstable DRD3 15 42 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccc(Cl)cc1Cl ZINC000217906314 GK In-Stock Unstable MTNR1A 25 43 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccc(Cl)cc1Cl ZINC000217906314 GK In-Stock Unstable MTNR1B 26 43 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccc(Cl)cc1Cl ZINC000217906314 GK In-Stock Unstable HDAC7 21 42 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccc(Cl)cc1Cl ZINC000217906314 GK In-Stock Unstable BOTA 28 45 CSCC[C@H](NC(=O)COc1ccc2c(C)cc(=O)oc2c1)c1nc2ccccc2n1C ZINC000217906411 JH In-Stock Unstable MAOA 59 49 CSCC[C@H](NC(=O)COc1ccc2c(C)cc(=O)oc2c1)c1nc2ccccc2n1C ZINC000217906411 JH In-Stock Unstable MAOB 30 49 CSCC[C@H](NC(=O)COc1ccc2c(C)cc(=O)oc2c1)c1nc2ccccc2n1C ZINC000217906411 JH In-Stock Unstable BCHE 18 45 COc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1OC ZINC000217906415 GJ In-Stock Unstable DRD3 16 44 COc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1OC ZINC000217906415 GJ In-Stock Unstable PYGL 0 40 COc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1OC ZINC000217906415 GJ In-Stock Unstable HDAC7 22 45 COc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1OC ZINC000217906415 GJ In-Stock Unstable PTGDR 29 41 COc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1OC ZINC000217906415 GJ In-Stock Unstable TTR 0 45 COc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1OC ZINC000217906415 GJ In-Stock Unstable PTGDR2 18 40 COc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1OC ZINC000217906415 GJ In-Stock Unstable BOTA 31 48 COc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1OC ZINC000217906415 GJ In-Stock Unstable CAN2 0 46 COc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1OC ZINC000217906415 GJ In-Stock Unstable CYSP_PLAFA 48 44 O=C(NCCc1noc(C(F)(F)F)n1)c1ccccc1N1CCCC1 ZINC000217906420 FF In-Stock Unstable KCNQ2 67 35 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccc(Cl)cc1Cl ZINC000217906508 FJ In-Stock Unstable SDH1 0 40 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccc(Cl)cc1Cl ZINC000217906508 FJ In-Stock Unstable KCNQ2 50 38 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccc(Cl)cc1Cl ZINC000217906508 FJ In-Stock Unstable BOTA 30 49 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccc(Cl)cc1Cl ZINC000217906508 FJ In-Stock Unstable CYSP_PLAFA 43 38 Cc1ccccc1OC[C@H](C)NC(=O)/C=C/c1ccc(Cl)cc1Cl ZINC000217906593 FJ In-Stock Unstable SDH1 0 40 Cc1ccccc1OC[C@H](C)NC(=O)/C=C/c1ccc(Cl)cc1Cl ZINC000217906593 FJ In-Stock Unstable KCNQ2 50 38 Cc1ccccc1OC[C@H](C)NC(=O)/C=C/c1ccc(Cl)cc1Cl ZINC000217906593 FJ In-Stock Unstable BOTA 30 49 Cc1ccccc1OC[C@H](C)NC(=O)/C=C/c1ccc(Cl)cc1Cl ZINC000217906593 FJ In-Stock Unstable CYSP_PLAFA 43 38 Cc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1 ZINC000217906707 FJ In-Stock Unstable KCNQ2 47 35 Cc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1 ZINC000217906707 FJ In-Stock Unstable BOTA 32 51 Cc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1 ZINC000217906792 FJ In-Stock Unstable KCNQ2 47 35 Cc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1 ZINC000217906792 FJ In-Stock Unstable BOTA 32 51 CSC[C@@](C)(O)CNC1=NS(=O)(=O)c2ccccc21 ZINC000217906875 DC On-Demand Unstable KCNA3 44 37 CC1CCN(c2ccc([C@@H](C)NC(=O)/C=C/c3ccc(Cl)cc3Cl)cc2)CC1 ZINC000217906881 HK In-Stock Unstable KCNQ2 56 45 CC1CCN(c2ccc([C@@H](C)NC(=O)/C=C/c3ccc(Cl)cc3Cl)cc2)CC1 ZINC000217906881 HK In-Stock Unstable BOTA 30 49 Cc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217906893 FE For-Sale Unstable CA2 108 58 Cc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217906893 FE For-Sale Unstable CA1 92 58 Cc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217906893 FE For-Sale Unstable CA7 54 51 Cc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217906893 FE For-Sale Unstable CA5B 48 48 Cc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217906893 FE For-Sale Unstable CA4 74 53 Cc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217906893 FE For-Sale Unstable CA5A 49 48 Cc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217906893 FE For-Sale Unstable CA14 45 51 Cc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217906893 FE For-Sale Unstable MMP2 15 40 Cc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217906893 FE For-Sale Unstable FBP1 15 42 Cc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217906893 FE For-Sale Unstable CA12 67 58 Cc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217906893 FE For-Sale Unstable CA9 78 58 Cc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217906893 FE For-Sale Unstable CYNT 27 46 Cc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217906893 FE For-Sale Unstable NCE103 36 49 Cc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217906893 FE For-Sale Unstable MTCA1 44 38 Cc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217906893 FE For-Sale Unstable P96878_MYCTU 58 44 Cc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217906893 FE For-Sale Unstable A6YCJ1_9METZ 24 48 CSC[C@](C)(O)CNC1=NS(=O)(=O)c2ccccc21 ZINC000217906939 DC On-Demand Unstable KCNA3 44 37 CC(=O)Nc1cccc(C(=O)N2CCCO[C@@H](CN3CCCC3)C2)c1 ZINC000217906951 ED In-Stock Unstable CCR3 24 45 CC(=O)Nc1cccc(C(=O)N2CCCO[C@@H](CN3CCCC3)C2)c1 ZINC000217906951 ED In-Stock Unstable EPHX2 22 42 CC(=O)Nc1cccc(C(=O)N2CCCO[C@@H](CN3CCCC3)C2)c1 ZINC000217906951 ED In-Stock Unstable RHOA 0 41 CC1CCN(c2ccc([C@H](C)NC(=O)/C=C/c3ccc(Cl)cc3Cl)cc2)CC1 ZINC000217906956 HK In-Stock Unstable KCNQ2 56 45 CC1CCN(c2ccc([C@H](C)NC(=O)/C=C/c3ccc(Cl)cc3Cl)cc2)CC1 ZINC000217906956 HK In-Stock Unstable BOTA 30 49 Cc1cccc(/C=C/NC(=O)Nc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1 ZINC000217906986 GK For-Sale Unstable KCNK3 40 35 CC(=O)Nc1cccc(C(=O)N2CCCO[C@H](CN3CCCC3)C2)c1 ZINC000217907011 ED In-Stock Unstable CCR3 24 45 CC(=O)Nc1cccc(C(=O)N2CCCO[C@H](CN3CCCC3)C2)c1 ZINC000217907011 ED In-Stock Unstable EPHX2 22 42 CC(=O)Nc1cccc(C(=O)N2CCCO[C@H](CN3CCCC3)C2)c1 ZINC000217907011 ED In-Stock Unstable RHOA 0 41 CC(C)Cc1cc(Cl)ccc1C(=O)O ZINC000217907069 BG For-Sale Unstable PTGER1 35 46 CC(C)Cc1cc(Cl)ccc1C(=O)O ZINC000217907069 BG For-Sale Unstable ACPS 0 45 CC(C)Cc1cc(Cl)ccc1C(=O)O ZINC000217907069 BG For-Sale Unstable AKR1C2 42 44 CC(C)Cc1cc(Cl)ccc1C(=O)O ZINC000217907069 BG For-Sale Unstable AKR1C1 45 44 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)/C=C/c3ccc(Cl)cc3Cl)cc2)C1 ZINC000217907080 HK In-Stock Unstable KCNQ2 54 45 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)/C=C/c3ccc(Cl)cc3Cl)cc2)C1 ZINC000217907080 HK In-Stock Unstable BOTA 28 46 CS(=O)(=O)Nc1ccc(C(=O)N[C@@H]2CCC[C@@H]2CO)cc1 ZINC000217907157 DC On-Demand Unstable PRKCA 22 41 CS(=O)(=O)Nc1ccc(C(=O)N[C@@H]2CCC[C@@H]2CO)cc1 ZINC000217907157 DC On-Demand Unstable PANK3 0 49 C[C@H](NC(=O)/C=C/c1ccc(Cl)cc1Cl)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217907172 HK In-Stock Unstable KCNQ2 54 45 C[C@H](NC(=O)/C=C/c1ccc(Cl)cc1Cl)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217907172 HK In-Stock Unstable BOTA 28 46 N#C/C(C=O)=C(\N)Nc1ccccc1 ZINC000217907198 AC For-Sale Unstable DHODH 39 40 C[C@@H]1CN(c2ccc(CBr)cn2)C[C@@H](C)N1C ZINC000217907263 CF For-Sale Unstable SORD 50 37 N#C/C(C=O)=C(/N)Nc1ccccc1 ZINC000217907276 AC For-Sale Unstable DHODH 39 40 Cc1ccc2c(c1)[C@@H](NC(=O)/C=C/c1ccc(Cl)cc1Cl)CC(C)(C)O2 ZINC000217907299 GK In-Stock Unstable BOTA 26 45 CSC[C@@](C)(O)CNC(=O)Nc1cccc2ccccc12 ZINC000217907304 DG On-Demand Unstable TRPV1 28 42 Cc1cccc(/C=C/NC(=O)Nc2ccc(C(N)=O)cc2)c1 ZINC000217907306 CF For-Sale Unstable MMP1 0 44 Cc1cccc(/C=C/NC(=O)Nc2ccc(C(N)=O)cc2)c1 ZINC000217907306 CF For-Sale Unstable KCNK3 59 40 Cc1cccc(/C=C/NC(=O)Nc2ccc(C(N)=O)cc2)c1 ZINC000217907306 CF For-Sale Unstable KCNK9 44 40 CC(C)COC(=O)N[C@@H](CCC(=O)OC(C)(C)C)C(=O)O ZINC000217907309 DD For-Sale Unstable FPR1 38 40 CC(C)COC(=O)N[C@@H](CCC(=O)OC(C)(C)C)C(=O)O ZINC000217907309 DD For-Sale Unstable PSMB5 23 44 CC(C)COC(=O)N[C@@H](CCC(=O)OC(C)(C)C)C(=O)O ZINC000217907309 DD For-Sale Unstable NOD1 67 35 N#Cc1cccc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217907339 CG For-Sale Unstable PTGER2 22 44 N#Cc1cccc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217907339 CG For-Sale Unstable PTGER4 27 52 N#Cc1cccc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217907339 CG For-Sale Unstable PTGER3 29 53 N#Cc1cccc(OCc2ccccc2/C=C\C(=O)O)c1 ZINC000217907339 CG For-Sale Unstable FFAR1 23 43 C[C@H]1CN(c2ccc(CBr)cn2)C[C@@H](C)N1C ZINC000217907343 CF For-Sale Unstable SORD 50 37 COC(=O)[C@@H](C)CN1CCC[C@@H](C)C1 ZINC000217907349 AD In-Stock Unstable BIRC2 40 34 COc1cc([C@H](C)N2C[C@@H]3CCCN3C[C@@H]2C)ccc1O ZINC000217907372 CF For-Sale Unstable CHRM2 28 45 CSC[C@](C)(O)CNC(=O)Nc1cccc2ccccc12 ZINC000217907376 DG On-Demand Unstable TRPV1 28 42 Cc1ccc2c(c1)[C@H](NC(=O)/C=C/c1ccc(Cl)cc1Cl)CC(C)(C)O2 ZINC000217907385 GK In-Stock Unstable BOTA 26 45 Cc1cccc(/C=C/NC(=O)Nc2ccc(F)c(Cl)c2)c1 ZINC000217907400 DJ For-Sale Unstable KIT 18 42 Cc1cccc(/C=C/NC(=O)Nc2ccc(F)c(Cl)c2)c1 ZINC000217907400 DJ For-Sale Unstable KDR 15 42 Cc1cccc(/C=C/NC(=O)Nc2ccc(F)c(Cl)c2)c1 ZINC000217907400 DJ For-Sale Unstable MMP1 0 42 Cc1cccc(/C=C/NC(=O)Nc2ccc(F)c(Cl)c2)c1 ZINC000217907400 DJ For-Sale Unstable IDO1 15 42 Cc1cccc(/C=C/NC(=O)Nc2ccc(F)c(Cl)c2)c1 ZINC000217907400 DJ For-Sale Unstable P95276_MYCTO 0 41 Cc1cccc(/C=C/NC(=O)Nc2ccc(F)c(Cl)c2)c1 ZINC000217907400 DJ For-Sale Unstable KCNK3 48 40 C[C@H]1CN(c2ccc(CBr)cn2)C[C@H](C)N1C ZINC000217907417 CF For-Sale Unstable SORD 50 37 COc1ccc(C(=O)N[C@@H]2CCC[C@@H]2CO)cn1 ZINC000217907451 CC On-Demand Unstable SSTR3 24 40 COc1ccc(C(=O)N[C@@H]2CCC[C@@H]2CO)cn1 ZINC000217907451 CC On-Demand Unstable HPGDS 31 40 CCC[C@@H](O)CNCCCF ZINC000217907456 AD For-Sale Unstable SPPS 41 36 CCN(CCNC(=O)c1cc(Cl)ccc1N)C1CC1 ZINC000217907459 CE For-Sale Unstable HTR4 15 42 Cc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)/C=C/c1ccc(Cl)cc1Cl ZINC000217907487 GK In-Stock Unstable BOTA 27 45 CCN(CC)c1ccc(NC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217907502 DJ For-Sale Unstable GHSR 0 40 COc1ccc(C(=O)N[C@H]2CCC[C@@H]2CO)cn1 ZINC000217907518 CC For-Sale Unstable SSTR3 25 40 COc1ccc(C(=O)N[C@H]2CCC[C@@H]2CO)cn1 ZINC000217907518 CC For-Sale Unstable HPGDS 33 40 CCC[C@H](O)CNCCCF ZINC000217907534 AD For-Sale Unstable SPPS 41 36 COc1ccc(NC(=O)CN2C(=O)c3ccccc3N3C(=O)c4c(ccc(OC)c4OC)[C@H]23)cc1 ZINC000217907544 JG In-Stock Unstable TSHR 66 37 Cc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)/C=C/c1ccc(Cl)cc1Cl ZINC000217907569 GK In-Stock Unstable BOTA 27 45 COc1ccc(C(=O)N[C@@H]2CCC[C@H]2CO)cn1 ZINC000217907609 CC For-Sale Unstable SSTR3 25 40 COc1ccc(C(=O)N[C@@H]2CCC[C@H]2CO)cn1 ZINC000217907609 CC For-Sale Unstable HPGDS 33 40 COC(=O)c1cc(C(=O)O)oc1Br ZINC000217907619 BD In-Stock Unstable GPR35 60 35 COc1ccc(NC(=O)CN2C(=O)c3ccccc3N3C(=O)c4c(ccc(OC)c4OC)[C@@H]23)cc1 ZINC000217907626 JG In-Stock Unstable TSHR 66 37 COc1ccc(C(=O)N[C@H]2CCC[C@H]2CO)cn1 ZINC000217907690 CC For-Sale Unstable SSTR3 25 40 COc1ccc(C(=O)N[C@H]2CCC[C@H]2CO)cn1 ZINC000217907690 CC For-Sale Unstable HPGDS 33 40 COc1ccc2c(c1)[C@@H](NC(=O)/C=C/c1ccc(Cl)cc1Cl)CC(C)(C)O2 ZINC000217907694 HK In-Stock Unstable BOTA 26 42 COc1ccc2c(c1)[C@@H](NC(=O)/C=C/c1ccc(Cl)cc1Cl)CC(C)(C)O2 ZINC000217907694 HK In-Stock Unstable CYSP_PLAFA 40 44 CSC[C@@](C)(O)CNC(=O)Nc1ccc(F)cc1F ZINC000217907709 CE On-Demand Unstable P2RY1 18 40 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)Nc1nccs1 ZINC000217907754 HH In-Stock Unstable MAP 0 40 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)Nc1nccs1 ZINC000217907754 HH In-Stock Unstable MAP1 68 39 COc1ccccc1N1CCN(C(=O)N/C=C/c2cccc(C)c2)CC1 ZINC000217907763 FH For-Sale Unstable DRD1 36 44 COc1ccccc1N1CCN(C(=O)N/C=C/c2cccc(C)c2)CC1 ZINC000217907763 FH For-Sale Unstable DRD3 24 40 COc1ccccc1N1CCN(C(=O)N/C=C/c2cccc(C)c2)CC1 ZINC000217907763 FH For-Sale Unstable TACR3 0 42 COc1ccc2c(c1)[C@H](NC(=O)/C=C/c1ccc(Cl)cc1Cl)CC(C)(C)O2 ZINC000217907773 HK In-Stock Unstable BOTA 26 42 COc1ccc2c(c1)[C@H](NC(=O)/C=C/c1ccc(Cl)cc1Cl)CC(C)(C)O2 ZINC000217907773 HK In-Stock Unstable CYSP_PLAFA 40 44 O=C(O)/C=C\c1cncc(C(=O)NCC2CCCCC2)c1 ZINC000217907774 CE For-Sale Unstable CACNA1I 51 35 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)Nc1nccs1 ZINC000217907833 HH In-Stock Unstable MAP 0 40 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)Nc1nccs1 ZINC000217907833 HH In-Stock Unstable MAP1 68 39 CC[C@@H](C)N(C)CCNS(=O)(=O)c1ccnc(Cl)c1 ZINC000217907866 DD For-Sale Unstable CHUK 16 40 O=C(O)/C=C\c1cncc(C(=O)Nc2ccc(Cl)cn2)c1 ZINC000217907870 DE For-Sale Anodyne KLKB1 31 41 O=C(O)/C=C\c1cncc(C(=O)Nc2ccc(Cl)cn2)c1 ZINC000217907870 DE For-Sale Anodyne F10 48 43 O=C(O)/C=C\c1cncc(C(=O)Nc2ccc(Cl)cn2)c1 ZINC000217907870 DE For-Sale Anodyne SCN10A 49 40 O=C(O)/C=C\c1cncc(C(=O)Nc2ccc(Cl)cn2)c1 ZINC000217907870 DE For-Sale Anodyne LUCI_LUCLA 43 47 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)/C=C/c1ccc(Cl)cc1Cl ZINC000217907876 HK In-Stock Unstable BOTA 26 42 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)/C=C/c1ccc(Cl)cc1Cl ZINC000217907876 HK In-Stock Unstable CYSP_PLAFA 47 44 COc1ccccc1CN[C@@H]1C[C@@H](C)N(C)C[C@@H]1C ZINC000217907899 CF For-Sale Unstable TACR3 25 41 CC[C@H](C)N(C)CCNS(=O)(=O)c1ccnc(Cl)c1 ZINC000217907924 DD For-Sale Unstable CHUK 16 40 O=C(O)/C=C\c1cncc(C(=O)Nc2ccncc2)c1 ZINC000217907929 CD For-Sale Anodyne KCNK3 71 44 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)/C=C/c1ccc(Cl)cc1Cl ZINC000217907932 HK In-Stock Unstable BOTA 26 42 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)/C=C/c1ccc(Cl)cc1Cl ZINC000217907932 HK In-Stock Unstable CYSP_PLAFA 47 44 COc1ccccc1CN[C@H]1C[C@@H](C)N(C)C[C@@H]1C ZINC000217907977 CF For-Sale Unstable TACR3 25 41 COc1ccccc1CN[C@@H]1C[C@H](C)N(C)C[C@@H]1C ZINC000217908042 CF For-Sale Unstable TACR3 25 41 CC[C@@H](NC(=O)/C=C/c1ccc(Cl)cc1Cl)c1ccc(C)c(C)c1 ZINC000217908065 FK In-Stock Unstable KCNQ2 47 38 CC[C@@H](NC(=O)/C=C/c1ccc(Cl)cc1Cl)c1ccc(C)c(C)c1 ZINC000217908065 FK In-Stock Unstable BOTA 32 52 C#CCOc1ccc(-c2cccc(CC(=O)O)c2)cc1 ZINC000217908087 CF For-Sale Unstable THRA 23 40 C#CCOc1ccc(-c2cccc(CC(=O)O)c2)cc1 ZINC000217908087 CF For-Sale Unstable PPARD 15 44 C#CCOc1ccc(-c2cccc(CC(=O)O)c2)cc1 ZINC000217908087 CF For-Sale Unstable PLA2G4B 33 44 C#CCOc1ccc(-c2cccc(CC(=O)O)c2)cc1 ZINC000217908087 CF For-Sale Unstable FFAR1 58 49 C#CCOc1ccc(-c2cccc(CC(=O)O)c2)cc1 ZINC000217908087 CF For-Sale Unstable FFAR4 52 35 C#CCOc1ccc(-c2cccc(CC(=O)O)c2)cc1 ZINC000217908087 CF For-Sale Unstable HAO2 49 42 COc1ccc([C@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1 ZINC000217908102 KH In-Stock Unstable AKR1B1 0 44 COc1ccc([C@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1 ZINC000217908102 KH In-Stock Unstable PRKDC 20 42 COc1ccc([C@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1 ZINC000217908102 KH In-Stock Unstable RORC 0 42 CC[C@H](NC(=O)/C=C/c1ccc(Cl)cc1Cl)c1ccc(C)c(C)c1 ZINC000217908121 FK In-Stock Unstable KCNQ2 47 38 CC[C@H](NC(=O)/C=C/c1ccc(Cl)cc1Cl)c1ccc(C)c(C)c1 ZINC000217908121 FK In-Stock Unstable BOTA 32 52 Cc1cccc(/C=C/NC(=O)NC2CCCCCC2)c1 ZINC000217908136 CH For-Sale Unstable FAAH 20 52 Cc1cccc(/C=C/NC(=O)NC2CCCCCC2)c1 ZINC000217908136 CH For-Sale Unstable EPHX2 29 45 COc1ccccc1CN[C@H]1C[C@H](C)N(C)C[C@@H]1C ZINC000217908140 CF For-Sale Unstable TACR3 25 41 COc1cc(F)c(CCN)cc1Br ZINC000217908173 BE For-Sale Unstable HTR2A 16 69 COc1cc(F)c(CCN)cc1Br ZINC000217908173 BE For-Sale Unstable HTR2C 16 69 COc1ccc([C@@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1 ZINC000217908184 KH In-Stock Unstable AKR1B1 0 44 COc1ccc([C@@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1 ZINC000217908184 KH In-Stock Unstable PRKDC 20 42 COc1ccc([C@@H](CC(=O)N2CCOCC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc1 ZINC000217908184 KH In-Stock Unstable RORC 55 42 Cc1cncc(C(=O)N[C@H]2CCC[C@@H]2CO)c1 ZINC000217908225 BD For-Sale Unstable SSTR5 27 43 CC[C@@H](NC(=O)/C=C/c1ccc(Cl)cc1Cl)c1ccc(C)cc1C ZINC000217908236 FK In-Stock Unstable BOTA 32 51 COc1ccc(N[C@@H]2C[C@@H](C)N(C)C[C@@H]2C)c(OC)c1 ZINC000217908242 CF For-Sale Unstable CYP1B1 33 40 Cc1nc2ccccc2n1CCC(=O)NCc1nnnn1-c1ccccc1 ZINC000217908250 FE In-Stock Unstable HTR7 22 41 CN1CCN(C(=O)C[C@H](c2ccccc2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)CC1 ZINC000217908294 KH In-Stock Unstable ABCB1 15 48 Nc1nc(Cl)c2c(I)cn([C@H]3C[C@H](O)[C@@H](CO)O3)c2n1 ZINC000217908302 HC For-Sale Unstable TK1 39 51 Nc1nc(Cl)c2c(I)cn([C@H]3C[C@H](O)[C@@H](CO)O3)c2n1 ZINC000217908302 HC For-Sale Unstable ADK 20 40 Nc1nc(Cl)c2c(I)cn([C@H]3C[C@H](O)[C@@H](CO)O3)c2n1 ZINC000217908302 HC For-Sale Unstable POLB 42 34 COc1ccc(N[C@H]2C[C@@H](C)N(C)C[C@@H]2C)c(OC)c1 ZINC000217908318 CF For-Sale Unstable CYP1B1 33 40 CC[C@H](NC(=O)/C=C/c1ccc(Cl)cc1Cl)c1ccc(C)cc1C ZINC000217908322 FK In-Stock Unstable BOTA 32 51 Cc1cncc(C(=O)N[C@@H]2CCC[C@H]2CO)c1 ZINC000217908329 BD For-Sale Unstable SSTR5 27 43 Cc1cccc(/C=C/NC(=O)Nc2cc(Cl)cc(Cl)c2)c1 ZINC000217908335 DK For-Sale Unstable MMP1 0 43 Cc1cccc(/C=C/NC(=O)Nc2cc(Cl)cc(Cl)c2)c1 ZINC000217908335 DK For-Sale Unstable KCNK3 44 39 COc1ccc(N[C@@H]2C[C@H](C)N(C)C[C@@H]2C)c(OC)c1 ZINC000217908365 CF For-Sale Unstable CYP1B1 33 40 CN1CCN(C(=O)C[C@@H](c2ccccc2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)CC1 ZINC000217908370 KH In-Stock Unstable ABCB1 15 48 Cc1cncc(C(=O)N[C@H]2CCC[C@H]2CO)c1 ZINC000217908391 BD For-Sale Unstable SSTR5 27 43 CC[C@@H](NC(=O)/C=C/c1ccc(Cl)cc1Cl)c1ccc(OC)c(OC)c1 ZINC000217908403 GK In-Stock Unstable BOTA 33 50 CC[C@@H](NC(=O)/C=C/c1ccc(Cl)cc1Cl)c1ccc(OC)c(OC)c1 ZINC000217908403 GK In-Stock Unstable CYSP_PLAFA 55 46 CCOc1ccccc1NC(=O)N/C=C/c1cccc(C)c1 ZINC000217908428 CI For-Sale Unstable KCNK3 27 43 CCOc1ccccc1NC(=O)N/C=C/c1cccc(C)c1 ZINC000217908428 CI For-Sale Unstable KCNK9 34 43 COc1ccc(/C=C\C(=O)O)c(CSCCCO)c1 ZINC000217908432 CE For-Sale Unstable PTGER2 31 45 COc1ccc(/C=C\C(=O)O)c(CSCCCO)c1 ZINC000217908432 CE For-Sale Unstable PTGER4 15 45 COc1ccc(N[C@H]2C[C@H](C)N(C)C[C@@H]2C)c(OC)c1 ZINC000217908463 CF For-Sale Unstable CYP1B1 33 40 CC[C@H](NC(=O)/C=C/c1ccc(Cl)cc1Cl)c1ccc(OC)c(OC)c1 ZINC000217908486 GK In-Stock Unstable BOTA 33 50 CC[C@H](NC(=O)/C=C/c1ccc(Cl)cc1Cl)c1ccc(OC)c(OC)c1 ZINC000217908486 GK In-Stock Unstable CYSP_PLAFA 55 46 Cc1cccc(/C=C/NC(=O)Nc2cc(C)cc(C)c2)c1 ZINC000217908554 CI For-Sale Unstable MMP1 0 49 Cc1cccc(/C=C/NC(=O)Nc2cc(C)cc(C)c2)c1 ZINC000217908554 CI For-Sale Unstable KCNK3 49 38 CC[C@@H](NC(=O)/C=C/c1ccc(Cl)cc1Cl)c1ccc(S(C)(=O)=O)cc1 ZINC000217908589 HJ In-Stock Unstable KCNQ2 47 38 CC[C@@H](NC(=O)/C=C/c1ccc(Cl)cc1Cl)c1ccc(S(C)(=O)=O)cc1 ZINC000217908589 HJ In-Stock Unstable BOTA 30 50 CC[C@H](NC(=O)/C=C/c1ccc(Cl)cc1Cl)c1ccc(S(C)(=O)=O)cc1 ZINC000217908658 HJ In-Stock Unstable KCNQ2 47 38 CC[C@H](NC(=O)/C=C/c1ccc(Cl)cc1Cl)c1ccc(S(C)(=O)=O)cc1 ZINC000217908658 HJ In-Stock Unstable BOTA 30 50 CCC[C@@H](O)CNCC(=O)OCC ZINC000217908672 AC For-Sale Unstable CARP_RHICH 45 32 COc1ccc(OCCNC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217908693 EG For-Sale Unstable HRH2 24 41 COc1ccc(OCCNC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217908693 EG For-Sale Unstable MTNR1A 83 49 COc1ccc(OCCNC(=O)N/C=C/c2cccc(C)c2)cc1 ZINC000217908693 EG For-Sale Unstable MTNR1B 71 49 CCC[C@H](O)CNCC(=O)OCC ZINC000217908783 AC For-Sale Unstable CARP_RHICH 45 32 Cn1nc(CN(C(=O)c2ccccc2F)C2CCCC2)c2c1CCC2 ZINC000217908785 EH In-Stock Unstable ACE 40 37 Cc1cccc(-c2noc(CNC(=O)/C=C/c3ccc(Cl)cc3Cl)n2)c1 ZINC000217908794 GJ In-Stock Unstable BOTA 28 44 O=C(N[C@@H]1CCC[C@@H]1CO)c1csc2ccccc12 ZINC000217908839 CF For-Sale Unstable C5AR1 24 42 Cn1nc(CN(C(=O)c2cccc(Cl)c2)C2CCCC2)c2c1CCC2 ZINC000217908916 FI In-Stock Unstable ACE 43 39 Cn1nc(CN(C(=O)c2cccc(Cl)c2)C2CCCC2)c2c1CCC2 ZINC000217908916 FI In-Stock Unstable SLC6A9 19 43 Cc1ccc(-c2noc(CNC(=O)/C=C/c3ccc(Cl)cc3Cl)n2)cc1 ZINC000217908919 GJ In-Stock Unstable HPSE 20 41 Cc1ccc(-c2noc(CNC(=O)/C=C/c3ccc(Cl)cc3Cl)n2)cc1 ZINC000217908919 GJ In-Stock Unstable BOTA 30 46 O=C(N[C@H]1CCC[C@@H]1CO)c1csc2ccccc12 ZINC000217908945 CF For-Sale Unstable C5AR1 24 42 Cc1nn(-c2ccccn2)c(C)c1CC(=O)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217908959 GF In-Stock Unstable P2RX7 33 48 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccc(Cl)cc3Cl)n2)cc1 ZINC000217909002 HI In-Stock Unstable HPSE 23 40 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccc(Cl)cc3Cl)n2)cc1 ZINC000217909002 HI In-Stock Unstable PDK1 53 45 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccc(Cl)cc3Cl)n2)cc1 ZINC000217909002 HI In-Stock Unstable BOTA 30 44 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccc(Cl)cc3Cl)n2)cc1 ZINC000217909002 HI In-Stock Unstable CYSP_PLAFA 39 41 O=C(N[C@@H]1CCC[C@H]1CO)c1csc2ccccc12 ZINC000217909030 CF For-Sale Unstable C5AR1 24 42 CCCCCCCCCNC[C@@H](O)CCC ZINC000217909056 BG For-Sale Unstable S1PR3 18 41 CCCCCCCCCNC[C@@H](O)CCC ZINC000217909056 BG For-Sale Unstable S1PR2 44 41 CCCCCCCCCNC[C@@H](O)CCC ZINC000217909056 BG For-Sale Unstable Q8WS26_TRYCR 45 52 CCCCCCCCCNC[C@@H](O)CCC ZINC000217909056 BG For-Sale Unstable CQSS 45 38 O=C(N[C@H]1CCC[C@H]1CO)c1csc2ccccc12 ZINC000217909117 CF On-Demand Unstable C5AR1 30 42 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccc(Cl)cc3Cl)n2)c(OC)c1 ZINC000217909127 II In-Stock Unstable PDK1 33 41 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccc(Cl)cc3Cl)n2)c(OC)c1 ZINC000217909127 II In-Stock Unstable BOTA 26 40 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccc(Cl)cc3Cl)n2)c(OC)c1 ZINC000217909127 II In-Stock Unstable CYSP_PLAFA 49 46 Cc1cccc(/C=C/NC(=O)NC23CC4CC(CC(C4)C2)C3)c1 ZINC000217909129 DI For-Sale Unstable EPHX2 106 60 CCCCCCCCCNC[C@H](O)CCC ZINC000217909149 BG For-Sale Unstable S1PR3 18 41 CCCCCCCCCNC[C@H](O)CCC ZINC000217909149 BG For-Sale Unstable S1PR2 44 41 CCCCCCCCCNC[C@H](O)CCC ZINC000217909149 BG For-Sale Unstable Q8WS26_TRYCR 45 52 CCCCCCCCCNC[C@H](O)CCC ZINC000217909149 BG For-Sale Unstable CQSS 45 38 COc1ccc(/C=C\C(=O)O)cc1CSCCCO ZINC000217909177 CE For-Sale Unstable AKR1C3 38 40 CCO[C@@H]1C[C@@H](NC(=O)NC2CCCC2)C1(C)C ZINC000217909184 CE For-Sale Unstable EPHX2 21 44 O=C(/C=C/c1ccc(Cl)cc1Cl)NCc1nc(-c2ccc(Cl)cc2)no1 ZINC000217909224 HK In-Stock Unstable HPSE 23 43 O=C(/C=C/c1ccc(Cl)cc1Cl)NCc1nc(-c2ccc(Cl)cc2)no1 ZINC000217909224 HK In-Stock Unstable BOTA 31 49 CC(C)[C@@H]1CN(c2cnc3ccc(F)cc3n2)CCN1 ZINC000217909229 CE For-Sale Unstable PRKCQ 26 42 C[C@H](Oc1ccccc1)C(=O)N(Cc1nn(C)c2c1CCC2)C1CCCC1 ZINC000217909231 FH In-Stock Unstable GHSR 24 40 Cc1cccc(/C=C/NC(=O)Nc2cccc3cccnc23)c1 ZINC000217909235 DI For-Sale Unstable PFHDAC1 0 43 CCO[C@H]1C[C@@H](NC(=O)NC2CCCC2)C1(C)C ZINC000217909263 CE For-Sale Unstable EPHX2 21 44 C[C@@H](Oc1ccccc1)C(=O)N(Cc1nn(C)c2c1CCC2)C1CCCC1 ZINC000217909315 FH In-Stock Unstable GHSR 24 40 CC(C)[C@H]1CN(c2cnc3ccc(F)cc3n2)CCN1 ZINC000217909319 CE For-Sale Unstable PRKCQ 26 42 CCO[C@@H]1C[C@H](NC(=O)NC2CCCC2)C1(C)C ZINC000217909349 CE For-Sale Unstable EPHX2 21 44 O=c1cc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)oc(CN2CCN(Cc3cccc(Cl)c3)CC2)c1O ZINC000217909368 KG In-Stock Unstable CHRNA4 30 56 COc1ccc(O)c(CN2C[C@@H]3CCCCN3C[C@@H]2C)c1 ZINC000217909409 CE On-Demand Unstable SIGMAR1 0 43 O=C(O)/C=C\c1cncc(C(=O)N2CCC(O)CC2)c1 ZINC000217909411 CC For-Sale Unstable L3MBTL1 0 43 O=C(O)/C=C\c1cncc(C(=O)N2CCC(O)CC2)c1 ZINC000217909411 CC For-Sale Unstable L3MBTL3 43 34 CCO[C@H]1C[C@H](NC(=O)NC2CCCC2)C1(C)C ZINC000217909423 CE For-Sale Unstable EPHX2 21 44 CC(C)[C@@H]1CCN(c2cnc3ccccc3n2)CCN1 ZINC000217909447 CE For-Sale Unstable SORD 27 49 COc1ccc(CSCCCO)cc1/C=C\C(=O)O ZINC000217909449 CE For-Sale Unstable PTGER2 28 43 COc1ccc(CSCCCO)cc1/C=C\C(=O)O ZINC000217909449 CE For-Sale Unstable PTGER4 16 43 COc1ccc(CSCCCO)cc1/C=C\C(=O)O ZINC000217909449 CE For-Sale Unstable LTB4R 40 44 O=C(CCCCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCCc1c[nH]cn1 ZINC000217909488 JG In-Stock Unstable HRH2 46 42 O=C(CCCCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCCc1c[nH]cn1 ZINC000217909488 JG In-Stock Unstable HRH1 20 43 O=C(CCCCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCCc1c[nH]cn1 ZINC000217909488 JG In-Stock Unstable HRH3 44 52 O=C(CCCCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCCc1c[nH]cn1 ZINC000217909488 JG In-Stock Unstable HRH4 28 40 Cc1cccc(/C=C/NC(=O)N2c3ccccc3C[C@H]2C)c1 ZINC000217909492 CI For-Sale Unstable DRD4 28 53 CC(C)[C@H]1CCN(c2cnc3ccccc3n2)CCN1 ZINC000217909513 CE For-Sale Unstable SORD 27 49 O=C(O)/C=C\c1cncc(C(=O)Nc2cccc(Cl)c2)c1 ZINC000217909517 DG For-Sale Anodyne MAOB 0 53 O=C(O)/C=C\c1cncc(C(=O)Nc2cccc(Cl)c2)c1 ZINC000217909517 DG For-Sale Anodyne PPIA 17 45 O=C(O)/C=C\c1cncc(C(=O)Nc2cccc(Cl)c2)c1 ZINC000217909517 DG For-Sale Anodyne GRM5 15 46 O=C(O)/C=C\c1cncc(C(=O)Nc2cccc(Cl)c2)c1 ZINC000217909517 DG For-Sale Anodyne SCN10A 41 40 O=C(O)/C=C\c1cncc(C(=O)Nc2cccc(Cl)c2)c1 ZINC000217909517 DG For-Sale Anodyne CSF1R 23 45 O=C(O)/C=C\c1cncc(C(=O)Nc2cccc(Cl)c2)c1 ZINC000217909517 DG For-Sale Anodyne TAAR1 18 52 O=C(O)/C=C\c1cncc(C(=O)Nc2cccc(Cl)c2)c1 ZINC000217909517 DG For-Sale Anodyne KCNK3 103 50 O=C(O)/C=C\c1cncc(C(=O)Nc2cccc(Cl)c2)c1 ZINC000217909517 DG For-Sale Anodyne KCNK9 53 47 CNC(=O)c1ccc(CN[C@@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217909530 CE For-Sale Unstable SSTR3 16 42 O=S(=O)(c1ccccc1)N(CCF)c1ccncc1 ZINC000217909539 CE For-Sale Unstable NR1I2 22 41 O=S(=O)(c1ccccc1)N(CCF)c1ccncc1 ZINC000217909539 CE For-Sale Unstable NR1H2 15 41 O=S(=O)(c1ccccc1)N(CCF)c1ccncc1 ZINC000217909539 CE For-Sale Unstable RORC 15 46 O=C(CCCCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCCc1c[nH]cn1 ZINC000217909557 JG In-Stock Unstable HRH2 46 42 O=C(CCCCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCCc1c[nH]cn1 ZINC000217909557 JG In-Stock Unstable HRH1 20 43 O=C(CCCCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCCc1c[nH]cn1 ZINC000217909557 JG In-Stock Unstable HRH3 44 52 O=C(CCCCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCCc1c[nH]cn1 ZINC000217909557 JG In-Stock Unstable HRH4 28 40 Cc1cc(N)cc(N2CCC(N3CCCC3)CC2)c1 ZINC000217909574 CF For-Sale Unstable HRH3 19 43 Cc1cc(N)cc(N2CCC(N3CCCC3)CC2)c1 ZINC000217909574 CF For-Sale Unstable L3MBTL3 104 54 Cc1cccc(/C=C/NC(=O)N2c3ccccc3C[C@@H]2C)c1 ZINC000217909579 CI For-Sale Unstable DRD4 28 53 C#CCN1C(=O)C(=O)c2ccccc2C1=O ZINC000217909583 BC In-Stock Unstable ALDH1A1 60 42 C#CCN1C(=O)C(=O)c2ccccc2C1=O ZINC000217909583 BC In-Stock Unstable ALDH3A1 37 40 O=C(O)/C=C\c1cncc(C(=O)Nc2cccc(F)c2)c1 ZINC000217909606 CF For-Sale Anodyne SCN10A 22 40 O=C(O)/C=C\c1cncc(C(=O)Nc2cccc(F)c2)c1 ZINC000217909606 CF For-Sale Anodyne CSF1R 17 43 O=C(O)/C=C\c1cncc(C(=O)Nc2cccc(F)c2)c1 ZINC000217909606 CF For-Sale Anodyne TAAR1 26 41 O=C(O)/C=C\c1cncc(C(=O)Nc2cccc(F)c2)c1 ZINC000217909606 CF For-Sale Anodyne KCNK3 103 50 O=C(O)/C=C\c1cncc(C(=O)Nc2cccc(F)c2)c1 ZINC000217909606 CF For-Sale Anodyne KCNK9 54 47 CNC(=O)c1ccc(CN[C@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217909607 CE For-Sale Unstable SSTR3 16 42 COc1ccc(-c2noc(CN(C)C(=O)/C=C/c3ccc(Cl)cc3Cl)n2)cc1 ZINC000217909643 HJ In-Stock Unstable CYSP_PLAFA 38 40 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)c1ccccc1 ZINC000217909652 HD In-Stock Unstable HTR1D 23 41 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)c1ccccc1 ZINC000217909652 HD In-Stock Unstable HTR1B 17 41 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)c1ccccc1 ZINC000217909652 HD In-Stock Unstable EDNRA 22 43 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)c1ccccc1 ZINC000217909652 HD In-Stock Unstable CCKAR 45 40 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)c1ccccc1 ZINC000217909652 HD In-Stock Unstable ECE1 41 37 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)c1ccccc1 ZINC000217909652 HD In-Stock Unstable SSTR3 49 34 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)c1ccccc1 ZINC000217909652 HD In-Stock Unstable CCKBR 42 40 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)N[C@H](CO)c1ccccc1 ZINC000217909652 HD In-Stock Unstable GHSR 56 39 N#CCN1C(=O)C(=O)c2ccccc2C1=O ZINC000217909669 BC In-Stock Unstable ALDH1A1 60 42 N#CCN1C(=O)C(=O)c2ccccc2C1=O ZINC000217909669 BC In-Stock Unstable ALDH3A1 37 40 CNC(=O)c1ccc(CN[C@@H]2C[C@H]3CC=C[C@H]32)cc1 ZINC000217909674 CE For-Sale Unstable SSTR3 16 42 CCCCCCCCCCCCOc1c2cccc1Cc1cccc(c1O)Cc1cccc(c1OCCCCCCCCCCCC)Cc1cccc(c1O)C2 ZINC000217909691 KK In-Stock Unstable THRA 58 37 CCCCCCCCCCCCOc1c2cccc1Cc1cccc(c1O)Cc1cccc(c1OCCCCCCCCCCCC)Cc1cccc(c1O)C2 ZINC000217909691 KK In-Stock Unstable INHA 52 34 CCCCCCCCCCCCOc1c2cccc1Cc1cccc(c1O)Cc1cccc(c1OCCCCCCCCCCCC)Cc1cccc(c1O)C2 ZINC000217909691 KK In-Stock Unstable THRB 41 37 CCCCCCCCCCCCOc1c2cccc1Cc1cccc(c1O)Cc1cccc(c1OCCCCCCCCCCCC)Cc1cccc(c1O)C2 ZINC000217909691 KK In-Stock Unstable LPAR2 45 33 CCCCCCCCCCCCOc1c2cccc1Cc1cccc(c1O)Cc1cccc(c1OCCCCCCCCCCCC)Cc1cccc(c1O)C2 ZINC000217909691 KK In-Stock Unstable PLA2G4B 84 39 CCCCCCCCCCCCOc1c2cccc1Cc1cccc(c1O)Cc1cccc(c1OCCCCCCCCCCCC)Cc1cccc(c1O)C2 ZINC000217909691 KK In-Stock Unstable S1PR2 44 33 Cc1cccc(/C=C/NC(=O)NC2CC2)c1 ZINC000217909695 BE For-Sale Unstable EPHX2 19 44 COc1ccc(-c2noc(CN(C)C(=O)/C=C/c3ccc(Cl)cc3Cl)n2)c(OC)c1 ZINC000217909741 IJ In-Stock Unstable CYSP_PLAFA 43 46 CNC(=O)c1ccc(CN[C@H]2C[C@H]3CC=C[C@@H]23)cc1 ZINC000217909766 CE For-Sale Unstable SSTR3 16 42 COc1ccccc1CNC(=O)N/C=C/c1cccc(C)c1 ZINC000217909783 CG For-Sale Unstable PHES 0 46 COc1ccccc1CNC(=O)N/C=C/c1cccc(C)c1 ZINC000217909783 CG For-Sale Unstable KCNK3 41 37 COC(=O)CN1C(=O)C(=O)c2ccccc2C1=O ZINC000217909787 BC In-Stock Unstable ALDH1A1 56 42 COC(=O)CN1C(=O)C(=O)c2ccccc2C1=O ZINC000217909787 BC In-Stock Unstable ALDH3A1 30 42 COC(=O)CN1C(=O)C(=O)c2ccccc2C1=O ZINC000217909787 BC In-Stock Unstable CES1 19 41 O=C(O)/C=C\c1cncc(C(=O)NCC(=O)NC2CC2)c1 ZINC000217909801 CC For-Sale Unstable CCR2 34 41 CN(Cc1nc(-c2ccc(Cl)cc2)no1)C(=O)/C=C/c1ccc(Cl)cc1Cl ZINC000217909827 HK In-Stock Unstable TSPO 15 46 COC(=O)[C@@H](NC(=O)c1cccc(-c2cc3ccccc3oc2=O)c1)C(C)C ZINC000217909839 GG In-Stock Unstable MAOB 17 41 O=C(O)CN1C(=O)C(=O)c2ccccc2C1=O ZINC000217909873 BB In-Stock Unstable PTGS1 26 41 O=C(O)CN1C(=O)C(=O)c2ccccc2C1=O ZINC000217909873 BB In-Stock Unstable AKR1B1 34 42 O=C(O)CN1C(=O)C(=O)c2ccccc2C1=O ZINC000217909873 BB In-Stock Unstable CDC25B 0 50 O=C(O)CN1C(=O)C(=O)c2ccccc2C1=O ZINC000217909873 BB In-Stock Unstable ALDH1A1 67 47 O=C(O)CN1C(=O)C(=O)c2ccccc2C1=O ZINC000217909873 BB In-Stock Unstable ALDH3A1 41 45 O=C(O)CN1C(=O)C(=O)c2ccccc2C1=O ZINC000217909873 BB In-Stock Unstable CES1 21 43 Cc1cccc(/C=C/NC(=O)N2CCN(c3ncccn3)CC2)c1 ZINC000217909915 DE For-Sale Unstable SLC6A7 0 46 Cc1cccc(/C=C/NC(=O)N2CCN(c3cccc(C)c3)CC2)c1 ZINC000217910019 EH For-Sale Unstable CCR1 0 44 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1 ZINC000217910032 GK In-Stock Unstable PYGL 0 43 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1 ZINC000217910032 GK In-Stock Unstable HDAC9 15 47 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1 ZINC000217910032 GK In-Stock Unstable HDAC7 23 47 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2Cl)cc1 ZINC000217910032 GK In-Stock Unstable BOTA 32 51 Cc1onc(-c2ccccc2Cl)c1C(=O)N(Cc1nn(C)c2c1CCC2)C1CCCC1 ZINC000217910040 IK In-Stock Unstable GPBAR1 42 53 COC(=O)C[C@@H](NC(=O)c1cc(C)nn1C)C(=O)O ZINC000217910058 CB For-Sale Unstable CTSV 45 35 CC[C@@H](C)N(C)CCNS(=O)(=O)c1c(C)cc(F)cc1C ZINC000217910064 DE On-Demand Unstable NR3C2 0 42 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCc1ccc(OC)c(OCc2ccccc2)c1 ZINC000217910080 KJ For-Sale Unstable PTGER1 48 34 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCc1ccc(OC)c(OCc2ccccc2)c1 ZINC000217910080 KJ For-Sale Unstable MTNR1B 19 41 CC[C@H](C)N(C)CCNS(=O)(=O)c1c(C)cc(F)cc1C ZINC000217910142 DE On-Demand Unstable NR3C2 0 42 CCOC(=O)N1CCC(NC(=O)N/C=C/c2cccc(C)c2)CC1 ZINC000217910158 EF For-Sale Unstable EPHX2 30 53 CCOC(=O)N1CCC(NC(=O)N/C=C/c2cccc(C)c2)CC1 ZINC000217910158 EF For-Sale Unstable CCR8 24 40 CN(CCCNC(=O)/C=C/c1ccc(Cl)cc1Cl)c1ccccc1 ZINC000217910161 FJ In-Stock Unstable HDAC9 22 47 CN(CCCNC(=O)/C=C/c1ccc(Cl)cc1Cl)c1ccccc1 ZINC000217910161 FJ In-Stock Unstable HDAC7 33 47 CN(CCCNC(=O)/C=C/c1ccc(Cl)cc1Cl)c1ccccc1 ZINC000217910161 FJ In-Stock Unstable BOTA 30 51 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCc1ccc(OC)c(OCc2ccccc2)c1 ZINC000217910170 KJ For-Sale Unstable PTGER1 48 34 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCc1ccc(OC)c(OCc2ccccc2)c1 ZINC000217910170 KJ For-Sale Unstable MTNR1B 19 41 CCO[C@@H]1C[C@@H](NC(=O)NC2CC2)C1(C)C ZINC000217910196 BD For-Sale Unstable EPHX2 21 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCc1ccc(OC)c(OCc2ccccc2)c1 ZINC000217910242 KJ For-Sale Unstable PTGER1 48 34 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCc1ccc(OC)c(OCc2ccccc2)c1 ZINC000217910242 KJ For-Sale Unstable MTNR1B 19 41 Cc1cccc(/C=C/NC(=O)N2CCN(c3cccc(Cl)c3)CC2)c1 ZINC000217910262 FI For-Sale Unstable HTR1A 17 42 Cc1cccc(/C=C/NC(=O)N2CCN(c3cccc(Cl)c3)CC2)c1 ZINC000217910262 FI For-Sale Unstable HTR2A 15 42 Cc1cccc(/C=C/NC(=O)N2CCN(c3cccc(Cl)c3)CC2)c1 ZINC000217910262 FI For-Sale Unstable CCR1 26 44 OC1CCC(NCCc2ccccn2)CC1 ZINC000217910267 BD On-Demand Unstable MERTK 27 40 O=C(/C=C/c1ccc(Cl)cc1Cl)NCCCN1CCCc2ccccc21 ZINC000217910268 GJ In-Stock Unstable DRD3 32 46 O=C(/C=C/c1ccc(Cl)cc1Cl)NCCCN1CCCc2ccccc21 ZINC000217910268 GJ In-Stock Unstable HDAC7 21 42 O=C(/C=C/c1ccc(Cl)cc1Cl)NCCCN1CCCc2ccccc21 ZINC000217910268 GJ In-Stock Unstable BOTA 24 45 Nc1nc2c(c(C(=O)NCCc3cccnc3)n1)CCCC2 ZINC000217910273 CD In-Stock Unstable PTAFR 29 45 Nc1nc2c(c(C(=O)NCCc3cccnc3)n1)CCCC2 ZINC000217910273 CD In-Stock Unstable BCHE 59 35 Nc1nc2c(c(C(=O)NCCc3cccnc3)n1)CCCC2 ZINC000217910273 CD In-Stock Unstable NAMPT 29 48 COC(=O)[C@@H]1CCc2c1c1ccccc1n2C ZINC000217910274 BE In-Stock Unstable TSPO 19 42 CCO[C@H]1C[C@@H](NC(=O)NC2CC2)C1(C)C ZINC000217910295 BD For-Sale Unstable EPHX2 21 40 Cc1cc(C(=O)N[C@@H]2CC[C@@H]3CNC[C@@H]3C2)n(C)n1 ZINC000217910320 CC For-Sale Unstable INHA 50 33 Cc1cc(C(=O)N[C@@H]2CC[C@@H]3CNC[C@@H]3C2)n(C)n1 ZINC000217910320 CC For-Sale Unstable MAPK13 43 32 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCc1ccc(OC)c(OCc2ccccc2)c1 ZINC000217910342 KJ For-Sale Unstable PTGER1 48 34 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCc1ccc(OC)c(OCc2ccccc2)c1 ZINC000217910342 KJ For-Sale Unstable MTNR1B 19 41 COC(=O)[C@H]1CCc2c1c1ccccc1n2C ZINC000217910344 BE In-Stock Unstable TSPO 19 42 CCO[C@@H]1C[C@H](NC(=O)NC2CC2)C1(C)C ZINC000217910354 BD For-Sale Unstable EPHX2 21 40 O=C(O)/C=C\c1cncc(C(=O)NCc2ccccc2)c1 ZINC000217910361 CE For-Sale Unstable SCN10A 34 40 O=C(O)/C=C\c1cncc(C(=O)NCc2ccccc2)c1 ZINC000217910361 CE For-Sale Unstable NAMPT 60 40 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccc(F)cc2)c1 ZINC000217910387 DH In-Stock Unstable ANPEP 19 41 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccc(F)cc2)c1 ZINC000217910387 DH In-Stock Unstable MMP2 17 50 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccc(F)cc2)c1 ZINC000217910387 DH In-Stock Unstable NR1H4 25 42 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccc(F)cc2)c1 ZINC000217910387 DH In-Stock Unstable MMP9 16 50 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccc(F)cc2)c1 ZINC000217910387 DH In-Stock Unstable HDAC7 44 33 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccc(F)cc2)c1 ZINC000217910387 DH In-Stock Unstable MMP1 0 41 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccc(F)cc2)c1 ZINC000217910387 DH In-Stock Unstable AMP1_PLAFQ 26 40 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccc(F)cc2)c1 ZINC000217910387 DH In-Stock Unstable PDS 49 38 Cc1cccc(/C=C/NC(=O)Nc2ccc(-c3nc4ccc(C)cc4s3)cc2)c1 ZINC000217910398 GK For-Sale Unstable CSNK1D 15 40 Cc1cccc(/C=C/NC(=O)Nc2ccc(-c3nc4ccc(C)cc4s3)cc2)c1 ZINC000217910398 GK For-Sale Unstable APP 26 53 Cc1cccc(/C=C/NC(=O)Nc2ccc(-c3nc4ccc(C)cc4s3)cc2)c1 ZINC000217910398 GK For-Sale Unstable LUCI_PHOPE 22 40 COc1ccc(CN2C[C@@H]3CCCCN3C[C@@H]2C)c(O)c1 ZINC000217910407 CE For-Sale Unstable CHRM2 15 49 COc1ccc(CN2C[C@@H]3CCCCN3C[C@@H]2C)c(O)c1 ZINC000217910407 CE For-Sale Unstable SIGMAR1 15 44 CCO[C@H]1C[C@H](NC(=O)NC2CC2)C1(C)C ZINC000217910410 BD For-Sale Unstable EPHX2 21 40 Cc1cccc(/C=C/NC(=O)Nc2ccc3c(c2)OCO3)c1 ZINC000217910504 CH For-Sale Unstable TRPV1 0 50 Cc1cccc(/C=C/NC(=O)Nc2ccc3c(c2)OCO3)c1 ZINC000217910504 CH For-Sale Unstable CCR2 0 42 Cc1cccc(/C=C/NC(=O)Nc2ccc3c(c2)OCO3)c1 ZINC000217910504 CH For-Sale Unstable DYRK2 52 37 Cc1cccc(/C=C/NC(=O)Nc2ccc3c(c2)OCO3)c1 ZINC000217910504 CH For-Sale Unstable KCNK3 40 35 CCOc1ccc(CNC(=O)/C=C/c2ccc(F)cc2)cc1OCC ZINC000217910505 EH In-Stock Unstable BDKRB2 46 33 CCOc1ccc(CNC(=O)/C=C/c2ccc(F)cc2)cc1OCC ZINC000217910505 EH In-Stock Unstable HDAC8 0 40 CCOc1ccc(CNC(=O)/C=C/c2ccc(F)cc2)cc1OCC ZINC000217910505 EH In-Stock Unstable AKR1C3 27 40 Cc1cc(C(=O)N[C@@H]2CC[C@H]3CNC[C@@H]3C2)n(C)n1 ZINC000217910510 CC For-Sale Unstable INHA 50 33 Cc1cc(C(=O)N[C@@H]2CC[C@H]3CNC[C@@H]3C2)n(C)n1 ZINC000217910510 CC For-Sale Unstable MAPK13 43 32 CCO[C@@H]1C[C@@H](NC(=O)NCc2ccccc2)C1(C)C ZINC000217910547 CF For-Sale Unstable ANPEP 16 40 CCO[C@@H]1C[C@@H](NC(=O)NCc2ccccc2)C1(C)C ZINC000217910547 CF For-Sale Unstable TIMP3 69 41 CCO[C@@H]1C[C@@H](NC(=O)NCc2ccccc2)C1(C)C ZINC000217910547 CF For-Sale Unstable PDS 50 36 CCO[C@H]1C[C@@H](NC(=O)NCc2ccccc2)C1(C)C ZINC000217910597 CF For-Sale Unstable ANPEP 16 40 CCO[C@H]1C[C@@H](NC(=O)NCc2ccccc2)C1(C)C ZINC000217910597 CF For-Sale Unstable TIMP3 69 41 CCO[C@H]1C[C@@H](NC(=O)NCc2ccccc2)C1(C)C ZINC000217910597 CF For-Sale Unstable PDS 50 36 COc1cc(CNC(=O)/C=C/c2ccc(F)cc2)ccc1OC(C)C ZINC000217910600 EH In-Stock Unstable TRPV1 15 44 COc1cc(CNC(=O)/C=C/c2ccc(F)cc2)ccc1OC(C)C ZINC000217910600 EH In-Stock Unstable HDAC8 0 46 COc1cc(CNC(=O)/C=C/c2ccc(F)cc2)ccc1OC(C)C ZINC000217910600 EH In-Stock Unstable NR1H4 18 40 COc1cc(CNC(=O)/C=C/c2ccc(F)cc2)ccc1OC(C)C ZINC000217910600 EH In-Stock Unstable HDAC1 0 42 O[C@@H]1CCC[C@H]1Cc1ccc(OCc2ccccc2)cc1 ZINC000217910601 CH For-Sale Unstable ALOX5 17 44 O[C@@H]1CCC[C@H]1Cc1ccc(OCc2ccccc2)cc1 ZINC000217910601 CH For-Sale Unstable MAOB 26 44 O[C@@H]1CCC[C@H]1Cc1ccc(OCc2ccccc2)cc1 ZINC000217910601 CH For-Sale Unstable KCNH2 18 42 O[C@@H]1CCC[C@H]1Cc1ccc(OCc2ccccc2)cc1 ZINC000217910601 CH For-Sale Unstable LTA4H 67 48 O[C@@H]1CCC[C@H]1Cc1ccc(OCc2ccccc2)cc1 ZINC000217910601 CH For-Sale Unstable ACR 26 41 O[C@@H]1CCC[C@H]1Cc1ccc(OCc2ccccc2)cc1 ZINC000217910601 CH For-Sale Unstable TAAR1 19 44 O[C@@H]1CCC[C@H]1Cc1ccc(OCc2ccccc2)cc1 ZINC000217910601 CH For-Sale Unstable FFAR1 35 47 CCO[C@@H]1C[C@H](NC(=O)NCc2ccccc2)C1(C)C ZINC000217910677 CF For-Sale Unstable ANPEP 16 40 CCO[C@@H]1C[C@H](NC(=O)NCc2ccccc2)C1(C)C ZINC000217910677 CF For-Sale Unstable TIMP3 69 41 CCO[C@@H]1C[C@H](NC(=O)NCc2ccccc2)C1(C)C ZINC000217910677 CF For-Sale Unstable PDS 50 36 C[C@H]1C[C@H](C)CCN1Cc1ccc(CCNC2CC2)cc1 ZINC000217910715 CH For-Sale Unstable HRH3 15 40 O=C(/C=C/c1ccc(F)cc1)NCCCc1ccccc1Cl ZINC000217910716 DI In-Stock Unstable DRD3 17 48 O=C(/C=C/c1ccc(F)cc1)NCCCc1ccccc1Cl ZINC000217910716 DI In-Stock Unstable PYGL 28 52 O=C(/C=C/c1ccc(F)cc1)NCCCc1ccccc1Cl ZINC000217910716 DI In-Stock Unstable MMP2 17 48 O=C(/C=C/c1ccc(F)cc1)NCCCc1ccccc1Cl ZINC000217910716 DI In-Stock Unstable HDAC2 18 41 O=C(/C=C/c1ccc(F)cc1)NCCCc1ccccc1Cl ZINC000217910716 DI In-Stock Unstable HDAC4 17 41 O=C(/C=C/c1ccc(F)cc1)NCCCc1ccccc1Cl ZINC000217910716 DI In-Stock Unstable HDAC9 42 41 O=C(/C=C/c1ccc(F)cc1)NCCCc1ccccc1Cl ZINC000217910716 DI In-Stock Unstable HDAC7 53 41 O=C(/C=C/c1ccc(F)cc1)NCCCc1ccccc1Cl ZINC000217910716 DI In-Stock Unstable MMP1 0 45 CCO[C@H]1C[C@H](NC(=O)NCc2ccccc2)C1(C)C ZINC000217910765 CF For-Sale Unstable ANPEP 16 40 CCO[C@H]1C[C@H](NC(=O)NCc2ccccc2)C1(C)C ZINC000217910765 CF For-Sale Unstable TIMP3 69 41 CCO[C@H]1C[C@H](NC(=O)NCc2ccccc2)C1(C)C ZINC000217910765 CF For-Sale Unstable PDS 50 36 C[C@H]1CCN(Cc2ccc(CCNC3CC3)cc2)[C@@H](C)C1 ZINC000217910782 CH For-Sale Unstable HRH3 15 40 O=C(/C=C/c1ccc(F)cc1)NCCCc1ccc(Cl)cc1 ZINC000217910799 DI In-Stock Unstable PYGL 27 51 O=C(/C=C/c1ccc(F)cc1)NCCCc1ccc(Cl)cc1 ZINC000217910799 DI In-Stock Unstable HDAC8 15 43 O=C(/C=C/c1ccc(F)cc1)NCCCc1ccc(Cl)cc1 ZINC000217910799 DI In-Stock Unstable HDAC1 20 47 O=C(/C=C/c1ccc(F)cc1)NCCCc1ccc(Cl)cc1 ZINC000217910799 DI In-Stock Unstable HDAC2 18 47 O=C(/C=C/c1ccc(F)cc1)NCCCc1ccc(Cl)cc1 ZINC000217910799 DI In-Stock Unstable HDAC4 17 47 O=C(/C=C/c1ccc(F)cc1)NCCCc1ccc(Cl)cc1 ZINC000217910799 DI In-Stock Unstable HDAC9 36 47 O=C(/C=C/c1ccc(F)cc1)NCCCc1ccc(Cl)cc1 ZINC000217910799 DI In-Stock Unstable HDAC7 54 47 O=C(/C=C/c1ccc(F)cc1)NCCCc1ccc(Cl)cc1 ZINC000217910799 DI In-Stock Unstable MMP1 0 43 O=C(/C=C/c1ccc(F)cc1)NCCCc1ccc(Cl)cc1 ZINC000217910799 DI In-Stock Unstable LEF 47 36 Cc1cccc(/C=C/NC(=O)N2CCc3ccccc32)c1 ZINC000217910812 CH For-Sale Unstable AVPR2 35 44 Cc1cccc(/C=C/NC(=O)N2CCc3ccccc32)c1 ZINC000217910812 CH For-Sale Unstable HSD17B3 18 40 CC(=O)Nc1ccc(NC(=O)c2csc(-c3cccc(Cl)c3)n2)c(C(F)(F)F)c1 ZINC000217910830 IK On-Demand Unstable MPL 41 33 CC(=O)Nc1ccc(NC(=O)c2csc(-c3cccc(Cl)c3)n2)c(C(F)(F)F)c1 ZINC000217910830 IK On-Demand Unstable GRM4 28 42 CC(=O)Nc1ccc(NC(=O)c2csc(-c3cccc(Cl)c3)n2)c(C(F)(F)F)c1 ZINC000217910830 IK On-Demand Unstable Q8MMZ8_EIMTE 42 35 O=C(O)/C=C\c1cncc(C(=O)Nc2ccc(Cl)cc2)c1 ZINC000217910878 DG For-Sale Anodyne SCN10A 52 48 O=C(O)/C=C\c1cncc(C(=O)Nc2ccc(Cl)cc2)c1 ZINC000217910878 DG For-Sale Anodyne Q25615_ONCVO 24 40 O=C(/C=C/c1ccc(F)cc1)NCCCc1ccc(F)cc1 ZINC000217910902 DH In-Stock Unstable PYGL 26 50 O=C(/C=C/c1ccc(F)cc1)NCCCc1ccc(F)cc1 ZINC000217910902 DH In-Stock Unstable HDAC8 33 43 O=C(/C=C/c1ccc(F)cc1)NCCCc1ccc(F)cc1 ZINC000217910902 DH In-Stock Unstable MMP2 15 56 O=C(/C=C/c1ccc(F)cc1)NCCCc1ccc(F)cc1 ZINC000217910902 DH In-Stock Unstable HDAC1 33 41 O=C(/C=C/c1ccc(F)cc1)NCCCc1ccc(F)cc1 ZINC000217910902 DH In-Stock Unstable HDAC2 22 43 O=C(/C=C/c1ccc(F)cc1)NCCCc1ccc(F)cc1 ZINC000217910902 DH In-Stock Unstable HDAC3 18 41 O=C(/C=C/c1ccc(F)cc1)NCCCc1ccc(F)cc1 ZINC000217910902 DH In-Stock Unstable HDAC4 34 41 O=C(/C=C/c1ccc(F)cc1)NCCCc1ccc(F)cc1 ZINC000217910902 DH In-Stock Unstable HDAC5 31 40 O=C(/C=C/c1ccc(F)cc1)NCCCc1ccc(F)cc1 ZINC000217910902 DH In-Stock Unstable HDAC6 21 41 O=C(/C=C/c1ccc(F)cc1)NCCCc1ccc(F)cc1 ZINC000217910902 DH In-Stock Unstable HDAC9 55 41 O=C(/C=C/c1ccc(F)cc1)NCCCc1ccc(F)cc1 ZINC000217910902 DH In-Stock Unstable HDAC7 55 41 O=C(/C=C/c1ccc(F)cc1)NCCCc1ccc(F)cc1 ZINC000217910902 DH In-Stock Unstable MMP1 0 48 O=C(/C=C/c1ccc(F)cc1)NCCCc1ccc(F)cc1 ZINC000217910902 DH In-Stock Unstable LEF 41 37 O=C(/C=C/c1ccc(F)cc1)NCCCc1ccc(F)cc1 ZINC000217910902 DH In-Stock Unstable TRPM2 0 43 CCCCCCCCOc1ccc([C@@H]2CC(=O)Oc3ccc4c(c32)OC(=C(C)C)C4=O)cc1 ZINC000217910909 IK In-Stock Unstable PLA2G4B 63 32 Cc1cccc(/C=C/NC(=O)Nc2ccc(I)cc2)c1 ZINC000217910923 GI For-Sale Unstable MMP1 0 43 Cc1cccc(/C=C/NC(=O)Nc2ccc(I)cc2)c1 ZINC000217910923 GI For-Sale Unstable KCNK3 40 35 CCCCCCCCOc1ccc([C@H]2CC(=O)Oc3ccc4c(c32)OC(=C(C)C)C4=O)cc1 ZINC000217910963 IK In-Stock Unstable PLA2G4B 68 32 Cc1cccc(/C=C/NC(=O)NCCc2c[nH]c3ccccc23)c1 ZINC000217911011 DH For-Sale Unstable TACR1 16 43 Cc1cccc(/C=C/NC(=O)NCCc2c[nH]c3ccccc23)c1 ZINC000217911011 DH For-Sale Unstable NQO2 25 43 Cc1cccc(/C=C/NC(=O)NCCc2c[nH]c3ccccc23)c1 ZINC000217911011 DH For-Sale Unstable CCKAR 51 42 Cc1cccc(/C=C/NC(=O)NCCc2c[nH]c3ccccc23)c1 ZINC000217911011 DH For-Sale Unstable CTSL 25 41 Cc1cccc(/C=C/NC(=O)NCCc2c[nH]c3ccccc23)c1 ZINC000217911011 DH For-Sale Unstable BRS3 27 41 Cc1cccc(/C=C/NC(=O)NCCc2c[nH]c3ccccc23)c1 ZINC000217911011 DH For-Sale Unstable NMBR 47 44 Cc1cccc(/C=C/NC(=O)NCCc2c[nH]c3ccccc23)c1 ZINC000217911011 DH For-Sale Unstable MTNR1A 26 46 Cc1cccc(/C=C/NC(=O)NCCc2c[nH]c3ccccc23)c1 ZINC000217911011 DH For-Sale Unstable MTNR1B 17 43 Cc1cccc(/C=C/NC(=O)NCCc2c[nH]c3ccccc23)c1 ZINC000217911011 DH For-Sale Unstable CCKBR 33 41 Cc1cccc(/C=C/NC(=O)NCCc2c[nH]c3ccccc23)c1 ZINC000217911011 DH For-Sale Unstable ALOX15 26 48 Cc1cccc(/C=C/NC(=O)NCCc2c[nH]c3ccccc23)c1 ZINC000217911011 DH For-Sale Unstable MMP9 15 51 COc1ccccc1CCCNC(=O)/C=C/c1ccc(F)cc1 ZINC000217911023 DH In-Stock Unstable DRD3 28 61 COc1ccccc1CCCNC(=O)/C=C/c1ccc(F)cc1 ZINC000217911023 DH In-Stock Unstable CCKAR 16 40 COc1ccccc1CCCNC(=O)/C=C/c1ccc(F)cc1 ZINC000217911023 DH In-Stock Unstable LTB4R 0 42 COc1ccccc1CCCNC(=O)/C=C/c1ccc(F)cc1 ZINC000217911023 DH In-Stock Unstable PYGL 0 42 COc1ccccc1CCCNC(=O)/C=C/c1ccc(F)cc1 ZINC000217911023 DH In-Stock Unstable MTNR1B 34 42 COc1ccccc1CCCNC(=O)/C=C/c1ccc(F)cc1 ZINC000217911023 DH In-Stock Unstable MMP2 17 46 COc1ccccc1CCCNC(=O)/C=C/c1ccc(F)cc1 ZINC000217911023 DH In-Stock Unstable MMP9 15 46 COc1ccccc1CCCNC(=O)/C=C/c1ccc(F)cc1 ZINC000217911023 DH In-Stock Unstable HDAC9 40 38 COc1ccccc1CCCNC(=O)/C=C/c1ccc(F)cc1 ZINC000217911023 DH In-Stock Unstable HDAC7 52 38 COc1ccccc1CCCNC(=O)/C=C/c1ccc(F)cc1 ZINC000217911023 DH In-Stock Unstable MMP1 0 43 COc1ccccc1CCCNC(=O)/C=C/c1ccc(F)cc1 ZINC000217911023 DH In-Stock Unstable HDA106 0 40 COc1ccccc1CCCNC(=O)/C=C/c1ccc(F)cc1 ZINC000217911023 DH In-Stock Unstable HD1B 0 40 COc1ccccc1CCCNC(=O)/C=C/c1ccc(F)cc1 ZINC000217911023 DH In-Stock Unstable MBTPS1 40 32 CC(=O)Nc1ccc(NC(=O)[C@@H]2COc3ccc(Cl)cc3C2)c(C(F)(F)F)c1 ZINC000217911051 HJ On-Demand Unstable ROCK2 31 53 O=C(O)/C=C\c1cncc(C(=O)Nc2ccc(F)cc2)c1 ZINC000217911058 CF For-Sale Anodyne CXCR2 0 42 O=C(O)/C=C\c1cncc(C(=O)Nc2ccc(F)cc2)c1 ZINC000217911058 CF For-Sale Anodyne KCNK3 21 42 O=C(Nc1nccs1)[C@@H]1CC(F)(F)CN1 ZINC000217911107 BD On-Demand Unstable MAP1 110 43 Cc1cc(C(=O)N(Cc2nn(C)c3c2CCC3)C2CCCC2)no1 ZINC000217911113 EF In-Stock Unstable S1PR3 0 56 CC(=O)Nc1ccc(NC(=O)[C@H]2COc3ccc(Cl)cc3C2)c(C(F)(F)F)c1 ZINC000217911135 HJ On-Demand Unstable ROCK2 31 53 CN(C)C(=O)CN1CCCN(C(=O)c2cccc(-c3ccccc3)c2)CC1 ZINC000217911141 FF In-Stock Unstable ABHD6 0 41 CN(C)C(=O)CN1CCCN(C(=O)c2cccc(-c3ccccc3)c2)CC1 ZINC000217911141 FF In-Stock Unstable SLC6A7 0 50 COc1cccc(CCCNC(=O)/C=C/c2ccc(F)cc2)c1 ZINC000217911142 DH In-Stock Unstable DRD3 19 51 COc1cccc(CCCNC(=O)/C=C/c2ccc(F)cc2)c1 ZINC000217911142 DH In-Stock Unstable PTAFR 24 50 COc1cccc(CCCNC(=O)/C=C/c2ccc(F)cc2)c1 ZINC000217911142 DH In-Stock Unstable PYGL 22 44 COc1cccc(CCCNC(=O)/C=C/c2ccc(F)cc2)c1 ZINC000217911142 DH In-Stock Unstable HDAC8 33 41 COc1cccc(CCCNC(=O)/C=C/c2ccc(F)cc2)c1 ZINC000217911142 DH In-Stock Unstable MTNR1A 73 60 COc1cccc(CCCNC(=O)/C=C/c2ccc(F)cc2)c1 ZINC000217911142 DH In-Stock Unstable MTNR1B 71 60 COc1cccc(CCCNC(=O)/C=C/c2ccc(F)cc2)c1 ZINC000217911142 DH In-Stock Unstable MMP2 17 46 COc1cccc(CCCNC(=O)/C=C/c2ccc(F)cc2)c1 ZINC000217911142 DH In-Stock Unstable HDAC1 28 42 COc1cccc(CCCNC(=O)/C=C/c2ccc(F)cc2)c1 ZINC000217911142 DH In-Stock Unstable HDAC6 24 41 COc1cccc(CCCNC(=O)/C=C/c2ccc(F)cc2)c1 ZINC000217911142 DH In-Stock Unstable MMP9 16 46 COc1cccc(CCCNC(=O)/C=C/c2ccc(F)cc2)c1 ZINC000217911142 DH In-Stock Unstable HDAC7 41 37 COc1cccc(CCCNC(=O)/C=C/c2ccc(F)cc2)c1 ZINC000217911142 DH In-Stock Unstable MMP1 0 40 COc1cccc(CCCNC(=O)/C=C/c2ccc(F)cc2)c1 ZINC000217911142 DH In-Stock Unstable AMP1_PLAFQ 27 41 COc1cccc(CCCNC(=O)/C=C/c2ccc(F)cc2)c1 ZINC000217911142 DH In-Stock Unstable HDA106 0 42 COc1cccc(CCCNC(=O)/C=C/c2ccc(F)cc2)c1 ZINC000217911142 DH In-Stock Unstable AKR1C3 25 40 COc1cccc(CCCNC(=O)/C=C/c2ccc(F)cc2)c1 ZINC000217911142 DH In-Stock Unstable HD1B 0 42 COc1cccc(CCCNC(=O)/C=C/c2ccc(F)cc2)c1 ZINC000217911142 DH In-Stock Unstable CRTM 59 47 Nc1ccc2[nH]c3c(c2c1)[C@H](C(=O)O)CC3 ZINC000217911206 BD In-Stock Unstable NGFR 0 48 CC(C)S(=O)(=O)c1ccc(CC(=O)N(Cc2nn(C)c3c2CCC3)C2CCCC2)cc1 ZINC000217911207 IH In-Stock Unstable CCR5 28 41 CC[C@@H](C)[C@@H](NC(=O)[C@@H](N)CCS(C)(=O)=O)C(=O)OC ZINC000217911226 DB For-Sale Unstable PAPA1_CARPA 46 34 CC[C@@H](C)[C@@H](NC(=O)[C@@H](N)CCS(C)(=O)=O)C(=O)OC ZINC000217911226 DB For-Sale Unstable ENPEP 88 46 COc1ccc(CCCNC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217911228 DH In-Stock Unstable PTGS2 0 51 COc1ccc(CCCNC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217911228 DH In-Stock Unstable DRD3 17 52 COc1ccc(CCCNC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217911228 DH In-Stock Unstable SCNN1A 15 40 COc1ccc(CCCNC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217911228 DH In-Stock Unstable PTAFR 17 43 COc1ccc(CCCNC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217911228 DH In-Stock Unstable AHR 29 40 COc1ccc(CCCNC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217911228 DH In-Stock Unstable PYGL 0 42 COc1ccc(CCCNC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217911228 DH In-Stock Unstable HDAC8 34 50 COc1ccc(CCCNC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217911228 DH In-Stock Unstable MTNR1A 39 41 COc1ccc(CCCNC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217911228 DH In-Stock Unstable MTNR1B 32 41 COc1ccc(CCCNC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217911228 DH In-Stock Unstable MMP2 15 47 COc1ccc(CCCNC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217911228 DH In-Stock Unstable HDAC1 30 42 COc1ccc(CCCNC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217911228 DH In-Stock Unstable HDAC6 23 50 COc1ccc(CCCNC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217911228 DH In-Stock Unstable HDAC9 46 37 COc1ccc(CCCNC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217911228 DH In-Stock Unstable HDAC7 51 37 COc1ccc(CCCNC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217911228 DH In-Stock Unstable LEF 46 37 Cc1ccc(CNC2CCN(C(=O)OC(C)(C)C)CC2)cn1 ZINC000217911233 DF On-Demand Unstable GPR119 42 42 C[C@@H](Cn1cccn1)C(=O)NCc1nnnn1-c1ccccc1 ZINC000217911278 DC In-Stock Unstable DAGLA 17 40 CC[C@H](C)[C@@H](NC(=O)[C@@H](N)CCS(C)(=O)=O)C(=O)OC ZINC000217911299 DB For-Sale Unstable PAPA1_CARPA 46 34 CC[C@H](C)[C@@H](NC(=O)[C@@H](N)CCS(C)(=O)=O)C(=O)OC ZINC000217911299 DB For-Sale Unstable ENPEP 88 46 Nc1ccc2[nH]c3c(c2c1)[C@@H](C(=O)O)CC3 ZINC000217911302 BD In-Stock Unstable NGFR 0 48 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217911326 EG In-Stock Unstable SDH1 0 50 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217911326 EG In-Stock Unstable AHR 25 40 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217911326 EG In-Stock Unstable HDAC8 17 50 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217911326 EG In-Stock Unstable CDC25B 0 44 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217911326 EG In-Stock Unstable MMP2 18 46 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217911326 EG In-Stock Unstable HDAC1 0 44 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217911326 EG In-Stock Unstable HDAC2 19 46 Cn1nc(CN(C(=O)c2cccc(C#N)c2)C2CCCC2)c2c1CCC2 ZINC000217911327 EG In-Stock Unstable ITK 17 41 CC(C)CCCCCCNCCc1ccncc1 ZINC000217911330 BH For-Sale Unstable GNRHR 22 42 CC(C)CCCCCCNCCc1ccncc1 ZINC000217911330 BH For-Sale Unstable FDFT1 0 40 CC(C)CCCCCCNCCc1ccncc1 ZINC000217911330 BH For-Sale Unstable GPM3 0 40 C[C@H](Cn1cccn1)C(=O)NCc1nnnn1-c1ccccc1 ZINC000217911351 DC In-Stock Unstable DAGLA 17 40 Cc1cccc(/C=C/NC(=O)Nc2ccc(C)cc2O)c1 ZINC000217911366 CH For-Sale Unstable MMP2 0 43 Cc1cccc(/C=C/NC(=O)Nc2ccc(C)cc2O)c1 ZINC000217911366 CH For-Sale Unstable MMP9 0 43 Cc1cccc(/C=C/NC(=O)Nc2ccc(C)cc2O)c1 ZINC000217911366 CH For-Sale Unstable MMP1 0 43 CC[C@@H](C)[C@H](NC(=O)[C@@H](N)CCS(C)(=O)=O)C(=O)OC ZINC000217911382 DB For-Sale Unstable PAPA1_CARPA 46 34 CC[C@@H](C)[C@H](NC(=O)[C@@H](N)CCS(C)(=O)=O)C(=O)OC ZINC000217911382 DB For-Sale Unstable ENPEP 88 46 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217911404 EG In-Stock Unstable SDH1 0 50 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217911404 EG In-Stock Unstable AHR 25 40 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217911404 EG In-Stock Unstable HDAC8 17 50 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217911404 EG In-Stock Unstable CDC25B 0 44 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217911404 EG In-Stock Unstable MMP2 18 46 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217911404 EG In-Stock Unstable HDAC1 0 44 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217911404 EG In-Stock Unstable HDAC2 19 46 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCCc1c[nH]cn1 ZINC000217911425 IF In-Stock Unstable TOP1 0 40 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCCc1c[nH]cn1 ZINC000217911425 IF In-Stock Unstable HRH2 46 42 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCCc1c[nH]cn1 ZINC000217911425 IF In-Stock Unstable HRH1 33 42 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCCc1c[nH]cn1 ZINC000217911425 IF In-Stock Unstable HRH3 46 53 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCCc1c[nH]cn1 ZINC000217911425 IF In-Stock Unstable HRH4 29 41 CC[C@H](C)[C@H](NC(=O)[C@@H](N)CCS(C)(=O)=O)C(=O)OC ZINC000217911456 DB For-Sale Unstable PAPA1_CARPA 46 34 CC[C@H](C)[C@H](NC(=O)[C@@H](N)CCS(C)(=O)=O)C(=O)OC ZINC000217911456 DB For-Sale Unstable ENPEP 88 46 COc1cccc(/C=C/c2cccc(N)c2)c1 ZINC000217911482 BG Annotated Unstable CYP1B1 76 58 COc1cccc(/C=C/c2cccc(N)c2)c1 ZINC000217911482 BG Annotated Unstable AHR 42 62 COc1cccc(/C=C/c2cccc(N)c2)c1 ZINC000217911482 BG Annotated Unstable CYP1A1 55 58 COc1cccc(/C=C/c2cccc(N)c2)c1 ZINC000217911482 BG Annotated Unstable TUBB2B 24 40 COc1cccc(/C=C/c2cccc(N)c2)c1 ZINC000217911482 BG Annotated Unstable CYP1A2 20 58 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCCc1c[nH]cn1 ZINC000217911498 IF In-Stock Unstable TOP1 0 40 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCCc1c[nH]cn1 ZINC000217911498 IF In-Stock Unstable HRH2 46 42 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCCc1c[nH]cn1 ZINC000217911498 IF In-Stock Unstable HRH1 33 42 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCCc1c[nH]cn1 ZINC000217911498 IF In-Stock Unstable HRH3 46 53 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCCc1c[nH]cn1 ZINC000217911498 IF In-Stock Unstable HRH4 29 41 CC(C)CCCCCCNCCc1ccccn1 ZINC000217911518 BH For-Sale Unstable GPM3 0 58 O=C(/C=C/c1ccc(F)cc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217911525 EJ In-Stock Anodyne LTB4R 0 60 O=C(/C=C/c1ccc(F)cc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217911525 EJ In-Stock Anodyne HDAC8 15 42 O=C(/C=C/c1ccc(F)cc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217911525 EJ In-Stock Anodyne MMP2 25 58 O=C(/C=C/c1ccc(F)cc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217911525 EJ In-Stock Anodyne HDAC1 26 47 O=C(/C=C/c1ccc(F)cc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217911525 EJ In-Stock Anodyne HDAC2 22 43 O=C(/C=C/c1ccc(F)cc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217911525 EJ In-Stock Anodyne HDAC6 16 43 O=C(/C=C/c1ccc(F)cc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217911525 EJ In-Stock Anodyne MMP9 22 58 O=C(/C=C/c1ccc(F)cc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217911525 EJ In-Stock Anodyne MMP1 28 58 O=C(/C=C/c1ccc(F)cc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217911525 EJ In-Stock Anodyne FABH 0 41 O=C(/C=C/c1ccc(F)cc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217911525 EJ In-Stock Anodyne HDA106 0 46 O=C(/C=C/c1ccc(F)cc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217911525 EJ In-Stock Anodyne TRPM2 0 50 C[C@H]1CN(C)[C@@H](C)C[C@@H]1NCc1cccc(C(F)(F)F)c1 ZINC000217911529 DH For-Sale Unstable CCR2 24 43 Cc1cc(C(=O)Nc2cccc(/C=C\C(=O)O)n2)n(C)n1 ZINC000217911531 CD For-Sale Unstable GRM5 21 47 CCCCNC(=O)N[C@@H]1C[C@@H](OCC)C1(C)C ZINC000217911550 BE For-Sale Unstable EPHX2 60 43 CC[C@@H](C)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)OC ZINC000217911587 CD For-Sale Unstable MME 31 40 CC[C@@H](C)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)OC ZINC000217911587 CD For-Sale Unstable PAPA1_CARPA 49 37 CC[C@@H](C)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)OC ZINC000217911587 CD For-Sale Unstable PGA 46 37 CC[C@@H](C)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)OC ZINC000217911587 CD For-Sale Unstable ENPEP 62 32 CC[C@@H](C)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)OC ZINC000217911587 CD For-Sale Unstable ACE2 43 36 CC[C@@H](C)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)OC ZINC000217911587 CD For-Sale Unstable POL 0 45 CC[C@@H](C)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)OC ZINC000217911587 CD For-Sale Unstable PENP_PENJA 0 40 COC(=O)C[C@H](c1ccccc1)c1oc(CN2CCOCC2)cc(=O)c1O ZINC000217911615 FD In-Stock Unstable CASR 56 39 CCCCNC(=O)N[C@H]1C[C@@H](OCC)C1(C)C ZINC000217911628 BE For-Sale Unstable EPHX2 60 43 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccc(F)cc2)c1 ZINC000217911644 EI In-Stock Unstable PYGL 21 40 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccc(F)cc2)c1 ZINC000217911644 EI In-Stock Unstable HDAC7 41 36 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccc(F)cc2)c1 ZINC000217911644 EI In-Stock Unstable CRTM 58 48 CC[C@H](C)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)OC ZINC000217911658 CD On-Demand Unstable BMP1 40 33 CC[C@H](C)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)OC ZINC000217911658 CD On-Demand Unstable PAPA1_CARPA 49 37 CC[C@H](C)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)OC ZINC000217911658 CD On-Demand Unstable PGA 41 35 CC[C@H](C)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)OC ZINC000217911658 CD On-Demand Unstable ENPEP 62 32 CC[C@H](C)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)OC ZINC000217911658 CD On-Demand Unstable ACE2 43 36 CC[C@H](C)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)OC ZINC000217911658 CD On-Demand Unstable POL 0 45 CC[C@H](C)[C@@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)OC ZINC000217911658 CD On-Demand Unstable PENP_PENJA 0 40 Cc1ccc(C(=O)N[C@@H]2CCC[C@@H]2CO)cc1Br ZINC000217911702 DF On-Demand Unstable MAPK14 44 43 Cc1ccc(C(=O)N[C@@H]2CCC[C@@H]2CO)cc1Br ZINC000217911702 DF On-Demand Unstable MAPK13 42 39 CCCCNC(=O)N[C@@H]1C[C@H](OCC)C1(C)C ZINC000217911721 BE For-Sale Unstable EPHX2 60 43 COC(=O)C[C@@H](c1ccccc1)c1oc(CN2CCOCC2)cc(=O)c1O ZINC000217911736 FD In-Stock Unstable CASR 56 39 CC(C)Oc1ccc(CCCNC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217911744 EI In-Stock Unstable PYGL 0 40 CC(C)Oc1ccc(CCCNC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217911744 EI In-Stock Unstable HDAC7 41 37 CC(C)Oc1ccc(CCCNC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217911744 EI In-Stock Unstable LEF 58 39 CC[C@@H](C)[C@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)OC ZINC000217911750 CD For-Sale Unstable MME 31 40 CC[C@@H](C)[C@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)OC ZINC000217911750 CD For-Sale Unstable BMP1 40 33 CC[C@@H](C)[C@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)OC ZINC000217911750 CD For-Sale Unstable PAPA1_CARPA 49 37 CC[C@@H](C)[C@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)OC ZINC000217911750 CD For-Sale Unstable PGA 46 37 CC[C@@H](C)[C@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)OC ZINC000217911750 CD For-Sale Unstable ENPEP 62 32 CC[C@@H](C)[C@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)OC ZINC000217911750 CD For-Sale Unstable ACE2 43 36 Cc1ccc(C(=O)N[C@H]2CCC[C@@H]2CO)cc1Br ZINC000217911758 DF For-Sale Unstable MAPK11 31 43 Cc1ccc(C(=O)N[C@H]2CCC[C@@H]2CO)cc1Br ZINC000217911758 DF For-Sale Unstable MAPK14 45 43 Cc1ccc(C(=O)N[C@H]2CCC[C@@H]2CO)cc1Br ZINC000217911758 DF For-Sale Unstable MAPK13 42 39 CCCCNC(=O)N[C@H]1C[C@H](OCC)C1(C)C ZINC000217911832 BE For-Sale Unstable EPHX2 60 43 CC[C@H](C)[C@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)OC ZINC000217911833 CD On-Demand Unstable BMP1 40 33 CC[C@H](C)[C@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)OC ZINC000217911833 CD On-Demand Unstable PAPA1_CARPA 49 37 CC[C@H](C)[C@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)OC ZINC000217911833 CD On-Demand Unstable PGA 41 35 CC[C@H](C)[C@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)OC ZINC000217911833 CD On-Demand Unstable ENPEP 62 32 CC[C@H](C)[C@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)OC ZINC000217911833 CD On-Demand Unstable ACE2 43 36 CC[C@H](C)[C@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)OC ZINC000217911833 CD On-Demand Unstable POL 0 45 CC[C@H](C)[C@H](NC(=O)C[C@@H](N)c1ccccc1)C(=O)OC ZINC000217911833 CD On-Demand Unstable PENP_PENJA 0 40 O=C(/C=C/c1ccc(F)cc1)Nc1ccc(OC2CCCC2)cc1 ZINC000217911840 EJ In-Stock Unstable MMP2 22 60 O=C(/C=C/c1ccc(F)cc1)Nc1ccc(OC2CCCC2)cc1 ZINC000217911840 EJ In-Stock Unstable MMP9 16 60 O=C(/C=C/c1ccc(F)cc1)Nc1ccc(OC2CCCC2)cc1 ZINC000217911840 EJ In-Stock Unstable EPHX2 19 49 O=C(/C=C/c1ccc(F)cc1)Nc1ccc(OC2CCCC2)cc1 ZINC000217911840 EJ In-Stock Unstable MMP1 27 60 O=C(/C=C/c1ccc(F)cc1)Nc1ccc(OC2CCCC2)cc1 ZINC000217911840 EJ In-Stock Unstable MCHR1 0 41 Cc1ccc(C(=O)N[C@@H]2CCC[C@H]2CO)cc1Br ZINC000217911874 DF For-Sale Unstable MAPK11 31 43 Cc1ccc(C(=O)N[C@@H]2CCC[C@H]2CO)cc1Br ZINC000217911874 DF For-Sale Unstable MAPK14 45 43 Cc1ccc(C(=O)N[C@@H]2CCC[C@H]2CO)cc1Br ZINC000217911874 DF For-Sale Unstable MAPK13 42 39 CCCCN(C(=O)Cc1c(C)nc2ccccc2c1-c1ccccc1)[C@@H]1CCS(=O)(=O)C1 ZINC000217911889 JJ On-Demand Unstable TSPO 45 38 CCCOc1ccc(CCC(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217911892 IH For-Sale Unstable FFAR4 40 34 Cc1cccc(/C=C/NC(=O)N2CCN(c3cccc(C)c3C)CC2)c1 ZINC000217911918 EI For-Sale Unstable ABCB1 16 43 Cc1ccc(C(=O)N[C@H]2CCC[C@H]2CO)cc1Br ZINC000217911947 DF For-Sale Unstable MAPK11 31 43 Cc1ccc(C(=O)N[C@H]2CCC[C@H]2CO)cc1Br ZINC000217911947 DF For-Sale Unstable MAPK14 45 43 Cc1ccc(C(=O)N[C@H]2CCC[C@H]2CO)cc1Br ZINC000217911947 DF For-Sale Unstable MAPK13 42 39 CC1(C)C[C@@H](NC(=O)/C=C/c2ccc(F)cc2)c2ccccc2O1 ZINC000217911967 EI In-Stock Unstable TRPV1 0 42 COC(=O)[C@@H]1Cc2[nH]c3ccccc3c2C1 ZINC000217911973 BE In-Stock Unstable PDE5A 25 50 CCCOc1ccc(CCC(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217911995 IH For-Sale Unstable FFAR4 40 34 CCCCN(C(=O)Cc1c(C)nc2ccccc2c1-c1ccccc1)[C@H]1CCS(=O)(=O)C1 ZINC000217911996 JJ On-Demand Unstable TSPO 45 38 CN1CC[C@H](CNC(=O)c2cncc(/C=C\C(=O)O)c2)C1 ZINC000217912008 CC For-Sale Unstable CACNA1I 73 41 Cc1cccc(/C=C/NC(=O)N2CCN(c3ccccc3)CC2)c1 ZINC000217912028 DG For-Sale Unstable FAAH 0 42 COC(=O)[C@H]1Cc2[nH]c3ccccc3c2C1 ZINC000217912037 BE In-Stock Unstable PDE5A 25 50 CC1(C)C[C@H](NC(=O)/C=C/c2ccc(F)cc2)c2ccccc2O1 ZINC000217912043 EI In-Stock Unstable TRPV1 0 42 CCCOc1ccc(CCC(=O)N2C[C@H](Oc3ccccc3F)C[C@H]2C(=O)OC)cc1 ZINC000217912089 IH For-Sale Unstable FFAR4 40 34 COc1ccc(CCN[C@@H]2C[C@@H](C)N(C)C[C@@H]2C)cc1 ZINC000217912124 CF On-Demand Unstable SLC18A2 15 40 CN(CC[S@@](=O)O)C(=O)OCc1ccccc1 ZINC000217912126 CD For-Sale Unstable PAPA1_CARPA 47 38 CN(CC[S@@](=O)O)C(=O)OCc1ccccc1 ZINC000217912126 CD For-Sale Unstable CAPNS1 53 34 CN(CC[S@@](=O)O)C(=O)OCc1ccccc1 ZINC000217912126 CD For-Sale Unstable CAPN2 58 33 CN(CC[S@@](=O)O)C(=O)OCc1ccccc1 ZINC000217912126 CD For-Sale Unstable NPR 67 36 Nc1cccc(/C=C/c2cccc(O)c2)c1 ZINC000217912136 BG Annotated Unstable CA7 15 64 CCCOc1ccc(CCC(=O)N2C[C@@H](Oc3ccccc3F)C[C@H]2C(=O)OC)cc1 ZINC000217912150 IH For-Sale Unstable FFAR4 40 34 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217912175 EH In-Stock Unstable PYGL 0 41 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217912175 EH In-Stock Unstable HDAC9 44 36 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217912175 EH In-Stock Unstable HDAC7 50 36 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217912175 EH In-Stock Unstable LEF 41 34 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217912175 EH In-Stock Unstable TRPM2 0 40 COc1ccc(CCN[C@H]2C[C@@H](C)N(C)C[C@@H]2C)cc1 ZINC000217912217 CF For-Sale Unstable SLC18A2 15 40 Cc1cccc(/C=C/NC(=O)Nc2c(C)cccc2C)c1 ZINC000217912238 CI For-Sale Unstable S1PR4 24 42 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccc(F)cc1 ZINC000217912264 EI In-Stock Unstable HDAC9 44 36 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccc(F)cc1 ZINC000217912264 EI In-Stock Unstable HDAC7 49 36 O=C(O)/C=C\c1cncc(C(=O)NCCn2ccnc2)c1 ZINC000217912281 CC For-Sale Unstable TBXAS1 44 49 O=C(O)/C=C\c1cncc(C(=O)NCCn2ccnc2)c1 ZINC000217912281 CC For-Sale Unstable CYP27B1 46 34 COc1ccc(CCN[C@@H]2C[C@H](C)N(C)C[C@@H]2C)cc1 ZINC000217912313 CF On-Demand Unstable SLC18A2 15 40 COc1ccc([N+](=O)[O-])cc1NC(=O)N/C=C/c1cccc(C)c1 ZINC000217912326 EH For-Sale Unstable CACNA1D 43 34 COc1ccc([N+](=O)[O-])cc1NC(=O)N/C=C/c1cccc(C)c1 ZINC000217912326 EH For-Sale Unstable PYGL 26 40 COc1ccc([N+](=O)[O-])cc1NC(=O)N/C=C/c1cccc(C)c1 ZINC000217912326 EH For-Sale Unstable KCNMA1 27 51 COc1ccc([N+](=O)[O-])cc1NC(=O)N/C=C/c1cccc(C)c1 ZINC000217912326 EH For-Sale Unstable TRPM8 0 55 O=C(O)/C=C\c1cncc(C(=O)Nc2ccccc2Cl)c1 ZINC000217912361 DG For-Sale Anodyne EPHB3 65 40 COc1ccc(CCN[C@H]2C[C@H](C)N(C)C[C@@H]2C)cc1 ZINC000217912378 CF For-Sale Unstable SLC18A2 15 40 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccc(F)cc1 ZINC000217912382 DH In-Stock Unstable SDH1 0 45 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccc(F)cc1 ZINC000217912382 DH In-Stock Unstable CDC25B 0 41 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccc(F)cc1 ZINC000217912382 DH In-Stock Unstable MMP2 19 46 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccc(F)cc1 ZINC000217912382 DH In-Stock Unstable HDAC1 20 42 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccc(F)cc1 ZINC000217912382 DH In-Stock Unstable HDAC2 17 42 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccc(F)cc1 ZINC000217912382 DH In-Stock Unstable MMP9 16 43 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccc(F)cc1 ZINC000217912382 DH In-Stock Unstable MMP1 0 46 OC[C@H]1Cc2sc(Br)cc2CN1 ZINC000217912385 BD For-Sale Unstable PNMT 48 59 C=CCOc1ccccc1C(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217912398 CE For-Sale Unstable HCN1 49 34 C=CCOc1ccccc1C(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217912398 CE For-Sale Unstable HCN4 42 34 OC[C@@H]1Cc2sc(Br)cc2CN1 ZINC000217912447 BD For-Sale Unstable PNMT 48 59 C=CCOc1ccccc1C(=O)N[C@H]1CCC[C@@H]1CO ZINC000217912455 CE For-Sale Unstable HCN1 49 34 C=CCOc1ccccc1C(=O)N[C@H]1CCC[C@@H]1CO ZINC000217912455 CE For-Sale Unstable HCN4 42 34 O=C(O)/C=C\c1cncc(C(=O)Nc2ccccc2F)c1 ZINC000217912471 CF For-Sale Anodyne HDAC1 0 40 Cc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217912484 DH In-Stock Unstable SDH1 0 50 Cc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217912484 DH In-Stock Unstable HDAC8 0 41 Cc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217912484 DH In-Stock Unstable CDC25B 0 42 Cc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217912484 DH In-Stock Unstable HDAC2 17 44 COc1ccc(S(=O)(=O)N(Cc2nn(C)c3c2CCC3)C2CCCC2)cc1 ZINC000217912501 GG In-Stock Unstable AVPR1B 31 51 CN(C)[C@@H]1CCCN(C(=O)CCCCc2ccccc2)CC1 ZINC000217912503 DG In-Stock Unstable SLC18A2 34 40 CN(C)[C@@H]1CCCN(C(=O)CCCCc2ccccc2)CC1 ZINC000217912503 DG In-Stock Unstable HRH3 0 40 CN(C)[C@@H]1CCCN(C(=O)CCCCc2ccccc2)CC1 ZINC000217912503 DG In-Stock Unstable SIGMAR1 23 45 CN(C)[C@@H]1CCCN(C(=O)CCCCc2ccccc2)CC1 ZINC000217912503 DG In-Stock Unstable TRY1_BOVIN 0 46 CN(C)[C@@H]1CCCN(C(=O)CCCCc2ccccc2)CC1 ZINC000217912503 DG In-Stock Unstable C3AR1 40 37 CN(C)[C@@H]1CCCN(C(=O)CCCCc2ccccc2)CC1 ZINC000217912503 DG In-Stock Unstable PREP 88 51 CN(C)[C@@H]1CCCN(C(=O)CCCCc2ccccc2)CC1 ZINC000217912503 DG In-Stock Unstable FAAH 53 41 CN(C)[C@@H]1CCCN(C(=O)CCCCc2ccccc2)CC1 ZINC000217912503 DG In-Stock Unstable CES1 51 37 C=CCOc1ccccc1C(=O)N[C@@H]1CCC[C@H]1CO ZINC000217912536 CE For-Sale Unstable HCN1 49 34 C=CCOc1ccccc1C(=O)N[C@@H]1CCC[C@H]1CO ZINC000217912536 CE For-Sale Unstable HCN4 42 34 Cc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217912557 DH In-Stock Unstable SDH1 0 50 Cc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217912557 DH In-Stock Unstable HDAC8 0 41 Cc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217912557 DH In-Stock Unstable CDC25B 0 42 Cc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217912557 DH In-Stock Unstable HDAC2 17 44 CN(C)[C@H]1CCCN(C(=O)CCCCc2ccccc2)CC1 ZINC000217912598 DG In-Stock Unstable SLC18A2 34 40 CN(C)[C@H]1CCCN(C(=O)CCCCc2ccccc2)CC1 ZINC000217912598 DG In-Stock Unstable HRH3 0 40 CN(C)[C@H]1CCCN(C(=O)CCCCc2ccccc2)CC1 ZINC000217912598 DG In-Stock Unstable SIGMAR1 23 45 CN(C)[C@H]1CCCN(C(=O)CCCCc2ccccc2)CC1 ZINC000217912598 DG In-Stock Unstable TRY1_BOVIN 0 46 CN(C)[C@H]1CCCN(C(=O)CCCCc2ccccc2)CC1 ZINC000217912598 DG In-Stock Unstable C3AR1 40 37 CN(C)[C@H]1CCCN(C(=O)CCCCc2ccccc2)CC1 ZINC000217912598 DG In-Stock Unstable PREP 88 51 CN(C)[C@H]1CCCN(C(=O)CCCCc2ccccc2)CC1 ZINC000217912598 DG In-Stock Unstable FAAH 53 41 CN(C)[C@H]1CCCN(C(=O)CCCCc2ccccc2)CC1 ZINC000217912598 DG In-Stock Unstable CES1 51 37 C=CCOc1ccccc1C(=O)N[C@H]1CCC[C@H]1CO ZINC000217912629 CE For-Sale Unstable HCN1 49 34 C=CCOc1ccccc1C(=O)N[C@H]1CCC[C@H]1CO ZINC000217912629 CE For-Sale Unstable HCN4 42 34 CC1CCN(c2ccc([C@@H](C)NC(=O)/C=C/c3ccc(F)cc3)cc2)CC1 ZINC000217912673 FJ In-Stock Unstable KCNQ2 50 38 CSc1ccc(C(=O)N2CCCO[C@@H](CN3CCCCC3)C2)cc1 ZINC000217912701 EG In-Stock Unstable L3MBTL3 53 37 CCN(C(=O)N/C=C/c1cccc(C)c1)c1cccc(C)c1 ZINC000217912705 CJ For-Sale Unstable NR1H4 47 41 Nc1ccc2[nH]c3c(c2c1)C[C@H](C(=O)O)C3 ZINC000217912723 BD In-Stock Unstable NGFR 0 44 CC1CCN(c2ccc([C@H](C)NC(=O)/C=C/c3ccc(F)cc3)cc2)CC1 ZINC000217912741 FJ In-Stock Unstable KCNQ2 50 38 CSc1ccc(C(=O)N2CCCO[C@H](CN3CCCCC3)C2)cc1 ZINC000217912788 EG In-Stock Unstable L3MBTL3 53 37 Nc1ccc2[nH]c3c(c2c1)C[C@@H](C(=O)O)C3 ZINC000217912805 BD In-Stock Unstable NGFR 0 44 CCCCN(C(=O)c1ccc(=O)n(Cc2ccccc2Cl)c1)[C@@H]1CCS(=O)(=O)C1 ZINC000217912823 IF On-Demand Unstable MBTPS1 60 37 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)/C=C/c3ccc(F)cc3)cc2)C1 ZINC000217912869 FJ In-Stock Unstable KCNQ2 49 38 CCCCN(C(=O)c1ccc(=O)n(Cc2ccccc2Cl)c1)[C@H]1CCS(=O)(=O)C1 ZINC000217912919 IF On-Demand Unstable MBTPS1 60 37 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCc1ccc(Cl)cc1Cl ZINC000217912936 II For-Sale Unstable MC4R 19 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCc1ccc(Cl)cc1Cl ZINC000217912936 II For-Sale Unstable P2RX7 40 38 C[C@H](NC(=O)/C=C/c1ccc(F)cc1)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217912954 FJ In-Stock Unstable KCNQ2 49 38 O=C(COc1ncnc2ccccc12)NCCc1noc([C@@H]2CCCO2)n1 ZINC000217913014 FD In-Stock Unstable SMO 46 35 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCc1ccc(Cl)cc1Cl ZINC000217913017 II For-Sale Unstable MC4R 19 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCc1ccc(Cl)cc1Cl ZINC000217913017 II For-Sale Unstable P2RX7 40 38 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)NCC3CCOCC3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217913051 KF In-Stock Unstable TUBA1A 18 68 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)NCC3CCOCC3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217913051 KF In-Stock Unstable TPPP 0 64 Cc1ccc2c(c1)[C@@H](NC(=O)/C=C/c1ccc(F)cc1)CC(C)(C)O2 ZINC000217913057 EJ In-Stock Unstable TRPV1 0 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCc1ccc(Cl)cc1Cl ZINC000217913086 II For-Sale Unstable MC4R 19 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCc1ccc(Cl)cc1Cl ZINC000217913086 II For-Sale Unstable P2RX7 40 38 O=C(COc1ncnc2ccccc12)NCCc1noc([C@H]2CCCO2)n1 ZINC000217913091 FD In-Stock Unstable SMO 46 35 Cc1cccc(/C=C/NC(=O)N2CCN(c3ccccc3F)CC2)c1 ZINC000217913097 EH For-Sale Unstable NPY2R 46 34 CN1CC[C@@H](NC(=O)NC2CCC2)C1=O ZINC000217913122 BC On-Demand Unstable EPHX2 24 47 Cc1ccc2c(c1)[C@H](NC(=O)/C=C/c1ccc(F)cc1)CC(C)(C)O2 ZINC000217913136 EJ In-Stock Unstable TRPV1 0 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCc1ccc(Cl)cc1Cl ZINC000217913149 II For-Sale Unstable MC4R 19 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCc1ccc(Cl)cc1Cl ZINC000217913149 II For-Sale Unstable P2RX7 40 38 CN1CC[C@H](NC(=O)NC2CCC2)C1=O ZINC000217913185 BC On-Demand Unstable EPHX2 24 47 Cc1cccc(C(=O)NCC[C@H](O)C2CCOCC2)c1 ZINC000217913234 CD In-Stock Unstable DRD4 43 36 Cc1cccc(C(=O)NCC[C@H](O)C2CCOCC2)c1 ZINC000217913234 CD In-Stock Unstable KCNK3 48 43 Cc1cccc(C(=O)NCC[C@H](O)C2CCOCC2)c1 ZINC000217913234 CD In-Stock Unstable KCNK9 48 43 Cc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)/C=C/c1ccc(F)cc1 ZINC000217913239 EJ In-Stock Unstable TRPV1 0 46 O=C(O)/C=C\c1cncc(C(=O)NCCc2cccs2)c1 ZINC000217913300 DE For-Sale Unstable ADAM17 0 40 Cc1cccc(C(=O)NCC[C@@H](O)C2CCOCC2)c1 ZINC000217913301 CD In-Stock Unstable DRD4 43 36 Cc1cccc(C(=O)NCC[C@@H](O)C2CCOCC2)c1 ZINC000217913301 CD In-Stock Unstable KCNK3 48 43 Cc1cccc(C(=O)NCC[C@@H](O)C2CCOCC2)c1 ZINC000217913301 CD In-Stock Unstable KCNK9 48 43 Cc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)/C=C/c1ccc(F)cc1 ZINC000217913312 EJ In-Stock Unstable TRPV1 0 46 CCO[C@@H]1C[C@@H](NC(=O)NC2CCC2)C1(C)C ZINC000217913328 BE For-Sale Unstable EPHX2 23 41 COC(=O)[C@H](CCSC)NC(=O)CCc1c(C)c2cc3c4c(oc3c(C)c2oc1=O)CCCC4 ZINC000217913345 JI In-Stock Unstable IMPDH1 0 45 CCO[C@H]1C[C@@H](NC(=O)NC2CCC2)C1(C)C ZINC000217913404 BE For-Sale Unstable EPHX2 23 41 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](CC(C)C)C(=O)NCCCO)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217913459 KG In-Stock Unstable TUBA1A 18 67 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](CC(C)C)C(=O)NCCCO)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217913459 KG In-Stock Unstable TPPP 0 63 CCO[C@@H]1C[C@H](NC(=O)NC2CCC2)C1(C)C ZINC000217913493 BE For-Sale Unstable EPHX2 23 41 CCOc1ccccc1[C@@H](C)N[C@@H]1CCCN(CC)C1 ZINC000217913497 CG On-Demand Unstable HCN1 44 35 CCOc1ccccc1[C@@H](C)N[C@@H]1CCCN(CC)C1 ZINC000217913497 CG On-Demand Unstable HCN4 43 35 Cc1cccc(/C=C/NC(=O)Nc2ccc(Br)c(C)c2)c1 ZINC000217913520 EJ For-Sale Unstable KCNK3 48 36 COCCCN(C)C(=O)N1[C@H](C(=O)O)C[C@@H]2CCCC[C@@H]21 ZINC000217913558 CD For-Sale Unstable ACE 15 55 CCO[C@H]1C[C@H](NC(=O)NC2CCC2)C1(C)C ZINC000217913562 BE For-Sale Unstable EPHX2 23 41 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)/C=C/c1ccc(F)cc1 ZINC000217913576 FI In-Stock Unstable TRPV1 0 44 CCOc1ccccc1[C@@H](C)N[C@H]1CCCN(CC)C1 ZINC000217913577 CG On-Demand Unstable HCN1 44 35 CCOc1ccccc1[C@@H](C)N[C@H]1CCCN(CC)C1 ZINC000217913577 CG On-Demand Unstable HCN4 43 35 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCc1ccc(Cl)c(Cl)c1 ZINC000217913583 II For-Sale Unstable OPRK1 16 40 COCCCN(C)C(=O)N1[C@H](C(=O)O)C[C@H]2CCCC[C@@H]21 ZINC000217913643 CD For-Sale Unstable ACE 15 55 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)/C=C/c1ccc(F)cc1 ZINC000217913653 FI In-Stock Unstable TRPV1 0 44 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCc1ccc(Cl)c(Cl)c1 ZINC000217913657 II For-Sale Unstable OPRK1 16 40 CCN(CCNC(=O)c1cc(N)cc(Cl)c1)C1CC1 ZINC000217913670 CE For-Sale Unstable CACNA1I 62 37 O=C(O)/C(S)=C/c1ccoc1 ZINC000217913682 AD For-Sale Anodyne CAPN1 61 52 CC[C@@H]1C[C@@H]1NC(=O)NC1CCC1 ZINC000217913683 AD For-Sale Unstable EPHX2 19 50 O=C(O)/C=C\c1cccc(CSCCCO)c1 ZINC000217913730 CE For-Sale Unstable LTB4R 18 44 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCc1ccc(Cl)c(Cl)c1 ZINC000217913740 II For-Sale Unstable OPRK1 16 40 CC[C@H]1C[C@@H]1NC(=O)NC1CCC1 ZINC000217913743 AD For-Sale Unstable EPHX2 19 50 CC[C@@H](NC(=O)/C=C/c1ccc(F)cc1)c1ccc(C)c(C)c1 ZINC000217913784 DJ In-Stock Unstable LEF 52 40 CCN(CCNC(=O)c1cccc(Cl)c1N)C1CC1 ZINC000217913807 CE For-Sale Unstable ECR 43 33 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCc1ccc(Cl)c(Cl)c1 ZINC000217913820 II For-Sale Unstable OPRK1 16 40 CC[C@@H]1C[C@H]1NC(=O)NC1CCC1 ZINC000217913846 AD On-Demand Unstable EPHX2 17 50 CC[C@H](NC(=O)/C=C/c1ccc(F)cc1)c1ccc(C)c(C)c1 ZINC000217913888 DJ In-Stock Unstable LEF 52 40 CC[C@H]1C[C@H]1NC(=O)NC1CCC1 ZINC000217913909 AD For-Sale Unstable EPHX2 19 50 Cc1cccc(NC(=O)c2cncc(/C=C\C(=O)O)c2)n1 ZINC000217913943 CE For-Sale Unstable GRM5 26 51 Cc1cccc(NC(=O)c2cncc(/C=C\C(=O)O)c2)n1 ZINC000217913943 CE For-Sale Unstable SORT1 23 46 C[C@H]1CN(C)[C@@H](C)C[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000217913990 DD For-Sale Unstable CA2 71 44 C[C@H]1CN(C)[C@@H](C)C[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000217913990 DD For-Sale Unstable CA6 17 42 C[C@H]1CN(C)[C@@H](C)C[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000217913990 DD For-Sale Unstable CA1 63 42 C[C@H]1CN(C)[C@@H](C)C[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000217913990 DD For-Sale Unstable CA7 47 42 C[C@H]1CN(C)[C@@H](C)C[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000217913990 DD For-Sale Unstable CA13 18 42 C[C@H]1CN(C)[C@@H](C)C[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000217913990 DD For-Sale Unstable CA5B 31 42 C[C@H]1CN(C)[C@@H](C)C[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000217913990 DD For-Sale Unstable CA4 41 42 C[C@H]1CN(C)[C@@H](C)C[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000217913990 DD For-Sale Unstable CA14 32 41 C[C@H]1CN(C)[C@@H](C)C[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000217913990 DD For-Sale Unstable CA12 51 43 C[C@H]1CN(C)[C@@H](C)C[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000217913990 DD For-Sale Unstable CA9 58 43 C[C@H]1CN(C)[C@@H](C)C[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000217913990 DD For-Sale Unstable CAH_METTE 24 42 C[C@H]1CN(C)[C@@H](C)C[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000217913990 DD For-Sale Unstable CYNT 39 40 C[C@H]1CN(C)[C@@H](C)C[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000217913990 DD For-Sale Unstable NCE103 16 42 C[C@H]1CN(C)[C@@H](C)C[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000217913990 DD For-Sale Unstable CA15 16 42 C[C@H]1CN(C)[C@@H](C)C[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000217913990 DD For-Sale Unstable MTCA1 24 42 C[C@H]1CN(C)[C@@H](C)C[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000217913990 DD For-Sale Unstable CA 0 42 C[C@H]1CN(C)[C@@H](C)C[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000217913990 DD For-Sale Unstable A6YCJ1_9METZ 23 42 C[C@H]1CN(C)[C@@H](C)C[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000217913990 DD For-Sale Unstable Q5TU56_ANOGA 0 42 COC(=O)[C@H](CC(C)C)NC(=O)c1cn(C)c(=O)c2ccccc12 ZINC000217913999 ED In-Stock Unstable FOLH1 47 37 COC(=O)[C@H](CC(C)C)NC(=O)c1cn(C)c(=O)c2ccccc12 ZINC000217913999 ED In-Stock Unstable CAPNS1 47 36 COC(=O)[C@H](CC(C)C)NC(=O)c1cn(C)c(=O)c2ccccc12 ZINC000217913999 ED In-Stock Unstable CAPN1 52 38 COC(=O)[C@H](CC(C)C)NC(=O)c1cn(C)c(=O)c2ccccc12 ZINC000217913999 ED In-Stock Unstable CAPN2 75 34 COC(=O)[C@H](CC(C)C)NC(=O)c1cn(C)c(=O)c2ccccc12 ZINC000217913999 ED In-Stock Unstable NPR 67 36 Cc1cccc(NC(=O)c2cncc(/C=C\C(=O)O)c2)c1 ZINC000217914003 CF For-Sale Unstable KIT 21 43 Cc1cccc(NC(=O)c2cncc(/C=C\C(=O)O)c2)c1 ZINC000217914003 CF For-Sale Unstable KDR 19 43 Cc1cccc(NC(=O)c2cncc(/C=C\C(=O)O)c2)c1 ZINC000217914003 CF For-Sale Unstable SCN10A 50 46 Cc1cccc(NC(=O)c2cncc(/C=C\C(=O)O)c2)c1 ZINC000217914003 CF For-Sale Unstable CSF1R 24 46 Cc1cccc(NC(=O)c2cncc(/C=C\C(=O)O)c2)c1 ZINC000217914003 CF For-Sale Unstable TAAR1 31 41 Cc1cccc(NC(=O)c2cncc(/C=C\C(=O)O)c2)c1 ZINC000217914003 CF For-Sale Unstable DDR1 28 43 Cc1cccc(NC(=O)c2cncc(/C=C\C(=O)O)c2)c1 ZINC000217914003 CF For-Sale Unstable KCNK3 123 51 Cc1cccc(NC(=O)c2cncc(/C=C\C(=O)O)c2)c1 ZINC000217914003 CF For-Sale Unstable KCNK9 70 51 O=C(O)/C=C\c1ccccc1CSCCCO ZINC000217914040 CE For-Sale Unstable PTGER2 44 50 O=C(O)/C=C\c1ccccc1CSCCCO ZINC000217914040 CE For-Sale Unstable PTGER4 21 50 O=C(O)/C=C\c1ccccc1CSCCCO ZINC000217914040 CE For-Sale Unstable PTGER3 19 50 O=C(O)/C=C\c1ccccc1CSCCCO ZINC000217914040 CE For-Sale Unstable PTGDR 18 48 CC1CCN(C(=O)c2cncc(/C=C\C(=O)O)c2)CC1 ZINC000217914093 CE For-Sale Unstable L3MBTL3 41 33 CC1CCN(C(=O)c2cncc(/C=C\C(=O)O)c2)CC1 ZINC000217914093 CE For-Sale Unstable TRPC6 40 34 O=C1C[C@@H](c2ccc(-c3ccc(C(=O)O)cc3)o2)c2c(c3ccccc3oc2=O)O1 ZINC000217914110 HI In-Stock Unstable VKORC1 0 40 O=C1C[C@@H](c2ccc(-c3ccc(C(=O)O)cc3)o2)c2c(c3ccccc3oc2=O)O1 ZINC000217914110 HI In-Stock Unstable TNKS 28 47 N=C(O[C@H]1O[C@H](COCc2ccccc2)[C@@H](OCc2ccccc2)[C@@H](OCc2ccccc2)[C@@H]1OCc1ccccc1)C(Cl)(Cl)Cl ZINC000217914137 KK For-Sale Unstable SSTR2 21 49 N=C(O[C@H]1O[C@H](COCc2ccccc2)[C@@H](OCc2ccccc2)[C@@H](OCc2ccccc2)[C@@H]1OCc1ccccc1)C(Cl)(Cl)Cl ZINC000217914137 KK For-Sale Unstable TACR2 19 41 Cc1ccc(CN[C@@H]2CCCN(C(=O)OC(C)(C)C)C2)cn1 ZINC000217914142 DF On-Demand Unstable GPR119 40 39 O=C1C[C@H](c2ccc(-c3ccc(C(=O)O)cc3)o2)c2c(c3ccccc3oc2=O)O1 ZINC000217914180 HI In-Stock Unstable VKORC1 0 40 O=C1C[C@H](c2ccc(-c3ccc(C(=O)O)cc3)o2)c2c(c3ccccc3oc2=O)O1 ZINC000217914180 HI In-Stock Unstable TNKS 28 47 Cc1cccc(/C=C/NC(=O)NC2CCN(Cc3ccccc3)CC2)c1 ZINC000217914261 EH For-Sale Unstable CHRM2 25 51 Cc1cccc(/C=C/NC(=O)NC2CCN(Cc3ccccc3)CC2)c1 ZINC000217914261 EH For-Sale Unstable CHRM1 16 57 Cc1cccc(/C=C/NC(=O)NC2CCN(Cc3ccccc3)CC2)c1 ZINC000217914261 EH For-Sale Unstable DRD2 28 55 Cc1cccc(/C=C/NC(=O)NC2CCN(Cc3ccccc3)CC2)c1 ZINC000217914261 EH For-Sale Unstable DRD4 65 58 Cc1cccc(/C=C/NC(=O)NC2CCN(Cc3ccccc3)CC2)c1 ZINC000217914261 EH For-Sale Unstable ACHE 45 48 Cc1cccc(/C=C/NC(=O)NC2CCN(Cc3ccccc3)CC2)c1 ZINC000217914261 EH For-Sale Unstable HRH2 29 41 Cc1cccc(/C=C/NC(=O)NC2CCN(Cc3ccccc3)CC2)c1 ZINC000217914261 EH For-Sale Unstable DRD3 28 55 Cc1cccc(/C=C/NC(=O)NC2CCN(Cc3ccccc3)CC2)c1 ZINC000217914261 EH For-Sale Unstable KCNH2 17 41 Cc1cccc(/C=C/NC(=O)NC2CCN(Cc3ccccc3)CC2)c1 ZINC000217914261 EH For-Sale Unstable CHRM3 35 57 Cc1cccc(/C=C/NC(=O)NC2CCN(Cc3ccccc3)CC2)c1 ZINC000217914261 EH For-Sale Unstable SIGMAR1 57 60 Cc1cccc(/C=C/NC(=O)NC2CCN(Cc3ccccc3)CC2)c1 ZINC000217914261 EH For-Sale Unstable SSTR5 58 39 Cc1cccc(/C=C/NC(=O)NC2CCN(Cc3ccccc3)CC2)c1 ZINC000217914261 EH For-Sale Unstable CCR3 52 46 Cc1cccc(/C=C/NC(=O)NC2CCN(Cc3ccccc3)CC2)c1 ZINC000217914261 EH For-Sale Unstable EPHX2 22 49 Cc1cccc(/C=C/NC(=O)NC2CCN(Cc3ccccc3)CC2)c1 ZINC000217914261 EH For-Sale Unstable CXCR3 31 40 Cc1cccc(/C=C/NC(=O)NC2CCN(Cc3ccccc3)CC2)c1 ZINC000217914261 EH For-Sale Unstable MCHR1 61 48 Cc1cccc(/C=C/NC(=O)NC2CCN(Cc3ccccc3)CC2)c1 ZINC000217914261 EH For-Sale Unstable CACNA1G 27 41 Cc1cccc(/C=C/NC(=O)NC2CCN(Cc3ccccc3)CC2)c1 ZINC000217914261 EH For-Sale Unstable CCR8 24 46 Cc1cccc(/C=C/NC(=O)NC2CCN(Cc3ccccc3)CC2)c1 ZINC000217914261 EH For-Sale Unstable ADIPOR1 0 42 Cc1cccc(/C=C/NC(=O)NC2CCN(Cc3ccccc3)CC2)c1 ZINC000217914261 EH For-Sale Unstable ADIPOR2 0 42 Cn1nc(CC(=O)N2CCn3nc(CO)cc3C2)c2ccccc2c1=O ZINC000217914267 FC In-Stock Unstable IMDH_CRYPV 28 42 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(OC)c(OC(C)C)c2)CC(=O)O4)cc1O ZINC000217914298 KK In-Stock Unstable AKR1B1 0 48 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(OC)c(OC(C)C)c2)CC(=O)O4)cc1O ZINC000217914298 KK In-Stock Unstable CYP1B1 57 36 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(OC)c(OC(C)C)c2)CC(=O)O4)cc1O ZINC000217914298 KK In-Stock Unstable CYP1A1 42 46 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccc(OC)c(OC(C)C)c2)CC(=O)O4)cc1O ZINC000217914298 KK In-Stock Unstable CYP1A2 33 41 Cc1cccc(/C=C/NC(=O)N2CCN(C(=O)c3ccco3)CC2)c1 ZINC000217914366 EF For-Sale Unstable ALDH1A1 17 45 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(OC)c(OC(C)C)c2)CC(=O)O4)cc1O ZINC000217914388 KK In-Stock Unstable AKR1B1 0 48 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(OC)c(OC(C)C)c2)CC(=O)O4)cc1O ZINC000217914388 KK In-Stock Unstable CYP1B1 57 36 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(OC)c(OC(C)C)c2)CC(=O)O4)cc1O ZINC000217914388 KK In-Stock Unstable CYP1A1 42 46 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccc(OC)c(OC(C)C)c2)CC(=O)O4)cc1O ZINC000217914388 KK In-Stock Unstable CYP1A2 33 41 CC[C@@H](NC(=O)/C=C/c1ccc(F)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217914411 FH In-Stock Unstable PTGS2 26 42 CC[C@@H](NC(=O)/C=C/c1ccc(F)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217914411 FH In-Stock Unstable CTSF 44 32 O=C(O)C[C@H](CN1CCC[C@@H](c2cccc(C(F)(F)F)c2)C1)C(F)(F)F ZINC000217914426 GJ For-Sale Unstable CCR2 70 39 O=C(O)C[C@H](CN1CCC[C@@H](c2cccc(C(F)(F)F)c2)C1)C(F)(F)F ZINC000217914426 GJ For-Sale Unstable LIPG 49 33 Cc1onc(-c2ccccc2Cl)c1C(=O)Nc1nc(CN2C[C@H](C)O[C@H](C)C2)cs1 ZINC000217914484 IJ On-Demand Unstable GHSR 17 50 Cc1onc(-c2ccccc2Cl)c1C(=O)Nc1nc(CN2C[C@H](C)O[C@H](C)C2)cs1 ZINC000217914484 IJ On-Demand Unstable GPBAR1 27 41 CC[C@H](NC(=O)/C=C/c1ccc(F)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217914488 FH In-Stock Unstable PTGS2 26 42 CC[C@H](NC(=O)/C=C/c1ccc(F)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217914488 FH In-Stock Unstable CTSF 44 32 C#CCOc1ccc(CN2CCC(N)CC2)cc1 ZINC000217914534 BD For-Sale Unstable LTA4H 47 44 C#CCOc1ccc(CN2CCC(N)CC2)cc1 ZINC000217914534 BD For-Sale Unstable HRH3 29 51 C#CCOc1ccc(CN2CCC(N)CC2)cc1 ZINC000217914534 BD For-Sale Unstable SIGMAR1 40 51 C#CCOc1ccc(CN2CCC(N)CC2)cc1 ZINC000217914534 BD For-Sale Unstable CHEK2 29 40 Cc1onc(-c2ccccc2Cl)c1C(=O)Nc1nc(CN2C[C@H](C)O[C@@H](C)C2)cs1 ZINC000217914568 IJ On-Demand Unstable GHSR 17 50 Cc1onc(-c2ccccc2Cl)c1C(=O)Nc1nc(CN2C[C@H](C)O[C@@H](C)C2)cs1 ZINC000217914568 IJ On-Demand Unstable GPBAR1 27 41 Cc1ccc(-c2noc(CNC(=O)/C=C/c3ccc(F)cc3)n2)cc1 ZINC000217914602 EH In-Stock Unstable HDAC8 0 51 Cc1ccc(-c2noc(CNC(=O)/C=C/c3ccc(F)cc3)n2)cc1 ZINC000217914602 EH In-Stock Unstable HDAC2 15 42 Cc1cccc(/C=C/NC(=O)N2CCN(Cc3ccc4c(c3)OCO4)CC2)c1 ZINC000217914605 GG For-Sale Unstable DRD4 21 48 Cc1cccc(/C=C/NC(=O)N2CCN(Cc3ccc4c(c3)OCO4)CC2)c1 ZINC000217914605 GG For-Sale Unstable SSTR3 70 32 Cc1cccc(/C=C/NC(=O)N2CCN(Cc3ccc4c(c3)OCO4)CC2)c1 ZINC000217914605 GG For-Sale Unstable MCHR1 26 45 NC[C@H](c1ccc(Cl)s1)N1CCC[C@@H]1c1cccnc1 ZINC000217914613 DH For-Sale Unstable CHRNA2 46 47 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCc1c(OC)ccc2ccccc12 ZINC000217914646 JI For-Sale Unstable AGTR2 44 33 Cc1onc(-c2ccccc2Cl)c1C(=O)Nc1nc(CN2C[C@@H](C)O[C@H](C)C2)cs1 ZINC000217914661 IJ On-Demand Unstable GHSR 17 50 Cc1onc(-c2ccccc2Cl)c1C(=O)Nc1nc(CN2C[C@@H](C)O[C@H](C)C2)cs1 ZINC000217914661 IJ On-Demand Unstable GPBAR1 27 41 O=C(c1cncc(O)c1)N1CCCS(=O)(=O)CC1 ZINC000217914673 CC For-Sale Unstable L3MBTL1 0 40 COc1cc(CN2CC[C@@H]3[C@@H](CCCN3C)C2)ccc1O ZINC000217914700 CE On-Demand Unstable SSTR5 57 37 COc1cccc(-c2noc(CNC(=O)/C=C/c3ccc(F)cc3)n2)c1 ZINC000217914721 FG In-Stock Unstable HDAC8 35 40 COc1cccc(-c2noc(CNC(=O)/C=C/c3ccc(F)cc3)n2)c1 ZINC000217914721 FG In-Stock Unstable HDAC1 0 41 COc1cccc(-c2noc(CNC(=O)/C=C/c3ccc(F)cc3)n2)c1 ZINC000217914721 FG In-Stock Unstable HDAC6 30 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCc1c(OC)ccc2ccccc12 ZINC000217914726 JI For-Sale Unstable AGTR2 44 33 CCOC(=O)N1CCN(C(=O)N/C=C/c2cccc(C)c2)CC1 ZINC000217914738 DE For-Sale Unstable P2RY12 60 41 O=C(CCc1ccccc1)NCC[C@H](O)C1CCOCC1 ZINC000217914744 CD In-Stock Unstable PAM 0 40 O=C(O)/C=C\c1cncc(C(=O)Nc2ccccc2)c1 ZINC000217914770 CE For-Sale Anodyne PRNP 26 40 O=C(O)/C=C\c1cncc(C(=O)Nc2ccccc2)c1 ZINC000217914770 CE For-Sale Anodyne ATR 47 34 O=C(O)/C=C\c1cncc(C(=O)Nc2ccccc2)c1 ZINC000217914770 CE For-Sale Anodyne KCNK3 99 45 O=C(O)/C=C\c1cncc(C(=O)Nc2ccccc2)c1 ZINC000217914770 CE For-Sale Anodyne KCNK9 52 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCc1c(OC)ccc2ccccc12 ZINC000217914804 JI For-Sale Unstable AGTR2 44 33 O=C(CCc1ccccc1)NCC[C@@H](O)C1CCOCC1 ZINC000217914821 CD In-Stock Unstable PAM 0 40 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccc(F)cc3)n2)cc1 ZINC000217914833 FG In-Stock Unstable HDAC8 0 52 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccc(F)cc3)n2)cc1 ZINC000217914833 FG In-Stock Unstable HDAC2 17 43 CCOC(=O)c1ccc(=O)n(-c2ccc(CN3CCC(N)CC3)cc2)c1 ZINC000217914851 FD For-Sale Unstable SSTR5 41 34 CCOC(=O)c1ccc(=O)n(-c2ccc(CN3CCC(N)CC3)cc2)c1 ZINC000217914851 FD For-Sale Unstable NOD2 17 40 Cc1ccc2nc([C@@H]3CCCN3C(=O)C(=O)c3ccco3)[nH]c2c1 ZINC000217914854 DG In-Stock Unstable PRCP 27 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCc1c(OC)ccc2ccccc12 ZINC000217914883 JI For-Sale Unstable AGTR2 44 33 Cc1ccc2nc([C@H]3CCCN3C(=O)C(=O)c3ccco3)[nH]c2c1 ZINC000217914920 DG In-Stock Unstable PRCP 27 40 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccc(F)cc3)n2)c(OC)c1 ZINC000217914952 GG In-Stock Unstable ABCG2 16 41 O=C(/C=C/c1ccc(F)cc1)NCc1nc(-c2ccccc2Cl)no1 ZINC000217915049 FH In-Stock Unstable GPBAR1 20 41 Cc1cccc(/C=C/NC(=O)Nc2ccc(C(F)(F)F)cc2)c1 ZINC000217915051 DJ For-Sale Unstable DHODH 30 40 Cc1cccc(/C=C/NC(=O)Nc2ccc(C(F)(F)F)cc2)c1 ZINC000217915051 DJ For-Sale Unstable TRPV1 20 42 Cc1cccc(/C=C/NC(=O)Nc2ccc(C(F)(F)F)cc2)c1 ZINC000217915051 DJ For-Sale Unstable EPHX2 28 42 Cc1cccc(/C=C/NC(=O)Nc2ccc(C(F)(F)F)cc2)c1 ZINC000217915051 DJ For-Sale Unstable KCNK3 41 35 C[C@H]1CN(C)[C@@H](C)C[C@@H]1Nc1ccc(C(N)=O)cc1 ZINC000217915078 CD For-Sale Unstable BRD4 0 40 C[C@H]1CN(C)[C@@H](C)C[C@@H]1Nc1ccc(C(N)=O)cc1 ZINC000217915078 CD For-Sale Unstable BRD2 29 40 C[C@H]1CN(C)[C@@H](C)C[C@@H]1Nc1ccc(C(N)=O)cc1 ZINC000217915078 CD For-Sale Unstable BRD3 28 40 C[C@@H](Cc1ccc(F)cc1)NC(=O)N[C@@H](C(=O)O)[C@H](C)O ZINC000217915084 CC For-Sale Unstable ACE 21 40 C[C@@H](Cc1ccc(F)cc1)NC(=O)N[C@@H](C(=O)O)[C@H](C)O ZINC000217915084 CC For-Sale Unstable MME 58 47 C[C@@H](Cc1ccc(F)cc1)NC(=O)N[C@@H](C(=O)O)[C@H](C)O ZINC000217915084 CC For-Sale Unstable CPA1 24 43 C[C@@H](Cc1ccc(F)cc1)NC(=O)N[C@@H](C(=O)O)[C@H](C)O ZINC000217915084 CC For-Sale Unstable ACE2 47 39 CC[C@@H](C)[C@@H](CO)NC(=O)CCc1c[nH]c2ccccc12 ZINC000217915096 CF In-Stock Unstable EDNRB 41 42 CC[C@@H](C)[C@@H](CO)NC(=O)CCc1c[nH]c2ccccc12 ZINC000217915096 CF In-Stock Unstable EDNRA 67 43 CC[C@@H](C)[C@@H](CO)NC(=O)CCc1c[nH]c2ccccc12 ZINC000217915096 CF In-Stock Unstable TACR1 49 45 CC[C@@H](C)[C@@H](CO)NC(=O)CCc1c[nH]c2ccccc12 ZINC000217915096 CF In-Stock Unstable MC4R 45 38 CC[C@@H](C)[C@@H](CO)NC(=O)CCc1c[nH]c2ccccc12 ZINC000217915096 CF In-Stock Unstable BMP1 27 43 CC[C@@H](C)[C@@H](CO)NC(=O)CCc1c[nH]c2ccccc12 ZINC000217915096 CF In-Stock Unstable TACR2 25 40 CC[C@@H](C)[C@@H](CO)NC(=O)CCc1c[nH]c2ccccc12 ZINC000217915096 CF In-Stock Unstable CTSL 33 49 CC[C@@H](C)[C@@H](CO)NC(=O)CCc1c[nH]c2ccccc12 ZINC000217915096 CF In-Stock Unstable BRS3 41 44 CC[C@@H](C)[C@@H](CO)NC(=O)CCc1c[nH]c2ccccc12 ZINC000217915096 CF In-Stock Unstable MMP8 51 39 CC[C@@H](C)[C@@H](CO)NC(=O)CCc1c[nH]c2ccccc12 ZINC000217915096 CF In-Stock Unstable MMP14 82 40 CC[C@@H](C)[C@@H](CO)NC(=O)CCc1c[nH]c2ccccc12 ZINC000217915096 CF In-Stock Unstable GHSR 26 40 CC[C@@H](C)[C@@H](CO)NC(=O)CCc1c[nH]c2ccccc12 ZINC000217915096 CF In-Stock Unstable MMP9 0 44 CC[C@@H](C)[C@@H](CO)NC(=O)CCc1c[nH]c2ccccc12 ZINC000217915096 CF In-Stock Unstable MMP1 0 43 CC[C@@H](C)[C@@H](CO)NC(=O)CCc1c[nH]c2ccccc12 ZINC000217915096 CF In-Stock Unstable MAGI3 0 41 CC[C@@H](C)[C@@H](CO)NC(=O)CCc1c[nH]c2ccccc12 ZINC000217915096 CF In-Stock Unstable SLC15A2 0 47 CC[C@@H](C)[C@@H](CO)NC(=O)CCc1c[nH]c2ccccc12 ZINC000217915096 CF In-Stock Unstable LASB 0 43 COc1ccc(CN2CC[C@@H]3[C@@H](CCCN3C)C2)cc1O ZINC000217915118 CE On-Demand Unstable SSTR5 44 35 COc1ccc(C(=O)NCC[C@H](O)C2CCOCC2)cc1 ZINC000217915124 CD In-Stock Unstable DRD4 42 33 C[C@@H](Cc1ccc(F)cc1)NC(=O)N[C@H](C(=O)O)[C@H](C)O ZINC000217915156 CC For-Sale Unstable ACE 21 40 C[C@@H](Cc1ccc(F)cc1)NC(=O)N[C@H](C(=O)O)[C@H](C)O ZINC000217915156 CC For-Sale Unstable MME 58 47 C[C@@H](Cc1ccc(F)cc1)NC(=O)N[C@H](C(=O)O)[C@H](C)O ZINC000217915156 CC For-Sale Unstable CPA1 24 43 C[C@@H](Cc1ccc(F)cc1)NC(=O)N[C@H](C(=O)O)[C@H](C)O ZINC000217915156 CC For-Sale Unstable ACE2 47 39 O=C(/C=C/c1ccc(F)cc1)NCc1nc(-c2cccc(Br)c2)no1 ZINC000217915189 HH In-Stock Unstable HDAC8 50 35 O=C(/C=C/c1ccc(F)cc1)NCc1nc(-c2cccc(Br)c2)no1 ZINC000217915189 HH In-Stock Unstable HDAC6 41 36 COc1ccc(C(=O)NCC[C@@H](O)C2CCOCC2)cc1 ZINC000217915190 CD In-Stock Unstable DRD4 42 33 O=C(c1ccc(O)c(Cl)c1)N1CCCS(=O)(=O)CC1 ZINC000217915224 DD On-Demand Unstable L3MBTL3 44 34 O=C(/C=C/c1ccc(F)cc1)NCc1nc(-c2cccs2)no1 ZINC000217915298 EG In-Stock Unstable ETHR 31 40 Cc1cccc(/C=C/NC(=O)Nc2cc(F)ccc2F)c1 ZINC000217915300 CI For-Sale Unstable MMP1 0 41 O=C(NCC[C@H](O)C1CCOCC1)c1ccc(Cl)cc1 ZINC000217915309 CE In-Stock Unstable UTS2 41 33 CSc1ccccc1C(=O)NC1CCN(C(=O)N2CCOCC2)CC1 ZINC000217915346 FE In-Stock Unstable HTR3A 23 41 CSc1ccccc1C(=O)NC1CCN(C(=O)N2CCOCC2)CC1 ZINC000217915346 FE In-Stock Unstable CNR2 16 43 CSc1ccccc1C(=O)NC1CCN(C(=O)N2CCOCC2)CC1 ZINC000217915346 FE In-Stock Unstable EPHX2 19 40 CSc1ccccc1C(=O)NC1CCN(C(=O)N2CCOCC2)CC1 ZINC000217915346 FE In-Stock Unstable CCR8 50 46 CSc1ccccc1C(=O)NC1CCN(C(=O)N2CCOCC2)CC1 ZINC000217915346 FE In-Stock Unstable AKR1C3 31 42 O=C(CC[C@@H]1NC(=O)N(Cc2ccccc2)C1=O)N[C@H](CO)Cc1ccccc1 ZINC000217915361 GD In-Stock Unstable MME 32 41 O=C(NCC[C@@H](O)C1CCOCC1)c1ccc(Cl)cc1 ZINC000217915381 CE In-Stock Unstable UTS2 41 33 Cc1ccc(NC(=O)c2cncc(/C=C\C(=O)O)c2)cc1 ZINC000217915384 CF For-Sale Unstable SCN10A 43 45 Cc1ccc(NC(=O)c2cncc(/C=C\C(=O)O)c2)cc1 ZINC000217915384 CF For-Sale Unstable KCNK3 68 38 Cc1ccc(NC(=O)c2cncc(/C=C\C(=O)O)c2)cc1 ZINC000217915384 CF For-Sale Unstable KCNK9 42 38 Cn1cc(C=O)c2c(N)ncnc21 ZINC000217915387 AC For-Sale Unstable ABL1 25 42 Cn1cc(C=O)c2c(N)ncnc21 ZINC000217915387 AC For-Sale Unstable PRKDC 61 42 Cn1cc(C=O)c2c(N)ncnc21 ZINC000217915387 AC For-Sale Unstable SRC 30 42 Cn1cc(C=O)c2c(N)ncnc21 ZINC000217915387 AC For-Sale Unstable PIK3CA 22 42 Cn1cc(C=O)c2c(N)ncnc21 ZINC000217915387 AC For-Sale Unstable PIK3CD 32 42 Cn1cc(C=O)c2c(N)ncnc21 ZINC000217915387 AC For-Sale Unstable MTOR 28 42 Cn1cc(C=O)c2c(N)ncnc21 ZINC000217915387 AC For-Sale Unstable HCK 38 42 Cn1cc(C=O)c2c(N)ncnc21 ZINC000217915387 AC For-Sale Unstable PIK3CG 24 42 Cn1cc(C=O)c2c(N)ncnc21 ZINC000217915387 AC For-Sale Unstable PIK3CB 24 42 Cn1cc(C=O)c2c(N)ncnc21 ZINC000217915387 AC For-Sale Unstable EIF2AK3 63 35 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1ccc(Cl)c(C(N)=O)c1 ZINC000217915390 DI For-Sale Unstable TRPM8 18 51 CN(Cc1nc(-c2ccccc2)no1)C(=O)/C=C/c1ccc(F)cc1 ZINC000217915406 EH In-Stock Unstable FABI 43 33 CN(Cc1nc(-c2ccccc2)no1)C(=O)/C=C/c1ccc(F)cc1 ZINC000217915406 EH In-Stock Unstable TSPO 15 44 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1ccc(Cl)c(C(N)=O)c1 ZINC000217915460 DI For-Sale Unstable TRPM8 18 51 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1ccc(Cl)c(C(N)=O)c1 ZINC000217915537 DI For-Sale Unstable TRPM8 18 51 Cc1cccc(-c2noc(CN(C)C(=O)/C=C/c3ccc(F)cc3)n2)c1 ZINC000217915555 FH In-Stock Unstable FABI 43 33 Cc1cccc(-c2noc(CN(C)C(=O)/C=C/c3ccc(F)cc3)n2)c1 ZINC000217915555 FH In-Stock Unstable GRM5 0 50 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1ccc(Cl)c(C(N)=O)c1 ZINC000217915576 DI For-Sale Unstable TRPM8 18 51 CS(=O)(=O)c1ccc(C2(N)CCCC2)c(F)c1 ZINC000217915612 CD For-Sale Unstable PTGS2 38 40 COC(=O)C[C@H](c1cc2ccc(OC)cc2[nH]c1=O)c1c(O)c2ccccc2oc1=O ZINC000217915645 HG In-Stock Unstable NQO1 45 52 CC1(C)OB(c2ccnc(OCCN3CCCC3)c2)OC1(C)C ZINC000217915652 DD For-Sale Unstable LTA4H 33 41 CC1(C)OB(c2ccnc(OCCN3CCCC3)c2)OC1(C)C ZINC000217915652 DD For-Sale Unstable PSMB2 46 35 CC1(C)OB(c2ccnc(OCCN3CCCC3)c2)OC1(C)C ZINC000217915652 DD For-Sale Unstable PSMB1 40 36 Cc1ccc(-c2noc(CN(C)C(=O)/C=C/c3ccc(F)cc3)n2)cc1 ZINC000217915656 FH In-Stock Unstable FABI 40 31 Cc1cccc(/C=C/NC(=O)N2CCN(c3ccccn3)CC2)c1 ZINC000217915708 DF For-Sale Unstable DRD4 26 42 Cc1cccc(/C=C/NC(=O)N2CCN(c3ccccn3)CC2)c1 ZINC000217915708 DF For-Sale Unstable P2RY12 21 40 COC(=O)C[C@@H](c1cc2ccc(OC)cc2[nH]c1=O)c1c(O)c2ccccc2oc1=O ZINC000217915742 HG In-Stock Unstable NQO1 45 52 CCN1Cc2ccccc2C[C@@H]1C(=O)N1CCC(n2cnnc2)CC1 ZINC000217915762 ED In-Stock Unstable PREP 42 47 CCN1Cc2ccccc2C[C@@H]1C(=O)N1CCC(n2cnnc2)CC1 ZINC000217915762 ED In-Stock Unstable ADAM9 63 35 COc1cccc(-c2noc(CN(C)C(=O)/C=C/c3ccc(F)cc3)n2)c1 ZINC000217915766 FH In-Stock Unstable FABI 40 30 CCN1Cc2ccccc2C[C@H]1C(=O)N1CCC(n2cnnc2)CC1 ZINC000217915838 ED In-Stock Unstable PREP 42 47 CCN1Cc2ccccc2C[C@H]1C(=O)N1CCC(n2cnnc2)CC1 ZINC000217915838 ED In-Stock Unstable ADAM9 63 35 O=C(NCC[C@H](O)C1CCOCC1)c1cc2ccccc2o1 ZINC000217915846 DE In-Stock Unstable NAMPT 16 43 O=C(Cc1cccc(O)c1)N1CCCS(=O)(=O)CC1 ZINC000217915895 CC On-Demand Unstable ECE2 0 42 O=C(NCC[C@@H](O)C1CCOCC1)c1cc2ccccc2o1 ZINC000217915925 DE In-Stock Unstable NAMPT 16 43 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)Nc3ccncc3)[C@H]21 ZINC000217915959 JG In-Stock Unstable TSHR 42 32 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)Nc3ccncc3)[C@H]21 ZINC000217915959 JG In-Stock Unstable ENPP1 40 33 Cc1csc(NC(=O)c2cncc(/C=C\C(=O)O)c2)n1 ZINC000217915970 CE For-Sale Unstable GCK 19 47 CC[C@H](C(=O)NCC[C@H](O)C1CCOCC1)c1ccccc1 ZINC000217916028 DE In-Stock Unstable KCNQ2 44 43 CC[C@H](C(=O)NCC[C@H](O)C1CCOCC1)c1ccccc1 ZINC000217916028 DE In-Stock Unstable KCNQ4 0 40 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)Nc3ccncc3)[C@@H]21 ZINC000217916057 JG In-Stock Unstable TSHR 42 32 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)Nc3ccncc3)[C@@H]21 ZINC000217916057 JG In-Stock Unstable ENPP1 40 33 CN(Cc1nc(-c2ccccc2Cl)no1)C(=O)/C=C/c1ccc(F)cc1 ZINC000217916062 FI In-Stock Unstable FABI 41 31 CN(Cc1nc(-c2ccccc2Cl)no1)C(=O)/C=C/c1ccc(F)cc1 ZINC000217916062 FI In-Stock Unstable GPBAR1 24 44 CC[C@@H](C(=O)NCC[C@H](O)C1CCOCC1)c1ccccc1 ZINC000217916090 DE In-Stock Unstable KCNQ2 44 43 CC[C@@H](C(=O)NCC[C@H](O)C1CCOCC1)c1ccccc1 ZINC000217916090 DE In-Stock Unstable KCNQ4 0 40 O=C(c1ccc([N+](=O)[O-])c(O)c1)N1CCCS(=O)(=O)CC1 ZINC000217916105 DC On-Demand Unstable L3MBTL1 0 45 CC[C@H](C(=O)NCC[C@@H](O)C1CCOCC1)c1ccccc1 ZINC000217916156 DE In-Stock Unstable KCNQ2 44 43 CC[C@H](C(=O)NCC[C@@H](O)C1CCOCC1)c1ccccc1 ZINC000217916156 DE In-Stock Unstable KCNQ4 0 40 CC1(C)CCc2cc(CC(=O)NCCCC(=O)O)ccc2O1 ZINC000217916170 DE In-Stock Unstable DAGLA 23 42 CCN(CCNC(=O)c1cc(N)n[nH]1)C1CC1 ZINC000217916183 BC For-Sale Unstable ALPL 46 33 COC(=O)c1cccc(NC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217916212 DH For-Sale Unstable KCNK3 87 44 COC(=O)c1cccc(NC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217916212 DH For-Sale Unstable KCNK9 54 44 O=C(c1ccc2[nH]cnc2c1)N1CCCS(=O)(=O)CC1 ZINC000217916235 CC On-Demand Unstable HPGD 49 40 CC[C@@H](C(=O)NCC[C@@H](O)C1CCOCC1)c1ccccc1 ZINC000217916238 DE In-Stock Unstable KCNQ2 44 43 CC[C@@H](C(=O)NCC[C@@H](O)C1CCOCC1)c1ccccc1 ZINC000217916238 DE In-Stock Unstable KCNQ4 0 40 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)N1CCC(C(N)=O)CC1)C(=O)OC2 ZINC000217916272 IF In-Stock Unstable IMPDH1 0 60 COc1c(C)c2c(c(OC)c1C/C=C(\C)CCC(=O)N1CCC(C(N)=O)CC1)C(=O)OC2 ZINC000217916272 IF In-Stock Unstable IMPDH2 0 60 C#CCCCOc1ccc(C(=O)N(C)C)cc1 ZINC000217916277 BE On-Demand Unstable PLA2G4B 63 38 C#CCCCOc1ccc(C(=O)N(C)C)cc1 ZINC000217916277 BE On-Demand Unstable ESRRG 44 33 COc1cc(-c2ccc3ncc(C(=O)C4CC4)c(Nc4ccc(N5CC[C@@H](N(C)C)C5)nc4)c3c2)cc(Cl)c1O ZINC000217916314 KK Annotated Unstable CSF1R 42 38 Cc1nn(Cc2ccccc2)c(C)c1CCC(=O)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217916388 HH In-Stock Unstable PANK1 0 41 COc1cc(-c2ccc3ncc(C(=O)C4CC4)c(Nc4ccc(N5CC[C@H](N(C)C)C5)nc4)c3c2)cc(Cl)c1O ZINC000217916402 KK Annotated Unstable CSF1R 42 38 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217916472 EJ In-Stock Unstable PYGL 24 45 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217916472 EJ In-Stock Unstable HDAC9 40 38 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217916472 EJ In-Stock Unstable HDAC7 51 38 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccc(F)cc2)cc1 ZINC000217916472 EJ In-Stock Unstable LEF 57 39 Cc1cccc(OC[C@@H]2CCCN(C(=O)c3cc(=O)cc(C)o3)C2)c1 ZINC000217916481 EG In-Stock Unstable CHRNA10 48 36 Cc1cccc(OC[C@H]2CCCN(C(=O)c3cc(=O)cc(C)o3)C2)c1 ZINC000217916504 EG In-Stock Unstable CHRNA10 48 36 CCC[C@@H](O)CNC[C@@H](O)COC(C)C ZINC000217916512 BC On-Demand Unstable ADRB2 0 55 CN(C)[C@@H]1CCN(c2ccc(Nc3c(C(=O)C4CC4)cnc4ccc(-c5cc(Cl)c(O)c(Cl)c5)cc34)cn2)C1 ZINC000217916513 KK Annotated Unstable MCHR1 19 42 CN(C)[C@H]1CCN(c2ccc(Nc3c(C(=O)C4CC4)cnc4ccc(-c5cc(Cl)c(O)c(Cl)c5)cc34)cn2)C1 ZINC000217916548 KK Annotated Unstable MCHR1 19 42 CCC[C@H](O)CNC[C@@H](O)COC(C)C ZINC000217916551 BC On-Demand Unstable ADRB2 0 55 O=C(/C=C/c1ccc(F)cc1)NCCCN1CCCc2ccccc21 ZINC000217916588 EH In-Stock Unstable DRD3 25 55 CCC[C@@H](O)CNC[C@H](O)COC(C)C ZINC000217916616 BC On-Demand Unstable ADRB2 0 55 COc1ccc(CN2CC[C@@H]3[C@@H](CCCN3C)C2)c(O)c1 ZINC000217916646 CE For-Sale Unstable CHRNA10 44 39 CC(C)(C)OC(=O)N[C@@H]1C[C@@H]2CCC(=O)C[C@@H]2C1 ZINC000217916676 CF In-Stock Unstable NAAA 15 48 CCOc1ccc(CNC(=O)/C=C/c2ccc(OC)cc2)cc1OCC ZINC000217916697 FH In-Stock Unstable PTGS2 0 49 CCOc1ccc(CNC(=O)/C=C/c2ccc(OC)cc2)cc1OCC ZINC000217916697 FH In-Stock Unstable BDKRB2 45 37 CCOc1ccc(CNC(=O)/C=C/c2ccc(OC)cc2)cc1OCC ZINC000217916697 FH In-Stock Unstable TRPV1 0 41 CCOc1ccc(CNC(=O)/C=C/c2ccc(OC)cc2)cc1OCC ZINC000217916697 FH In-Stock Unstable LTB4R 21 43 CCOc1ccc(CNC(=O)/C=C/c2ccc(OC)cc2)cc1OCC ZINC000217916697 FH In-Stock Unstable AHR 21 41 CCOc1ccc(CNC(=O)/C=C/c2ccc(OC)cc2)cc1OCC ZINC000217916697 FH In-Stock Unstable HDAC8 18 48 CCOc1ccc(CNC(=O)/C=C/c2ccc(OC)cc2)cc1OCC ZINC000217916697 FH In-Stock Unstable HDAC1 25 41 CCOc1ccc(CNC(=O)/C=C/c2ccc(OC)cc2)cc1OCC ZINC000217916697 FH In-Stock Unstable HDAC2 0 41 CCOc1ccc(CNC(=O)/C=C/c2ccc(OC)cc2)cc1OCC ZINC000217916697 FH In-Stock Unstable AKR1C3 17 40 CCOc1ccc(CNC(=O)/C=C/c2ccc(OC)cc2)cc1OCC ZINC000217916697 FH In-Stock Unstable HD1B 0 40 CCOc1ccc(CNC(=O)/C=C/c2ccc(OC)cc2)cc1OCC ZINC000217916697 FH In-Stock Unstable ABCG2 16 41 CCC[C@H](O)CNC[C@H](O)COC(C)C ZINC000217916699 BC On-Demand Unstable ADRB2 0 55 Cc1c(C(=O)Nc2cccc(Cl)c2N2CCOCC2)[nH]c2c1C(=O)CC(C)(C)C2 ZINC000217916727 HI On-Demand Unstable MAPK8 16 40 CC(C)(C)OC(=O)N[C@H]1C[C@@H]2CCC(=O)C[C@@H]2C1 ZINC000217916740 CF In-Stock Unstable NAAA 15 48 O=C(c1cc(I)ccc1O)N1CCn2ccnc2C1 ZINC000217916748 FD On-Demand Unstable P2RX7 26 51 O=C(N[C@@H]1CCC[C@@H]1CO)c1cc(Cl)cc([N+](=O)[O-])c1 ZINC000217916751 CE For-Sale Unstable CACNA1I 44 31 Cc1cccc(/C=C/NC(=O)NCc2ccccc2Br)c1 ZINC000217916761 EI For-Sale Unstable ANPEP 15 45 CCC(CC)[C@H](NC(=O)[C@H](N)[C@H](C)CC)c1ccccc1 ZINC000217916782 CH For-Sale Unstable MME 48 39 CCC(CC)[C@H](NC(=O)[C@H](N)[C@H](C)CC)c1ccccc1 ZINC000217916782 CH For-Sale Unstable ANPEP 59 34 CCC(CC)[C@H](NC(=O)[C@H](N)[C@H](C)CC)c1ccccc1 ZINC000217916782 CH For-Sale Unstable PGA 15 40 CCC(CC)[C@H](NC(=O)[C@H](N)[C@H](C)CC)c1ccccc1 ZINC000217916782 CH For-Sale Unstable CAPN1 41 42 CCC(CC)[C@H](NC(=O)[C@H](N)[C@H](C)CC)c1ccccc1 ZINC000217916782 CH For-Sale Unstable CAPN2 73 40 CCC(CC)[C@H](NC(=O)[C@H](N)[C@H](C)CC)c1ccccc1 ZINC000217916782 CH For-Sale Unstable ACE2 60 39 COc1ccc(/C=C/C(=O)NCc2ccc(OC(C)C)c(OC)c2)cc1 ZINC000217916798 FH In-Stock Unstable PTGS2 0 50 COc1ccc(/C=C/C(=O)NCc2ccc(OC(C)C)c(OC)c2)cc1 ZINC000217916798 FH In-Stock Unstable TRPV1 28 47 COc1ccc(/C=C/C(=O)NCc2ccc(OC(C)C)c(OC)c2)cc1 ZINC000217916798 FH In-Stock Unstable HDAC8 17 47 COc1ccc(/C=C/C(=O)NCc2ccc(OC(C)C)c(OC)c2)cc1 ZINC000217916798 FH In-Stock Unstable HDAC1 0 42 COc1ccc(/C=C/C(=O)NCc2ccc(OC(C)C)c(OC)c2)cc1 ZINC000217916798 FH In-Stock Unstable HDAC2 0 40 COc1ccc(/C=C/C(=O)NCc2ccc(OC(C)C)c(OC)c2)cc1 ZINC000217916798 FH In-Stock Unstable HDAC6 15 46 COc1ccc(/C=C/C(=O)NCc2ccc(OC(C)C)c(OC)c2)cc1 ZINC000217916798 FH In-Stock Unstable MT-ND1 25 43 COc1ccc(/C=C/C(=O)NCc2ccc(OC(C)C)c(OC)c2)cc1 ZINC000217916798 FH In-Stock Unstable ABCG2 22 42 CC(C)(C)OC(=O)N[C@H]1C[C@H]2CC(=O)CC[C@@H]2C1 ZINC000217916820 CF In-Stock Unstable NAAA 15 48 O=C(N[C@H]1CCC[C@@H]1CO)c1cc(Cl)cc([N+](=O)[O-])c1 ZINC000217916831 CE For-Sale Unstable CACNA1I 44 31 CCC(CC)[C@H](NC(=O)[C@H](N)[C@@H](C)CC)c1ccccc1 ZINC000217916852 CH For-Sale Unstable MME 48 39 CCC(CC)[C@H](NC(=O)[C@H](N)[C@@H](C)CC)c1ccccc1 ZINC000217916852 CH For-Sale Unstable ANPEP 59 34 CCC(CC)[C@H](NC(=O)[C@H](N)[C@@H](C)CC)c1ccccc1 ZINC000217916852 CH For-Sale Unstable PGA 15 40 CCC(CC)[C@H](NC(=O)[C@H](N)[C@@H](C)CC)c1ccccc1 ZINC000217916852 CH For-Sale Unstable CAPN1 41 42 CCC(CC)[C@H](NC(=O)[C@H](N)[C@@H](C)CC)c1ccccc1 ZINC000217916852 CH For-Sale Unstable CAPN2 73 40 CCC(CC)[C@H](NC(=O)[C@H](N)[C@@H](C)CC)c1ccccc1 ZINC000217916852 CH For-Sale Unstable ACE2 60 39 Cc1n[nH]c(C)c1CCNC(=O)c1cc(CO)ccn1 ZINC000217916865 CC In-Stock Unstable HAO2 74 34 Cc1cccc(/C=C/NC(=O)NCc2cccc(C)c2)c1 ZINC000217916880 CH For-Sale Unstable ANPEP 16 51 Cc1cccc(/C=C/NC(=O)NCc2cccc(C)c2)c1 ZINC000217916880 CH For-Sale Unstable FBP1 16 41 O=C(NCc1ccccc1S(=O)(=O)N1CCCCC1)c1ccnc2ccccc12 ZINC000217916889 HG On-Demand Unstable PREP 34 46 O=C(NCc1ccccc1S(=O)(=O)N1CCCCC1)c1ccnc2ccccc12 ZINC000217916889 HG On-Demand Unstable HNMT 66 40 O=C(NCc1ccccc1S(=O)(=O)N1CCCCC1)c1ccnc2ccccc12 ZINC000217916889 HG On-Demand Unstable EPHX2 20 43 O=C(NCc1ccccc1S(=O)(=O)N1CCCCC1)c1ccnc2ccccc12 ZINC000217916889 HG On-Demand Unstable FAP 0 56 O=C(NCc1ccccc1S(=O)(=O)N1CCCCC1)c1ccnc2ccccc12 ZINC000217916889 HG On-Demand Unstable NAMPT 44 41 O=C(N[C@@H]1CCC[C@H]1CO)c1cc(Cl)cc([N+](=O)[O-])c1 ZINC000217916898 CE For-Sale Unstable CACNA1I 44 31 CC(C)(C)OC(=O)N[C@@H]1C[C@H]2CC(=O)CC[C@@H]2C1 ZINC000217916904 CF In-Stock Unstable NAAA 15 48 O=C(Cc1ccc(Br)cc1)N1C[C@H]2CNC[C@@H](C2)C1 ZINC000217916916 DE For-Sale Unstable CHRNA7 23 54 COc1ccc(/C=C/C(=O)NCCCc2ccccc2Cl)cc1 ZINC000217916920 EI In-Stock Unstable PTGS2 0 51 COc1ccc(/C=C/C(=O)NCCCc2ccccc2Cl)cc1 ZINC000217916920 EI In-Stock Unstable PYGL 27 49 COc1ccc(/C=C/C(=O)NCCCc2ccccc2Cl)cc1 ZINC000217916920 EI In-Stock Unstable HDAC8 40 51 COc1ccc(/C=C/C(=O)NCCCc2ccccc2Cl)cc1 ZINC000217916920 EI In-Stock Unstable MTNR1A 59 40 COc1ccc(/C=C/C(=O)NCCCc2ccccc2Cl)cc1 ZINC000217916920 EI In-Stock Unstable MTNR1B 53 41 COc1ccc(/C=C/C(=O)NCCCc2ccccc2Cl)cc1 ZINC000217916920 EI In-Stock Unstable HDAC4 28 40 COc1ccc(/C=C/C(=O)NCCCc2ccccc2Cl)cc1 ZINC000217916920 EI In-Stock Unstable HDAC6 29 51 COc1ccc(/C=C/C(=O)NCCCc2ccccc2Cl)cc1 ZINC000217916920 EI In-Stock Unstable HDAC9 46 40 COc1ccc(/C=C/C(=O)NCCCc2ccccc2Cl)cc1 ZINC000217916920 EI In-Stock Unstable HDAC7 51 40 COc1ccc(/C=C/C(=O)NCCCc2ccccc2Cl)cc1 ZINC000217916920 EI In-Stock Unstable GPR183 0 42 COc1ccc(C(F)(F)F)c(C(C)=O)c1OC ZINC000217916961 BF For-Sale Unstable TUBB1 41 34 COc1cccc(CNC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217917002 CG For-Sale Unstable ROCK1 38 44 COc1cccc(CNC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217917002 CG For-Sale Unstable MTNR1A 51 48 COc1cccc(CNC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217917002 CG For-Sale Unstable MTNR1B 53 48 COc1cccc(CNC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217917002 CG For-Sale Unstable ROCK2 42 48 COc1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217917017 EI In-Stock Unstable PTGS2 26 53 COc1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217917017 EI In-Stock Unstable SCNN1A 53 42 COc1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217917017 EI In-Stock Unstable PYGL 26 48 COc1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217917017 EI In-Stock Unstable HDAC8 37 50 COc1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217917017 EI In-Stock Unstable HDAC1 29 42 COc1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217917017 EI In-Stock Unstable HDAC2 24 42 COc1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217917017 EI In-Stock Unstable HDAC4 24 40 COc1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217917017 EI In-Stock Unstable HDAC6 22 50 COc1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217917017 EI In-Stock Unstable CCR2 0 48 COc1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217917017 EI In-Stock Unstable HDAC9 40 40 COc1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217917017 EI In-Stock Unstable HDAC7 43 40 COc1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217917017 EI In-Stock Unstable U38 0 42 COc1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217917017 EI In-Stock Unstable PROKR1 54 38 COc1ccc(/C=C/C(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217917068 DH In-Stock Unstable PTGS2 0 51 COc1ccc(/C=C/C(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217917068 DH In-Stock Unstable DRD3 17 52 COc1ccc(/C=C/C(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217917068 DH In-Stock Unstable SCNN1A 15 40 COc1ccc(/C=C/C(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217917068 DH In-Stock Unstable PTAFR 17 43 COc1ccc(/C=C/C(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217917068 DH In-Stock Unstable AHR 29 40 COc1ccc(/C=C/C(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217917068 DH In-Stock Unstable PYGL 0 42 COc1ccc(/C=C/C(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217917068 DH In-Stock Unstable HDAC8 34 50 COc1ccc(/C=C/C(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217917068 DH In-Stock Unstable MTNR1A 39 41 COc1ccc(/C=C/C(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217917068 DH In-Stock Unstable MTNR1B 32 41 COc1ccc(/C=C/C(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217917068 DH In-Stock Unstable MMP2 15 47 COc1ccc(/C=C/C(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217917068 DH In-Stock Unstable HDAC1 30 42 COc1ccc(/C=C/C(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217917068 DH In-Stock Unstable HDAC6 23 50 COc1ccc(/C=C/C(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217917068 DH In-Stock Unstable HDAC9 46 37 COc1ccc(/C=C/C(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217917068 DH In-Stock Unstable HDAC7 51 37 COc1ccc(/C=C/C(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217917068 DH In-Stock Unstable LEF 46 37 CCC(CC)[C@@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217917096 CE For-Sale Unstable CTSC 24 41 CCN(C)C(=O)c1ccc(OC)cc1 ZINC000217917098 AD On-Demand Unstable OPRD1 15 51 CCN(C)C(=O)c1ccc(OC)cc1 ZINC000217917098 AD On-Demand Unstable BCHE 17 40 CCN(C)C(=O)c1ccc(OC)cc1 ZINC000217917098 AD On-Demand Unstable MTNR1A 45 35 CCN(C)C(=O)c1ccc(OC)cc1 ZINC000217917098 AD On-Demand Unstable MT-ND1 24 43 CCN(C)C(=O)c1ccc(OC)cc1 ZINC000217917098 AD On-Demand Unstable HSD17B2 19 47 CCN(C)C(=O)c1ccc(OC)cc1 ZINC000217917098 AD On-Demand Unstable H9B8T9_CAPHI 15 50 COc1ccc(CN2Cc3cnc(-c4ccccc4)nc3C2)cc1C(=O)O ZINC000217917111 FG In-Stock Unstable DRD4 28 41 COc1ccc(CN2Cc3cnc(-c4ccccc4)nc3C2)cc1C(=O)O ZINC000217917111 FG In-Stock Unstable ACHE 16 41 COc1ccc(CN2Cc3cnc(-c4ccccc4)nc3C2)cc1C(=O)O ZINC000217917111 FG In-Stock Unstable HRH1 18 46 COc1ccc(CN2Cc3cnc(-c4ccccc4)nc3C2)cc1C(=O)O ZINC000217917111 FG In-Stock Unstable AGTR2 40 34 COc1ccc(CN2Cc3cnc(-c4ccccc4)nc3C2)cc1C(=O)O ZINC000217917111 FG In-Stock Unstable SSTR5 53 38 COc1ccc(CN2Cc3cnc(-c4ccccc4)nc3C2)cc1C(=O)O ZINC000217917111 FG In-Stock Unstable ABCB1B 44 38 COc1ccc(CN2Cc3cnc(-c4ccccc4)nc3C2)cc1C(=O)O ZINC000217917111 FG In-Stock Unstable ABCB1 29 41 COc1ccc(CN2Cc3cnc(-c4ccccc4)nc3C2)cc1C(=O)O ZINC000217917111 FG In-Stock Unstable MCHR1 18 42 CCn1cc(NC(=O)c2cncc(/C=C\C(=O)O)c2)cn1 ZINC000217917124 CD For-Sale Unstable PANC 49 32 CCC(CC)[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217917132 CE For-Sale Unstable CTSC 24 41 COc1ccc(/C=C/C(=O)NCCCc2ccccc2OC)cc1 ZINC000217917174 EG In-Stock Unstable DRD2 15 61 COc1ccc(/C=C/C(=O)NCCCc2ccccc2OC)cc1 ZINC000217917174 EG In-Stock Unstable ACHE 0 43 COc1ccc(/C=C/C(=O)NCCCc2ccccc2OC)cc1 ZINC000217917174 EG In-Stock Unstable PTGS2 0 55 COc1ccc(/C=C/C(=O)NCCCc2ccccc2OC)cc1 ZINC000217917174 EG In-Stock Unstable DRD3 31 61 COc1ccc(/C=C/C(=O)NCCCc2ccccc2OC)cc1 ZINC000217917174 EG In-Stock Unstable LTB4R 0 42 COc1ccc(/C=C/C(=O)NCCCc2ccccc2OC)cc1 ZINC000217917174 EG In-Stock Unstable PYGL 0 42 COc1ccc(/C=C/C(=O)NCCCc2ccccc2OC)cc1 ZINC000217917174 EG In-Stock Unstable HDAC8 31 49 COc1ccc(/C=C/C(=O)NCCCc2ccccc2OC)cc1 ZINC000217917174 EG In-Stock Unstable MTNR1A 66 39 COc1ccc(/C=C/C(=O)NCCCc2ccccc2OC)cc1 ZINC000217917174 EG In-Stock Unstable MTNR1B 57 50 COc1ccc(/C=C/C(=O)NCCCc2ccccc2OC)cc1 ZINC000217917174 EG In-Stock Unstable MMP2 20 49 COc1ccc(/C=C/C(=O)NCCCc2ccccc2OC)cc1 ZINC000217917174 EG In-Stock Unstable HDAC2 26 41 COc1ccc(/C=C/C(=O)NCCCc2ccccc2OC)cc1 ZINC000217917174 EG In-Stock Unstable HDAC3 19 41 COc1ccc(/C=C/C(=O)NCCCc2ccccc2OC)cc1 ZINC000217917174 EG In-Stock Unstable HDAC4 25 41 COc1ccc(/C=C/C(=O)NCCCc2ccccc2OC)cc1 ZINC000217917174 EG In-Stock Unstable HDAC6 25 49 COc1ccc(/C=C/C(=O)NCCCc2ccccc2OC)cc1 ZINC000217917174 EG In-Stock Unstable MMP9 17 49 COc1ccc(/C=C/C(=O)NCCCc2ccccc2OC)cc1 ZINC000217917174 EG In-Stock Unstable HDAC9 45 41 COc1ccc(/C=C/C(=O)NCCCc2ccccc2OC)cc1 ZINC000217917174 EG In-Stock Unstable HDAC7 51 41 COc1ccc(/C=C/C(=O)NCCCc2ccccc2OC)cc1 ZINC000217917174 EG In-Stock Unstable ABCG2 24 42 COc1ccc(/C=C/C(=O)NCCCc2ccccc2OC)cc1 ZINC000217917174 EG In-Stock Unstable GPR183 0 46 O=C(NCC[C@H](O)C1CCOCC1)c1ccc2ccccc2c1 ZINC000217917178 DF In-Stock Unstable PLD1 27 40 O=C(NCC[C@H](O)C1CCOCC1)c1ccc2ccccc2c1 ZINC000217917178 DF In-Stock Unstable PLD2 36 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCc1ccc(OC)c(OC)c1OC ZINC000217917180 JG For-Sale Unstable AGTR2 40 35 O=C(Cc1cccc(Br)c1)N1C[C@H]2CNC[C@@H](C2)C1 ZINC000217917181 DE For-Sale Unstable CHRNA7 18 50 CCC[C@@H](O)CNCCCCCC(=O)O ZINC000217917205 BD For-Sale Unstable FABP2 0 47 CCC[C@@H](O)CNCCCCCC(=O)O ZINC000217917205 BD For-Sale Unstable PLA2G2C 0 40 CCC[C@@H](O)CNCCCCCC(=O)O ZINC000217917205 BD For-Sale Unstable PLA2G4A 0 41 CCC[C@@H](O)CNCCCCCC(=O)O ZINC000217917205 BD For-Sale Unstable S1PR2 29 40 CCC[C@@H](O)CNCCCCCC(=O)O ZINC000217917205 BD For-Sale Unstable EPHX2 0 42 CCC[C@@H](O)CNCCCCCC(=O)O ZINC000217917205 BD For-Sale Unstable Q6UB75_PIG 0 42 CCC[C@@H](O)CNCCCCCC(=O)O ZINC000217917205 BD For-Sale Unstable Q8WS26_TRYCR 34 40 CCC[C@@H](O)CNCCCCCC(=O)O ZINC000217917205 BD For-Sale Unstable SLC22A20 0 47 CCC[C@@H](O)CNCCCCCC(=O)O ZINC000217917205 BD For-Sale Unstable FPPS 0 40 CCC[C@@H](O)CNCCCCCC(=O)O ZINC000217917205 BD For-Sale Unstable SPPS 0 40 CCC[C@@H](O)CNCCCCCC(=O)O ZINC000217917205 BD For-Sale Unstable NOD1 42 33 CCC[C@@H](O)CNCCCCCC(=O)O ZINC000217917205 BD For-Sale Unstable CQSS 57 39 CCC(CC)[C@@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217917215 CE For-Sale Unstable CTSC 24 41 O=C(NCC[C@@H](O)C1CCOCC1)c1ccc2ccccc2c1 ZINC000217917239 DF In-Stock Unstable PLD1 27 40 O=C(NCC[C@@H](O)C1CCOCC1)c1ccc2ccccc2c1 ZINC000217917239 DF In-Stock Unstable PLD2 36 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCc1ccc(OC)c(OC)c1OC ZINC000217917244 JG For-Sale Unstable AGTR2 40 35 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC)c2)cc1 ZINC000217917250 EG In-Stock Unstable DRD4 40 30 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC)c2)cc1 ZINC000217917250 EG In-Stock Unstable PTGS2 0 53 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC)c2)cc1 ZINC000217917250 EG In-Stock Unstable DRD3 18 51 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC)c2)cc1 ZINC000217917250 EG In-Stock Unstable PTAFR 24 49 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC)c2)cc1 ZINC000217917250 EG In-Stock Unstable NQO2 23 40 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC)c2)cc1 ZINC000217917250 EG In-Stock Unstable FDFT1 0 43 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC)c2)cc1 ZINC000217917250 EG In-Stock Unstable CTSL 17 40 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC)c2)cc1 ZINC000217917250 EG In-Stock Unstable PYGL 23 44 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC)c2)cc1 ZINC000217917250 EG In-Stock Unstable HDAC8 58 49 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC)c2)cc1 ZINC000217917250 EG In-Stock Unstable MTNR1A 88 64 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC)c2)cc1 ZINC000217917250 EG In-Stock Unstable MTNR1B 70 61 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC)c2)cc1 ZINC000217917250 EG In-Stock Unstable MMP2 22 49 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC)c2)cc1 ZINC000217917250 EG In-Stock Unstable HDAC1 33 46 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC)c2)cc1 ZINC000217917250 EG In-Stock Unstable HDAC2 23 41 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC)c2)cc1 ZINC000217917250 EG In-Stock Unstable HDAC4 31 41 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC)c2)cc1 ZINC000217917250 EG In-Stock Unstable HDAC5 31 41 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC)c2)cc1 ZINC000217917250 EG In-Stock Unstable HDAC6 39 49 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC)c2)cc1 ZINC000217917250 EG In-Stock Unstable MMP9 24 49 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC)c2)cc1 ZINC000217917250 EG In-Stock Unstable HDAC9 40 41 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC)c2)cc1 ZINC000217917250 EG In-Stock Unstable HDAC7 43 41 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC)c2)cc1 ZINC000217917250 EG In-Stock Unstable AMP1_PLAFQ 20 43 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC)c2)cc1 ZINC000217917250 EG In-Stock Unstable HDA106 0 41 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC)c2)cc1 ZINC000217917250 EG In-Stock Unstable AKR1C3 22 42 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC)c2)cc1 ZINC000217917250 EG In-Stock Unstable HD1B 0 41 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC)c2)cc1 ZINC000217917250 EG In-Stock Unstable FOXO1 0 40 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC)c2)cc1 ZINC000217917250 EG In-Stock Unstable ABCG2 25 42 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC)c2)cc1 ZINC000217917250 EG In-Stock Unstable CRTM 69 50 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC)c2)cc1 ZINC000217917250 EG In-Stock Unstable GPR183 0 43 Cc1cccc(/C=C/NC(=O)NCc2cccc(Cl)c2)c1 ZINC000217917266 DI For-Sale Unstable CTSV 37 40 CCC[C@H](O)CNCCCCCC(=O)O ZINC000217917292 BD For-Sale Unstable FABP2 0 47 CCC[C@H](O)CNCCCCCC(=O)O ZINC000217917292 BD For-Sale Unstable PLA2G2C 0 40 CCC[C@H](O)CNCCCCCC(=O)O ZINC000217917292 BD For-Sale Unstable PLA2G4A 0 41 CCC[C@H](O)CNCCCCCC(=O)O ZINC000217917292 BD For-Sale Unstable S1PR2 29 40 CCC[C@H](O)CNCCCCCC(=O)O ZINC000217917292 BD For-Sale Unstable EPHX2 0 42 CCC[C@H](O)CNCCCCCC(=O)O ZINC000217917292 BD For-Sale Unstable Q6UB75_PIG 0 42 CCC[C@H](O)CNCCCCCC(=O)O ZINC000217917292 BD For-Sale Unstable Q8WS26_TRYCR 34 40 CCC[C@H](O)CNCCCCCC(=O)O ZINC000217917292 BD For-Sale Unstable SLC22A20 0 47 CCC[C@H](O)CNCCCCCC(=O)O ZINC000217917292 BD For-Sale Unstable FPPS 0 40 CCC[C@H](O)CNCCCCCC(=O)O ZINC000217917292 BD For-Sale Unstable SPPS 0 40 CCC[C@H](O)CNCCCCCC(=O)O ZINC000217917292 BD For-Sale Unstable NOD1 42 33 CCC[C@H](O)CNCCCCCC(=O)O ZINC000217917292 BD For-Sale Unstable CQSS 57 39 CCC(CC)[C@H](NC(=O)[C@H]1C[C@@H](O)CN1)c1ccccc1 ZINC000217917302 CE For-Sale Unstable CTSC 24 41 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCc1ccc(OC)c(OC)c1OC ZINC000217917314 JG For-Sale Unstable AGTR2 40 35 CCN(CC)c1ccc(C(=O)Nc2ccccc2OCC(F)(F)F)cc1 ZINC000217917342 FJ On-Demand Unstable ESRRG 21 42 CCN(CC)c1ccc(C(=O)Nc2ccccc2OCC(F)(F)F)cc1 ZINC000217917342 FJ On-Demand Unstable ABCG2 16 40 O=C(NCC[C@H](O)C1CCOCC1)c1ccc(F)cc1Cl ZINC000217917350 DE In-Stock Unstable P2RX7 26 41 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC)cc2)cc1 ZINC000217917361 EG In-Stock Unstable PTGS2 0 56 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC)cc2)cc1 ZINC000217917361 EG In-Stock Unstable DRD3 16 53 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC)cc2)cc1 ZINC000217917361 EG In-Stock Unstable SCNN1A 37 40 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC)cc2)cc1 ZINC000217917361 EG In-Stock Unstable PTAFR 19 47 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC)cc2)cc1 ZINC000217917361 EG In-Stock Unstable PYGL 23 47 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC)cc2)cc1 ZINC000217917361 EG In-Stock Unstable HDAC8 43 56 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC)cc2)cc1 ZINC000217917361 EG In-Stock Unstable MTNR1A 46 45 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC)cc2)cc1 ZINC000217917361 EG In-Stock Unstable MMP2 22 52 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC)cc2)cc1 ZINC000217917361 EG In-Stock Unstable HDAC1 34 42 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC)cc2)cc1 ZINC000217917361 EG In-Stock Unstable HDAC2 24 40 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC)cc2)cc1 ZINC000217917361 EG In-Stock Unstable HDAC4 37 40 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC)cc2)cc1 ZINC000217917361 EG In-Stock Unstable HDAC5 36 40 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC)cc2)cc1 ZINC000217917361 EG In-Stock Unstable HDAC6 29 56 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC)cc2)cc1 ZINC000217917361 EG In-Stock Unstable MMP9 22 52 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC)cc2)cc1 ZINC000217917361 EG In-Stock Unstable HDAC9 54 40 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC)cc2)cc1 ZINC000217917361 EG In-Stock Unstable HDAC7 53 40 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC)cc2)cc1 ZINC000217917361 EG In-Stock Unstable CA9 18 42 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC)cc2)cc1 ZINC000217917361 EG In-Stock Unstable CYP24A1 20 42 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC)cc2)cc1 ZINC000217917361 EG In-Stock Unstable HDA106 0 43 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC)cc2)cc1 ZINC000217917361 EG In-Stock Unstable HD1B 0 40 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC)cc2)cc1 ZINC000217917361 EG In-Stock Unstable ABCG2 16 41 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC)cc2)cc1 ZINC000217917361 EG In-Stock Unstable PROKR1 52 32 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC)cc2)cc1 ZINC000217917361 EG In-Stock Unstable CYP27B1 25 42 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC)cc2)cc1 ZINC000217917361 EG In-Stock Unstable TRPM2 0 43 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC)cc2)cc1 ZINC000217917361 EG In-Stock Unstable GPR183 0 43 Cc1cccc(/C=C/NC(=O)NCc2cccc(Br)c2)c1 ZINC000217917367 EI For-Sale Unstable ANPEP 15 48 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCc1ccc(OC)c(OC)c1OC ZINC000217917395 JG For-Sale Unstable AGTR2 40 35 O=C(NCC[C@@H](O)C1CCOCC1)c1ccc(F)cc1Cl ZINC000217917430 DE In-Stock Unstable P2RX7 26 41 O=C(Cc1ccccc1Br)N1C[C@H]2CNC[C@@H](C2)C1 ZINC000217917447 DE For-Sale Unstable CHRNA7 18 51 COc1ccc(/C=C/C(=O)N[C@@H](C)COc2ccc(OC)cc2)cc1 ZINC000217917462 EG In-Stock Unstable PTGS2 0 55 COc1ccc(/C=C/C(=O)N[C@@H](C)COc2ccc(OC)cc2)cc1 ZINC000217917462 EG In-Stock Unstable PTAFR 0 41 COc1ccc(/C=C/C(=O)N[C@@H](C)COc2ccc(OC)cc2)cc1 ZINC000217917462 EG In-Stock Unstable SDH1 0 41 COc1ccc(/C=C/C(=O)N[C@@H](C)COc2ccc(OC)cc2)cc1 ZINC000217917462 EG In-Stock Unstable HDAC8 25 56 COc1ccc(/C=C/C(=O)N[C@@H](C)COc2ccc(OC)cc2)cc1 ZINC000217917462 EG In-Stock Unstable MMP2 25 51 COc1ccc(/C=C/C(=O)N[C@@H](C)COc2ccc(OC)cc2)cc1 ZINC000217917462 EG In-Stock Unstable HDAC1 24 46 COc1ccc(/C=C/C(=O)N[C@@H](C)COc2ccc(OC)cc2)cc1 ZINC000217917462 EG In-Stock Unstable HDAC2 20 47 COc1ccc(/C=C/C(=O)N[C@@H](C)COc2ccc(OC)cc2)cc1 ZINC000217917462 EG In-Stock Unstable HDAC4 0 46 COc1ccc(/C=C/C(=O)N[C@@H](C)COc2ccc(OC)cc2)cc1 ZINC000217917462 EG In-Stock Unstable MMP9 19 51 COc1ccc(/C=C/C(=O)N[C@@H](C)COc2ccc(OC)cc2)cc1 ZINC000217917462 EG In-Stock Unstable GPR183 0 40 Cc1cccc(/C=C/NC(=O)NCc2ccc(Br)cc2)c1 ZINC000217917474 EI For-Sale Unstable ANPEP 17 44 CCCN(CC)CCNC(=O)CCC(C)=O ZINC000217917475 BD On-Demand Unstable PAOX 18 43 O=C(Nc1nc2c(s1)CCCCC2)c1cc(F)c(F)c(F)c1F ZINC000217917480 EI On-Demand Unstable SLC27A1 39 44 O=C(NCC[C@H](O)C1CCOCC1)c1nc2ccccc2s1 ZINC000217917526 DE In-Stock Unstable TRY1_BOVIN 41 38 O=C(NCC[C@H](O)C1CCOCC1)c1nc2ccccc2s1 ZINC000217917526 DE In-Stock Unstable TPSAB1 20 43 O=C(NCC[C@H](O)C1CCOCC1)c1nc2ccccc2s1 ZINC000217917526 DE In-Stock Unstable ST14 40 35 O=C(NCC[C@H](O)C1CCOCC1)c1nc2ccccc2s1 ZINC000217917526 DE In-Stock Unstable TMPRSS6 59 35 CC(C)(C)OC(=O)N[C@@H]1Cc2n[nH]c(C(=O)O)c2C1 ZINC000217917527 CD In-Stock Unstable HCAR2 17 51 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccc(OC)cc2)cc1 ZINC000217917543 EG In-Stock Unstable PTGS2 0 55 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccc(OC)cc2)cc1 ZINC000217917543 EG In-Stock Unstable PTAFR 0 41 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccc(OC)cc2)cc1 ZINC000217917543 EG In-Stock Unstable SDH1 0 41 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccc(OC)cc2)cc1 ZINC000217917543 EG In-Stock Unstable HDAC8 25 56 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccc(OC)cc2)cc1 ZINC000217917543 EG In-Stock Unstable MMP2 25 51 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccc(OC)cc2)cc1 ZINC000217917543 EG In-Stock Unstable HDAC1 24 46 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccc(OC)cc2)cc1 ZINC000217917543 EG In-Stock Unstable HDAC2 20 47 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccc(OC)cc2)cc1 ZINC000217917543 EG In-Stock Unstable HDAC4 0 46 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccc(OC)cc2)cc1 ZINC000217917543 EG In-Stock Unstable MMP9 19 51 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccc(OC)cc2)cc1 ZINC000217917543 EG In-Stock Unstable GPR183 0 40 O=C(c1ccc2[nH]c3c(c2c1)CCCC3)N1CCc2c([nH]c3ccccc23)C1 ZINC000217917556 FJ In-Stock Unstable FABI 60 39 O=C(c1ccc2[nH]c3c(c2c1)CCCC3)N1CCc2c([nH]c3ccccc23)C1 ZINC000217917556 FJ In-Stock Unstable DRD5 23 42 O=C(c1ccc2[nH]c3c(c2c1)CCCC3)N1CCc2c([nH]c3ccccc23)C1 ZINC000217917556 FJ In-Stock Unstable PARP1 19 43 CC(C)(C)OC(=O)N[C@H]1Cc2n[nH]c(C(=O)O)c2C1 ZINC000217917581 CD In-Stock Unstable HCAR2 17 51 CCC(CC)C(=O)Nc1nc2c(s1)CCCCC2 ZINC000217917600 CH On-Demand Unstable SLC27A1 39 42 Cc1cccc(/C=C/NC(=O)NCCc2ccccc2C)c1 ZINC000217917603 CH For-Sale Unstable MTNR1A 37 41 O=C(NCC[C@@H](O)C1CCOCC1)c1nc2ccccc2s1 ZINC000217917624 DE In-Stock Unstable TRY1_BOVIN 41 38 O=C(NCC[C@@H](O)C1CCOCC1)c1nc2ccccc2s1 ZINC000217917624 DE In-Stock Unstable TPSAB1 20 43 O=C(NCC[C@@H](O)C1CCOCC1)c1nc2ccccc2s1 ZINC000217917624 DE In-Stock Unstable ST14 40 35 O=C(NCC[C@@H](O)C1CCOCC1)c1nc2ccccc2s1 ZINC000217917624 DE In-Stock Unstable TMPRSS6 59 35 COc1ccc2nc(N[C@@H]3CCC[C@@H](C)[C@@H]3C)sc2c1 ZINC000217917627 CJ For-Sale Unstable CSNK1D 32 46 COc1ccc2nc(N[C@@H]3CCC[C@@H](C)[C@@H]3C)sc2c1 ZINC000217917627 CJ For-Sale Unstable ITK 0 50 COc1ccc2nc(N[C@@H]3CCC[C@@H](C)[C@@H]3C)sc2c1 ZINC000217917627 CJ For-Sale Unstable LUCI_PHOPE 31 40 COc1ccc2nc(N[C@@H]3CCC[C@@H](C)[C@@H]3C)sc2c1 ZINC000217917627 CJ For-Sale Unstable ISPD 0 41 O=C(Cc1ccc(F)c(F)c1)N[C@H]1CCC[C@H]1CO ZINC000217917635 CD On-Demand Unstable SSTR3 0 44 COc1ccc(/C=C/C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217917663 FJ In-Stock Unstable LTB4R 0 56 COc1ccc(/C=C/C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217917663 FJ In-Stock Unstable HDAC8 35 51 COc1ccc(/C=C/C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217917663 FJ In-Stock Unstable MMP2 27 61 COc1ccc(/C=C/C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217917663 FJ In-Stock Unstable HDAC1 26 53 COc1ccc(/C=C/C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217917663 FJ In-Stock Unstable HDAC2 23 40 COc1ccc(/C=C/C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217917663 FJ In-Stock Unstable HDAC6 26 51 COc1ccc(/C=C/C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217917663 FJ In-Stock Unstable MMP9 25 61 COc1ccc(/C=C/C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217917663 FJ In-Stock Unstable TUBB2B 21 41 COc1ccc(/C=C/C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217917663 FJ In-Stock Unstable HDA106 0 46 COc1ccc(/C=C/C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217917663 FJ In-Stock Unstable HD1B 0 40 COc1ccc(/C=C/C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217917663 FJ In-Stock Unstable ABCG2 18 41 COc1ccc(/C=C/C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217917663 FJ In-Stock Unstable AKR1C2 49 44 COc1ccc(/C=C/C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217917663 FJ In-Stock Unstable TRPM2 0 50 COc1ccc(/C=C/C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217917663 FJ In-Stock Unstable GPR183 0 42 COc1ccc(/C=C/C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217917663 FJ In-Stock Unstable A0A060INS8_CAPHI 0 47 C[C@H]1CN(C)[C@@H](C)C[C@@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000217917671 CD For-Sale Unstable CA2 52 43 C[C@H]1CN(C)[C@@H](C)C[C@@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000217917671 CD For-Sale Unstable CA1 47 42 C[C@H]1CN(C)[C@@H](C)C[C@@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000217917671 CD For-Sale Unstable CA7 37 40 C[C@H]1CN(C)[C@@H](C)C[C@@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000217917671 CD For-Sale Unstable CA12 40 43 C[C@H]1CN(C)[C@@H](C)C[C@@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000217917671 CD For-Sale Unstable CA9 42 40 C[C@H]1CN(C)[C@@H](C)C[C@@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000217917671 CD For-Sale Unstable CAH_METTE 18 40 C[C@H]1CN(C)[C@@H](C)C[C@@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000217917671 CD For-Sale Unstable CYNT 40 36 C[C@H]1CN(C)[C@@H](C)C[C@@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000217917671 CD For-Sale Unstable MTCA1 43 35 C[C@H]1CN(C)[C@@H](C)C[C@@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000217917671 CD For-Sale Unstable P96878_MYCTU 53 35 Cc1onc(-c2ccccc2Cl)c1C(=O)Nc1nc2c(s1)CCCCC2 ZINC000217917676 GK On-Demand Unstable GHSR 15 52 Cc1onc(-c2ccccc2Cl)c1C(=O)Nc1nc2c(s1)CCCCC2 ZINC000217917676 GK On-Demand Unstable GPBAR1 31 44 Cc1onc(-c2ccccc2Cl)c1C(=O)Nc1nc2c(s1)CCCCC2 ZINC000217917676 GK On-Demand Unstable BLAACC-4 0 42 Cc1onc(-c2ccccc2Cl)c1C(=O)Nc1nc2c(s1)CCCCC2 ZINC000217917676 GK On-Demand Unstable SUGE 0 42 Cc1onc(-c2ccccc2Cl)c1C(=O)Nc1nc2c(s1)CCCCC2 ZINC000217917676 GK On-Demand Unstable BLA_LAT-2 0 42 CCOc1ccc([C@@H](C)NC(=O)[C@H](N)[C@@H](C)CC)cc1 ZINC000217917697 CF For-Sale Unstable ACACA 73 57 CCOc1ccc([C@@H](C)NC(=O)[C@H](N)[C@@H](C)CC)cc1 ZINC000217917697 CF For-Sale Unstable ACACB 29 57 CCOc1ccc([C@@H](C)NC(=O)[C@H](N)[C@@H](C)CC)cc1 ZINC000217917697 CF For-Sale Unstable ACE2 56 38 O=C1C[C@@H](c2coc3ccccc3c2=O)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217917714 JI In-Stock Unstable AKR1B1 0 41 O=C1C[C@@H](c2coc3ccccc3c2=O)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217917714 JI In-Stock Unstable CYP1A1 28 40 O=C1C[C@@H](c2coc3ccccc3c2=O)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217917714 JI In-Stock Unstable CYP1A2 15 40 O=C1C[C@@H](c2coc3ccccc3c2=O)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217917714 JI In-Stock Unstable TNKS 31 41 O=C(Cc1ccccc1Br)NC1C[C@@H]2CC[C@@H](C1)N2 ZINC000217917716 DE On-Demand Unstable CA9 18 41 COc1ccccc1CCNC(=O)N/C=C/c1cccc(C)c1 ZINC000217917720 DH For-Sale Unstable MTNR1A 70 42 COc1ccccc1CCNC(=O)N/C=C/c1cccc(C)c1 ZINC000217917720 DH For-Sale Unstable MTNR1B 54 42 COc1ccc(CCC(=O)NCC[C@H](O)C2CCOCC2)cc1 ZINC000217917758 DD In-Stock Unstable BMP1 35 41 COc1ccc(CCC(=O)NCC[C@H](O)C2CCOCC2)cc1 ZINC000217917758 DD In-Stock Unstable MTNR1A 43 35 COc1ccc(CCC(=O)NCC[C@H](O)C2CCOCC2)cc1 ZINC000217917758 DD In-Stock Unstable MMP2 63 33 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC(C)C)c2)cc1 ZINC000217917759 FI In-Stock Unstable DRD3 17 47 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC(C)C)c2)cc1 ZINC000217917759 FI In-Stock Unstable PTAFR 23 47 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC(C)C)c2)cc1 ZINC000217917759 FI In-Stock Unstable PYGL 0 40 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC(C)C)c2)cc1 ZINC000217917759 FI In-Stock Unstable HDAC8 41 44 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC(C)C)c2)cc1 ZINC000217917759 FI In-Stock Unstable MTNR1A 55 55 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC(C)C)c2)cc1 ZINC000217917759 FI In-Stock Unstable MTNR1B 45 53 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC(C)C)c2)cc1 ZINC000217917759 FI In-Stock Unstable MMP2 15 44 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC(C)C)c2)cc1 ZINC000217917759 FI In-Stock Unstable HDAC1 23 41 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC(C)C)c2)cc1 ZINC000217917759 FI In-Stock Unstable HDAC6 27 44 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC(C)C)c2)cc1 ZINC000217917759 FI In-Stock Unstable HDAC7 40 38 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC(C)C)c2)cc1 ZINC000217917759 FI In-Stock Unstable AMP1_PLAFQ 23 42 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC(C)C)c2)cc1 ZINC000217917759 FI In-Stock Unstable CRTM 64 48 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC(C)C)c2)cc1 ZINC000217917759 FI In-Stock Unstable GPR183 0 40 C[C@H]1CN(C)[C@@H](C)C[C@@H]1Nc1cccc(S(N)(=O)=O)c1 ZINC000217917764 CD For-Sale Unstable CA2 16 41 C[C@H]1CN(C)[C@@H](C)C[C@@H]1Nc1cccc(S(N)(=O)=O)c1 ZINC000217917764 CD For-Sale Unstable CA4 20 42 COc1ccc2nc(N[C@@H]3CCC[C@H](C)[C@@H]3C)sc2c1 ZINC000217917778 CJ For-Sale Unstable CSNK1D 32 46 COc1ccc2nc(N[C@@H]3CCC[C@H](C)[C@@H]3C)sc2c1 ZINC000217917778 CJ For-Sale Unstable ITK 0 50 COc1ccc2nc(N[C@@H]3CCC[C@H](C)[C@@H]3C)sc2c1 ZINC000217917778 CJ For-Sale Unstable LUCI_PHOPE 31 40 COc1ccc2nc(N[C@@H]3CCC[C@H](C)[C@@H]3C)sc2c1 ZINC000217917778 CJ For-Sale Unstable ISPD 0 41 O=C1C[C@H](c2coc3ccccc3c2=O)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217917787 JI In-Stock Unstable AKR1B1 0 41 O=C1C[C@H](c2coc3ccccc3c2=O)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217917787 JI In-Stock Unstable CYP1A1 28 40 O=C1C[C@H](c2coc3ccccc3c2=O)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217917787 JI In-Stock Unstable CYP1A2 15 40 O=C1C[C@H](c2coc3ccccc3c2=O)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217917787 JI In-Stock Unstable TNKS 31 41 O=C(Cc1ccccc1Br)NC1C[C@@H]2CC[C@H](C1)N2 ZINC000217917801 DE On-Demand Unstable CA9 18 41 C[C@@H](CN)c1ccc(CN2CC[C@@H](N3CCCC3)C2)cc1 ZINC000217917806 CE For-Sale Unstable L3MBTL3 66 45 Cc1cccc(/C=C/NC(=O)NCCc2ccccc2F)c1 ZINC000217917827 CH For-Sale Unstable MTNR1A 40 37 COc1ccc(CCC(=O)NCC[C@@H](O)C2CCOCC2)cc1 ZINC000217917840 DD In-Stock Unstable BMP1 35 41 COc1ccc(CCC(=O)NCC[C@@H](O)C2CCOCC2)cc1 ZINC000217917840 DD In-Stock Unstable MTNR1A 50 35 COc1ccc(CCC(=O)NCC[C@@H](O)C2CCOCC2)cc1 ZINC000217917840 DD In-Stock Unstable MTNR1B 41 35 COc1ccc(CCC(=O)NCC[C@@H](O)C2CCOCC2)cc1 ZINC000217917840 DD In-Stock Unstable MMP2 63 33 O=C(c1cc(Br)ccc1O)N1CCC2(CCCC2)CC1 ZINC000217917854 EH On-Demand Unstable PYK 74 32 CCC[C@@H](C)C(=O)Nc1nc2c(s1)CCCCC2 ZINC000217917864 CH On-Demand Unstable SLC27A1 39 43 CCOc1ccc([C@@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2)cc1 ZINC000217917866 CC On-Demand Unstable ACACA 22 40 CCOc1ccc([C@@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2)cc1 ZINC000217917866 CC On-Demand Unstable ACACB 32 49 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC(C)C)cc2)cc1 ZINC000217917868 FI In-Stock Unstable PTAFR 17 43 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC(C)C)cc2)cc1 ZINC000217917868 FI In-Stock Unstable PYGL 0 41 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC(C)C)cc2)cc1 ZINC000217917868 FI In-Stock Unstable HDAC8 30 48 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC(C)C)cc2)cc1 ZINC000217917868 FI In-Stock Unstable HDAC1 23 41 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC(C)C)cc2)cc1 ZINC000217917868 FI In-Stock Unstable HDAC2 0 41 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC(C)C)cc2)cc1 ZINC000217917868 FI In-Stock Unstable HDAC6 17 48 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC(C)C)cc2)cc1 ZINC000217917868 FI In-Stock Unstable HDAC7 40 38 O=C(Cc1ccccc1Br)NC1C[C@H]2CC[C@H](C1)N2 ZINC000217917880 DE On-Demand Unstable CA9 18 41 C[C@H](CN)c1ccc(CN2CC[C@@H](N3CCCC3)C2)cc1 ZINC000217917887 CE For-Sale Unstable L3MBTL3 66 45 COC(=O)C[C@H](c1ccc(OC(C)C)c(OC)c1)c1c(O)c2ccccc2oc1=O ZINC000217917897 HH In-Stock Unstable NQO1 53 49 N[C@@H]1Cc2n[nH]c(C(=O)O)c2C1 ZINC000217917907 AB In-Stock Unstable HCAR2 22 61 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc2nccc(C)c2c1 ZINC000217917914 HH For-Sale Unstable HCRTR1 48 37 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc2nccc(C)c2c1 ZINC000217917914 HH For-Sale Unstable HCRTR2 53 37 CCC[C@H](C)C(=O)Nc1nc2c(s1)CCCCC2 ZINC000217917923 CH On-Demand Unstable SLC27A1 37 40 CCOc1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2)cc1 ZINC000217917934 CC On-Demand Unstable ACACA 22 40 CCOc1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2)cc1 ZINC000217917934 CC On-Demand Unstable ACACB 32 49 CCOc1ccc(CC(=O)NCC[C@H](O)C2CCOCC2)cc1 ZINC000217917959 DD In-Stock Unstable NQO2 16 40 COc1ccc(/C=C/C(=O)Nc2ccc(OC3CCCC3)cc2)cc1 ZINC000217917961 EJ In-Stock Unstable HDAC8 26 51 COc1ccc(/C=C/C(=O)Nc2ccc(OC3CCCC3)cc2)cc1 ZINC000217917961 EJ In-Stock Unstable MMP2 27 67 COc1ccc(/C=C/C(=O)Nc2ccc(OC3CCCC3)cc2)cc1 ZINC000217917961 EJ In-Stock Unstable HDAC1 34 51 COc1ccc(/C=C/C(=O)Nc2ccc(OC3CCCC3)cc2)cc1 ZINC000217917961 EJ In-Stock Unstable MMP9 24 67 COc1ccc(/C=C/C(=O)Nc2ccc(OC3CCCC3)cc2)cc1 ZINC000217917961 EJ In-Stock Unstable MMP1 25 49 COc1ccc(/C=C/C(=O)Nc2ccc(OC3CCCC3)cc2)cc1 ZINC000217917961 EJ In-Stock Unstable MCHR1 19 45 COc1ccc(/C=C/C(=O)Nc2ccc(OC3CCCC3)cc2)cc1 ZINC000217917961 EJ In-Stock Unstable METAP2 0 48 COc1ccc(/C=C/C(=O)Nc2ccc(OC3CCCC3)cc2)cc1 ZINC000217917961 EJ In-Stock Unstable EXSA 0 44 COc1ccc(/C=C/C(=O)Nc2ccc(OC3CCCC3)cc2)cc1 ZINC000217917961 EJ In-Stock Unstable GPR183 0 43 Cc1cccc(/C=C/NC(=O)NCCc2ccccc2Cl)c1 ZINC000217917969 DI For-Sale Unstable MTNR1A 33 40 CCCCNC(=O)[C@@H](C)NC[C@@H](O)CCC ZINC000217917973 BD For-Sale Unstable DPP7 0 41 N[C@H]1Cc2n[nH]c(C(=O)O)c2C1 ZINC000217917985 AB In-Stock Unstable HCAR2 22 61 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc2nccc(C)c2c1 ZINC000217917986 HH For-Sale Unstable HCRTR1 48 37 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc2nccc(C)c2c1 ZINC000217917986 HH For-Sale Unstable HCRTR2 53 37 COC(=O)C[C@@H](c1ccc(OC(C)C)c(OC)c1)c1c(O)c2ccccc2oc1=O ZINC000217917996 HH In-Stock Unstable NQO1 53 49 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable ACE 52 64 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable TYR 27 45 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable SSTR2 36 45 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable GNRHR 25 50 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable OPRM1 35 63 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable OPRD1 36 63 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable MME 94 59 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable ANPEP 34 43 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable EDNRB 116 60 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable EDNRA 121 63 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable TACR1 64 50 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable MC4R 68 57 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable BMP1 38 49 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable TACR2 52 58 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable CTSB 22 45 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable CCKAR 132 53 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable NTSR1 38 40 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable CTSL 35 42 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable BRS3 47 51 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable TIMP3 20 55 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable C3AR1 26 46 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable TACR3 15 44 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable NMBR 32 49 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable MC3R 90 53 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable MC5R 101 53 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable MMP2 37 50 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable MMP3 17 44 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable MMP8 70 47 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable MMP14 105 47 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable GRPR 93 51 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable ECE1 90 59 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable REN 17 43 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable LNPEP 29 46 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable SSTR3 27 42 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable MMP11 103 47 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable FURIN 23 44 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable CCKBR 94 66 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable GHSR 71 53 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable CAPN1 19 57 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable MMP9 35 52 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable ACE2 77 39 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable MC1R 129 57 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable ADAM9 44 46 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable CTSC 16 56 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable C5AR1 59 44 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable ST14 15 48 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable MMP7 29 42 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable MMP1 26 52 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable FPR1 85 53 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable NPR 40 59 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable ADAM12 15 46 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable SSSIM 28 42 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable BLA1_STEMA 72 37 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable KISS1R 88 42 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable ERAP2 51 47 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable PSMB8 26 41 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable TMPRSS6 17 40 CSCC[C@H](NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O ZINC000217917999 GD Annotated Unstable HPN 35 48 CC(C)[C@@H]1CN(c2cnc3ccc(Cl)cc3n2)CCN1 ZINC000217918005 CF For-Sale Unstable PRKCQ 24 42 CCOc1ccc([C@@H](C)NC(=O)[C@H]2C[C@@H](O)CN2)cc1 ZINC000217918023 CC On-Demand Unstable ACACA 22 40 CCOc1ccc([C@@H](C)NC(=O)[C@H]2C[C@@H](O)CN2)cc1 ZINC000217918023 CC On-Demand Unstable ACACB 32 49 CCOc1ccc(CC(=O)NCC[C@@H](O)C2CCOCC2)cc1 ZINC000217918024 DD In-Stock Unstable NQO2 16 40 CCCCNC(=O)[C@H](C)NC[C@@H](O)CCC ZINC000217918035 BD For-Sale Unstable DPP7 0 41 O=C(CCOc1ccccc1)Nc1nc2c(s1)CCCCC2 ZINC000217918042 DH On-Demand Unstable SLC27A1 42 46 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc2nccc(C)c2c1 ZINC000217918070 HH For-Sale Unstable HCRTR1 48 37 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc2nccc(C)c2c1 ZINC000217918070 HH For-Sale Unstable HCRTR2 53 37 Cc1cccc(/C=C/NC(=O)NCCc2ccccc2Br)c1 ZINC000217918072 FI For-Sale Unstable MTNR1A 29 40 CC(C)[C@H]1CN(c2cnc3ccc(Cl)cc3n2)CCN1 ZINC000217918073 CF For-Sale Unstable PRKCQ 24 42 CCCCCCCCCC[C@@H](O)[C@@H]1CCC[C@@H](C)C1 ZINC000217918075 CK For-Sale Unstable MT-ND1 40 35 CCN1CCC[C@H](N[C@H](c2ccccc2)C(C)C)C1 ZINC000217918082 CG On-Demand Unstable BIRC2 45 41 COc1ccc(/C=C/C(=O)N[C@@H]2CC(C)(C)Oc3ccccc32)cc1 ZINC000217918084 EI In-Stock Unstable MMP2 16 45 COC(=O)C[C@H](c1ccc(OC)c(CO)c1)c1c(O)c2ccccc2oc1=O ZINC000217918088 GF In-Stock Unstable NQO1 60 51 CC(=O)Nc1cccc(N[C@H]2C[C@H](C)N(C)C[C@@H]2C)c1 ZINC000217918093 CF For-Sale Unstable CSNK2A1 23 40 CC(=O)Nc1cccc(N[C@H]2C[C@H](C)N(C)C[C@@H]2C)c1 ZINC000217918093 CF For-Sale Unstable KCNK3 87 35 CC(=O)Nc1cccc(N[C@H]2C[C@H](C)N(C)C[C@@H]2C)c1 ZINC000217918093 CF For-Sale Unstable KCNK9 57 35 CN(Cc1ccco1)C(=O)c1cncc(/C=C\C(=O)O)c1 ZINC000217918095 CE For-Sale Unstable FABI 40 30 CCOc1ccc([C@H](C)NC(=O)[C@H]2C[C@@H](O)CN2)cc1 ZINC000217918100 CC On-Demand Unstable ACACA 22 40 CCOc1ccc([C@H](C)NC(=O)[C@H]2C[C@@H](O)CN2)cc1 ZINC000217918100 CC On-Demand Unstable ACACB 32 49 CCCCNC(=O)[C@@H](C)NC[C@H](O)CCC ZINC000217918124 BD For-Sale Unstable DPP7 0 41 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc2nccc(C)c2c1 ZINC000217918141 HH For-Sale Unstable HCRTR1 48 37 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc2nccc(C)c2c1 ZINC000217918141 HH For-Sale Unstable HCRTR2 53 37 CCCCCCCCCC[C@H](O)[C@@H]1CCC[C@@H](C)C1 ZINC000217918147 CK For-Sale Unstable MT-ND1 40 35 CCN1CCC[C@@H](N[C@H](c2ccccc2)C(C)C)C1 ZINC000217918149 CG On-Demand Unstable BIRC2 45 41 COc1ccc(/C=C/C(=O)N[C@H]2CC(C)(C)Oc3ccccc32)cc1 ZINC000217918152 EI In-Stock Unstable MMP2 16 45 COC(=O)C[C@@H](c1ccc(OC)c(CO)c1)c1c(O)c2ccccc2oc1=O ZINC000217918153 GF In-Stock Unstable NQO1 60 51 Cc1nc(N)sc1C(=O)NCCN1CCNC1=O ZINC000217918178 CB In-Stock Unstable SCD1 32 40 Cc1nc(N)sc1C(=O)NCCN1CCNC1=O ZINC000217918178 CB In-Stock Unstable SCD 27 40 CC(C)[C@@H](C(=O)Nc1nc2c(s1)CCCCC2)N1C(=O)c2ccccc2C1=O ZINC000217918182 GH On-Demand Unstable SLC27A1 40 47 Cc1cccc(/C=C/NC(=O)NCCc2cccc(C)c2)c1 ZINC000217918183 CH For-Sale Unstable FBP1 15 41 CCCCNC(=O)[C@H](C)NC[C@H](O)CCC ZINC000217918205 BD For-Sale Unstable DPP7 0 41 CCCCCCCCCC[C@@H](O)[C@H]1CCC[C@@H](C)C1 ZINC000217918240 CK For-Sale Unstable MT-ND1 40 35 CC(C)[C@H](C(=O)Nc1nc2c(s1)CCCCC2)N1C(=O)c2ccccc2C1=O ZINC000217918255 GH On-Demand Unstable SLC27A1 40 47 COc1ccccc1OCC(=O)NCC[C@H](O)C1CCOCC1 ZINC000217918274 DD In-Stock Unstable MBTPS1 44 32 COc1cccc(CCNC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217918284 DH For-Sale Unstable DRD4 40 33 COc1cccc(CCNC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217918284 DH For-Sale Unstable CTSL 20 41 COc1cccc(CCNC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217918284 DH For-Sale Unstable MTNR1A 94 55 COc1cccc(CCNC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217918284 DH For-Sale Unstable MTNR1B 85 55 COc1cccc(CCNC(=O)N/C=C/c2cccc(C)c2)c1 ZINC000217918284 DH For-Sale Unstable CRTM 41 37 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(OC)cc2)cc1 ZINC000217918290 EH In-Stock Unstable DRD3 15 48 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(OC)cc2)cc1 ZINC000217918290 EH In-Stock Unstable PTAFR 17 42 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(OC)cc2)cc1 ZINC000217918290 EH In-Stock Unstable SCN2A 18 42 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(OC)cc2)cc1 ZINC000217918290 EH In-Stock Unstable AHR 22 45 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(OC)cc2)cc1 ZINC000217918290 EH In-Stock Unstable PYGL 0 42 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(OC)cc2)cc1 ZINC000217918290 EH In-Stock Unstable HDAC8 35 49 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(OC)cc2)cc1 ZINC000217918290 EH In-Stock Unstable MTNR1A 29 41 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(OC)cc2)cc1 ZINC000217918290 EH In-Stock Unstable HDAC1 31 43 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(OC)cc2)cc1 ZINC000217918290 EH In-Stock Unstable HDAC6 19 49 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(OC)cc2)cc1 ZINC000217918290 EH In-Stock Unstable MMP9 15 46 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(OC)cc2)cc1 ZINC000217918290 EH In-Stock Unstable HDAC7 41 38 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(OC)cc2)cc1 ZINC000217918290 EH In-Stock Unstable TRPM2 0 41 CCCCCCCCCC[C@H](O)[C@H]1CCC[C@@H](C)C1 ZINC000217918315 CK For-Sale Unstable MT-ND1 40 35 O=C(NCC1C[C@@H]2CC[C@H](C1)N2)c1cccc(Br)c1 ZINC000217918329 DF For-Sale Unstable CACNA1I 45 42 O=C(Nc1nc2c(s1)CCCCC2)c1ccccc1SCC(=O)N1CCCC1 ZINC000217918335 HI On-Demand Unstable SLC27A1 37 41 COc1cccc(N(CCF)S(=O)(=O)c2ccccc2)c1 ZINC000217918355 DF For-Sale Unstable OXTR 16 40 COc1cccc(N(CCF)S(=O)(=O)c2ccccc2)c1 ZINC000217918355 DF For-Sale Unstable MTNR1B 16 40 COc1cccc(N(CCF)S(=O)(=O)c2ccccc2)c1 ZINC000217918355 DF For-Sale Unstable NR1H2 15 43 COc1ccc([C@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2oc(C)cc(=O)c2O)cc1 ZINC000217918359 JI In-Stock Unstable DRD5 17 41 COc1ccc([C@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2oc(C)cc(=O)c2O)cc1 ZINC000217918359 JI In-Stock Unstable CYP1B1 15 41 COc1ccc([C@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2oc(C)cc(=O)c2O)cc1 ZINC000217918359 JI In-Stock Unstable RORC 45 38 COc1ccccc1OCC(=O)NCC[C@@H](O)C1CCOCC1 ZINC000217918388 DD In-Stock Unstable MBTPS1 44 32 CCCCCCCCCCCC[C@@H](O)[C@@H]1CCC[C@@H](C)C1 ZINC000217918393 CK For-Sale Unstable MT-ND1 40 35 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccc(OC)cc1 ZINC000217918401 FI In-Stock Unstable DRD3 21 53 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccc(OC)cc1 ZINC000217918401 FI In-Stock Unstable LTB4R 28 43 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccc(OC)cc1 ZINC000217918401 FI In-Stock Unstable HDAC8 17 44 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccc(OC)cc1 ZINC000217918401 FI In-Stock Unstable MTNR1A 75 55 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccc(OC)cc1 ZINC000217918401 FI In-Stock Unstable MTNR1B 63 55 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccc(OC)cc1 ZINC000217918401 FI In-Stock Unstable HDAC6 15 44 CN(C(=O)CSc1ccccc1C(=O)Nc1nc2c(s1)CCCCC2)C1CCCCC1 ZINC000217918425 JK On-Demand Unstable SLC27A1 36 41 COc1ccc([C@@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2oc(C)cc(=O)c2O)cc1 ZINC000217918432 JI In-Stock Unstable DRD5 17 41 COc1ccc([C@@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2oc(C)cc(=O)c2O)cc1 ZINC000217918432 JI In-Stock Unstable CYP1B1 15 41 COc1ccc([C@@H](CC(=O)N2CCc3c([nH]c4ccccc34)C2)c2oc(C)cc(=O)c2O)cc1 ZINC000217918432 JI In-Stock Unstable RORC 45 38 CCCCCCCCCCCC[C@H](O)[C@@H]1CCC[C@@H](C)C1 ZINC000217918467 CK For-Sale Unstable MT-ND1 40 35 COc1cccc(OCC(=O)NCC[C@H](O)C2CCOCC2)c1 ZINC000217918477 DD In-Stock Unstable DRD4 41 32 COc1cccc(OCC(=O)NCC[C@H](O)C2CCOCC2)c1 ZINC000217918477 DD In-Stock Unstable MTNR1A 66 43 COc1cccc(OCC(=O)NCC[C@H](O)C2CCOCC2)c1 ZINC000217918477 DD In-Stock Unstable MTNR1B 53 41 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccccc2C)cc1 ZINC000217918498 EH In-Stock Unstable PTGS2 0 50 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccccc2C)cc1 ZINC000217918498 EH In-Stock Unstable HDAC8 42 47 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccccc2C)cc1 ZINC000217918498 EH In-Stock Unstable MMP2 22 50 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccccc2C)cc1 ZINC000217918498 EH In-Stock Unstable HDAC1 16 41 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccccc2C)cc1 ZINC000217918498 EH In-Stock Unstable HDAC2 18 44 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccccc2C)cc1 ZINC000217918498 EH In-Stock Unstable HDAC6 27 47 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccccc2C)cc1 ZINC000217918498 EH In-Stock Unstable MMP9 19 50 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccccc2C)cc1 ZINC000217918498 EH In-Stock Unstable TUBB1 21 40 Cc1cccc(/C=C/NC(=O)NCCc2cccc(Cl)c2)c1 ZINC000217918509 DI For-Sale Unstable FBP1 21 40 O=C(Cc1ccc(S(=O)(=O)N2CCCC2)s1)Nc1nc2c(s1)CCCCC2 ZINC000217918511 IG On-Demand Unstable SLC27A1 45 48 COc1cc2c(cc1OC)CC(=O)N(CC(=O)NCC1CC1)C=C2 ZINC000217918540 ED In-Stock Unstable HCN2 0 41 CCCCCCCCCCCC[C@@H](O)[C@H]1CCC[C@@H](C)C1 ZINC000217918542 CK For-Sale Unstable MT-ND1 40 35 COc1cccc(OCC(=O)NCC[C@@H](O)C2CCOCC2)c1 ZINC000217918572 DD In-Stock Unstable DRD4 41 32 COc1cccc(OCC(=O)NCC[C@@H](O)C2CCOCC2)c1 ZINC000217918572 DD In-Stock Unstable MTNR1A 85 43 COc1cccc(OCC(=O)NCC[C@@H](O)C2CCOCC2)c1 ZINC000217918572 DD In-Stock Unstable MTNR1B 73 43 O=C(Nc1nc2c(s1)CCCCC2)c1cc2c(s1)CCC2 ZINC000217918598 DI On-Demand Unstable SLC27A1 30 42 COc1ccc(/C=C/C(=O)N[C@@H](C)COc2ccc(C)cc2)cc1 ZINC000217918601 EH In-Stock Unstable PTAFR 0 40 COc1ccc(/C=C/C(=O)N[C@@H](C)COc2ccc(C)cc2)cc1 ZINC000217918601 EH In-Stock Unstable HDAC8 22 54 COc1ccc(/C=C/C(=O)N[C@@H](C)COc2ccc(C)cc2)cc1 ZINC000217918601 EH In-Stock Unstable MMP2 17 47 COc1ccc(/C=C/C(=O)N[C@@H](C)COc2ccc(C)cc2)cc1 ZINC000217918601 EH In-Stock Unstable HDAC1 0 43 COc1ccc(/C=C/C(=O)N[C@@H](C)COc2ccc(C)cc2)cc1 ZINC000217918601 EH In-Stock Unstable HDAC2 19 44 COc1ccc(/C=C/C(=O)N[C@@H](C)COc2ccc(C)cc2)cc1 ZINC000217918601 EH In-Stock Unstable MMP9 16 47 COc1ccc(/C=C/C(=O)N[C@@H](C)COc2ccc(C)cc2)cc1 ZINC000217918601 EH In-Stock Unstable GPR183 0 45 CCCCCCCCCCCC[C@H](O)[C@H]1CCC[C@@H](C)C1 ZINC000217918608 CK For-Sale Unstable MT-ND1 40 35 O=C(NCC1C[C@@H]2CC[C@H](C1)N2)c1ccc(Br)cc1 ZINC000217918617 DF For-Sale Unstable CACNA1I 46 33 O=C(Cc1ccc(F)cc1F)N[C@H]1CCC[C@H]1CO ZINC000217918637 CD On-Demand Unstable SSTR3 24 40 COC(=O)[C@H](C)NC(=O)CC/C(C)=C/Cc1c(OC)c(C)c2c(c1OC)C(=O)OC2 ZINC000217918656 HF In-Stock Unstable IMPDH1 0 73 COC(=O)[C@H](C)NC(=O)CC/C(C)=C/Cc1c(OC)c(C)c2c(c1OC)C(=O)OC2 ZINC000217918656 HF In-Stock Unstable IMPDH2 0 73 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccc(C)cc2)cc1 ZINC000217918679 EH In-Stock Unstable PTAFR 0 40 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccc(C)cc2)cc1 ZINC000217918679 EH In-Stock Unstable HDAC8 22 54 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccc(C)cc2)cc1 ZINC000217918679 EH In-Stock Unstable MMP2 17 47 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccc(C)cc2)cc1 ZINC000217918679 EH In-Stock Unstable HDAC1 0 43 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccc(C)cc2)cc1 ZINC000217918679 EH In-Stock Unstable HDAC2 19 44 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccc(C)cc2)cc1 ZINC000217918679 EH In-Stock Unstable MMP9 16 47 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccc(C)cc2)cc1 ZINC000217918679 EH In-Stock Unstable GPR183 0 45 O=C(COc1ccc(Cl)cc1)NCC[C@H](O)C1CCOCC1 ZINC000217918680 EE In-Stock Unstable TRAR 32 48 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable ALOX5 27 43 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable ACE 38 53 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable MAOB 25 51 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable OPRM1 51 42 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable PPARG 39 43 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable OPRD1 50 42 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable PPARA 47 48 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable ADRB3 20 41 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable MME 109 53 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable LTA4H 43 56 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable ANPEP 61 34 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable HRAS 54 37 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable TACR2 26 41 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable PTGER3 59 38 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable CTSB 56 55 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable PAPA1_CARPA 75 42 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable CYSP_TRYCR 53 42 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable CTSK 36 42 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable CTSL 51 52 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable CACNA1B 42 41 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable CCR3 15 50 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable SCN2A 20 47 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable NPFFR2 41 34 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable ADAM17 21 40 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable TIMP3 76 36 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable LPAR1 31 47 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable CAPNS1 67 41 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable MMP2 21 54 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable MMP3 27 45 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable MMP8 16 45 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable GRIA1 61 41 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable PLA2G4B 66 35 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable ECE1 19 49 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable HLA-DRB1 61 37 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable REN 15 42 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable LNPEP 24 45 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable CTSS 18 41 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable CAPN1 88 45 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable MMP9 29 47 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable CAPN2 106 55 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable ACE2 76 53 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable ADAMTS4 40 38 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable FPR1 39 40 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable CTRB_BOVIN 52 39 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable NPR 61 43 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable AMP1_PLAFQ 30 48 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable LPAR3 43 51 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable TAAR1 21 45 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable FFAR1 66 47 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable FFAR4 40 38 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable ERAP2 30 40 CCCCN[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)OC ZINC000217918739 EH For-Sale Unstable NPFFR1 62 34 CN(C)S(=O)(=O)c1ccc(N2CCCC2)c(C(=O)Nc2nc3c(s2)CCCCC3)c1 ZINC000217918756 IH On-Demand Unstable SLC27A1 38 40 O=C(COc1ccc(Cl)cc1)NCC[C@@H](O)C1CCOCC1 ZINC000217918764 EE In-Stock Unstable TRAR 32 48 COc1ccc(/C=C/C(=O)N[C@@H](C)c2ccc(N3CCC(C)CC3)cc2)cc1 ZINC000217918774 GJ In-Stock Unstable HDAC1 15 40 COc1ccc(/C=C/C(=O)N[C@H](C)c2ccc(N3CCC(C)CC3)cc2)cc1 ZINC000217918849 GJ In-Stock Unstable HDAC1 15 40 O=C(NCC[C@H](O)C1CCOCC1)c1cc(-c2ccccc2)on1 ZINC000217918864 EE In-Stock Unstable HDAC10 19 52 O=C1CC[C@H]2CN([C@@H]3CCCc4cc(O)ccc43)CCN12 ZINC000217918865 CE For-Sale Unstable DRD5 20 48 CNC1C[C@@H]2CC[C@H](C1)N2CCc1cccc(Br)c1 ZINC000217918922 DG For-Sale Unstable ACHP_LYMST 15 42 CNC1C[C@@H]2CC[C@H](C1)N2CCc1cccc(Br)c1 ZINC000217918922 DG For-Sale Unstable Q8WSF8_APLCA 18 42 O=C(NCC[C@@H](O)C1CCOCC1)c1cc(-c2ccccc2)on1 ZINC000217918951 EE In-Stock Unstable HDAC10 19 52 COc1ccc(/C=C/C(=O)N[C@@H](C)c2ccc(N3CCC[C@@H](C)C3)cc2)cc1 ZINC000217918967 GJ In-Stock Unstable HDAC8 21 44 CCO[C@@H]1C[C@@H](NC(=O)c2ccc(O)c(Cl)c2)C1(C)C ZINC000217918983 CF For-Sale Unstable ADCYAP1R1 66 35 CCc1cccc2c1CCCO2 ZINC000217918989 AF For-Sale Unstable MTNR1A 17 47 C[C@@H]1CCC[C@H]([C@@H](O)CCCc2ccccc2)C1 ZINC000217919051 BI For-Sale Unstable SLC18A2 58 44 C[C@@H]1CCC[C@H]([C@@H](O)CCCc2ccccc2)C1 ZINC000217919051 BI For-Sale Unstable SIGMAR1 18 40 C[C@@H]1CCC[C@H]([C@@H](O)CCCc2ccccc2)C1 ZINC000217919051 BI For-Sale Unstable MMP3 19 43 COc1ccc(/C=C/C(=O)N[C@H](C)c2ccc(N3CCC[C@@H](C)C3)cc2)cc1 ZINC000217919052 GJ In-Stock Unstable HDAC8 21 44 CCO[C@H]1C[C@@H](NC(=O)c2ccc(O)c(Cl)c2)C1(C)C ZINC000217919065 CF For-Sale Unstable ADCYAP1R1 66 35 O=C(NCC[C@H](O)C1CCOCC1)c1cccc(C(F)(F)F)c1 ZINC000217919072 EF In-Stock Unstable CCR2 84 48 O=C(NCC[C@H](O)C1CCOCC1)c1cccc(C(F)(F)F)c1 ZINC000217919072 EF In-Stock Unstable BRAF 27 40 O=C(NCC[C@H](O)C1CCOCC1)c1cccc(C(F)(F)F)c1 ZINC000217919072 EF In-Stock Unstable GPR52 0 41 CNC[C@@H](C)c1ccc(CN2CCC[C@@H](C)CC2)cc1 ZINC000217919084 CH For-Sale Unstable HRH3 17 43 COc1ccc2[nH]c(=O)c([C@H](CC(=O)N3CCOCC3)c3c(O)c(O)c(O)c4c(=O)cc(-c5ccccc5)oc34)cc2c1 ZINC000217919099 KH In-Stock Unstable RORC 41 35 CCN(C(=O)c1cncc(/C=C\C(=O)O)c1)C1CCCC1 ZINC000217919113 CF For-Sale Unstable ACE 48 35 C[C@H]1CCC[C@H]([C@@H](O)CCCc2ccccc2)C1 ZINC000217919117 BI For-Sale Unstable SLC18A2 58 44 C[C@H]1CCC[C@H]([C@@H](O)CCCc2ccccc2)C1 ZINC000217919117 BI For-Sale Unstable SIGMAR1 18 40 C[C@H]1CCC[C@H]([C@@H](O)CCCc2ccccc2)C1 ZINC000217919117 BI For-Sale Unstable MMP3 19 43 Cc1ccc(NC(=O)N/C=C/c2cccc(C)c2)nc1 ZINC000217919129 CG For-Sale Unstable LUCI_LUCLA 36 42 CC(C)(C)NC(=O)Nc1ccc([N+](=O)[O-])cc1Br ZINC000217919139 DG For-Sale Unstable TBXA2R 30 48 CC(C)(C)NC(=O)Nc1ccc([N+](=O)[O-])cc1Br ZINC000217919139 DG For-Sale Unstable DDX3X 0 43 O=C(NCC[C@@H](O)C1CCOCC1)c1cccc(C(F)(F)F)c1 ZINC000217919141 EF In-Stock Unstable CCR2 84 48 O=C(NCC[C@@H](O)C1CCOCC1)c1cccc(C(F)(F)F)c1 ZINC000217919141 EF In-Stock Unstable BRAF 27 40 O=C(NCC[C@@H](O)C1CCOCC1)c1cccc(C(F)(F)F)c1 ZINC000217919141 EF In-Stock Unstable GPR52 0 41 CCO[C@@H]1C[C@H](NC(=O)c2ccc(O)c(Cl)c2)C1(C)C ZINC000217919157 CF For-Sale Unstable ADCYAP1R1 66 35 CCCCNC(=O)CNC[C@@H](O)CCC ZINC000217919161 BC For-Sale Unstable NOD1 40 37 CNC1C[C@@H]2CC[C@H](C1)N2CCc1ccc(Br)cc1 ZINC000217919181 DG For-Sale Unstable Q8WSF8_APLCA 17 41 COc1ccc2[nH]c(=O)c([C@@H](CC(=O)N3CCOCC3)c3c(O)c(O)c(O)c4c(=O)cc(-c5ccccc5)oc34)cc2c1 ZINC000217919188 KH In-Stock Unstable RORC 41 35 C[C@@H]1CCC[C@@H]([C@@H](O)CCCc2ccccc2)C1 ZINC000217919195 BI For-Sale Unstable SLC18A2 58 44 C[C@@H]1CCC[C@@H]([C@@H](O)CCCc2ccccc2)C1 ZINC000217919195 BI For-Sale Unstable SIGMAR1 18 40 C[C@@H]1CCC[C@@H]([C@@H](O)CCCc2ccccc2)C1 ZINC000217919195 BI For-Sale Unstable MMP3 19 43 C[C@H](CN)c1ccc(CN2CCC[C@@H](C)CC2)cc1 ZINC000217919209 CG For-Sale Unstable HRH3 20 43 CCCCNC(=O)CNC[C@H](O)CCC ZINC000217919230 BC For-Sale Unstable NOD1 40 37 CCO[C@H]1C[C@H](NC(=O)c2ccc(O)c(Cl)c2)C1(C)C ZINC000217919240 CF For-Sale Unstable ADCYAP1R1 66 35 CCCCNC(=O)Nc1ccc([N+](=O)[O-])cc1Br ZINC000217919247 DG For-Sale Unstable TBXA2R 29 52 CCCCNC(=O)Nc1ccc([N+](=O)[O-])cc1Br ZINC000217919247 DG For-Sale Unstable ACAT 0 46 O=C(NCC[C@H](O)C1CCOCC1)c1ccccc1C(F)(F)F ZINC000217919254 EF In-Stock Unstable RBP4 51 32 C[C@H]1CCC[C@@H]([C@@H](O)CCCc2ccccc2)C1 ZINC000217919278 BI For-Sale Unstable SLC18A2 58 44 C[C@H]1CCC[C@@H]([C@@H](O)CCCc2ccccc2)C1 ZINC000217919278 BI For-Sale Unstable SIGMAR1 18 40 C[C@H]1CCC[C@@H]([C@@H](O)CCCc2ccccc2)C1 ZINC000217919278 BI For-Sale Unstable MMP3 19 43 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccnc3ccccc23)CC(=O)O4)cc1O ZINC000217919311 JJ In-Stock Unstable AKR1B1 0 44 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccnc3ccccc23)CC(=O)O4)cc1O ZINC000217919311 JJ In-Stock Unstable CYP1B1 49 36 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2ccnc3ccccc23)CC(=O)O4)cc1O ZINC000217919311 JJ In-Stock Unstable CYP1A1 36 42 O=C(NCC[C@@H](O)C1CCOCC1)c1ccccc1C(F)(F)F ZINC000217919320 EF In-Stock Unstable RBP4 51 32 CCNC[C@@H](C)c1ccc(CN2CCC[C@@H](C)CC2)cc1 ZINC000217919329 CI For-Sale Unstable HRH3 18 41 Cc1cccc(/C=C/NC(=O)Nc2ccc(Br)cn2)c1 ZINC000217919337 EH For-Sale Unstable EGFR 21 41 COc1ccc(/C=C/C(=O)N[C@@H]2CC(C)(C)Oc3cc(C)ccc32)cc1 ZINC000217919344 FI In-Stock Unstable GPR183 0 42 Cc1cccc(C)c1NC(=O)Nc1ccccc1C(C)(C)C ZINC000217919384 CK For-Sale Unstable CXCL8 35 42 Cc1cccc(C)c1NC(=O)Nc1ccccc1C(C)(C)C ZINC000217919384 CK For-Sale Unstable MAPK14 16 40 Cc1cccc(C)c1NC(=O)Nc1ccccc1C(C)(C)C ZINC000217919384 CK For-Sale Unstable TRPV1 15 47 Cc1cccc(C)c1NC(=O)Nc1ccccc1C(C)(C)C ZINC000217919384 CK For-Sale Unstable P2RY1 25 42 Cc1cccc(C)c1NC(=O)Nc1ccccc1C(C)(C)C ZINC000217919384 CK For-Sale Unstable PYGL 44 42 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccnc3ccccc23)CC(=O)O4)cc1O ZINC000217919395 JJ In-Stock Unstable AKR1B1 0 44 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccnc3ccccc23)CC(=O)O4)cc1O ZINC000217919395 JJ In-Stock Unstable CYP1B1 49 36 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2ccnc3ccccc23)CC(=O)O4)cc1O ZINC000217919395 JJ In-Stock Unstable CYP1A1 36 42 CCNC[C@H](C)c1ccc(CN2CCC[C@@H](C)CC2)cc1 ZINC000217919407 CI For-Sale Unstable HRH3 18 41 COc1ccc(/C=C/C(=O)N[C@H]2CC(C)(C)Oc3cc(C)ccc32)cc1 ZINC000217919426 FI In-Stock Unstable GPR183 0 42 Cc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cn2)c1 ZINC000217919461 CH For-Sale Unstable F10 40 40 O=S(=O)(c1ccccc1)N(CCF)c1ccc(Cl)cc1 ZINC000217919466 DH For-Sale Unstable OXTR 23 47 O=S(=O)(c1ccccc1)N(CCF)c1ccc(Cl)cc1 ZINC000217919466 DH For-Sale Unstable NR1H3 15 44 O=S(=O)(c1ccccc1)N(CCF)c1ccc(Cl)cc1 ZINC000217919466 DH For-Sale Unstable NR1I2 24 46 O=S(=O)(c1ccccc1)N(CCF)c1ccc(Cl)cc1 ZINC000217919466 DH For-Sale Unstable NR1H2 24 44 O=S(=O)(c1ccccc1)N(CCF)c1ccc(Cl)cc1 ZINC000217919466 DH For-Sale Unstable RORC 18 49 CC(C)(C)OC(=O)NCCNC(=O)c1cccc(Cl)c1N ZINC000217919468 DE For-Sale Unstable ECR 55 39 CCCCNC(=O)Nc1ccc(Cl)cc1[N+](=O)[O-] ZINC000217919474 CG For-Sale Unstable TBXA2R 18 40 O=C(CCNC(=O)NC12CC3CC(CC(C3)C1)C2)Nc1nc2c(s1)CCCCC2 ZINC000217919547 HI On-Demand Unstable EPHX2 75 46 O=C(CCNC(=O)NC12CC3CC(CC(C3)C1)C2)Nc1nc2c(s1)CCCCC2 ZINC000217919547 HI On-Demand Unstable SLC27A1 32 41 Cc1cccc(/C=C/NC(=O)Nc2cc(Cl)ccn2)c1 ZINC000217919567 CH For-Sale Unstable TYK2 50 37 O=C(NCC[C@H](O)C1CCOCC1)c1cc(Cl)ccc1Cl ZINC000217919645 EF In-Stock Unstable P2RX7 25 44 O=C(NCC[C@H](O)C1CCOCC1)c1cc(Cl)ccc1Cl ZINC000217919645 EF In-Stock Unstable ALPL 41 34 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cc(OC)c(OC)c(OC)c2)CC(=O)O4)cc1O ZINC000217919685 KI In-Stock Unstable ALOX5 0 55 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cc(OC)c(OC)c(OC)c2)CC(=O)O4)cc1O ZINC000217919685 KI In-Stock Unstable AKR1B1 25 55 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cc(OC)c(OC)c(OC)c2)CC(=O)O4)cc1O ZINC000217919685 KI In-Stock Unstable CYP1B1 75 45 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cc(OC)c(OC)c(OC)c2)CC(=O)O4)cc1O ZINC000217919685 KI In-Stock Unstable CYP1A1 54 48 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cc(OC)c(OC)c(OC)c2)CC(=O)O4)cc1O ZINC000217919685 KI In-Stock Unstable CYP1A2 43 45 O=C(Nc1cccc(C(F)(F)F)c1)OCCCl ZINC000217919701 CG For-Sale Unstable KIT 16 42 O=C(Nc1cccc(C(F)(F)F)c1)OCCCl ZINC000217919701 CG For-Sale Unstable KDR 19 44 O=C(Nc1cccc(C(F)(F)F)c1)OCCCl ZINC000217919701 CG For-Sale Unstable NPY5R 16 40 O=C(Nc1cccc(C(F)(F)F)c1)OCCCl ZINC000217919701 CG For-Sale Unstable EPHX2 15 46 O=C(Nc1cccc(C(F)(F)F)c1)OCCCl ZINC000217919701 CG For-Sale Unstable TEK 28 44 O=C(Nc1cccc(C(F)(F)F)c1)OCCCl ZINC000217919701 CG For-Sale Unstable BTK 19 41 O=C(Nc1cccc(C(F)(F)F)c1)OCCCl ZINC000217919701 CG For-Sale Unstable RIPK1 39 41 O=C(Nc1cccc(C(F)(F)F)c1)OCCCl ZINC000217919701 CG For-Sale Unstable TRPM4 0 43 O=C(Nc1cccc(C(F)(F)F)c1)OCCCl ZINC000217919701 CG For-Sale Unstable PSBA 0 52 O=C(Nc1cccc(C(F)(F)F)c1)OCCCl ZINC000217919701 CG For-Sale Unstable KCNK3 42 47 O=C(Nc1cccc(C(F)(F)F)c1)OCCCl ZINC000217919701 CG For-Sale Unstable PDS 47 44 O=C(NCC[C@@H](O)C1CCOCC1)c1cc(Cl)ccc1Cl ZINC000217919731 EF In-Stock Unstable P2RX7 25 44 O=C(NCC[C@@H](O)C1CCOCC1)c1cc(Cl)ccc1Cl ZINC000217919731 EF In-Stock Unstable ALPL 41 34 COc1ccc(-n2c(C)nnc2SCC(=O)Nc2nc3c(s2)CCCCC3)cc1 ZINC000217919745 II On-Demand Unstable AXIN2 0 42 COc1ccc(-n2c(C)nnc2SCC(=O)Nc2nc3c(s2)CCCCC3)cc1 ZINC000217919745 II On-Demand Unstable SLC27A1 41 50 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cc(OC)c(OC)c(OC)c2)CC(=O)O4)cc1O ZINC000217919755 KI In-Stock Unstable ALOX5 0 55 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cc(OC)c(OC)c(OC)c2)CC(=O)O4)cc1O ZINC000217919755 KI In-Stock Unstable AKR1B1 25 55 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cc(OC)c(OC)c(OC)c2)CC(=O)O4)cc1O ZINC000217919755 KI In-Stock Unstable CYP1B1 75 45 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cc(OC)c(OC)c(OC)c2)CC(=O)O4)cc1O ZINC000217919755 KI In-Stock Unstable CYP1A1 54 48 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cc(OC)c(OC)c(OC)c2)CC(=O)O4)cc1O ZINC000217919755 KI In-Stock Unstable CYP1A2 43 45 Cc1cccc(/C=C/NC(=O)NCCCc2ccccc2)c1 ZINC000217919789 CH For-Sale Unstable MTNR1A 36 42 Cc1cccc(/C=C/NC(=O)NCCCc2ccccc2)c1 ZINC000217919789 CH For-Sale Unstable MTNR1B 39 42 Cc1cccc(/C=C/NC(=O)NCCCc2ccccc2)c1 ZINC000217919789 CH For-Sale Unstable FBP1 15 44 Cc1cccc(/C=C/NC(=O)NCCCc2ccccc2)c1 ZINC000217919789 CH For-Sale Unstable SCN5A 0 46 Cc1cccc(/C=C/NC(=O)NCCCc2ccccc2)c1 ZINC000217919789 CH For-Sale Unstable AMP1_PLAFQ 25 42 Cc1cccc(/C=C/NC(=O)NCCCc2ccccc2)c1 ZINC000217919789 CH For-Sale Unstable CRTM 44 40 O=C(NC12CC3CC(CC(C3)C1)C2)OCCCl ZINC000217919799 CF For-Sale Unstable EPHX2 97 50 CCCOc1ccc([C@@H](O)[C@@H]2CCC[C@@H](C)C2)cc1 ZINC000217919836 CI For-Sale Unstable ACACA 39 43 COc1ccc(CCN2C[C@H](C(=O)N[C@H](CO)c3ccccc3)CC2=O)cc1OC ZINC000217919859 HD In-Stock Unstable HCRTR1 17 41 COc1ccc(CCN2C[C@H](C(=O)N[C@H](CO)c3ccccc3)CC2=O)cc1OC ZINC000217919859 HD In-Stock Unstable CCR5 25 43 CCCC1CCC(Nc2cc(C(=O)OC)ccn2)CC1 ZINC000217919878 CH On-Demand Unstable PRKD1 65 36 Cc1cccc(/C=C/NC(=O)NCCCCc2ccccc2)c1 ZINC000217919888 DI For-Sale Unstable SCN2A 17 41 Cc1cccc(/C=C/NC(=O)NCCCCc2ccccc2)c1 ZINC000217919888 DI For-Sale Unstable MTNR1A 29 41 Cc1cccc(/C=C/NC(=O)NCCCCc2ccccc2)c1 ZINC000217919888 DI For-Sale Unstable MTNR1B 41 41 Cc1cccc(/C=C/NC(=O)NCCCCc2ccccc2)c1 ZINC000217919888 DI For-Sale Unstable HDAC1 19 40 Cc1cccc(/C=C/NC(=O)NCCCCc2ccccc2)c1 ZINC000217919888 DI For-Sale Unstable HDAC6 22 40 Cc1cccc(/C=C/NC(=O)NCCCCc2ccccc2)c1 ZINC000217919888 DI For-Sale Unstable FAAH 24 48 Cc1cccc(/C=C/NC(=O)NCCCCc2ccccc2)c1 ZINC000217919888 DI For-Sale Unstable FBP1 16 46 Cc1cccc(/C=C/NC(=O)NCCCCc2ccccc2)c1 ZINC000217919888 DI For-Sale Unstable SCN5A 0 47 Cc1cccc(/C=C/NC(=O)NCCCCc2ccccc2)c1 ZINC000217919888 DI For-Sale Unstable HDAC7 20 40 Cc1cccc(/C=C/NC(=O)NCCCCc2ccccc2)c1 ZINC000217919888 DI For-Sale Unstable AMP1_PLAFQ 24 41 Cc1cccc(/C=C/NC(=O)NCCCCc2ccccc2)c1 ZINC000217919888 DI For-Sale Unstable HDA106 0 41 Cc1cccc(/C=C/NC(=O)NCCCCc2ccccc2)c1 ZINC000217919888 DI For-Sale Unstable ACAT 0 44 CCCOc1ccc([C@H](O)[C@@H]2CCC[C@@H](C)C2)cc1 ZINC000217919921 CI For-Sale Unstable ACACA 39 43 CC[C@@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(C)c(C)c1 ZINC000217919939 DJ In-Stock Unstable PTGS2 0 51 CC[C@@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(C)c(C)c1 ZINC000217919939 DJ In-Stock Unstable HDAC8 19 48 CC[C@@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(C)c(C)c1 ZINC000217919939 DJ In-Stock Unstable HDAC1 0 41 CC[C@@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(C)c(C)c1 ZINC000217919939 DJ In-Stock Unstable TUBB1 25 41 CC[C@@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(C)c(C)c1 ZINC000217919939 DJ In-Stock Unstable GPR183 0 45 COc1ccc(CCN2C[C@@H](C(=O)N[C@H](CO)c3ccccc3)CC2=O)cc1OC ZINC000217919943 HD In-Stock Unstable HCRTR1 17 41 COc1ccc(CCN2C[C@@H](C(=O)N[C@H](CO)c3ccccc3)CC2=O)cc1OC ZINC000217919943 HD In-Stock Unstable CCR5 25 43 CCCOc1ccc([C@@H](O)[C@H]2CCC[C@@H](C)C2)cc1 ZINC000217920010 CI For-Sale Unstable ACACA 39 43 CC[C@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(C)c(C)c1 ZINC000217920012 DJ In-Stock Unstable PTGS2 0 51 CC[C@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(C)c(C)c1 ZINC000217920012 DJ In-Stock Unstable HDAC8 19 48 CC[C@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(C)c(C)c1 ZINC000217920012 DJ In-Stock Unstable HDAC1 17 41 CC[C@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(C)c(C)c1 ZINC000217920012 DJ In-Stock Unstable TUBB1 25 41 CC[C@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(C)c(C)c1 ZINC000217920012 DJ In-Stock Unstable GPR183 0 45 O=C(NC12CC3CC(CC(C3)C1)C2)OCCBr ZINC000217920020 DG For-Sale Unstable EPHX2 98 50 O=C(COc1ccc2ccccc2c1)NCC[C@H](O)C1CCOCC1 ZINC000217920030 EF In-Stock Unstable CYSP_TRYCR 0 47 CCCOc1ccc([C@H](O)[C@H]2CCC[C@@H](C)C2)cc1 ZINC000217920089 CI For-Sale Unstable ACACA 39 43 O=C(COc1ccc2ccccc2c1)NCC[C@@H](O)C1CCOCC1 ZINC000217920103 EF In-Stock Unstable CYSP_TRYCR 0 47 CC[C@@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(C)cc1C ZINC000217920117 DJ In-Stock Unstable GPR183 0 40 CC(C)Sc1ccccc1C(=O)Nc1nc2c(s1)CCCCC2 ZINC000217920134 EK On-Demand Unstable SLC27A1 32 44 C[C@@H]1CCC[C@@H](CNc2ncccc2[N+](=O)[O-])C1 ZINC000217920174 BG On-Demand Unstable PRKCQ 51 44 CC[C@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(C)cc1C ZINC000217920195 DJ In-Stock Unstable GPR183 0 40 CC[C@@H]1CN(C(=O)OC(C)(C)C)CC[C@@H]1C(=O)O ZINC000217920209 CE For-Sale Unstable GPR119 43 43 CC(C)C[C@H](NC(=O)C[C@@H]1NC(=O)c2ccccc2NC1=O)c1nc2ccccc2[nH]1 ZINC000217920225 HF In-Stock Unstable MMP7 21 50 C[C@H]1CCC[C@@H](CNc2ncccc2[N+](=O)[O-])C1 ZINC000217920256 BG On-Demand Unstable PRKCQ 51 44 Cn1ccc(NC(=O)c2cncc(/C=C\C(=O)O)c2)n1 ZINC000217920257 CD For-Sale Unstable GCK 20 43 Oc1ccc2c(c1)CCC[C@@H]2N1CC[C@@H]2CCCC[C@@H]21 ZINC000217920263 CI For-Sale Unstable DRD5 16 45 Oc1ccc2c(c1)CCC[C@@H]2N1CC[C@@H]2CCCC[C@@H]21 ZINC000217920263 CI For-Sale Unstable HSD17B1 53 37 CCN1CCC[C@H](NC(=O)[C@@H](Br)C(C)C)C1 ZINC000217920292 CE For-Sale Unstable BIRC2 50 41 CC[C@H]1CN(C(=O)OC(C)(C)C)CC[C@@H]1C(=O)O ZINC000217920295 CE For-Sale Unstable GPR119 43 43 CC(C)C[C@H](NC(=O)C[C@H]1NC(=O)c2ccccc2NC1=O)c1nc2ccccc2[nH]1 ZINC000217920317 HF In-Stock Unstable MMP7 21 50 CC[C@@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217920320 FH In-Stock Unstable PTGS2 0 54 CC[C@@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217920320 FH In-Stock Unstable CYP1B1 55 38 CC[C@@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217920320 FH In-Stock Unstable HDAC8 0 49 CC[C@@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217920320 FH In-Stock Unstable HDAC1 0 47 CC[C@@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217920320 FH In-Stock Unstable TUBB1 42 38 CC[C@@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217920320 FH In-Stock Unstable PTPA 0 42 CC[C@@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217920320 FH In-Stock Unstable ABCG2 21 46 C1=C[C@@H]2[C@@H](C1)C[C@H]2Nc1ccccc1N1CCCCC1 ZINC000217920328 CI For-Sale Unstable KCNQ2 70 39 C[C@@H]1CCC[C@H](CNc2ncccc2[N+](=O)[O-])C1 ZINC000217920337 BG On-Demand Unstable PRKCQ 51 44 Oc1ccc2c(c1)CCC[C@H]2N1CC[C@@H]2CCCC[C@@H]21 ZINC000217920344 CI For-Sale Unstable HSD17B1 53 37 Cc1cccc(/C=C/NC(=O)N2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000217920353 GF For-Sale Unstable TGM2 74 41 Cc1cccc(/C=C/NC(=O)N2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000217920353 GF For-Sale Unstable F13A1 92 41 Cc1cccc(/C=C/NC(=O)N2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000217920353 GF For-Sale Unstable AKR1C3 49 38 CN[C@@H]1[C@@H](O)O[C@@H](CO)[C@H](O)[C@H]1O ZINC000217920367 AA For-Sale Unstable B4GALT1 64 33 CCN1CCC[C@@H](NC(=O)[C@@H](Br)C(C)C)C1 ZINC000217920368 CE For-Sale Unstable BIRC2 50 41 CC[C@@H]1CN(C(=O)OC(C)(C)C)CC[C@H]1C(=O)O ZINC000217920377 CE For-Sale Unstable GPR119 43 43 C[C@H]1CCC[C@H](CNc2ncccc2[N+](=O)[O-])C1 ZINC000217920408 BG On-Demand Unstable PRKCQ 51 44 CC[C@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217920409 FH In-Stock Unstable PTGS2 0 54 CC[C@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217920409 FH In-Stock Unstable CYP1B1 55 38 CC[C@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217920409 FH In-Stock Unstable HDAC8 0 49 CC[C@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217920409 FH In-Stock Unstable HDAC1 0 47 CC[C@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217920409 FH In-Stock Unstable TUBB1 42 38 CC[C@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217920409 FH In-Stock Unstable PTPA 0 42 CC[C@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(OC)c(OC)c1 ZINC000217920409 FH In-Stock Unstable ABCG2 21 46 C1=C[C@@H]2[C@H](C1)C[C@H]2Nc1ccccc1N1CCCCC1 ZINC000217920412 CI For-Sale Unstable KCNQ2 70 39 O=C(Nc1ccc(Cl)c(Cl)c1)OCCCCCl ZINC000217920431 CJ For-Sale Unstable AGPAT2 41 36 COCc1n[nH]c(-c2cccc(NC(=O)CCCCCNc3ccc4c(cc3=O)[C@@H](NC(C)=O)CCc3cc(OC)c(OC)c(OC)c3-4)c2)n1 ZINC000217920434 KK In-Stock Unstable TUBA1A 15 53 CCN1CCC[C@H](NC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217920452 CF For-Sale Unstable CHRM1 28 43 CCN1CCC[C@H](NC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217920452 CF For-Sale Unstable DRD2 19 43 CCN1CCC[C@H](NC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217920452 CF For-Sale Unstable DRD4 18 42 CCN1CCC[C@H](NC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217920452 CF For-Sale Unstable SLC6A1 136 44 CCN1CCC[C@H](NC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217920452 CF For-Sale Unstable KCNQ2 54 39 CCN1CCC[C@H](NC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217920452 CF For-Sale Unstable CCR5 48 38 CCN1CCC[C@H](NC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217920452 CF For-Sale Unstable CCR2 15 41 CCN1CCC[C@H](NC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217920452 CF For-Sale Unstable XIAP 60 39 CCN1CCC[C@H](NC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217920452 CF For-Sale Unstable BIRC2 71 51 CCN1CCC[C@H](NC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217920452 CF For-Sale Unstable BIRC8 44 31 CCN1CCC[C@H](NC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217920452 CF For-Sale Unstable NMUR2 0 40 CCN1CCC[C@H](NC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217920452 CF For-Sale Unstable NMUR1 0 40 Cc1ccc(S(=O)(=O)N2CCN(C(=O)N/C=C/c3cccc(C)c3)CC2)cc1 ZINC000217920454 GF For-Sale Unstable TGM2 76 41 Cc1ccc(S(=O)(=O)N2CCN(C(=O)N/C=C/c3cccc(C)c3)CC2)cc1 ZINC000217920454 GF For-Sale Unstable F13A1 95 41 CC[C@H]1CN(C(=O)OC(C)(C)C)CC[C@H]1C(=O)O ZINC000217920462 CE For-Sale Unstable GPR119 43 43 O=C(c1ccccc1-c1ccccc1F)N1CCN(c2ncc[nH]c2=O)CC1 ZINC000217920482 GF In-Stock Unstable PARP1 27 40 O=C(c1ccccc1-c1ccccc1F)N1CCN(c2ncc[nH]c2=O)CC1 ZINC000217920482 GF In-Stock Unstable SLC6A7 0 49 O=C(Cc1csc(NC(=O)c2cccs2)n1)Nc1nc2c(s1)CCCCC2 ZINC000217920494 HI On-Demand Unstable SLC27A1 34 44 CC[C@@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217920520 FG In-Stock Unstable PTGS2 18 44 CC[C@@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217920520 FG In-Stock Unstable BMP1 46 38 CC[C@@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217920520 FG In-Stock Unstable MMP13 32 40 CC[C@@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217920520 FG In-Stock Unstable HDAC8 0 47 CC[C@@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217920520 FG In-Stock Unstable MMP2 25 44 CC[C@@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217920520 FG In-Stock Unstable HDAC1 0 50 CC[C@@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217920520 FG In-Stock Unstable MMP9 29 40 CCN1CCC[C@@H](NC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217920537 CF For-Sale Unstable CHRM1 28 43 CCN1CCC[C@@H](NC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217920537 CF For-Sale Unstable DRD2 19 43 CCN1CCC[C@@H](NC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217920537 CF For-Sale Unstable DRD4 18 42 CCN1CCC[C@@H](NC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217920537 CF For-Sale Unstable SLC6A1 136 44 CCN1CCC[C@@H](NC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217920537 CF For-Sale Unstable KCNQ2 54 39 CCN1CCC[C@@H](NC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217920537 CF For-Sale Unstable CCR5 48 38 CCN1CCC[C@@H](NC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217920537 CF For-Sale Unstable CCR2 15 41 CCN1CCC[C@@H](NC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217920537 CF For-Sale Unstable XIAP 60 39 CCN1CCC[C@@H](NC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217920537 CF For-Sale Unstable BIRC2 71 51 CCN1CCC[C@@H](NC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217920537 CF For-Sale Unstable BIRC8 44 31 CCN1CCC[C@@H](NC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217920537 CF For-Sale Unstable NMUR2 0 40 CCN1CCC[C@@H](NC(=O)[C@@H](Cl)c2ccccc2)C1 ZINC000217920537 CF For-Sale Unstable NMUR1 0 40 O=C(Nc1cccc(C(F)(F)F)c1)OCCCCCl ZINC000217920543 CI For-Sale Unstable KIT 17 42 O=C(Nc1cccc(C(F)(F)F)c1)OCCCCCl ZINC000217920543 CI For-Sale Unstable ATF1 40 37 O=C(Nc1cccc(C(F)(F)F)c1)OCCCCCl ZINC000217920543 CI For-Sale Unstable KDR 19 47 O=C(Nc1cccc(C(F)(F)F)c1)OCCCCCl ZINC000217920543 CI For-Sale Unstable EPHX2 21 48 O=C(Nc1cccc(C(F)(F)F)c1)OCCCCCl ZINC000217920543 CI For-Sale Unstable TEK 32 47 O=C(Nc1cccc(C(F)(F)F)c1)OCCCCCl ZINC000217920543 CI For-Sale Unstable BTK 20 41 O=C(Nc1cccc(C(F)(F)F)c1)OCCCCCl ZINC000217920543 CI For-Sale Unstable RIPK1 51 41 O=C(Nc1cccc(C(F)(F)F)c1)OCCCCCl ZINC000217920543 CI For-Sale Unstable TRPM4 0 40 O=C(Nc1cccc(C(F)(F)F)c1)OCCCCCl ZINC000217920543 CI For-Sale Unstable PSBA 0 49 O=C(Nc1cccc(C(F)(F)F)c1)OCCCCCl ZINC000217920543 CI For-Sale Unstable KCNK3 31 42 O=C(Nc1cccc(C(F)(F)F)c1)OCCCCCl ZINC000217920543 CI For-Sale Unstable PDS 45 45 COC(=O)N1CCN(C(=O)N/C=C/c2cccc(C)c2)CC1 ZINC000217920560 DE For-Sale Unstable GPR183 0 41 CC[C@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217920604 FG In-Stock Unstable PTGS2 18 44 CC[C@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217920604 FG In-Stock Unstable BMP1 46 38 CC[C@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217920604 FG In-Stock Unstable MMP13 32 40 CC[C@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217920604 FG In-Stock Unstable HDAC8 0 47 CC[C@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217920604 FG In-Stock Unstable MMP2 25 44 CC[C@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217920604 FG In-Stock Unstable HDAC1 0 50 CC[C@H](NC(=O)/C=C/c1ccc(OC)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217920604 FG In-Stock Unstable MMP9 29 40 COc1ccc(OC)c(CC(=O)Nc2nc3c(s2)CCCCC3)c1 ZINC000217920607 EH On-Demand Unstable CSNK1D 47 56 COc1ccc(OC)c(CC(=O)Nc2nc3c(s2)CCCCC3)c1 ZINC000217920607 EH On-Demand Unstable MAPK9 0 45 COc1ccc(OC)c(CC(=O)Nc2nc3c(s2)CCCCC3)c1 ZINC000217920607 EH On-Demand Unstable MAPK8 17 43 COc1ccc(OC)c(CC(=O)Nc2nc3c(s2)CCCCC3)c1 ZINC000217920607 EH On-Demand Unstable CA9 16 42 COc1ccc(OC)c(CC(=O)Nc2nc3c(s2)CCCCC3)c1 ZINC000217920607 EH On-Demand Unstable SLC27A1 45 48 O=C(Nc1ccc([N+](=O)[O-])cc1)OCCCCCl ZINC000217920659 CG For-Sale Unstable ACR 17 44 Cc1cc(C(=O)Nc2nc3c(s2)CCCCC3)c(C)n1C1CC1 ZINC000217920679 EI On-Demand Unstable SLC27A1 25 42 COc1ccc(/C=C/C(=O)NCc2nc(-c3ccc(C)cc3)no2)cc1 ZINC000217920685 EG In-Stock Unstable HDAC8 0 53 COc1ccc(/C=C/C(=O)NCc2nc(-c3ccc(C)cc3)no2)cc1 ZINC000217920685 EG In-Stock Unstable HDAC1 0 40 COc1ccc(/C=C/C(=O)NCc2nc(-c3ccc(C)cc3)no2)cc1 ZINC000217920685 EG In-Stock Unstable AXIN2 0 41 COc1ccc(/C=C/C(=O)NCc2nc(-c3ccc(C)cc3)no2)cc1 ZINC000217920685 EG In-Stock Unstable GPR183 0 43 Cn1c(C(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc2ccc(Cl)cc21 ZINC000217920770 GG In-Stock Unstable CHRNA4 28 46 O=C(NC12CC3CC(CC(C3)C1)C2)OCCCCCl ZINC000217920771 CH For-Sale Unstable EPHX2 97 50 O=C(NC12CC3CC(CC(C3)C1)C2)OCCCCCl ZINC000217920771 CH For-Sale Unstable P95276_MYCTO 0 40 O=C(NCC[C@H](O)C1CCOCC1)c1ccc(OC(F)(F)F)cc1 ZINC000217920777 EE In-Stock Unstable GCGR 38 41 O=C(NCC[C@H](O)C1CCOCC1)c1ccc(OC(F)(F)F)cc1 ZINC000217920777 EE In-Stock Unstable TRPV1 0 50 O=C(NCC[C@H](O)C1CCOCC1)c1ccc(OC(F)(F)F)cc1 ZINC000217920777 EE In-Stock Unstable CTSS 25 41 O=C(NCC[C@H](O)C1CCOCC1)c1ccc(OC(F)(F)F)cc1 ZINC000217920777 EE In-Stock Unstable GIPR 45 37 COc1ccc(/C=C/C(=O)NCc2nc(-c3cccc(OC)c3)no2)cc1 ZINC000217920804 FG In-Stock Unstable HDAC8 54 45 COc1ccc(/C=C/C(=O)NCc2nc(-c3cccc(OC)c3)no2)cc1 ZINC000217920804 FG In-Stock Unstable HDAC1 26 41 COc1ccc(/C=C/C(=O)NCc2nc(-c3cccc(OC)c3)no2)cc1 ZINC000217920804 FG In-Stock Unstable HDAC2 15 41 COc1ccc(/C=C/C(=O)NCc2nc(-c3cccc(OC)c3)no2)cc1 ZINC000217920804 FG In-Stock Unstable HDAC6 43 45 O=C(NCC[C@@H](O)C1CCOCC1)c1ccc(OC(F)(F)F)cc1 ZINC000217920864 EE In-Stock Unstable GCGR 38 41 O=C(NCC[C@@H](O)C1CCOCC1)c1ccc(OC(F)(F)F)cc1 ZINC000217920864 EE In-Stock Unstable TRPV1 0 50 O=C(NCC[C@@H](O)C1CCOCC1)c1ccc(OC(F)(F)F)cc1 ZINC000217920864 EE In-Stock Unstable CTSS 25 41 O=C(NCC[C@@H](O)C1CCOCC1)c1ccc(OC(F)(F)F)cc1 ZINC000217920864 EE In-Stock Unstable GIPR 45 37 CSCC[C@@H](CO)NC(=O)CC[C@@H]1NC(=O)N(CCc2ccccc2)C1=O ZINC000217920876 GD In-Stock Unstable PAM 0 41 COc1ccccc1NC(=O)OCCCCCl ZINC000217920891 CG For-Sale Unstable HRH3 15 44 COc1cccc(/C=C/C(=O)N[C@@H]2CCC[C@@H]2CO)c1 ZINC000217920899 CD On-Demand Unstable HD1B 0 42 O=C(Nc1nc2c(s1)CCCCC2)c1ccnc2ccccc12 ZINC000217920902 DI On-Demand Unstable FAP 0 44 O=C(Nc1nc2c(s1)CCCCC2)c1ccnc2ccccc12 ZINC000217920902 DI On-Demand Unstable SLC27A1 30 47 COc1ccc(/C=C/C(=O)NCc2nc(-c3ccc(OC)cc3)no2)cc1 ZINC000217920908 FG In-Stock Unstable HDAC8 0 56 COc1ccc(/C=C/C(=O)NCc2nc(-c3ccc(OC)cc3)no2)cc1 ZINC000217920908 FG In-Stock Unstable HDAC1 0 41 COc1ccc(/C=C/C(=O)NCc2nc(-c3ccc(OC)cc3)no2)cc1 ZINC000217920908 FG In-Stock Unstable HDAC2 19 46 COc1ccc(/C=C/C(=O)NCc2nc(-c3ccc(OC)cc3)no2)cc1 ZINC000217920908 FG In-Stock Unstable AXIN2 0 40 O=C(Cc1c(F)cccc1Cl)NCC[C@H](O)C1CCOCC1 ZINC000217920985 EE In-Stock Unstable P2RX7 15 43 Cc1ccc(NC(=O)c2cncc(/C=C\C(=O)O)c2)nc1 ZINC000217921006 CE For-Sale Unstable LUCI_LUCLA 43 43 CCS(=O)(=O)N1CCC(C(=O)Nc2nc3c(s2)CCCCC3)(c2ccccc2)CC1 ZINC000217921009 IH On-Demand Unstable SLC27A1 45 51 O=C(Nc1cccc2ccccc12)OCCCCCl ZINC000217921012 CI For-Sale Unstable TRPV1 32 44 COc1ccc(/C=C/C(=O)NCc2nc(-c3ccc(OC)cc3OC)no2)cc1 ZINC000217921017 GG In-Stock Unstable IMPDH2 0 42 COc1ccc(/C=C/C(=O)NCc2nc(-c3ccc(OC)cc3OC)no2)cc1 ZINC000217921017 GG In-Stock Unstable ABCG2 17 44 NC[C@@H]1CCC[C@@H]1N1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217921065 BF For-Sale Unstable CYP2D26 0 40 O=C(Cc1c(F)cccc1Cl)NCC[C@@H](O)C1CCOCC1 ZINC000217921071 EE In-Stock Unstable P2RX7 15 43 O=C(Nc1nc2c(s1)CCCCC2)c1ccccc1SCc1nnnn1-c1ccccc1 ZINC000217921094 JJ On-Demand Unstable SLC27A1 28 46 Cc1cccc(/C=C/NC(=O)N2CCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000217921137 EG For-Sale Unstable GPR119 34 50 NC[C@H]1CCC[C@@H]1N1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217921141 BF For-Sale Unstable CYP2D26 0 40 COc1ccc(/C=C/C(=O)NCc2nc(-c3ccc(Cl)cc3)no2)cc1 ZINC000217921150 FH In-Stock Unstable PTGS2 0 40 COc1ccc(/C=C/C(=O)NCc2nc(-c3ccc(Cl)cc3)no2)cc1 ZINC000217921150 FH In-Stock Unstable HDAC8 0 52 COc1ccc(/C=C/C(=O)NCc2nc(-c3ccc(Cl)cc3)no2)cc1 ZINC000217921150 FH In-Stock Unstable HDAC1 0 41 COc1ccc(/C=C/C(=O)NCc2nc(-c3ccc(Cl)cc3)no2)cc1 ZINC000217921150 FH In-Stock Unstable HDAC2 20 45 COc1ccc(/C=C/C(=O)NCc2nc(-c3ccc(Cl)cc3)no2)cc1 ZINC000217921150 FH In-Stock Unstable PDK1 34 40 COC(=O)C[C@H](c1cc(OC)c(OC)c(OC)c1)c1c(Cc2ccc3c(c2)CCC(C)(C)O3)[nH][nH]c1=O ZINC000217921203 KI In-Stock Unstable NDUFA4 0 45 O=C(CCn1cnc2ccccc21)Nc1nc2c(s1)CCCCC2 ZINC000217921205 EH On-Demand Unstable SLC27A1 45 50 NC[C@@H]1CCC[C@H]1N1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217921208 BF For-Sale Unstable CYP2D26 0 40 Cc1cccc(/C=C/NC(=O)NC2CCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000217921236 FH For-Sale Unstable GPR119 37 53 C[C@@H]1CCC[C@@H](CNc2ccccn2)C1 ZINC000217921238 BG On-Demand Unstable GPR39 0 47 COc1ccc(/C=C/C(=O)NCc2nc(-c3cccc(Br)c3)no2)cc1 ZINC000217921261 HH In-Stock Unstable HDAC8 56 46 COc1ccc(/C=C/C(=O)NCc2nc(-c3cccc(Br)c3)no2)cc1 ZINC000217921261 HH In-Stock Unstable HDAC1 25 41 COc1ccc(/C=C/C(=O)NCc2nc(-c3cccc(Br)c3)no2)cc1 ZINC000217921261 HH In-Stock Unstable HDAC6 43 46 CCN1CCC[C@H](NC(=O)[C@@H](N)CC(N)=O)C1 ZINC000217921273 BA On-Demand Unstable BIRC2 42 35 COC(=O)C[C@@H](c1cc(OC)c(OC)c(OC)c1)c1c(Cc2ccc3c(c2)CCC(C)(C)O3)[nH][nH]c1=O ZINC000217921297 KI In-Stock Unstable NDUFA4 0 45 O=C(Nc1ccc(F)cc1[N+](=O)[O-])NC1CCCCC1 ZINC000217921299 CG For-Sale Unstable EPHX2 30 55 C[C@H]1CCC[C@@H](CNc2ccccn2)C1 ZINC000217921317 BG On-Demand Unstable GPR39 0 47 CCN1CCC[C@@H](NC(=O)[C@@H](N)CC(N)=O)C1 ZINC000217921355 BA On-Demand Unstable BIRC2 42 35 COc1cccc(/C=C/NC(=O)Nc2ccc(OC)c(OC)c2)c1 ZINC000217921356 EH For-Sale Unstable CYP1B1 56 40 COc1cccc(/C=C/NC(=O)Nc2ccc(OC)c(OC)c2)c1 ZINC000217921356 EH For-Sale Unstable KDR 25 43 COc1cccc(/C=C/NC(=O)Nc2ccc(OC)c(OC)c2)c1 ZINC000217921356 EH For-Sale Unstable MTNR1A 30 46 COc1cccc(/C=C/NC(=O)Nc2ccc(OC)c(OC)c2)c1 ZINC000217921356 EH For-Sale Unstable MTNR1B 37 46 COc1cccc(/C=C/NC(=O)Nc2ccc(OC)c(OC)c2)c1 ZINC000217921356 EH For-Sale Unstable CYP1A1 40 44 COc1cccc(/C=C/NC(=O)Nc2ccc(OC)c(OC)c2)c1 ZINC000217921356 EH For-Sale Unstable PDGFRA 42 43 COc1cccc(/C=C/NC(=O)Nc2ccc(OC)c(OC)c2)c1 ZINC000217921356 EH For-Sale Unstable IMPDH2 0 45 COc1cccc(/C=C/NC(=O)Nc2ccc(OC)c(OC)c2)c1 ZINC000217921356 EH For-Sale Unstable Q8MMZ8_EIMTE 0 44 COc1cccc(/C=C/NC(=O)Nc2ccc(OC)c(OC)c2)c1 ZINC000217921356 EH For-Sale Unstable ABCG2 24 45 COc1cccc(/C=C/NC(=O)Nc2ccc(OC)c(OC)c2)c1 ZINC000217921356 EH For-Sale Unstable ENPP1 71 35 COc1ccc(/C=C/C(=O)N(C)Cc2nc(-c3ccc(C)cc3)no2)cc1 ZINC000217921385 FH In-Stock Unstable AXIN2 0 40 COc1ccc(/C=C/C(=O)N(C)Cc2nc(-c3ccc(C)cc3)no2)cc1 ZINC000217921385 FH In-Stock Unstable GPR183 0 42 C[C@@H]1CCC[C@H](CNc2ccccn2)C1 ZINC000217921403 BG On-Demand Unstable GPR39 0 47 CC(C)(C)NC(=O)Nc1ccc(F)cc1[N+](=O)[O-] ZINC000217921408 CF For-Sale Unstable COLA 15 40 Cn1cc(Br)cc1C(=O)Nc1nc2c(s1)CCCCC2 ZINC000217921473 FH On-Demand Unstable SLC27A1 29 40 Cc1ccc(CN2CC[C@@H](N)[C@@H](C)C2)cn1 ZINC000217921481 BD On-Demand Unstable PDE1C 20 42 COc1ccc(/C=C/C(=O)N(C)Cc2nc(-c3cccc(OC)c3)no2)cc1 ZINC000217921483 GG In-Stock Unstable FABI 40 30 COc1ccc(/C=C/C(=O)N(C)Cc2nc(-c3cccc(OC)c3)no2)cc1 ZINC000217921483 GG In-Stock Unstable HSD17B2 18 41 COc1cccc(/C=C/NC(=O)NCCCN2CCCC2=O)c1 ZINC000217921484 DD For-Sale Unstable DRD4 47 36 COc1cccc(/C=C/NC(=O)NCCCN2CCCC2=O)c1 ZINC000217921484 DD For-Sale Unstable HRH2 28 42 COc1cccc(/C=C/NC(=O)NCCCN2CCCC2=O)c1 ZINC000217921484 DD For-Sale Unstable NQO2 15 47 COc1cccc(/C=C/NC(=O)NCCCN2CCCC2=O)c1 ZINC000217921484 DD For-Sale Unstable MTR1B_CHICK 0 47 COc1cccc(/C=C/NC(=O)NCCCN2CCCC2=O)c1 ZINC000217921484 DD For-Sale Unstable CCR3 16 42 COc1cccc(/C=C/NC(=O)NCCCN2CCCC2=O)c1 ZINC000217921484 DD For-Sale Unstable MTNR1A 43 47 COc1cccc(/C=C/NC(=O)NCCCN2CCCC2=O)c1 ZINC000217921484 DD For-Sale Unstable MTNR1B 44 41 COc1cccc(/C=C/NC(=O)NCCCN2CCCC2=O)c1 ZINC000217921484 DD For-Sale Unstable TYRO3 24 41 C[C@H]1CCC[C@H](CNc2ccccn2)C1 ZINC000217921490 BG On-Demand Unstable GPR39 0 47 C[C@@H](CCc1ccc(O)cc1)N1CC[C@@H]2CCCC[C@@H]21 ZINC000217921522 CH For-Sale Unstable BIRC2 47 38 CCCNC(=O)Nc1ccc(F)cc1[N+](=O)[O-] ZINC000217921542 BE For-Sale Unstable COLA 15 41 CCN1CCC[C@H](NC(=O)C[C@@H](N)c2ccccc2)C1 ZINC000217921554 CD On-Demand Unstable CHRM1 26 42 CCN1CCC[C@H](NC(=O)C[C@@H](N)c2ccccc2)C1 ZINC000217921554 CD On-Demand Unstable SLC6A1 54 37 CCN1CCC[C@H](NC(=O)C[C@@H](N)c2ccccc2)C1 ZINC000217921554 CD On-Demand Unstable SIGMAR1 22 41 CCN1CCC[C@H](NC(=O)C[C@@H](N)c2ccccc2)C1 ZINC000217921554 CD On-Demand Unstable XIAP 48 39 CCN1CCC[C@H](NC(=O)C[C@@H](N)c2ccccc2)C1 ZINC000217921554 CD On-Demand Unstable BIRC2 54 46 NC[C@@H]1CCCC[C@@H]1N1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217921560 CG For-Sale Unstable CYP2D26 0 41 Cc1ccc(CN2CC[C@H](N)[C@@H](C)C2)cn1 ZINC000217921567 BD On-Demand Unstable PDE1C 20 42 O=C(N[C@@H](C(=O)Nc1nc2c(s1)CCCCC2)c1ccccc1)c1ccccc1 ZINC000217921576 HJ On-Demand Unstable MTTP 66 37 O=C(N[C@@H](C(=O)Nc1nc2c(s1)CCCCC2)c1ccccc1)c1ccccc1 ZINC000217921576 HJ On-Demand Unstable SLC27A1 29 46 C[C@@H]1CCC[C@@H](CNc2ncccn2)C1 ZINC000217921592 BF On-Demand Unstable GRIN2B 15 40 C[C@@H]1CCC[C@@H](CNc2ncccn2)C1 ZINC000217921592 BF On-Demand Unstable GPR39 0 40 COc1cccc(/C=C/NC(=O)Nc2ccc(Br)cc2)c1 ZINC000217921594 EI For-Sale Unstable MTNR1A 28 50 COc1cccc(/C=C/NC(=O)Nc2ccc(Br)cc2)c1 ZINC000217921594 EI For-Sale Unstable MTNR1B 34 50 COc1cccc(/C=C/NC(=O)Nc2ccc(Br)cc2)c1 ZINC000217921594 EI For-Sale Unstable FPR2 17 40 COc1cccc(/C=C/NC(=O)Nc2ccc(Br)cc2)c1 ZINC000217921594 EI For-Sale Unstable AKR1C3 17 41 COc1cccc(/C=C/NC(=O)Nc2ccc(Br)cc2)c1 ZINC000217921594 EI For-Sale Unstable AKR1C2 45 41 C[C@H](CCc1ccc(O)cc1)N1CC[C@@H]2CCCC[C@@H]21 ZINC000217921603 CH For-Sale Unstable BIRC2 47 38 COc1ccc(/C=C/C(=O)N(C)Cc2nc(-c3ccc(OC)cc3)no2)cc1 ZINC000217921606 GG In-Stock Unstable AXIN2 0 40 COc1ccc([C@@H]2CC(=O)Oc3c2c(=O)oc2ccccc32)cc1OC ZINC000217921629 FG In-Stock Unstable CYP1B1 46 35 CCN1CCC[C@@H](NC(=O)C[C@@H](N)c2ccccc2)C1 ZINC000217921637 CD On-Demand Unstable CHRM1 26 42 CCN1CCC[C@@H](NC(=O)C[C@@H](N)c2ccccc2)C1 ZINC000217921637 CD On-Demand Unstable SLC6A1 54 37 CCN1CCC[C@@H](NC(=O)C[C@@H](N)c2ccccc2)C1 ZINC000217921637 CD On-Demand Unstable SIGMAR1 22 41 CCN1CCC[C@@H](NC(=O)C[C@@H](N)c2ccccc2)C1 ZINC000217921637 CD On-Demand Unstable XIAP 48 39 CCN1CCC[C@@H](NC(=O)C[C@@H](N)c2ccccc2)C1 ZINC000217921637 CD On-Demand Unstable BIRC2 54 46 NC[C@H]1CCCC[C@@H]1N1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217921638 CG For-Sale Unstable CYP2D26 0 41 CN[C@@H]1CCN(Cc2ccc(C)nc2)C[C@@H]1C ZINC000217921644 BD For-Sale Unstable PDE1C 28 43 CN[C@@H]1CCN(Cc2ccc(C)nc2)C[C@@H]1C ZINC000217921644 BD For-Sale Unstable PDE9A 0 43 C[C@H]1CCC[C@@H](CNc2ncccn2)C1 ZINC000217921664 BF On-Demand Unstable GRIN2B 15 40 C[C@H]1CCC[C@@H](CNc2ncccn2)C1 ZINC000217921664 BF On-Demand Unstable GPR39 0 40 O=C(N[C@H](C(=O)Nc1nc2c(s1)CCCCC2)c1ccccc1)c1ccccc1 ZINC000217921667 HJ On-Demand Unstable MTTP 66 37 O=C(N[C@H](C(=O)Nc1nc2c(s1)CCCCC2)c1ccccc1)c1ccccc1 ZINC000217921667 HJ On-Demand Unstable SLC27A1 29 46 COc1cccc(/C=C/NC(=O)Nc2cccc(C(=O)O)c2)c1 ZINC000217921699 DG For-Sale Unstable DRD4 40 30 COc1cccc(/C=C/NC(=O)Nc2cccc(C(=O)O)c2)c1 ZINC000217921699 DG For-Sale Unstable CYP1B1 21 40 COc1cccc(/C=C/NC(=O)Nc2cccc(C(=O)O)c2)c1 ZINC000217921699 DG For-Sale Unstable MTNR1A 25 45 COc1cccc(/C=C/NC(=O)Nc2cccc(C(=O)O)c2)c1 ZINC000217921699 DG For-Sale Unstable MTNR1B 31 45 COc1cccc(/C=C/NC(=O)Nc2cccc(C(=O)O)c2)c1 ZINC000217921699 DG For-Sale Unstable NR1H4 25 46 COc1cccc(/C=C/NC(=O)Nc2cccc(C(=O)O)c2)c1 ZINC000217921699 DG For-Sale Unstable CCKBR 15 47 COc1cccc(/C=C/NC(=O)Nc2cccc(C(=O)O)c2)c1 ZINC000217921699 DG For-Sale Unstable EPHX2 19 41 COc1cccc(/C=C/NC(=O)Nc2cccc(C(=O)O)c2)c1 ZINC000217921699 DG For-Sale Unstable TTR 0 40 COc1cccc(/C=C/NC(=O)Nc2cccc(C(=O)O)c2)c1 ZINC000217921699 DG For-Sale Unstable Q8MMZ8_EIMTE 0 43 COc1cccc(/C=C/NC(=O)Nc2cccc(C(=O)O)c2)c1 ZINC000217921699 DG For-Sale Unstable TAAR1 37 41 COc1cccc(/C=C/NC(=O)Nc2cccc(C(=O)O)c2)c1 ZINC000217921699 DG For-Sale Unstable AKR1C3 58 53 COc1cccc(/C=C/NC(=O)Nc2cccc(C(=O)O)c2)c1 ZINC000217921699 DG For-Sale Unstable AKR1C2 48 38 COc1cccc(/C=C/NC(=O)Nc2cccc(C(=O)O)c2)c1 ZINC000217921699 DG For-Sale Unstable IMDH_CRYPV 41 39 COc1cccc(/C=C/NC(=O)Nc2cccc(C(=O)O)c2)c1 ZINC000217921699 DG For-Sale Unstable KCNK3 79 49 COc1cccc(/C=C/NC(=O)Nc2cccc(C(=O)O)c2)c1 ZINC000217921699 DG For-Sale Unstable KCNK9 48 33 COc1ccc([C@H]2CC(=O)Oc3c2c(=O)oc2ccccc32)cc1OC ZINC000217921709 FG In-Stock Unstable CYP1B1 46 35 NC[C@@H]1CCCC[C@H]1N1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217921722 CG For-Sale Unstable CYP2D26 0 41 CC(C)CCCCCCNC(=O)NC1CCCCC1 ZINC000217921723 CI For-Sale Unstable EPHX2 36 70 CN[C@H]1CCN(Cc2ccc(C)nc2)C[C@@H]1C ZINC000217921728 BD For-Sale Unstable PDE1C 28 43 CN[C@H]1CCN(Cc2ccc(C)nc2)C[C@@H]1C ZINC000217921728 BD For-Sale Unstable PDE9A 0 43 C[C@@H]1CCC[C@H](CNc2ncccn2)C1 ZINC000217921744 BF On-Demand Unstable GRIN2B 15 40 C[C@@H]1CCC[C@H](CNc2ncccn2)C1 ZINC000217921744 BF On-Demand Unstable GPR39 0 40 O=C(c1cccc(Cn2cccn2)c1)N1CCn2nc(CO)cc2C1 ZINC000217921752 ED In-Stock Unstable FABI 41 35 O=C(CCc1ccc(C(F)(F)F)cc1)NCC[C@H](O)C1CCOCC1 ZINC000217921779 FF In-Stock Unstable LUXR 31 41 CCN1CCC[C@H](NC(=O)[C@@H](N)CCS(C)(=O)=O)C1 ZINC000217921799 CB For-Sale Unstable BIRC2 41 35 C[C@H]1CCC[C@H](CNc2ncccn2)C1 ZINC000217921804 BF On-Demand Unstable GRIN2B 15 40 C[C@H]1CCC[C@H](CNc2ncccn2)C1 ZINC000217921804 BF On-Demand Unstable GPR39 0 40 COc1ccc(/C=C/C(=O)N(C)Cc2nc(-c3ccccc3Cl)no2)cc1 ZINC000217921808 GI In-Stock Unstable GPBAR1 24 46 COc1cccc(/C=C/NC(=O)Nc2ccccc2[N+](=O)[O-])c1 ZINC000217921813 DG For-Sale Unstable TAAR1 26 44 COc1cccc(/C=C/NC(=O)Nc2ccccc2[N+](=O)[O-])c1 ZINC000217921813 DG For-Sale Unstable AKR1C2 26 43 CNC[C@@H](C)c1ccc(CN2CCCCC[C@@H]2C)cc1 ZINC000217921826 CH For-Sale Unstable HRH3 36 53 CCOC(=O)CNC(=O)NCCCCCCC(C)C ZINC000217921839 CE For-Sale Unstable EPHX2 54 43 O=C(CCc1ccc(C(F)(F)F)cc1)NCC[C@@H](O)C1CCOCC1 ZINC000217921871 FF In-Stock Unstable LUXR 31 41 CCN1CCC[C@@H](NC(=O)[C@@H](N)CCS(C)(=O)=O)C1 ZINC000217921900 CB For-Sale Unstable BIRC2 41 35 O=C(Nc1nc2c(s1)CCCCC2)c1occc1CSc1ccccc1 ZINC000217921902 GK On-Demand Unstable SLC27A1 28 45 COC(=O)c1cc(CN2CCC(N)CC2)cc(C(=O)NCCOCCO)c1 ZINC000217921904 GC For-Sale Unstable ACHE 15 42 COC(=O)c1cc(CN2CCC(N)CC2)cc(C(=O)NCCOCCO)c1 ZINC000217921904 GC For-Sale Unstable SSTR5 43 34 COC(=O)c1cc(CN2CCC(N)CC2)cc(C(=O)NCCOCCO)c1 ZINC000217921904 GC For-Sale Unstable CACNA1I 68 42 C[C@H](CN)c1ccc(CN2CCCCC[C@@H]2C)cc1 ZINC000217921941 CH For-Sale Unstable HRH3 39 56 COc1cccc(/C=C/NC(=O)Nc2cccc(O)c2)c1 ZINC000217921943 CG For-Sale Unstable MTNR1A 29 47 COc1cccc(/C=C/NC(=O)Nc2cccc(O)c2)c1 ZINC000217921943 CG For-Sale Unstable MTNR1B 33 47 COc1cccc(/C=C/NC(=O)Nc2cccc(O)c2)c1 ZINC000217921943 CG For-Sale Unstable TAAR1 30 40 COc1cccc(/C=C/NC(=O)Nc2cccc(O)c2)c1 ZINC000217921943 CG For-Sale Unstable KCNK3 29 42 COc1cccc(/C=C/NC(=O)Nc2ccc(C)cc2)c1 ZINC000217922049 CH For-Sale Unstable KIT 23 42 COc1cccc(/C=C/NC(=O)Nc2ccc(C)cc2)c1 ZINC000217922049 CH For-Sale Unstable CYP1B1 15 40 COc1cccc(/C=C/NC(=O)Nc2ccc(C)cc2)c1 ZINC000217922049 CH For-Sale Unstable KDR 21 42 COc1cccc(/C=C/NC(=O)Nc2ccc(C)cc2)c1 ZINC000217922049 CH For-Sale Unstable MTNR1A 31 51 COc1cccc(/C=C/NC(=O)Nc2ccc(C)cc2)c1 ZINC000217922049 CH For-Sale Unstable MTNR1B 36 51 COc1cccc(/C=C/NC(=O)Nc2ccc(C)cc2)c1 ZINC000217922049 CH For-Sale Unstable TEK 24 42 COc1cccc(/C=C/NC(=O)Nc2ccc(C)cc2)c1 ZINC000217922049 CH For-Sale Unstable Q8MMZ8_EIMTE 0 45 COc1cccc(/C=C/NC(=O)Nc2ccc(C)cc2)c1 ZINC000217922049 CH For-Sale Unstable AKR1C3 17 40 COc1cccc(/C=C/NC(=O)Nc2ccc(C)cc2)c1 ZINC000217922049 CH For-Sale Unstable AKR1C2 41 38 COc1cccc(/C=C/NC(=O)Nc2ccc(C)cc2)c1 ZINC000217922049 CH For-Sale Unstable KCNK3 26 42 CCCCNC(=O)NCCCCCCC(C)C ZINC000217922077 BH For-Sale Unstable CPT1A 23 43 CCCCNC(=O)NCCCCCCC(C)C ZINC000217922077 BH For-Sale Unstable EPHX2 71 48 CCCCNC(=O)NCCCCCCC(C)C ZINC000217922077 BH For-Sale Unstable Q6UB75_PIG 0 40 CCCCNC(=O)NCCCCCCC(C)C ZINC000217922077 BH For-Sale Unstable ASAH1 79 33 CCCCNC(=O)NCCCCCCC(C)C ZINC000217922077 BH For-Sale Unstable ACAT 0 41 CCCCNC(=O)NCCCCCCC(C)C ZINC000217922077 BH For-Sale Unstable NOD1 62 43 CCCCNC(=O)NCCCCCCC(C)C ZINC000217922077 BH For-Sale Unstable CQSS 52 34 CC(C)(C)OC(=O)NC1CCN(Cc2ccc(OCCOCCOCCOCCN=[N+]=[N-])cc2)CC1 ZINC000217922104 KH For-Sale Unstable LTA4H 26 41 CC(C)(C)OC(=O)NC1CCN(Cc2ccc(OCCOCCOCCOCCN=[N+]=[N-])cc2)CC1 ZINC000217922104 KH For-Sale Unstable HRH3 16 44 CC(C)(C)OC(=O)NC1CCN(Cc2ccc(OCCOCCOCCOCCN=[N+]=[N-])cc2)CC1 ZINC000217922104 KH For-Sale Unstable SIGMAR1 23 43 CC(C)(C)OC(=O)NC1CCN(Cc2ccc(OCCOCCOCCOCCN=[N+]=[N-])cc2)CC1 ZINC000217922104 KH For-Sale Unstable SSTR5 48 38 CC(C)(C)OC(=O)NC1CCN(Cc2ccc(OCCOCCOCCOCCN=[N+]=[N-])cc2)CC1 ZINC000217922104 KH For-Sale Unstable SLC6A5 30 41 CC(C)(C)OC(=O)NC1CCN(Cc2ccc(OCCOCCOCCOCCN=[N+]=[N-])cc2)CC1 ZINC000217922104 KH For-Sale Unstable MCHR1 34 45 COc1ccc(/C=C/C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217922124 EJ In-Stock Unstable DRD3 15 50 COc1ccc(/C=C/C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217922124 EJ In-Stock Unstable PTAFR 18 43 COc1ccc(/C=C/C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217922124 EJ In-Stock Unstable BMP1 28 41 COc1ccc(/C=C/C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217922124 EJ In-Stock Unstable PYGL 0 43 COc1ccc(/C=C/C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217922124 EJ In-Stock Unstable HDAC8 30 48 COc1ccc(/C=C/C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217922124 EJ In-Stock Unstable HDAC1 24 41 COc1ccc(/C=C/C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217922124 EJ In-Stock Unstable HDAC2 0 41 COc1ccc(/C=C/C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217922124 EJ In-Stock Unstable HDAC4 0 41 COc1ccc(/C=C/C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217922124 EJ In-Stock Unstable HDAC6 16 48 COc1ccc(/C=C/C(=O)NCCCc2ccc(C(C)C)cc2)cc1 ZINC000217922124 EJ In-Stock Unstable HDAC7 40 36 Cc1nc(-c2cccs2)ccc1C(=O)Nc1nc2c(s1)CCCCC2 ZINC000217922134 FK On-Demand Unstable SLC27A1 28 41 O=C(O)/C=C\c1cncc(C(=O)NCC2CCCC2)c1 ZINC000217922148 CE For-Sale Unstable CACNA1I 55 35 COc1cccc(/C=C/NC(=O)NCCC(=O)O)c1 ZINC000217922163 CD For-Sale Unstable DRD4 42 32 COc1cccc(/C=C/NC(=O)NCCC(=O)O)c1 ZINC000217922163 CD For-Sale Unstable MTNR1A 86 45 COc1cccc(/C=C/NC(=O)NCCC(=O)O)c1 ZINC000217922163 CD For-Sale Unstable MTNR1B 78 45 CCCNC(=O)NCCCCCCC(C)C ZINC000217922200 BG On-Demand Unstable EPHX2 23 43 CNC[C@@H](C)c1ccc(CN2CC[C@@H](COC)C2)cc1 ZINC000217922212 CE For-Sale Unstable SIGMAR1 20 42 CCN1CCC[C@H](NC(=O)[C@@](C)(N)C2CC2)C1 ZINC000217922225 BC For-Sale Unstable BIRC2 40 35 COc1ccc(/C=C/C(=O)NCCCN(C)c2ccccc2)cc1 ZINC000217922243 DG In-Stock Unstable PTGS2 0 50 COc1ccc(/C=C/C(=O)NCCCN(C)c2ccccc2)cc1 ZINC000217922243 DG In-Stock Unstable DRD3 18 53 COc1ccc(/C=C/C(=O)NCCCN(C)c2ccccc2)cc1 ZINC000217922243 DG In-Stock Unstable PYGL 22 42 COc1ccc(/C=C/C(=O)NCCCN(C)c2ccccc2)cc1 ZINC000217922243 DG In-Stock Unstable HDAC8 32 49 COc1ccc(/C=C/C(=O)NCCCN(C)c2ccccc2)cc1 ZINC000217922243 DG In-Stock Unstable MMP2 20 52 COc1ccc(/C=C/C(=O)NCCCN(C)c2ccccc2)cc1 ZINC000217922243 DG In-Stock Unstable HDAC1 26 41 COc1ccc(/C=C/C(=O)NCCCN(C)c2ccccc2)cc1 ZINC000217922243 DG In-Stock Unstable HDAC2 24 43 COc1ccc(/C=C/C(=O)NCCCN(C)c2ccccc2)cc1 ZINC000217922243 DG In-Stock Unstable HDAC4 24 43 COc1ccc(/C=C/C(=O)NCCCN(C)c2ccccc2)cc1 ZINC000217922243 DG In-Stock Unstable HDAC6 29 49 COc1ccc(/C=C/C(=O)NCCCN(C)c2ccccc2)cc1 ZINC000217922243 DG In-Stock Unstable MMP9 25 52 COc1ccc(/C=C/C(=O)NCCCN(C)c2ccccc2)cc1 ZINC000217922243 DG In-Stock Unstable HDAC9 40 43 COc1ccc(/C=C/C(=O)NCCCN(C)c2ccccc2)cc1 ZINC000217922243 DG In-Stock Unstable HDAC7 51 43 COc1ccc(/C=C/C(=O)NCCCN(C)c2ccccc2)cc1 ZINC000217922243 DG In-Stock Unstable GPR183 0 43 O=C(O)/C=C\c1cncc(C(=O)NCc2ccncc2)c1 ZINC000217922245 CD For-Sale Unstable NAMPT 57 39 COc1cccc(/C=C/NC(=O)Nc2ccc(N)cc2)c1 ZINC000217922270 CG For-Sale Unstable KIT 16 43 COc1cccc(/C=C/NC(=O)Nc2ccc(N)cc2)c1 ZINC000217922270 CG For-Sale Unstable KDR 18 40 COc1cccc(/C=C/NC(=O)Nc2ccc(N)cc2)c1 ZINC000217922270 CG For-Sale Unstable MTNR1A 31 50 COc1cccc(/C=C/NC(=O)Nc2ccc(N)cc2)c1 ZINC000217922270 CG For-Sale Unstable MTNR1B 34 50 COc1cccc(/C=C/NC(=O)Nc2ccc(N)cc2)c1 ZINC000217922270 CG For-Sale Unstable ACR 30 41 COc1cccc(/C=C/NC(=O)Nc2ccc(N)cc2)c1 ZINC000217922270 CG For-Sale Unstable AKR1C2 40 32 CNC[C@H](C)c1ccc(CN2CC[C@@H](COC)C2)cc1 ZINC000217922288 CE For-Sale Unstable SIGMAR1 20 42 CCN1CCC[C@@H](NC(=O)[C@@](C)(N)C2CC2)C1 ZINC000217922310 BC For-Sale Unstable BIRC2 40 35 CN(Cc1cnccn1)C(=O)c1cc(=O)n(-c2ccccc2)[nH]1 ZINC000217922322 DD In-Stock Unstable CTSA 55 42 CN1CCCN(Cc2ccccc2)C[C@@H]1C(=O)O ZINC000217922328 BD For-Sale Unstable ACE 67 38 CN1CCCN(Cc2ccccc2)C[C@@H]1C(=O)O ZINC000217922328 BD For-Sale Unstable DRD2 30 44 CN1CCCN(Cc2ccccc2)C[C@@H]1C(=O)O ZINC000217922328 BD For-Sale Unstable DRD4 53 44 CN1CCCN(Cc2ccccc2)C[C@@H]1C(=O)O ZINC000217922328 BD For-Sale Unstable ACHE 34 40 CN1CCCN(Cc2ccccc2)C[C@@H]1C(=O)O ZINC000217922328 BD For-Sale Unstable HTR2A 15 41 CN1CCCN(Cc2ccccc2)C[C@@H]1C(=O)O ZINC000217922328 BD For-Sale Unstable SLC6A1 119 40 CN1CCCN(Cc2ccccc2)C[C@@H]1C(=O)O ZINC000217922328 BD For-Sale Unstable DRD3 36 42 CN1CCCN(Cc2ccccc2)C[C@@H]1C(=O)O ZINC000217922328 BD For-Sale Unstable FABP4 40 38 CN1CCCN(Cc2ccccc2)C[C@@H]1C(=O)O ZINC000217922328 BD For-Sale Unstable HRH3 28 42 CN1CCCN(Cc2ccccc2)C[C@@H]1C(=O)O ZINC000217922328 BD For-Sale Unstable SIGMAR1 76 52 CN1CCCN(Cc2ccccc2)C[C@@H]1C(=O)O ZINC000217922328 BD For-Sale Unstable BCHE 16 40 CN1CCCN(Cc2ccccc2)C[C@@H]1C(=O)O ZINC000217922328 BD For-Sale Unstable SLC18A3 23 41 CN1CCCN(Cc2ccccc2)C[C@@H]1C(=O)O ZINC000217922328 BD For-Sale Unstable NPFFR1 48 37 NC(=O)[C@H]1CCCN1C(=O)c1cncc(/C=C\C(=O)O)c1 ZINC000217922329 CC For-Sale Unstable PREP 47 40 COc1ccc(/C=C/C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217922363 FH In-Stock Unstable DRD2 28 60 COc1ccc(/C=C/C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217922363 FH In-Stock Unstable DRD4 40 33 COc1ccc(/C=C/C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217922363 FH In-Stock Unstable DRD3 45 60 COc1ccc(/C=C/C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217922363 FH In-Stock Unstable PYGL 23 40 COc1ccc(/C=C/C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217922363 FH In-Stock Unstable HDAC8 21 41 COc1ccc(/C=C/C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217922363 FH In-Stock Unstable HDAC1 28 40 COc1ccc(/C=C/C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217922363 FH In-Stock Unstable HDAC4 0 40 COc1ccc(/C=C/C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217922363 FH In-Stock Unstable HDAC6 16 41 COc1ccc(/C=C/C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217922363 FH In-Stock Unstable MMP9 27 42 COc1ccc(/C=C/C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217922363 FH In-Stock Unstable GPR183 0 42 COc1cccc(/C=C/NC(=O)N(C(C)=O)c2ccc(N)cc2)c1 ZINC000217922370 EG For-Sale Unstable MTNR1A 22 45 COc1cccc(/C=C/NC(=O)N(C(C)=O)c2ccc(N)cc2)c1 ZINC000217922370 EG For-Sale Unstable MTNR1B 27 45 Cc1cc(NC(=O)COc2cccc3ccccc23)n(-c2ccc([N+](=O)[O-])cc2)n1 ZINC000217922403 HI On-Demand Unstable TNF 46 35 Cc1cc(NC(=O)COc2cccc3ccccc23)n(-c2ccc([N+](=O)[O-])cc2)n1 ZINC000217922403 HI On-Demand Unstable DDR2 18 44 COC[C@@H]1CCN(Cc2ccc([C@@H](C)CN)cc2)C1 ZINC000217922420 CE For-Sale Unstable SLC6A3 15 42 COC[C@@H]1CCN(Cc2ccc([C@@H](C)CN)cc2)C1 ZINC000217922420 CE For-Sale Unstable SIGMAR1 19 40 NC(=O)[C@@H]1CCCN1C(=O)c1cncc(/C=C\C(=O)O)c1 ZINC000217922422 CC For-Sale Unstable PREP 47 40 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922447 BD For-Sale Unstable ACE 23 40 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922447 BD For-Sale Unstable ELANE 34 43 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922447 BD For-Sale Unstable CTRA_BOVIN 40 31 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922447 BD For-Sale Unstable HRAS 41 33 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922447 BD For-Sale Unstable CASP3 18 44 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922447 BD For-Sale Unstable BMP1 65 38 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922447 BD For-Sale Unstable GALR1 43 30 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922447 BD For-Sale Unstable KLK3 74 40 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922447 BD For-Sale Unstable CTSB 61 42 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922447 BD For-Sale Unstable PAPA1_CARPA 62 34 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922447 BD For-Sale Unstable CYSP_TRYCR 61 42 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922447 BD For-Sale Unstable CTSK 43 49 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922447 BD For-Sale Unstable CTSL 43 46 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922447 BD For-Sale Unstable PGA 21 40 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922447 BD For-Sale Unstable CAPNS1 66 40 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922447 BD For-Sale Unstable MMP11 40 33 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922447 BD For-Sale Unstable CTSS 25 45 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922447 BD For-Sale Unstable CAPN1 93 48 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922447 BD For-Sale Unstable CASP1 27 42 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922447 BD For-Sale Unstable CAPN2 122 43 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922447 BD For-Sale Unstable PLAU 15 41 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922447 BD For-Sale Unstable CASP6 24 42 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922447 BD For-Sale Unstable CASP9 31 42 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922447 BD For-Sale Unstable NPR 66 39 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922447 BD For-Sale Unstable PSMB5 49 40 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922447 BD For-Sale Unstable BIRC2 34 40 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922447 BD For-Sale Unstable MBTPS1 40 35 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922447 BD For-Sale Unstable Q9NAW4_PLAFA 35 41 COC(=O)[C@@H]1[C@@H]2CC(=O)[C@@H]1C[C@@H]2Br ZINC000217922451 BD In-Stock Unstable SLC6A1 48 33 C=COCCCNC(=O)NC1CCCCC1 ZINC000217922469 BE For-Sale Unstable EPHX2 23 71 COc1cccc(/C=C/NC(=O)Nc2ccc(NC(C)=O)cc2)c1 ZINC000217922472 EG For-Sale Unstable CYP1B1 31 42 COc1cccc(/C=C/NC(=O)Nc2ccc(NC(C)=O)cc2)c1 ZINC000217922472 EG For-Sale Unstable MTNR1A 46 60 COc1cccc(/C=C/NC(=O)Nc2ccc(NC(C)=O)cc2)c1 ZINC000217922472 EG For-Sale Unstable MTNR1B 48 60 COc1cccc(/C=C/NC(=O)Nc2ccc(NC(C)=O)cc2)c1 ZINC000217922472 EG For-Sale Unstable CYP1A1 21 42 COc1cccc(/C=C/NC(=O)Nc2ccc(NC(C)=O)cc2)c1 ZINC000217922472 EG For-Sale Unstable ACR 20 41 COc1cccc(/C=C/NC(=O)Nc2ccc(NC(C)=O)cc2)c1 ZINC000217922472 EG For-Sale Unstable Q8MMZ8_EIMTE 0 47 COc1cccc(/C=C/NC(=O)Nc2ccc(NC(C)=O)cc2)c1 ZINC000217922472 EG For-Sale Unstable TAAR1 28 40 COc1cccc(/C=C/NC(=O)Nc2ccc(NC(C)=O)cc2)c1 ZINC000217922472 EG For-Sale Unstable IDO1 29 41 COc1cccc(/C=C/NC(=O)Nc2ccc(NC(C)=O)cc2)c1 ZINC000217922472 EG For-Sale Unstable AKR1C2 45 34 COc1cccc(/C=C/NC(=O)Nc2ccc(NC(C)=O)cc2)c1 ZINC000217922472 EG For-Sale Unstable IMDH_CRYPV 17 40 COc1ccc(/C=C/C(=O)NCc2ccc(OC)c(OC)c2OC)cc1OC ZINC000217922479 GG In-Stock Unstable CYP1B1 28 44 COc1ccc(/C=C/C(=O)NCc2ccc(OC)c(OC)c2OC)cc1OC ZINC000217922479 GG In-Stock Unstable SLC9A1 55 31 COc1ccc(/C=C/C(=O)NCc2ccc(OC)c(OC)c2OC)cc1OC ZINC000217922479 GG In-Stock Unstable MMP2 0 44 COc1ccc(/C=C/C(=O)NCc2ccc(OC)c(OC)c2OC)cc1OC ZINC000217922479 GG In-Stock Unstable CYP1A1 28 44 COc1ccc(/C=C/C(=O)NCc2ccc(OC)c(OC)c2OC)cc1OC ZINC000217922479 GG In-Stock Unstable TUBB1 62 47 COc1ccc(/C=C/C(=O)NCc2ccc(OC)c(OC)c2OC)cc1OC ZINC000217922479 GG In-Stock Unstable ABCG2 17 47 O=C(O)/C=C\c1cncc(C(=O)NCc2cccnc2)c1 ZINC000217922514 CD For-Sale Unstable TBXAS1 51 45 O=C(O)/C=C\c1cncc(C(=O)NCc2cccnc2)c1 ZINC000217922514 CD For-Sale Unstable PTAFR 28 41 O=C(O)/C=C\c1cncc(C(=O)NCc2cccnc2)c1 ZINC000217922514 CD For-Sale Unstable NAMPT 95 46 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922531 BD For-Sale Unstable ACE 23 40 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922531 BD For-Sale Unstable ELANE 34 43 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922531 BD For-Sale Unstable CTRA_BOVIN 40 31 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922531 BD For-Sale Unstable HRAS 41 33 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922531 BD For-Sale Unstable CASP3 18 44 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922531 BD For-Sale Unstable BMP1 65 38 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922531 BD For-Sale Unstable GALR1 43 30 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922531 BD For-Sale Unstable KLK3 74 40 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922531 BD For-Sale Unstable CTSB 61 42 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922531 BD For-Sale Unstable PAPA1_CARPA 62 34 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922531 BD For-Sale Unstable CYSP_TRYCR 61 42 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922531 BD For-Sale Unstable CTSK 43 49 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922531 BD For-Sale Unstable CTSL 43 46 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922531 BD For-Sale Unstable PGA 21 40 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922531 BD For-Sale Unstable CAPNS1 66 40 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922531 BD For-Sale Unstable MMP11 40 33 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922531 BD For-Sale Unstable CTSS 25 45 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922531 BD For-Sale Unstable CAPN1 93 48 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922531 BD For-Sale Unstable CASP1 27 42 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922531 BD For-Sale Unstable CAPN2 122 43 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922531 BD For-Sale Unstable PLAU 15 41 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922531 BD For-Sale Unstable CASP6 24 42 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922531 BD For-Sale Unstable CASP9 31 42 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922531 BD For-Sale Unstable NPR 66 39 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922531 BD For-Sale Unstable PSMB5 49 40 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922531 BD For-Sale Unstable BIRC2 34 40 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922531 BD For-Sale Unstable MBTPS1 40 35 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCNC1 ZINC000217922531 BD For-Sale Unstable Q9NAW4_PLAFA 35 41 CCNC[C@@H](C)c1ccc(CN2CC[C@@H](COC)C2)cc1 ZINC000217922536 CF For-Sale Unstable SIGMAR1 17 41 COC(=O)[C@H]1[C@@H]2CC(=O)[C@@H]1C[C@@H]2Br ZINC000217922546 BD In-Stock Unstable SLC6A1 48 33 CCOc1ccc(CNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1OCC ZINC000217922553 GH In-Stock Unstable TRPV1 15 43 CCOc1ccc(CNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1OCC ZINC000217922553 GH In-Stock Unstable APP 19 40 CCOc1ccc(CNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1OCC ZINC000217922553 GH In-Stock Unstable TUBB1 52 44 CCOc1ccc(CNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1OCC ZINC000217922553 GH In-Stock Unstable MT-ND1 24 42 CCOc1ccc(CNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1OCC ZINC000217922553 GH In-Stock Unstable AKR1C3 35 44 CCOc1ccc(CNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1OCC ZINC000217922553 GH In-Stock Unstable ABCG2 20 45 CCOc1ccc(CNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1OCC ZINC000217922553 GH In-Stock Unstable DRTS_TRYCR 45 34 COc1cccc(/C=C/NC(=O)Nc2ccc(S(=O)(=O)O)cc2)c1 ZINC000217922594 EF For-Sale Unstable CA1 41 38 COc1cccc(/C=C/NC(=O)Nc2ccc(S(=O)(=O)O)cc2)c1 ZINC000217922594 EF For-Sale Unstable MTNR1A 24 47 COc1cccc(/C=C/NC(=O)Nc2ccc(S(=O)(=O)O)cc2)c1 ZINC000217922594 EF For-Sale Unstable MTNR1B 27 47 COc1cccc(/C=C/NC(=O)Nc2ccc(S(=O)(=O)O)cc2)c1 ZINC000217922594 EF For-Sale Unstable CA12 30 45 COc1cccc(/C=C/NC(=O)Nc2ccc(S(=O)(=O)O)cc2)c1 ZINC000217922594 EF For-Sale Unstable CA9 26 40 COc1cccc(/C=C/NC(=O)Nc2ccc(S(=O)(=O)O)cc2)c1 ZINC000217922594 EF For-Sale Unstable IDO1 28 42 COc1cccc(/C=C/NC(=O)Nc2ccc(S(=O)(=O)O)cc2)c1 ZINC000217922594 EF For-Sale Unstable AKR1C2 45 34 COc1cccc(/C=C/NC(=O)Nc2ccc(S(=O)(=O)O)cc2)c1 ZINC000217922594 EF For-Sale Unstable MTCA1 35 45 COc1cccc(/C=C/NC(=O)Nc2ccc(S(=O)(=O)O)cc2)c1 ZINC000217922594 EF For-Sale Unstable P96878_MYCTU 45 45 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922614 BD For-Sale Unstable ACE 23 40 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922614 BD For-Sale Unstable ELANE 34 43 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922614 BD For-Sale Unstable CTRA_BOVIN 40 31 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922614 BD For-Sale Unstable HRAS 41 33 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922614 BD For-Sale Unstable CASP3 18 44 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922614 BD For-Sale Unstable BMP1 65 38 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922614 BD For-Sale Unstable GALR1 43 30 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922614 BD For-Sale Unstable KLK3 74 40 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922614 BD For-Sale Unstable CTSB 61 42 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922614 BD For-Sale Unstable PAPA1_CARPA 62 34 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922614 BD For-Sale Unstable CYSP_TRYCR 61 42 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922614 BD For-Sale Unstable CTSK 43 49 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922614 BD For-Sale Unstable CTSL 43 46 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922614 BD For-Sale Unstable PGA 21 40 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922614 BD For-Sale Unstable CAPNS1 66 40 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922614 BD For-Sale Unstable MMP11 40 33 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922614 BD For-Sale Unstable CTSS 25 45 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922614 BD For-Sale Unstable CAPN1 93 48 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922614 BD For-Sale Unstable CASP1 27 42 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922614 BD For-Sale Unstable CAPN2 122 43 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922614 BD For-Sale Unstable PLAU 15 41 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922614 BD For-Sale Unstable CASP6 24 42 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922614 BD For-Sale Unstable CASP9 31 42 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922614 BD For-Sale Unstable NPR 66 39 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922614 BD For-Sale Unstable PSMB5 49 40 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922614 BD For-Sale Unstable BIRC2 34 40 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922614 BD For-Sale Unstable MBTPS1 40 35 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922614 BD For-Sale Unstable Q9NAW4_PLAFA 35 41 CCNC[C@H](C)c1ccc(CN2CC[C@@H](COC)C2)cc1 ZINC000217922618 CF For-Sale Unstable SIGMAR1 17 41 Nc1cc(F)cc(C(=O)OCC2CCCCC2)c1F ZINC000217922623 CG On-Demand Unstable HTR4 34 47 COc1ccc(/C=C/C(=O)NCc2ccc(OC(C)C)c(OC)c2)cc1OC ZINC000217922625 GH In-Stock Unstable TRPV1 24 54 COc1ccc(/C=C/C(=O)NCc2ccc(OC(C)C)c(OC)c2)cc1OC ZINC000217922625 GH In-Stock Unstable TUBB1 41 36 COc1ccc(/C=C/C(=O)NCc2ccc(OC(C)C)c(OC)c2)cc1OC ZINC000217922625 GH In-Stock Unstable MT-ND1 24 42 COc1ccc(/C=C/C(=O)NCc2ccc(OC(C)C)c(OC)c2)cc1OC ZINC000217922625 GH In-Stock Unstable AKR1C3 31 44 COc1ccc(/C=C/C(=O)NCc2ccc(OC(C)C)c(OC)c2)cc1OC ZINC000217922625 GH In-Stock Unstable ABCG2 18 45 CC(C)c1nc(CCNC(=O)c2cc(Cl)ccc2O)cs1 ZINC000217922647 DH On-Demand Unstable KCNMA1 23 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc(Oc2ccc(F)cc2)c1 ZINC000217922663 JJ For-Sale Unstable CFTR 51 48 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922692 BD For-Sale Unstable ACE 23 40 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922692 BD For-Sale Unstable ELANE 34 43 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922692 BD For-Sale Unstable CTRA_BOVIN 40 31 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922692 BD For-Sale Unstable HRAS 41 33 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922692 BD For-Sale Unstable CASP3 18 44 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922692 BD For-Sale Unstable BMP1 65 38 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922692 BD For-Sale Unstable GALR1 43 30 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922692 BD For-Sale Unstable KLK3 74 40 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922692 BD For-Sale Unstable CTSB 61 42 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922692 BD For-Sale Unstable PAPA1_CARPA 62 34 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922692 BD For-Sale Unstable CYSP_TRYCR 61 42 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922692 BD For-Sale Unstable CTSK 43 49 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922692 BD For-Sale Unstable CTSL 43 46 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922692 BD For-Sale Unstable PGA 21 40 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922692 BD For-Sale Unstable CAPNS1 66 40 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922692 BD For-Sale Unstable MMP11 40 33 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922692 BD For-Sale Unstable CTSS 25 45 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922692 BD For-Sale Unstable CAPN1 93 48 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922692 BD For-Sale Unstable CASP1 27 42 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922692 BD For-Sale Unstable CAPN2 122 43 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922692 BD For-Sale Unstable PLAU 15 41 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922692 BD For-Sale Unstable CASP6 24 42 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922692 BD For-Sale Unstable CASP9 31 42 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922692 BD For-Sale Unstable NPR 66 39 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922692 BD For-Sale Unstable PSMB5 49 40 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922692 BD For-Sale Unstable BIRC2 34 40 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922692 BD For-Sale Unstable MBTPS1 40 35 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCNC1 ZINC000217922692 BD For-Sale Unstable Q9NAW4_PLAFA 35 41 COc1cccc(/C=C/NC(=O)Nc2cccc(S(=O)(=O)O)c2)c1 ZINC000217922713 EF For-Sale Unstable MTNR1A 24 43 COc1cccc(/C=C/NC(=O)Nc2cccc(S(=O)(=O)O)c2)c1 ZINC000217922713 EF For-Sale Unstable MTNR1B 26 43 COc1ccc(/C=C/C(=O)NCCCc2ccccc2Cl)cc1OC ZINC000217922738 FI In-Stock Unstable TOP2A 17 43 COc1ccc(/C=C/C(=O)NCCCc2ccccc2Cl)cc1OC ZINC000217922738 FI In-Stock Unstable DRD3 21 48 COc1ccc(/C=C/C(=O)NCCCc2ccccc2Cl)cc1OC ZINC000217922738 FI In-Stock Unstable CYP1B1 18 41 COc1ccc(/C=C/C(=O)NCCCc2ccccc2Cl)cc1OC ZINC000217922738 FI In-Stock Unstable BCHE 15 43 COc1ccc(/C=C/C(=O)NCCCc2ccccc2Cl)cc1OC ZINC000217922738 FI In-Stock Unstable PYGL 29 52 COc1ccc(/C=C/C(=O)NCCCc2ccccc2Cl)cc1OC ZINC000217922738 FI In-Stock Unstable MTNR1B 30 44 COc1ccc(/C=C/C(=O)NCCCc2ccccc2Cl)cc1OC ZINC000217922738 FI In-Stock Unstable MMP2 0 42 COc1ccc(/C=C/C(=O)NCCCc2ccccc2Cl)cc1OC ZINC000217922738 FI In-Stock Unstable CYP1A1 21 41 COc1ccc(/C=C/C(=O)NCCCc2ccccc2Cl)cc1OC ZINC000217922738 FI In-Stock Unstable HDAC1 17 42 COc1ccc(/C=C/C(=O)NCCCc2ccccc2Cl)cc1OC ZINC000217922738 FI In-Stock Unstable ABCG2 18 45 COc1ccc(/C=C/C(=O)NCCCc2ccccc2Cl)cc1OC ZINC000217922738 FI In-Stock Unstable CAN2 0 40 COc1ccc(/C=C/C(=O)NCCCc2ccccc2Cl)cc1OC ZINC000217922738 FI In-Stock Unstable CYSP_PLAFA 37 44 Nc1cc(F)cc(C(=O)OCC2CCOCC2)c1F ZINC000217922739 CE On-Demand Unstable HTR4 31 42 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc(Oc2ccc(F)cc2)c1 ZINC000217922747 JJ For-Sale Unstable CFTR 51 48 Cc1cc(NC(=O)COc2ccc(Br)cc2Cl)n(-c2ccc([N+](=O)[O-])cc2)n1 ZINC000217922750 JJ On-Demand Unstable S1PR4 0 45 CC(C)OCc1ccc(C(=O)N[C@@H]2CCC[C@@H]2CO)cc1 ZINC000217922751 CF On-Demand Unstable SSTR3 26 43 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable ACE 39 44 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable SLC6A1 22 51 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable SLC6A3 18 51 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable CELA1 31 45 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable ELANE 37 45 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable TACR1 18 42 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable CTSD 17 42 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable CTRA_BOVIN 54 33 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable HRAS 41 33 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable CASP3 20 44 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable BMP1 64 38 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable KLK3 83 40 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable CTSB 75 48 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable PAPA1_CARPA 78 44 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable CYSP_TRYCR 60 44 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable CTSG 41 33 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable CTSK 59 49 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable CTSL 55 48 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable PGA 22 43 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable PREP 27 53 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable AMY2 45 32 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable CAPNS1 77 41 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable CELA2A 41 33 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable REN 52 38 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable MMP11 44 34 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable CTSS 32 48 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable GHSR 30 40 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable CAPN1 101 48 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable CASP1 28 42 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable CAPN2 154 45 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable PLAU 17 41 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable CASP6 24 42 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable CASP9 31 42 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable TPSAB1 43 38 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable NPR 84 38 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable NAAA 37 41 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable PSMB5 49 40 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable BIRC2 33 40 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable SLC12A5 53 34 C[C@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922803 BE For-Sale Unstable Q9NAW4_PLAFA 34 41 CCCCCCCCC[C@@H](O)[C@@H]1CCC[C@@H](C)C1 ZINC000217922815 CK For-Sale Unstable MT-ND1 40 35 COc1cccc(/C=C/NC(=O)N2CCNCC2)c1 ZINC000217922822 CD For-Sale Unstable DRD4 42 32 COc1cccc(/C=C/NC(=O)N2CCNCC2)c1 ZINC000217922822 CD For-Sale Unstable MTNR1A 26 40 COc1cccc(/C=C/NC(=O)N2CCNCC2)c1 ZINC000217922822 CD For-Sale Unstable MTNR1B 36 40 COc1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1OC ZINC000217922828 FI In-Stock Unstable DRD3 17 51 COc1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1OC ZINC000217922828 FI In-Stock Unstable SCNN1A 58 38 COc1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1OC ZINC000217922828 FI In-Stock Unstable BCHE 15 42 COc1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1OC ZINC000217922828 FI In-Stock Unstable PYGL 0 51 COc1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1OC ZINC000217922828 FI In-Stock Unstable HDAC8 18 45 COc1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1OC ZINC000217922828 FI In-Stock Unstable MMP2 0 44 COc1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1OC ZINC000217922828 FI In-Stock Unstable HDAC1 15 43 COc1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1OC ZINC000217922828 FI In-Stock Unstable TUBB1 42 35 COc1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1OC ZINC000217922828 FI In-Stock Unstable HDAC7 40 38 COc1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1OC ZINC000217922828 FI In-Stock Unstable AKR1C3 27 42 COc1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1OC ZINC000217922828 FI In-Stock Unstable FOXO1 0 41 COc1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1OC ZINC000217922828 FI In-Stock Unstable ABCG2 17 44 COc1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1OC ZINC000217922828 FI In-Stock Unstable CAN2 0 41 COc1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1OC ZINC000217922828 FI In-Stock Unstable CYSP_PLAFA 38 41 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc(Oc2ccc(F)cc2)c1 ZINC000217922833 JJ For-Sale Unstable CFTR 51 48 CCCCCCOC(=O)c1cc(F)cc(N)c1F ZINC000217922850 CG On-Demand Unstable THRA 42 33 CCCCCCOC(=O)c1cc(F)cc(N)c1F ZINC000217922850 CG On-Demand Unstable THRB 40 33 CCCCCCOC(=O)c1cc(F)cc(N)c1F ZINC000217922850 CG On-Demand Unstable PLA2G4B 43 31 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable ACE 39 44 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable SLC6A1 22 51 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable SLC6A3 18 51 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable CELA1 31 45 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable ELANE 37 45 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable TACR1 18 42 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable CTSD 17 42 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable CTRA_BOVIN 54 33 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable HRAS 41 33 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable CASP3 20 44 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable BMP1 64 38 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable KLK3 83 40 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable CTSB 75 48 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable PAPA1_CARPA 78 44 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable CYSP_TRYCR 60 44 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable CTSG 41 33 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable CTSK 59 49 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable CTSL 55 48 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable PGA 22 43 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable PREP 27 53 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable AMY2 45 32 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable CAPNS1 77 41 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable CELA2A 41 33 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable REN 52 38 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable MMP11 44 34 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable CTSS 32 48 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable GHSR 30 40 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable CAPN1 101 48 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable CASP1 28 42 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable CAPN2 154 45 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable PLAU 17 41 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable CASP6 24 42 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable CASP9 31 42 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable TPSAB1 43 38 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable NPR 84 38 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable NAAA 37 41 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable PSMB5 49 40 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable BIRC2 33 40 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable SLC12A5 53 34 C[C@@H](NC(=O)OCc1ccccc1)[C@@H]1CCCN1 ZINC000217922882 BE For-Sale Unstable Q9NAW4_PLAFA 34 41 COc1ccccc1-c1cc(C(=O)NC[C@@H]2CCCN3CCCC[C@H]23)n(C)n1 ZINC000217922901 GG In-Stock Unstable ACKR3 62 32 COc1ccccc1-c1cc(C(=O)NC[C@@H]2CCCN3CCCC[C@H]23)n(C)n1 ZINC000217922901 GG In-Stock Unstable MT-CYB 41 40 CCCCCCCCC[C@H](O)[C@@H]1CCC[C@@H](C)C1 ZINC000217922906 CK For-Sale Unstable MT-ND1 40 35 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc(Oc2ccc(F)cc2)c1 ZINC000217922919 JJ For-Sale Unstable CFTR 51 48 CCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217922927 BE For-Sale Unstable DRD4 43 33 CCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217922927 BE For-Sale Unstable HRH2 17 40 CCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217922927 BE For-Sale Unstable CYP1B1 24 42 CCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217922927 BE For-Sale Unstable AHR 24 43 CCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217922927 BE For-Sale Unstable MTNR1A 107 50 CCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217922927 BE For-Sale Unstable MTNR1B 93 47 CCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217922927 BE For-Sale Unstable CYP1A1 21 42 O=C(NCC[C@H](O)C1CCOCC1)c1ccc(C(F)(F)F)nc1 ZINC000217922941 EE In-Stock Unstable EPHX2 0 42 COc1ccc(/C=C/C(=O)NCCCc2ccc(F)cc2)cc1OC ZINC000217922951 EH In-Stock Unstable TOP2A 16 42 COc1ccc(/C=C/C(=O)NCCCc2ccc(F)cc2)cc1OC ZINC000217922951 EH In-Stock Unstable DRD3 18 52 COc1ccc(/C=C/C(=O)NCCCc2ccc(F)cc2)cc1OC ZINC000217922951 EH In-Stock Unstable BCHE 15 42 COc1ccc(/C=C/C(=O)NCCCc2ccc(F)cc2)cc1OC ZINC000217922951 EH In-Stock Unstable PYGL 24 45 COc1ccc(/C=C/C(=O)NCCCc2ccc(F)cc2)cc1OC ZINC000217922951 EH In-Stock Unstable HDAC8 18 45 COc1ccc(/C=C/C(=O)NCCCc2ccc(F)cc2)cc1OC ZINC000217922951 EH In-Stock Unstable MMP2 0 44 COc1ccc(/C=C/C(=O)NCCCc2ccc(F)cc2)cc1OC ZINC000217922951 EH In-Stock Unstable HDAC1 15 43 COc1ccc(/C=C/C(=O)NCCCc2ccc(F)cc2)cc1OC ZINC000217922951 EH In-Stock Unstable TUBB1 43 37 COc1ccc(/C=C/C(=O)NCCCc2ccc(F)cc2)cc1OC ZINC000217922951 EH In-Stock Unstable AKR1C3 29 43 COc1ccc(/C=C/C(=O)NCCCc2ccc(F)cc2)cc1OC ZINC000217922951 EH In-Stock Unstable ABCG2 20 44 CC[C@H](CCO)NC(=O)[C@@H](N)[C@H](C)CC ZINC000217922967 BC For-Sale Unstable ENPEP 66 36 CC[C@H](CCO)NC(=O)[C@@H](N)[C@H](C)CC ZINC000217922967 BC For-Sale Unstable ACE2 26 41 CC[C@H](CCO)NC(=O)[C@@H](N)[C@H](C)CC ZINC000217922967 BC For-Sale Unstable SLC15A2 0 46 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable ACE 39 44 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable SLC6A1 22 51 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable SLC6A3 18 51 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable CELA1 31 45 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable ELANE 37 45 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable TACR1 18 42 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable CTSD 17 42 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable CTRA_BOVIN 54 33 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable HRAS 41 33 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable CASP3 20 44 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable BMP1 64 38 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable KLK3 83 40 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable CTSB 75 48 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable PAPA1_CARPA 78 44 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable CYSP_TRYCR 60 44 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable CTSG 41 33 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable CTSK 59 49 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable CTSL 55 48 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable PGA 22 43 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable PREP 27 53 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable AMY2 45 32 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable CAPNS1 77 41 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable CELA2A 41 33 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable REN 52 38 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable MMP11 44 34 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable CTSS 32 48 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable GHSR 30 40 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable CAPN1 101 48 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable CASP1 28 42 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable CAPN2 154 45 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable PLAU 17 41 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable CASP6 24 42 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable CASP9 31 42 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable TPSAB1 43 38 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable NPR 84 38 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable NAAA 37 41 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable PSMB5 49 40 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable BIRC2 33 40 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable SLC12A5 53 34 C[C@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217922969 BE For-Sale Unstable Q9NAW4_PLAFA 34 41 Cc1cc(NC(=O)COc2ccc(F)cc2Cl)n(-c2ccc([N+](=O)[O-])cc2)n1 ZINC000217922983 HH On-Demand Unstable S1PR4 15 45 CCCCCCCCC[C@@H](O)[C@H]1CCC[C@@H](C)C1 ZINC000217922986 CK For-Sale Unstable MT-ND1 40 35 O=C(NCC[C@@H](O)C1CCOCC1)c1ccc(C(F)(F)F)nc1 ZINC000217923027 EE In-Stock Unstable EPHX2 0 42 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable ACE 39 44 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable SLC6A1 22 51 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable SLC6A3 18 51 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable CELA1 31 45 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable ELANE 37 45 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable TACR1 18 42 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable CTSD 17 42 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable CTRA_BOVIN 54 33 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable HRAS 41 33 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable CASP3 20 44 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable BMP1 64 38 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable KLK3 83 40 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable CTSB 75 48 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable PAPA1_CARPA 78 44 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable CYSP_TRYCR 60 44 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable CTSG 41 33 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable CTSK 59 49 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable CTSL 55 48 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable PGA 22 43 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable PREP 27 53 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable AMY2 45 32 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable CAPNS1 77 41 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable CELA2A 41 33 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable REN 52 38 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable MMP11 44 34 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable CTSS 32 48 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable GHSR 30 40 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable CAPN1 101 48 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable CASP1 28 42 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable CAPN2 154 45 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable PLAU 17 41 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable CASP6 24 42 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable CASP9 31 42 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable TPSAB1 43 38 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable NPR 84 38 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable NAAA 37 41 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable PSMB5 49 40 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable BIRC2 33 40 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable SLC12A5 53 34 C[C@@H](NC(=O)OCc1ccccc1)[C@H]1CCCN1 ZINC000217923040 BE For-Sale Unstable Q9NAW4_PLAFA 34 41 COc1cccc(/C=C/NC(=O)Nc2ccc(C(C)C)cc2)c1 ZINC000217923041 DJ For-Sale Unstable CA1 24 43 COc1cccc(/C=C/NC(=O)Nc2ccc(C(C)C)cc2)c1 ZINC000217923041 DJ For-Sale Unstable MTNR1A 28 48 COc1cccc(/C=C/NC(=O)Nc2ccc(C(C)C)cc2)c1 ZINC000217923041 DJ For-Sale Unstable MTNR1B 34 48 COc1ccccc1CCCNC(=O)/C=C/c1ccc(OC)c(OC)c1 ZINC000217923051 FG In-Stock Unstable TOP2A 17 43 COc1ccccc1CCCNC(=O)/C=C/c1ccc(OC)c(OC)c1 ZINC000217923051 FG In-Stock Unstable ACHE 0 46 COc1ccccc1CCCNC(=O)/C=C/c1ccc(OC)c(OC)c1 ZINC000217923051 FG In-Stock Unstable DRD3 30 50 COc1ccccc1CCCNC(=O)/C=C/c1ccc(OC)c(OC)c1 ZINC000217923051 FG In-Stock Unstable CYP1B1 20 44 COc1ccccc1CCCNC(=O)/C=C/c1ccc(OC)c(OC)c1 ZINC000217923051 FG In-Stock Unstable BCHE 15 45 COc1ccccc1CCCNC(=O)/C=C/c1ccc(OC)c(OC)c1 ZINC000217923051 FG In-Stock Unstable PYGL 25 46 COc1ccccc1CCCNC(=O)/C=C/c1ccc(OC)c(OC)c1 ZINC000217923051 FG In-Stock Unstable HDAC8 24 41 COc1ccccc1CCCNC(=O)/C=C/c1ccc(OC)c(OC)c1 ZINC000217923051 FG In-Stock Unstable MTNR1A 34 42 COc1ccccc1CCCNC(=O)/C=C/c1ccc(OC)c(OC)c1 ZINC000217923051 FG In-Stock Unstable MTNR1B 47 49 COc1ccccc1CCCNC(=O)/C=C/c1ccc(OC)c(OC)c1 ZINC000217923051 FG In-Stock Unstable MMP2 16 45 COc1ccccc1CCCNC(=O)/C=C/c1ccc(OC)c(OC)c1 ZINC000217923051 FG In-Stock Unstable CYP1A1 23 44 COc1ccccc1CCCNC(=O)/C=C/c1ccc(OC)c(OC)c1 ZINC000217923051 FG In-Stock Unstable HDAC1 22 44 COc1ccccc1CCCNC(=O)/C=C/c1ccc(OC)c(OC)c1 ZINC000217923051 FG In-Stock Unstable MMP9 15 45 COc1ccccc1CCCNC(=O)/C=C/c1ccc(OC)c(OC)c1 ZINC000217923051 FG In-Stock Unstable TUBB1 42 37 COc1ccccc1CCCNC(=O)/C=C/c1ccc(OC)c(OC)c1 ZINC000217923051 FG In-Stock Unstable HDAC7 40 38 COc1ccccc1CCCNC(=O)/C=C/c1ccc(OC)c(OC)c1 ZINC000217923051 FG In-Stock Unstable PTPA 0 44 COc1ccccc1CCCNC(=O)/C=C/c1ccc(OC)c(OC)c1 ZINC000217923051 FG In-Stock Unstable ABCG2 20 46 COc1ccccc1CCCNC(=O)/C=C/c1ccc(OC)c(OC)c1 ZINC000217923051 FG In-Stock Unstable CYSP_PLAFA 18 42 CCCCCCCCC[C@H](O)[C@H]1CCC[C@@H](C)C1 ZINC000217923063 CK For-Sale Unstable MT-ND1 40 35 O=C(Nc1c(F)c(F)cc(F)c1F)NC1CCCCC1 ZINC000217923074 CH For-Sale Unstable EPHX2 49 60 CC[C@@H](CCO)NC(=O)[C@@H](C)CCCN ZINC000217923089 BC For-Sale Unstable KLK3 45 33 CC[C@@H](CCO)NC(=O)[C@@H](C)CCCN ZINC000217923089 BC For-Sale Unstable GSP 0 40 CC[C@@H](CCO)NC(=O)[C@@H](C)CCCN ZINC000217923089 BC For-Sale Unstable NOD1 43 40 CNC(=O)c1cccc(N[C@@H]2C[C@@H]3CC=C[C@H]32)c1 ZINC000217923140 BE For-Sale Unstable KCNK3 50 34 CCCCCCCC[C@@H](O)[C@@H]1CCC[C@@H](C)C1 ZINC000217923143 BJ For-Sale Unstable MT-ND1 40 35 COc1cccc(/C=C/NC(=O)Nc2ccccc2OC)c1 ZINC000217923155 CG For-Sale Unstable CYP1B1 55 39 COc1cccc(/C=C/NC(=O)Nc2ccccc2OC)c1 ZINC000217923155 CG For-Sale Unstable MTNR1A 32 44 COc1cccc(/C=C/NC(=O)Nc2ccccc2OC)c1 ZINC000217923155 CG For-Sale Unstable MTNR1B 36 45 COc1cccc(/C=C/NC(=O)Nc2ccccc2OC)c1 ZINC000217923155 CG For-Sale Unstable CYP1A1 38 45 COc1cccc(/C=C/NC(=O)Nc2ccccc2OC)c1 ZINC000217923155 CG For-Sale Unstable ABCG2 21 45 CC(C)(C)OC(=O)N1CC[C@@H]1c1cccc(N)c1 ZINC000217923159 BF For-Sale Unstable GPR119 27 43 COc1ccc(CCCNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923168 FG In-Stock Unstable PTGS2 0 54 COc1ccc(CCCNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923168 FG In-Stock Unstable DRD3 17 50 COc1ccc(CCCNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923168 FG In-Stock Unstable SCNN1A 65 42 COc1ccc(CCCNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923168 FG In-Stock Unstable PTAFR 18 44 COc1ccc(CCCNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923168 FG In-Stock Unstable CYP1B1 41 46 COc1ccc(CCCNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923168 FG In-Stock Unstable BCHE 15 45 COc1ccc(CCCNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923168 FG In-Stock Unstable PYGL 24 46 COc1ccc(CCCNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923168 FG In-Stock Unstable HDAC8 35 46 COc1ccc(CCCNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923168 FG In-Stock Unstable MTNR1A 48 44 COc1ccc(CCCNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923168 FG In-Stock Unstable MTNR1B 42 44 COc1ccc(CCCNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923168 FG In-Stock Unstable CYP1A1 30 46 COc1ccc(CCCNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923168 FG In-Stock Unstable HDAC1 23 44 COc1ccc(CCCNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923168 FG In-Stock Unstable HDAC2 24 43 COc1ccc(CCCNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923168 FG In-Stock Unstable HDAC6 21 45 COc1ccc(CCCNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923168 FG In-Stock Unstable TUBB1 55 37 COc1ccc(CCCNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923168 FG In-Stock Unstable PTPA 0 44 COc1ccc(CCCNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923168 FG In-Stock Unstable ABCG2 29 46 COc1ccc(CCCNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923168 FG In-Stock Unstable PROKR1 43 31 COc1ccc(CCCNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923168 FG In-Stock Unstable CYSP_PLAFA 36 40 CC[C@H](CCO)NC(=O)[C@@H](C)CCCN ZINC000217923180 BC For-Sale Unstable KLK3 45 33 CC[C@H](CCO)NC(=O)[C@@H](C)CCCN ZINC000217923180 BC For-Sale Unstable GSP 0 40 CC[C@H](CCO)NC(=O)[C@@H](C)CCCN ZINC000217923180 BC For-Sale Unstable NOD1 43 40 Cc1n[nH]c(C)c1CNC(=O)c1ccc(O)cc1F ZINC000217923209 CD In-Stock Unstable P2RX7 17 52 Cc1n[nH]c(C)c1CNC(=O)c1ccc(O)cc1F ZINC000217923209 CD In-Stock Unstable HAO2 48 35 CCCCCCCC[C@H](O)[C@@H]1CCC[C@@H](C)C1 ZINC000217923220 BJ For-Sale Unstable MT-ND1 40 35 CC(C)(C)OC(=O)N1CC[C@H]1c1cccc(N)c1 ZINC000217923235 BF For-Sale Unstable GPR119 27 43 CNC(=O)c1cccc(N[C@H]2C[C@@H]3CC=C[C@H]32)c1 ZINC000217923237 BE For-Sale Unstable KCNK3 50 34 COc1cccc(/C=C/NC(=O)Nc2ccccc2C)c1 ZINC000217923264 CH For-Sale Unstable MTNR1A 31 42 COc1cccc(/C=C/NC(=O)Nc2ccccc2C)c1 ZINC000217923264 CH For-Sale Unstable MTNR1B 32 42 CC[C@@H](CCO)NC(=O)[C@H](C)CCCN ZINC000217923270 BC For-Sale Unstable KLK3 45 33 CC[C@@H](CCO)NC(=O)[C@H](C)CCCN ZINC000217923270 BC For-Sale Unstable GSP 0 40 CC[C@@H](CCO)NC(=O)[C@H](C)CCCN ZINC000217923270 BC For-Sale Unstable NOD1 43 40 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923277 FG In-Stock Unstable CYP1B1 41 43 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923277 FG In-Stock Unstable HDAC8 18 45 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923277 FG In-Stock Unstable CYP1A1 30 43 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923277 FG In-Stock Unstable TUBB1 58 38 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923277 FG In-Stock Unstable PTPA 0 46 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923277 FG In-Stock Unstable ABCG2 22 46 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923277 FG In-Stock Unstable CYSP_PLAFA 35 40 CCCCCCCC[C@@H](O)[C@H]1CCC[C@@H](C)C1 ZINC000217923302 BJ For-Sale Unstable MT-ND1 40 35 Cc1cc(NC(=O)CCc2ccc3c(c2)OCCO3)n(-c2ccc([N+](=O)[O-])cc2)n1 ZINC000217923305 HG On-Demand Unstable LUXR 20 40 CNC(=O)c1cccc(N[C@@H]2C[C@H]3CC=C[C@H]32)c1 ZINC000217923310 BE For-Sale Unstable KCNK3 50 34 CC(C)(C)OC(=O)N1CC[C@@H]1c1ccccc1N ZINC000217923353 BF For-Sale Unstable GPR119 27 40 CC[C@H](CCO)NC(=O)[C@H](C)CCCN ZINC000217923359 BC For-Sale Unstable KLK3 45 33 CC[C@H](CCO)NC(=O)[C@H](C)CCCN ZINC000217923359 BC For-Sale Unstable GSP 0 40 CC[C@H](CCO)NC(=O)[C@H](C)CCCN ZINC000217923359 BC For-Sale Unstable NOD1 43 40 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923366 FG In-Stock Unstable CYP1B1 41 43 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923366 FG In-Stock Unstable HDAC8 18 45 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923366 FG In-Stock Unstable CYP1A1 30 43 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923366 FG In-Stock Unstable TUBB1 58 38 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923366 FG In-Stock Unstable PTPA 0 46 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923366 FG In-Stock Unstable ABCG2 22 46 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923366 FG In-Stock Unstable CYSP_PLAFA 35 40 CN1CCC(NC(=O)c2cncc(/C=C\C(=O)O)c2)CC1 ZINC000217923367 CD For-Sale Unstable SSTR5 42 41 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c(Cl)c2)c1 ZINC000217923373 EJ For-Sale Unstable UL80 16 40 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c(Cl)c2)c1 ZINC000217923373 EJ For-Sale Unstable GUAB 0 40 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c(Cl)c2)c1 ZINC000217923373 EJ For-Sale Unstable RAF1 26 45 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c(Cl)c2)c1 ZINC000217923373 EJ For-Sale Unstable KDR 15 41 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c(Cl)c2)c1 ZINC000217923373 EJ For-Sale Unstable MTNR1A 25 48 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c(Cl)c2)c1 ZINC000217923373 EJ For-Sale Unstable MTNR1B 30 48 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c(Cl)c2)c1 ZINC000217923373 EJ For-Sale Unstable PDGFRA 21 41 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c(Cl)c2)c1 ZINC000217923373 EJ For-Sale Unstable TAAR1 30 52 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c(Cl)c2)c1 ZINC000217923373 EJ For-Sale Unstable IMDH_CRYPV 42 41 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c(Cl)c2)c1 ZINC000217923373 EJ For-Sale Unstable P95276_MYCTO 0 44 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c(Cl)c2)c1 ZINC000217923373 EJ For-Sale Unstable PPX1 0 40 CCCCCCCC[C@H](O)[C@H]1CCC[C@@H](C)C1 ZINC000217923387 BJ For-Sale Unstable MT-ND1 40 35 CNC(=O)c1cccc(N[C@H]2C[C@H]3CC=C[C@@H]23)c1 ZINC000217923399 BE For-Sale Unstable KCNK3 50 34 Cc1cc(NC(=O)Cc2ccc(OCc3c(C)noc3C)cc2)n(-c2ccc(Cl)cc2)n1 ZINC000217923403 JK On-Demand Unstable P2RX7 20 47 Cc1cc(NC(=O)Cc2ccc(OCc3c(C)noc3C)cc2)n(-c2ccc(Cl)cc2)n1 ZINC000217923403 JK On-Demand Unstable RORC 15 56 CCCCNC(=O)Nc1c(F)c(F)cc(F)c1F ZINC000217923428 CG For-Sale Unstable ASAH1 74 35 CCCCNC(=O)Nc1c(F)c(F)cc(F)c1F ZINC000217923428 CG For-Sale Unstable ACAT 0 64 CC(C)(C)OC(=O)N1CC[C@H]1c1ccccc1N ZINC000217923447 BF For-Sale Unstable GPR119 27 40 COc1cccc(/C=C/NC(=O)Nc2ccc(C)c(Cl)c2)c1 ZINC000217923473 DI For-Sale Unstable DRD4 42 33 COc1cccc(/C=C/NC(=O)Nc2ccc(C)c(Cl)c2)c1 ZINC000217923473 DI For-Sale Unstable MTNR1A 25 43 COc1cccc(/C=C/NC(=O)Nc2ccc(C)c(Cl)c2)c1 ZINC000217923473 DI For-Sale Unstable MTNR1B 30 44 COc1cccc(/C=C/NC(=O)Nc2ccc(C)c(Cl)c2)c1 ZINC000217923473 DI For-Sale Unstable Q8MMZ8_EIMTE 0 41 COc1cccc(/C=C/NC(=O)Nc2ccc(C)c(Cl)c2)c1 ZINC000217923473 DI For-Sale Unstable TAAR1 25 42 COc1cccc(/C=C/NC(=O)Nc2ccc(C)c(Cl)c2)c1 ZINC000217923473 DI For-Sale Unstable AKR1C2 42 36 CC(=O)Nc1cccc(C(=O)N[C@@H]2CCC[C@@H]2CO)c1 ZINC000217923474 CD On-Demand Unstable CCR3 24 46 CC(=O)Nc1cccc(C(=O)N[C@@H]2CCC[C@@H]2CO)c1 ZINC000217923474 CD On-Demand Unstable SSTR3 28 40 CC(=O)Nc1cccc(C(=O)N[C@@H]2CCC[C@@H]2CO)c1 ZINC000217923474 CD On-Demand Unstable PARP15 0 40 CC(=O)Nc1cccc(C(=O)N[C@@H]2CCC[C@@H]2CO)c1 ZINC000217923474 CD On-Demand Unstable KCNK3 81 35 CC(=O)Nc1cccc(C(=O)N[C@@H]2CCC[C@@H]2CO)c1 ZINC000217923474 CD On-Demand Unstable KCNK9 57 40 CC(=O)Nc1cccc(C(=O)N[C@@H]2CCC[C@@H]2CO)c1 ZINC000217923474 CD On-Demand Unstable PARP10 0 44 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC(C)C)c2)cc1OC ZINC000217923477 GI In-Stock Unstable TOP2A 16 42 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC(C)C)c2)cc1OC ZINC000217923477 GI In-Stock Unstable DRD3 15 43 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC(C)C)c2)cc1OC ZINC000217923477 GI In-Stock Unstable PTAFR 24 46 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC(C)C)c2)cc1OC ZINC000217923477 GI In-Stock Unstable PYGL 0 41 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC(C)C)c2)cc1OC ZINC000217923477 GI In-Stock Unstable MTNR1A 32 52 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC(C)C)c2)cc1OC ZINC000217923477 GI In-Stock Unstable MTNR1B 36 52 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC(C)C)c2)cc1OC ZINC000217923477 GI In-Stock Unstable AKR1C3 29 43 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC(C)C)c2)cc1OC ZINC000217923477 GI In-Stock Unstable ABCG2 17 40 COc1ccc(/C=C/C(=O)NCCCc2cccc(OC(C)C)c2)cc1OC ZINC000217923477 GI In-Stock Unstable CRTM 46 46 Cc1cc(S(=O)(=O)NCC[C@H](O)C2CCOCC2)ccc1F ZINC000217923498 ED In-Stock Unstable LEF 75 59 Cc1cc(NC(=O)c2ccc3c(c2)OCCCO3)n(-c2ccc(Cl)cc2)n1 ZINC000217923519 GI On-Demand Unstable F10 21 40 Cc1cc(NC(=O)c2ccc3c(c2)OCCCO3)n(-c2ccc(Cl)cc2)n1 ZINC000217923519 GI On-Demand Unstable PLK1 15 44 CC(C)(C)OC(=O)N1CC[C@@H]1c1ccc(N)cc1 ZINC000217923568 BF For-Sale Unstable GPR119 32 41 COc1cccc(/C=C/NC(=O)Nc2c(C)cccc2C(C)C)c1 ZINC000217923586 DJ For-Sale Unstable SOAT1 50 43 COc1cccc(/C=C/NC(=O)Nc2c(C)cccc2C(C)C)c1 ZINC000217923586 DJ For-Sale Unstable ACAT 0 45 Cc1cc(S(=O)(=O)NCC[C@@H](O)C2CCOCC2)ccc1F ZINC000217923590 ED In-Stock Unstable LEF 75 59 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@H](C(=O)Nc3nc(-c4cccnc4)cs3)C(C)C)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217923602 KK In-Stock Unstable TUBA1A 16 55 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC(C)C)cc2)cc1OC ZINC000217923607 GI In-Stock Unstable DRD3 15 42 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC(C)C)cc2)cc1OC ZINC000217923607 GI In-Stock Unstable PYGL 0 42 COc1ccc(/C=C/C(=O)NCCCc2ccc(OC(C)C)cc2)cc1OC ZINC000217923607 GI In-Stock Unstable ABCG2 17 41 C[C@@H]1CCC[C@H]([C@@H](O)c2ccc(Cl)c(Cl)c2)C1 ZINC000217923655 CJ For-Sale Unstable SLC6A3 15 50 CC(C)(C)OC(=O)N1CC[C@H]1c1ccc(N)cc1 ZINC000217923661 BF For-Sale Unstable GPR119 32 41 N[C@@H]1CCCC[C@@H]1N1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217923693 BF For-Sale Unstable CYP2D26 0 47 COc1cccc(/C=C/NC(=O)Nc2ccccc2C(F)(F)F)c1 ZINC000217923696 EJ For-Sale Unstable TAAR1 18 42 NC(=O)c1cccc(N[C@@H]2C[C@@H]3CC=C[C@H]32)c1 ZINC000217923701 BE For-Sale Unstable MVFR 0 40 NC(=O)c1cccc(N[C@@H]2C[C@@H]3CC=C[C@H]32)c1 ZINC000217923701 BE For-Sale Unstable PARP10 0 40 O=C1C[C@H](c2ccc(O)cc2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217923714 HI In-Stock Unstable VEGFA 24 43 O=C1C[C@H](c2ccc(O)cc2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217923714 HI In-Stock Unstable AKR1B1 0 48 O=C1C[C@H](c2ccc(O)cc2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217923714 HI In-Stock Unstable CYP1B1 36 46 O=C1C[C@H](c2ccc(O)cc2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217923714 HI In-Stock Unstable CYP1A1 34 46 O=C1C[C@H](c2ccc(O)cc2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217923714 HI In-Stock Unstable CYP1A2 23 43 CCn1nccc1NC(=O)[C@@H](C)Oc1ccc(Cl)cc1Cl ZINC000217923730 EH On-Demand Unstable IMDH_CRYPV 32 50 C[C@H]1CCC[C@H]([C@@H](O)c2ccc(Cl)c(Cl)c2)C1 ZINC000217923732 CJ For-Sale Unstable SLC6A3 15 50 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc(OCc2ccccc2)c1 ZINC000217923770 II For-Sale Unstable PTGER1 42 35 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc(OCc2ccccc2)c1 ZINC000217923770 II For-Sale Unstable GYS1 50 46 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc(OCc2ccccc2)c1 ZINC000217923770 II For-Sale Unstable CFTR 48 37 N[C@H]1CCCC[C@@H]1N1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217923783 BF For-Sale Unstable CYP2D26 0 47 NC(=O)c1cccc(N[C@H]2C[C@@H]3CC=C[C@H]32)c1 ZINC000217923785 BE For-Sale Unstable MVFR 0 40 NC(=O)c1cccc(N[C@H]2C[C@@H]3CC=C[C@H]32)c1 ZINC000217923785 BE For-Sale Unstable PARP10 0 40 O=C1C[C@@H](c2ccc(O)cc2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217923800 HI In-Stock Unstable VEGFA 24 43 O=C1C[C@@H](c2ccc(O)cc2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217923800 HI In-Stock Unstable AKR1B1 0 48 O=C1C[C@@H](c2ccc(O)cc2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217923800 HI In-Stock Unstable CYP1B1 36 46 O=C1C[C@@H](c2ccc(O)cc2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217923800 HI In-Stock Unstable CYP1A1 34 46 O=C1C[C@@H](c2ccc(O)cc2)c2c(cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc23)O1 ZINC000217923800 HI In-Stock Unstable CYP1A2 23 43 COc1cccc(/C=C/NC(=O)Nc2ccc(C(=O)O)cc2)c1 ZINC000217923806 DG For-Sale Unstable UL80 30 43 COc1cccc(/C=C/NC(=O)Nc2ccc(C(=O)O)cc2)c1 ZINC000217923806 DG For-Sale Unstable RAF1 24 44 COc1cccc(/C=C/NC(=O)Nc2ccc(C(=O)O)cc2)c1 ZINC000217923806 DG For-Sale Unstable MTNR1A 26 49 COc1cccc(/C=C/NC(=O)Nc2ccc(C(=O)O)cc2)c1 ZINC000217923806 DG For-Sale Unstable MTNR1B 34 49 COc1cccc(/C=C/NC(=O)Nc2ccc(C(=O)O)cc2)c1 ZINC000217923806 DG For-Sale Unstable ACR 32 43 COc1cccc(/C=C/NC(=O)Nc2ccc(C(=O)O)cc2)c1 ZINC000217923806 DG For-Sale Unstable Q8MMZ8_EIMTE 27 44 COc1cccc(/C=C/NC(=O)Nc2ccc(C(=O)O)cc2)c1 ZINC000217923806 DG For-Sale Unstable TAAR1 32 40 COc1cccc(/C=C/NC(=O)Nc2ccc(C(=O)O)cc2)c1 ZINC000217923806 DG For-Sale Unstable AKR1C3 51 45 COc1cccc(/C=C/NC(=O)Nc2ccc(C(=O)O)cc2)c1 ZINC000217923806 DG For-Sale Unstable AKR1C2 58 43 COc1cccc(/C=C/NC(=O)Nc2ccc(C(=O)O)cc2)c1 ZINC000217923806 DG For-Sale Unstable IMDH_CRYPV 28 42 CCn1nccc1NC(=O)[C@H](C)Oc1ccc(Cl)cc1Cl ZINC000217923811 EH On-Demand Unstable IMDH_CRYPV 32 50 C[C@@H]1CCC[C@@H]([C@@H](O)c2ccc(Cl)c(Cl)c2)C1 ZINC000217923824 CJ For-Sale Unstable SLC6A3 15 50 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc(OCc2ccccc2)c1 ZINC000217923847 II For-Sale Unstable PTGER1 42 35 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc(OCc2ccccc2)c1 ZINC000217923847 II For-Sale Unstable GYS1 50 46 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc(OCc2ccccc2)c1 ZINC000217923847 II For-Sale Unstable CFTR 48 37 N[C@@H]1CCCC[C@H]1N1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217923872 BF For-Sale Unstable CYP2D26 0 47 NC(=O)c1cccc(N[C@@H]2C[C@H]3CC=C[C@H]32)c1 ZINC000217923877 BE For-Sale Unstable MVFR 0 40 NC(=O)c1cccc(N[C@@H]2C[C@H]3CC=C[C@H]32)c1 ZINC000217923877 BE For-Sale Unstable PARP10 0 40 O=C(O)/C=C\c1cncc(C(=O)Nc2cccnc2)c1 ZINC000217923881 CD For-Sale Anodyne TBXAS1 27 45 O=C(O)/C=C\c1cncc(C(=O)Nc2cccnc2)c1 ZINC000217923881 CD For-Sale Anodyne RPS6KA3 28 40 O=C(O)/C=C\c1cncc(C(=O)Nc2cccnc2)c1 ZINC000217923881 CD For-Sale Anodyne CSF1R 15 46 O=C(O)/C=C\c1cncc(C(=O)Nc2cccnc2)c1 ZINC000217923881 CD For-Sale Anodyne NAMPT 24 54 O=C(O)/C=C\c1cncc(C(=O)Nc2cccnc2)c1 ZINC000217923881 CD For-Sale Anodyne KCNK3 76 42 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923917 FH In-Stock Unstable TOP2A 15 40 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923917 FH In-Stock Unstable DRD3 15 43 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923917 FH In-Stock Unstable CYP1B1 18 40 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923917 FH In-Stock Unstable BCHE 15 41 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923917 FH In-Stock Unstable PYGL 0 43 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923917 FH In-Stock Unstable HDAC8 16 45 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923917 FH In-Stock Unstable MTNR1B 24 40 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923917 FH In-Stock Unstable CYP1A1 20 40 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923917 FH In-Stock Unstable TUBB1 54 41 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923917 FH In-Stock Unstable AKR1C3 25 42 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(OC)c(OC)c2)cc1 ZINC000217923917 FH In-Stock Unstable ABCG2 21 42 C[C@H]1CCC[C@@H]([C@@H](O)c2ccc(Cl)c(Cl)c2)C1 ZINC000217923918 CJ For-Sale Unstable SLC6A3 15 50 COc1cccc(/C=C/NC(=O)Nc2cccc(Cl)c2C)c1 ZINC000217923924 DI For-Sale Unstable PTGER3 18 41 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc(OCc2ccccc2)c1 ZINC000217923937 II For-Sale Unstable PTGER1 42 35 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc(OCc2ccccc2)c1 ZINC000217923937 II For-Sale Unstable GYS1 50 46 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc(OCc2ccccc2)c1 ZINC000217923937 II For-Sale Unstable CFTR 48 37 CCCCCCCOC(=O)c1cc(F)cc(N)c1F ZINC000217923950 CH On-Demand Unstable PLA2G4B 43 31 NC(=O)c1cccc(N[C@H]2C[C@H]3CC=C[C@@H]23)c1 ZINC000217923958 BE For-Sale Unstable MVFR 0 40 NC(=O)c1cccc(N[C@H]2C[C@H]3CC=C[C@@H]23)c1 ZINC000217923958 BE For-Sale Unstable PARP10 0 40 Cc1cc(NC(=O)CCc2ccc3c(c2)OCCO3)n(-c2ccc(Cl)cc2)n1 ZINC000217924000 GI On-Demand Unstable NOS2 62 33 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc(OCc2ccccc2)c1 ZINC000217924008 II For-Sale Unstable PTGER1 42 35 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc(OCc2ccccc2)c1 ZINC000217924008 II For-Sale Unstable GYS1 50 46 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc(OCc2ccccc2)c1 ZINC000217924008 II For-Sale Unstable CFTR 48 37 CCOC(=O)c1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217924033 EH For-Sale Unstable CA1 23 45 CCOC(=O)c1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217924033 EH For-Sale Unstable MTNR1A 33 50 CCOC(=O)c1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217924033 EH For-Sale Unstable MTNR1B 37 50 CCOC(=O)c1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217924033 EH For-Sale Unstable ACR 69 49 CCOC(=O)c1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217924033 EH For-Sale Unstable SENP1 0 45 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccc(OC)c(OC)c1 ZINC000217924038 GI In-Stock Unstable DRD3 23 45 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccc(OC)c(OC)c1 ZINC000217924038 GI In-Stock Unstable BCHE 16 44 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccc(OC)c(OC)c1 ZINC000217924038 GI In-Stock Unstable PYGL 0 41 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccc(OC)c(OC)c1 ZINC000217924038 GI In-Stock Unstable MTNR1A 46 53 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccc(OC)c(OC)c1 ZINC000217924038 GI In-Stock Unstable MTNR1B 47 53 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccc(OC)c(OC)c1 ZINC000217924038 GI In-Stock Unstable ABCB1 15 40 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccc(OC)c(OC)c1 ZINC000217924038 GI In-Stock Unstable AKR1C3 22 42 CC(=O)N[C@@H]1CCN(Cc2ccccc2)C1=O ZINC000217924086 BC On-Demand Unstable NA 52 38 CC(=O)N[C@@H]1CCN(Cc2ccccc2)C1=O ZINC000217924086 BC On-Demand Unstable ACE 57 38 CC(=O)N[C@@H]1CCN(Cc2ccccc2)C1=O ZINC000217924086 BC On-Demand Unstable DRD4 24 40 CC(=O)N[C@@H]1CCN(Cc2ccccc2)C1=O ZINC000217924086 BC On-Demand Unstable DRD3 16 41 CC(=O)N[C@@H]1CCN(Cc2ccccc2)C1=O ZINC000217924086 BC On-Demand Unstable F10 25 44 CC(=O)N[C@@H]1CCN(Cc2ccccc2)C1=O ZINC000217924086 BC On-Demand Unstable MME 29 44 CC(=O)N[C@@H]1CCN(Cc2ccccc2)C1=O ZINC000217924086 BC On-Demand Unstable SIGMAR1 45 45 CC(=O)N[C@@H]1CCN(Cc2ccccc2)C1=O ZINC000217924086 BC On-Demand Unstable APP 15 40 CC(=O)N[C@@H]1CCN(Cc2ccccc2)C1=O ZINC000217924086 BC On-Demand Unstable BIRC2 42 38 CC(=O)N[C@@H]1CCN(Cc2ccccc2)C1=O ZINC000217924086 BC On-Demand Unstable BIRC8 40 31 Cc1ccc(S(=O)(=O)NCC[C@H](O)C2CCOCC2)cc1Cl ZINC000217924088 EE In-Stock Unstable LEF 20 42 COc1cccc(/C=C/NC(=O)Nc2ccccc2Cl)c1 ZINC000217924132 DI For-Sale Unstable PTGER3 26 44 COc1cccc(/C=C/NC(=O)Nc2ccccc2Cl)c1 ZINC000217924132 DI For-Sale Unstable MTNR1A 29 41 COc1cccc(/C=C/NC(=O)Nc2ccccc2Cl)c1 ZINC000217924132 DI For-Sale Unstable MTNR1B 31 41 COc1cccc(/C=C/NC(=O)Nc2ccccc2Cl)c1 ZINC000217924132 DI For-Sale Unstable EPHB3 36 43 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccccc2C)cc1OC ZINC000217924140 FH In-Stock Unstable CYP1B1 21 44 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccccc2C)cc1OC ZINC000217924140 FH In-Stock Unstable MTNR1B 15 42 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccccc2C)cc1OC ZINC000217924140 FH In-Stock Unstable MMP2 16 44 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccccc2C)cc1OC ZINC000217924140 FH In-Stock Unstable CYP1A1 22 44 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccccc2C)cc1OC ZINC000217924140 FH In-Stock Unstable TUBB1 48 38 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccccc2C)cc1OC ZINC000217924140 FH In-Stock Unstable AKR1C3 27 41 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccccc2C)cc1OC ZINC000217924140 FH In-Stock Unstable PTPA 0 44 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccccc2C)cc1OC ZINC000217924140 FH In-Stock Unstable ABCG2 15 44 Cc1ccc(S(=O)(=O)NCC[C@@H](O)C2CCOCC2)cc1Cl ZINC000217924162 EE In-Stock Unstable LEF 20 42 Nc1cc(Cl)ccc1N1CC[C@H](NC(=O)C(F)(F)F)C1 ZINC000217924163 DE For-Sale Unstable MTNR1A 30 40 Nc1cc(Cl)ccc1N1CC[C@H](NC(=O)C(F)(F)F)C1 ZINC000217924163 DE For-Sale Unstable MTNR1B 19 40 Nc1cc(Cl)ccc1N1CC[C@H](NC(=O)C(F)(F)F)C1 ZINC000217924163 DE For-Sale Unstable LIPG 43 32 CC(=O)N[C@H]1CCN(Cc2ccccc2)C1=O ZINC000217924168 BC On-Demand Unstable NA 52 38 CC(=O)N[C@H]1CCN(Cc2ccccc2)C1=O ZINC000217924168 BC On-Demand Unstable ACE 57 38 CC(=O)N[C@H]1CCN(Cc2ccccc2)C1=O ZINC000217924168 BC On-Demand Unstable DRD4 24 40 CC(=O)N[C@H]1CCN(Cc2ccccc2)C1=O ZINC000217924168 BC On-Demand Unstable DRD3 16 41 CC(=O)N[C@H]1CCN(Cc2ccccc2)C1=O ZINC000217924168 BC On-Demand Unstable F10 25 44 CC(=O)N[C@H]1CCN(Cc2ccccc2)C1=O ZINC000217924168 BC On-Demand Unstable MME 29 44 CC(=O)N[C@H]1CCN(Cc2ccccc2)C1=O ZINC000217924168 BC On-Demand Unstable SIGMAR1 45 45 CC(=O)N[C@H]1CCN(Cc2ccccc2)C1=O ZINC000217924168 BC On-Demand Unstable APP 15 40 CC(=O)N[C@H]1CCN(Cc2ccccc2)C1=O ZINC000217924168 BC On-Demand Unstable BIRC2 42 38 CC(=O)N[C@H]1CCN(Cc2ccccc2)C1=O ZINC000217924168 BC On-Demand Unstable BIRC8 40 31 COc1cc(C(=O)N[C@@H]2CCC[C@@H]2CO)ccc1F ZINC000217924186 CD On-Demand Unstable SSTR3 26 43 COc1cc(C(=O)N[C@@H]2CCC[C@@H]2CO)ccc1F ZINC000217924186 CD On-Demand Unstable ACKR3 52 34 C[C@@H](CCN(C)C)NC(=O)c1cncc(/C=C\C(=O)O)c1 ZINC000217924187 CD For-Sale Unstable UTS2 62 34 O=C(N[C@H](CO)c1ccccc1)[C@@H]1CC(=O)N(Cc2ccc3c(c2)OCO3)C1 ZINC000217924216 GD In-Stock Unstable BACE2 0 40 O=C(N[C@H](CO)c1ccccc1)[C@@H]1CC(=O)N(Cc2ccc3c(c2)OCO3)C1 ZINC000217924216 GD In-Stock Unstable NOS2 74 33 O=C(N[C@H](CO)c1ccccc1)[C@@H]1CC(=O)N(Cc2ccc3c(c2)OCO3)C1 ZINC000217924216 GD In-Stock Unstable MCHR1 19 42 COc1ccc(/C=C/C(=O)N[C@@H](C)COc2ccc(C)cc2)cc1OC ZINC000217924248 FH In-Stock Unstable TUBB1 52 37 COc1ccc(/C=C/C(=O)N[C@@H](C)COc2ccc(C)cc2)cc1OC ZINC000217924248 FH In-Stock Unstable PTPA 0 42 COc1ccc(/C=C/C(=O)N[C@@H](C)COc2ccc(C)cc2)cc1OC ZINC000217924248 FH In-Stock Unstable ABCG2 18 43 Nc1cc(Cl)ccc1N1CC[C@@H](NC(=O)C(F)(F)F)C1 ZINC000217924249 DE For-Sale Unstable MTNR1A 30 40 Nc1cc(Cl)ccc1N1CC[C@@H](NC(=O)C(F)(F)F)C1 ZINC000217924249 DE For-Sale Unstable MTNR1B 19 40 Nc1cc(Cl)ccc1N1CC[C@@H](NC(=O)C(F)(F)F)C1 ZINC000217924249 DE For-Sale Unstable LIPG 43 32 COc1cccc(/C=C/NC(=O)Nc2ccccc2C(C)C)c1 ZINC000217924257 DJ For-Sale Unstable MTNR1A 30 41 COc1cccc(/C=C/NC(=O)Nc2ccccc2C(C)C)c1 ZINC000217924257 DJ For-Sale Unstable MTNR1B 32 41 COc1cccc(/C=C/NC(=O)Nc2ccccc2C(C)C)c1 ZINC000217924257 DJ For-Sale Unstable TRPM8 0 47 COc1cccc(/C=C/NC(=O)Nc2ccccc2C(C)C)c1 ZINC000217924257 DJ For-Sale Unstable ACAT 0 40 C[C@H](CCN(C)C)NC(=O)c1cncc(/C=C\C(=O)O)c1 ZINC000217924276 CD For-Sale Unstable UTS2 62 34 O=S(=O)(NCC[C@H](O)C1CCOCC1)c1cccc2ccccc12 ZINC000217924292 EE In-Stock Unstable NPY2R 46 44 O=S(=O)(NCC[C@H](O)C1CCOCC1)c1cccc2ccccc12 ZINC000217924292 EE In-Stock Unstable NPY5R 20 43 O=S(=O)(NCC[C@H](O)C1CCOCC1)c1cccc2ccccc12 ZINC000217924292 EE In-Stock Unstable Q95J97_RABIT 0 40 O=C(N[C@H](CO)c1ccccc1)[C@H]1CC(=O)N(Cc2ccc3c(c2)OCO3)C1 ZINC000217924302 GD In-Stock Unstable BACE2 0 40 O=C(N[C@H](CO)c1ccccc1)[C@H]1CC(=O)N(Cc2ccc3c(c2)OCO3)C1 ZINC000217924302 GD In-Stock Unstable NOS2 74 33 O=C(N[C@H](CO)c1ccccc1)[C@H]1CC(=O)N(Cc2ccc3c(c2)OCO3)C1 ZINC000217924302 GD In-Stock Unstable MCHR1 19 42 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccc(C)cc2)cc1OC ZINC000217924332 FH In-Stock Unstable TUBB1 52 37 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccc(C)cc2)cc1OC ZINC000217924332 FH In-Stock Unstable PTPA 0 42 COc1ccc(/C=C/C(=O)N[C@H](C)COc2ccc(C)cc2)cc1OC ZINC000217924332 FH In-Stock Unstable ABCG2 18 43 O=S(=O)(NCC[C@@H](O)C1CCOCC1)c1cccc2ccccc12 ZINC000217924373 EE In-Stock Unstable NPY2R 46 44 O=S(=O)(NCC[C@@H](O)C1CCOCC1)c1cccc2ccccc12 ZINC000217924373 EE In-Stock Unstable NPY5R 20 43 O=S(=O)(NCC[C@@H](O)C1CCOCC1)c1cccc2ccccc12 ZINC000217924373 EE In-Stock Unstable Q95J97_RABIT 0 40 COc1cccc(/C=C/NC(=O)Nc2cccc(Cl)c2Cl)c1 ZINC000217924381 EJ For-Sale Unstable MTNR1A 33 43 COc1cccc(/C=C/NC(=O)Nc2cccc(Cl)c2Cl)c1 ZINC000217924381 EJ For-Sale Unstable MTNR1B 34 43 COc1cccc(/C=C/NC(=O)Nc2cccc(Cl)c2Cl)c1 ZINC000217924381 EJ For-Sale Unstable CYSP_PLAFA 18 40 CCN(CCNC(=O)c1cc(N)ccc1Cl)C1CC1 ZINC000217924388 CE On-Demand Unstable HTR4 21 43 CCN(CCNC(=O)c1cc(N)ccc1Cl)C1CC1 ZINC000217924388 CE On-Demand Unstable P2RX7 18 48 C[C@H]1CN(C)[C@@H](C)C[C@@H]1Nc1ccc2c(c1)C(=O)NC2=O ZINC000217924422 CD For-Sale Unstable CDK4 0 42 O=S(=O)(NCC[C@H](O)C1CCOCC1)c1ccc(F)c(Cl)c1 ZINC000217924468 FD In-Stock Unstable LEF 34 44 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)Cc1ccc(NC(C)=O)cc1 ZINC000217924486 HF For-Sale Unstable TSHR 63 38 COc1cccc(/C=C/NC(=O)Nc2cc(Cl)ccc2Cl)c1 ZINC000217924489 EJ For-Sale Unstable TAAR1 17 41 C[C@@H]1CCC[C@@H](CNc2ncc([N+](=O)[O-])cc2C#N)C1 ZINC000217924501 CG On-Demand Unstable PRKCQ 45 38 N[C@@H]1CCC[C@@H]1N1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217924505 BE For-Sale Unstable CYP2D26 0 45 Cc1cc(NC(=O)C2C[C@@H]3CCC[C@H](C2)C3=O)n(-c2cccc(C(F)(F)F)c2)n1 ZINC000217924532 HJ On-Demand Unstable NPY5R 15 41 O=C(N[C@@H]1CCC[C@@H]1CO)c1ccc2cc[nH]c2c1 ZINC000217924536 CE For-Sale Unstable SSTR3 32 42 O=S(=O)(NCC[C@@H](O)C1CCOCC1)c1ccc(F)c(Cl)c1 ZINC000217924549 FD In-Stock Unstable LEF 34 44 CN(Cc1cccnc1)Cc1ccccc1/C=C\C(=O)O ZINC000217924556 CF For-Sale Unstable PTGER2 49 43 CN(Cc1cccnc1)Cc1ccccc1/C=C\C(=O)O ZINC000217924556 CF For-Sale Unstable TBXAS1 34 49 CN(Cc1cccnc1)Cc1ccccc1/C=C\C(=O)O ZINC000217924556 CF For-Sale Unstable PTGER4 24 44 CN(Cc1cccnc1)Cc1ccccc1/C=C\C(=O)O ZINC000217924556 CF For-Sale Unstable PTGER3 20 44 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)Cc1ccc(NC(C)=O)cc1 ZINC000217924572 HF For-Sale Unstable TSHR 63 38 C[C@H]1CCC[C@@H](CNc2ncc([N+](=O)[O-])cc2C#N)C1 ZINC000217924591 CG On-Demand Unstable PRKCQ 45 38 N[C@H]1CCC[C@@H]1N1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217924594 BE For-Sale Unstable CYP2D26 0 45 COc1cccc(/C=C/NC(=O)Nc2ccc(OC)c(Cl)c2)c1 ZINC000217924600 EI For-Sale Unstable CYP1B1 27 42 COc1cccc(/C=C/NC(=O)Nc2ccc(OC)c(Cl)c2)c1 ZINC000217924600 EI For-Sale Unstable MTNR1A 24 44 COc1cccc(/C=C/NC(=O)Nc2ccc(OC)c(Cl)c2)c1 ZINC000217924600 EI For-Sale Unstable MTNR1B 31 44 COc1cccc(/C=C/NC(=O)Nc2ccc(OC)c(Cl)c2)c1 ZINC000217924600 EI For-Sale Unstable CYP1A1 24 42 COc1cccc(/C=C/NC(=O)Nc2ccc(OC)c(Cl)c2)c1 ZINC000217924600 EI For-Sale Unstable Q8MMZ8_EIMTE 0 41 COc1cccc(/C=C/NC(=O)Nc2ccc(OC)c(Cl)c2)c1 ZINC000217924600 EI For-Sale Unstable TAAR1 22 42 COc1cccc(/C=C/NC(=O)Nc2ccc(OC)c(Cl)c2)c1 ZINC000217924600 EI For-Sale Unstable CYSP_PLAFA 42 39 CCCCOC(=O)c1cc(F)cc(N)c1F ZINC000217924605 BF On-Demand Unstable Q9FYV8_MAIZE 19 40 O=C(N[C@H]1CCC[C@@H]1CO)c1ccc2cc[nH]c2c1 ZINC000217924625 CE For-Sale Unstable SSTR3 32 42 COc1ccc(/C=C/C(=O)N[C@@H](C)c2ccc(N3CCC[C@@H](C)C3)cc2)cc1OC ZINC000217924640 HJ In-Stock Unstable KCNQ2 21 44 COc1ccc(/C=C/C(=O)N[C@@H](C)c2ccc(N3CCC[C@@H](C)C3)cc2)cc1OC ZINC000217924640 HJ In-Stock Unstable RORC 40 39 COc1ccccc1-c1ncc(-c2ccccc2)[nH]1 ZINC000217924652 CH Annotated Unstable LUCI_PHOPE 23 43 COc1ccccc1-c1ncc(-c2ccccc2)[nH]1 ZINC000217924652 CH Annotated Unstable SMO 59 46 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)Cc1ccc(NC(C)=O)cc1 ZINC000217924656 HF For-Sale Unstable TSHR 63 38 CN(Cc1ccc(/C=C\C(=O)O)cc1)Cc1cccnc1 ZINC000217924668 CF For-Sale Unstable TBXAS1 35 70 CN(Cc1ccc(/C=C\C(=O)O)cc1)Cc1cccnc1 ZINC000217924668 CF For-Sale Unstable NR1D1 40 39 C[C@@H]1CCC[C@H](CNc2ncc([N+](=O)[O-])cc2C#N)C1 ZINC000217924669 CG On-Demand Unstable PRKCQ 45 38 N[C@@H]1CCC[C@H]1N1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217924684 BE For-Sale Unstable CYP2D26 0 45 COc1cccc(/C=C/NC(=O)Nc2cccc(C(F)(F)F)c2)c1 ZINC000217924703 EJ For-Sale Unstable KIT 17 43 COc1cccc(/C=C/NC(=O)Nc2cccc(C(F)(F)F)c2)c1 ZINC000217924703 EJ For-Sale Unstable UL80 22 43 COc1cccc(/C=C/NC(=O)Nc2cccc(C(F)(F)F)c2)c1 ZINC000217924703 EJ For-Sale Unstable RAF1 26 41 COc1cccc(/C=C/NC(=O)Nc2cccc(C(F)(F)F)c2)c1 ZINC000217924703 EJ For-Sale Unstable KDR 24 41 COc1cccc(/C=C/NC(=O)Nc2cccc(C(F)(F)F)c2)c1 ZINC000217924703 EJ For-Sale Unstable MTNR1A 22 43 COc1cccc(/C=C/NC(=O)Nc2cccc(C(F)(F)F)c2)c1 ZINC000217924703 EJ For-Sale Unstable MTNR1B 28 43 COc1cccc(/C=C/NC(=O)Nc2cccc(C(F)(F)F)c2)c1 ZINC000217924703 EJ For-Sale Unstable EPHX2 16 45 COc1cccc(/C=C/NC(=O)Nc2cccc(C(F)(F)F)c2)c1 ZINC000217924703 EJ For-Sale Unstable TEK 40 41 COc1cccc(/C=C/NC(=O)Nc2cccc(C(F)(F)F)c2)c1 ZINC000217924703 EJ For-Sale Unstable BTK 17 44 COc1cccc(/C=C/NC(=O)Nc2cccc(C(F)(F)F)c2)c1 ZINC000217924703 EJ For-Sale Unstable TAAR1 37 43 COc1cccc(/C=C/NC(=O)Nc2cccc(C(F)(F)F)c2)c1 ZINC000217924703 EJ For-Sale Unstable AKR1C3 17 51 COc1cccc(/C=C/NC(=O)Nc2cccc(C(F)(F)F)c2)c1 ZINC000217924703 EJ For-Sale Unstable AKR1C2 23 51 COc1cccc(/C=C/NC(=O)Nc2cccc(C(F)(F)F)c2)c1 ZINC000217924703 EJ For-Sale Unstable KCNK3 41 40 O=C(N[C@@H]1CCC[C@H]1CO)c1ccc2cc[nH]c2c1 ZINC000217924713 CE For-Sale Unstable SSTR3 32 42 COc1ccc(/C=C/C(=O)N[C@H](C)c2ccc(N3CCC[C@@H](C)C3)cc2)cc1OC ZINC000217924732 HJ In-Stock Unstable KCNQ2 21 44 COc1ccc(/C=C/C(=O)N[C@H](C)c2ccc(N3CCC[C@@H](C)C3)cc2)cc1OC ZINC000217924732 HJ In-Stock Unstable RORC 40 39 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)Cc1ccc(NC(C)=O)cc1 ZINC000217924741 HF For-Sale Unstable TSHR 63 38 C[C@H]1CCC[C@H](CNc2ncc([N+](=O)[O-])cc2C#N)C1 ZINC000217924757 CG On-Demand Unstable PRKCQ 45 38 Cc1cc(NC(=O)Cc2ccc(OCc3c(C)noc3C)cc2)n(-c2cccc(C(F)(F)F)c2)n1 ZINC000217924758 JK On-Demand Unstable P2RX7 15 40 Cc1cc(NC(=O)Cc2ccc(OCc3c(C)noc3C)cc2)n(-c2cccc(C(F)(F)F)c2)n1 ZINC000217924758 JK On-Demand Unstable PDS 40 31 CN(C)[C@H](CN)[C@H]1CCN(C(=O)OC(C)(C)C)C1 ZINC000217924764 CD For-Sale Unstable GPR119 31 40 O=C(N[C@H]1CCC[C@H]1CO)c1ccc2cc[nH]c2c1 ZINC000217924769 CE On-Demand Unstable SSTR3 31 42 CN(Cc1cccnc1)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217924783 CF For-Sale Unstable TBXAS1 38 57 CN(Cc1cccnc1)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217924783 CF For-Sale Unstable AKR1C3 40 39 CN(Cc1cccnc1)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217924783 CF For-Sale Unstable NR1D1 40 40 COc1cccc(/C=C/NC(=O)Nc2ccccc2C#N)c1 ZINC000217924815 CG For-Sale Unstable TAAR1 20 41 CN(C)[C@H](CN)[C@@H]1CCN(C(=O)OC(C)(C)C)C1 ZINC000217924850 CD For-Sale Unstable GPR119 31 40 Cc1cc(NC(=O)Cn2c(=O)ccn(Cc3ccccc3)c2=O)n(-c2cccc(C(F)(F)F)c2)n1 ZINC000217924873 JG On-Demand Unstable NPY5R 15 44 COc1ccc(/C=C\C(=O)O)cc1CN(C)CC(F)(F)F ZINC000217924886 DF For-Sale Unstable TUBB1 42 37 COc1ccc(/C=C\C(=O)O)cc1CN(C)CC(F)(F)F ZINC000217924886 DF For-Sale Unstable AKR1C3 39 40 CCOC(=O)c1ccccc1NC(=O)N/C=C/c1cccc(OC)c1 ZINC000217924920 EH For-Sale Unstable MTNR1A 31 42 CCOC(=O)c1ccccc1NC(=O)N/C=C/c1cccc(OC)c1 ZINC000217924920 EH For-Sale Unstable MTNR1B 32 42 CN(C)[C@@H](CN)[C@H]1CCN(C(=O)OC(C)(C)C)C1 ZINC000217924925 CD For-Sale Unstable GPR119 31 40 CC[C@@H](CCO)NC(=O)[C@@H](N)CCC(=O)O ZINC000217924933 BB For-Sale Unstable FOLH1 15 56 CC[C@@H](CCO)NC(=O)[C@@H](N)CCC(=O)O ZINC000217924933 BB For-Sale Unstable GRM8 15 45 CC[C@@H](CCO)NC(=O)[C@@H](N)CCC(=O)O ZINC000217924933 BB For-Sale Unstable GRIK3 20 45 Cc1cc(NC(=O)CCc2ccc3c(c2)OCCO3)n(-c2cccc(C(F)(F)F)c2)n1 ZINC000217924993 IJ On-Demand Unstable NPY5R 15 42 Cc1cc(NC(=O)CCc2ccc3c(c2)OCCO3)n(-c2cccc(C(F)(F)F)c2)n1 ZINC000217924993 IJ On-Demand Unstable LUXR 19 41 CN(C)[C@@H](CN)[C@@H]1CCN(C(=O)OC(C)(C)C)C1 ZINC000217925014 CD For-Sale Unstable GPR119 31 40 CC[C@H](CCO)NC(=O)[C@@H](N)CCC(=O)O ZINC000217925020 BB For-Sale Unstable FOLH1 15 56 CC[C@H](CCO)NC(=O)[C@@H](N)CCC(=O)O ZINC000217925020 BB For-Sale Unstable GRM8 15 45 CC[C@H](CCO)NC(=O)[C@@H](N)CCC(=O)O ZINC000217925020 BB For-Sale Unstable GRIK3 20 45 COc1cccc(/C=C/NC(=O)Nc2ccc(O)cc2)c1 ZINC000217925026 CG For-Sale Unstable CYP1B1 23 41 COc1cccc(/C=C/NC(=O)Nc2ccc(O)cc2)c1 ZINC000217925026 CG For-Sale Unstable MTNR1A 33 51 COc1cccc(/C=C/NC(=O)Nc2ccc(O)cc2)c1 ZINC000217925026 CG For-Sale Unstable MTNR1B 37 51 COc1cccc(/C=C/NC(=O)Nc2ccc(O)cc2)c1 ZINC000217925026 CG For-Sale Unstable MMP2 0 54 COc1cccc(/C=C/NC(=O)Nc2ccc(O)cc2)c1 ZINC000217925026 CG For-Sale Unstable CYP1A1 17 41 COc1cccc(/C=C/NC(=O)Nc2ccc(O)cc2)c1 ZINC000217925026 CG For-Sale Unstable MMP9 0 50 COc1cccc(/C=C/NC(=O)Nc2ccc(O)cc2)c1 ZINC000217925026 CG For-Sale Unstable MMP1 0 50 COc1cccc(/C=C/NC(=O)Nc2ccc(O)cc2)c1 ZINC000217925026 CG For-Sale Unstable Q8MMZ8_EIMTE 0 45 COc1cccc(/C=C/NC(=O)Nc2ccc(O)cc2)c1 ZINC000217925026 CG For-Sale Unstable AKR1C2 41 33 COc1ccc([C@@H]2CC(=O)Oc3c(C(C)=O)c(O)c4c(C)cc(=O)oc4c32)cc1OC ZINC000217925062 HG In-Stock Unstable NTBBF1.1 0 41 COc1ccc(CCS(=O)(=O)NCC[C@H](O)C2CCOCC2)cc1 ZINC000217925080 FD In-Stock Unstable BMP1 48 34 COc1ccc(CCS(=O)(=O)NCC[C@H](O)C2CCOCC2)cc1 ZINC000217925080 FD In-Stock Unstable MMP13 31 53 COc1ccc(CCS(=O)(=O)NCC[C@H](O)C2CCOCC2)cc1 ZINC000217925080 FD In-Stock Unstable MMP8 20 46 COc1ccc(CCS(=O)(=O)NCC[C@H](O)C2CCOCC2)cc1 ZINC000217925080 FD In-Stock Unstable MMP12 21 53 CC[C@@H](CCO)NC(=O)[C@H](N)CCC(=O)O ZINC000217925115 BB For-Sale Unstable FOLH1 15 56 CC[C@@H](CCO)NC(=O)[C@H](N)CCC(=O)O ZINC000217925115 BB For-Sale Unstable GRM8 15 45 CC[C@@H](CCO)NC(=O)[C@H](N)CCC(=O)O ZINC000217925115 BB For-Sale Unstable GRIK3 20 45 COc1cccc(/C=C/NC(=O)Nc2cc(Cl)ccc2OC)c1 ZINC000217925126 EI For-Sale Unstable CYP1B1 27 42 COc1cccc(/C=C/NC(=O)Nc2cc(Cl)ccc2OC)c1 ZINC000217925126 EI For-Sale Unstable MTNR1A 24 42 COc1cccc(/C=C/NC(=O)Nc2cc(Cl)ccc2OC)c1 ZINC000217925126 EI For-Sale Unstable MTNR1B 28 42 COc1cccc(/C=C/NC(=O)Nc2cc(Cl)ccc2OC)c1 ZINC000217925126 EI For-Sale Unstable CYP1A1 24 42 COc1cccc(/C=C/NC(=O)Nc2cc(Cl)ccc2OC)c1 ZINC000217925126 EI For-Sale Unstable RBP4 23 41 COc1cccc(/C=C/NC(=O)Nc2cc(Cl)ccc2OC)c1 ZINC000217925126 EI For-Sale Unstable CYSP_PLAFA 45 39 Nc1cc(F)cc(C(=O)OCc2cccc(Cl)c2)c1F ZINC000217925154 CH On-Demand Unstable MAOB 26 40 COc1ccc([C@H]2CC(=O)Oc3c(C(C)=O)c(O)c4c(C)cc(=O)oc4c32)cc1OC ZINC000217925159 HG In-Stock Unstable NTBBF1.1 0 41 COc1ccc(CCS(=O)(=O)NCC[C@@H](O)C2CCOCC2)cc1 ZINC000217925164 FD In-Stock Unstable BMP1 48 34 COc1ccc(CCS(=O)(=O)NCC[C@@H](O)C2CCOCC2)cc1 ZINC000217925164 FD In-Stock Unstable MMP13 31 53 COc1ccc(CCS(=O)(=O)NCC[C@@H](O)C2CCOCC2)cc1 ZINC000217925164 FD In-Stock Unstable MMP8 20 46 COc1ccc(CCS(=O)(=O)NCC[C@@H](O)C2CCOCC2)cc1 ZINC000217925164 FD In-Stock Unstable MMP12 21 53 Cc1nc(CC(C)C)cc(C(=O)N2CCC[C@@H]2c2ccccn2)n1 ZINC000217925174 DG In-Stock Unstable ADAM17 0 41 Cc1nc(CC(C)C)cc(C(=O)N2CCC[C@@H]2c2ccccn2)n1 ZINC000217925174 DG In-Stock Unstable COLA 86 38 Cc1nc(CC(C)C)cc(C(=O)N2CCC[C@@H]2c2ccccn2)n1 ZINC000217925174 DG In-Stock Unstable CPT1A 81 38 CC[C@H](CCO)NC(=O)[C@H](N)CCC(=O)O ZINC000217925194 BB For-Sale Unstable FOLH1 15 56 CC[C@H](CCO)NC(=O)[C@H](N)CCC(=O)O ZINC000217925194 BB For-Sale Unstable GRM8 15 45 CC[C@H](CCO)NC(=O)[C@H](N)CCC(=O)O ZINC000217925194 BB For-Sale Unstable GRIK3 20 45 COc1ccc2c(c1)[C@@H](NC(=O)/C=C/c1ccc(OC)c(OC)c1)CC(C)(C)O2 ZINC000217925198 GI In-Stock Unstable ABCG2 18 42 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc(NC(C)=O)cc1 ZINC000217925223 HF For-Sale Unstable CFTR 41 34 CCCCc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217925239 DJ For-Sale Unstable INHA 52 40 CCCCc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217925239 DJ For-Sale Unstable SCN2A 17 45 CCCCc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217925239 DJ For-Sale Unstable MTNR1A 47 49 CCCCc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217925239 DJ For-Sale Unstable MTNR1B 50 49 CCCCc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217925239 DJ For-Sale Unstable CFTR 45 36 CCCCc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217925239 DJ For-Sale Unstable P96878_MYCTU 16 45 CCCCc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217925239 DJ For-Sale Unstable ACAT 0 47 Cc1nc(CC(C)C)cc(C(=O)N2CCC[C@H]2c2ccccn2)n1 ZINC000217925253 DG In-Stock Unstable ADAM17 0 41 Cc1nc(CC(C)C)cc(C(=O)N2CCC[C@H]2c2ccccn2)n1 ZINC000217925253 DG In-Stock Unstable COLA 86 38 Cc1nc(CC(C)C)cc(C(=O)N2CCC[C@H]2c2ccccn2)n1 ZINC000217925253 DG In-Stock Unstable CPT1A 81 38 COC(=O)C[C@H](c1cccc(OC)c1OCCc1ccccc1)c1c(O)c2ccccc2oc1=O ZINC000217925274 JJ In-Stock Unstable NQO1 39 45 COC(=O)C[C@H](c1cccc(OC)c1OCCc1ccccc1)c1c(O)c2ccccc2oc1=O ZINC000217925274 JJ In-Stock Unstable ABCG2 17 41 COc1ccc2c(c1)[C@H](NC(=O)/C=C/c1ccc(OC)c(OC)c1)CC(C)(C)O2 ZINC000217925277 GI In-Stock Unstable ABCG2 18 42 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc(NC(C)=O)cc1 ZINC000217925301 HF For-Sale Unstable CFTR 41 34 N#C[C@@H]1CCCC[C@@H]1N1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217925348 BH For-Sale Unstable CYP2D26 0 41 COc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217925351 CG For-Sale Unstable CYP1B1 47 42 COc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217925351 CG For-Sale Unstable CA1 48 39 COc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217925351 CG For-Sale Unstable AHR 33 43 COc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217925351 CG For-Sale Unstable RAF1 27 50 COc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217925351 CG For-Sale Unstable KDR 27 41 COc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217925351 CG For-Sale Unstable MTNR1A 56 53 COc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217925351 CG For-Sale Unstable MTNR1B 56 53 COc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217925351 CG For-Sale Unstable CYP1A1 30 45 COc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217925351 CG For-Sale Unstable ACR 20 41 COc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217925351 CG For-Sale Unstable CA12 21 44 COc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217925351 CG For-Sale Unstable PDGFRA 42 41 COc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217925351 CG For-Sale Unstable CA9 22 44 COc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217925351 CG For-Sale Unstable Q8MMZ8_EIMTE 27 50 COc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217925351 CG For-Sale Unstable AKR1C3 22 43 COc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217925351 CG For-Sale Unstable AKR1C2 50 38 COc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217925351 CG For-Sale Unstable IMDH_CRYPV 18 45 COC(=O)C[C@@H](c1cccc(OC)c1OCCc1ccccc1)c1c(O)c2ccccc2oc1=O ZINC000217925361 JJ In-Stock Unstable NQO1 39 45 COC(=O)C[C@@H](c1cccc(OC)c1OCCc1ccccc1)c1c(O)c2ccccc2oc1=O ZINC000217925361 JJ In-Stock Unstable ABCG2 17 41 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc(NC(C)=O)cc1 ZINC000217925377 HF For-Sale Unstable CFTR 41 34 CCCN(Cc1ccccc1/C=C\C(=O)O)CC1CC1 ZINC000217925383 CG For-Sale Unstable PTGER2 38 44 CCCN(Cc1ccccc1/C=C\C(=O)O)CC1CC1 ZINC000217925383 CG For-Sale Unstable PTGER4 0 44 CCCN(Cc1ccccc1/C=C\C(=O)O)CC1CC1 ZINC000217925383 CG For-Sale Unstable PTGER3 15 44 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)/C=C/c1ccc(OC)c(OC)c1 ZINC000217925401 GI In-Stock Unstable PTPA 0 44 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)/C=C/c1ccc(OC)c(OC)c1 ZINC000217925401 GI In-Stock Unstable ABCG2 20 42 N#C[C@H]1CCCC[C@@H]1N1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217925440 BH For-Sale Unstable CYP2D26 0 41 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cc2Cl)c1 ZINC000217925442 EJ For-Sale Unstable TAAR1 18 41 O=C(/C=C/c1ccc(Br)cc1)N[C@H]1CCC[C@H]1CO ZINC000217925460 DF On-Demand Unstable HDAC8 0 42 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc(NC(C)=O)cc1 ZINC000217925461 HF For-Sale Unstable CFTR 41 34 COc1cccc2c1ccn2CCNC(=O)Cc1cn(C)c2ccccc12 ZINC000217925467 FH In-Stock Unstable CNR1 0 41 COc1cccc2c1ccn2CCNC(=O)Cc1cn(C)c2ccccc12 ZINC000217925467 FH In-Stock Unstable CYSLTR1 47 33 COc1cccc2c1ccn2CCNC(=O)Cc1cn(C)c2ccccc12 ZINC000217925467 FH In-Stock Unstable CNR2 15 41 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)/C=C/c1ccc(OC)c(OC)c1 ZINC000217925470 GI In-Stock Unstable PTPA 0 44 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)/C=C/c1ccc(OC)c(OC)c1 ZINC000217925470 GI In-Stock Unstable ABCG2 20 42 CCN(CCOC)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217925493 CE For-Sale Unstable LTB4R 17 42 CCN(CCOC)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217925493 CE For-Sale Unstable SQLE 48 32 N#C[C@@H]1CCCC[C@H]1N1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217925523 BH For-Sale Unstable CYP2D26 0 41 COc1cccc(/C=C/NC(=O)NCCc2ccc(O)cc2)c1 ZINC000217925545 DF For-Sale Unstable MTNR1A 102 47 COc1cccc(/C=C/NC(=O)NCCc2ccc(O)cc2)c1 ZINC000217925545 DF For-Sale Unstable MTNR1B 92 47 COc1cccc(/C=C/NC(=O)NCCc2ccc(O)cc2)c1 ZINC000217925545 DF For-Sale Unstable SLC6A5 22 42 COc1cccc(/C=C/NC(=O)NCCc2ccc(O)cc2)c1 ZINC000217925545 DF For-Sale Unstable NCE103 16 45 COc1cccc(/C=C/NC(=O)NCCc2ccc(O)cc2)c1 ZINC000217925545 DF For-Sale Unstable ABCG2 21 43 N[C@H]1CNC[C@H]1c1cc(Cl)ccc1F ZINC000217925583 BD For-Sale Unstable HTR2B 15 43 COc1ccnc(NC[C@@H]2CCC[C@@H](C)C2)n1 ZINC000217925610 BF On-Demand Unstable PKNB 17 43 CCN(CCOC)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217925623 CE For-Sale Unstable ERG2 18 44 CCN(CCOC)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217925623 CE For-Sale Unstable AHR 15 41 COc1cccc(/C=C/NC(=O)NC(C)C)c1 ZINC000217925639 BE For-Sale Unstable CYP1B1 28 43 COc1cccc(/C=C/NC(=O)NC(C)C)c1 ZINC000217925639 BE For-Sale Unstable AHR 15 44 COc1cccc(/C=C/NC(=O)NC(C)C)c1 ZINC000217925639 BE For-Sale Unstable MTNR1A 41 45 COc1cccc(/C=C/NC(=O)NC(C)C)c1 ZINC000217925639 BE For-Sale Unstable MTNR1B 44 45 COc1cccc(/C=C/NC(=O)NC(C)C)c1 ZINC000217925639 BE For-Sale Unstable CYP1A1 24 43 COc1cccc(/C=C/NC(=O)NC(C)C)c1 ZINC000217925639 BE For-Sale Unstable NR1H4 29 40 O=S(=O)(NCC[C@H](O)C1CCOCC1)c1ccc(C(F)(F)F)cc1 ZINC000217925652 FE In-Stock Unstable CACNA1B 15 40 C[C@H]1CN(C)[C@H](C)C[C@H]1N[C@H](C)c1ccc(F)cc1 ZINC000217925659 CG For-Sale Unstable SLC6A3 16 40 CC[C@@H](CCO)NC(=O)CCC[C@@H](C)N ZINC000217925667 BC For-Sale Unstable PLA2G2C 0 40 CC[C@@H](CCO)NC(=O)CCC[C@@H](C)N ZINC000217925667 BC For-Sale Unstable Q6UB75_PIG 0 42 CC[C@@H](CCO)NC(=O)CCC[C@@H](C)N ZINC000217925667 BC For-Sale Unstable NOD1 89 39 N[C@@H]1CNC[C@H]1c1cc(Cl)ccc1F ZINC000217925676 BD For-Sale Unstable HTR2B 15 43 COc1ccnc(NC[C@H]2CCC[C@@H](C)C2)n1 ZINC000217925694 BF On-Demand Unstable PKNB 17 43 CC[C@@H]1CO[C@H](C)CN1Cc1ccccc1/C=C\C(=O)O ZINC000217925710 CF For-Sale Unstable PTGER2 30 40 CC[C@@H]1CO[C@H](C)CN1Cc1ccccc1/C=C\C(=O)O ZINC000217925710 CF For-Sale Unstable PTGER4 15 40 CC[C@@H]1CO[C@H](C)CN1Cc1ccccc1/C=C\C(=O)O ZINC000217925710 CF For-Sale Unstable PTGER3 16 40 O=S(=O)(NCC[C@@H](O)C1CCOCC1)c1ccc(C(F)(F)F)cc1 ZINC000217925723 FE In-Stock Unstable CACNA1B 15 40 C[C@H](N[C@@H]1C[C@@H](C)N(C)C[C@@H]1C)c1ccc(F)cc1 ZINC000217925730 CG For-Sale Unstable SLC6A3 16 40 CC[C@H](CCO)NC(=O)CCC[C@@H](C)N ZINC000217925732 BC For-Sale Unstable PLA2G2C 0 40 CC[C@H](CCO)NC(=O)CCC[C@@H](C)N ZINC000217925732 BC For-Sale Unstable Q6UB75_PIG 0 42 CC[C@H](CCO)NC(=O)CCC[C@@H](C)N ZINC000217925732 BC For-Sale Unstable NOD1 89 39 Cc1nc(Br)nc2ccc(Cl)cc12 ZINC000217925749 CG For-Sale Unstable PRS 17 41 COc1cccc(/C=C/NC(=O)N(Cc2ccccc2)C(C)C)c1 ZINC000217925752 DI For-Sale Unstable TSPO 41 33 COc1cccc(/C=C/NC(=O)N(Cc2ccccc2)C(C)C)c1 ZINC000217925752 DI For-Sale Unstable G6PC 27 47 COc1cccc(/C=C/NC(=O)N(Cc2ccccc2)C(C)C)c1 ZINC000217925752 DI For-Sale Unstable MTNR1A 49 43 COc1cccc(/C=C/NC(=O)N(Cc2ccccc2)C(C)C)c1 ZINC000217925752 DI For-Sale Unstable MTNR1B 53 43 COc1cccc(/C=C/NC(=O)N(Cc2ccccc2)C(C)C)c1 ZINC000217925752 DI For-Sale Unstable ROCK2 27 46 COc1cccc(/C=C/NC(=O)N(Cc2ccccc2)C(C)C)c1 ZINC000217925752 DI For-Sale Unstable NR1H4 44 37 COc1cccc(/C=C/NC(=O)N(Cc2ccccc2)C(C)C)c1 ZINC000217925752 DI For-Sale Unstable PTGES 22 48 CC[C@@H](NC(=O)/C=C/c1ccc(OC)c(OC)c1)c1ccc(C)cc1C ZINC000217925755 FJ In-Stock Unstable TUBB1 42 35 N[C@@H]1CNC[C@@H]1c1cc(Cl)ccc1F ZINC000217925756 BD For-Sale Unstable HTR2B 15 43 COc1ccnc(NC[C@@H]2CCC[C@H](C)C2)n1 ZINC000217925763 BF On-Demand Unstable PKNB 17 43 NCCNC(=O)/C=C\c1ccc(Br)cc1 ZINC000217925775 CD For-Sale Unstable PYGL 22 47 NCCNC(=O)/C=C\c1ccc(Br)cc1 ZINC000217925775 CD For-Sale Unstable HDAC8 43 43 NCCNC(=O)/C=C\c1ccc(Br)cc1 ZINC000217925775 CD For-Sale Unstable MMP2 16 49 NCCNC(=O)/C=C\c1ccc(Br)cc1 ZINC000217925775 CD For-Sale Unstable HDAC1 41 37 NCCNC(=O)/C=C\c1ccc(Br)cc1 ZINC000217925775 CD For-Sale Unstable HDAC6 22 43 NCCNC(=O)/C=C\c1ccc(Br)cc1 ZINC000217925775 CD For-Sale Unstable HDAC9 59 39 NCCNC(=O)/C=C\c1ccc(Br)cc1 ZINC000217925775 CD For-Sale Unstable HDAC7 52 39 C[C@H]1CN(C)[C@H](C)C[C@@H]1N[C@H](C)c1ccc(F)cc1 ZINC000217925812 CG For-Sale Unstable SLC6A3 16 40 CC[C@@H](CCO)NC(=O)CCC[C@H](C)N ZINC000217925820 BC For-Sale Unstable PLA2G2C 0 40 CC[C@@H](CCO)NC(=O)CCC[C@H](C)N ZINC000217925820 BC For-Sale Unstable Q6UB75_PIG 0 42 CC[C@@H](CCO)NC(=O)CCC[C@H](C)N ZINC000217925820 BC For-Sale Unstable NOD1 89 39 CC[C@H](NC(=O)/C=C/c1ccc(OC)c(OC)c1)c1ccc(C)cc1C ZINC000217925832 FJ In-Stock Unstable TUBB1 42 35 COc1ccnc(NC[C@H]2CCC[C@H](C)C2)n1 ZINC000217925844 BF On-Demand Unstable PKNB 17 43 COc1cccc(/C=C/NC(=O)N(C)C2CCCCC2)c1 ZINC000217925847 CH For-Sale Unstable MTNR1A 28 42 COc1cccc(/C=C/NC(=O)N(C)C2CCCCC2)c1 ZINC000217925847 CH For-Sale Unstable MTNR1B 31 42 COc1cccc(/C=C/NC(=O)N(C)C2CCCCC2)c1 ZINC000217925847 CH For-Sale Unstable NR1H4 24 41 Cc1nc(Br)nc2cc(Cl)ccc12 ZINC000217925865 CG For-Sale Unstable ACHE 18 40 C[C@H](N[C@H]1C[C@@H](C)N(C)C[C@@H]1C)c1ccc(F)cc1 ZINC000217925895 CG For-Sale Unstable SLC6A3 16 40 CC[C@H](CCO)NC(=O)CCC[C@H](C)N ZINC000217925899 BC For-Sale Unstable PLA2G2C 0 40 CC[C@H](CCO)NC(=O)CCC[C@H](C)N ZINC000217925899 BC For-Sale Unstable Q6UB75_PIG 0 42 CC[C@H](CCO)NC(=O)CCC[C@H](C)N ZINC000217925899 BC For-Sale Unstable NOD1 89 39 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccccc1C(=O)c1ccc(F)cc1 ZINC000217925909 JI For-Sale Unstable PLA2G4A 35 47 CC[C@@H](NC(=O)/C=C/c1ccc(OC)c(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217925936 GI In-Stock Unstable CYP1B1 19 41 CC[C@@H](NC(=O)/C=C/c1ccc(OC)c(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217925936 GI In-Stock Unstable MMP2 0 49 CC[C@@H](NC(=O)/C=C/c1ccc(OC)c(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217925936 GI In-Stock Unstable CYP1A1 22 41 CC[C@@H](NC(=O)/C=C/c1ccc(OC)c(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217925936 GI In-Stock Unstable TUBB1 56 38 CC[C@@H](NC(=O)/C=C/c1ccc(OC)c(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217925936 GI In-Stock Unstable PDE10A 29 41 CC[C@@H](NC(=O)/C=C/c1ccc(OC)c(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217925936 GI In-Stock Unstable ABCG2 17 48 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccccc1C(=O)c1ccc(F)cc1 ZINC000217925984 JI For-Sale Unstable PLA2G4A 35 47 CC[C@H](NC(=O)/C=C/c1ccc(OC)c(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217926017 GI In-Stock Unstable CYP1B1 19 41 CC[C@H](NC(=O)/C=C/c1ccc(OC)c(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217926017 GI In-Stock Unstable MMP2 0 49 CC[C@H](NC(=O)/C=C/c1ccc(OC)c(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217926017 GI In-Stock Unstable CYP1A1 22 41 CC[C@H](NC(=O)/C=C/c1ccc(OC)c(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217926017 GI In-Stock Unstable TUBB1 56 38 CC[C@H](NC(=O)/C=C/c1ccc(OC)c(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217926017 GI In-Stock Unstable PDE10A 29 41 CC[C@H](NC(=O)/C=C/c1ccc(OC)c(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217926017 GI In-Stock Unstable ABCG2 17 48 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccccc1C(=O)c1ccc(F)cc1 ZINC000217926075 JI For-Sale Unstable PLA2G4A 35 47 O=C(Cn1cnc2ccsc2c1=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217926078 GD In-Stock Unstable CHRNA4 27 43 Nc1cc(F)cc(C(=O)OCC2CCCC2)c1F ZINC000217926094 CF On-Demand Unstable HTR4 35 45 CC[C@@H](NC(=O)/C=C/c1ccc(OC)c(OC)c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217926142 HG In-Stock Unstable ABCG2 15 44 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccccc1C(=O)c1ccc(F)cc1 ZINC000217926158 JI For-Sale Unstable PLA2G4A 35 47 CCCCCCCCOC(=O)c1cc(F)cc(N)c1F ZINC000217926170 CI On-Demand Unstable PLA2G4B 43 31 CCN(CCNC(=O)c1ccc(N)c(Cl)c1)C1CC1 ZINC000217926176 CE For-Sale Unstable HTR4 21 42 CC[C@H](C)[C@H](C(=O)N[C@H](CO)c1ccccc1)N1Cc2ccccc2C1=O ZINC000217926199 FF In-Stock Unstable GPR88 0 44 CC[C@H](NC(=O)/C=C/c1ccc(OC)c(OC)c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217926222 HG In-Stock Unstable ABCG2 15 44 CCOC(=O)C1CCN(C(=O)N/C=C/c2cccc(OC)c2)CC1 ZINC000217926248 EF For-Sale Unstable DRD4 40 31 CCOC(=O)C1CCN(C(=O)N/C=C/c2cccc(OC)c2)CC1 ZINC000217926248 EF For-Sale Unstable FDFT1 0 43 CCC1CCN(Cc2ccc(F)cc2/C=C\C(=O)O)CC1 ZINC000217926255 CH For-Sale Unstable SIGMAR1 31 41 CCC1CCN(Cc2ccc(F)cc2/C=C\C(=O)O)CC1 ZINC000217926255 CH For-Sale Unstable CCR3 44 40 Cc1cccc2c(Cl)nc(Br)nc12 ZINC000217926302 CG For-Sale Unstable TNKS 30 41 Cc1cccc2c(Cl)nc(Br)nc12 ZINC000217926302 CG For-Sale Unstable TNKS2 20 41 COc1cccc(-c2noc(CNC(=O)/C=C/c3ccc(OC)c(OC)c3)n2)c1 ZINC000217926341 GG In-Stock Unstable PTPA 0 42 CCC1CCN(Cc2ccc(F)c(/C=C\C(=O)O)c2)CC1 ZINC000217926355 CH For-Sale Unstable ACHE 31 42 CCC1CCN(Cc2ccc(F)c(/C=C\C(=O)O)c2)CC1 ZINC000217926355 CH For-Sale Unstable SIGMAR1 43 44 CCC1CCN(Cc2ccc(F)c(/C=C\C(=O)O)c2)CC1 ZINC000217926355 CH For-Sale Unstable CCR1 0 40 CCC1CCN(Cc2ccc(F)c(/C=C\C(=O)O)c2)CC1 ZINC000217926355 CH For-Sale Unstable CCR3 50 42 CCC1CCN(Cc2ccc(F)c(/C=C\C(=O)O)c2)CC1 ZINC000217926355 CH For-Sale Unstable MCHR1 30 40 COc1cccc(/C=C/NC(=O)NC2CCCCC2)c1 ZINC000217926362 CG For-Sale Unstable MTNR1A 37 40 COc1cccc(/C=C/NC(=O)NC2CCCCC2)c1 ZINC000217926362 CG For-Sale Unstable MTNR1B 40 40 COc1cccc(/C=C/NC(=O)NC2CCCCC2)c1 ZINC000217926362 CG For-Sale Unstable NR1H4 22 40 COc1cccc(/C=C/NC(=O)NC2CCCCC2)c1 ZINC000217926362 CG For-Sale Unstable FAAH 26 46 COc1cccc(/C=C/NC(=O)NC2CCCCC2)c1 ZINC000217926362 CG For-Sale Unstable EPHX2 28 50 COC(=O)c1ccnc(-n2ccc([N+](=O)[O-])n2)c1 ZINC000217926383 BC For-Sale Unstable KDM3A 0 47 COC(=O)c1ccnc(-n2ccc([N+](=O)[O-])n2)c1 ZINC000217926383 BC For-Sale Unstable KDM5C 0 47 O=C([C@@H]1C[C@@H](O)CN1)N1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217926444 CC For-Sale Unstable DPP4 15 43 O=C([C@@H]1C[C@@H](O)CN1)N1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217926444 CC For-Sale Unstable DPP9 0 43 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccc(OC)c(OC)c3)n2)c(OC)c1 ZINC000217926462 IG In-Stock Unstable CYP1B1 30 40 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccc(OC)c(OC)c3)n2)c(OC)c1 ZINC000217926462 IG In-Stock Unstable CYP1A1 22 40 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccc(OC)c(OC)c3)n2)c(OC)c1 ZINC000217926462 IG In-Stock Unstable ABCG2 19 42 COc1cccc(/C=C/NC(=O)N2CCC(C)CC2)c1 ZINC000217926468 CG For-Sale Unstable DRD4 40 30 COc1cccc(/C=C/NC(=O)N2CCC(C)CC2)c1 ZINC000217926468 CG For-Sale Unstable MTNR1A 27 40 COc1cccc(/C=C/NC(=O)N2CCC(C)CC2)c1 ZINC000217926468 CG For-Sale Unstable MTNR1B 37 40 O=C(O)/C=C\c1cccc(OCCN2CCCSCC2)c1 ZINC000217926472 DF For-Sale Unstable ESR1 40 36 O=C(O)/C=C\c1cccc(OCCN2CCCSCC2)c1 ZINC000217926472 DF For-Sale Unstable ESR2 29 46 O=C(O)/C=C\c1cccc(OCCN2CCCSCC2)c1 ZINC000217926472 DF For-Sale Unstable LTA4H 44 46 O=C(O)/C=C\c1cccc(OCCN2CCCSCC2)c1 ZINC000217926472 DF For-Sale Unstable HRH3 24 40 O=C(O)/C=C\c1cccc(OCCN2CCCSCC2)c1 ZINC000217926472 DF For-Sale Unstable PSMB2 51 42 O=C(O)/C=C\c1cccc(OCCN2CCCSCC2)c1 ZINC000217926472 DF For-Sale Unstable PSMB5 17 42 O=C(O)/C=C\c1cccc(OCCN2CCCSCC2)c1 ZINC000217926472 DF For-Sale Unstable PSMB1 44 42 O=C([C@H]1C[C@H](O)CN1)N1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217926513 CC For-Sale Unstable DPP4 15 43 O=C([C@H]1C[C@H](O)CN1)N1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217926513 CC For-Sale Unstable DPP9 0 43 COc1cccc(/C=C/NC(=O)N2CCC(C(=O)O)CC2)c1 ZINC000217926568 DE For-Sale Unstable DRD4 43 33 COc1ccc(/C=C/C(=O)NCc2nc(-c3ccccc3Cl)no2)cc1OC ZINC000217926569 GH In-Stock Unstable BDKRB2 59 34 COc1ccc(/C=C/C(=O)NCc2nc(-c3ccccc3Cl)no2)cc1OC ZINC000217926569 GH In-Stock Unstable CYSP_PLAFA 19 43 O=C(O)/C=C\c1cccc(CN2CCC(CO)CC2)c1 ZINC000217926571 CD For-Sale Unstable DRD2 19 45 O=C(O)/C=C\c1cccc(CN2CCC(CO)CC2)c1 ZINC000217926571 CD For-Sale Unstable DRD4 41 45 O=C(O)/C=C\c1cccc(CN2CCC(CO)CC2)c1 ZINC000217926571 CD For-Sale Unstable ACHE 50 47 O=C(O)/C=C\c1cccc(CN2CCC(CO)CC2)c1 ZINC000217926571 CD For-Sale Unstable CHRM3 23 41 O=C(O)/C=C\c1cccc(CN2CCC(CO)CC2)c1 ZINC000217926571 CD For-Sale Unstable GRIN2B 27 40 O=C(O)/C=C\c1cccc(CN2CCC(CO)CC2)c1 ZINC000217926571 CD For-Sale Unstable SIGMAR1 63 51 O=C(O)/C=C\c1cccc(CN2CCC(CO)CC2)c1 ZINC000217926571 CD For-Sale Unstable CCR3 46 41 O=C([C@H]1C[C@@H](O)CN1)N1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217926588 CC For-Sale Unstable DPP4 15 43 O=C([C@H]1C[C@@H](O)CN1)N1CC[C@@H]2CCCC[C@@H]2C1 ZINC000217926588 CC For-Sale Unstable DPP9 0 43 CCC(C)(C)c1ccc(Oc2ccc(NC(=O)Cn3cnc(C#N)n3)cc2)cc1 ZINC000217926598 GI On-Demand Unstable PFKFB3 57 38 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1cccc(CO)c1 ZINC000217926612 CI For-Sale Unstable TRPM8 18 49 O=C(O)/C=C\c1cc(F)ccc1CN1CCC(CO)CC1 ZINC000217926670 CE For-Sale Unstable SIGMAR1 29 42 O=C(O)/C=C\c1cc(F)ccc1CN1CCC(CO)CC1 ZINC000217926670 CE For-Sale Unstable CCR3 37 40 COc1cccc(/C=C/NC(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)c1 ZINC000217926672 IJ For-Sale Unstable OPRD1 15 45 COc1cccc(/C=C/NC(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)c1 ZINC000217926672 IJ For-Sale Unstable MTNR1B 35 41 COc1cccc(/C=C/NC(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)c1 ZINC000217926672 IJ For-Sale Unstable NMUR2 0 44 COc1cccc(/C=C/NC(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)c1 ZINC000217926672 IJ For-Sale Unstable NMUR1 0 44 Cc1cc(NC[C@@H]2CCC[C@@H](C)C2)n2ncnc2n1 ZINC000217926684 CF On-Demand Unstable DHOD 0 52 COc1cccc(-c2noc(CN(C)C(=O)/C=C/c3ccc(OC)c(OC)c3)n2)c1 ZINC000217926694 HG In-Stock Unstable PTPA 0 41 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1cccc(CO)c1 ZINC000217926695 CI For-Sale Unstable TRPM8 18 49 COc1cnc2c(ccn2S(=O)(=O)c2ccccc2)c1Cl ZINC000217926749 DF For-Sale Unstable HTR6 15 43 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1cccc(CO)c1 ZINC000217926768 CI For-Sale Unstable TRPM8 18 49 Cc1cc(NC[C@H]2CCC[C@@H](C)C2)n2ncnc2n1 ZINC000217926771 CF On-Demand Unstable DHOD 0 52 COc1cccc(/C=C/NC(=O)NCC(C)C)c1 ZINC000217926778 BF For-Sale Unstable DRD4 40 30 COc1cccc(/C=C/NC(=O)NCC(C)C)c1 ZINC000217926778 BF For-Sale Unstable CYP1B1 20 41 COc1cccc(/C=C/NC(=O)NCC(C)C)c1 ZINC000217926778 BF For-Sale Unstable MTNR1A 77 50 COc1cccc(/C=C/NC(=O)NCC(C)C)c1 ZINC000217926778 BF For-Sale Unstable MTNR1B 75 50 COc1cccc(/C=C/NC(=O)NCC(C)C)c1 ZINC000217926778 BF For-Sale Unstable CYP1A1 18 41 O=C(O)/C=C\c1cc(CN2CCC(CO)CC2)ccc1F ZINC000217926779 CE For-Sale Unstable ACHE 27 41 O=C(O)/C=C\c1cc(CN2CCC(CO)CC2)ccc1F ZINC000217926779 CE For-Sale Unstable SIGMAR1 41 45 O=C(O)/C=C\c1cc(CN2CCC(CO)CC2)ccc1F ZINC000217926779 CE For-Sale Unstable CCR3 41 40 O=C(O)/C=C\c1cc(CN2CCC(CO)CC2)ccc1F ZINC000217926779 CE For-Sale Unstable MCHR1 25 40 COc1cc2c(cc1OC)[C@@H](c1ccccc1)N(C(=O)Cn1cnc(C#N)n1)CC2 ZINC000217926810 HE On-Demand Unstable HCRTR1 15 40 COc1cc2c(cc1OC)[C@@H](c1ccccc1)N(C(=O)Cn1cnc(C#N)n1)CC2 ZINC000217926810 HE On-Demand Unstable MTNR1B 38 46 COc1ccc(-c2noc(CN(C)C(=O)/C=C/c3ccc(OC)c(OC)c3)n2)c(OC)c1 ZINC000217926815 IG In-Stock Unstable ABCG2 18 41 O=c1nc[nH]c2nc(Cl)cc(Cl)c12 ZINC000217926834 BD For-Sale Anodyne PRIM_HHV11 40 38 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1cccc(CO)c1 ZINC000217926847 CI For-Sale Unstable TRPM8 18 49 Cc1cc(NC[C@@H]2CCC[C@H](C)C2)n2ncnc2n1 ZINC000217926858 CF On-Demand Unstable DHOD 0 52 O=C(O)/C=C\c1cc(F)ccc1CN1CCCCCC1 ZINC000217926862 CG For-Sale Unstable SLC6A1 49 42 C[C@@H](c1ccc(Cl)cc1)N(C)[C@H](C)C(=O)OC(C)(C)C ZINC000217926870 CI For-Sale Unstable UTS2 44 33 COCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217926882 CD For-Sale Unstable DRD4 45 34 COCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217926882 CD For-Sale Unstable CYP1B1 24 41 COCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217926882 CD For-Sale Unstable AHR 19 43 COCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217926882 CD For-Sale Unstable MTNR1A 93 51 COCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217926882 CD For-Sale Unstable MTNR1B 86 51 COCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217926882 CD For-Sale Unstable CYP1A1 18 41 COc1cc2c(cc1OC)[C@H](c1ccccc1)N(C(=O)Cn1cnc(C#N)n1)CC2 ZINC000217926885 HE On-Demand Unstable HCRTR1 15 40 COc1cc2c(cc1OC)[C@H](c1ccccc1)N(C(=O)Cn1cnc(C#N)n1)CC2 ZINC000217926885 HE On-Demand Unstable MTNR1B 38 46 CC[C@@H](CCO)NC(=O)[C@@H](C)CN ZINC000217926924 AB For-Sale Unstable SLC15A2 41 37 Cc1cc(NC[C@H]2CCC[C@H](C)C2)n2ncnc2n1 ZINC000217926930 CF On-Demand Unstable DHOD 0 52 O=C(O)/C=C\c1cc(CN2CCCCCC2)ccc1F ZINC000217926957 CG For-Sale Unstable HRH3 19 41 O=C(O)/C=C\c1cc(CN2CCCCCC2)ccc1F ZINC000217926957 CG For-Sale Unstable SIGMAR1 19 41 O=C(O)/C=C\c1cc(CN2CCCCCC2)ccc1F ZINC000217926957 CG For-Sale Unstable CCR1 0 42 O=C(CN1CC[C@H]2CCCC[C@@H]2C1)N1CCNCC1 ZINC000217926979 CC For-Sale Unstable GNAI1 0 43 O=C(CN1CC[C@H]2CCCC[C@@H]2C1)N1CCNCC1 ZINC000217926979 CC For-Sale Unstable GNAI3 0 43 O=C(CN1CC[C@H]2CCCC[C@@H]2C1)N1CCNCC1 ZINC000217926979 CC For-Sale Unstable GNAO1 0 43 CCCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217926993 BF For-Sale Unstable DRD4 42 32 CCCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217926993 BF For-Sale Unstable HRH2 23 43 CCCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217926993 BF For-Sale Unstable AHR 20 42 CCCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217926993 BF For-Sale Unstable MTNR1A 103 51 CCCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217926993 BF For-Sale Unstable MTNR1B 95 51 CCCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217926993 BF For-Sale Unstable FAAH 15 43 CCCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217926993 BF For-Sale Unstable ACAT 0 44 CC[C@H](CCO)NC(=O)[C@@H](C)CN ZINC000217927012 AB For-Sale Unstable SLC15A2 41 37 COc1ccc(/C=C/C(=O)NCCCc2ccc(C(C)C)cc2)cc1OC ZINC000217927045 FJ In-Stock Unstable DRD3 16 46 COc1ccc(/C=C/C(=O)NCCCc2ccc(C(C)C)cc2)cc1OC ZINC000217927045 FJ In-Stock Unstable TRPV1 0 51 COc1ccc(/C=C/C(=O)NCCCc2ccc(C(C)C)cc2)cc1OC ZINC000217927045 FJ In-Stock Unstable PYGL 0 46 COc1ccc(/C=C/C(=O)NCCCc2ccc(C(C)C)cc2)cc1OC ZINC000217927045 FJ In-Stock Unstable ABCG2 16 42 COc1cc(N2CCN(C(=O)OC(C)(C)C)CC2)ccc1Nc1nc(Cl)nc(N)c1C(N)=O ZINC000217927052 JF For-Sale Unstable INSR 20 42 COc1cc(N2CCN(C(=O)OC(C)(C)C)CC2)ccc1Nc1nc(Cl)nc(N)c1C(N)=O ZINC000217927052 JF For-Sale Unstable IGF1R 74 43 COc1cc(N2CCN(C(=O)OC(C)(C)C)CC2)ccc1Nc1nc(Cl)nc(N)c1C(N)=O ZINC000217927052 JF For-Sale Unstable PTK2 21 40 COc1cc(N2CCN(C(=O)OC(C)(C)C)CC2)ccc1Nc1nc(Cl)nc(N)c1C(N)=O ZINC000217927052 JF For-Sale Unstable MAPK10 23 44 COc1cc(N2CCN(C(=O)OC(C)(C)C)CC2)ccc1Nc1nc(Cl)nc(N)c1C(N)=O ZINC000217927052 JF For-Sale Unstable ZAP70 22 41 COc1cc(N2CCN(C(=O)OC(C)(C)C)CC2)ccc1Nc1nc(Cl)nc(N)c1C(N)=O ZINC000217927052 JF For-Sale Unstable TTK 40 38 COc1cc(N2CCN(C(=O)OC(C)(C)C)CC2)ccc1Nc1nc(Cl)nc(N)c1C(N)=O ZINC000217927052 JF For-Sale Unstable ALK 26 42 COc1cc(N2CCN(C(=O)OC(C)(C)C)CC2)ccc1Nc1nc(Cl)nc(N)c1C(N)=O ZINC000217927052 JF For-Sale Unstable GPR119 21 41 CSCC[C@H](NC(=O)c1ccc2c(ccn2Cc2ccccc2)c1)C(=O)O ZINC000217927074 GH In-Stock Unstable DHFR 43 36 CSCC[C@H](NC(=O)c1ccc2c(ccn2Cc2ccccc2)c1)C(=O)O ZINC000217927074 GH In-Stock Unstable TYMS 52 36 CSCC[C@H](NC(=O)c1ccc2c(ccn2Cc2ccccc2)c1)C(=O)O ZINC000217927074 GH In-Stock Unstable ACE 24 45 CSCC[C@H](NC(=O)c1ccc2c(ccn2Cc2ccccc2)c1)C(=O)O ZINC000217927074 GH In-Stock Unstable MME 23 45 CSCC[C@H](NC(=O)c1ccc2c(ccn2Cc2ccccc2)c1)C(=O)O ZINC000217927074 GH In-Stock Unstable CCKAR 35 48 CSCC[C@H](NC(=O)c1ccc2c(ccn2Cc2ccccc2)c1)C(=O)O ZINC000217927074 GH In-Stock Unstable CCKBR 59 41 CSCC[C@H](NC(=O)c1ccc2c(ccn2Cc2ccccc2)c1)C(=O)O ZINC000217927074 GH In-Stock Unstable GART 52 37 CSCC[C@H](NC(=O)c1ccc2c(ccn2Cc2ccccc2)c1)C(=O)O ZINC000217927074 GH In-Stock Unstable FPR1 40 39 CSCC[C@H](NC(=O)c1ccc2c(ccn2Cc2ccccc2)c1)C(=O)O ZINC000217927074 GH In-Stock Unstable BLA1_STEMA 43 35 N#Cc1ncn(CC(=O)N2CCN(c3ccc(C(F)(F)F)cc3[N+](=O)[O-])CC2)n1 ZINC000217927079 HD On-Demand Unstable SLC6A9 15 47 N#Cc1ncn(CC(=O)N2CCN(c3ccc(C(F)(F)F)cc3[N+](=O)[O-])CC2)n1 ZINC000217927079 HD On-Demand Unstable LIPG 40 33 CCOCCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217927088 CE For-Sale Unstable HRH2 26 41 CCOCCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217927088 CE For-Sale Unstable MTNR1A 80 47 CCOCCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217927088 CE For-Sale Unstable MTNR1B 75 47 CCCC(CCC)C(=O)N1[C@H](C(=O)O)C[C@@H]2CCCC[C@@H]21 ZINC000217927099 CG For-Sale Unstable ACE 36 67 CC[C@@H](CCO)NC(=O)[C@H](C)CN ZINC000217927102 AB For-Sale Unstable SLC15A2 41 37 COc1ccc(/C=C/C(=O)NCCCN2CCCc3ccccc32)cc1OC ZINC000217927159 GH In-Stock Unstable DRD2 30 53 COc1ccc(/C=C/C(=O)NCCCN2CCCc3ccccc32)cc1OC ZINC000217927159 GH In-Stock Unstable DRD1 0 51 COc1ccc(/C=C/C(=O)NCCCN2CCCc3ccccc32)cc1OC ZINC000217927159 GH In-Stock Unstable HTR2A 15 51 COc1ccc(/C=C/C(=O)NCCCN2CCCc3ccccc32)cc1OC ZINC000217927159 GH In-Stock Unstable DRD3 49 53 COc1ccc(/C=C/C(=O)NCCCN2CCCc3ccccc32)cc1OC ZINC000217927159 GH In-Stock Unstable BCHE 20 44 COc1ccc(/C=C/C(=O)NCCCN2CCCc3ccccc32)cc1OC ZINC000217927159 GH In-Stock Unstable ACKR3 40 33 CCCC(CCC)C(=O)N1[C@H](C(=O)O)C[C@H]2CCCC[C@@H]21 ZINC000217927179 CG For-Sale Unstable ACE 36 67 O=C(N[C@H]1CCC[C@H]1CO)c1cc(C(F)(F)F)ccc1F ZINC000217927182 DF On-Demand Unstable CCR2 33 41 O=C(N[C@H]1CCC[C@H]1CO)c1cc(C(F)(F)F)ccc1F ZINC000217927182 DF On-Demand Unstable LIPG 47 39 CN1CCN(C(=O)C[C@H](c2cccnc2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)CC1 ZINC000217927188 KG In-Stock Unstable PTAFR 26 42 CC[C@H](CCO)NC(=O)[C@H](C)CN ZINC000217927192 AB For-Sale Unstable SLC15A2 41 37 CC[C@@H](C)NC(=O)N/C=C/c1cccc(OC)c1 ZINC000217927204 BF For-Sale Unstable AHR 18 41 CC[C@@H](C)NC(=O)N/C=C/c1cccc(OC)c1 ZINC000217927204 BF For-Sale Unstable MTNR1A 44 47 CC[C@@H](C)NC(=O)N/C=C/c1cccc(OC)c1 ZINC000217927204 BF For-Sale Unstable MTNR1B 47 47 NC(=O)CCCCCn1c(SCc2ccc3ccccc3n2)nc2ccccc2c1=O ZINC000217927226 II On-Demand Unstable HTR3A 15 41 CCCCN(CC)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217927240 CG For-Sale Unstable THRA 0 41 CCCCN(CC)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217927240 CG For-Sale Unstable LTB4R 22 40 CCCCN(CC)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217927240 CG For-Sale Unstable PLA2G4B 59 40 CCCCN(CC)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217927240 CG For-Sale Unstable SQLE 40 31 CCCCN(CC)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217927240 CG For-Sale Unstable AKR1C3 26 42 CN1CCN(C(=O)C[C@@H](c2cccnc2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)CC1 ZINC000217927257 KG In-Stock Unstable PTAFR 26 42 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CNC(=O)c1cccc(OC)c1 ZINC000217927265 ID For-Sale Unstable DRD4 53 41 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CNC(=O)c1cccc(OC)c1 ZINC000217927265 ID For-Sale Unstable DRD3 19 45 N#CCNC(=O)c1ccc(B(O)O)cc1 ZINC000217927274 BA In-Stock Unstable PAPA1_CARPA 26 42 N#CCNC(=O)c1ccc(B(O)O)cc1 ZINC000217927274 BA In-Stock Unstable CTSL 21 42 N#CCNC(=O)c1ccc(B(O)O)cc1 ZINC000217927274 BA In-Stock Unstable CTSS 19 42 CN(C)S(=O)(=O)c1ccc2c(c1)CCN2C(=O)/C=C/c1ccc2c(c1)OCO2 ZINC000217927280 HE In-Stock Unstable DYRK2 40 31 CC[C@H](C)NC(=O)N/C=C/c1cccc(OC)c1 ZINC000217927290 BF For-Sale Unstable AHR 18 41 CC[C@H](C)NC(=O)N/C=C/c1cccc(OC)c1 ZINC000217927290 BF For-Sale Unstable MTNR1A 44 47 CC[C@H](C)NC(=O)N/C=C/c1cccc(OC)c1 ZINC000217927290 BF For-Sale Unstable MTNR1B 47 47 CCCCN(CC)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217927342 CG On-Demand Unstable THRA 27 46 CCCCN(CC)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217927342 CG On-Demand Unstable ACHE 0 60 CCCCN(CC)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217927342 CG On-Demand Unstable ERG2 18 44 CCCCN(CC)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217927342 CG On-Demand Unstable KCNQ1 0 44 CCCCN(CC)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217927342 CG On-Demand Unstable PLA2G4B 85 38 CCCCN(CC)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217927342 CG On-Demand Unstable FAAH 22 40 CCCCN(CC)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217927342 CG On-Demand Unstable AKR1C3 0 43 CCCCN(CC)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217927342 CG On-Demand Unstable NORA 0 46 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CNC(=O)c1cccc(OC)c1 ZINC000217927343 ID For-Sale Unstable DRD4 53 41 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CNC(=O)c1cccc(OC)c1 ZINC000217927343 ID For-Sale Unstable DRD3 19 45 O=S(=O)(NCC[C@H](O)C1CCOCC1)c1ccc(-n2cccn2)cc1 ZINC000217927353 FD In-Stock Unstable AMP1_PLAFQ 40 31 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc(OC(C)C)c2)CC(=O)O4)cc1O ZINC000217927364 JK In-Stock Unstable AKR1B1 0 43 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc(OC(C)C)c2)CC(=O)O4)cc1O ZINC000217927364 JK In-Stock Unstable CYP1B1 47 35 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@@H](c2cccc(OC(C)C)c2)CC(=O)O4)cc1O ZINC000217927364 JK In-Stock Unstable CYP1A1 37 43 C[C@@H]1CCC[C@@H](CNc2ccc(C(N)=O)cn2)C1 ZINC000217927377 BE On-Demand Unstable GCK 15 40 CCN(C)C(=O)CNC(=O)[C@@H](C#N)Cc1ccccc1 ZINC000217927389 CC For-Sale Unstable MME 81 42 CCN(C)C(=O)CNC(=O)[C@@H](C#N)Cc1ccccc1 ZINC000217927389 CC For-Sale Unstable ANPEP 39 42 CCN(C)C(=O)CNC(=O)[C@@H](C#N)Cc1ccccc1 ZINC000217927389 CC For-Sale Unstable CTSB 42 41 CCN(C)C(=O)CNC(=O)[C@@H](C#N)Cc1ccccc1 ZINC000217927389 CC For-Sale Unstable PAPA1_CARPA 51 42 CCN(C)C(=O)CNC(=O)[C@@H](C#N)Cc1ccccc1 ZINC000217927389 CC For-Sale Unstable CTSF 43 32 CCN(C)C(=O)CNC(=O)[C@@H](C#N)Cc1ccccc1 ZINC000217927389 CC For-Sale Unstable CTSK 17 41 CCN(C)C(=O)CNC(=O)[C@@H](C#N)Cc1ccccc1 ZINC000217927389 CC For-Sale Unstable CTSL 32 42 CCN(C)C(=O)CNC(=O)[C@@H](C#N)Cc1ccccc1 ZINC000217927389 CC For-Sale Unstable CTSS 21 42 CCN(C)C(=O)CNC(=O)[C@@H](C#N)Cc1ccccc1 ZINC000217927389 CC For-Sale Unstable CTSC 40 43 CCN(C)C(=O)CNC(=O)[C@@H](C#N)Cc1ccccc1 ZINC000217927389 CC For-Sale Unstable AMP1_PLAFQ 45 38 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccc3c(c2)OCO3)c1 ZINC000217927391 EH In-Stock Unstable EDNRB 33 41 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccc3c(c2)OCO3)c1 ZINC000217927391 EH In-Stock Unstable EDNRA 35 41 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccc3c(c2)OCO3)c1 ZINC000217927391 EH In-Stock Unstable DYRK2 50 36 COc1cccc(/C=C/NC(=O)N2CCCc3ccccc32)c1 ZINC000217927397 DH For-Sale Unstable DRD4 43 35 COc1cccc(/C=C/NC(=O)N2CCCc3ccccc32)c1 ZINC000217927397 DH For-Sale Unstable AVPR2 40 54 CCN(Cc1ccc(/C=C\C(=O)O)cc1)c1ccccc1 ZINC000217927416 CH For-Sale Unstable NR1H4 41 43 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CNC(=O)c1cccc(OC)c1 ZINC000217927417 ID For-Sale Unstable DRD4 53 41 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CNC(=O)c1cccc(OC)c1 ZINC000217927417 ID For-Sale Unstable DRD3 19 45 O=S(=O)(NCC[C@@H](O)C1CCOCC1)c1ccc(-n2cccn2)cc1 ZINC000217927420 FD In-Stock Unstable AMP1_PLAFQ 40 31 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc(OC(C)C)c2)CC(=O)O4)cc1O ZINC000217927436 JK In-Stock Unstable AKR1B1 0 43 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc(OC(C)C)c2)CC(=O)O4)cc1O ZINC000217927436 JK In-Stock Unstable CYP1B1 47 35 COc1ccc(-c2cc(=O)c3c(O)cc4c(c3o2)[C@H](c2cccc(OC(C)C)c2)CC(=O)O4)cc1O ZINC000217927436 JK In-Stock Unstable CYP1A1 37 43 C[C@H]1CCC[C@@H](CNc2ccc(C(N)=O)cn2)C1 ZINC000217927460 BE On-Demand Unstable GCK 15 40 CCN(C)C(=O)CNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000217927471 CC For-Sale Unstable MME 81 42 CCN(C)C(=O)CNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000217927471 CC For-Sale Unstable ANPEP 39 42 CCN(C)C(=O)CNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000217927471 CC For-Sale Unstable CTSB 42 41 CCN(C)C(=O)CNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000217927471 CC For-Sale Unstable PAPA1_CARPA 51 42 CCN(C)C(=O)CNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000217927471 CC For-Sale Unstable CTSF 43 32 CCN(C)C(=O)CNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000217927471 CC For-Sale Unstable CTSK 17 41 CCN(C)C(=O)CNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000217927471 CC For-Sale Unstable CTSL 32 42 CCN(C)C(=O)CNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000217927471 CC For-Sale Unstable CTSS 21 42 CCN(C)C(=O)CNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000217927471 CC For-Sale Unstable CTSC 40 43 CCN(C)C(=O)CNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000217927471 CC For-Sale Unstable AMP1_PLAFQ 45 38 COc1cccc(/C=C/NC(=O)NCCc2ccccc2)c1 ZINC000217927501 CG For-Sale Unstable DRD4 41 32 COc1cccc(/C=C/NC(=O)NCCc2ccccc2)c1 ZINC000217927501 CG For-Sale Unstable NQO2 30 41 COc1cccc(/C=C/NC(=O)NCCc2ccccc2)c1 ZINC000217927501 CG For-Sale Unstable G6PC 24 43 COc1cccc(/C=C/NC(=O)NCCc2ccccc2)c1 ZINC000217927501 CG For-Sale Unstable HDAC8 19 40 COc1cccc(/C=C/NC(=O)NCCc2ccccc2)c1 ZINC000217927501 CG For-Sale Unstable MTNR1A 130 52 COc1cccc(/C=C/NC(=O)NCCc2ccccc2)c1 ZINC000217927501 CG For-Sale Unstable MTNR1B 119 52 COc1cccc(/C=C/NC(=O)NCCc2ccccc2)c1 ZINC000217927501 CG For-Sale Unstable MMP2 15 52 COc1cccc(/C=C/NC(=O)NCCc2ccccc2)c1 ZINC000217927501 CG For-Sale Unstable HDAC6 15 40 COc1cccc(/C=C/NC(=O)NCCc2ccccc2)c1 ZINC000217927501 CG For-Sale Unstable FAAH 17 45 COc1cccc(/C=C/NC(=O)NCCc2ccccc2)c1 ZINC000217927501 CG For-Sale Unstable AKR1C3 30 42 COc1cccc(/C=C/NC(=O)NCCc2ccccc2)c1 ZINC000217927501 CG For-Sale Unstable CRTM 58 38 COc1cccc(/C=C/NC(=O)NCCc2ccccc2)c1 ZINC000217927501 CG For-Sale Unstable PDS 49 37 CCN(Cc1cccc(/C=C\C(=O)O)c1)c1ccccc1 ZINC000217927504 CH For-Sale Unstable PTGER2 27 43 CCN(Cc1cccc(/C=C\C(=O)O)c1)c1ccccc1 ZINC000217927504 CH For-Sale Unstable NR1H4 50 39 CCN(Cc1cccc(/C=C\C(=O)O)c1)c1ccccc1 ZINC000217927504 CH For-Sale Unstable AKR1C3 32 45 COc1ccc(CNC(=O)/C=C/c2ccc3c(c2)OCO3)c(OC)c1OC ZINC000217927505 FF In-Stock Unstable EDNRB 37 46 COc1ccc(CNC(=O)/C=C/c2ccc3c(c2)OCO3)c(OC)c1OC ZINC000217927505 FF In-Stock Unstable F3 19 41 COc1ccc(CNC(=O)/C=C/c2ccc3c(c2)OCO3)c(OC)c1OC ZINC000217927505 FF In-Stock Unstable TUBB1 47 42 COc1ccc(CNC(=O)/C=C/c2ccc3c(c2)OCO3)c(OC)c1OC ZINC000217927505 FF In-Stock Unstable DYRK2 52 34 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CNC(=O)c1cccc(OC)c1 ZINC000217927506 ID For-Sale Unstable DRD4 53 41 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CNC(=O)c1cccc(OC)c1 ZINC000217927506 ID For-Sale Unstable DRD3 19 45 C[C@@H]1CCC[C@H](CNc2ccc(C(N)=O)cn2)C1 ZINC000217927538 BE On-Demand Unstable GCK 15 40 CS(=O)(=O)C1(C#N)CCN(Cc2ccccc2)CC1 ZINC000217927560 CD In-Stock Unstable DRD2 0 43 CS(=O)(=O)C1(C#N)CCN(Cc2ccccc2)CC1 ZINC000217927560 CD In-Stock Unstable DRD3 0 43 CS(=O)(=O)C1(C#N)CCN(Cc2ccccc2)CC1 ZINC000217927560 CD In-Stock Unstable ADAM17 0 41 CS(=O)(=O)C1(C#N)CCN(Cc2ccccc2)CC1 ZINC000217927560 CD In-Stock Unstable NPFFR1 58 39 COc1cccc(/C=C/NC(=O)NC2CCCC2)c1 ZINC000217927601 CF For-Sale Unstable MTNR1A 41 41 COc1cccc(/C=C/NC(=O)NC2CCCC2)c1 ZINC000217927601 CF For-Sale Unstable MTNR1B 43 41 COc1cccc(/C=C/NC(=O)NC2CCCC2)c1 ZINC000217927601 CF For-Sale Unstable FAAH 25 44 COc1cccc(/C=C/NC(=O)NC2CCCC2)c1 ZINC000217927601 CF For-Sale Unstable EPHX2 22 48 O=C(N[C@@H]1CCC[C@@H]1CO)c1cccc(Cl)n1 ZINC000217927616 CD For-Sale Unstable SSTR3 29 40 CCOc1ccc(CNC(=O)/C=C/c2ccc3c(c2)OCO3)cc1OCC ZINC000217927617 FH In-Stock Unstable NOS2 57 33 CCOc1ccc(CNC(=O)/C=C/c2ccc3c(c2)OCO3)cc1OCC ZINC000217927617 FH In-Stock Unstable DYRK2 49 35 C[C@H]1CCC[C@H](CNc2ccc(C(N)=O)cn2)C1 ZINC000217927620 BE On-Demand Unstable GCK 15 40 O=C(O)/C=C\c1cccc(OCCN2CCC(O)CC2)c1 ZINC000217927624 CD For-Sale Unstable HRH2 28 42 O=C(O)/C=C\c1cccc(OCCN2CCC(O)CC2)c1 ZINC000217927624 CD For-Sale Unstable HRH1 19 42 O=C(O)/C=C\c1cccc(OCCN2CCC(O)CC2)c1 ZINC000217927624 CD For-Sale Unstable ESR2 22 42 O=C(O)/C=C\c1cccc(OCCN2CCC(O)CC2)c1 ZINC000217927624 CD For-Sale Unstable LTA4H 41 44 O=C(O)/C=C\c1cccc(OCCN2CCC(O)CC2)c1 ZINC000217927624 CD For-Sale Unstable HRH3 24 43 O=C(O)/C=C\c1cccc(OCCN2CCC(O)CC2)c1 ZINC000217927624 CD For-Sale Unstable SIGMAR1 20 45 O=C(O)/C=C\c1cccc(OCCN2CCC(O)CC2)c1 ZINC000217927624 CD For-Sale Unstable PSMB2 46 39 O=C(O)/C=C\c1cccc(OCCN2CCC(O)CC2)c1 ZINC000217927624 CD For-Sale Unstable PSMB1 40 39 C[C@H]1CN(C)[C@@H](C)C[C@@H]1NCCc1c[nH]c2ccccc12 ZINC000217927628 CG For-Sale Unstable HTR1A 0 47 C[C@H]1CN(C)[C@@H](C)C[C@@H]1NCCc1c[nH]c2ccccc12 ZINC000217927628 CG For-Sale Unstable HTR1D 26 41 C[C@H]1CN(C)[C@@H](C)C[C@@H]1NCCc1c[nH]c2ccccc12 ZINC000217927628 CG For-Sale Unstable HTR1B 20 41 C[C@H]1CN(C)[C@@H](C)C[C@@H]1NCCc1c[nH]c2ccccc12 ZINC000217927628 CG For-Sale Unstable MC4R 24 40 C[C@H]1CN(C)[C@@H](C)C[C@@H]1NCCc1c[nH]c2ccccc12 ZINC000217927628 CG For-Sale Unstable MPO 29 41 CCS(=O)(=O)C1(C#N)CCN(Cc2ccccc2)CC1 ZINC000217927675 CD In-Stock Unstable DRD2 0 43 CCS(=O)(=O)C1(C#N)CCN(Cc2ccccc2)CC1 ZINC000217927675 CD In-Stock Unstable DRD3 0 43 CCS(=O)(=O)C1(C#N)CCN(Cc2ccccc2)CC1 ZINC000217927675 CD In-Stock Unstable NPFFR1 56 40 O=C(N[C@H]1CCC[C@@H]1CO)c1cccc(Cl)n1 ZINC000217927692 CD For-Sale Unstable SSTR3 29 40 COc1cccc(/C=C/NC(=O)NCc2ccccc2Cl)c1 ZINC000217927709 DH For-Sale Unstable DRD4 44 37 COc1cccc(/C=C/NC(=O)NCc2ccccc2Cl)c1 ZINC000217927709 DH For-Sale Unstable PTGER3 28 45 COc1cccc(/C=C/NC(=O)NCc2ccccc2Cl)c1 ZINC000217927709 DH For-Sale Unstable P2RX7 34 40 COc1cccc(/C=C/NC(=O)NCc2ccccc2Cl)c1 ZINC000217927709 DH For-Sale Unstable MTNR1A 58 41 COc1cccc(/C=C/NC(=O)NCc2ccccc2Cl)c1 ZINC000217927709 DH For-Sale Unstable MTNR1B 54 41 O=C(O)/C=C\c1ccccc1CN1CCS(=O)(=O)CC1 ZINC000217927725 CD For-Sale Unstable PTGER2 39 48 O=C(O)/C=C\c1ccccc1CN1CCS(=O)(=O)CC1 ZINC000217927725 CD For-Sale Unstable PTGER4 17 40 O=C(O)/C=C\c1ccccc1CN1CCS(=O)(=O)CC1 ZINC000217927725 CD For-Sale Unstable PTGER3 20 48 COc1cc(CNC(=O)/C=C/c2ccc3c(c2)OCO3)ccc1OC(C)C ZINC000217927726 FH In-Stock Unstable EDNRB 42 42 COc1cc(CNC(=O)/C=C/c2ccc3c(c2)OCO3)ccc1OC(C)C ZINC000217927726 FH In-Stock Unstable EDNRA 49 38 COc1cc(CNC(=O)/C=C/c2ccc3c(c2)OCO3)ccc1OC(C)C ZINC000217927726 FH In-Stock Unstable TRPV1 16 42 COc1cc(CNC(=O)/C=C/c2ccc3c(c2)OCO3)ccc1OC(C)C ZINC000217927726 FH In-Stock Unstable DYRK2 42 33 C[C@@H]1CCC[C@@H](CNc2ccc(C#N)cn2)C1 ZINC000217927727 BG On-Demand Unstable PK7 0 42 O=CC[C@H](CSc1ccccc1)NC(=O)OCc1ccccc1 ZINC000217927736 EH For-Sale Unstable CELA1 18 41 O=CC[C@H](CSc1ccccc1)NC(=O)OCc1ccccc1 ZINC000217927736 EH For-Sale Unstable BMP1 54 35 O=CC[C@H](CSc1ccccc1)NC(=O)OCc1ccccc1 ZINC000217927736 EH For-Sale Unstable KLK3 82 41 O=CC[C@H](CSc1ccccc1)NC(=O)OCc1ccccc1 ZINC000217927736 EH For-Sale Unstable CTSB 66 44 O=CC[C@H](CSc1ccccc1)NC(=O)OCc1ccccc1 ZINC000217927736 EH For-Sale Unstable PAPA1_CARPA 58 39 O=CC[C@H](CSc1ccccc1)NC(=O)OCc1ccccc1 ZINC000217927736 EH For-Sale Unstable CYSP_TRYCR 59 42 O=CC[C@H](CSc1ccccc1)NC(=O)OCc1ccccc1 ZINC000217927736 EH For-Sale Unstable CTSK 43 47 O=CC[C@H](CSc1ccccc1)NC(=O)OCc1ccccc1 ZINC000217927736 EH For-Sale Unstable CTSL 49 46 O=CC[C@H](CSc1ccccc1)NC(=O)OCc1ccccc1 ZINC000217927736 EH For-Sale Unstable CAPNS1 65 37 O=CC[C@H](CSc1ccccc1)NC(=O)OCc1ccccc1 ZINC000217927736 EH For-Sale Unstable MMP11 43 30 O=CC[C@H](CSc1ccccc1)NC(=O)OCc1ccccc1 ZINC000217927736 EH For-Sale Unstable CTSS 23 43 O=CC[C@H](CSc1ccccc1)NC(=O)OCc1ccccc1 ZINC000217927736 EH For-Sale Unstable CAPN1 93 47 O=CC[C@H](CSc1ccccc1)NC(=O)OCc1ccccc1 ZINC000217927736 EH For-Sale Unstable CASP1 23 43 O=CC[C@H](CSc1ccccc1)NC(=O)OCc1ccccc1 ZINC000217927736 EH For-Sale Unstable CAPN2 131 44 O=CC[C@H](CSc1ccccc1)NC(=O)OCc1ccccc1 ZINC000217927736 EH For-Sale Unstable NPR 67 34 O=CC[C@H](CSc1ccccc1)NC(=O)OCc1ccccc1 ZINC000217927736 EH For-Sale Unstable PSMB5 35 40 COc1ccc(OC)c(N(C)[C@@H](C)C(=O)O)c1 ZINC000217927757 BD In-Stock Unstable AKR1C3 20 44 COc1ccc(OC)c(N(C)[C@@H](C)C(=O)O)c1 ZINC000217927757 BD In-Stock Unstable AKR1C2 41 33 CC(C)[C@@H](CO)NC(=O)C[C@@H]1NC(=O)N(Cc2ccccc2)C1=O ZINC000217927766 EC In-Stock Unstable GALR1 46 33 O=C(N[C@@H]1CCC[C@H]1CO)c1cccc(Cl)n1 ZINC000217927768 CD For-Sale Unstable SSTR3 29 40 CS(=O)(=O)C1(CN)CCN(Cc2ccccc2)CC1 ZINC000217927777 CD In-Stock Unstable DRD3 17 42 CS(=O)(=O)C1(CN)CCN(Cc2ccccc2)CC1 ZINC000217927777 CD In-Stock Unstable OPRL1 15 47 CS(=O)(=O)C1(CN)CCN(Cc2ccccc2)CC1 ZINC000217927777 CD In-Stock Unstable SIGMAR1 78 49 CS(=O)(=O)C1(CN)CCN(Cc2ccccc2)CC1 ZINC000217927777 CD In-Stock Unstable ADAM17 16 42 CS(=O)(=O)C1(CN)CCN(Cc2ccccc2)CC1 ZINC000217927777 CD In-Stock Unstable EBP 17 42 CS(=O)(=O)C1(CN)CCN(Cc2ccccc2)CC1 ZINC000217927777 CD In-Stock Unstable NPFFR1 57 39 CS(=O)(=O)C1(CN)CCN(Cc2ccccc2)CC1 ZINC000217927777 CD In-Stock Unstable EBPL 0 42 C[C@H]1CCC[C@@H](CNc2ccc(C#N)cn2)C1 ZINC000217927807 BG On-Demand Unstable PK7 0 42 COc1cccc(/C=C/NC(=O)NCCc2ccc(OC)c(OC)c2)c1 ZINC000217927818 FG For-Sale Unstable CYP1B1 28 41 COc1cccc(/C=C/NC(=O)NCCc2ccc(OC)c(OC)c2)c1 ZINC000217927818 FG For-Sale Unstable MTNR1A 100 48 COc1cccc(/C=C/NC(=O)NCCc2ccc(OC)c(OC)c2)c1 ZINC000217927818 FG For-Sale Unstable MTNR1B 96 53 COc1cccc(/C=C/NC(=O)NCCc2ccc(OC)c(OC)c2)c1 ZINC000217927818 FG For-Sale Unstable CYP1A1 27 41 COc1cccc(/C=C/NC(=O)NCCc2ccc(OC)c(OC)c2)c1 ZINC000217927818 FG For-Sale Unstable ABCG2 27 43 O=C(O)/C=C\c1ccc(CN2CCS(=O)(=O)CC2)cc1 ZINC000217927830 CD For-Sale Unstable SIGMAR1 19 44 O=C(/C=C/c1ccc2c(c1)OCO2)NCCCc1ccccc1Cl ZINC000217927839 EH In-Stock Unstable DRD3 18 54 O=C(/C=C/c1ccc2c(c1)OCO2)NCCCc1ccccc1Cl ZINC000217927839 EH In-Stock Unstable PYGL 28 52 O=C(/C=C/c1ccc2c(c1)OCO2)NCCCc1ccccc1Cl ZINC000217927839 EH In-Stock Unstable DYRK2 46 33 O=C(N[C@H]1CCC[C@H]1CO)c1cccc(Cl)n1 ZINC000217927854 CD On-Demand Unstable SSTR3 29 40 C[C@H]1Cc2ccccc2N1[C@H](C)C(=O)OC(C)(C)C ZINC000217927857 CG For-Sale Unstable TPP2 57 36 CC(C)[C@@H](CO)NC(=O)CC[C@@H]1NC(=O)N(Cc2ccc3c(c2)OCO3)C1=O ZINC000217927873 GC In-Stock Unstable SSTR3 97 33 CC(C)[C@@H](CO)NC(=O)CC[C@@H]1NC(=O)N(Cc2ccc3c(c2)OCO3)C1=O ZINC000217927873 GC In-Stock Unstable MCHR1 18 40 C[C@@H]1CCC[C@H](CNc2ccc(C#N)cn2)C1 ZINC000217927888 BG On-Demand Unstable PK7 0 42 CCS(=O)(=O)C1(CN)CCN(Cc2ccccc2)CC1 ZINC000217927889 CD In-Stock Unstable DRD3 16 41 CCS(=O)(=O)C1(CN)CCN(Cc2ccccc2)CC1 ZINC000217927889 CD In-Stock Unstable OPRL1 15 46 CCS(=O)(=O)C1(CN)CCN(Cc2ccccc2)CC1 ZINC000217927889 CD In-Stock Unstable SIGMAR1 78 47 CCS(=O)(=O)C1(CN)CCN(Cc2ccccc2)CC1 ZINC000217927889 CD In-Stock Unstable NPFFR2 33 40 CCS(=O)(=O)C1(CN)CCN(Cc2ccccc2)CC1 ZINC000217927889 CD In-Stock Unstable ADAM17 18 41 CCS(=O)(=O)C1(CN)CCN(Cc2ccccc2)CC1 ZINC000217927889 CD In-Stock Unstable EBP 17 41 CCS(=O)(=O)C1(CN)CCN(Cc2ccccc2)CC1 ZINC000217927889 CD In-Stock Unstable MCHR2 40 33 CCS(=O)(=O)C1(CN)CCN(Cc2ccccc2)CC1 ZINC000217927889 CD In-Stock Unstable NPFFR1 57 41 COCCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217927926 CE For-Sale Unstable DRD4 44 33 COCCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217927926 CE For-Sale Unstable HRH2 26 43 COCCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217927926 CE For-Sale Unstable MTNR1A 87 50 COCCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217927926 CE For-Sale Unstable MTNR1B 81 50 O=C(O)/C=C\c1ccc(CN2CCS(=O)(=O)CC2)c(F)c1 ZINC000217927940 DD For-Sale Unstable GPR183 0 40 O=C(/C=C/c1ccc2c(c1)OCO2)NCCCc1ccc(Cl)cc1 ZINC000217927941 EH In-Stock Unstable PYGL 27 50 O=C(/C=C/c1ccc2c(c1)OCO2)NCCCc1ccc(Cl)cc1 ZINC000217927941 EH In-Stock Unstable DYRK2 46 34 C[C@H]1CN(C)[C@@H](C)C[C@@H]1NCCCc1ccccc1 ZINC000217927946 CF For-Sale Unstable SIGMAR1 25 49 C[C@H]1CCC[C@H](CNc2ccc(C#N)cn2)C1 ZINC000217927976 BG On-Demand Unstable PK7 0 42 CCOC(=O)C1(S(C)(=O)=O)CCN(Cc2ccccc2)CC1 ZINC000217927981 ED In-Stock Unstable CHRM2 18 42 CCOC(=O)C1(S(C)(=O)=O)CCN(Cc2ccccc2)CC1 ZINC000217927981 ED In-Stock Unstable DRD4 36 40 CCOC(=O)C1(S(C)(=O)=O)CCN(Cc2ccccc2)CC1 ZINC000217927981 ED In-Stock Unstable DRD3 25 42 CCOC(=O)C1(S(C)(=O)=O)CCN(Cc2ccccc2)CC1 ZINC000217927981 ED In-Stock Unstable OPRK1 15 40 CCOC(=O)C1(S(C)(=O)=O)CCN(Cc2ccccc2)CC1 ZINC000217927981 ED In-Stock Unstable OPRL1 17 42 CCOC(=O)C1(S(C)(=O)=O)CCN(Cc2ccccc2)CC1 ZINC000217927981 ED In-Stock Unstable SIGMAR1 74 53 CCOC(=O)C1(S(C)(=O)=O)CCN(Cc2ccccc2)CC1 ZINC000217927981 ED In-Stock Unstable MMP13 18 50 CCOC(=O)C1(S(C)(=O)=O)CCN(Cc2ccccc2)CC1 ZINC000217927981 ED In-Stock Unstable NPFFR2 42 41 CCOC(=O)C1(S(C)(=O)=O)CCN(Cc2ccccc2)CC1 ZINC000217927981 ED In-Stock Unstable ADAM17 28 50 CCOC(=O)C1(S(C)(=O)=O)CCN(Cc2ccccc2)CC1 ZINC000217927981 ED In-Stock Unstable MMP14 17 46 CCOC(=O)C1(S(C)(=O)=O)CCN(Cc2ccccc2)CC1 ZINC000217927981 ED In-Stock Unstable MMP9 15 50 CCOC(=O)C1(S(C)(=O)=O)CCN(Cc2ccccc2)CC1 ZINC000217927981 ED In-Stock Unstable MCHR2 41 32 CCOC(=O)C1(S(C)(=O)=O)CCN(Cc2ccccc2)CC1 ZINC000217927981 ED In-Stock Unstable CCR8 49 37 CCOC(=O)C1(S(C)(=O)=O)CCN(Cc2ccccc2)CC1 ZINC000217927981 ED In-Stock Unstable NPFFR1 65 42 CCOC(=O)C1(S(C)(=O)=O)CCN(Cc2ccccc2)CC1 ZINC000217927981 ED In-Stock Unstable SLC12A5 72 37 CCOC(=O)C1(S(C)(=O)=O)CCN(Cc2ccccc2)CC1 ZINC000217927981 ED In-Stock Unstable PA 21 41 CCCCOCCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217928014 DG For-Sale Unstable HRH2 25 42 CCCCOCCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217928014 DG For-Sale Unstable MTNR1A 109 46 CCCCOCCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217928014 DG For-Sale Unstable MTNR1B 98 46 CCCCOCCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217928014 DG For-Sale Unstable ACAT 0 43 CC[C@@H](CCO)NC(=O)[C@@H](N)CC(=O)O ZINC000217928034 BB For-Sale Unstable ENPEP 56 32 O=C(/C=C/c1ccc2c(c1)OCO2)NCCCc1ccc(F)cc1 ZINC000217928042 EG In-Stock Unstable PYGL 25 44 O=C(/C=C/c1ccc2c(c1)OCO2)NCCCc1ccc(F)cc1 ZINC000217928042 EG In-Stock Unstable HDAC7 46 35 O=C(/C=C/c1ccc2c(c1)OCO2)NCCCc1ccc(F)cc1 ZINC000217928042 EG In-Stock Unstable DYRK2 46 36 COc1ccc(CN(C)CC(F)(F)F)cc1/C=C\C(=O)O ZINC000217928052 DF For-Sale Unstable PTGER2 28 42 COc1ccc(CN(C)CC(F)(F)F)cc1/C=C\C(=O)O ZINC000217928052 DF For-Sale Unstable PTGER4 17 42 O=C(NCC[C@H](O)C1CCOCC1)Nc1ccccc1 ZINC000217928077 CD In-Stock Unstable ACAT 0 40 O=C(NCC[C@H](O)C1CCOCC1)Nc1ccccc1 ZINC000217928077 CD In-Stock Unstable P95276_MYCTO 0 40 CCOC(=O)C1(S(=O)(=O)CC)CCN(Cc2ccccc2)CC1 ZINC000217928087 EE In-Stock Unstable CHRM2 20 42 CCOC(=O)C1(S(=O)(=O)CC)CCN(Cc2ccccc2)CC1 ZINC000217928087 EE In-Stock Unstable DRD2 15 42 CCOC(=O)C1(S(=O)(=O)CC)CCN(Cc2ccccc2)CC1 ZINC000217928087 EE In-Stock Unstable DRD4 35 40 CCOC(=O)C1(S(=O)(=O)CC)CCN(Cc2ccccc2)CC1 ZINC000217928087 EE In-Stock Unstable ACHE 24 40 CCOC(=O)C1(S(=O)(=O)CC)CCN(Cc2ccccc2)CC1 ZINC000217928087 EE In-Stock Unstable DRD3 24 42 CCOC(=O)C1(S(=O)(=O)CC)CCN(Cc2ccccc2)CC1 ZINC000217928087 EE In-Stock Unstable OPRK1 15 40 CCOC(=O)C1(S(=O)(=O)CC)CCN(Cc2ccccc2)CC1 ZINC000217928087 EE In-Stock Unstable OPRL1 18 42 CCOC(=O)C1(S(=O)(=O)CC)CCN(Cc2ccccc2)CC1 ZINC000217928087 EE In-Stock Unstable CHRM3 15 47 CCOC(=O)C1(S(=O)(=O)CC)CCN(Cc2ccccc2)CC1 ZINC000217928087 EE In-Stock Unstable SIGMAR1 76 53 CCOC(=O)C1(S(=O)(=O)CC)CCN(Cc2ccccc2)CC1 ZINC000217928087 EE In-Stock Unstable MMP13 22 53 CCOC(=O)C1(S(=O)(=O)CC)CCN(Cc2ccccc2)CC1 ZINC000217928087 EE In-Stock Unstable NPFFR2 42 41 CCOC(=O)C1(S(=O)(=O)CC)CCN(Cc2ccccc2)CC1 ZINC000217928087 EE In-Stock Unstable ADAM17 33 53 CCOC(=O)C1(S(=O)(=O)CC)CCN(Cc2ccccc2)CC1 ZINC000217928087 EE In-Stock Unstable MMP14 18 48 CCOC(=O)C1(S(=O)(=O)CC)CCN(Cc2ccccc2)CC1 ZINC000217928087 EE In-Stock Unstable MMP9 20 53 CCOC(=O)C1(S(=O)(=O)CC)CCN(Cc2ccccc2)CC1 ZINC000217928087 EE In-Stock Unstable MCHR2 40 31 CCOC(=O)C1(S(=O)(=O)CC)CCN(Cc2ccccc2)CC1 ZINC000217928087 EE In-Stock Unstable CCR8 49 37 CCOC(=O)C1(S(=O)(=O)CC)CCN(Cc2ccccc2)CC1 ZINC000217928087 EE In-Stock Unstable NPFFR1 65 42 CCOC(=O)C1(S(=O)(=O)CC)CCN(Cc2ccccc2)CC1 ZINC000217928087 EE In-Stock Unstable SLC12A5 71 36 CCOC(=O)C1(S(=O)(=O)CC)CCN(Cc2ccccc2)CC1 ZINC000217928087 EE In-Stock Unstable PA 21 41 CC[C@H](CCO)NC(=O)[C@@H](N)CC(=O)O ZINC000217928112 BB For-Sale Unstable ENPEP 56 32 COc1cccc(/C=C/NC(=O)NCc2cccnc2)c1 ZINC000217928118 CF For-Sale Unstable PTAFR 38 47 COc1cccc(/C=C/NC(=O)NCc2cccnc2)c1 ZINC000217928118 CF For-Sale Unstable TRPV1 0 44 COc1cccc(/C=C/NC(=O)NCc2cccnc2)c1 ZINC000217928118 CF For-Sale Unstable MMP13 26 40 COc1cccc(/C=C/NC(=O)NCc2cccnc2)c1 ZINC000217928118 CF For-Sale Unstable ROCK1 41 45 COc1cccc(/C=C/NC(=O)NCc2cccnc2)c1 ZINC000217928118 CF For-Sale Unstable MTNR1A 46 44 COc1cccc(/C=C/NC(=O)NCc2cccnc2)c1 ZINC000217928118 CF For-Sale Unstable MTNR1B 48 44 COc1cccc(/C=C/NC(=O)NCc2cccnc2)c1 ZINC000217928118 CF For-Sale Unstable ROCK2 47 49 COc1cccc(/C=C/NC(=O)NCc2cccnc2)c1 ZINC000217928118 CF For-Sale Unstable NAMPT 65 47 NCCCCCCCN1CC[C@H]2CCCC[C@@H]2C1 ZINC000217928124 CG For-Sale Unstable GNAO1 0 40 COc1ccccc1CCCNC(=O)/C=C/c1ccc2c(c1)OCO2 ZINC000217928152 EG In-Stock Unstable DRD2 21 69 COc1ccccc1CCCNC(=O)/C=C/c1ccc2c(c1)OCO2 ZINC000217928152 EG In-Stock Unstable DRD3 37 69 COc1ccccc1CCCNC(=O)/C=C/c1ccc2c(c1)OCO2 ZINC000217928152 EG In-Stock Unstable EDNRB 40 41 COc1ccccc1CCCNC(=O)/C=C/c1ccc2c(c1)OCO2 ZINC000217928152 EG In-Stock Unstable BCHE 15 41 COc1ccccc1CCCNC(=O)/C=C/c1ccc2c(c1)OCO2 ZINC000217928152 EG In-Stock Unstable PYGL 23 41 COc1ccccc1CCCNC(=O)/C=C/c1ccc2c(c1)OCO2 ZINC000217928152 EG In-Stock Unstable PLK1 0 40 COc1ccccc1CCCNC(=O)/C=C/c1ccc2c(c1)OCO2 ZINC000217928152 EG In-Stock Unstable MTNR1B 38 42 COc1ccccc1CCCNC(=O)/C=C/c1ccc2c(c1)OCO2 ZINC000217928152 EG In-Stock Unstable DYRK2 50 34 O=C(NCC[C@@H](O)C1CCOCC1)Nc1ccccc1 ZINC000217928168 CD In-Stock Unstable ACAT 0 40 O=C(NCC[C@@H](O)C1CCOCC1)Nc1ccccc1 ZINC000217928168 CD In-Stock Unstable P95276_MYCTO 0 40 CC[C@@H](CCO)NC(=O)[C@H](N)CC(=O)O ZINC000217928200 BB For-Sale Unstable ENPEP 56 32 CS(=O)(=O)C1(CO)CCN(Cc2ccccc2)CC1 ZINC000217928201 CD In-Stock Unstable CHRM2 18 45 CS(=O)(=O)C1(CO)CCN(Cc2ccccc2)CC1 ZINC000217928201 CD In-Stock Unstable DRD2 20 46 CS(=O)(=O)C1(CO)CCN(Cc2ccccc2)CC1 ZINC000217928201 CD In-Stock Unstable DRD4 45 37 CS(=O)(=O)C1(CO)CCN(Cc2ccccc2)CC1 ZINC000217928201 CD In-Stock Unstable DRD3 25 45 CS(=O)(=O)C1(CO)CCN(Cc2ccccc2)CC1 ZINC000217928201 CD In-Stock Unstable OPRD1 15 40 CS(=O)(=O)C1(CO)CCN(Cc2ccccc2)CC1 ZINC000217928201 CD In-Stock Unstable OPRK1 23 44 CS(=O)(=O)C1(CO)CCN(Cc2ccccc2)CC1 ZINC000217928201 CD In-Stock Unstable OPRL1 21 48 CS(=O)(=O)C1(CO)CCN(Cc2ccccc2)CC1 ZINC000217928201 CD In-Stock Unstable SIGMAR1 92 50 CS(=O)(=O)C1(CO)CCN(Cc2ccccc2)CC1 ZINC000217928201 CD In-Stock Unstable NPFFR2 43 43 CS(=O)(=O)C1(CO)CCN(Cc2ccccc2)CC1 ZINC000217928201 CD In-Stock Unstable ADAM17 21 45 CS(=O)(=O)C1(CO)CCN(Cc2ccccc2)CC1 ZINC000217928201 CD In-Stock Unstable EBP 17 40 CS(=O)(=O)C1(CO)CCN(Cc2ccccc2)CC1 ZINC000217928201 CD In-Stock Unstable MCHR2 52 38 CS(=O)(=O)C1(CO)CCN(Cc2ccccc2)CC1 ZINC000217928201 CD In-Stock Unstable NPFFR1 67 43 CS(=O)(=O)C1(CO)CCN(Cc2ccccc2)CC1 ZINC000217928201 CD In-Stock Unstable SLC12A5 55 34 CS(=O)(=O)C1(CO)CCN(Cc2ccccc2)CC1 ZINC000217928201 CD In-Stock Unstable PA 21 41 COc1cccc(/C=C/NC(=O)NC(C)(C)C)c1 ZINC000217928230 BF For-Sale Unstable CYP1B1 35 43 COc1cccc(/C=C/NC(=O)NC(C)(C)C)c1 ZINC000217928230 BF For-Sale Unstable AHR 15 44 COc1cccc(/C=C/NC(=O)NC(C)(C)C)c1 ZINC000217928230 BF For-Sale Unstable MTNR1A 38 44 COc1cccc(/C=C/NC(=O)NC(C)(C)C)c1 ZINC000217928230 BF For-Sale Unstable MTNR1B 39 44 COc1cccc(/C=C/NC(=O)NC(C)(C)C)c1 ZINC000217928230 BF For-Sale Unstable CYP1A1 26 43 COc1cccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)c1 ZINC000217928259 EG In-Stock Unstable DRD4 41 32 COc1cccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)c1 ZINC000217928259 EG In-Stock Unstable DRD3 20 57 COc1cccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)c1 ZINC000217928259 EG In-Stock Unstable EDNRB 48 44 COc1cccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)c1 ZINC000217928259 EG In-Stock Unstable EDNRA 43 36 COc1cccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)c1 ZINC000217928259 EG In-Stock Unstable PTAFR 18 41 COc1cccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)c1 ZINC000217928259 EG In-Stock Unstable BMP1 47 37 COc1cccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)c1 ZINC000217928259 EG In-Stock Unstable PYGL 22 42 COc1cccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)c1 ZINC000217928259 EG In-Stock Unstable MTNR1A 60 56 COc1cccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)c1 ZINC000217928259 EG In-Stock Unstable MTNR1B 44 56 COc1cccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)c1 ZINC000217928259 EG In-Stock Unstable DYRK2 50 35 COc1cccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)c1 ZINC000217928259 EG In-Stock Unstable CRTM 57 43 CC[C@H](CCO)NC(=O)[C@H](N)CC(=O)O ZINC000217928277 BB For-Sale Unstable ENPEP 56 32 O=C(NCC[C@H](O)C1CCOCC1)NC1CCCCC1 ZINC000217928295 CD In-Stock Unstable EPHX2 16 46 O=C(N[C@@H]1CCC[C@@H]1CO)c1ccc2ncccc2c1 ZINC000217928304 CE For-Sale Unstable ADAM17 28 40 O=C(N[C@@H]1CCC[C@@H]1CO)c1ccc2ncccc2c1 ZINC000217928304 CE For-Sale Unstable SSTR3 29 43 CCS(=O)(=O)C1(CO)CCN(Cc2ccccc2)CC1 ZINC000217928324 CD In-Stock Unstable CHRM2 18 44 CCS(=O)(=O)C1(CO)CCN(Cc2ccccc2)CC1 ZINC000217928324 CD In-Stock Unstable DRD2 18 44 CCS(=O)(=O)C1(CO)CCN(Cc2ccccc2)CC1 ZINC000217928324 CD In-Stock Unstable DRD4 42 39 CCS(=O)(=O)C1(CO)CCN(Cc2ccccc2)CC1 ZINC000217928324 CD In-Stock Unstable DRD3 22 44 CCS(=O)(=O)C1(CO)CCN(Cc2ccccc2)CC1 ZINC000217928324 CD In-Stock Unstable OPRK1 21 43 CCS(=O)(=O)C1(CO)CCN(Cc2ccccc2)CC1 ZINC000217928324 CD In-Stock Unstable OPRL1 22 47 CCS(=O)(=O)C1(CO)CCN(Cc2ccccc2)CC1 ZINC000217928324 CD In-Stock Unstable CHRM3 15 48 CCS(=O)(=O)C1(CO)CCN(Cc2ccccc2)CC1 ZINC000217928324 CD In-Stock Unstable SIGMAR1 91 49 CCS(=O)(=O)C1(CO)CCN(Cc2ccccc2)CC1 ZINC000217928324 CD In-Stock Unstable NPFFR2 43 43 CCS(=O)(=O)C1(CO)CCN(Cc2ccccc2)CC1 ZINC000217928324 CD In-Stock Unstable ADAM17 22 45 CCS(=O)(=O)C1(CO)CCN(Cc2ccccc2)CC1 ZINC000217928324 CD In-Stock Unstable MCHR2 50 33 CCS(=O)(=O)C1(CO)CCN(Cc2ccccc2)CC1 ZINC000217928324 CD In-Stock Unstable NPFFR1 67 44 CCS(=O)(=O)C1(CO)CCN(Cc2ccccc2)CC1 ZINC000217928324 CD In-Stock Unstable SLC12A5 45 32 CCS(=O)(=O)C1(CO)CCN(Cc2ccccc2)CC1 ZINC000217928324 CD In-Stock Unstable PA 21 40 COc1cccc(/C=C/NC(=O)N2CCC(Cc3ccccc3)CC2)c1 ZINC000217928331 FI For-Sale Unstable DRD4 41 32 COc1cccc(/C=C/NC(=O)N2CCC(Cc3ccccc3)CC2)c1 ZINC000217928331 FI For-Sale Unstable ACHE 18 46 COc1cccc(/C=C/NC(=O)N2CCC(Cc3ccccc3)CC2)c1 ZINC000217928331 FI For-Sale Unstable GRIN2B 80 45 COc1cccc(/C=C/NC(=O)N2CCC(Cc3ccccc3)CC2)c1 ZINC000217928331 FI For-Sale Unstable SIGMAR1 28 53 COc1cccc(/C=C/NC(=O)N2CCC(Cc3ccccc3)CC2)c1 ZINC000217928331 FI For-Sale Unstable CCR3 60 53 COc1cccc(/C=C/NC(=O)N2CCC(Cc3ccccc3)CC2)c1 ZINC000217928331 FI For-Sale Unstable MTNR1B 41 38 COc1cccc(/C=C/NC(=O)N2CCC(Cc3ccccc3)CC2)c1 ZINC000217928331 FI For-Sale Unstable AMP1_PLAFQ 24 46 COc1cccc(/C=C/NC(=O)N2CCC(Cc3ccccc3)CC2)c1 ZINC000217928331 FI For-Sale Unstable ACKR3 46 34 COc1ccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217928362 EG In-Stock Unstable DRD3 17 57 COc1ccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217928362 EG In-Stock Unstable EDNRB 63 49 COc1ccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217928362 EG In-Stock Unstable EDNRA 62 39 COc1ccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217928362 EG In-Stock Unstable BMP1 61 41 COc1ccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217928362 EG In-Stock Unstable PYGL 23 42 COc1ccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217928362 EG In-Stock Unstable HDAC8 26 41 COc1ccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217928362 EG In-Stock Unstable PLK1 0 49 COc1ccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217928362 EG In-Stock Unstable MTNR1A 44 41 COc1ccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217928362 EG In-Stock Unstable NR1H4 15 40 COc1ccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217928362 EG In-Stock Unstable HDAC1 18 43 COc1ccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217928362 EG In-Stock Unstable HDAC2 0 40 COc1ccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217928362 EG In-Stock Unstable HDAC6 17 41 COc1ccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217928362 EG In-Stock Unstable DYRK1A 20 40 COc1ccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217928362 EG In-Stock Unstable CLK1 30 40 COc1ccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217928362 EG In-Stock Unstable DYRK2 57 39 O=C(N[C@H]1CCC[C@@H]1CO)c1ccc2ncccc2c1 ZINC000217928368 CE For-Sale Unstable ADAM17 28 40 O=C(N[C@H]1CCC[C@@H]1CO)c1ccc2ncccc2c1 ZINC000217928368 CE For-Sale Unstable SSTR3 29 43 O=C(NCC[C@@H](O)C1CCOCC1)NC1CCCCC1 ZINC000217928373 CD In-Stock Unstable EPHX2 16 46 CS(=O)(=O)C1(C(N)=S)CCN(Cc2ccccc2)CC1 ZINC000217928427 DD In-Stock Unstable DRD2 0 43 CS(=O)(=O)C1(C(N)=S)CCN(Cc2ccccc2)CC1 ZINC000217928427 DD In-Stock Unstable DRD3 0 42 CS(=O)(=O)C1(C(N)=S)CCN(Cc2ccccc2)CC1 ZINC000217928427 DD In-Stock Unstable OPRL1 16 44 CS(=O)(=O)C1(C(N)=S)CCN(Cc2ccccc2)CC1 ZINC000217928427 DD In-Stock Unstable SIGMAR1 71 45 CS(=O)(=O)C1(C(N)=S)CCN(Cc2ccccc2)CC1 ZINC000217928427 DD In-Stock Unstable MMP13 17 50 CS(=O)(=O)C1(C(N)=S)CCN(Cc2ccccc2)CC1 ZINC000217928427 DD In-Stock Unstable NPFFR2 43 42 CS(=O)(=O)C1(C(N)=S)CCN(Cc2ccccc2)CC1 ZINC000217928427 DD In-Stock Unstable ADAM17 25 50 CS(=O)(=O)C1(C(N)=S)CCN(Cc2ccccc2)CC1 ZINC000217928427 DD In-Stock Unstable NPFFR1 66 42 COc1cccc(/C=C/NC(=O)N(C)C2CCN(C)CC2)c1 ZINC000217928434 DE For-Sale Unstable DRD4 41 31 COc1cccc(/C=C/NC(=O)N(C)C2CCN(C)CC2)c1 ZINC000217928434 DE For-Sale Unstable MTNR1A 25 41 COc1cccc(/C=C/NC(=O)N(C)C2CCN(C)CC2)c1 ZINC000217928434 DE For-Sale Unstable MTNR1B 33 41 COc1cccc(/C=C/NC(=O)N(C)C2CCN(C)CC2)c1 ZINC000217928434 DE For-Sale Unstable ACKR3 62 34 O=C(N[C@@H]1CCC[C@H]1CO)c1ccc2ncccc2c1 ZINC000217928444 CE For-Sale Unstable ADAM17 28 40 O=C(N[C@@H]1CCC[C@H]1CO)c1ccc2ncccc2c1 ZINC000217928444 CE For-Sale Unstable SSTR3 29 43 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217928495 FG In-Stock Unstable EDNRB 60 46 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217928495 FG In-Stock Unstable EDNRA 64 38 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217928495 FG In-Stock Unstable BMP1 55 37 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217928495 FG In-Stock Unstable KCNQ2 21 43 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217928495 FG In-Stock Unstable DYRK1A 19 40 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217928495 FG In-Stock Unstable CLK1 31 40 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217928495 FG In-Stock Unstable DYRK2 57 39 Cn1nc(C(C)(C)C)cc1C(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217928519 FE In-Stock Unstable CHRNA4 27 50 Cn1nc(C(C)(C)C)cc1C(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217928519 FE In-Stock Unstable CTSV 44 30 O=C(N[C@H]1CCC[C@H]1CO)c1ccc2ncccc2c1 ZINC000217928525 CE On-Demand Unstable ADAM17 25 40 CCS(=O)(=O)C1(C(N)=S)CCN(Cc2ccccc2)CC1 ZINC000217928529 ED In-Stock Unstable CHRM2 15 41 CCS(=O)(=O)C1(C(N)=S)CCN(Cc2ccccc2)CC1 ZINC000217928529 ED In-Stock Unstable DRD3 0 41 CCS(=O)(=O)C1(C(N)=S)CCN(Cc2ccccc2)CC1 ZINC000217928529 ED In-Stock Unstable OPRL1 16 43 CCS(=O)(=O)C1(C(N)=S)CCN(Cc2ccccc2)CC1 ZINC000217928529 ED In-Stock Unstable SIGMAR1 68 44 CCS(=O)(=O)C1(C(N)=S)CCN(Cc2ccccc2)CC1 ZINC000217928529 ED In-Stock Unstable MMP13 17 49 CCS(=O)(=O)C1(C(N)=S)CCN(Cc2ccccc2)CC1 ZINC000217928529 ED In-Stock Unstable NPFFR2 43 42 CCS(=O)(=O)C1(C(N)=S)CCN(Cc2ccccc2)CC1 ZINC000217928529 ED In-Stock Unstable ADAM17 26 49 CCS(=O)(=O)C1(C(N)=S)CCN(Cc2ccccc2)CC1 ZINC000217928529 ED In-Stock Unstable MCHR2 47 31 CCS(=O)(=O)C1(C(N)=S)CCN(Cc2ccccc2)CC1 ZINC000217928529 ED In-Stock Unstable NPFFR1 67 44 CCN(CCNC(=O)c1cc(N)cn1C)C1CC1 ZINC000217928532 CC For-Sale Unstable HRAS 50 34 COc1ccc(CCNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217928540 EG For-Sale Unstable DRD4 41 31 COc1ccc(CCNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217928540 EG For-Sale Unstable CYP1B1 23 41 COc1ccc(CCNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217928540 EG For-Sale Unstable NQO2 42 44 COc1ccc(CCNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217928540 EG For-Sale Unstable AHR 27 40 COc1ccc(CCNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217928540 EG For-Sale Unstable MTNR1A 143 49 COc1ccc(CCNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217928540 EG For-Sale Unstable MTNR1B 123 49 COc1ccc(CCNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217928540 EG For-Sale Unstable CYP1A1 21 41 COc1ccc(CCNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217928540 EG For-Sale Unstable ROCK2 18 44 COc1ccc(CCNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217928540 EG For-Sale Unstable PTGDR 23 41 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217928588 FG In-Stock Unstable EDNRB 60 46 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217928588 FG In-Stock Unstable EDNRA 64 38 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217928588 FG In-Stock Unstable BMP1 55 37 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217928588 FG In-Stock Unstable KCNQ2 21 43 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217928588 FG In-Stock Unstable DYRK1A 19 40 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217928588 FG In-Stock Unstable CLK1 31 40 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217928588 FG In-Stock Unstable DYRK2 57 39 O=C(CSCCc1ccccc1)N[C@@H]1CCC[C@@H]1CO ZINC000217928628 CE For-Sale Unstable SIGMAR1 19 40 CS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928634 CD In-Stock Unstable CHRM2 19 47 CS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928634 CD In-Stock Unstable DRD2 24 47 CS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928634 CD In-Stock Unstable DRD4 54 39 CS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928634 CD In-Stock Unstable ACHE 30 40 CS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928634 CD In-Stock Unstable DRD3 27 47 CS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928634 CD In-Stock Unstable OPRK1 18 43 CS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928634 CD In-Stock Unstable OPRL1 27 44 CS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928634 CD In-Stock Unstable CHRM3 19 51 CS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928634 CD In-Stock Unstable SIGMAR1 91 49 CS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928634 CD In-Stock Unstable MMP13 20 53 CS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928634 CD In-Stock Unstable NPFFR2 42 42 CS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928634 CD In-Stock Unstable ADAM17 28 53 CS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928634 CD In-Stock Unstable MMP9 16 53 CS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928634 CD In-Stock Unstable TRPV4 15 40 CS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928634 CD In-Stock Unstable MCHR2 50 34 CS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928634 CD In-Stock Unstable CCR8 44 39 CS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928634 CD In-Stock Unstable NPFFR1 66 42 CS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928634 CD In-Stock Unstable SLC12A5 52 34 CS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928634 CD In-Stock Unstable PA 22 43 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc2ccc(C)nc12 ZINC000217928635 HH For-Sale Unstable HCRTR1 57 41 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc2ccc(C)nc12 ZINC000217928635 HH For-Sale Unstable HCRTR2 59 41 COc1cccc(/C=C/NC(=O)NC[C@@H]2CCCO2)c1 ZINC000217928654 CE For-Sale Unstable DRD4 40 30 COc1cccc(/C=C/NC(=O)NC[C@@H]2CCCO2)c1 ZINC000217928654 CE For-Sale Unstable MTNR1A 51 39 COc1cccc(/C=C/NC(=O)NC[C@@H]2CCCO2)c1 ZINC000217928654 CE For-Sale Unstable MTNR1B 47 39 COc1cccc(/C=C/NC(=O)NC[C@@H]2CCCO2)c1 ZINC000217928654 CE For-Sale Unstable ACKR3 44 32 Cc1cccc(NC(=O)NCC[C@H](O)C2CCOCC2)c1 ZINC000217928672 CE In-Stock Unstable CASR 0 41 Cc1cccc(NC(=O)NCC[C@H](O)C2CCOCC2)c1 ZINC000217928672 CE In-Stock Unstable CCKAR 24 44 Cc1cccc(NC(=O)NCC[C@H](O)C2CCOCC2)c1 ZINC000217928672 CE In-Stock Unstable EPHX2 17 40 Cc1cccc(NC(=O)NCC[C@H](O)C2CCOCC2)c1 ZINC000217928672 CE In-Stock Unstable ACAT 0 44 Cc1cccc(NC(=O)NCC[C@H](O)C2CCOCC2)c1 ZINC000217928672 CE In-Stock Unstable KCNK3 52 38 Cc1cccc(NC(=O)NCC[C@H](O)C2CCOCC2)c1 ZINC000217928672 CE In-Stock Unstable KCNK9 47 38 O=C(CSCCc1ccccc1)N[C@H]1CCC[C@@H]1CO ZINC000217928693 CE For-Sale Unstable SIGMAR1 19 40 O=C(/C=C/c1ccc2c(c1)OCO2)Nc1ccccc1C(=O)c1ccccc1 ZINC000217928694 FI In-Stock Unstable LTB4R 0 49 O=C(/C=C/c1ccc2c(c1)OCO2)Nc1ccccc1C(=O)c1ccccc1 ZINC000217928694 FI In-Stock Unstable PLK1 0 47 O=C(/C=C/c1ccc2c(c1)OCO2)Nc1ccccc1C(=O)c1ccccc1 ZINC000217928694 FI In-Stock Unstable MMP2 20 44 O=C(/C=C/c1ccc2c(c1)OCO2)Nc1ccccc1C(=O)c1ccccc1 ZINC000217928694 FI In-Stock Unstable HDAC1 15 43 O=C(/C=C/c1ccc2c(c1)OCO2)Nc1ccccc1C(=O)c1ccccc1 ZINC000217928694 FI In-Stock Unstable MMP9 18 44 O=C(/C=C/c1ccc2c(c1)OCO2)Nc1ccccc1C(=O)c1ccccc1 ZINC000217928694 FI In-Stock Unstable MMP1 24 45 O=C(/C=C/c1ccc2c(c1)OCO2)Nc1ccccc1C(=O)c1ccccc1 ZINC000217928694 FI In-Stock Unstable DYRK2 49 34 O=C(/C=C/c1ccc2c(c1)OCO2)Nc1ccccc1C(=O)c1ccccc1 ZINC000217928694 FI In-Stock Unstable TRPM2 0 42 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc2ccc(C)nc12 ZINC000217928712 HH For-Sale Unstable HCRTR1 57 41 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc2ccc(C)nc12 ZINC000217928712 HH For-Sale Unstable HCRTR2 59 41 COc1cccc(/C=C/NC(=O)NC[C@H]2CCCO2)c1 ZINC000217928732 CE For-Sale Unstable DRD4 40 30 COc1cccc(/C=C/NC(=O)NC[C@H]2CCCO2)c1 ZINC000217928732 CE For-Sale Unstable MTNR1A 51 39 COc1cccc(/C=C/NC(=O)NC[C@H]2CCCO2)c1 ZINC000217928732 CE For-Sale Unstable MTNR1B 47 39 COc1cccc(/C=C/NC(=O)NC[C@H]2CCCO2)c1 ZINC000217928732 CE For-Sale Unstable ACKR3 44 32 CCS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928739 DD In-Stock Unstable CHRM2 21 46 CCS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928739 DD In-Stock Unstable DRD2 20 46 CCS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928739 DD In-Stock Unstable DRD4 50 41 CCS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928739 DD In-Stock Unstable ACHE 31 40 CCS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928739 DD In-Stock Unstable DRD3 23 46 CCS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928739 DD In-Stock Unstable OPRK1 16 42 CCS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928739 DD In-Stock Unstable OPRL1 26 43 CCS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928739 DD In-Stock Unstable CHRM3 21 50 CCS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928739 DD In-Stock Unstable SIGMAR1 89 47 CCS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928739 DD In-Stock Unstable MMP13 20 52 CCS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928739 DD In-Stock Unstable NPFFR2 43 42 CCS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928739 DD In-Stock Unstable ADAM17 27 52 CCS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928739 DD In-Stock Unstable MMP14 17 47 CCS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928739 DD In-Stock Unstable MMP9 15 52 CCS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928739 DD In-Stock Unstable MCHR2 50 33 CCS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928739 DD In-Stock Unstable CCR8 43 38 CCS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928739 DD In-Stock Unstable NPFFR1 66 44 CCS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928739 DD In-Stock Unstable SLC12A5 45 33 CCS(=O)(=O)C1(C(=O)O)CCN(Cc2ccccc2)CC1 ZINC000217928739 DD In-Stock Unstable PA 22 42 CCC(CO)(CO)NC[C@@H](O)COc1ccc(C)cc1 ZINC000217928741 CC For-Sale Unstable ADRB2 50 61 CCC(CO)(CO)NC[C@@H](O)COc1ccc(C)cc1 ZINC000217928741 CC For-Sale Unstable ADRB1 49 48 CCC(CO)(CO)NC[C@@H](O)COc1ccc(C)cc1 ZINC000217928741 CC For-Sale Unstable ADRB3 23 40 CCC(CO)(CO)NC[C@@H](O)COc1ccc(C)cc1 ZINC000217928741 CC For-Sale Unstable CYP2D6 19 40 Cc1cccc(NC(=O)NCC[C@@H](O)C2CCOCC2)c1 ZINC000217928754 CE In-Stock Unstable CASR 0 41 Cc1cccc(NC(=O)NCC[C@@H](O)C2CCOCC2)c1 ZINC000217928754 CE In-Stock Unstable CCKAR 24 44 Cc1cccc(NC(=O)NCC[C@@H](O)C2CCOCC2)c1 ZINC000217928754 CE In-Stock Unstable EPHX2 17 40 Cc1cccc(NC(=O)NCC[C@@H](O)C2CCOCC2)c1 ZINC000217928754 CE In-Stock Unstable ACAT 0 44 Cc1cccc(NC(=O)NCC[C@@H](O)C2CCOCC2)c1 ZINC000217928754 CE In-Stock Unstable KCNK3 52 38 Cc1cccc(NC(=O)NCC[C@@H](O)C2CCOCC2)c1 ZINC000217928754 CE In-Stock Unstable KCNK9 47 38 O=C(CSCCc1ccccc1)N[C@@H]1CCC[C@H]1CO ZINC000217928767 CE For-Sale Unstable SIGMAR1 19 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc2ccc(C)nc12 ZINC000217928787 HH For-Sale Unstable HCRTR1 57 41 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc2ccc(C)nc12 ZINC000217928787 HH For-Sale Unstable HCRTR2 59 41 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)c1 ZINC000217928799 FH In-Stock Unstable DYRK2 48 34 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)c1 ZINC000217928799 FH In-Stock Unstable CRTM 56 44 Cc1noc2nc(C(C)C)cc(C(=O)Nc3ccc(Cl)cc3)c12 ZINC000217928805 EJ On-Demand Unstable NR2E3 53 34 Cc1noc2nc(C(C)C)cc(C(=O)Nc3ccc(Cl)cc3)c12 ZINC000217928805 EJ On-Demand Unstable Q25615_ONCVO 46 36 CCN(CCOC)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217928815 CE For-Sale Unstable TUBB1 42 37 CCN(CCOC)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217928815 CE For-Sale Unstable AKR1C3 22 40 CCC(CO)(CO)NC[C@H](O)COc1ccc(C)cc1 ZINC000217928823 CC For-Sale Unstable ADRB2 50 61 CCC(CO)(CO)NC[C@H](O)COc1ccc(C)cc1 ZINC000217928823 CC For-Sale Unstable ADRB1 49 48 CCC(CO)(CO)NC[C@H](O)COc1ccc(C)cc1 ZINC000217928823 CC For-Sale Unstable ADRB3 23 40 CCC(CO)(CO)NC[C@H](O)COc1ccc(C)cc1 ZINC000217928823 CC For-Sale Unstable CYP2D6 19 40 N#Cc1cc(Cl)ccc1N1CCC[C@@H]2CCCC[C@H]21 ZINC000217928830 CI For-Sale Unstable AR 26 43 C[C@@H]1CCC[C@@H](CNc2cc(Cl)nc(N)n2)C1 ZINC000217928831 CF On-Demand Unstable HRH4 27 41 CC[C@H](CCO)NC(=O)[C@@H](C)[C@@H](N)c1ccccc1 ZINC000217928835 CD For-Sale Unstable MME 53 40 CC[C@H](CCO)NC(=O)[C@@H](C)[C@@H](N)c1ccccc1 ZINC000217928835 CD For-Sale Unstable ANPEP 68 36 CC[C@H](CCO)NC(=O)[C@@H](C)[C@@H](N)c1ccccc1 ZINC000217928835 CD For-Sale Unstable ACE2 51 33 CC[C@H](CCO)NC(=O)[C@@H](C)[C@@H](N)c1ccccc1 ZINC000217928835 CD For-Sale Unstable CTSC 32 43 O=C(CSCCc1ccccc1)N[C@H]1CCC[C@H]1CO ZINC000217928836 CE For-Sale Unstable SIGMAR1 19 40 COc1cccc(/C=C/NC(=O)NCc2ccc(Cl)cc2)c1 ZINC000217928842 DH For-Sale Unstable DRD4 43 38 COc1cccc(/C=C/NC(=O)NCc2ccc(Cl)cc2)c1 ZINC000217928842 DH For-Sale Unstable MTNR1A 51 43 COc1cccc(/C=C/NC(=O)NCc2ccc(Cl)cc2)c1 ZINC000217928842 DH For-Sale Unstable MTNR1B 51 43 COc1cccc(/C=C/NC(=O)NCc2ccc(Cl)cc2)c1 ZINC000217928842 DH For-Sale Unstable ROCK2 23 41 COc1cccc(/C=C/NC(=O)NCc2ccc(Cl)cc2)c1 ZINC000217928842 DH For-Sale Unstable PDS 65 41 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc2ccc(C)nc12 ZINC000217928870 HH For-Sale Unstable HCRTR1 57 41 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc2ccc(C)nc12 ZINC000217928870 HH For-Sale Unstable HCRTR2 59 41 C[C@H]1CCC[C@@H](CNc2cc(Cl)nc(N)n2)C1 ZINC000217928905 CF On-Demand Unstable HRH4 27 41 N#Cc1cc(Cl)ccc1N1CCC[C@H]2CCCC[C@H]21 ZINC000217928917 CI For-Sale Unstable AR 26 43 CC(C)Oc1ccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217928919 FH In-Stock Unstable EDNRB 30 42 CC(C)Oc1ccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217928919 FH In-Stock Unstable BMP1 40 35 CC(C)Oc1ccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217928919 FH In-Stock Unstable PYGL 0 40 CC(C)Oc1ccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217928919 FH In-Stock Unstable DYRK2 53 35 CCC(CO)(CO)NC[C@@H](O)COc1cccc(C)c1 ZINC000217928944 CC For-Sale Unstable ADRB2 45 64 CCC(CO)(CO)NC[C@@H](O)COc1cccc(C)c1 ZINC000217928944 CC For-Sale Unstable ADRB1 40 64 CCC(CO)(CO)NC[C@@H](O)COc1cccc(C)c1 ZINC000217928944 CC For-Sale Unstable PDS 47 41 CCN(CCOC)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217928945 CE For-Sale Unstable ACHE 18 45 CCN(CCOC)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217928945 CE For-Sale Unstable PTGER2 29 41 CCN(CCOC)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217928945 CE For-Sale Unstable PTGER4 17 41 COc1cccc(/C=C/NC(=O)N[C@@H](C)c2ccccc2)c1 ZINC000217928952 CH For-Sale Unstable ACACA 22 46 COc1cccc(/C=C/NC(=O)N[C@@H](C)c2ccccc2)c1 ZINC000217928952 CH For-Sale Unstable ACACB 17 50 COc1cccc(/C=C/NC(=O)N[C@@H](C)c2ccccc2)c1 ZINC000217928952 CH For-Sale Unstable MTNR1A 32 41 COc1cccc(/C=C/NC(=O)N[C@@H](C)c2ccccc2)c1 ZINC000217928952 CH For-Sale Unstable MTNR1B 39 41 C[C@@H]1CCC[C@H](CNc2cc(Cl)nc(N)n2)C1 ZINC000217928983 CF On-Demand Unstable HRH4 27 41 CC[C@H](CCO)NC(=O)[C@H](C)[C@@H](N)c1ccccc1 ZINC000217928996 CD For-Sale Unstable MME 53 40 CC[C@H](CCO)NC(=O)[C@H](C)[C@@H](N)c1ccccc1 ZINC000217928996 CD For-Sale Unstable ANPEP 68 36 CC[C@H](CCO)NC(=O)[C@H](C)[C@@H](N)c1ccccc1 ZINC000217928996 CD For-Sale Unstable ACE2 51 33 CC[C@H](CCO)NC(=O)[C@H](C)[C@@H](N)c1ccccc1 ZINC000217928996 CD For-Sale Unstable CTSC 32 43 CCC(CO)(CO)NC[C@H](O)COc1cccc(C)c1 ZINC000217929026 CC For-Sale Unstable ADRB2 45 64 CCC(CO)(CO)NC[C@H](O)COc1cccc(C)c1 ZINC000217929026 CC For-Sale Unstable ADRB1 40 64 CCC(CO)(CO)NC[C@H](O)COc1cccc(C)c1 ZINC000217929026 CC For-Sale Unstable PDS 47 41 COc1cccc(/C=C/NC(=O)N[C@H](C)c2ccccc2)c1 ZINC000217929031 CH For-Sale Unstable ACACA 22 46 COc1cccc(/C=C/NC(=O)N[C@H](C)c2ccccc2)c1 ZINC000217929031 CH For-Sale Unstable ACACB 17 50 COc1cccc(/C=C/NC(=O)N[C@H](C)c2ccccc2)c1 ZINC000217929031 CH For-Sale Unstable MTNR1A 32 41 COc1cccc(/C=C/NC(=O)N[C@H](C)c2ccccc2)c1 ZINC000217929031 CH For-Sale Unstable MTNR1B 39 41 CC(C)S(=O)(=O)CC(=O)N(C)[C@@H]1CCNC1 ZINC000217929038 BB On-Demand Unstable SLC6A2 29 42 COC(=O)COc1ccc([C@@H](CC(=O)OC)C2=C(O)C(=O)c3ccccc3C2=O)cc1OC ZINC000217929044 JF In-Stock Unstable TNF 22 43 CCN(Cc1ccco1)Cc1ccccc1/C=C\C(=O)O ZINC000217929054 CG For-Sale Unstable PTGER2 39 44 CCN(Cc1ccco1)Cc1ccccc1/C=C\C(=O)O ZINC000217929054 CG For-Sale Unstable PTGER4 0 44 CCN(Cc1ccco1)Cc1ccccc1/C=C\C(=O)O ZINC000217929054 CG For-Sale Unstable PTGER3 16 45 O=C(/C=C/c1ccc2c(c1)OCO2)Nc1ccc(OC2CCCC2)cc1 ZINC000217929055 FI In-Stock Unstable MMP2 0 45 O=C(/C=C/c1ccc2c(c1)OCO2)Nc1ccc(OC2CCCC2)cc1 ZINC000217929055 FI In-Stock Unstable MMP9 0 41 O=C(/C=C/c1ccc2c(c1)OCO2)Nc1ccc(OC2CCCC2)cc1 ZINC000217929055 FI In-Stock Unstable IMPDH2 0 41 O=C(/C=C/c1ccc2c(c1)OCO2)Nc1ccc(OC2CCCC2)cc1 ZINC000217929055 FI In-Stock Unstable MMP1 0 41 O=C(/C=C/c1ccc2c(c1)OCO2)Nc1ccc(OC2CCCC2)cc1 ZINC000217929055 FI In-Stock Unstable DYRK2 49 35 O=C(NCC[C@H](O)C1CCOCC1)Nc1cccc(Cl)c1 ZINC000217929064 DF In-Stock Unstable CASR 15 58 O=C(NCC[C@H](O)C1CCOCC1)Nc1cccc(Cl)c1 ZINC000217929064 DF In-Stock Unstable EPHX2 21 52 C[C@H]1CCC[C@H](CNc2cc(Cl)nc(N)n2)C1 ZINC000217929065 CF On-Demand Unstable HRH4 27 41 CC(C)(C)OC(=O)N1CC(F)(c2ccc(C#N)cc2)C1 ZINC000217929066 CF For-Sale Unstable GPR119 28 44 CC(C)S(=O)(=O)CC(=O)N(C)[C@H]1CCNC1 ZINC000217929118 BB On-Demand Unstable SLC6A2 29 42 COC(=O)COc1ccc([C@H](CC(=O)OC)C2=C(O)C(=O)c3ccccc3C2=O)cc1OC ZINC000217929131 JF In-Stock Unstable TNF 22 43 COc1cccc(/C=C/NC(=O)NC(c2ccccc2)c2ccccc2)c1 ZINC000217929146 FJ For-Sale Unstable MTNR1A 34 41 COc1cccc(/C=C/NC(=O)NC(c2ccccc2)c2ccccc2)c1 ZINC000217929146 FJ For-Sale Unstable MTNR1B 40 41 CCC(CO)(CO)NC[C@@H](O)COc1ccccc1C ZINC000217929147 CC For-Sale Unstable ADRB2 43 63 CCC(CO)(CO)NC[C@@H](O)COc1ccccc1C ZINC000217929147 CC For-Sale Unstable ADRB1 37 40 CCC(CO)(CO)NC[C@@H](O)COc1ccccc1C ZINC000217929147 CC For-Sale Unstable VDR 15 40 CCC(CO)(CO)NC[C@@H](O)COc1ccccc1C ZINC000217929147 CC For-Sale Unstable CASR 43 40 CCC(CO)(CO)NC[C@@H](O)COc1ccccc1C ZINC000217929147 CC For-Sale Unstable CYP2D6 25 55 O=C(NCC[C@@H](O)C1CCOCC1)Nc1cccc(Cl)c1 ZINC000217929155 DF In-Stock Unstable CASR 15 58 O=C(NCC[C@@H](O)C1CCOCC1)Nc1cccc(Cl)c1 ZINC000217929155 DF In-Stock Unstable EPHX2 21 52 N#Cc1ccc(Cl)cc1N1CCC[C@@H]2CCCC[C@H]21 ZINC000217929160 CI For-Sale Unstable AR 29 40 N#Cc1ccc(Cl)cc1N1CCC[C@@H]2CCCC[C@H]21 ZINC000217929160 CI For-Sale Unstable NOS3 15 40 COC(=O)c1ccnc(NC[C@@H]2CCC[C@@H](C)C2)c1 ZINC000217929173 CG On-Demand Unstable KDM5C 0 42 CC1(C)C[C@@H](NC(=O)/C=C/c2ccc3c(c2)OCO3)c2ccccc2O1 ZINC000217929176 FH In-Stock Unstable PLM1_PLAFA 15 45 CC1(C)C[C@@H](NC(=O)/C=C/c2ccc3c(c2)OCO3)c2ccccc2O1 ZINC000217929176 FH In-Stock Unstable DYRK2 45 34 Cc1noc2nc(C(C)C)cc(C(=O)Nc3c(C(C)C)cccc3C(C)C)c12 ZINC000217929182 GK On-Demand Unstable SOAT1 42 37 CCC(CO)(CO)NC[C@H](O)COc1ccccc1C ZINC000217929228 CC For-Sale Unstable ADRB2 43 63 CCC(CO)(CO)NC[C@H](O)COc1ccccc1C ZINC000217929228 CC For-Sale Unstable ADRB1 37 40 CCC(CO)(CO)NC[C@H](O)COc1ccccc1C ZINC000217929228 CC For-Sale Unstable VDR 15 40 CCC(CO)(CO)NC[C@H](O)COc1ccccc1C ZINC000217929228 CC For-Sale Unstable CASR 43 40 CCC(CO)(CO)NC[C@H](O)COc1ccccc1C ZINC000217929228 CC For-Sale Unstable CYP2D6 25 55 N#Cc1ccc(Cl)cc1N1CCC[C@H]2CCCC[C@H]21 ZINC000217929237 CI For-Sale Unstable AR 29 40 N#Cc1ccc(Cl)cc1N1CCC[C@H]2CCCC[C@H]21 ZINC000217929237 CI For-Sale Unstable NOS3 15 40 COC(=O)C[C@H](c1ccc(OC)c(OC)c1OC)c1c(O)c2ccccc2oc1=O ZINC000217929244 HG In-Stock Unstable NQO1 48 50 COC(=O)c1ccnc(NC[C@H]2CCC[C@@H](C)C2)c1 ZINC000217929247 CG On-Demand Unstable KDM5C 0 42 COc1ccc(CNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217929251 DG For-Sale Unstable CYP1B1 37 40 COc1ccc(CNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217929251 DG For-Sale Unstable TRPV1 23 47 COc1ccc(CNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217929251 DG For-Sale Unstable MMP13 26 45 COc1ccc(CNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217929251 DG For-Sale Unstable AHR 28 42 COc1ccc(CNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217929251 DG For-Sale Unstable ROCK1 29 41 COc1ccc(CNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217929251 DG For-Sale Unstable MTNR1A 96 50 COc1ccc(CNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217929251 DG For-Sale Unstable MTNR1B 89 50 COc1ccc(CNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217929251 DG For-Sale Unstable CYP1A1 26 43 COc1ccc(CNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217929251 DG For-Sale Unstable ROCK2 32 43 COc1ccc(CNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217929251 DG For-Sale Unstable NR1H4 25 40 COc1ccc(CNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217929251 DG For-Sale Unstable CA9 15 41 COc1ccc(CNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217929251 DG For-Sale Unstable U38 0 44 COc1ccc(CNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217929251 DG For-Sale Unstable PDS 46 41 CC1(C)C[C@H](NC(=O)/C=C/c2ccc3c(c2)OCO3)c2ccccc2O1 ZINC000217929260 FH In-Stock Unstable PLM1_PLAFA 15 45 CC1(C)C[C@H](NC(=O)/C=C/c2ccc3c(c2)OCO3)c2ccccc2O1 ZINC000217929260 FH In-Stock Unstable DYRK2 45 34 CCN(Cc1cccc(/C=C\C(=O)O)c1)Cc1ccco1 ZINC000217929264 CG For-Sale Unstable AKR1C3 37 40 Cc1cc(Cl)ccc1NC(=O)c1cc(C(C)C)nc2onc(C)c12 ZINC000217929280 EJ On-Demand Unstable H9CNL0_SPOEX 0 45 CC[C@@H](CCO)NC(=O)[C@@H](N)CCCOC ZINC000217929318 BC For-Sale Unstable DPP7 35 40 CCC(CO)(CO)NC[C@@H](O)COc1ccccc1 ZINC000217929331 CC For-Sale Unstable ADRB2 72 60 CCC(CO)(CO)NC[C@@H](O)COc1ccccc1 ZINC000217929331 CC For-Sale Unstable ADRB1 72 46 CCC(CO)(CO)NC[C@@H](O)COc1ccccc1 ZINC000217929331 CC For-Sale Unstable ADRB3 44 43 CCC(CO)(CO)NC[C@@H](O)COc1ccccc1 ZINC000217929331 CC For-Sale Unstable CASR 42 58 CCC(CO)(CO)NC[C@@H](O)COc1ccccc1 ZINC000217929331 CC For-Sale Unstable CYP2D6 24 51 CCC(CO)(CO)NC[C@@H](O)COc1ccccc1 ZINC000217929331 CC For-Sale Unstable ABCB1 18 40 CCC(CO)(CO)NC[C@@H](O)COc1ccccc1 ZINC000217929331 CC For-Sale Unstable PDS 50 37 COC(=O)c1ccnc(NC[C@@H]2CCC[C@H](C)C2)c1 ZINC000217929340 CG On-Demand Unstable KDM5C 0 42 COC(=O)C[C@@H](c1ccc(OC)c(OC)c1OC)c1c(O)c2ccccc2oc1=O ZINC000217929342 HG In-Stock Unstable NQO1 48 50 CC1(C)OB(c2ccc(F)c(-c3ccc(S(N)(=O)=O)cc3)c2)OC1(C)C ZINC000217929345 GE For-Sale Unstable PTGS2 69 49 CC1(C)OB(c2ccc(F)c(-c3ccc(S(N)(=O)=O)cc3)c2)OC1(C)C ZINC000217929345 GE For-Sale Unstable CA7 16 44 CC1(C)OB(c2ccc(F)c(-c3ccc(S(N)(=O)=O)cc3)c2)OC1(C)C ZINC000217929345 GE For-Sale Unstable CA9 17 51 CC1(C)OB(c2ccc(F)c(-c3ccc(S(N)(=O)=O)cc3)c2)OC1(C)C ZINC000217929345 GE For-Sale Unstable CA15 20 44 COc1cccc(/C=C/NC(=O)N2CCN(C(C)=O)CC2)c1 ZINC000217929357 DD For-Sale Unstable DRD4 42 32 COc1cccc(/C=C/NC(=O)N2CCN(C(C)=O)CC2)c1 ZINC000217929357 DD For-Sale Unstable CYP1B1 20 41 COc1cccc(/C=C/NC(=O)N2CCN(C(C)=O)CC2)c1 ZINC000217929357 DD For-Sale Unstable MTNR1A 37 43 COc1cccc(/C=C/NC(=O)N2CCN(C(C)=O)CC2)c1 ZINC000217929357 DD For-Sale Unstable MTNR1B 42 43 COc1cccc(/C=C/NC(=O)N2CCN(C(C)=O)CC2)c1 ZINC000217929357 DD For-Sale Unstable CYP1A1 19 41 CCOc1ccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217929365 FH In-Stock Unstable EDNRB 35 41 CCOc1ccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217929365 FH In-Stock Unstable EDNRA 41 36 CCOc1ccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217929365 FH In-Stock Unstable PYGL 0 41 CCOc1ccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217929365 FH In-Stock Unstable DYRK2 53 35 O=C(O)/C=C\c1ccc(OCCN2CCCSCC2)cc1 ZINC000217929367 DF For-Sale Unstable ESR1 71 38 O=C(O)/C=C\c1ccc(OCCN2CCCSCC2)cc1 ZINC000217929367 DF For-Sale Unstable ESR2 50 38 O=C(O)/C=C\c1ccc(OCCN2CCCSCC2)cc1 ZINC000217929367 DF For-Sale Unstable LTA4H 60 44 O=C(O)/C=C\c1ccc(OCCN2CCCSCC2)cc1 ZINC000217929367 DF For-Sale Unstable HRH3 45 54 O=C(O)/C=C\c1ccc(OCCN2CCCSCC2)cc1 ZINC000217929367 DF For-Sale Unstable PSMB2 48 45 O=C(O)/C=C\c1ccc(OCCN2CCCSCC2)cc1 ZINC000217929367 DF For-Sale Unstable PSMB1 51 46 CC[C@H](CCO)NC(=O)[C@@H](N)CCCOC ZINC000217929395 BC For-Sale Unstable DPP7 35 40 CCC(CO)(CO)NC[C@H](O)COc1ccccc1 ZINC000217929405 CC For-Sale Unstable ADRB2 72 60 CCC(CO)(CO)NC[C@H](O)COc1ccccc1 ZINC000217929405 CC For-Sale Unstable ADRB1 72 46 CCC(CO)(CO)NC[C@H](O)COc1ccccc1 ZINC000217929405 CC For-Sale Unstable ADRB3 44 43 CCC(CO)(CO)NC[C@H](O)COc1ccccc1 ZINC000217929405 CC For-Sale Unstable CASR 42 58 CCC(CO)(CO)NC[C@H](O)COc1ccccc1 ZINC000217929405 CC For-Sale Unstable CYP2D6 24 51 CCC(CO)(CO)NC[C@H](O)COc1ccccc1 ZINC000217929405 CC For-Sale Unstable ABCB1 18 40 CCC(CO)(CO)NC[C@H](O)COc1ccccc1 ZINC000217929405 CC For-Sale Unstable PDS 50 37 COC(=O)c1ccnc(NC[C@H]2CCC[C@H](C)C2)c1 ZINC000217929426 CG On-Demand Unstable KDM5C 0 42 CCOc1ccc(NC(=O)NCC[C@H](O)C2CCOCC2)cc1 ZINC000217929433 DE In-Stock Unstable ADRB1 20 41 CCOc1ccc(NC(=O)NCC[C@H](O)C2CCOCC2)cc1 ZINC000217929433 DE In-Stock Unstable MTOR 41 35 O=C(/C=C\c1ccc(Cl)cc1)CCl ZINC000217929461 BG For-Sale Unstable F3 24 41 O=C(/C=C\c1ccc(Cl)cc1)CCl ZINC000217929461 BG For-Sale Unstable SSSIM 17 52 COc1cccc(/C=C/NC(=O)NCc2ccc3c(c2)OCO3)c1 ZINC000217929465 EF For-Sale Unstable PDE5A 0 42 COc1cccc(/C=C/NC(=O)NCc2ccc3c(c2)OCO3)c1 ZINC000217929465 EF For-Sale Unstable EDNRB 67 46 COc1cccc(/C=C/NC(=O)NCc2ccc3c(c2)OCO3)c1 ZINC000217929465 EF For-Sale Unstable EDNRA 57 37 COc1cccc(/C=C/NC(=O)NCc2ccc3c(c2)OCO3)c1 ZINC000217929465 EF For-Sale Unstable BMP1 56 42 COc1cccc(/C=C/NC(=O)NCc2ccc3c(c2)OCO3)c1 ZINC000217929465 EF For-Sale Unstable SCN9A 0 41 O=C(O)/C=C\c1ccccc1CN1CCC[C@H](CO)C1 ZINC000217929473 CD For-Sale Unstable SLC6A1 134 43 O=C(O)/C=C\c1ccccc1CN1CCC[C@H](CO)C1 ZINC000217929473 CD For-Sale Unstable PTGER2 29 42 O=C(O)/C=C\c1ccccc1CN1CCC[C@H](CO)C1 ZINC000217929473 CD For-Sale Unstable PTGER3 17 42 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccc2c(c1)OCO2 ZINC000217929478 FH In-Stock Unstable DRD3 18 58 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccc2c(c1)OCO2 ZINC000217929478 FH In-Stock Unstable MTNR1B 40 38 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccc2c(c1)OCO2 ZINC000217929478 FH In-Stock Unstable DYRK2 41 36 CC[C@@H](CCO)NC(=O)[C@H](N)CCCOC ZINC000217929480 BC For-Sale Unstable DPP7 35 40 C[C@@H](O)c1cc2n(n1)CCN(CCN1CCN(c3ccccc3)CC1)C2 ZINC000217929491 FD In-Stock Unstable HTR1A 40 45 C[C@@H](O)c1cc2n(n1)CCN(CCN1CCN(c3ccccc3)CC1)C2 ZINC000217929491 FD In-Stock Unstable DRD2 24 45 C[C@@H](O)c1cc2n(n1)CCN(CCN1CCN(c3ccccc3)CC1)C2 ZINC000217929491 FD In-Stock Unstable HTR2A 32 45 C[C@@H](O)c1cc2n(n1)CCN(CCN1CCN(c3ccccc3)CC1)C2 ZINC000217929491 FD In-Stock Unstable HTR7 62 40 CCOc1ccc(NC(=O)NCC[C@@H](O)C2CCOCC2)cc1 ZINC000217929506 DE In-Stock Unstable ADRB1 20 41 CCOc1ccc(NC(=O)NCC[C@@H](O)C2CCOCC2)cc1 ZINC000217929506 DE In-Stock Unstable MTOR 41 35 O=C(/C=C\c1ccc(Br)cc1)CCl ZINC000217929541 CG For-Sale Unstable SSSIM 16 50 O=C(/C=C\c1ccc(Br)cc1)CCl ZINC000217929541 CG For-Sale Unstable GPR183 0 43 CC[C@H](CCO)NC(=O)[C@H](N)CCCOC ZINC000217929550 BC For-Sale Unstable DPP7 35 40 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccc2c(c1)OCO2 ZINC000217929554 EG In-Stock Unstable KCNQ2 23 46 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccc2c(c1)OCO2 ZINC000217929554 EG In-Stock Unstable DYRK2 49 32 COc1cccc(/C=C/NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217929569 EE For-Sale Unstable CA2 89 52 COc1cccc(/C=C/NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217929569 EE For-Sale Unstable CA1 87 55 COc1cccc(/C=C/NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217929569 EE For-Sale Unstable CA7 41 44 COc1cccc(/C=C/NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217929569 EE For-Sale Unstable CA4 56 47 COc1cccc(/C=C/NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217929569 EE For-Sale Unstable CA14 38 43 COc1cccc(/C=C/NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217929569 EE For-Sale Unstable MTNR1A 26 46 COc1cccc(/C=C/NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217929569 EE For-Sale Unstable MTNR1B 30 46 COc1cccc(/C=C/NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217929569 EE For-Sale Unstable CA12 79 55 COc1cccc(/C=C/NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217929569 EE For-Sale Unstable CA9 87 47 COc1cccc(/C=C/NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217929569 EE For-Sale Unstable UREA_CANEN 35 54 COc1cccc(/C=C/NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217929569 EE For-Sale Unstable IDO1 30 41 COc1cccc(/C=C/NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217929569 EE For-Sale Unstable NCE103 50 40 COc1cccc(/C=C/NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217929569 EE For-Sale Unstable MTCA1 60 55 COc1cccc(/C=C/NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217929569 EE For-Sale Unstable P96878_MYCTU 73 55 C[C@H](O)c1cc2n(n1)CCN(CCN1CCN(c3ccccc3)CC1)C2 ZINC000217929578 FD In-Stock Unstable HTR1A 40 45 C[C@H](O)c1cc2n(n1)CCN(CCN1CCN(c3ccccc3)CC1)C2 ZINC000217929578 FD In-Stock Unstable DRD2 24 45 C[C@H](O)c1cc2n(n1)CCN(CCN1CCN(c3ccccc3)CC1)C2 ZINC000217929578 FD In-Stock Unstable HTR2A 32 45 C[C@H](O)c1cc2n(n1)CCN(CCN1CCN(c3ccccc3)CC1)C2 ZINC000217929578 FD In-Stock Unstable HTR7 62 40 O=C(O)/C=C\c1ccc(CN2CCC[C@H](CO)C2)cc1 ZINC000217929581 CD For-Sale Unstable SLC6A1 55 33 O=C(O)/C=C\c1ccc(CN2CCC[C@H](CO)C2)cc1 ZINC000217929581 CD For-Sale Unstable SIGMAR1 23 46 O=C(NC[C@@H]1CCCN2CCCC[C@H]12)c1cc2c(Cl)cccc2[nH]1 ZINC000217929608 EH In-Stock Unstable PYGL 40 36 CCc1ccc(/C=C\C(=O)CCl)cc1 ZINC000217929618 BG For-Sale Unstable SSSIM 15 47 CC[C@@H](CCO)NC(=O)[C@@H](N)c1cccs1 ZINC000217929652 BD For-Sale Unstable CTSC 42 38 Cc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217929662 EG In-Stock Unstable KCNQ2 21 43 Cc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217929662 EG In-Stock Unstable DYRK2 59 35 COc1cccc(/C=C/NC(=O)NCc2ccccc2)c1 ZINC000217929681 CG For-Sale Unstable DRD4 40 31 COc1cccc(/C=C/NC(=O)NCc2ccccc2)c1 ZINC000217929681 CG For-Sale Unstable HRH2 15 40 COc1cccc(/C=C/NC(=O)NCc2ccccc2)c1 ZINC000217929681 CG For-Sale Unstable ANPEP 23 46 COc1cccc(/C=C/NC(=O)NCc2ccccc2)c1 ZINC000217929681 CG For-Sale Unstable CYP1B1 22 40 COc1cccc(/C=C/NC(=O)NCc2ccccc2)c1 ZINC000217929681 CG For-Sale Unstable G6PC 25 44 COc1cccc(/C=C/NC(=O)NCc2ccccc2)c1 ZINC000217929681 CG For-Sale Unstable MMP13 26 40 COc1cccc(/C=C/NC(=O)NCc2ccccc2)c1 ZINC000217929681 CG For-Sale Unstable ROCK1 32 41 COc1cccc(/C=C/NC(=O)NCc2ccccc2)c1 ZINC000217929681 CG For-Sale Unstable MTNR1A 79 48 COc1cccc(/C=C/NC(=O)NCc2ccccc2)c1 ZINC000217929681 CG For-Sale Unstable MTNR1B 77 48 COc1cccc(/C=C/NC(=O)NCc2ccccc2)c1 ZINC000217929681 CG For-Sale Unstable CYP1A1 16 40 COc1cccc(/C=C/NC(=O)NCc2ccccc2)c1 ZINC000217929681 CG For-Sale Unstable ROCK2 38 46 COc1cccc(/C=C/NC(=O)NCc2ccccc2)c1 ZINC000217929681 CG For-Sale Unstable AKR1C3 17 40 COc1cccc(/C=C/NC(=O)NCc2ccccc2)c1 ZINC000217929681 CG For-Sale Unstable PDS 77 48 CC(C)(C)OC(=O)Nc1ccc(C2CC2)c2ccccc12 ZINC000217929683 CK In-Stock Unstable CCR8 66 34 CCOc1ccc(/C=C\C(=O)CCl)cc1 ZINC000217929698 BF For-Sale Unstable AHR 20 48 O=C(O)/C=C\c1ccc(CN2CCC[C@H](CO)C2)c(F)c1 ZINC000217929701 CE For-Sale Unstable SLC6A1 63 34 COc1ccc(CCCNC(=O)C[C@H]2CN(C)CCN2C)cc1 ZINC000217929704 DD In-Stock Unstable BMP1 50 36 COc1ccc(CCCNC(=O)C[C@H]2CN(C)CCN2C)cc1 ZINC000217929704 DD In-Stock Unstable MMP13 24 40 COc1ccc(CCCNC(=O)C[C@H]2CN(C)CCN2C)cc1 ZINC000217929704 DD In-Stock Unstable MTNR1A 39 41 COc1ccc(CCCNC(=O)C[C@H]2CN(C)CCN2C)cc1 ZINC000217929704 DD In-Stock Unstable MTNR1B 32 41 COc1ccc(CCCNC(=O)C[C@H]2CN(C)CCN2C)cc1 ZINC000217929704 DD In-Stock Unstable MMP3 32 40 COc1ccc(CCCNC(=O)C[C@H]2CN(C)CCN2C)cc1 ZINC000217929704 DD In-Stock Unstable SLC6A5 20 40 COc1cc([C@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc(OC)c1OC ZINC000217929715 KH In-Stock Unstable CYP1B1 64 42 COc1cc([C@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc(OC)c1OC ZINC000217929715 KH In-Stock Unstable CYP1A1 48 42 COc1cc([C@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc(OC)c1OC ZINC000217929715 KH In-Stock Unstable CYP1A2 41 42 COc1cc([C@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc(OC)c1OC ZINC000217929715 KH In-Stock Unstable RORC 49 35 CC[C@H](CCO)NC(=O)[C@@H](N)c1cccs1 ZINC000217929731 BD For-Sale Unstable CTSC 42 38 Cc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217929736 EG In-Stock Unstable KCNQ2 21 43 Cc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217929736 EG In-Stock Unstable DYRK2 59 35 CNC(=O)c1cccc(N[C@@H]2C[C@@H](C)N(C)C[C@@H]2C)c1 ZINC000217929749 CE For-Sale Unstable KCNK3 47 33 CC(C)(C)c1ccc(NC(=O)NCC[C@H](O)C2CCOCC2)cc1 ZINC000217929787 EG In-Stock Unstable DOT1L 44 33 COc1cccc(/C=C/NC(=O)N[C@@H](C)C23CC4CC(CC(C4)C2)C3)c1 ZINC000217929791 FJ For-Sale Unstable EPHX2 22 46 COc1cc([C@@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc(OC)c1OC ZINC000217929800 KH In-Stock Unstable CYP1B1 64 42 COc1cc([C@@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc(OC)c1OC ZINC000217929800 KH In-Stock Unstable CYP1A1 48 42 COc1cc([C@@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc(OC)c1OC ZINC000217929800 KH In-Stock Unstable CYP1A2 41 42 COc1cc([C@@H](CC(=O)N2CCN(C)CC2)c2c(O)c(O)c(O)c3c(=O)cc(-c4ccccc4)oc23)cc(OC)c1OC ZINC000217929800 KH In-Stock Unstable RORC 49 35 CC[C@@H](CCO)NC(=O)[C@H](N)c1cccs1 ZINC000217929806 BD For-Sale Unstable CTSC 42 38 COc1ccc(CN2CCCC[C@H]2C)cc1/C=C\C(=O)O ZINC000217929816 CG For-Sale Unstable HRH3 41 40 CNC(=O)c1cccc(N[C@H]2C[C@@H](C)N(C)C[C@@H]2C)c1 ZINC000217929825 CE For-Sale Unstable KCNK3 47 33 Cc1noc2nc(C(C)C)cc(C(=O)Nc3ccc(S(=O)(=O)N4CCCCC4)cc3)c12 ZINC000217929840 II On-Demand Unstable LPL 50 40 Cc1noc2nc(C(C)C)cc(C(=O)Nc3ccc(S(=O)(=O)N4CCCCC4)cc3)c12 ZINC000217929840 II On-Demand Unstable TGM2 48 37 Cc1noc2nc(C(C)C)cc(C(=O)Nc3ccc(S(=O)(=O)N4CCCCC4)cc3)c12 ZINC000217929840 II On-Demand Unstable F13A1 63 41 Cc1noc2nc(C(C)C)cc(C(=O)Nc3ccc(S(=O)(=O)N4CCCCC4)cc3)c12 ZINC000217929840 II On-Demand Unstable MERTK 27 41 Cc1noc2nc(C(C)C)cc(C(=O)Nc3ccc(S(=O)(=O)N4CCCCC4)cc3)c12 ZINC000217929840 II On-Demand Unstable LIPG 20 40 CC(C)(C)c1ccc(NC(=O)NCC[C@@H](O)C2CCOCC2)cc1 ZINC000217929851 EG In-Stock Unstable DOT1L 44 33 CC1CCN(c2ccc([C@@H](C)NC(=O)/C=C/c3ccc4c(c3)OCO4)cc2)CC1 ZINC000217929852 GJ In-Stock Unstable KCNQ2 44 52 COc1cccc(/C=C/NC(=O)N[C@H](C)C23CC4CC(CC(C4)C2)C3)c1 ZINC000217929874 FJ For-Sale Unstable EPHX2 22 46 CC[C@H](CCO)NC(=O)[C@H](N)c1cccs1 ZINC000217929885 BD For-Sale Unstable CTSC 42 38 CC(C)S(=O)(=O)CC(=O)N1CCC[C@@H]1CN ZINC000217929893 BB On-Demand Unstable FAP 0 40 CNC(=O)c1cccc(N[C@@H]2C[C@H](C)N(C)C[C@@H]2C)c1 ZINC000217929909 CE For-Sale Unstable KCNK3 47 33 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCCCc1nc2ccccc2[nH]1 ZINC000217929910 JI In-Stock Unstable CYSP_TRYCR 0 41 COc1ccc(CN2CCCC[C@@H]2C)cc1/C=C\C(=O)O ZINC000217929916 CG For-Sale Unstable HRH3 38 40 CC1CCN(c2ccc([C@H](C)NC(=O)/C=C/c3ccc4c(c3)OCO4)cc2)CC1 ZINC000217929933 GJ In-Stock Unstable KCNQ2 44 52 COc1ccc(NC(=O)c2ccc(NC(=O)c3cc(C(C)C)nc4onc(C)c34)cc2)cc1 ZINC000217929951 IK On-Demand Unstable KCNK3 67 38 COc1ccc(NC(=O)c2ccc(NC(=O)c3cc(C(C)C)nc4onc(C)c34)cc2)cc1 ZINC000217929951 IK On-Demand Unstable KCNK9 52 35 COc1ccc(CCNC(=O)NCC[C@H](O)C2CCOCC2)cc1 ZINC000217929953 ED In-Stock Unstable MTNR1A 41 37 CC(C)S(=O)(=O)CC(=O)N1CCC[C@H]1CN ZINC000217929963 BB On-Demand Unstable FAP 0 40 COc1cccc(/C=C/NC(=O)Nc2cccc3c(O)cccc23)c1 ZINC000217929971 EI For-Sale Unstable TRPV1 21 45 COc1cccc(/C=C/NC(=O)Nc2cccc3c(O)cccc23)c1 ZINC000217929971 EI For-Sale Unstable MTNR1A 33 43 COc1cccc(/C=C/NC(=O)Nc2cccc3c(O)cccc23)c1 ZINC000217929971 EI For-Sale Unstable MTNR1B 33 43 CNC(=O)c1cccc(N[C@H]2C[C@H](C)N(C)C[C@@H]2C)c1 ZINC000217929986 CE For-Sale Unstable KCNK3 47 33 O=C(CCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCCCc1nc2ccccc2[nH]1 ZINC000217930011 JI In-Stock Unstable CYSP_TRYCR 0 41 C[C@@H]1CCCCN1Cc1ccc(/C=C\C(=O)O)cc1F ZINC000217930025 CG For-Sale Unstable GPR183 0 40 COc1ccc(CCNC(=O)NCC[C@@H](O)C2CCOCC2)cc1 ZINC000217930038 ED In-Stock Unstable MTNR1A 41 37 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)/C=C/c3ccc4c(c3)OCO4)cc2)C1 ZINC000217930056 GJ In-Stock Unstable KCNQ2 35 50 COc1cc(S(C)(=O)=O)ccc1B1OC(C)(C)C(C)(C)O1 ZINC000217930082 DD For-Sale Unstable PTGS2 18 40 COc1cccc(/C=C/NC(=O)Nc2ccc(O)cc2C)c1 ZINC000217930089 CH For-Sale Unstable MTNR1A 25 42 COc1cccc(/C=C/NC(=O)Nc2ccc(O)cc2C)c1 ZINC000217930089 CH For-Sale Unstable MTNR1B 28 42 C[C@H]1CCCCN1Cc1ccc(/C=C\C(=O)O)cc1F ZINC000217930103 CG For-Sale Unstable GPR183 0 40 CCOC(=O)c1ccc(NC(=O)c2cc(C(C)C)nc3onc(C)c23)cc1 ZINC000217930139 FI On-Demand Unstable F3 73 35 CCOC(=O)c1ccc(NC(=O)c2cc(C(C)C)nc3onc(C)c23)cc1 ZINC000217930139 FI On-Demand Unstable ACR 40 34 C[C@H](NC(=O)/C=C/c1ccc2c(c1)OCO2)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217930144 GJ In-Stock Unstable KCNQ2 35 50 C[C@H](NC(=O)/C=C/c1ccc2c(c1)OCO2)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217930144 GJ In-Stock Unstable SSTR3 42 35 C[C@H](NC(=O)/C=C/c1ccc2c(c1)OCO2)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217930144 GJ In-Stock Unstable RORC 37 42 COc1cccc(/C=C/NC(=O)N2CCOCC2)c1 ZINC000217930204 CD For-Sale Unstable DRD4 42 33 COc1cccc(/C=C/NC(=O)N2CCOCC2)c1 ZINC000217930204 CD For-Sale Unstable MTNR1A 30 40 COc1cccc(/C=C/NC(=O)N2CCOCC2)c1 ZINC000217930204 CD For-Sale Unstable MTNR1B 37 40 COc1cccc(/C=C/NC(=O)N2CCOCC2)c1 ZINC000217930204 CD For-Sale Unstable BRPF1 0 41 C[C@@H]1CN(CCOc2ccc(/C=C\C(=O)O)cc2)CCO1 ZINC000217930206 CD On-Demand Unstable HRH3 23 43 C[C@@H]1CN(CCOc2ccc(/C=C\C(=O)O)cc2)CCO1 ZINC000217930206 CD On-Demand Unstable PSMB2 47 38 C[C@@H]1CN(CCOc2ccc(/C=C\C(=O)O)cc2)CCO1 ZINC000217930206 CD On-Demand Unstable PSMB1 41 38 O=C(CCc1nc2ccccc2[nH]1)N[C@H]1CCC[C@H]1CO ZINC000217930247 CD On-Demand Unstable CYSP_TRYCR 0 41 O=C(CCc1nc2ccccc2[nH]1)N[C@H]1CCC[C@H]1CO ZINC000217930247 CD On-Demand Unstable ISPE 0 41 Cc1ccc2c(c1)[C@@H](NC(=O)/C=C/c1ccc3c(c1)OCO3)CC(C)(C)O2 ZINC000217930255 FI In-Stock Unstable DYRK2 46 35 CCC(CO)(CO)NC[C@@H](O)COCc1ccccc1 ZINC000217930278 CC For-Sale Unstable ADRB2 23 44 CCC(CO)(CO)NC[C@@H](O)COCc1ccccc1 ZINC000217930278 CC For-Sale Unstable CASR 37 57 C[C@H]1CN(CCOc2ccc(/C=C\C(=O)O)cc2)CCO1 ZINC000217930286 CD On-Demand Unstable HRH3 23 43 C[C@H]1CN(CCOc2ccc(/C=C\C(=O)O)cc2)CCO1 ZINC000217930286 CD On-Demand Unstable PSMB2 47 38 C[C@H]1CN(CCOc2ccc(/C=C\C(=O)O)cc2)CCO1 ZINC000217930286 CD On-Demand Unstable PSMB1 41 38 O=C(CCCCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCc1ccccn1 ZINC000217930297 JI In-Stock Unstable HTR7 15 48 O=C(CCCCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)NCc1ccccn1 ZINC000217930297 JI In-Stock Unstable SCN9A 0 44 COc1cccc(/C=C/NC(=O)NCC(=O)O)c1 ZINC000217930303 CD For-Sale Unstable DRD4 40 31 COc1cccc(/C=C/NC(=O)NCC(=O)O)c1 ZINC000217930303 CD For-Sale Unstable CYP1B1 29 42 COc1cccc(/C=C/NC(=O)NCC(=O)O)c1 ZINC000217930303 CD For-Sale Unstable AHR 23 43 COc1cccc(/C=C/NC(=O)NCC(=O)O)c1 ZINC000217930303 CD For-Sale Unstable MTNR1A 75 49 COc1cccc(/C=C/NC(=O)NCC(=O)O)c1 ZINC000217930303 CD For-Sale Unstable MTNR1B 72 49 COc1cccc(/C=C/NC(=O)NCC(=O)O)c1 ZINC000217930303 CD For-Sale Unstable CYP1A1 22 42 Cc1ccc2c(c1)[C@H](NC(=O)/C=C/c1ccc3c(c1)OCO3)CC(C)(C)O2 ZINC000217930331 FI In-Stock Unstable DYRK2 46 35 Cc1cccc(N2CCN(CC(=O)N3CCC[C@@H]3c3ccccn3)CC2)c1 ZINC000217930348 FF In-Stock Unstable HTR1A 40 46 Cc1cccc(N2CCN(CC(=O)N3CCC[C@@H]3c3ccccn3)CC2)c1 ZINC000217930348 FF In-Stock Unstable DRD4 28 48 Cc1cccc(N2CCN(CC(=O)N3CCC[C@@H]3c3ccccn3)CC2)c1 ZINC000217930348 FF In-Stock Unstable HTR2A 25 45 Cc1cccc(N2CCN(CC(=O)N3CCC[C@@H]3c3ccccn3)CC2)c1 ZINC000217930348 FF In-Stock Unstable HTR7 27 40 Cc1cccc(N2CCN(CC(=O)N3CCC[C@@H]3c3ccccn3)CC2)c1 ZINC000217930348 FF In-Stock Unstable PRCP 23 41 Cc1cccc(N2CCN(CC(=O)N3CCC[C@@H]3c3ccccn3)CC2)c1 ZINC000217930348 FF In-Stock Unstable CPT1A 99 38 C[C@@H](N[C@@](C)(CO)c1ccccc1)C(=O)OC(C)(C)C ZINC000217930356 CE For-Sale Unstable AMY2 62 37 C[C@@H](N[C@@](C)(CO)c1ccccc1)C(=O)OC(C)(C)C ZINC000217930356 CE For-Sale Unstable KIF11 20 43 CCC(CO)(CO)NC[C@H](O)COCc1ccccc1 ZINC000217930363 CC For-Sale Unstable ADRB2 23 44 CCC(CO)(CO)NC[C@H](O)COCc1ccccc1 ZINC000217930363 CC For-Sale Unstable CASR 37 57 CCCCN(CC)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217930374 CG For-Sale Unstable ACHE 0 47 CCCCN(CC)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217930374 CG For-Sale Unstable BCHE 0 45 CCCCN(CC)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217930374 CG For-Sale Unstable TUBB1 42 37 CCCCN(CC)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217930374 CG For-Sale Unstable AKR1C3 29 44 O=C(CCCCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCc1ccccn1 ZINC000217930384 JI In-Stock Unstable HTR7 15 48 O=C(CCCCCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)NCc1ccccn1 ZINC000217930384 JI In-Stock Unstable SCN9A 0 44 COc1cccc(/C=C/NC(=O)N(CCO)CCO)c1 ZINC000217930409 CC For-Sale Unstable DRD4 40 30 COc1cccc(/C=C/NC(=O)N(CCO)CCO)c1 ZINC000217930409 CC For-Sale Unstable CYP1B1 20 41 COc1cccc(/C=C/NC(=O)N(CCO)CCO)c1 ZINC000217930409 CC For-Sale Unstable MTNR1A 48 45 COc1cccc(/C=C/NC(=O)N(CCO)CCO)c1 ZINC000217930409 CC For-Sale Unstable MTNR1B 46 45 COc1cccc(/C=C/NC(=O)N(CCO)CCO)c1 ZINC000217930409 CC For-Sale Unstable CYP1A1 18 41 COc1cccc(/C=C/NC(=O)N(CCO)CCO)c1 ZINC000217930409 CC For-Sale Unstable ROCK2 19 42 CCOc1ccc(/C=C\c2csc(N)n2)cc1 ZINC000217930425 BG For-Sale Unstable AHR 25 47 Cc1cccc(N2CCN(CC(=O)N3CCC[C@H]3c3ccccn3)CC2)c1 ZINC000217930431 FF In-Stock Unstable HTR1A 40 46 Cc1cccc(N2CCN(CC(=O)N3CCC[C@H]3c3ccccn3)CC2)c1 ZINC000217930431 FF In-Stock Unstable DRD4 28 48 Cc1cccc(N2CCN(CC(=O)N3CCC[C@H]3c3ccccn3)CC2)c1 ZINC000217930431 FF In-Stock Unstable HTR2A 25 45 Cc1cccc(N2CCN(CC(=O)N3CCC[C@H]3c3ccccn3)CC2)c1 ZINC000217930431 FF In-Stock Unstable HTR7 27 40 Cc1cccc(N2CCN(CC(=O)N3CCC[C@H]3c3ccccn3)CC2)c1 ZINC000217930431 FF In-Stock Unstable PRCP 23 41 Cc1cccc(N2CCN(CC(=O)N3CCC[C@H]3c3ccccn3)CC2)c1 ZINC000217930431 FF In-Stock Unstable CPT1A 99 38 C[C@H](N[C@@](C)(CO)c1ccccc1)C(=O)OC(C)(C)C ZINC000217930435 CE For-Sale Unstable AMY2 62 37 C[C@H](N[C@@](C)(CO)c1ccccc1)C(=O)OC(C)(C)C ZINC000217930435 CE For-Sale Unstable KIF11 20 43 Cc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)/C=C/c1ccc2c(c1)OCO2 ZINC000217930440 FI In-Stock Unstable DYRK2 40 35 CCCCN(CC)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217930490 CG For-Sale Unstable ACHE 23 45 CCCCN(CC)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217930490 CG For-Sale Unstable PTGER2 29 41 CCCCN(CC)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217930490 CG For-Sale Unstable PTGER4 0 41 COc1ccc(/C=C\c2csc(N)n2)cc1 ZINC000217930504 BF For-Sale Unstable CYP1B1 48 47 COc1ccc(/C=C\c2csc(N)n2)cc1 ZINC000217930504 BF For-Sale Unstable AHR 39 47 COc1ccc(/C=C\c2csc(N)n2)cc1 ZINC000217930504 BF For-Sale Unstable CYP1A1 34 47 COc1ccc(/C=C\c2csc(N)n2)cc1 ZINC000217930504 BF For-Sale Unstable MAPT 16 60 COc1cccc(/C=C/NC(=O)N[C@@H](C)C(=O)O)c1 ZINC000217930508 CD For-Sale Unstable MTNR1A 33 42 COc1cccc(/C=C/NC(=O)N[C@@H](C)C(=O)O)c1 ZINC000217930508 CD For-Sale Unstable MTNR1B 36 42 Cc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)/C=C/c1ccc2c(c1)OCO2 ZINC000217930520 FI In-Stock Unstable DYRK2 40 35 C[C@@H](N[C@](C)(CO)c1ccccc1)C(=O)OC(C)(C)C ZINC000217930522 CE For-Sale Unstable AMY2 62 37 C[C@@H](N[C@](C)(CO)c1ccccc1)C(=O)OC(C)(C)C ZINC000217930522 CE For-Sale Unstable KIF11 20 43 O=C(NCC[C@H](O)C1CCOCC1)Nc1ccccc1C(F)(F)F ZINC000217930543 EG In-Stock Unstable RBP4 62 34 CN(C)CCN(C)C1CCN(C(=O)[C@H](O)c2ccc3ccccc3c2)CC1 ZINC000217930554 FE In-Stock Unstable TRY2_BOVIN 44 33 CN(C)CCN(C)C1CCN(C(=O)[C@H](O)c2ccc3ccccc3c2)CC1 ZINC000217930554 FE In-Stock Unstable UTS2 54 43 C[C@H]1CN(C)[C@@H](C)C[C@@H]1Nc1ccc2c(c1)NC(=O)CO2 ZINC000217930571 CE For-Sale Unstable NR3C2 35 42 Nc1nc(/C=C\c2c[nH]c3cc([N+](=O)[O-])ccc23)cs1 ZINC000217930590 CG For-Sale Unstable TDO2 0 47 COc1cccc(/C=C/NC(=O)N[C@H](C)C(=O)O)c1 ZINC000217930591 CD For-Sale Unstable MTNR1A 33 42 COc1cccc(/C=C/NC(=O)N[C@H](C)C(=O)O)c1 ZINC000217930591 CD For-Sale Unstable MTNR1B 36 42 C[C@H](N[C@](C)(CO)c1ccccc1)C(=O)OC(C)(C)C ZINC000217930601 CE For-Sale Unstable AMY2 62 37 C[C@H](N[C@](C)(CO)c1ccccc1)C(=O)OC(C)(C)C ZINC000217930601 CE For-Sale Unstable KIF11 20 43 O=C(O)/C=C\c1cccc(CN2CCS(=O)(=O)CC2)c1 ZINC000217930602 CD For-Sale Unstable SIGMAR1 29 45 O=C(NCC[C@@H](O)C1CCOCC1)Nc1ccccc1C(F)(F)F ZINC000217930627 EG In-Stock Unstable RBP4 62 34 COc1ccc2c(c1)[C@@H](NC(=O)/C=C/c1ccc3c(c1)OCO3)CC(C)(C)O2 ZINC000217930634 GH In-Stock Unstable EDNRB 46 38 COc1ccc2c(c1)[C@@H](NC(=O)/C=C/c1ccc3c(c1)OCO3)CC(C)(C)O2 ZINC000217930634 GH In-Stock Unstable EDNRA 48 37 COc1ccc2c(c1)[C@@H](NC(=O)/C=C/c1ccc3c(c1)OCO3)CC(C)(C)O2 ZINC000217930634 GH In-Stock Unstable DYRK2 41 39 Cc1nc([C@@H]2CCCN(C(=O)c3csc(-c4cccs4)n3)C2)no1 ZINC000217930682 FH In-Stock Unstable ETHR 53 41 Cc1nc([C@@H]2CCCN(C(=O)c3csc(-c4cccs4)n3)C2)no1 ZINC000217930682 FH In-Stock Unstable TRPC6 46 33 CCCCSCC(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217930684 BD On-Demand Unstable EST1_PIG 43 37 COc1cccc(/C=C/NC(=O)NCCCCCC(=O)O)c1 ZINC000217930705 DF For-Sale Unstable MTNR1A 76 47 COc1cccc(/C=C/NC(=O)NCCCCCC(=O)O)c1 ZINC000217930705 DF For-Sale Unstable MTNR1B 73 47 COc1cccc(/C=C/NC(=O)NCCCCCC(=O)O)c1 ZINC000217930705 DF For-Sale Unstable HDAC9 32 40 COc1cccc(/C=C/NC(=O)NCCCCCC(=O)O)c1 ZINC000217930705 DF For-Sale Unstable HDAC7 30 40 COc1ccc2c(c1)[C@H](NC(=O)/C=C/c1ccc3c(c1)OCO3)CC(C)(C)O2 ZINC000217930709 GH In-Stock Unstable EDNRB 46 38 COc1ccc2c(c1)[C@H](NC(=O)/C=C/c1ccc3c(c1)OCO3)CC(C)(C)O2 ZINC000217930709 GH In-Stock Unstable EDNRA 48 37 COc1ccc2c(c1)[C@H](NC(=O)/C=C/c1ccc3c(c1)OCO3)CC(C)(C)O2 ZINC000217930709 GH In-Stock Unstable DYRK2 41 39 COc1ccc(/C=C\c2csc(N)n2)cc1C ZINC000217930747 BG For-Sale Unstable TUBB1 33 43 O=C(NCC[C@H](O)C1CCOCC1)Nc1cccc(C(F)(F)F)c1 ZINC000217930754 EG In-Stock Unstable CCR3 22 48 O=C(NCC[C@H](O)C1CCOCC1)Nc1cccc(C(F)(F)F)c1 ZINC000217930754 EG In-Stock Unstable RAF1 20 42 O=C(NCC[C@H](O)C1CCOCC1)Nc1cccc(C(F)(F)F)c1 ZINC000217930754 EG In-Stock Unstable EPHX2 29 46 O=C(NCC[C@H](O)C1CCOCC1)Nc1cccc(C(F)(F)F)c1 ZINC000217930754 EG In-Stock Unstable Q8MMZ8_EIMTE 0 42 CCCCSCC(=O)N[C@H]1CCC[C@@H]1CO ZINC000217930758 BD For-Sale Unstable EST1_PIG 43 37 Cc1nc([C@H]2CCCN(C(=O)c3csc(-c4cccs4)n3)C2)no1 ZINC000217930782 FH In-Stock Unstable ETHR 53 41 Cc1nc([C@H]2CCCN(C(=O)c3csc(-c4cccs4)n3)C2)no1 ZINC000217930782 FH In-Stock Unstable TRPC6 46 33 CCN(CC)S(=O)(=O)c1ccc(Cl)c(NC(=O)c2cc(C(C)C)nc3onc(C)c23)c1 ZINC000217930783 JJ On-Demand Unstable MURF 0 40 Cc1cc(CO[C@H]2C[C@H](C)CC[C@H]2C(C)C)oc1C(=O)O ZINC000217930798 CI For-Sale Unstable SERPINE1 40 40 CC[C@H](CCO)NC(=O)[C@@H](C)[C@@H](C)N ZINC000217930802 BC For-Sale Unstable ENPEP 51 32 COc1cccc(/C=C/NC(=O)N[C@H](C(=O)O)C(C)C)c1 ZINC000217930823 CE For-Sale Unstable MTNR1A 30 41 COc1cccc(/C=C/NC(=O)N[C@H](C(=O)O)C(C)C)c1 ZINC000217930823 CE For-Sale Unstable MTNR1B 35 41 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)/C=C/c1ccc2c(c1)OCO2 ZINC000217930833 GH In-Stock Unstable EDNRB 57 39 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)/C=C/c1ccc2c(c1)OCO2 ZINC000217930833 GH In-Stock Unstable EDNRA 55 38 CCCCSCC(=O)N[C@@H]1CCC[C@H]1CO ZINC000217930834 BD For-Sale Unstable EST1_PIG 43 37 O=C(NCC[C@@H](O)C1CCOCC1)Nc1cccc(C(F)(F)F)c1 ZINC000217930837 EG In-Stock Unstable CCR3 22 48 O=C(NCC[C@@H](O)C1CCOCC1)Nc1cccc(C(F)(F)F)c1 ZINC000217930837 EG In-Stock Unstable RAF1 20 42 O=C(NCC[C@@H](O)C1CCOCC1)Nc1cccc(C(F)(F)F)c1 ZINC000217930837 EG In-Stock Unstable EPHX2 29 46 O=C(NCC[C@@H](O)C1CCOCC1)Nc1cccc(C(F)(F)F)c1 ZINC000217930837 EG In-Stock Unstable Q8MMZ8_EIMTE 0 42 Cc1cc(CO[C@H]2C[C@@H](C)CC[C@H]2C(C)C)oc1C(=O)O ZINC000217930875 CI For-Sale Unstable SERPINE1 40 40 COc1cccc(/C=C/NC(=O)N[C@@H](C(=O)O)C(C)C)c1 ZINC000217930897 CE For-Sale Unstable MTNR1A 30 41 COc1cccc(/C=C/NC(=O)N[C@@H](C(=O)O)C(C)C)c1 ZINC000217930897 CE For-Sale Unstable MTNR1B 35 41 CCCCSCC(=O)N[C@H]1CCC[C@H]1CO ZINC000217930913 BD For-Sale Unstable EST1_PIG 43 37 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)/C=C/c1ccc2c(c1)OCO2 ZINC000217930923 GH In-Stock Unstable EDNRB 44 39 O=C(c1cc[nH]n1)N1CCC[C@@H](Cn2ccnc2)C1 ZINC000217930932 CD In-Stock Unstable CAMC 0 44 CC[C@H](CCO)NC(=O)[C@H](C)[C@@H](C)N ZINC000217930974 BC For-Sale Unstable ENPEP 51 32 Cc1noc2nc(C(C)C)cc(C(=O)Nc3cccc(S(=O)(=O)N(C)C)c3)c12 ZINC000217931003 HG On-Demand Unstable KCNK3 43 34 Cc1noc2nc(C(C)C)cc(C(=O)Nc3cccc(S(=O)(=O)N(C)C)c3)c12 ZINC000217931003 HG On-Demand Unstable KCNK9 43 34 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cc(-c2ccccc2)n[nH]1 ZINC000217931004 HG For-Sale Unstable TACR3 21 46 COc1cccc(/C=C/NC(=O)NCCCC(=O)O)c1 ZINC000217931005 CD For-Sale Unstable DRD4 41 31 COc1cccc(/C=C/NC(=O)NCCCC(=O)O)c1 ZINC000217931005 CD For-Sale Unstable MTNR1A 83 49 COc1cccc(/C=C/NC(=O)NCCCC(=O)O)c1 ZINC000217931005 CD For-Sale Unstable MTNR1B 79 49 O=C(c1cc[nH]n1)N1CCC[C@H](Cn2ccnc2)C1 ZINC000217931029 CD In-Stock Unstable CAMC 0 44 CC[C@@H](NC(=O)/C=C/c1ccc2c(c1)OCO2)c1ccc(C)c(C)c1 ZINC000217931051 EI In-Stock Unstable KCNQ2 22 46 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cc(-c2ccccc2)n[nH]1 ZINC000217931089 HG For-Sale Unstable TACR3 21 46 COc1cccc(/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O)c1 ZINC000217931106 DE For-Sale Unstable FOLH1 62 44 COc1cccc(/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O)c1 ZINC000217931106 DE For-Sale Unstable MME 23 40 COc1cccc(/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O)c1 ZINC000217931106 DE For-Sale Unstable ANPEP 37 50 COc1cccc(/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O)c1 ZINC000217931106 DE For-Sale Unstable CTSK 26 42 COc1cccc(/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O)c1 ZINC000217931106 DE For-Sale Unstable CTSL 15 42 COc1cccc(/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O)c1 ZINC000217931106 DE For-Sale Unstable MTNR1A 34 41 COc1cccc(/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O)c1 ZINC000217931106 DE For-Sale Unstable MTNR1B 38 41 COc1cccc(/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O)c1 ZINC000217931106 DE For-Sale Unstable CAPN1 45 39 COc1cccc(/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O)c1 ZINC000217931106 DE For-Sale Unstable FPR1 74 41 COc1cccc(/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O)c1 ZINC000217931106 DE For-Sale Unstable NPR 42 35 COc1cccc(/C=C/NC(=O)N[C@@H](CC(C)C)C(=O)O)c1 ZINC000217931106 DE For-Sale Unstable CPG2 0 43 CC[C@H](NC(=O)/C=C/c1ccc2c(c1)OCO2)c1ccc(C)c(C)c1 ZINC000217931122 EI In-Stock Unstable KCNQ2 22 46 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cc(-c2ccccc2)n[nH]1 ZINC000217931161 HG For-Sale Unstable TACR3 21 46 CCN(CCO)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217931167 CD For-Sale Unstable SQLE 40 31 COc1cccc(/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O)c1 ZINC000217931183 DE For-Sale Unstable FOLH1 62 44 COc1cccc(/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O)c1 ZINC000217931183 DE For-Sale Unstable MME 23 40 COc1cccc(/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O)c1 ZINC000217931183 DE For-Sale Unstable ANPEP 37 50 COc1cccc(/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O)c1 ZINC000217931183 DE For-Sale Unstable CTSK 26 42 COc1cccc(/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O)c1 ZINC000217931183 DE For-Sale Unstable CTSL 15 42 COc1cccc(/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O)c1 ZINC000217931183 DE For-Sale Unstable MTNR1A 34 41 COc1cccc(/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O)c1 ZINC000217931183 DE For-Sale Unstable MTNR1B 38 41 COc1cccc(/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O)c1 ZINC000217931183 DE For-Sale Unstable CAPN1 45 39 COc1cccc(/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O)c1 ZINC000217931183 DE For-Sale Unstable FPR1 74 41 COc1cccc(/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O)c1 ZINC000217931183 DE For-Sale Unstable NPR 42 35 COc1cccc(/C=C/NC(=O)N[C@H](CC(C)C)C(=O)O)c1 ZINC000217931183 DE For-Sale Unstable CPG2 0 43 CC[C@@H](NC(=O)/C=C/c1ccc2c(c1)OCO2)c1ccc(C)cc1C ZINC000217931216 EI In-Stock Unstable DYRK2 45 34 COc1cc(CN2CCN3CCN(C)C[C@@H]3C2)ccc1F ZINC000217931218 CD In-Stock Unstable DRD4 15 41 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cc(-c2ccccc2)n[nH]1 ZINC000217931249 HG For-Sale Unstable TACR3 21 46 COc1cccc(/C=C/NC(=O)N[C@@H](CCSC)C(=O)O)c1 ZINC000217931277 DE For-Sale Unstable FPR1 40 44 COc1cccc(/C=C/NC(=O)N[C@@H](CCSC)C(=O)O)c1 ZINC000217931277 DE For-Sale Unstable CPG2 0 46 CC[C@H](NC(=O)/C=C/c1ccc2c(c1)OCO2)c1ccc(C)cc1C ZINC000217931290 EI In-Stock Unstable DYRK2 45 34 COc1ccc(/C=C\C(=O)O)cc1CN(CCO)CCO ZINC000217931300 CC For-Sale Unstable PTGER2 0 43 COc1ccc(/C=C\C(=O)O)cc1CN(CCO)CCO ZINC000217931300 CC For-Sale Unstable TUBB1 52 40 COc1ccc(/C=C\C(=O)O)cc1CN(CCO)CCO ZINC000217931300 CC For-Sale Unstable AKR1C3 30 41 COc1ccc(/C=C\C(=O)O)cc1CN(CCO)CCO ZINC000217931300 CC For-Sale Unstable ABCG2 17 42 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)C(c1ccccc1)c1ccccc1 ZINC000217931360 II For-Sale Unstable AGTR2 111 48 COc1cccc(/C=C/NC(=O)N[C@H](CCSC)C(=O)O)c1 ZINC000217931361 DE For-Sale Unstable FPR1 40 44 COc1cccc(/C=C/NC(=O)N[C@H](CCSC)C(=O)O)c1 ZINC000217931361 DE For-Sale Unstable CPG2 0 46 COc1ccc(CN(CCO)CCO)cc1/C=C\C(=O)O ZINC000217931394 CC For-Sale Unstable PTGER2 37 44 COc1ccc(CN(CCO)CCO)cc1/C=C\C(=O)O ZINC000217931394 CC For-Sale Unstable PTGER4 22 44 COc1ccc(CN(CCO)CCO)cc1/C=C\C(=O)O ZINC000217931394 CC For-Sale Unstable PTGER3 17 44 COc1ccc(CN(CCO)CCO)cc1/C=C\C(=O)O ZINC000217931394 CC For-Sale Unstable AKR1B10 30 40 CC[C@@H](NC(=O)/C=C/c1ccc2c(c1)OCO2)c1ccc(OC)c(OC)c1 ZINC000217931395 FH In-Stock Unstable KCNQ2 22 45 CC[C@@H](NC(=O)/C=C/c1ccc2c(c1)OCO2)c1ccc(OC)c(OC)c1 ZINC000217931395 FH In-Stock Unstable F3 19 41 CC[C@@H](NC(=O)/C=C/c1ccc2c(c1)OCO2)c1ccc(OC)c(OC)c1 ZINC000217931395 FH In-Stock Unstable PDE10A 24 45 CC[C@@H](NC(=O)/C=C/c1ccc2c(c1)OCO2)c1ccc(OC)c(OC)c1 ZINC000217931395 FH In-Stock Unstable DYRK2 47 35 CC[C@@H](NC(=O)/C=C/c1ccc2c(c1)OCO2)c1ccc(OC)c(OC)c1 ZINC000217931395 FH In-Stock Unstable RORC 32 40 CC(C)(C)OC(=O)N1CCC(CN)(S(C)(=O)=O)CC1 ZINC000217931411 CC In-Stock Unstable GPR119 30 41 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)C(c1ccccc1)c1ccccc1 ZINC000217931438 II For-Sale Unstable AGTR2 111 48 Cc1noc2nc(C(C)C)cc(C(=O)Nc3ccccc3-c3nc4ccccc4[nH]3)c12 ZINC000217931456 HK On-Demand Unstable NR2E3 63 36 Cc1noc2nc(C(C)C)cc(C(=O)Nc3ccccc3-c3nc4ccccc4[nH]3)c12 ZINC000217931456 HK On-Demand Unstable SHH 23 41 Cc1noc2nc(C(C)C)cc(C(=O)Nc3ccccc3-c3nc4ccccc4[nH]3)c12 ZINC000217931456 HK On-Demand Unstable STK33 55 39 CN(C)C(=O)NCC(=O)NCCc1cccnc1 ZINC000217931463 CC In-Stock Unstable TBXAS1 38 42 CN(C)C(=O)NCC(=O)NCCc1cccnc1 ZINC000217931463 CC In-Stock Unstable PTAFR 30 45 CN(C)C(=O)NCC(=O)NCCc1cccnc1 ZINC000217931463 CC In-Stock Unstable NAMPT 31 40 COc1cccc(/C=C/NC(=O)N[C@@H](C)c2ccc(OC)c(OC)c2)c1 ZINC000217931469 FH For-Sale Unstable MTNR1A 17 43 CC[C@H](NC(=O)/C=C/c1ccc2c(c1)OCO2)c1ccc(OC)c(OC)c1 ZINC000217931471 FH In-Stock Unstable KCNQ2 22 45 CC[C@H](NC(=O)/C=C/c1ccc2c(c1)OCO2)c1ccc(OC)c(OC)c1 ZINC000217931471 FH In-Stock Unstable F3 19 41 CC[C@H](NC(=O)/C=C/c1ccc2c(c1)OCO2)c1ccc(OC)c(OC)c1 ZINC000217931471 FH In-Stock Unstable PDE10A 24 45 CC[C@H](NC(=O)/C=C/c1ccc2c(c1)OCO2)c1ccc(OC)c(OC)c1 ZINC000217931471 FH In-Stock Unstable DYRK2 47 35 CC[C@H](NC(=O)/C=C/c1ccc2c(c1)OCO2)c1ccc(OC)c(OC)c1 ZINC000217931471 FH In-Stock Unstable RORC 32 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)C(c1ccccc1)c1ccccc1 ZINC000217931517 II For-Sale Unstable AGTR2 111 48 Cn1cccc1[C@H](O)CCNC(=O)c1ccsc1 ZINC000217931520 CD In-Stock Unstable ITGAV 17 40 COc1cccc(/C=C/NC(=O)N[C@H](C)c2ccc(OC)c(OC)c2)c1 ZINC000217931534 FH For-Sale Unstable MTNR1A 17 43 CC[C@@H](NC(=O)/C=C/c1ccc2c(c1)OCO2)c1ccc(S(C)(=O)=O)cc1 ZINC000217931576 GG In-Stock Unstable KCNQ2 22 45 CC[C@@H](NC(=O)/C=C/c1ccc2c(c1)OCO2)c1ccc(S(C)(=O)=O)cc1 ZINC000217931576 GG In-Stock Unstable DYRK2 51 35 COc1cccc(/C=C2/CC(=O)NC2=O)c1 ZINC000217931578 BD For-Sale Unstable AKR1B1 23 45 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)C(c1ccccc1)c1ccccc1 ZINC000217931606 II For-Sale Unstable AGTR2 111 48 Cn1cccc1[C@@H](O)CCNC(=O)c1ccsc1 ZINC000217931608 CD In-Stock Unstable ITGAV 17 40 Cc1ccnn1CC(=O)N1CCCC[C@@H]1c1nc2cc(F)ccc2[nH]1 ZINC000217931613 EF In-Stock Unstable PRCP 64 46 Cc1ccnn1CC(=O)N1CCCC[C@@H]1c1nc2cc(F)ccc2[nH]1 ZINC000217931613 EF In-Stock Unstable COLA 76 39 Cc1ccnn1CC(=O)N1CCCC[C@@H]1c1nc2cc(F)ccc2[nH]1 ZINC000217931613 EF In-Stock Unstable CPT1A 67 37 CC(C)(C)OC(=O)N1CCC(C=O)(S(C)(=O)=O)CC1 ZINC000217931627 CC In-Stock Unstable GPR119 27 41 COc1ccc([C@@H](C)NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217931649 EH For-Sale Unstable CYP1B1 23 41 COc1ccc([C@@H](C)NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217931649 EH For-Sale Unstable ACACA 25 46 COc1ccc([C@@H](C)NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217931649 EH For-Sale Unstable ACACB 26 56 COc1ccc([C@@H](C)NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217931649 EH For-Sale Unstable AHR 19 40 COc1ccc([C@@H](C)NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217931649 EH For-Sale Unstable MTNR1A 44 45 COc1ccc([C@@H](C)NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217931649 EH For-Sale Unstable MTNR1B 45 45 COc1ccc([C@@H](C)NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217931649 EH For-Sale Unstable CYP1A1 21 41 O=C1C/C(=C/c2ccc(Cl)c(F)c2)C(=O)N1 ZINC000217931655 BD For-Sale Unstable HPGD 41 33 CC[C@H](NC(=O)/C=C/c1ccc2c(c1)OCO2)c1ccc(S(C)(=O)=O)cc1 ZINC000217931662 GG In-Stock Unstable KCNQ2 22 45 CC[C@H](NC(=O)/C=C/c1ccc2c(c1)OCO2)c1ccc(S(C)(=O)=O)cc1 ZINC000217931662 GG In-Stock Unstable DYRK2 51 35 COCCOCc1nc2cc(Cl)ccc2[nH]1 ZINC000217931666 BE For-Sale Unstable PIN1 25 41 Cc1ccnn1CC(=O)N1CCCC[C@H]1c1nc2cc(F)ccc2[nH]1 ZINC000217931682 EF In-Stock Unstable PRCP 64 46 Cc1ccnn1CC(=O)N1CCCC[C@H]1c1nc2cc(F)ccc2[nH]1 ZINC000217931682 EF In-Stock Unstable COLA 76 39 Cc1ccnn1CC(=O)N1CCCC[C@H]1c1nc2cc(F)ccc2[nH]1 ZINC000217931682 EF In-Stock Unstable CPT1A 67 37 Cc1ccccc1-c1cc(C(=O)N(C)C2CCN(C)CC2)c2cnn(C(C)C)c2n1 ZINC000217931696 HI On-Demand Unstable EZH2 20 40 C[C@H](NC(=O)Cc1ccc2c(c1)CCC(C)(C)O2)C(=O)O ZINC000217931705 CD In-Stock Unstable NDUFA4 0 40 C[C@H](NC(=O)Cc1ccc2c(c1)CCC(C)(C)O2)C(=O)O ZINC000217931705 CD In-Stock Unstable DAGLA 23 43 Cn1cccc1[C@H](O)CCNC(=O)C1CCCCC1 ZINC000217931707 CE In-Stock Unstable SLC6A1 49 35 CCCCN(CCO)Cc1ccccc1/C=C\C(=O)O ZINC000217931714 CE For-Sale Unstable PTGER2 15 41 CCCCN(CCO)Cc1ccccc1/C=C\C(=O)O ZINC000217931714 CE For-Sale Unstable PTGER3 17 46 CCCCN(CCO)Cc1ccccc1/C=C\C(=O)O ZINC000217931714 CE For-Sale Unstable PLM2_PLAFA 25 40 COc1ccc([C@H](C)NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217931715 EH For-Sale Unstable CYP1B1 23 41 COc1ccc([C@H](C)NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217931715 EH For-Sale Unstable ACACA 25 46 COc1ccc([C@H](C)NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217931715 EH For-Sale Unstable ACACB 26 56 COc1ccc([C@H](C)NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217931715 EH For-Sale Unstable AHR 19 40 COc1ccc([C@H](C)NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217931715 EH For-Sale Unstable MTNR1A 44 45 COc1ccc([C@H](C)NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217931715 EH For-Sale Unstable MTNR1B 45 45 COc1ccc([C@H](C)NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217931715 EH For-Sale Unstable CYP1A1 21 41 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cc(OC)c(OC)c(OC)c1 ZINC000217931726 IF For-Sale Unstable ACKR3 41 35 Cc1cccc(-c2noc(CNC(=O)/C=C/c3ccc4c(c3)OCO4)n2)c1 ZINC000217931762 FG In-Stock Unstable HDAC8 45 33 Cc1cccc(-c2noc(CNC(=O)/C=C/c3ccc4c(c3)OCO4)n2)c1 ZINC000217931762 FG In-Stock Unstable DYRK2 51 35 Cn1cccc1[C@@H](O)CCNC(=O)C1CCCCC1 ZINC000217931780 CE In-Stock Unstable SLC6A1 49 35 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cc(OC)c(OC)c(OC)c1 ZINC000217931798 IF For-Sale Unstable ACKR3 41 35 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1O ZINC000217931826 II In-Stock Unstable AKR1B1 22 46 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1O ZINC000217931826 II In-Stock Unstable CYP1B1 67 39 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1O ZINC000217931826 II In-Stock Unstable CYP1A1 50 48 COc1ccc([C@@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1O ZINC000217931826 II In-Stock Unstable CYP1A2 42 50 Cc1ccc(-c2noc(CNC(=O)/C=C/c3ccc4c(c3)OCO4)n2)cc1 ZINC000217931866 FG In-Stock Unstable DYRK2 56 36 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cc(OC)c(OC)c(OC)c1 ZINC000217931872 IF For-Sale Unstable ACKR3 41 35 CC1CN(c2ccnc(Cl)n2)C1 ZINC000217931898 AD For-Sale Unstable SORD 70 36 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1O ZINC000217931907 II In-Stock Unstable AKR1B1 22 46 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1O ZINC000217931907 II In-Stock Unstable CYP1B1 67 39 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1O ZINC000217931907 II In-Stock Unstable CYP1A1 50 48 COc1ccc([C@H]2CC(=O)Oc3cc(O)c4c(=O)cc(-c5ccc(O)cc5)oc4c32)cc1O ZINC000217931907 II In-Stock Unstable CYP1A2 42 50 CC[C@@H](CCO)NC(=O)CNC(=O)CN ZINC000217931948 BA For-Sale Unstable UREB 0 44 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cc(OC)c(OC)c(OC)c1 ZINC000217931961 IF For-Sale Unstable ACKR3 41 35 COc1cccc(-c2noc(CNC(=O)/C=C/c3ccc4c(c3)OCO4)n2)c1 ZINC000217931968 GF In-Stock Unstable EDNRB 56 39 COc1cccc(-c2noc(CNC(=O)/C=C/c3ccc4c(c3)OCO4)n2)c1 ZINC000217931968 GF In-Stock Unstable EDNRA 55 39 COc1cccc(-c2noc(CNC(=O)/C=C/c3ccc4c(c3)OCO4)n2)c1 ZINC000217931968 GF In-Stock Unstable DYRK2 45 35 C[Si](C)(C)c1ccc(NC(=O)Oc2ccccc2)cc1 ZINC000217931971 CH For-Sale Unstable ACHE 20 52 C[Si](C)(C)c1ccc(NC(=O)Oc2ccccc2)cc1 ZINC000217931971 CH For-Sale Unstable BCHE 19 54 C[Si](C)(C)c1ccc(NC(=O)Oc2ccccc2)cc1 ZINC000217931971 CH For-Sale Unstable RAF1 17 42 C[Si](C)(C)c1ccc(NC(=O)Oc2ccccc2)cc1 ZINC000217931971 CH For-Sale Unstable FAAH 32 56 C[Si](C)(C)c1ccc(NC(=O)Oc2ccccc2)cc1 ZINC000217931971 CH For-Sale Unstable ACR 59 44 C[Si](C)(C)c1ccc(NC(=O)Oc2ccccc2)cc1 ZINC000217931971 CH For-Sale Unstable Q8MMZ8_EIMTE 21 42 CC[C@H](CCO)NC(=O)CNC(=O)CN ZINC000217932013 BA For-Sale Unstable UREB 0 44 COC(=O)C[C@H](c1cc(OC)c(OC)cc1OC)c1c(O)c2ccccc2oc1=O ZINC000217932017 HG In-Stock Unstable NQO1 64 51 COCCN(CCOC)Cc1ccccc1/C=C\C(=O)O ZINC000217932050 CD For-Sale Unstable PTGER2 62 50 COCCN(CCOC)Cc1ccccc1/C=C\C(=O)O ZINC000217932050 CD For-Sale Unstable PTGER4 29 43 COCCN(CCOC)Cc1ccccc1/C=C\C(=O)O ZINC000217932050 CD For-Sale Unstable PTGER3 25 50 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccc4c(c3)OCO4)n2)cc1 ZINC000217932059 GF In-Stock Unstable EDNRB 70 40 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccc4c(c3)OCO4)n2)cc1 ZINC000217932059 GF In-Stock Unstable EDNRA 67 39 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccc4c(c3)OCO4)n2)cc1 ZINC000217932059 GF In-Stock Unstable BMP1 57 35 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccc4c(c3)OCO4)n2)cc1 ZINC000217932059 GF In-Stock Unstable TERT 0 42 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccc4c(c3)OCO4)n2)cc1 ZINC000217932059 GF In-Stock Unstable DYRK2 59 39 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccc2ccccc2c1 ZINC000217932060 HH For-Sale Unstable COLA 43 36 COC(=O)C[C@@H](c1cc(OC)c(OC)cc1OC)c1c(O)c2ccccc2oc1=O ZINC000217932097 HG In-Stock Unstable NQO1 64 51 O=C(O)C1(S(=O)(=O)c2cccs2)CCOCC1 ZINC000217932140 CD In-Stock Unstable MMP2 16 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccc2ccccc2c1 ZINC000217932144 HH For-Sale Unstable COLA 43 36 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccc4c(c3)OCO4)n2)c(OC)c1 ZINC000217932155 HF In-Stock Unstable EDNRB 59 40 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccc4c(c3)OCO4)n2)c(OC)c1 ZINC000217932155 HF In-Stock Unstable EDNRA 56 38 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1ccc(Cl)cc1F ZINC000217932176 CK For-Sale Unstable TRPM8 17 53 O=C([C@@H]1CCCN1C[C@@H]1CCCCO1)N1CCNCC1 ZINC000217932183 CC For-Sale Unstable PREP 24 41 CCc1ccc([C@@H](C)NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217932194 DI For-Sale Unstable ACACA 25 40 CCc1ccc([C@@H](C)NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217932194 DI For-Sale Unstable ACACB 29 48 CCc1ccc([C@@H](C)NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217932194 DI For-Sale Unstable MTNR1A 33 40 CCc1ccc([C@@H](C)NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217932194 DI For-Sale Unstable MTNR1B 36 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccc2ccccc2c1 ZINC000217932237 HH For-Sale Unstable COLA 43 36 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1ccc(Cl)cc1F ZINC000217932258 CK For-Sale Unstable TRPM8 17 53 O=C(NCc1cnc2cnccn12)c1ccc(Cl)s1 ZINC000217932259 CE In-Stock Unstable F10 25 44 CCc1ccc([C@H](C)NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217932274 DI For-Sale Unstable ACACA 25 40 CCc1ccc([C@H](C)NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217932274 DI For-Sale Unstable ACACB 29 48 CCc1ccc([C@H](C)NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217932274 DI For-Sale Unstable MTNR1A 33 40 CCc1ccc([C@H](C)NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217932274 DI For-Sale Unstable MTNR1B 36 40 Cn1cccc1[C@H](O)CCNC(=O)c1cccc(C#N)c1 ZINC000217932278 CD In-Stock Unstable DRD4 43 33 COCCN(CCOC)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217932283 CD For-Sale Unstable PTGER2 29 42 COCCN(CCOC)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217932283 CD For-Sale Unstable LTB4R 17 51 COCCN(CCOC)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217932283 CD For-Sale Unstable NR1H4 47 36 COCCN(CCOC)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217932283 CD For-Sale Unstable AKR1C3 32 42 CCCCCCC/C(C)=C1/CC(=O)NC1=O ZINC000217932294 BF For-Sale Unstable CQSS 53 32 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccc2ccccc2c1 ZINC000217932322 HH For-Sale Unstable COLA 43 36 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1ccc(Cl)cc1F ZINC000217932335 CK For-Sale Unstable TRPM8 17 53 C[C@@H]1CCC[C@@H](CNc2cccnc2[N+](=O)[O-])C1 ZINC000217932356 BG On-Demand Unstable PRKCQ 43 38 Cn1cccc1[C@@H](O)CCNC(=O)c1cccc(C#N)c1 ZINC000217932358 CD In-Stock Unstable DRD4 43 33 O=C(/C=C/c1ccc2c(c1)OCO2)NCc1nc(-c2ccc(Cl)cc2)no1 ZINC000217932369 GG In-Stock Unstable DYRK2 41 32 COC(=O)C[C@H]1c2cc3c(cc2Oc2nc4cc(OC)ccc4cc21)OCO3 ZINC000217932401 GH In-Stock Unstable EDNRB 58 40 COC(=O)C[C@H]1c2cc3c(cc2Oc2nc4cc(OC)ccc4cc21)OCO3 ZINC000217932401 GH In-Stock Unstable EDNRA 56 40 O=C1NCCCC[C@H]1N1CCC[C@H]1C(=O)N1CCNCC1 ZINC000217932413 CB For-Sale Unstable PREP 28 42 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1ccc(Cl)cc1F ZINC000217932414 CK For-Sale Unstable TRPM8 17 53 O=C(c1ccc(N2CCCC2)cc1)N1CCN(c2ncc[nH]c2=O)CC1 ZINC000217932424 FD In-Stock Unstable L3MBTL1 0 44 O=C(c1ccc(N2CCCC2)cc1)N1CCN(c2ncc[nH]c2=O)CC1 ZINC000217932424 FD In-Stock Unstable L3MBTL3 47 44 O=C(c1ccc(N2CCCC2)cc1)N1CCN(c2ncc[nH]c2=O)CC1 ZINC000217932424 FD In-Stock Unstable L3MBTL4 0 44 O=C(c1ccc(N2CCCC2)cc1)N1CCN(c2ncc[nH]c2=O)CC1 ZINC000217932424 FD In-Stock Unstable MBTD1 0 44 O=C(c1ccc(N2CCCC2)cc1)N1CCN(c2ncc[nH]c2=O)CC1 ZINC000217932424 FD In-Stock Unstable TP53BP1 0 44 O=C(c1ccc(N2CCCC2)cc1)N1CCN(c2ncc[nH]c2=O)CC1 ZINC000217932424 FD In-Stock Unstable SLC6A7 0 47 C[C@H]1CCC[C@@H](CNc2cccnc2[N+](=O)[O-])C1 ZINC000217932433 BG On-Demand Unstable PRKCQ 43 38 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cnn(-c2ccccc2)n1 ZINC000217932439 HE For-Sale Unstable HCRTR1 44 37 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cnn(-c2ccccc2)n1 ZINC000217932439 HE For-Sale Unstable HCRTR2 48 37 Cn1cccc1[C@H](O)CCNC(=O)/C=C/c1ccccc1 ZINC000217932459 CE In-Stock Unstable HDAC8 52 36 Cn1cccc1[C@H](O)CCNC(=O)/C=C/c1ccccc1 ZINC000217932459 CE In-Stock Unstable MMP2 17 51 Cn1cccc1[C@H](O)CCNC(=O)/C=C/c1ccccc1 ZINC000217932459 CE In-Stock Unstable HDAC1 24 40 Cn1cccc1[C@H](O)CCNC(=O)/C=C/c1ccccc1 ZINC000217932459 CE In-Stock Unstable HDAC6 40 43 Cn1cccc1[C@H](O)CCNC(=O)/C=C/c1ccccc1 ZINC000217932459 CE In-Stock Unstable MMP9 15 51 Cn1cccc1[C@H](O)CCNC(=O)/C=C/c1ccccc1 ZINC000217932459 CE In-Stock Unstable HDAC9 20 40 Cn1cccc1[C@H](O)CCNC(=O)/C=C/c1ccccc1 ZINC000217932459 CE In-Stock Unstable HDAC7 29 40 Cn1cccc1[C@H](O)CCNC(=O)/C=C/c1ccccc1 ZINC000217932459 CE In-Stock Unstable HDA106 0 41 COC(=O)C[C@@H]1c2cc3c(cc2Oc2nc4cc(OC)ccc4cc21)OCO3 ZINC000217932491 GH In-Stock Unstable EDNRB 45 38 COC(=O)C[C@@H]1c2cc3c(cc2Oc2nc4cc(OC)ccc4cc21)OCO3 ZINC000217932491 GH In-Stock Unstable EDNRA 43 38 O=C(/C=C/c1ccc2c(c1)OCO2)NCc1nc(-c2cccc(Br)c2)no1 ZINC000217932496 IH In-Stock Unstable HDAC8 43 32 C[C@@H]1CCC[C@H](CNc2cccnc2[N+](=O)[O-])C1 ZINC000217932518 BG On-Demand Unstable PRKCQ 43 38 Cn1cccc1[C@@H](O)CCNC(=O)/C=C/c1ccccc1 ZINC000217932524 CE In-Stock Unstable HDAC8 52 36 Cn1cccc1[C@@H](O)CCNC(=O)/C=C/c1ccccc1 ZINC000217932524 CE In-Stock Unstable MMP2 17 51 Cn1cccc1[C@@H](O)CCNC(=O)/C=C/c1ccccc1 ZINC000217932524 CE In-Stock Unstable HDAC1 24 40 Cn1cccc1[C@@H](O)CCNC(=O)/C=C/c1ccccc1 ZINC000217932524 CE In-Stock Unstable HDAC6 40 43 Cn1cccc1[C@@H](O)CCNC(=O)/C=C/c1ccccc1 ZINC000217932524 CE In-Stock Unstable MMP9 15 51 Cn1cccc1[C@@H](O)CCNC(=O)/C=C/c1ccccc1 ZINC000217932524 CE In-Stock Unstable HDAC9 20 40 Cn1cccc1[C@@H](O)CCNC(=O)/C=C/c1ccccc1 ZINC000217932524 CE In-Stock Unstable HDAC7 29 40 Cn1cccc1[C@@H](O)CCNC(=O)/C=C/c1ccccc1 ZINC000217932524 CE In-Stock Unstable HDA106 0 41 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cnn(-c2ccccc2)n1 ZINC000217932535 HE For-Sale Unstable HCRTR1 44 37 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cnn(-c2ccccc2)n1 ZINC000217932535 HE For-Sale Unstable HCRTR2 48 37 CCc1cccc(CC)c1NC(=O)N/C=C/c1cccc(OC)c1 ZINC000217932557 DJ For-Sale Unstable AHR 18 41 CCc1cccc(CC)c1NC(=O)N/C=C/c1cccc(OC)c1 ZINC000217932557 DJ For-Sale Unstable MTNR1A 55 44 CCc1cccc(CC)c1NC(=O)N/C=C/c1cccc(OC)c1 ZINC000217932557 DJ For-Sale Unstable MTNR1B 51 44 C[C@H]1CCC[C@H](CNc2cccnc2[N+](=O)[O-])C1 ZINC000217932589 BG On-Demand Unstable PRKCQ 43 38 Cn1cccc1[C@H](O)CCNC(=O)CCc1ccccc1 ZINC000217932627 CE In-Stock Unstable MMP3 15 42 Cn1cccc1[C@H](O)CCNC(=O)CCc1ccccc1 ZINC000217932627 CE In-Stock Unstable PAM 0 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cnn(-c2ccccc2)n1 ZINC000217932629 HE For-Sale Unstable HCRTR1 44 37 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cnn(-c2ccccc2)n1 ZINC000217932629 HE For-Sale Unstable HCRTR2 48 37 COc1cccc(/C=C/NC(=O)Nc2ccc(Oc3ccccc3)cc2)c1 ZINC000217932660 FK For-Sale Unstable PDGFRB 22 40 COc1cccc(/C=C/NC(=O)Nc2ccc(Oc3ccccc3)cc2)c1 ZINC000217932660 FK For-Sale Unstable CYP1B1 27 41 COc1cccc(/C=C/NC(=O)Nc2ccc(Oc3ccccc3)cc2)c1 ZINC000217932660 FK For-Sale Unstable CA1 49 45 COc1cccc(/C=C/NC(=O)Nc2ccc(Oc3ccccc3)cc2)c1 ZINC000217932660 FK For-Sale Unstable RAF1 42 55 COc1cccc(/C=C/NC(=O)Nc2ccc(Oc3ccccc3)cc2)c1 ZINC000217932660 FK For-Sale Unstable KDR 27 43 COc1cccc(/C=C/NC(=O)Nc2ccc(Oc3ccccc3)cc2)c1 ZINC000217932660 FK For-Sale Unstable MTNR1A 41 59 COc1cccc(/C=C/NC(=O)Nc2ccc(Oc3ccccc3)cc2)c1 ZINC000217932660 FK For-Sale Unstable MTNR1B 46 59 COc1cccc(/C=C/NC(=O)Nc2ccc(Oc3ccccc3)cc2)c1 ZINC000217932660 FK For-Sale Unstable CYP1A1 24 41 COc1cccc(/C=C/NC(=O)Nc2ccc(Oc3ccccc3)cc2)c1 ZINC000217932660 FK For-Sale Unstable NPY5R 26 43 COc1cccc(/C=C/NC(=O)Nc2ccc(Oc3ccccc3)cc2)c1 ZINC000217932660 FK For-Sale Unstable CA12 17 45 COc1cccc(/C=C/NC(=O)Nc2ccc(Oc3ccccc3)cc2)c1 ZINC000217932660 FK For-Sale Unstable PDGFRA 53 43 COc1cccc(/C=C/NC(=O)Nc2ccc(Oc3ccccc3)cc2)c1 ZINC000217932660 FK For-Sale Unstable CA9 17 45 COc1cccc(/C=C/NC(=O)Nc2ccc(Oc3ccccc3)cc2)c1 ZINC000217932660 FK For-Sale Unstable Q8MMZ8_EIMTE 55 55 COc1cccc(/C=C/NC(=O)Nc2ccc(Oc3ccccc3)cc2)c1 ZINC000217932660 FK For-Sale Unstable AKR1C3 23 41 COc1cccc(/C=C/NC(=O)Nc2ccc(Oc3ccccc3)cc2)c1 ZINC000217932660 FK For-Sale Unstable AKR1C2 52 36 CCCOc1ccc(/C(C)=C2/CC(=O)NC2=O)cc1 ZINC000217932702 CE For-Sale Unstable PLA2G4B 70 37 Cn1cccc1[C@@H](O)CCNC(=O)CCc1ccccc1 ZINC000217932711 CE In-Stock Unstable MMP3 15 42 Cn1cccc1[C@@H](O)CCNC(=O)CCc1ccccc1 ZINC000217932711 CE In-Stock Unstable PAM 0 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cnn(-c2ccccc2)n1 ZINC000217932715 HE For-Sale Unstable HCRTR1 44 37 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cnn(-c2ccccc2)n1 ZINC000217932715 HE For-Sale Unstable HCRTR2 48 37 NS(=O)(=O)c1ccc(C(=O)N2CCCC[C@@H]2CC(=O)O)cc1 ZINC000217932721 EC In-Stock Unstable CA2 51 62 NS(=O)(=O)c1ccc(C(=O)N2CCCC[C@@H]2CC(=O)O)cc1 ZINC000217932721 EC In-Stock Unstable CA1 43 45 NS(=O)(=O)c1ccc(C(=O)N2CCCC[C@@H]2CC(=O)O)cc1 ZINC000217932721 EC In-Stock Unstable PREP 21 40 NS(=O)(=O)c1ccc(C(=O)N2CCCC[C@@H]2CC(=O)O)cc1 ZINC000217932721 EC In-Stock Unstable CA4 50 41 NS(=O)(=O)c1ccc(C(=O)N2CCCC[C@@H]2CC(=O)O)cc1 ZINC000217932721 EC In-Stock Unstable NCE103 22 45 NS(=O)(=O)c1ccc(C(=O)N2CCCC[C@@H]2CC(=O)O)cc1 ZINC000217932721 EC In-Stock Unstable CA 0 45 NS(=O)(=O)c1ccc(C(=O)N2CCCC[C@@H]2CC(=O)O)cc1 ZINC000217932721 EC In-Stock Unstable L3MBTL1 0 40 NS(=O)(=O)c1ccc(C(=O)N2CCCC[C@@H]2CC(=O)O)cc1 ZINC000217932721 EC In-Stock Unstable L3MBTL3 55 36 NS(=O)(=O)c1ccc(C(=O)N2CCCC[C@@H]2CC(=O)O)cc1 ZINC000217932721 EC In-Stock Unstable MBTD1 0 40 NS(=O)(=O)c1ccc(C(=O)N2CCCC[C@@H]2CC(=O)O)cc1 ZINC000217932721 EC In-Stock Unstable Q5TU56_ANOGA 0 45 CN(Cc1nc(-c2ccccc2)no1)C(=O)/C=C/c1ccc2c(c1)OCO2 ZINC000217932742 FG In-Stock Unstable FABI 43 33 CN(Cc1nc(-c2ccccc2)no1)C(=O)/C=C/c1ccc2c(c1)OCO2 ZINC000217932742 FG In-Stock Unstable DYRK2 45 34 O=C(O)/C=C\c1cccc(CN2CCC[C@H](CO)C2)c1 ZINC000217932766 CD For-Sale Unstable SLC6A1 71 34 O=C(O)/C=C\c1cccc(CN2CCC[C@H](CO)C2)c1 ZINC000217932766 CD For-Sale Unstable SIGMAR1 32 46 O=C(O)/C=C\c1cccc(CN2CCC[C@H](CO)C2)c1 ZINC000217932766 CD For-Sale Unstable CCR3 28 42 COC(=O)c1ccnc(NCC2CCC(C)CC2)c1 ZINC000217932769 CG On-Demand Unstable KDM3A 0 46 COC(=O)c1ccnc(NCC2CCC(C)CC2)c1 ZINC000217932769 CG On-Demand Unstable KDM5C 0 46 COC(=O)c1ccnc(NCC2CCC(C)CC2)c1 ZINC000217932769 CG On-Demand Unstable GPR39 0 40 COc1cccc(/C=C/NC(=O)Nc2cc(Cl)ccc2C)c1 ZINC000217932773 DI For-Sale Unstable S1PR4 25 44 NS(=O)(=O)c1ccc(C(=O)N2CCCC[C@H]2CC(=O)O)cc1 ZINC000217932806 EC In-Stock Unstable CA2 51 62 NS(=O)(=O)c1ccc(C(=O)N2CCCC[C@H]2CC(=O)O)cc1 ZINC000217932806 EC In-Stock Unstable CA1 43 45 NS(=O)(=O)c1ccc(C(=O)N2CCCC[C@H]2CC(=O)O)cc1 ZINC000217932806 EC In-Stock Unstable PREP 21 40 NS(=O)(=O)c1ccc(C(=O)N2CCCC[C@H]2CC(=O)O)cc1 ZINC000217932806 EC In-Stock Unstable CA4 50 41 NS(=O)(=O)c1ccc(C(=O)N2CCCC[C@H]2CC(=O)O)cc1 ZINC000217932806 EC In-Stock Unstable NCE103 22 45 NS(=O)(=O)c1ccc(C(=O)N2CCCC[C@H]2CC(=O)O)cc1 ZINC000217932806 EC In-Stock Unstable CA 0 45 NS(=O)(=O)c1ccc(C(=O)N2CCCC[C@H]2CC(=O)O)cc1 ZINC000217932806 EC In-Stock Unstable L3MBTL1 0 40 NS(=O)(=O)c1ccc(C(=O)N2CCCC[C@H]2CC(=O)O)cc1 ZINC000217932806 EC In-Stock Unstable L3MBTL3 55 36 NS(=O)(=O)c1ccc(C(=O)N2CCCC[C@H]2CC(=O)O)cc1 ZINC000217932806 EC In-Stock Unstable MBTD1 0 40 NS(=O)(=O)c1ccc(C(=O)N2CCCC[C@H]2CC(=O)O)cc1 ZINC000217932806 EC In-Stock Unstable Q5TU56_ANOGA 0 45 O=S1(=O)CCCN(C[C@@H](O)COCc2ccccc2)CC1 ZINC000217932824 DC On-Demand Unstable ABCB1 58 45 O=S1(=O)CCCN(C[C@@H](O)COCc2ccccc2)CC1 ZINC000217932824 DC On-Demand Unstable HSP90AB1 34 41 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccc(-c2ccccc2)cc1 ZINC000217932825 II For-Sale Unstable CPT1A 111 38 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccc(-c2ccccc2)cc1 ZINC000217932825 II For-Sale Unstable CPT2 40 38 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccc(-c2ccccc2)cc1 ZINC000217932825 II For-Sale Unstable GYS1 50 38 Cc1cccc(-c2noc(CN(C)C(=O)/C=C/c3ccc4c(c3)OCO4)n2)c1 ZINC000217932842 GG In-Stock Unstable FABI 42 32 CC[C@@H](CCO)NC(=O)CC1(CN)CCC1 ZINC000217932858 BC For-Sale Unstable CACNA2D1 0 40 COc1cccc(/C=C/NC(=O)Nc2cc(OC)ccc2OC)c1 ZINC000217932865 EH For-Sale Unstable CYP1B1 63 39 COc1cccc(/C=C/NC(=O)Nc2cc(OC)ccc2OC)c1 ZINC000217932865 EH For-Sale Unstable MTNR1A 41 47 COc1cccc(/C=C/NC(=O)Nc2cc(OC)ccc2OC)c1 ZINC000217932865 EH For-Sale Unstable MTNR1B 43 47 COc1cccc(/C=C/NC(=O)Nc2cc(OC)ccc2OC)c1 ZINC000217932865 EH For-Sale Unstable CYP1A1 45 48 COc1cccc(/C=C/NC(=O)Nc2cc(OC)ccc2OC)c1 ZINC000217932865 EH For-Sale Unstable AKR1C3 22 42 COc1cccc(/C=C/NC(=O)Nc2cc(OC)ccc2OC)c1 ZINC000217932865 EH For-Sale Unstable ABCG2 20 45 COc1cccc(/C=C/NC(=O)Nc2cc(OC)ccc2OC)c1 ZINC000217932865 EH For-Sale Unstable AKR1C2 51 37 O=C(O)/C=C\c1cc(F)ccc1CN1CCC[C@H](CO)C1 ZINC000217932890 CE For-Sale Unstable SLC6A1 100 43 O=C(O)/C=C\c1cc(F)ccc1CN1CCC[C@H](CO)C1 ZINC000217932890 CE For-Sale Unstable CCR3 40 35 O=S1(=O)CCCN(C[C@H](O)COCc2ccccc2)CC1 ZINC000217932901 DC On-Demand Unstable ABCB1 58 45 O=S1(=O)CCCN(C[C@H](O)COCc2ccccc2)CC1 ZINC000217932901 DC On-Demand Unstable HSP90AB1 34 41 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccc(-c2ccccc2)cc1 ZINC000217932903 II For-Sale Unstable CPT1A 111 38 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccc(-c2ccccc2)cc1 ZINC000217932903 II For-Sale Unstable CPT2 40 38 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccc(-c2ccccc2)cc1 ZINC000217932903 II For-Sale Unstable GYS1 50 38 CN1CCC(N(C)C(=O)[C@@H]2CCCN(S(=O)(=O)c3ccc(Br)cc3)C2)CC1 ZINC000217932907 JE On-Demand Unstable AKR1C3 30 45 CN1CCC(N(C)C(=O)[C@@H]2CCCN(S(=O)(=O)c3ccc(Br)cc3)C2)CC1 ZINC000217932907 JE On-Demand Unstable AKR1C1 22 45 CC[C@H](CCO)NC(=O)CC1(CN)CCC1 ZINC000217932948 BC For-Sale Unstable CACNA2D1 0 40 Cc1ccc(-c2noc(CN(C)C(=O)/C=C/c3ccc4c(c3)OCO4)n2)cc1 ZINC000217932953 GG In-Stock Unstable FABI 41 31 Cc1ccc(-c2noc(CN(C)C(=O)/C=C/c3ccc4c(c3)OCO4)n2)cc1 ZINC000217932953 GG In-Stock Unstable DYRK2 52 36 CCc1cccc(C)c1NC(=O)N/C=C/c1cccc(OC)c1 ZINC000217932972 DI For-Sale Unstable S1PR4 0 40 CCc1cccc(C)c1NC(=O)N/C=C/c1cccc(OC)c1 ZINC000217932972 DI For-Sale Unstable MTNR1A 37 41 CCc1cccc(C)c1NC(=O)N/C=C/c1cccc(OC)c1 ZINC000217932972 DI For-Sale Unstable MTNR1B 37 41 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccc(-c2ccccc2)cc1 ZINC000217932976 II For-Sale Unstable CPT1A 111 38 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccc(-c2ccccc2)cc1 ZINC000217932976 II For-Sale Unstable CPT2 40 38 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccc(-c2ccccc2)cc1 ZINC000217932976 II For-Sale Unstable GYS1 50 38 O=C([C@H]1CCCN1[C@H]1CS(=O)(=O)C[C@H]1O)N1CCNCC1 ZINC000217932979 DA For-Sale Unstable PREP 27 44 CN1CCC(N(C)C(=O)[C@H]2CCCN(S(=O)(=O)c3ccc(Br)cc3)C2)CC1 ZINC000217932994 JE On-Demand Unstable AKR1C3 30 45 CN1CCC(N(C)C(=O)[C@H]2CCCN(S(=O)(=O)c3ccc(Br)cc3)C2)CC1 ZINC000217932994 JE On-Demand Unstable AKR1C1 22 45 O=C(O)/C=C\c1cc(CN2CCC[C@H](CO)C2)ccc1F ZINC000217932995 CE For-Sale Unstable SLC6A1 76 35 O=C(O)/C=C\c1cc(CN2CCC[C@H](CO)C2)ccc1F ZINC000217932995 CE For-Sale Unstable CCR3 50 38 O=C([C@H]1CCCN1[C@H]1CS(=O)(=O)C[C@@H]1O)N1CCNCC1 ZINC000217933051 DA For-Sale Unstable PREP 27 44 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccc(-c2ccccc2)cc1 ZINC000217933054 II For-Sale Unstable CPT1A 111 38 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccc(-c2ccccc2)cc1 ZINC000217933054 II For-Sale Unstable CPT2 40 38 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccc(-c2ccccc2)cc1 ZINC000217933054 II For-Sale Unstable GYS1 50 38 COc1cccc(-c2noc(CN(C)C(=O)/C=C/c3ccc4c(c3)OCO4)n2)c1 ZINC000217933056 GG In-Stock Unstable EDNRB 33 44 COc1cccc(/C=C/NC(=O)Nc2c(C)cc(C)cc2C)c1 ZINC000217933064 DI For-Sale Unstable PYGL 36 42 COc1cccc(/C=C/NC(=O)Nc2c(C)cc(C)cc2C)c1 ZINC000217933064 DI For-Sale Unstable MTNR1A 26 42 COc1cccc(/C=C/NC(=O)Nc2c(C)cc(C)cc2C)c1 ZINC000217933064 DI For-Sale Unstable MTNR1B 31 42 Cc1cc(-c2cc(C(=O)N(C)C3CCN(C)CC3)c3cnn(C(C)C)c3n2)c(C)s1 ZINC000217933103 IJ On-Demand Unstable EZH2 19 40 C[C@@H]1CCCCN1Cc1ccc(F)cc1/C=C\C(=O)O ZINC000217933114 CG For-Sale Unstable HRH3 22 41 O=C([C@H]1CCCN1[C@@H]1CS(=O)(=O)C[C@H]1O)N1CCNCC1 ZINC000217933117 DA For-Sale Unstable PREP 27 44 COc1ccc(-c2noc(CN(C)C(=O)/C=C/c3ccc4c(c3)OCO4)n2)cc1 ZINC000217933150 GG In-Stock Unstable EDNRB 48 46 COc1ccc(-c2noc(CN(C)C(=O)/C=C/c3ccc4c(c3)OCO4)n2)cc1 ZINC000217933150 GG In-Stock Unstable EDNRA 43 36 COc1ccc(-c2noc(CN(C)C(=O)/C=C/c3ccc4c(c3)OCO4)n2)cc1 ZINC000217933150 GG In-Stock Unstable BMP1 43 34 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc(S(N)(=O)=O)cc1 ZINC000217933169 HD For-Sale Unstable CA2 23 40 COC(=O)c1ccccc1NC(=O)N/C=C/c1cccc(OC)c1 ZINC000217933178 EG For-Sale Unstable MTNR1A 29 40 COC(=O)c1ccccc1NC(=O)N/C=C/c1cccc(OC)c1 ZINC000217933178 EG For-Sale Unstable MTNR1B 30 40 COC(=O)c1ccccc1NC(=O)N/C=C/c1cccc(OC)c1 ZINC000217933178 EG For-Sale Unstable AKR1C3 17 45 Cn1cccc1[C@H](O)CCNC(=O)c1cccc(Cl)c1 ZINC000217933183 CF In-Stock Unstable CPT1A 43 30 Cn1cccc1[C@H](O)CCNC(=O)c1cccc(Cl)c1 ZINC000217933183 CF In-Stock Unstable CCKBR 22 46 C[C@H]1CCCCN1Cc1ccc(F)cc1/C=C\C(=O)O ZINC000217933203 CG For-Sale Unstable HRH3 22 41 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc(S(N)(=O)=O)cc1 ZINC000217933255 HD For-Sale Unstable CA2 23 40 Cn1cccc1[C@@H](O)CCNC(=O)c1cccc(Cl)c1 ZINC000217933263 CF In-Stock Unstable CPT1A 43 30 Cn1cccc1[C@@H](O)CCNC(=O)c1cccc(Cl)c1 ZINC000217933263 CF In-Stock Unstable CCKBR 22 46 COc1ccc(-c2noc(CN(C)C(=O)/C=C/c3ccc4c(c3)OCO4)n2)c(OC)c1 ZINC000217933264 HG In-Stock Unstable EDNRB 41 47 COc1ccc(-c2noc(CN(C)C(=O)/C=C/c3ccc4c(c3)OCO4)n2)c(OC)c1 ZINC000217933264 HG In-Stock Unstable EDNRA 44 37 COc1cccc(/C=C/NC(=O)Nc2ccc(F)cc2)c1 ZINC000217933288 CH For-Sale Unstable CYP1B1 25 42 COc1cccc(/C=C/NC(=O)Nc2ccc(F)cc2)c1 ZINC000217933288 CH For-Sale Unstable CCR3 16 40 COc1cccc(/C=C/NC(=O)Nc2ccc(F)cc2)c1 ZINC000217933288 CH For-Sale Unstable AHR 20 41 COc1cccc(/C=C/NC(=O)Nc2ccc(F)cc2)c1 ZINC000217933288 CH For-Sale Unstable KDR 18 40 COc1cccc(/C=C/NC(=O)Nc2ccc(F)cc2)c1 ZINC000217933288 CH For-Sale Unstable MTNR1A 29 53 COc1cccc(/C=C/NC(=O)Nc2ccc(F)cc2)c1 ZINC000217933288 CH For-Sale Unstable MTNR1B 35 53 COc1cccc(/C=C/NC(=O)Nc2ccc(F)cc2)c1 ZINC000217933288 CH For-Sale Unstable ROCK2 18 40 COc1cccc(/C=C/NC(=O)Nc2ccc(F)cc2)c1 ZINC000217933288 CH For-Sale Unstable Q8MMZ8_EIMTE 0 47 COc1cccc(/C=C/NC(=O)Nc2ccc(F)cc2)c1 ZINC000217933288 CH For-Sale Unstable TAAR1 30 43 COc1cccc(/C=C/NC(=O)Nc2ccc(F)cc2)c1 ZINC000217933288 CH For-Sale Unstable AKR1C2 40 32 C[C@@H]1CCCCN1Cc1ccc(F)c(/C=C\C(=O)O)c1 ZINC000217933318 CG For-Sale Unstable HRH3 42 42 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc(S(N)(=O)=O)cc1 ZINC000217933329 HD For-Sale Unstable CA2 23 40 O=C1C/C(=C/c2ccc(-c3cccc(Br)c3)s2)C(=O)N1 ZINC000217933362 EH For-Sale Unstable PRF1 46 41 CCCC(CCC)C(=O)O[C@@H]1C[C@H]2CC[C@@]1(C)C2(C)C ZINC000217933373 CJ For-Sale Unstable ELANE 0 46 CN(Cc1nc(-c2ccccc2Cl)no1)C(=O)/C=C/c1ccc2c(c1)OCO2 ZINC000217933381 GH In-Stock Unstable FABI 41 31 C[C@H]1CCCCN1Cc1ccc(F)c(/C=C\C(=O)O)c1 ZINC000217933401 CG For-Sale Unstable HRH3 42 42 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c([N+](=O)[O-])c2)c1 ZINC000217933402 EI For-Sale Unstable MTNR1B 19 40 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c([N+](=O)[O-])c2)c1 ZINC000217933402 EI For-Sale Unstable TAAR1 32 58 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c([N+](=O)[O-])c2)c1 ZINC000217933402 EI For-Sale Unstable IMDH_CRYPV 41 46 O=S(=O)(Nc1nc2c(s1)CCCCC2)c1ccc2ccccc2c1 ZINC000217933414 FI On-Demand Unstable TRY2_BOVIN 62 37 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc(S(N)(=O)=O)cc1 ZINC000217933415 HD For-Sale Unstable CA2 23 40 O=C(NCCCn1ccccc1=O)[C@@H](c1ccc(F)cc1)N1CCCCC1 ZINC000217933437 FF In-Stock Unstable ADRA1D 30 40 O=C(NCCCn1ccccc1=O)[C@@H](c1ccc(F)cc1)N1CCCCC1 ZINC000217933437 FF In-Stock Unstable ADRA1B 24 40 O=C(NCCCn1ccccc1=O)[C@@H](c1ccc(F)cc1)N1CCCCC1 ZINC000217933437 FF In-Stock Unstable KCNQ2 36 40 COc1ccc(/C=C\C(=O)CCl)c(OC)c1 ZINC000217933456 BF For-Sale Unstable PTGS2 0 48 COc1ccc(/C=C\C(=O)CCl)c(OC)c1 ZINC000217933456 BF For-Sale Unstable CYP1B1 67 60 COc1ccc(/C=C\C(=O)CCl)c(OC)c1 ZINC000217933456 BF For-Sale Unstable MTNR1A 41 41 COc1ccc(/C=C\C(=O)CCl)c(OC)c1 ZINC000217933456 BF For-Sale Unstable MTNR1B 33 41 COc1ccc(/C=C\C(=O)CCl)c(OC)c1 ZINC000217933456 BF For-Sale Unstable CYP1A1 55 60 COc1ccc(/C=C\C(=O)CCl)c(OC)c1 ZINC000217933456 BF For-Sale Unstable CYP1A2 23 60 COc1ccc(/C=C\C(=O)CCl)c(OC)c1 ZINC000217933456 BF For-Sale Unstable ABCG2 22 50 COc1ccc(/C=C\C(=O)CCl)c(OC)c1 ZINC000217933456 BF For-Sale Unstable AKR1B10 32 42 COc1ccc(/C=C\C(=O)CCl)c(OC)c1 ZINC000217933456 BF For-Sale Unstable CYSP_PLAFA 66 57 CCCC(CCC)C(=O)O[C@H]1C[C@H]2CC[C@@]1(C)C2(C)C ZINC000217933458 CJ For-Sale Unstable ELANE 0 46 CC(C)C[C@@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccccc4)oc3c21 ZINC000217933460 FJ In-Stock Unstable CYP1B1 19 41 CC(C)C[C@@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccccc4)oc3c21 ZINC000217933460 FJ In-Stock Unstable CYP1A1 27 50 CC(C)C[C@@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccccc4)oc3c21 ZINC000217933460 FJ In-Stock Unstable ABCB1 15 43 CC(C)C[C@@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccccc4)oc3c21 ZINC000217933460 FJ In-Stock Unstable CYP1A2 20 50 O=C(NCCCn1ccccc1=O)[C@H](c1ccc(F)cc1)N1CCCCC1 ZINC000217933503 FF In-Stock Unstable ADRA1D 30 40 O=C(NCCCn1ccccc1=O)[C@H](c1ccc(F)cc1)N1CCCCC1 ZINC000217933503 FF In-Stock Unstable ADRA1B 24 40 O=C(NCCCn1ccccc1=O)[C@H](c1ccc(F)cc1)N1CCCCC1 ZINC000217933503 FF In-Stock Unstable KCNQ2 36 40 Cc1ccc([N+](=O)[O-])cc1S(=O)(=O)Nc1nc2c(s1)CCCCC2 ZINC000217933505 FG On-Demand Unstable PIK3CA 0 44 Cc1ccc([N+](=O)[O-])cc1S(=O)(=O)Nc1nc2c(s1)CCCCC2 ZINC000217933505 FG On-Demand Unstable NFKBIA 0 48 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cc2ccccc2[nH]1 ZINC000217933525 GG For-Sale Unstable HRH4 16 44 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cc2ccccc2[nH]1 ZINC000217933525 GG For-Sale Unstable AKR1C3 32 42 COc1cccc(/C=C/NC(=O)Nc2ccc([N+](=O)[O-])cc2OC)c1 ZINC000217933527 EG For-Sale Unstable CACNA1D 46 34 COc1cccc(/C=C/NC(=O)Nc2ccc([N+](=O)[O-])cc2OC)c1 ZINC000217933527 EG For-Sale Unstable KCNMA1 23 51 COc1cccc(/C=C/NC(=O)Nc2ccc([N+](=O)[O-])cc2OC)c1 ZINC000217933527 EG For-Sale Unstable TAAR1 22 44 COc1cccc(/C=C/NC(=O)Nc2ccc([N+](=O)[O-])cc2OC)c1 ZINC000217933527 EG For-Sale Unstable TRPM8 0 52 COc1cccc(/C=C/NC(=O)Nc2ccc([N+](=O)[O-])cc2OC)c1 ZINC000217933527 EG For-Sale Unstable AKR1C2 15 42 CC(C)C[C@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccccc4)oc3c21 ZINC000217933546 FJ In-Stock Unstable CYP1B1 19 41 CC(C)C[C@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccccc4)oc3c21 ZINC000217933546 FJ In-Stock Unstable CYP1A1 26 50 CC(C)C[C@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccccc4)oc3c21 ZINC000217933546 FJ In-Stock Unstable ABCB1 15 43 CC(C)C[C@H]1CC(=O)Oc2cc(O)c3c(=O)cc(-c4ccccc4)oc3c21 ZINC000217933546 FJ In-Stock Unstable CYP1A2 19 50 Cc1ccc(S(=O)(=O)Nc2nc3c(s2)CCCCC3)cc1 ZINC000217933589 DH On-Demand Unstable CA1 19 48 Cc1ccc(S(=O)(=O)Nc2nc3c(s2)CCCCC3)cc1 ZINC000217933589 DH On-Demand Unstable CA4 27 48 Cc1ccc(S(=O)(=O)Nc2nc3c(s2)CCCCC3)cc1 ZINC000217933589 DH On-Demand Unstable FFAR4 26 41 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cc2ccccc2[nH]1 ZINC000217933598 GG For-Sale Unstable HRH4 16 44 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cc2ccccc2[nH]1 ZINC000217933598 GG For-Sale Unstable AKR1C3 32 42 O=C(/C=C\c1ccc2c(c1)CCO2)CCl ZINC000217933611 BE For-Sale Unstable GPR183 0 48 COc1ccc(CN2CCO[C@H](C)C2)cc1/C=C\C(=O)O ZINC000217933633 CE For-Sale Unstable DRD4 27 45 COc1ccc(CN2CCO[C@H](C)C2)cc1/C=C\C(=O)O ZINC000217933633 CE For-Sale Unstable DRD3 15 40 COc1cccc(/C=C/NC(=O)Nc2ccc([N+](=O)[O-])cc2)c1 ZINC000217933637 DG For-Sale Unstable MTNR1A 21 46 COc1cccc(/C=C/NC(=O)Nc2ccc([N+](=O)[O-])cc2)c1 ZINC000217933637 DG For-Sale Unstable MTNR1B 28 46 COc1cccc(/C=C/NC(=O)Nc2ccc([N+](=O)[O-])cc2)c1 ZINC000217933637 DG For-Sale Unstable TAAR1 27 47 COc1cccc(/C=C/NC(=O)Nc2ccc([N+](=O)[O-])cc2)c1 ZINC000217933637 DG For-Sale Unstable AKR1C3 17 45 COc1cccc(/C=C/NC(=O)Nc2ccc([N+](=O)[O-])cc2)c1 ZINC000217933637 DG For-Sale Unstable TRPM8 0 56 COc1cccc(/C=C/NC(=O)Nc2ccc([N+](=O)[O-])cc2)c1 ZINC000217933637 DG For-Sale Unstable AKR1C2 37 45 COc1cccc(/C=C/NC(=O)Nc2ccc([N+](=O)[O-])cc2)c1 ZINC000217933637 DG For-Sale Unstable EXSA 0 40 CC1(C)CCc2cc(CC(=O)N[C@H](CO)c3ccccc3)ccc2O1 ZINC000217933649 EG In-Stock Unstable DAGLA 23 44 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cc2ccccc2[nH]1 ZINC000217933676 GG For-Sale Unstable HRH4 16 44 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cc2ccccc2[nH]1 ZINC000217933676 GG For-Sale Unstable AKR1C3 32 42 O=C(c1cccnc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217933721 CD On-Demand Unstable HRH3 26 45 O=C(c1cccnc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217933721 CD On-Demand Unstable CCR3 21 42 O=C(c1cccnc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217933721 CD On-Demand Unstable L3MBTL1 0 60 O=C(c1cccnc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217933721 CD On-Demand Unstable L3MBTL3 103 60 O=C(c1cccnc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217933721 CD On-Demand Unstable L3MBTL4 0 43 O=C(c1cccnc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217933721 CD On-Demand Unstable MBTD1 0 53 O=C(c1cccnc1O)N1CC[C@@H](N2CCCCC2)C1 ZINC000217933721 CD On-Demand Unstable TP53BP1 0 60 COc1ccc(CN2CCO[C@@H](C)C2)cc1/C=C\C(=O)O ZINC000217933730 CE For-Sale Unstable DRD4 27 45 COc1ccc(CN2CCO[C@@H](C)C2)cc1/C=C\C(=O)O ZINC000217933730 CE For-Sale Unstable DRD3 15 40 Cn1cccc1[C@H](O)CCNC(=O)c1ccc(Cl)s1 ZINC000217933740 CF In-Stock Unstable F10 23 46 COc1cccc(/C=C/NC(=O)Nc2cccc([N+](=O)[O-])c2)c1 ZINC000217933744 DG For-Sale Unstable CACNA1D 67 36 COc1cccc(/C=C/NC(=O)Nc2cccc([N+](=O)[O-])c2)c1 ZINC000217933744 DG For-Sale Unstable MTNR1A 18 43 COc1cccc(/C=C/NC(=O)Nc2cccc([N+](=O)[O-])c2)c1 ZINC000217933744 DG For-Sale Unstable MTNR1B 25 43 COc1cccc(/C=C/NC(=O)Nc2cccc([N+](=O)[O-])c2)c1 ZINC000217933744 DG For-Sale Unstable TAAR1 33 57 COc1cccc(/C=C/NC(=O)Nc2cccc([N+](=O)[O-])c2)c1 ZINC000217933744 DG For-Sale Unstable AKR1C3 17 52 COc1cccc(/C=C/NC(=O)Nc2cccc([N+](=O)[O-])c2)c1 ZINC000217933744 DG For-Sale Unstable DDX3X 0 48 COc1cccc(/C=C/NC(=O)Nc2cccc([N+](=O)[O-])c2)c1 ZINC000217933744 DG For-Sale Unstable TRPM8 0 67 COc1cccc(/C=C/NC(=O)Nc2cccc([N+](=O)[O-])c2)c1 ZINC000217933744 DG For-Sale Unstable AKR1C2 28 52 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cc2ccccc2[nH]1 ZINC000217933756 GG For-Sale Unstable HRH4 16 44 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cc2ccccc2[nH]1 ZINC000217933756 GG For-Sale Unstable AKR1C3 32 42 O=S(=O)(Nc1nc2c(s1)CCCCC2)c1ccc(F)cc1F ZINC000217933761 EG On-Demand Unstable SLC27A1 37 41 O=C(c1cccnc1O)N1CC[C@H](N2CCCCC2)C1 ZINC000217933801 CD On-Demand Unstable HRH3 26 45 O=C(c1cccnc1O)N1CC[C@H](N2CCCCC2)C1 ZINC000217933801 CD On-Demand Unstable CCR3 21 42 O=C(c1cccnc1O)N1CC[C@H](N2CCCCC2)C1 ZINC000217933801 CD On-Demand Unstable L3MBTL1 0 60 O=C(c1cccnc1O)N1CC[C@H](N2CCCCC2)C1 ZINC000217933801 CD On-Demand Unstable L3MBTL3 103 60 O=C(c1cccnc1O)N1CC[C@H](N2CCCCC2)C1 ZINC000217933801 CD On-Demand Unstable L3MBTL4 0 43 O=C(c1cccnc1O)N1CC[C@H](N2CCCCC2)C1 ZINC000217933801 CD On-Demand Unstable MBTD1 0 53 O=C(c1cccnc1O)N1CC[C@H](N2CCCCC2)C1 ZINC000217933801 CD On-Demand Unstable TP53BP1 0 60 Cn1cccc1[C@@H](O)CCNC(=O)c1ccc(Cl)s1 ZINC000217933824 CF In-Stock Unstable F10 23 46 O=S(=O)(Nc1nc2c(s1)CCCCC2)c1cc(F)cc(F)c1 ZINC000217933847 EG On-Demand Unstable SLC27A1 37 42 COc1cccc(/C=C/NC(=O)Nc2cc([N+](=O)[O-])ccc2Cl)c1 ZINC000217933848 EI For-Sale Unstable TAAR1 23 44 COc1cccc(/C=C/NC(=O)Nc2cc([N+](=O)[O-])ccc2Cl)c1 ZINC000217933848 EI For-Sale Unstable TRPM8 0 52 COc1cccc(/C=C/NC(=O)Nc2cc([N+](=O)[O-])ccc2Cl)c1 ZINC000217933848 EI For-Sale Unstable AKR1C2 15 42 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217933905 FI In-Stock Unstable KCNQ2 22 45 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217933905 FI In-Stock Unstable PYGL 25 45 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccc3c(c2)OCO3)cc1 ZINC000217933905 FI In-Stock Unstable DYRK2 48 35 O=S(=O)(Nc1nc2c(s1)CCCCC2)c1ccc(F)c(F)c1 ZINC000217933923 EG On-Demand Unstable CA2 16 41 O=S(=O)(Nc1nc2c(s1)CCCCC2)c1ccc(F)c(F)c1 ZINC000217933923 EG On-Demand Unstable CA4 16 41 COc1ccc2occ([C@H](CC(=O)NCCc3ccc(O)c(O)c3)c3c(O)nc4ccccn4c3=O)c(=O)c2c1 ZINC000217933959 KF In-Stock Unstable MTNR1A 48 40 COc1cccc(/C=C/NC(=O)NCCCl)c1 ZINC000217933965 CE For-Sale Unstable DRD4 44 34 COc1cccc(/C=C/NC(=O)NCCCl)c1 ZINC000217933965 CE For-Sale Unstable CYP1B1 34 41 COc1cccc(/C=C/NC(=O)NCCCl)c1 ZINC000217933965 CE For-Sale Unstable AHR 15 46 COc1cccc(/C=C/NC(=O)NCCCl)c1 ZINC000217933965 CE For-Sale Unstable MTNR1A 86 46 COc1cccc(/C=C/NC(=O)NCCCl)c1 ZINC000217933965 CE For-Sale Unstable MTNR1B 78 46 COc1cccc(/C=C/NC(=O)NCCCl)c1 ZINC000217933965 CE For-Sale Unstable CYP1A1 26 44 COc1cc(CNC2CCN(C(=O)OC(C)(C)C)CC2)ccn1 ZINC000217933992 DF On-Demand Unstable GPR119 40 36 O=C(/C=C/c1ccc2c(c1)OCO2)NCCCN1CCCc2ccccc21 ZINC000217934017 FG In-Stock Unstable DRD3 18 58 O=C(/C=C/c1ccc2c(c1)OCO2)NCCCN1CCCc2ccccc21 ZINC000217934017 FG In-Stock Unstable DYRK2 54 36 O=C(/C=C\c1c[nH]c2cc(Cl)ccc12)CCl ZINC000217934034 CH For-Sale Unstable TDO2 0 51 COc1ccc2occ([C@@H](CC(=O)NCCc3ccc(O)c(O)c3)c3c(O)nc4ccccn4c3=O)c(=O)c2c1 ZINC000217934040 KF In-Stock Unstable MTNR1A 48 40 Nc1[nH]nc(C(=O)N2CCC[C@@H]2c2ccccn2)c1Cl ZINC000217934069 CE In-Stock Unstable COLA 57 37 Nc1[nH]nc(C(=O)N2CCC[C@@H]2c2ccccn2)c1Cl ZINC000217934069 CE In-Stock Unstable CPT1A 54 37 COc1cccc(/C=C/NC(=O)N2CCN(c3ccc(F)cc3)CC2)c1 ZINC000217934075 FG For-Sale Unstable DRD4 47 40 COc1cccc(/C=C/NC(=O)N2CCN(c3ccc(F)cc3)CC2)c1 ZINC000217934075 FG For-Sale Unstable ABCB1 0 41 Cc1cccc(S(=O)(=O)Nc2nc3c(s2)CCCCC3)c1 ZINC000217934090 DH On-Demand Unstable SLC27A1 22 40 Cn1cccc1[C@H](O)CCNC(=O)Cc1ccccc1Cl ZINC000217934099 DE In-Stock Unstable CXCL8 41 33 CN[C@H]1CCCN(CCS(=O)(=O)C(C)C)C1 ZINC000217934115 BC For-Sale Unstable BIRC2 44 35 CN1CCC(Oc2ccc(NC(=O)/C=C/c3ccc4c(c3)OCO4)cc2)CC1 ZINC000217934123 GH In-Stock Unstable PRSS2 64 32 CN1CCC(Oc2ccc(NC(=O)/C=C/c3ccc4c(c3)OCO4)cc2)CC1 ZINC000217934123 GH In-Stock Unstable DYRK2 68 38 Nc1[nH]nc(C(=O)N2CCC[C@H]2c2ccccn2)c1Cl ZINC000217934142 CE In-Stock Unstable COLA 57 37 Nc1[nH]nc(C(=O)N2CCC[C@H]2c2ccccn2)c1Cl ZINC000217934142 CE In-Stock Unstable CPT1A 54 37 O=C(CCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)Nc1nccs1 ZINC000217934150 HG In-Stock Unstable MAP 0 41 O=C(CCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@H]12)Nc1nccs1 ZINC000217934150 HG In-Stock Unstable MAP1 82 39 Cn1cccc1[C@@H](O)CCNC(=O)Cc1ccccc1Cl ZINC000217934176 DE In-Stock Unstable CXCL8 41 33 CN[C@@H]1CCCN(CCS(=O)(=O)C(C)C)C1 ZINC000217934188 BC For-Sale Unstable BIRC2 44 35 COc1cccc(/C=C/NC(=O)Nc2ccccc2O)c1 ZINC000217934189 CG For-Sale Unstable CYP1B1 27 40 COc1cccc(/C=C/NC(=O)Nc2ccccc2O)c1 ZINC000217934189 CG For-Sale Unstable MTNR1A 34 42 COc1cccc(/C=C/NC(=O)Nc2ccccc2O)c1 ZINC000217934189 CG For-Sale Unstable MTNR1B 34 42 COc1cccc(/C=C/NC(=O)Nc2ccccc2O)c1 ZINC000217934189 CG For-Sale Unstable CYP1A1 16 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)Cn1cccn1 ZINC000217934203 ED For-Sale Unstable HCRTR2 41 35 O=C(CCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)Nc1nccs1 ZINC000217934218 HG In-Stock Unstable MAP 0 41 O=C(CCN1C(=O)c2ccccc2N2C(=O)c3ccccc3[C@@H]12)Nc1nccs1 ZINC000217934218 HG In-Stock Unstable MAP1 82 39 CN(Cc1ccncc1)Cc1ccccc1/C=C\C(=O)O ZINC000217934227 CF For-Sale Unstable PTGER2 52 46 CN(Cc1ccncc1)Cc1ccccc1/C=C\C(=O)O ZINC000217934227 CF For-Sale Unstable PTGER3 21 47 CN1CCN(c2ccc(CNC(=O)/C=C/c3ccc4c(c3)OCO4)cc2)CC1 ZINC000217934250 GE In-Stock Unstable NOS2 60 35 CN1CCN(c2ccc(CNC(=O)/C=C/c3ccc4c(c3)OCO4)cc2)CC1 ZINC000217934250 GE In-Stock Unstable HDAC1 36 47 CN1CCN(c2ccc(CNC(=O)/C=C/c3ccc4c(c3)OCO4)cc2)CC1 ZINC000217934250 GE In-Stock Unstable DYRK2 56 38 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)Cn1cccn1 ZINC000217934286 ED For-Sale Unstable HCRTR2 41 35 CCOc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217934295 DH For-Sale Unstable CYP1B1 18 40 CCOc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217934295 DH For-Sale Unstable AHR 21 44 CCOc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217934295 DH For-Sale Unstable MTNR1A 51 47 CCOc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217934295 DH For-Sale Unstable MTNR1B 50 50 CCOc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217934295 DH For-Sale Unstable AKR1C2 41 33 O=S(=O)(Nc1nc2c(s1)CCCCC2)c1cccc(Cl)c1 ZINC000217934350 EH On-Demand Unstable FBP1 26 44 COc1ccc(/C=C\c2csc(N)n2)c(OC)c1 ZINC000217934365 CF For-Sale Unstable CYP1B1 63 59 COc1ccc(/C=C\c2csc(N)n2)c(OC)c1 ZINC000217934365 CF For-Sale Unstable CYP1A1 55 59 COc1ccc(/C=C\c2csc(N)n2)c(OC)c1 ZINC000217934365 CF For-Sale Unstable CYP1A2 22 59 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)Cn1cccn1 ZINC000217934368 ED For-Sale Unstable HCRTR2 41 35 CCCC[C@@H](C(=O)OC)N1CCC[C@@H](OCC)C1 ZINC000217934374 CE On-Demand Unstable GBA2 44 32 S=C(NCCSCc1cccc(Cl)c1)Nc1ccccc1 ZINC000217934379 EJ In-Stock Unstable CACNA2D1 0 47 CCCCOC(=O)c1ccccc1NC(=O)N/C=C/c1cccc(OC)c1 ZINC000217934404 FI For-Sale Unstable MTNR1A 41 40 CCCCOC(=O)c1ccccc1NC(=O)N/C=C/c1cccc(OC)c1 ZINC000217934404 FI For-Sale Unstable MTNR1B 40 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)Cn1cccn1 ZINC000217934450 ED For-Sale Unstable HCRTR2 41 35 CN(Cc1ccncc1)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217934455 CF For-Sale Unstable PTGER2 24 40 CN(Cc1ccncc1)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217934455 CF For-Sale Unstable NR1H4 42 37 CN(Cc1ccncc1)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217934455 CF For-Sale Unstable AKR1C3 41 40 Cc1ccc(C)c(S(=O)(=O)Nc2nc3c(s2)CCCCC3)c1 ZINC000217934458 EH On-Demand Unstable SLC27A1 24 41 CCCC[C@H](C(=O)OC)N1CCC[C@@H](OCC)C1 ZINC000217934466 CE On-Demand Unstable GBA2 44 32 CN(C)S(=O)(=O)c1ccc2c(c1)CCN2C(=S)Nc1ccccc1 ZINC000217934512 FF In-Stock Unstable BETA-TUBULIN 0 42 COc1cccc(/C=C/NC(=O)Nc2ccc(C(C)=O)cc2)c1 ZINC000217934516 DH For-Sale Unstable CA1 17 42 COc1cccc(/C=C/NC(=O)Nc2ccc(C(C)=O)cc2)c1 ZINC000217934516 DH For-Sale Unstable MTNR1A 28 50 COc1cccc(/C=C/NC(=O)Nc2ccc(C(C)=O)cc2)c1 ZINC000217934516 DH For-Sale Unstable MTNR1B 34 50 COc1cccc(/C=C/NC(=O)Nc2ccc(C(C)=O)cc2)c1 ZINC000217934516 DH For-Sale Unstable ACR 32 44 COc1cccc(/C=C/NC(=O)Nc2ccc(C(C)=O)cc2)c1 ZINC000217934516 DH For-Sale Unstable TAAR1 30 43 COc1cccc(/C=C/NC(=O)Nc2ccc(C(C)=O)cc2)c1 ZINC000217934516 DH For-Sale Unstable AKR1C3 29 43 COc1cccc(/C=C/NC(=O)Nc2ccc(C(C)=O)cc2)c1 ZINC000217934516 DH For-Sale Unstable AKR1C2 46 43 COc1cccc(/C=C/NC(=O)Nc2ccc(C(C)=O)cc2)c1 ZINC000217934516 DH For-Sale Unstable IMDH_CRYPV 20 40 COc1cc2oc(=O)cc(C)c2cc1CCC(=O)N[C@@H](CC(C)C)c1nc2ccccc2[nH]1 ZINC000217934534 IJ In-Stock Unstable MMP7 20 40 CCN(CCO)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217934573 CD For-Sale Unstable ERG2 18 44 COc1cccc(/C=C/NC(=O)Nc2cccc(C(C)=O)c2)c1 ZINC000217934613 DH For-Sale Unstable CYP1B1 27 42 COc1cccc(/C=C/NC(=O)Nc2cccc(C(C)=O)c2)c1 ZINC000217934613 DH For-Sale Unstable MTNR1A 29 47 COc1cccc(/C=C/NC(=O)Nc2cccc(C(C)=O)c2)c1 ZINC000217934613 DH For-Sale Unstable MTNR1B 34 47 COc1cccc(/C=C/NC(=O)Nc2cccc(C(C)=O)c2)c1 ZINC000217934613 DH For-Sale Unstable CYP1A1 22 42 COc1cccc(/C=C/NC(=O)Nc2cccc(C(C)=O)c2)c1 ZINC000217934613 DH For-Sale Unstable TAAR1 33 45 COc1cccc(/C=C/NC(=O)Nc2cccc(C(C)=O)c2)c1 ZINC000217934613 DH For-Sale Unstable AKR1C3 38 45 COc1cccc(/C=C/NC(=O)Nc2cccc(C(C)=O)c2)c1 ZINC000217934613 DH For-Sale Unstable KCNK3 77 48 COc1cccc(/C=C/NC(=O)Nc2cccc(C(C)=O)c2)c1 ZINC000217934613 DH For-Sale Unstable KCNK9 44 34 Cc1[nH]c2ccccc2c1C(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217934618 CE For-Sale Unstable SSTR3 26 41 COc1cc(CNC(=S)Nc2ccccc2)ccc1OC(C)C ZINC000217934632 EH In-Stock Unstable TRPV1 29 45 COc1cc2nc(C)n(CC(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)c(=O)c2cc1OC ZINC000217934638 JD In-Stock Unstable CHRNA4 26 42 COC(=O)c1ccc(C(=O)NCC[C@@H](O)c2cccn2C)cc1 ZINC000217934664 DD In-Stock Unstable EPHX2 15 40 Cc1[nH]c2ccccc2c1C(=O)N[C@H]1CCC[C@@H]1CO ZINC000217934696 CE For-Sale Unstable SSTR3 26 41 CCCC[C@@H](C(=O)OC)N1CCC[C@@H](OCCC)C1 ZINC000217934717 CF For-Sale Unstable GBA2 45 33 COC(=O)c1ccc(C(=O)NCC[C@H](O)c2cccn2C)cc1 ZINC000217934749 DD In-Stock Unstable EPHX2 15 40 Cc1[nH]c2ccccc2c1C(=O)N[C@@H]1CCC[C@H]1CO ZINC000217934767 CE For-Sale Unstable SSTR3 26 41 COc1ccc(/C=C\c2csc(N)n2)cc1F ZINC000217934787 CG For-Sale Unstable TUBB1 39 52 CCCC[C@H](C(=O)OC)N1CCC[C@@H](OCCC)C1 ZINC000217934798 CF For-Sale Unstable GBA2 45 33 Cc1ccc(S(=O)(=O)Nc2nc3c(s2)CCCCC3)c(C)c1 ZINC000217934801 EH On-Demand Unstable SLC27A1 24 41 COc1cccc(/C=C/NC(=O)Nc2cccc(C)c2C)c1 ZINC000217934824 CI For-Sale Unstable MTNR1A 27 41 COc1cccc(/C=C/NC(=O)Nc2cccc(C)c2C)c1 ZINC000217934824 CI For-Sale Unstable MTNR1B 29 41 Cc1[nH]c2ccccc2c1C(=O)N[C@H]1CCC[C@H]1CO ZINC000217934854 CE For-Sale Unstable SSTR3 26 41 S=C(NCCCc1ccc(Cl)cc1)Nc1ccccc1 ZINC000217934861 DI In-Stock Unstable EPHX1 0 45 S=C(NCCCc1ccc(Cl)cc1)Nc1ccccc1 ZINC000217934861 DI In-Stock Unstable ADRB1 17 49 S=C(NCCCc1ccc(Cl)cc1)Nc1ccccc1 ZINC000217934861 DI In-Stock Unstable ADRB3 17 49 S=C(NCCCc1ccc(Cl)cc1)Nc1ccccc1 ZINC000217934861 DI In-Stock Unstable SLC6A5 15 42 CCOC(=O)c1ccc(S(=O)(=O)Nc2nc3c(s2)CCCCC3)cc1 ZINC000217934882 GG On-Demand Unstable CA2 19 46 CCOC(=O)c1ccc(S(=O)(=O)Nc2nc3c(s2)CCCCC3)cc1 ZINC000217934882 GG On-Demand Unstable CA1 18 46 CCOC(=O)c1ccc(S(=O)(=O)Nc2nc3c(s2)CCCCC3)cc1 ZINC000217934882 GG On-Demand Unstable CA4 34 46 CCOC(=O)c1ccc(S(=O)(=O)Nc2nc3c(s2)CCCCC3)cc1 ZINC000217934882 GG On-Demand Unstable NS5B 0 41 CCOC(=O)c1ccc(S(=O)(=O)Nc2nc3c(s2)CCCCC3)cc1 ZINC000217934882 GG On-Demand Unstable SLC27A1 35 40 CCCCN(CCO)Cc1ccc(/C=C\C(=O)O)cc1 ZINC000217934892 CE For-Sale Unstable PLM2_PLAFA 57 38 COc1cccc(/C=C/NC(=O)Nc2ccc(C)cc2C)c1 ZINC000217934942 CI For-Sale Unstable MTNR1A 26 40 COc1cccc(/C=C/NC(=O)Nc2ccc(C)cc2C)c1 ZINC000217934942 CI For-Sale Unstable MTNR1B 28 40 Fc1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217934969 CH In-Stock Unstable ADRB1 16 49 Fc1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217934969 CH In-Stock Unstable ADRB3 17 49 Fc1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217934969 CH In-Stock Unstable CCR3 20 46 COc1cccc(/C=C/NC(=O)Nc2cc(C)ccc2OC)c1 ZINC000217935043 DH For-Sale Unstable CYP1B1 40 37 COc1cccc(/C=C/NC(=O)Nc2cc(C)ccc2OC)c1 ZINC000217935043 DH For-Sale Unstable MTNR1A 26 42 COc1cccc(/C=C/NC(=O)Nc2cc(C)ccc2OC)c1 ZINC000217935043 DH For-Sale Unstable MTNR1B 30 42 COc1cccc(/C=C/NC(=O)Nc2cc(C)ccc2OC)c1 ZINC000217935043 DH For-Sale Unstable CYP1A1 27 42 COc1cccc(/C=C/NC(=O)Nc2cc(C)ccc2OC)c1 ZINC000217935043 DH For-Sale Unstable ABCG2 16 43 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)NCCc3ccccc3)[C@H]21 ZINC000217935062 JH In-Stock Unstable TSHR 48 35 COc1ccccc1CCCNC(=S)Nc1ccccc1 ZINC000217935065 DH In-Stock Unstable EPHX1 0 41 COc1ccccc1CCCNC(=S)Nc1ccccc1 ZINC000217935065 DH In-Stock Unstable MTNR1A 28 40 COc1ccccc1CCCNC(=S)Nc1ccccc1 ZINC000217935065 DH In-Stock Unstable MTNR1B 41 41 COc1ccccc1CCCNC(=S)Nc1ccccc1 ZINC000217935065 DH In-Stock Unstable QPCT 38 41 C/C(CCc1ccccc1)=C1\CC(=O)NC1=O ZINC000217935110 BD For-Sale Unstable SLC12A5 18 40 CCCCN(CCO)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217935123 CE For-Sale Unstable AKR1C3 29 44 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CCC(=O)NCCc3ccccc3)[C@@H]21 ZINC000217935141 JH In-Stock Unstable TSHR 48 35 COc1cccc(/C=C/NC(=O)Nc2cccc(C)c2)c1 ZINC000217935142 CH For-Sale Unstable CCKAR 27 45 COc1cccc(/C=C/NC(=O)Nc2cccc(C)c2)c1 ZINC000217935142 CH For-Sale Unstable KDR 20 41 COc1cccc(/C=C/NC(=O)Nc2cccc(C)c2)c1 ZINC000217935142 CH For-Sale Unstable MTNR1A 28 47 COc1cccc(/C=C/NC(=O)Nc2cccc(C)c2)c1 ZINC000217935142 CH For-Sale Unstable MTNR1B 33 47 COc1cccc(/C=C/NC(=O)Nc2cccc(C)c2)c1 ZINC000217935142 CH For-Sale Unstable CCKBR 27 45 COc1cccc(/C=C/NC(=O)Nc2cccc(C)c2)c1 ZINC000217935142 CH For-Sale Unstable TAAR1 31 41 COc1cccc(/C=C/NC(=O)Nc2cccc(C)c2)c1 ZINC000217935142 CH For-Sale Unstable AKR1C3 16 47 COc1cccc(/C=C/NC(=O)Nc2cccc(C)c2)c1 ZINC000217935142 CH For-Sale Unstable AKR1C2 33 47 COc1cccc(/C=C/NC(=O)Nc2cccc(C)c2)c1 ZINC000217935142 CH For-Sale Unstable KCNK3 76 52 COc1cccc(/C=C/NC(=O)Nc2cccc(C)c2)c1 ZINC000217935142 CH For-Sale Unstable KCNK9 62 39 O=S(=O)(Nc1nc2c(s1)CCCCC2)c1ccc(Cl)s1 ZINC000217935172 EH On-Demand Unstable CCR4 52 33 COc1cccc(CCCNC(=S)Nc2ccccc2)c1 ZINC000217935183 DH In-Stock Unstable EPHX1 0 40 COc1cccc(CCCNC(=S)Nc2ccccc2)c1 ZINC000217935183 DH In-Stock Unstable ADRB1 18 50 COc1cccc(CCCNC(=S)Nc2ccccc2)c1 ZINC000217935183 DH In-Stock Unstable HRH2 28 44 COc1cccc(CCCNC(=S)Nc2ccccc2)c1 ZINC000217935183 DH In-Stock Unstable GRIN2B 0 40 COc1cccc(CCCNC(=S)Nc2ccccc2)c1 ZINC000217935183 DH In-Stock Unstable ADRB3 20 50 COc1cccc(CCCNC(=S)Nc2ccccc2)c1 ZINC000217935183 DH In-Stock Unstable FDFT1 15 46 COc1cccc(CCCNC(=S)Nc2ccccc2)c1 ZINC000217935183 DH In-Stock Unstable CCR3 15 43 COc1cccc(CCCNC(=S)Nc2ccccc2)c1 ZINC000217935183 DH In-Stock Unstable MTNR1A 50 62 COc1cccc(CCCNC(=S)Nc2ccccc2)c1 ZINC000217935183 DH In-Stock Unstable MTNR1B 42 62 COc1cccc(CCCNC(=S)Nc2ccccc2)c1 ZINC000217935183 DH In-Stock Unstable ABCB1 0 45 COc1cccc(CCCNC(=S)Nc2ccccc2)c1 ZINC000217935183 DH In-Stock Unstable AMP1_PLAFQ 24 46 COc1cccc(CCCNC(=S)Nc2ccccc2)c1 ZINC000217935183 DH In-Stock Unstable FPR2 15 41 COc1cccc(CCCNC(=S)Nc2ccccc2)c1 ZINC000217935183 DH In-Stock Unstable QPCT 48 45 COc1cccc(CCCNC(=S)Nc2ccccc2)c1 ZINC000217935183 DH In-Stock Unstable NCE103 22 41 COc1cccc(CCCNC(=S)Nc2ccccc2)c1 ZINC000217935183 DH In-Stock Unstable CRTM 69 46 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc2cc[nH]c2c1 ZINC000217935248 GG For-Sale Unstable GHSR 16 51 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)c1 ZINC000217935252 FK For-Sale Unstable GUAB 0 47 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)c1 ZINC000217935252 FK For-Sale Unstable RAF1 43 51 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)c1 ZINC000217935252 FK For-Sale Unstable MTNR1A 15 41 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)c1 ZINC000217935252 FK For-Sale Unstable MTNR1B 21 41 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)c1 ZINC000217935252 FK For-Sale Unstable Q8MMZ8_EIMTE 68 51 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)c1 ZINC000217935252 FK For-Sale Unstable BRAF 17 41 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)c1 ZINC000217935252 FK For-Sale Unstable TAAR1 25 43 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)c1 ZINC000217935252 FK For-Sale Unstable IMDH_CRYPV 48 49 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)c1 ZINC000217935252 FK For-Sale Unstable BLM 0 42 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable ACE 29 46 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable OPRM1 40 52 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable OPRD1 44 51 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable MME 75 48 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable ANPEP 27 44 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable NPR1 41 36 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable TACR1 20 48 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable FCER2 42 35 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable TACR2 32 49 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable KLK3 17 41 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable PAPA1_CARPA 61 45 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable CYSP_TRYCR 40 35 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable CCKAR 19 44 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable CTSK 25 45 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable CTSL 54 51 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable NPFFR2 23 41 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable TACR3 34 57 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable GRIA1 21 42 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable REN 16 44 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable PCSK5 39 43 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable FURIN 77 52 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable CCKBR 18 42 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable CTSS 35 51 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable CAPN1 35 41 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable CAPN2 41 36 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable ACE2 48 34 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable FPR1 66 46 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable NPR 59 34 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable AMP1_PLAFQ 43 31 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable PSMB5 46 42 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable BLA1_STEMA 41 39 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable KISS1R 55 35 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable POLG_WNV 59 37 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable NPFFR1 32 41 COC(=O)CNC(=O)[C@@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935296 EC On-Demand Unstable PDS 44 33 COc1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217935297 DH In-Stock Unstable EPHX1 0 43 COc1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217935297 DH In-Stock Unstable ADRB2 15 54 COc1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217935297 DH In-Stock Unstable ADRB1 23 54 COc1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217935297 DH In-Stock Unstable ADRB3 32 54 COc1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217935297 DH In-Stock Unstable BMP1 23 41 COc1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217935297 DH In-Stock Unstable CA1 23 42 COc1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217935297 DH In-Stock Unstable SIGMAR1 15 51 COc1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217935297 DH In-Stock Unstable SCN2A 32 46 COc1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217935297 DH In-Stock Unstable MTNR1A 40 43 COc1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217935297 DH In-Stock Unstable MTNR1B 43 45 COc1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217935297 DH In-Stock Unstable QPCT 40 53 COc1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217935297 DH In-Stock Unstable NCE103 17 42 COc1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217935297 DH In-Stock Unstable CRTM 40 37 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc2cc[nH]c2c1 ZINC000217935333 GG For-Sale Unstable GHSR 16 51 CN(Cc1ccoc1)Cc1ccccc1/C=C\C(=O)O ZINC000217935337 CG For-Sale Unstable PTGER2 45 44 CN(Cc1ccoc1)Cc1ccccc1/C=C\C(=O)O ZINC000217935337 CG For-Sale Unstable PTGER4 23 46 CN(Cc1ccoc1)Cc1ccccc1/C=C\C(=O)O ZINC000217935337 CG For-Sale Unstable PTGER3 18 48 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable ACE 29 46 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable OPRM1 40 52 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable OPRD1 44 51 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable MME 75 48 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable ANPEP 27 44 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable NPR1 41 36 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable TACR1 20 48 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable FCER2 42 35 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable TACR2 32 49 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable KLK3 17 41 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable PAPA1_CARPA 61 45 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable CYSP_TRYCR 40 35 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable CCKAR 19 44 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable CTSK 25 45 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable CTSL 54 51 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable NPFFR2 23 41 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable TACR3 34 57 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable GRIA1 21 42 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable REN 16 44 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable PCSK5 39 43 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable FURIN 77 52 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable CCKBR 18 42 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable CTSS 35 51 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable CAPN1 35 41 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable CAPN2 41 36 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable ACE2 48 34 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable FPR1 66 46 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable NPR 59 34 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable AMP1_PLAFQ 43 31 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable PSMB5 46 42 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable BLA1_STEMA 41 39 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable KISS1R 55 35 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable POLG_WNV 59 37 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable NPFFR1 32 41 COC(=O)CNC(=O)[C@H](CCSC)NC(=O)Cc1ccccc1 ZINC000217935356 EC On-Demand Unstable PDS 44 33 COc1ccc(OC[C@@H](C)NC(=S)Nc2ccccc2)cc1 ZINC000217935403 DG In-Stock Unstable EPHX1 0 42 COc1ccc(OC[C@@H](C)NC(=S)Nc2ccccc2)cc1 ZINC000217935403 DG In-Stock Unstable ADRB2 21 53 COc1ccc(OC[C@@H](C)NC(=S)Nc2ccccc2)cc1 ZINC000217935403 DG In-Stock Unstable ADRB1 28 53 COc1ccc(OC[C@@H](C)NC(=S)Nc2ccccc2)cc1 ZINC000217935403 DG In-Stock Unstable ADRB3 31 53 COc1ccc(OC[C@@H](C)NC(=S)Nc2ccccc2)cc1 ZINC000217935403 DG In-Stock Unstable SDH1 0 41 COc1ccc(OC[C@@H](C)NC(=S)Nc2ccccc2)cc1 ZINC000217935403 DG In-Stock Unstable O69638_MYCTO 0 46 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc2cc[nH]c2c1 ZINC000217935424 GG For-Sale Unstable GHSR 16 51 COc1cccc(/C=C/NC(=O)Nc2ccc(N)c(Cl)c2)c1 ZINC000217935471 DH For-Sale Unstable MTNR1A 21 43 COc1cccc(/C=C/NC(=O)Nc2ccc(N)c(Cl)c2)c1 ZINC000217935471 DH For-Sale Unstable MTNR1B 25 43 COc1cccc(/C=C/NC(=O)Nc2ccc(N)c(Cl)c2)c1 ZINC000217935471 DH For-Sale Unstable TAAR1 21 41 COc1ccc(OC[C@H](C)NC(=S)Nc2ccccc2)cc1 ZINC000217935481 DG In-Stock Unstable EPHX1 0 42 COc1ccc(OC[C@H](C)NC(=S)Nc2ccccc2)cc1 ZINC000217935481 DG In-Stock Unstable ADRB2 21 53 COc1ccc(OC[C@H](C)NC(=S)Nc2ccccc2)cc1 ZINC000217935481 DG In-Stock Unstable ADRB1 28 53 COc1ccc(OC[C@H](C)NC(=S)Nc2ccccc2)cc1 ZINC000217935481 DG In-Stock Unstable ADRB3 31 53 COc1ccc(OC[C@H](C)NC(=S)Nc2ccccc2)cc1 ZINC000217935481 DG In-Stock Unstable SDH1 0 41 COc1ccc(OC[C@H](C)NC(=S)Nc2ccccc2)cc1 ZINC000217935481 DG In-Stock Unstable O69638_MYCTO 0 46 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc2cc[nH]c2c1 ZINC000217935503 GG For-Sale Unstable GHSR 16 51 CCOc1cc(/C=C2/CC(=O)NC2=O)ccc1OC ZINC000217935530 CD For-Sale Unstable ESRRA 50 41 CCOc1cc(/C=C2/CC(=O)NC2=O)ccc1OC ZINC000217935530 CD For-Sale Unstable HPGD 49 42 COCCN(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217935562 CD For-Sale Unstable FDPS 34 46 COCCN(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217935562 CD For-Sale Unstable PTGER2 24 40 COCCN(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217935562 CD For-Sale Unstable LTB4R 19 46 COc1cccc(/C=C/NC(=O)Nc2ccc(I)cc2C)c1 ZINC000217935574 HI For-Sale Unstable BRPF1 0 40 Cn1cccc1[C@H](O)CCNC(=O)c1cc(-c2ccccc2)on1 ZINC000217935592 EF In-Stock Unstable HDAC10 20 54 CC(C)Oc1cccc(CCCNC(=S)Nc2ccccc2)c1 ZINC000217935598 EI In-Stock Unstable HRH2 31 43 CC(C)Oc1cccc(CCCNC(=S)Nc2ccccc2)c1 ZINC000217935598 EI In-Stock Unstable FDFT1 0 46 CC(C)Oc1cccc(CCCNC(=S)Nc2ccccc2)c1 ZINC000217935598 EI In-Stock Unstable CCKAR 0 40 CC(C)Oc1cccc(CCCNC(=S)Nc2ccccc2)c1 ZINC000217935598 EI In-Stock Unstable MTNR1B 30 40 CC(C)Oc1cccc(CCCNC(=S)Nc2ccccc2)c1 ZINC000217935598 EI In-Stock Unstable AMP1_PLAFQ 40 48 CC(C)Oc1cccc(CCCNC(=S)Nc2ccccc2)c1 ZINC000217935598 EI In-Stock Unstable CRTM 70 48 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCCc1ccccc1 ZINC000217935604 GG For-Sale Unstable FKBP1A 41 36 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCCc1ccccc1 ZINC000217935604 GG For-Sale Unstable PREP 54 41 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCCc1ccccc1 ZINC000217935604 GG For-Sale Unstable FAAH 41 38 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCCc1ccccc1 ZINC000217935604 GG For-Sale Unstable CES1 48 36 Cn1cccc1[C@@H](O)CCNC(=O)c1cc(-c2ccccc2)on1 ZINC000217935672 EF In-Stock Unstable HDAC10 20 54 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCCc1ccccc1 ZINC000217935674 GG For-Sale Unstable FKBP1A 41 36 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCCc1ccccc1 ZINC000217935674 GG For-Sale Unstable PREP 54 41 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCCc1ccccc1 ZINC000217935674 GG For-Sale Unstable FAAH 41 38 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCCc1ccccc1 ZINC000217935674 GG For-Sale Unstable CES1 48 36 COCCN(C)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217935677 CD On-Demand Unstable FDPS 30 46 COCCN(C)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217935677 CD On-Demand Unstable LTA4H 19 40 COCCN(C)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217935677 CD On-Demand Unstable AHR 15 40 COc1cccc(/C=C/NC(=O)Nc2cccc(Cl)c2)c1 ZINC000217935694 DI For-Sale Unstable MTNR1A 27 46 COc1cccc(/C=C/NC(=O)Nc2cccc(Cl)c2)c1 ZINC000217935694 DI For-Sale Unstable MTNR1B 32 46 COc1cccc(/C=C/NC(=O)Nc2cccc(Cl)c2)c1 ZINC000217935694 DI For-Sale Unstable TAAR1 33 45 COc1cccc(/C=C/NC(=O)Nc2cccc(Cl)c2)c1 ZINC000217935694 DI For-Sale Unstable AKR1C2 27 48 COc1cccc(/C=C/NC(=O)Nc2cccc(Cl)c2)c1 ZINC000217935694 DI For-Sale Unstable IMDH_CRYPV 17 40 COc1cccc(/C=C/NC(=O)Nc2cccc(Cl)c2)c1 ZINC000217935694 DI For-Sale Unstable PSBA 0 44 COc1cccc(/C=C/NC(=O)Nc2cccc(Cl)c2)c1 ZINC000217935694 DI For-Sale Unstable KCNK3 36 42 C[S+](C)CC(=O)Nc1ccccc1 ZINC000217935698 AD Annotated Unstable LTA4H 34 41 C[S+](C)CC(=O)Nc1ccccc1 ZINC000217935698 AD Annotated Unstable HDAC8 27 49 C[S+](C)CC(=O)Nc1ccccc1 ZINC000217935698 AD Annotated Unstable HDAC10 42 49 C[S+](C)CC(=O)Nc1ccccc1 ZINC000217935698 AD Annotated Unstable CA5B 16 40 C[S+](C)CC(=O)Nc1ccccc1 ZINC000217935698 AD Annotated Unstable CA5A 18 40 C[S+](C)CC(=O)Nc1ccccc1 ZINC000217935698 AD Annotated Unstable MMP3 19 40 C[S+](C)CC(=O)Nc1ccccc1 ZINC000217935698 AD Annotated Unstable HDAC1 21 49 C[S+](C)CC(=O)Nc1ccccc1 ZINC000217935698 AD Annotated Unstable HDAC2 30 49 C[S+](C)CC(=O)Nc1ccccc1 ZINC000217935698 AD Annotated Unstable HDAC3 32 49 C[S+](C)CC(=O)Nc1ccccc1 ZINC000217935698 AD Annotated Unstable HDAC6 32 40 C[S+](C)CC(=O)Nc1ccccc1 ZINC000217935698 AD Annotated Unstable FUCA1 19 43 C[S+](C)CC(=O)Nc1ccccc1 ZINC000217935698 AD Annotated Unstable SLC1A1 17 40 C[S+](C)CC(=O)Nc1ccccc1 ZINC000217935698 AD Annotated Unstable HDAC11 47 49 C[S+](C)CC(=O)Nc1ccccc1 ZINC000217935698 AD Annotated Unstable SLC1A2 26 40 C[S+](C)CC(=O)Nc1ccccc1 ZINC000217935698 AD Annotated Unstable KCNK3 43 34 CC(C)Oc1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217935705 EI In-Stock Unstable ADRB1 23 46 CC(C)Oc1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217935705 EI In-Stock Unstable ADRB3 24 46 CC(C)Oc1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217935705 EI In-Stock Unstable SCN2A 24 40 COC(=O)C[C@@H](c1c(O)c2ccccc2oc1=O)C(C)C ZINC000217935720 CF In-Stock Unstable NQO1 42 45 O=S(=O)(Nc1nc2c(s1)CCCCC2)c1ccccc1Br ZINC000217935746 GH On-Demand Unstable SLC27A1 26 41 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCCc1ccccc1 ZINC000217935748 GG For-Sale Unstable FKBP1A 41 36 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCCc1ccccc1 ZINC000217935748 GG For-Sale Unstable PREP 54 41 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCCc1ccccc1 ZINC000217935748 GG For-Sale Unstable FAAH 41 38 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCCc1ccccc1 ZINC000217935748 GG For-Sale Unstable CES1 48 36 Cn1cccc1[C@H](O)CCNC(=O)c1cccc(C(F)(F)F)c1 ZINC000217935784 EF In-Stock Unstable DRD4 41 31 Cn1cccc1[C@H](O)CCNC(=O)c1cccc(C(F)(F)F)c1 ZINC000217935784 EF In-Stock Unstable CCR2 81 43 Cn1cccc1[C@H](O)CCNC(=O)c1cccc(C(F)(F)F)c1 ZINC000217935784 EF In-Stock Unstable GPR52 0 41 COC(=O)C[C@H](c1c(O)c2ccccc2oc1=O)C(C)C ZINC000217935795 CF In-Stock Unstable NQO1 42 45 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cc2)c1 ZINC000217935802 DI For-Sale Unstable UL80 19 41 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cc2)c1 ZINC000217935802 DI For-Sale Unstable AHR 15 50 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cc2)c1 ZINC000217935802 DI For-Sale Unstable GUAB 0 41 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cc2)c1 ZINC000217935802 DI For-Sale Unstable MTNR1A 29 50 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cc2)c1 ZINC000217935802 DI For-Sale Unstable MTNR1B 34 50 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cc2)c1 ZINC000217935802 DI For-Sale Unstable Q8MMZ8_EIMTE 0 44 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cc2)c1 ZINC000217935802 DI For-Sale Unstable TAAR1 24 43 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cc2)c1 ZINC000217935802 DI For-Sale Unstable AKR1C3 19 41 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cc2)c1 ZINC000217935802 DI For-Sale Unstable AKR1C2 42 41 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cc2)c1 ZINC000217935802 DI For-Sale Unstable IMDH_CRYPV 21 40 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cc2)c1 ZINC000217935802 DI For-Sale Unstable P95276_MYCTO 0 40 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cc2)c1 ZINC000217935802 DI For-Sale Unstable SENP1 0 45 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCCc1ccccc1 ZINC000217935828 GG For-Sale Unstable FKBP1A 41 36 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCCc1ccccc1 ZINC000217935828 GG For-Sale Unstable PREP 54 41 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCCc1ccccc1 ZINC000217935828 GG For-Sale Unstable FAAH 41 38 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCCc1ccccc1 ZINC000217935828 GG For-Sale Unstable CES1 48 36 Cn1cccc1[C@@H](O)CCNC(=O)c1cccc(C(F)(F)F)c1 ZINC000217935848 EF In-Stock Unstable DRD4 41 31 Cn1cccc1[C@@H](O)CCNC(=O)c1cccc(C(F)(F)F)c1 ZINC000217935848 EF In-Stock Unstable CCR2 81 43 Cn1cccc1[C@@H](O)CCNC(=O)c1cccc(C(F)(F)F)c1 ZINC000217935848 EF In-Stock Unstable GPR52 0 41 C=CCN(CC=C)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217935913 CG For-Sale Unstable MTNR1A 41 44 C=CCN(CC=C)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217935913 CG For-Sale Unstable MTNR1B 42 44 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccc(OC)cc1 ZINC000217935919 HE For-Sale Unstable COLA 80 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccc(OC)cc1 ZINC000217935919 HE For-Sale Unstable CPT1A 69 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccc(OC)cc1 ZINC000217935919 HE For-Sale Unstable CPT2 36 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccc(OC)cc1 ZINC000217935919 HE For-Sale Unstable MMP3 20 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccc(OC)cc1 ZINC000217935919 HE For-Sale Unstable MMP1 17 40 C/C(=C1/CC(=O)NC1=O)c1cccnc1 ZINC000217935938 BC For-Sale Unstable TBXAS1 23 40 CCCCCc1ccc(N[C@@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217935950 CJ For-Sale Unstable SPHK1 15 40 Cn1cccc1[C@H](O)CCNC(=O)c1cc2ccccc2oc1=O ZINC000217935955 ED In-Stock Unstable MAOB 16 49 Cn1cccc1[C@H](O)CCNC(=O)c1cc2ccccc2oc1=O ZINC000217935955 ED In-Stock Unstable POLR1A 53 32 COc1cc(CN[C@@]23C[C@@H]4C[C@@H](C[C@@](O)(C4)C2)C3)ccc1OCC(N)=O ZINC000217935968 FD In-Stock Unstable DRTS_TRYCR 43 30 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccc(OC)cc1 ZINC000217936001 HE For-Sale Unstable COLA 80 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccc(OC)cc1 ZINC000217936001 HE For-Sale Unstable CPT1A 69 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccc(OC)cc1 ZINC000217936001 HE For-Sale Unstable CPT2 36 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccc(OC)cc1 ZINC000217936001 HE For-Sale Unstable MMP3 20 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccc(OC)cc1 ZINC000217936001 HE For-Sale Unstable MMP1 17 40 CCOc1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217936004 DI In-Stock Unstable ADRB1 28 49 CCOc1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217936004 DI In-Stock Unstable ADRB3 35 49 CCOc1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217936004 DI In-Stock Unstable CA1 21 40 CCOc1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217936004 DI In-Stock Unstable SCN2A 37 49 CCOc1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217936004 DI In-Stock Unstable FAAH 18 40 CCOc1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217936004 DI In-Stock Unstable S1PR5 17 41 CCOc1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217936004 DI In-Stock Unstable TAAR1 18 41 CCOc1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217936004 DI In-Stock Unstable QPCT 32 47 CCOc1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217936004 DI In-Stock Unstable PPO2 36 42 CCOc1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217936004 DI In-Stock Unstable NCE103 17 40 NC(=O)[C@H]1CCCN(Cc2ccccc2/C=C\C(=O)O)C1 ZINC000217936007 CD For-Sale Unstable SLC6A1 174 49 NC(=O)[C@H]1CCCN(Cc2ccccc2/C=C\C(=O)O)C1 ZINC000217936007 CD For-Sale Unstable PTGER2 33 42 NC(=O)[C@H]1CCCN(Cc2ccccc2/C=C\C(=O)O)C1 ZINC000217936007 CD For-Sale Unstable PTGER4 0 42 NC(=O)[C@H]1CCCN(Cc2ccccc2/C=C\C(=O)O)C1 ZINC000217936007 CD For-Sale Unstable PTGER3 16 42 COc1ccc(Br)cc1S(=O)(=O)Nc1nc2c(s1)CCCCC2 ZINC000217936011 HH On-Demand Unstable ALPL 15 47 COc1cccc(/C=C/NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000217936025 FG For-Sale Unstable HTR1A 24 44 COc1cccc(/C=C/NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000217936025 FG For-Sale Unstable DRD2 34 41 COc1cccc(/C=C/NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000217936025 FG For-Sale Unstable DRD4 61 45 COc1cccc(/C=C/NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000217936025 FG For-Sale Unstable ACHE 32 47 COc1cccc(/C=C/NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000217936025 FG For-Sale Unstable HRH2 30 41 COc1cccc(/C=C/NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000217936025 FG For-Sale Unstable DRD3 30 40 COc1cccc(/C=C/NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000217936025 FG For-Sale Unstable SIGMAR1 60 59 COc1cccc(/C=C/NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000217936025 FG For-Sale Unstable MMP13 18 42 COc1cccc(/C=C/NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000217936025 FG For-Sale Unstable CCR3 26 41 COc1cccc(/C=C/NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000217936025 FG For-Sale Unstable NPFFR2 27 44 COc1cccc(/C=C/NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000217936025 FG For-Sale Unstable MLNR 21 40 COc1cccc(/C=C/NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000217936025 FG For-Sale Unstable MTNR1B 50 39 COc1cccc(/C=C/NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000217936025 FG For-Sale Unstable FAAH 39 57 COc1cccc(/C=C/NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000217936025 FG For-Sale Unstable MMP9 15 42 COc1cccc(/C=C/NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000217936025 FG For-Sale Unstable MCHR1 32 44 COc1cccc(/C=C/NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000217936025 FG For-Sale Unstable CACNA1G 25 41 COc1cccc(/C=C/NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000217936025 FG For-Sale Unstable MGLL 0 43 COc1cccc(/C=C/NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000217936025 FG For-Sale Unstable CCR8 29 43 COc1cccc(/C=C/NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000217936025 FG For-Sale Unstable ABHD6 0 43 COc1cccc(/C=C/NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000217936025 FG For-Sale Unstable NPFFR1 40 44 COc1cccc(/C=C/NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000217936025 FG For-Sale Unstable GPR183 0 42 Cn1cccc1[C@@H](O)CCNC(=O)c1cc2ccccc2oc1=O ZINC000217936037 ED In-Stock Unstable MAOB 16 49 Cn1cccc1[C@@H](O)CCNC(=O)c1cc2ccccc2oc1=O ZINC000217936037 ED In-Stock Unstable POLR1A 53 32 CCCCCc1ccc(N[C@H]2C[C@@H]3CC=C[C@H]32)cc1 ZINC000217936039 CJ For-Sale Unstable SPHK1 15 40 O=C(NCC1(O)CCC1)Nc1cc(Cl)cc(Cl)c1 ZINC000217936071 CG On-Demand Unstable ACAT 0 43 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccc(OC)cc1 ZINC000217936095 HE For-Sale Unstable COLA 80 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccc(OC)cc1 ZINC000217936095 HE For-Sale Unstable CPT1A 69 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccc(OC)cc1 ZINC000217936095 HE For-Sale Unstable CPT2 36 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccc(OC)cc1 ZINC000217936095 HE For-Sale Unstable MMP3 20 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccc(OC)cc1 ZINC000217936095 HE For-Sale Unstable MMP1 17 40 CCCOc1ccccc1CCCNC(=S)Nc1ccccc1 ZINC000217936098 EI In-Stock Unstable MTNR1B 36 41 CCCOc1ccccc1CCCNC(=S)Nc1ccccc1 ZINC000217936098 EI In-Stock Unstable QPCT 23 40 CCCCCc1ccc(N[C@@H]2C[C@H]3CC=C[C@H]32)cc1 ZINC000217936117 CJ For-Sale Unstable SPHK1 15 40 NC(=O)[C@H]1CCCN(Cc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217936122 CD For-Sale Unstable SLC6A1 140 40 NC(=O)[C@H]1CCCN(Cc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217936122 CD For-Sale Unstable SIGMAR1 19 45 COc1cccc(/C=C/NC(=O)N2CCN(C)CC2)c1 ZINC000217936128 CD For-Sale Unstable DRD4 44 33 COc1cccc(/C=C/NC(=O)N2CCN(C)CC2)c1 ZINC000217936128 CD For-Sale Unstable MTNR1A 36 41 COc1cccc(/C=C/NC(=O)N2CCN(C)CC2)c1 ZINC000217936128 CD For-Sale Unstable MTNR1B 45 41 CSCC[C@H](Nc1nc(C)cc(C)n1)C(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217936172 IE In-Stock Unstable CHRNA4 26 42 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccc(OC)cc1 ZINC000217936181 HE For-Sale Unstable COLA 80 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccc(OC)cc1 ZINC000217936181 HE For-Sale Unstable CPT1A 69 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccc(OC)cc1 ZINC000217936181 HE For-Sale Unstable CPT2 36 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccc(OC)cc1 ZINC000217936181 HE For-Sale Unstable MMP3 20 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccc(OC)cc1 ZINC000217936181 HE For-Sale Unstable MMP1 17 40 CCCCCc1ccc(N[C@H]2C[C@H]3CC=C[C@@H]23)cc1 ZINC000217936205 CJ For-Sale Unstable SPHK1 15 40 Cc1ccc(OC[C@@H](C)NC(=S)Nc2ccccc2)cc1 ZINC000217936223 DH In-Stock Unstable ADRB2 19 42 Cc1ccc(OC[C@@H](C)NC(=S)Nc2ccccc2)cc1 ZINC000217936223 DH In-Stock Unstable ADRB1 27 51 Cc1ccc(OC[C@@H](C)NC(=S)Nc2ccccc2)cc1 ZINC000217936223 DH In-Stock Unstable ADRB3 24 51 Cc1ccc(OC[C@@H](C)NC(=S)Nc2ccccc2)cc1 ZINC000217936223 DH In-Stock Unstable SDH1 0 41 Cc1ccc(OC[C@@H](C)NC(=S)Nc2ccccc2)cc1 ZINC000217936223 DH In-Stock Unstable O69638_MYCTO 0 46 NC(=O)[C@H]1CCCN(Cc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217936225 CD For-Sale Unstable SLC6A1 150 40 NC(=O)[C@H]1CCCN(Cc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217936225 CD For-Sale Unstable SIGMAR1 26 45 COc1cccc(/C=C/NC(=O)N2CCCCC2)c1 ZINC000217936230 CF For-Sale Unstable DRD4 43 33 COc1cccc(/C=C/NC(=O)N2CCCCC2)c1 ZINC000217936230 CF For-Sale Unstable MTNR1A 35 42 COc1cccc(/C=C/NC(=O)N2CCCCC2)c1 ZINC000217936230 CF For-Sale Unstable MTNR1B 44 42 CSCC[C@@H](Nc1nc(C)cc(C)n1)C(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217936241 IE In-Stock Unstable CHRNA4 26 42 COc1cccc(/C=C/NC(=O)NC2CCCCCCCCCCC2)c1 ZINC000217936307 FK For-Sale Unstable MTNR1A 37 40 COc1cccc(/C=C/NC(=O)NC2CCCCCCCCCCC2)c1 ZINC000217936307 FK For-Sale Unstable MTNR1B 40 40 COc1cccc(/C=C/NC(=O)NC2CCCCCCCCCCC2)c1 ZINC000217936307 FK For-Sale Unstable NR1H4 22 40 COc1cccc(/C=C/NC(=O)NC2CCCCCCCCCCC2)c1 ZINC000217936307 FK For-Sale Unstable FAAH 26 46 COc1cccc(/C=C/NC(=O)NC2CCCCCCCCCCC2)c1 ZINC000217936307 FK For-Sale Unstable EPHX2 28 50 Cc1ccc(OC[C@H](C)NC(=S)Nc2ccccc2)cc1 ZINC000217936311 DH In-Stock Unstable ADRB2 19 42 Cc1ccc(OC[C@H](C)NC(=S)Nc2ccccc2)cc1 ZINC000217936311 DH In-Stock Unstable ADRB1 27 51 Cc1ccc(OC[C@H](C)NC(=S)Nc2ccccc2)cc1 ZINC000217936311 DH In-Stock Unstable ADRB3 24 51 Cc1ccc(OC[C@H](C)NC(=S)Nc2ccccc2)cc1 ZINC000217936311 DH In-Stock Unstable SDH1 0 41 Cc1ccc(OC[C@H](C)NC(=S)Nc2ccccc2)cc1 ZINC000217936311 DH In-Stock Unstable O69638_MYCTO 0 46 Cn1cccc1[C@H](O)CCNC(=O)/C=C/c1ccc2c(c1)OCO2 ZINC000217936328 EE In-Stock Unstable DYRK2 56 37 C/C(=C1/CC(=O)NC1=O)c1cccc(C(F)(F)F)c1 ZINC000217936337 CF For-Sale Unstable CCR2 51 35 COc1cc2c(cc1OC)CN(C(=O)c1cnc3ccc(Cl)cc3c1O)CC2 ZINC000217936338 GH In-Stock Unstable ABCB1B 59 35 COc1cc2c(cc1OC)CN(C(=O)c1cnc3ccc(Cl)cc3c1O)CC2 ZINC000217936338 GH In-Stock Unstable ABCB1 17 43 Cn1cccc1[C@@H](O)CCNC(=O)/C=C/c1ccc2c(c1)OCO2 ZINC000217936408 EE In-Stock Unstable DYRK2 56 37 COc1cccc(/C=C/NC(=O)NCCN2CCOCC2)c1 ZINC000217936409 DD For-Sale Unstable HTR1A 19 48 COc1cccc(/C=C/NC(=O)NCCN2CCOCC2)c1 ZINC000217936409 DD For-Sale Unstable DRD2 18 43 COc1cccc(/C=C/NC(=O)NCCN2CCOCC2)c1 ZINC000217936409 DD For-Sale Unstable CNR1 0 43 COc1cccc(/C=C/NC(=O)NCCN2CCOCC2)c1 ZINC000217936409 DD For-Sale Unstable DRD4 59 46 COc1cccc(/C=C/NC(=O)NCCN2CCOCC2)c1 ZINC000217936409 DD For-Sale Unstable DRD3 32 48 COc1cccc(/C=C/NC(=O)NCCN2CCOCC2)c1 ZINC000217936409 DD For-Sale Unstable CNR2 15 43 COc1cccc(/C=C/NC(=O)NCCN2CCOCC2)c1 ZINC000217936409 DD For-Sale Unstable CASR 43 46 COc1cccc(/C=C/NC(=O)NCCN2CCOCC2)c1 ZINC000217936409 DD For-Sale Unstable SIGMAR1 15 40 COc1cccc(/C=C/NC(=O)NCCN2CCOCC2)c1 ZINC000217936409 DD For-Sale Unstable MTNR1A 64 39 COc1cccc(/C=C/NC(=O)NCCN2CCOCC2)c1 ZINC000217936409 DD For-Sale Unstable MTNR1B 61 39 COc1cccc(/C=C/NC(=O)NCCN2CCOCC2)c1 ZINC000217936409 DD For-Sale Unstable EPHX2 24 42 COc1cccc(/C=C/NC(=O)NCCN2CCOCC2)c1 ZINC000217936409 DD For-Sale Unstable ACKR3 39 42 C[C@@H]1CN(Cc2ccc(F)c(/C=C\C(=O)O)c2)CCO1 ZINC000217936462 CE For-Sale Unstable DRD4 16 40 C[C@@H]1CN(Cc2ccc(F)c(/C=C\C(=O)O)c2)CCO1 ZINC000217936462 CE For-Sale Unstable CCR1 24 41 C[C@@H]1CN(Cc2ccc(F)c(/C=C\C(=O)O)c2)CCO1 ZINC000217936462 CE For-Sale Unstable MLNR 44 33 O=S(=O)(Nc1nc2c(s1)CCCCC2)c1cc(F)ccc1F ZINC000217936473 EG On-Demand Unstable SLC27A1 39 43 CS(=O)(=O)[C@@H]1CCC(CN)(CN)C1 ZINC000217936481 BB In-Stock Unstable CACNA2D1 43 41 Cc1nonc1CC(=O)N1CCCN(Cc2cccnc2)CC1 ZINC000217936487 DD In-Stock Unstable C3AR1 41 37 COc1ccc(CC(=O)NCC[C@@H](O)c2cccn2C)cc1OC ZINC000217936504 ED In-Stock Unstable TRPV1 0 42 COc1ccc(CC(=O)NCC[C@@H](O)c2cccn2C)cc1OC ZINC000217936504 ED In-Stock Unstable NCE103 22 47 COc1ccc(CC(=O)NCC[C@@H](O)c2cccn2C)cc1OC ZINC000217936504 ED In-Stock Unstable CAN2 0 47 COc1cccc(/C=C/NC(=O)NCc2ccco2)c1 ZINC000217936505 CF For-Sale Unstable MTNR1A 47 41 COc1cccc(/C=C/NC(=O)NCc2ccco2)c1 ZINC000217936505 CF For-Sale Unstable MTNR1B 44 41 C[C@H]1CN(Cc2ccc(F)c(/C=C\C(=O)O)c2)CCO1 ZINC000217936551 CE For-Sale Unstable DRD4 16 40 C[C@H]1CN(Cc2ccc(F)c(/C=C\C(=O)O)c2)CCO1 ZINC000217936551 CE For-Sale Unstable CCR1 24 41 C[C@H]1CN(Cc2ccc(F)c(/C=C\C(=O)O)c2)CCO1 ZINC000217936551 CE For-Sale Unstable MLNR 44 33 CS(=O)(=O)[C@H]1CCC(CN)(CN)C1 ZINC000217936562 BB In-Stock Unstable CACNA2D1 43 41 COc1ccc(CC(=O)NCC[C@H](O)c2cccn2C)cc1OC ZINC000217936585 ED In-Stock Unstable TRPV1 0 42 COc1ccc(CC(=O)NCC[C@H](O)c2cccn2C)cc1OC ZINC000217936585 ED In-Stock Unstable NCE103 22 47 COc1ccc(CC(=O)NCC[C@H](O)c2cccn2C)cc1OC ZINC000217936585 ED In-Stock Unstable CAN2 0 47 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=S)Nc3ccccc3)cc2)C1 ZINC000217936596 FJ In-Stock Unstable HRH3 22 40 COc1cccc(/C=C/NC(=O)N2CCN(CCN)CC2)c1 ZINC000217936614 DC For-Sale Unstable DRD4 52 40 COc1cccc(/C=C/NC(=O)N2CCN(CCN)CC2)c1 ZINC000217936614 DC For-Sale Unstable DRD3 21 40 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](C)C(=O)Nc3nc4c(s3)CCC4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217936623 KI In-Stock Unstable TUBA1A 17 62 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](C)C(=O)Nc3nc4c(s3)CCC4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217936623 KI In-Stock Unstable TPPP 0 58 Cc1ccc(=O)cc(C)c1 ZINC000217936649 AD For-Sale Unstable CYP2A5 0 43 CCCCN(CC)Cc1ccc(F)c(/C=C\C(=O)O)c1 ZINC000217936658 CH For-Sale Unstable PLM2_PLAFA 40 33 C=CCC[C@@H](CCC(=O)OC)NC(=O)OC(C)(C)C ZINC000217936663 CF For-Sale Unstable CTSK 18 43 CS(=O)(=O)[C@@H]1CC[C@@](CN)(CO)C1 ZINC000217936664 BB In-Stock Unstable CACNA2D1 47 44 O=C1C/C(=C\c2ccc(-c3ccccc3)cc2)C(=O)N1 ZINC000217936671 CF For-Sale Unstable PRKCA 15 41 O=C1C/C(=C\c2ccc(-c3ccccc3)cc2)C(=O)N1 ZINC000217936671 CF For-Sale Unstable PIM2 0 49 O=C1C/C(=C\c2ccc(-c3ccccc3)cc2)C(=O)N1 ZINC000217936671 CF For-Sale Unstable HPGD 31 46 C[C@H](NC(=S)Nc1ccccc1)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217936696 FJ In-Stock Unstable HRH3 0 40 COc1cccc(/C=C/NC(=O)NCCN2CCNCC2)c1 ZINC000217936715 DC For-Sale Unstable HTR1A 18 45 COc1cccc(/C=C/NC(=O)NCCN2CCNCC2)c1 ZINC000217936715 DC For-Sale Unstable DRD2 16 43 COc1cccc(/C=C/NC(=O)NCCN2CCNCC2)c1 ZINC000217936715 DC For-Sale Unstable DRD4 58 44 COc1cccc(/C=C/NC(=O)NCCN2CCNCC2)c1 ZINC000217936715 DC For-Sale Unstable DRD3 31 45 COc1cccc(/C=C/NC(=O)NCCN2CCNCC2)c1 ZINC000217936715 DC For-Sale Unstable CCR3 16 42 COc1cccc(/C=C/NC(=O)NCCN2CCNCC2)c1 ZINC000217936715 DC For-Sale Unstable MTNR1A 54 39 COc1cccc(/C=C/NC(=O)NCCN2CCNCC2)c1 ZINC000217936715 DC For-Sale Unstable MTNR1B 53 39 Cn1nc(-c2ccc(Cl)cc2Cl)cc1C(=O)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217936730 HI In-Stock Unstable CNR1 54 32 Cn1nc(-c2ccc(Cl)cc2Cl)cc1C(=O)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217936730 HI In-Stock Unstable IL2RA 51 36 Cn1nc(-c2ccc(Cl)cc2Cl)cc1C(=O)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217936730 HI In-Stock Unstable CNR2 17 40 Cn1nc(-c2ccc(Cl)cc2Cl)cc1C(=O)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217936730 HI In-Stock Unstable ALPL 46 36 CS(=O)(=O)[C@H]1CC[C@@](CN)(CO)C1 ZINC000217936750 BB In-Stock Unstable CACNA2D1 47 44 NC(=O)C1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217936761 CD For-Sale Unstable PTGER2 39 45 NC(=O)C1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217936761 CD For-Sale Unstable PTGER4 0 45 NC(=O)C1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217936761 CD For-Sale Unstable SIGMAR1 28 43 NC(=O)C1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217936761 CD For-Sale Unstable PTGER3 18 45 C[C@@H](CCO)SCc1cccc(/C=C\C(=O)O)c1 ZINC000217936782 CF For-Sale Unstable AKR1C3 40 42 COc1cccc(/C=C/NC(=O)NCc2ccc(C)cc2)c1 ZINC000217936815 CG For-Sale Unstable MTNR1A 54 43 COc1cccc(/C=C/NC(=O)NCc2ccc(C)cc2)c1 ZINC000217936815 CG For-Sale Unstable MTNR1B 55 43 COc1cccc(/C=C/NC(=O)NCc2ccc(C)cc2)c1 ZINC000217936815 CG For-Sale Unstable PDS 40 39 CS(=O)(=O)[C@@H]1CC[C@](CN)(CO)C1 ZINC000217936824 BB In-Stock Unstable CACNA2D1 47 44 COC(=O)C[C@H](c1ccc(C(=O)O)cc1)c1c(O)c2ccccc2oc1=O ZINC000217936832 FF In-Stock Unstable NQO1 67 54 COc1cc(/C=C2/CC(=O)NC2=O)cc(OC)c1 ZINC000217936833 BD For-Sale Unstable CYP1A1 22 41 C[C@H](CCO)SCc1cccc(/C=C\C(=O)O)c1 ZINC000217936857 CF For-Sale Unstable AKR1C3 40 42 NC(=O)C1CCN(Cc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217936867 CD For-Sale Unstable DRD4 31 43 NC(=O)C1CCN(Cc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217936867 CD For-Sale Unstable LTA4H 17 45 NC(=O)C1CCN(Cc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217936867 CD For-Sale Unstable HRH3 15 50 NC(=O)C1CCN(Cc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217936867 CD For-Sale Unstable SIGMAR1 40 50 CS(=O)(=O)[C@H]1CC[C@](CN)(CO)C1 ZINC000217936899 BB In-Stock Unstable CACNA2D1 47 44 COc1cccc(/C=C/NC(=O)NCc2ccncc2)c1 ZINC000217936913 CF For-Sale Unstable TRPV1 0 47 COc1cccc(/C=C/NC(=O)NCc2ccncc2)c1 ZINC000217936913 CF For-Sale Unstable ROCK1 29 48 COc1cccc(/C=C/NC(=O)NCc2ccncc2)c1 ZINC000217936913 CF For-Sale Unstable MTNR1A 52 43 COc1cccc(/C=C/NC(=O)NCc2ccncc2)c1 ZINC000217936913 CF For-Sale Unstable MTNR1B 53 43 COc1cccc(/C=C/NC(=O)NCc2ccncc2)c1 ZINC000217936913 CF For-Sale Unstable ROCK2 35 54 COc1cccc(/C=C/NC(=O)NCc2ccncc2)c1 ZINC000217936913 CF For-Sale Unstable NAMPT 22 42 COC(=O)C[C@@H](c1ccc(C(=O)O)cc1)c1c(O)c2ccccc2oc1=O ZINC000217936916 FF In-Stock Unstable NQO1 67 54 O=C1C/C(=C/c2ccc(-c3cccc(Cl)c3)s2)C(=O)N1 ZINC000217936920 DG For-Sale Unstable PRF1 46 41 Cc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=S)Nc1ccccc1 ZINC000217936974 EJ In-Stock Unstable TRPV1 0 40 CCC[C@@H](C)N(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217936979 CG For-Sale Unstable AKR1C3 37 40 CS(=O)(=O)[C@@H]1CC[C@](CN)(C(=O)O)C1 ZINC000217936996 BB In-Stock Unstable CACNA2D1 48 36 COc1cccc(/C=C/NC(=O)NCc2ccccn2)c1 ZINC000217937011 CF For-Sale Unstable MTNR1A 43 41 COc1cccc(/C=C/NC(=O)NCc2ccccn2)c1 ZINC000217937011 CF For-Sale Unstable MTNR1B 44 43 COc1cccc(/C=C/NC(=O)NCc2ccccn2)c1 ZINC000217937011 CF For-Sale Unstable ROCK2 18 40 Cc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=S)Nc1ccccc1 ZINC000217937053 EJ In-Stock Unstable TRPV1 0 40 CCC[C@H](C)N(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217937059 CG For-Sale Unstable AKR1C3 37 40 CO[C@@H]1CCCC[C@@H]1N[C@@H](C)c1cccc2ccccc12 ZINC000217937067 CI For-Sale Unstable CASR 0 60 CS(=O)(=O)[C@H]1CC[C@](CN)(C(=O)O)C1 ZINC000217937070 BB In-Stock Unstable CACNA2D1 48 36 CCN(CCCN(C)C)c1ccc(F)cc1CBr ZINC000217937133 DG For-Sale Unstable MPO 15 41 COc1cccc(/C=C/NC(=O)NCCCN2CCOCC2)c1 ZINC000217937134 DD For-Sale Unstable HTR1A 30 45 COc1cccc(/C=C/NC(=O)NCCCN2CCOCC2)c1 ZINC000217937134 DD For-Sale Unstable DRD2 31 46 COc1cccc(/C=C/NC(=O)NCCCN2CCOCC2)c1 ZINC000217937134 DD For-Sale Unstable DRD4 52 41 COc1cccc(/C=C/NC(=O)NCCCN2CCOCC2)c1 ZINC000217937134 DD For-Sale Unstable HRH2 26 42 COc1cccc(/C=C/NC(=O)NCCCN2CCOCC2)c1 ZINC000217937134 DD For-Sale Unstable HTR2A 26 48 COc1cccc(/C=C/NC(=O)NCCCN2CCOCC2)c1 ZINC000217937134 DD For-Sale Unstable HTR2C 25 42 COc1cccc(/C=C/NC(=O)NCCCN2CCOCC2)c1 ZINC000217937134 DD For-Sale Unstable DRD3 60 46 COc1cccc(/C=C/NC(=O)NCCCN2CCOCC2)c1 ZINC000217937134 DD For-Sale Unstable AVPR1B 28 41 COc1cccc(/C=C/NC(=O)NCCCN2CCOCC2)c1 ZINC000217937134 DD For-Sale Unstable CASR 39 44 COc1cccc(/C=C/NC(=O)NCCCN2CCOCC2)c1 ZINC000217937134 DD For-Sale Unstable HTR7 25 40 COc1cccc(/C=C/NC(=O)NCCCN2CCOCC2)c1 ZINC000217937134 DD For-Sale Unstable TACR2 30 45 COc1cccc(/C=C/NC(=O)NCCCN2CCOCC2)c1 ZINC000217937134 DD For-Sale Unstable FGFR1 15 41 COc1cccc(/C=C/NC(=O)NCCCN2CCOCC2)c1 ZINC000217937134 DD For-Sale Unstable SIGMAR1 16 42 COc1cccc(/C=C/NC(=O)NCCCN2CCOCC2)c1 ZINC000217937134 DD For-Sale Unstable NPY1R 15 40 COc1cccc(/C=C/NC(=O)NCCCN2CCOCC2)c1 ZINC000217937134 DD For-Sale Unstable CCR3 37 46 COc1cccc(/C=C/NC(=O)NCCCN2CCOCC2)c1 ZINC000217937134 DD For-Sale Unstable CHRNA7 0 43 COc1cccc(/C=C/NC(=O)NCCCN2CCOCC2)c1 ZINC000217937134 DD For-Sale Unstable MTNR1A 60 42 COc1cccc(/C=C/NC(=O)NCCCN2CCOCC2)c1 ZINC000217937134 DD For-Sale Unstable MTNR1B 59 42 COc1cccc(/C=C/NC(=O)NCCCN2CCOCC2)c1 ZINC000217937134 DD For-Sale Unstable EPHX2 28 45 COc1cccc(/C=C/NC(=O)NCCCN2CCOCC2)c1 ZINC000217937134 DD For-Sale Unstable ACKR3 35 45 CO[C@@H]1CCCC[C@H]1N[C@@H](C)c1cccc2ccccc12 ZINC000217937147 CI For-Sale Unstable CASR 0 60 CS(=O)(=O)[C@@H]1CC[C@@](CN)(C(=O)O)C1 ZINC000217937155 BB In-Stock Unstable CACNA2D1 48 36 CCC[C@@H](C)N(C)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217937167 CG On-Demand Unstable PLA2G4B 60 32 CCC[C@@H](C)N(C)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217937167 CG On-Demand Unstable AKR1C3 16 40 CCC[C@@H](C)N(C)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217937167 CG On-Demand Unstable NORA 0 48 CS(=O)(=O)[C@H]1CC[C@@](CN)(C(=O)O)C1 ZINC000217937234 BB In-Stock Unstable CACNA2D1 48 36 C[C@H](NC(=O)[C@@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937240 CG On-Demand Unstable F2 41 36 C[C@H](NC(=O)[C@@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937240 CG On-Demand Unstable ACE 41 38 C[C@H](NC(=O)[C@@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937240 CG On-Demand Unstable FKBP1A 28 40 C[C@H](NC(=O)[C@@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937240 CG On-Demand Unstable ELANE 62 42 C[C@H](NC(=O)[C@@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937240 CG On-Demand Unstable TRY1_BOVIN 53 34 C[C@H](NC(=O)[C@@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937240 CG On-Demand Unstable XIAP 114 46 C[C@H](NC(=O)[C@@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937240 CG On-Demand Unstable BIRC3 71 48 C[C@H](NC(=O)[C@@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937240 CG On-Demand Unstable BIRC2 79 42 C[C@H](NC(=O)[C@@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937240 CG On-Demand Unstable BIRC8 68 48 C[C@H](NC(=O)[C@@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937240 CG On-Demand Unstable BRCA1 52 32 CCC[C@H](C)N(C)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217937246 CG On-Demand Unstable PLA2G4B 60 32 CCC[C@H](C)N(C)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217937246 CG On-Demand Unstable AKR1C3 16 40 CCC[C@H](C)N(C)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217937246 CG On-Demand Unstable NORA 0 48 CCN(C(=O)N/C=C/c1cccc(OC)c1)c1ccccc1 ZINC000217937258 CH For-Sale Unstable TSPO 43 35 CCN(C(=O)N/C=C/c1cccc(OC)c1)c1ccccc1 ZINC000217937258 CH For-Sale Unstable MTNR1A 46 45 CCN(C(=O)N/C=C/c1cccc(OC)c1)c1ccccc1 ZINC000217937258 CH For-Sale Unstable MTNR1B 47 45 CCN(C(=O)N/C=C/c1cccc(OC)c1)c1ccccc1 ZINC000217937258 CH For-Sale Unstable NR1H4 45 39 C[C@@H](NC(=O)[C@@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937311 CG On-Demand Unstable F2 41 36 C[C@@H](NC(=O)[C@@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937311 CG On-Demand Unstable ACE 41 38 C[C@@H](NC(=O)[C@@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937311 CG On-Demand Unstable FKBP1A 28 40 C[C@@H](NC(=O)[C@@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937311 CG On-Demand Unstable ELANE 62 42 C[C@@H](NC(=O)[C@@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937311 CG On-Demand Unstable TRY1_BOVIN 53 34 C[C@@H](NC(=O)[C@@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937311 CG On-Demand Unstable CTSK 20 40 C[C@@H](NC(=O)[C@@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937311 CG On-Demand Unstable XIAP 114 46 C[C@@H](NC(=O)[C@@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937311 CG On-Demand Unstable BIRC3 71 48 C[C@@H](NC(=O)[C@@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937311 CG On-Demand Unstable BIRC2 79 42 C[C@@H](NC(=O)[C@@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937311 CG On-Demand Unstable BIRC8 68 48 C[C@@H](NC(=O)[C@@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937311 CG On-Demand Unstable BRCA1 52 32 CCN(CCO)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217937366 CD For-Sale Unstable ACHE 0 43 CCN(CCO)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217937366 CD For-Sale Unstable TUBB1 42 38 CCN(CCO)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217937366 CD For-Sale Unstable AKR1C3 22 41 COc1cccc(/C=C/NC(=O)N(C)Cc2ccccc2)c1 ZINC000217937374 CH For-Sale Unstable TSPO 43 35 COc1cccc(/C=C/NC(=O)N(C)Cc2ccccc2)c1 ZINC000217937374 CH For-Sale Unstable G6PC 29 50 COc1cccc(/C=C/NC(=O)N(C)Cc2ccccc2)c1 ZINC000217937374 CH For-Sale Unstable ROCK1 24 42 COc1cccc(/C=C/NC(=O)N(C)Cc2ccccc2)c1 ZINC000217937374 CH For-Sale Unstable MTNR1A 48 43 COc1cccc(/C=C/NC(=O)N(C)Cc2ccccc2)c1 ZINC000217937374 CH For-Sale Unstable MTNR1B 51 43 COc1cccc(/C=C/NC(=O)N(C)Cc2ccccc2)c1 ZINC000217937374 CH For-Sale Unstable ROCK2 33 44 COc1cccc(/C=C/NC(=O)N(C)Cc2ccccc2)c1 ZINC000217937374 CH For-Sale Unstable NR1H4 44 41 COc1cccc(/C=C/NC(=O)N(C)Cc2ccccc2)c1 ZINC000217937374 CH For-Sale Unstable HSD17B2 24 48 COc1cccc(/C=C/NC(=O)N(C)Cc2ccccc2)c1 ZINC000217937374 CH For-Sale Unstable AKR1C3 18 40 COc1cccc(/C=C/NC(=O)N(C)Cc2ccccc2)c1 ZINC000217937374 CH For-Sale Unstable CRTM 40 37 COc1cccc(/C=C/NC(=O)N(C)Cc2ccccc2)c1 ZINC000217937374 CH For-Sale Unstable PTGES 19 46 COc1cccc(/C=C/NC(=O)N(C)Cc2ccccc2)c1 ZINC000217937374 CH For-Sale Unstable LIMK2 19 49 COc1ccc(CN2C(=O)N[C@@H](CC(=O)N[C@H](CO)Cc3ccccc3)C2=O)cc1 ZINC000217937393 HD In-Stock Unstable MMP1 18 43 C[C@H](NC(=O)[C@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937401 CG On-Demand Unstable F2 41 36 C[C@H](NC(=O)[C@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937401 CG On-Demand Unstable ACE 41 38 C[C@H](NC(=O)[C@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937401 CG On-Demand Unstable FKBP1A 28 40 C[C@H](NC(=O)[C@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937401 CG On-Demand Unstable ELANE 62 42 C[C@H](NC(=O)[C@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937401 CG On-Demand Unstable TRY1_BOVIN 53 34 C[C@H](NC(=O)[C@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937401 CG On-Demand Unstable CTSK 20 40 C[C@H](NC(=O)[C@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937401 CG On-Demand Unstable XIAP 114 46 C[C@H](NC(=O)[C@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937401 CG On-Demand Unstable BIRC3 71 48 C[C@H](NC(=O)[C@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937401 CG On-Demand Unstable BIRC2 79 42 C[C@H](NC(=O)[C@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937401 CG On-Demand Unstable BIRC8 68 48 C[C@H](NC(=O)[C@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937401 CG On-Demand Unstable BRCA1 52 32 O=C(/C=C\c1ccc2c(c1)CCC(=O)N2)CCl ZINC000217937414 BE For-Sale Unstable FABI 44 33 COc1ccc(Br)c(C(=O)NCC[C@@H](O)c2cccn2C)c1 ZINC000217937418 FF In-Stock Unstable DRD4 42 32 Cc1noc2nc(C(C)C)cc(C(=O)Nc3cccc(I)c3)c12 ZINC000217937440 HJ On-Demand Unstable KCNK3 81 38 Cc1noc2nc(C(C)C)cc(C(=O)Nc3cccc(I)c3)c12 ZINC000217937440 HJ On-Demand Unstable KCNK9 69 37 CCN(CCO)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217937472 CD For-Sale Unstable ACHE 0 47 CCN(CCO)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217937472 CD For-Sale Unstable PTGER2 25 42 CCN(CCO)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217937472 CD For-Sale Unstable PTGER4 15 42 COc1cccc(/C=C/NC(=O)NCc2cccc(CN)c2)c1 ZINC000217937479 DF For-Sale Unstable ROCK1 27 41 COc1cccc(/C=C/NC(=O)NCc2cccc(CN)c2)c1 ZINC000217937479 DF For-Sale Unstable MTNR1A 50 44 COc1cccc(/C=C/NC(=O)NCc2cccc(CN)c2)c1 ZINC000217937479 DF For-Sale Unstable MTNR1B 49 44 COc1cccc(/C=C/NC(=O)NCc2cccc(CN)c2)c1 ZINC000217937479 DF For-Sale Unstable ROCK2 34 42 O=C(CCc1nc(-c2ccc(Cl)cc2)no1)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217937488 HH In-Stock Unstable COLA 0 40 O=C(CCc1nc(-c2ccc(Cl)cc2)no1)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217937488 HH In-Stock Unstable CPT1A 16 40 O=C(CCc1nc(-c2ccc(Cl)cc2)no1)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217937488 HH In-Stock Unstable SPHK1 42 40 O=C(CCc1nc(-c2ccc(Cl)cc2)no1)NC[C@@H]1CCCN2CCCC[C@H]12 ZINC000217937488 HH In-Stock Unstable HCAR2 23 41 O=C(/C=C\c1c[nH]c2cc(F)ccc12)CCl ZINC000217937497 BG For-Sale Unstable MPO 66 37 O=C(/C=C\c1c[nH]c2cc(F)ccc12)CCl ZINC000217937497 BG For-Sale Unstable CAPN1 23 53 C[C@@H](NC(=O)[C@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937499 CG On-Demand Unstable F2 41 36 C[C@@H](NC(=O)[C@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937499 CG On-Demand Unstable ACE 41 38 C[C@@H](NC(=O)[C@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937499 CG On-Demand Unstable FKBP1A 28 40 C[C@@H](NC(=O)[C@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937499 CG On-Demand Unstable ELANE 62 42 C[C@@H](NC(=O)[C@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937499 CG On-Demand Unstable TRY1_BOVIN 53 34 C[C@@H](NC(=O)[C@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937499 CG On-Demand Unstable CTSK 20 40 C[C@@H](NC(=O)[C@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937499 CG On-Demand Unstable XIAP 114 46 C[C@@H](NC(=O)[C@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937499 CG On-Demand Unstable BIRC3 71 48 C[C@@H](NC(=O)[C@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937499 CG On-Demand Unstable BIRC2 79 42 C[C@@H](NC(=O)[C@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937499 CG On-Demand Unstable BIRC8 68 48 C[C@@H](NC(=O)[C@H]1CCCN1C1CCCC1)c1ccccc1 ZINC000217937499 CG On-Demand Unstable BRCA1 52 32 COc1ccc(Br)c(C(=O)NCC[C@H](O)c2cccn2C)c1 ZINC000217937500 FF In-Stock Unstable DRD4 42 32 COc1cccc(/C=C/NC(=O)Nc2nc(C)cs2)c1 ZINC000217937588 CG For-Sale Unstable MTNR1A 21 40 COc1cccc(/C=C/NC(=O)Nc2nc(C)cs2)c1 ZINC000217937588 CG For-Sale Unstable MTNR1B 24 40 COc1cccc(/C=C/NC(=O)Nc2nc(C)cs2)c1 ZINC000217937588 CG For-Sale Unstable GCK 18 48 Cn1cccc1[C@H](O)CCNC(=O)c1cc(C2CC2)on1 ZINC000217937603 CD In-Stock Unstable S1PR3 17 41 Cc1noc2nc(C(C)C)cc(C(=O)Nc3ccccc3N3CCCCC3)c12 ZINC000217937647 GJ On-Demand Unstable KCNQ2 85 44 Cc1noc2nc(C(C)C)cc(C(=O)Nc3ccccc3N3CCCCC3)c12 ZINC000217937647 GJ On-Demand Unstable CSF1R 31 48 Cc1noc2nc(C(C)C)cc(C(=O)Nc3ccccc3N3CCCCC3)c12 ZINC000217937647 GJ On-Demand Unstable BRPF1 0 42 CC(C)CN(Cc1ccccc1/C=C\C(=O)O)CC(C)C ZINC000217937657 CH For-Sale Unstable PTGER2 48 51 CC(C)CN(Cc1ccccc1/C=C\C(=O)O)CC(C)C ZINC000217937657 CH For-Sale Unstable PTGER4 0 51 CC(C)CN(Cc1ccccc1/C=C\C(=O)O)CC(C)C ZINC000217937657 CH For-Sale Unstable PTGER3 19 51 CC(C)CN(Cc1ccccc1/C=C\C(=O)O)CC(C)C ZINC000217937657 CH For-Sale Unstable PTGDR 0 49 Cn1cccc1[C@@H](O)CCNC(=O)c1cc(C2CC2)on1 ZINC000217937682 CD In-Stock Unstable S1PR3 17 41 COc1cccc(/C=C/NC(=O)Nc2ccc(C#N)cc2)c1 ZINC000217937703 CG For-Sale Unstable MTNR1A 22 47 COc1cccc(/C=C/NC(=O)Nc2ccc(C#N)cc2)c1 ZINC000217937703 CG For-Sale Unstable MTNR1B 30 47 O=C(CCn1ccnc1)N[C@@H]1CCC[C@@H]1CO ZINC000217937709 BC For-Sale Unstable TBXAS1 28 40 CC[C@@H](NC(=S)Nc1ccccc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217937721 EH In-Stock Unstable PTGS2 21 50 CC[C@@H](NC(=S)Nc1ccccc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217937721 EH In-Stock Unstable CA1 21 46 CC[C@@H](NC(=S)Nc1ccccc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217937721 EH In-Stock Unstable CA4 15 42 CC(C)CN(Cc1ccc(/C=C\C(=O)O)cc1)CC(C)C ZINC000217937763 CH For-Sale Unstable NR1H4 26 40 CCN(CC)S(=O)(=O)c1cc(NC(=O)c2cc(C(C)C)nc3onc(C)c23)ccc1C ZINC000217937775 II On-Demand Unstable SMG1 30 40 O=C(CCn1ccnc1)N[C@H]1CCC[C@@H]1CO ZINC000217937795 BC For-Sale Unstable TBXAS1 28 40 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCc1ccccc1 ZINC000217937796 GE In-Stock Unstable HTR1D 35 43 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCc1ccccc1 ZINC000217937796 GE In-Stock Unstable HTR1B 27 43 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCc1ccccc1 ZINC000217937796 GE In-Stock Unstable SSTR2 47 37 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCc1ccccc1 ZINC000217937796 GE In-Stock Unstable EDNRA 19 42 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCc1ccccc1 ZINC000217937796 GE In-Stock Unstable TACR1 30 45 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCc1ccccc1 ZINC000217937796 GE In-Stock Unstable MC4R 56 50 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCc1ccccc1 ZINC000217937796 GE In-Stock Unstable SSTR4 42 37 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCc1ccccc1 ZINC000217937796 GE In-Stock Unstable TACR2 59 42 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCc1ccccc1 ZINC000217937796 GE In-Stock Unstable CCKAR 56 41 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCc1ccccc1 ZINC000217937796 GE In-Stock Unstable BRS3 28 48 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCc1ccccc1 ZINC000217937796 GE In-Stock Unstable MC3R 43 39 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCc1ccccc1 ZINC000217937796 GE In-Stock Unstable MC5R 39 41 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCc1ccccc1 ZINC000217937796 GE In-Stock Unstable MMP14 55 33 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCc1ccccc1 ZINC000217937796 GE In-Stock Unstable ECE1 40 37 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCc1ccccc1 ZINC000217937796 GE In-Stock Unstable SSTR3 58 38 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCc1ccccc1 ZINC000217937796 GE In-Stock Unstable MMP11 54 33 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCc1ccccc1 ZINC000217937796 GE In-Stock Unstable CCKBR 64 40 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCc1ccccc1 ZINC000217937796 GE In-Stock Unstable GHSR 57 39 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCc1ccccc1 ZINC000217937796 GE In-Stock Unstable MC1R 55 39 O=C(C[C@@H]1NC(=O)N(CCc2c[nH]c3ccccc23)C1=O)NCc1ccccc1 ZINC000217937796 GE In-Stock Unstable KISS1R 40 33 CC[C@H](NC(=S)Nc1ccccc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217937801 EH In-Stock Unstable PTGS2 21 50 CC[C@H](NC(=S)Nc1ccccc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217937801 EH In-Stock Unstable CA1 21 46 CC[C@H](NC(=S)Nc1ccccc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217937801 EH In-Stock Unstable CA4 15 42 COc1cccc(/C=C/NC(=O)Nc2cccc(OC)c2)c1 ZINC000217937815 CG For-Sale Unstable CYP1B1 45 43 COc1cccc(/C=C/NC(=O)Nc2cccc(OC)c2)c1 ZINC000217937815 CG For-Sale Unstable AHR 15 44 COc1cccc(/C=C/NC(=O)Nc2cccc(OC)c2)c1 ZINC000217937815 CG For-Sale Unstable MTNR1A 39 55 COc1cccc(/C=C/NC(=O)Nc2cccc(OC)c2)c1 ZINC000217937815 CG For-Sale Unstable MTNR1B 41 55 COc1cccc(/C=C/NC(=O)Nc2cccc(OC)c2)c1 ZINC000217937815 CG For-Sale Unstable CYP1A1 29 43 COc1cccc(/C=C/NC(=O)Nc2cccc(OC)c2)c1 ZINC000217937815 CG For-Sale Unstable EPHX2 17 49 COc1cccc(/C=C/NC(=O)Nc2cccc(OC)c2)c1 ZINC000217937815 CG For-Sale Unstable IMPDH2 0 42 COc1cccc(/C=C/NC(=O)Nc2cccc(OC)c2)c1 ZINC000217937815 CG For-Sale Unstable TAAR1 35 46 COc1cccc(/C=C/NC(=O)Nc2cccc(OC)c2)c1 ZINC000217937815 CG For-Sale Unstable AKR1C3 25 45 COc1cccc(/C=C/NC(=O)Nc2cccc(OC)c2)c1 ZINC000217937815 CG For-Sale Unstable AKR1C2 42 37 COc1cccc(/C=C/NC(=O)Nc2cccc(OC)c2)c1 ZINC000217937815 CG For-Sale Unstable PSBA 0 52 COc1cccc(/C=C/NC(=O)Nc2cccc(OC)c2)c1 ZINC000217937815 CG For-Sale Unstable KCNK3 41 46 COc1cccc(/C=C/NC(=O)Nc2cccc(OC)c2)c1 ZINC000217937815 CG For-Sale Unstable KCNK9 42 40 C[C@@H](CCO)SCc1ccccc1/C=C\C(=O)O ZINC000217937828 CF For-Sale Unstable PTGER2 43 47 C[C@@H](CCO)SCc1ccccc1/C=C\C(=O)O ZINC000217937828 CF For-Sale Unstable PTGER4 0 47 C[C@@H](CCO)SCc1ccccc1/C=C\C(=O)O ZINC000217937828 CF For-Sale Unstable PTGER3 16 48 COc1ccc([N+](=O)[O-])cc1N[C@@H]1C[C@@H](C)N(C)C[C@@H]1C ZINC000217937862 CF For-Sale Unstable KCNMA1 20 44 O=C(CCn1ccnc1)N[C@@H]1CCC[C@H]1CO ZINC000217937864 BC For-Sale Unstable TBXAS1 28 40 C[C@H](CCO)SCc1ccccc1/C=C\C(=O)O ZINC000217937901 CF For-Sale Unstable PTGER2 43 47 C[C@H](CCO)SCc1ccccc1/C=C\C(=O)O ZINC000217937901 CF For-Sale Unstable PTGER4 0 47 C[C@H](CCO)SCc1ccccc1/C=C\C(=O)O ZINC000217937901 CF For-Sale Unstable PTGER3 16 48 COc1ccc(-c2noc(CNC(=S)Nc3ccccc3)n2)c(OC)c1 ZINC000217937922 FG In-Stock Unstable MAPKAPK2 0 41 COc1cccc(/C=C/NC(=O)Nc2cc(Cl)ccc2O)c1 ZINC000217937923 DH For-Sale Unstable KCNMA1 26 42 O=C(CCn1ccnc1)N[C@H]1CCC[C@H]1CO ZINC000217937942 BC For-Sale Unstable TBXAS1 28 40 COc1ccc([N+](=O)[O-])cc1N[C@H]1C[C@@H](C)N(C)C[C@@H]1C ZINC000217937952 CF For-Sale Unstable KCNMA1 20 44 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cc(Br)ccc1Cl ZINC000217937956 JI For-Sale Unstable HCRTR2 40 38 CCO[C@@H]1C[C@@H](NC(=O)NC2CCCCC2)C1(C)C ZINC000217937969 CF For-Sale Unstable EPHX2 20 47 CCOc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1OCC ZINC000217938011 FI For-Sale Unstable MTNR1A 34 43 CCOc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1OCC ZINC000217938011 FI For-Sale Unstable MTNR1B 42 43 CCOc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1OCC ZINC000217938011 FI For-Sale Unstable IMPDH2 0 40 CCOc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1OCC ZINC000217938011 FI For-Sale Unstable KCNK3 31 40 CCOc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1OCC ZINC000217938011 FI For-Sale Unstable KCNK9 23 40 O=C(O)CCCCCNCl ZINC000217938013 AD For-Sale Unstable FABP4 19 48 O=C(O)CCCCCNCl ZINC000217938013 AD For-Sale Unstable FABP5 16 48 O=C(O)CCCCCNCl ZINC000217938013 AD For-Sale Unstable KDM2A 43 35 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cc(Br)ccc1Cl ZINC000217938031 JI For-Sale Unstable HCRTR2 40 38 COc1ccc([N+](=O)[O-])cc1N[C@@H]1C[C@H](C)N(C)C[C@@H]1C ZINC000217938034 CF For-Sale Unstable KCNMA1 20 44 CCO[C@H]1C[C@@H](NC(=O)NC2CCCCC2)C1(C)C ZINC000217938035 CF For-Sale Unstable EPHX2 20 47 COc1ccccc1NC(=O)c1ccc(NC(=O)c2cc(C(C)C)nc3onc(C)c23)cc1 ZINC000217938058 IK On-Demand Unstable PRNP 40 36 COc1ccccc1NC(=O)c1ccc(NC(=O)c2cc(C(C)C)nc3onc(C)c23)cc1 ZINC000217938058 IK On-Demand Unstable NR1H4 21 46 COc1ccccc1NC(=O)c1ccc(NC(=O)c2cc(C(C)C)nc3onc(C)c23)cc1 ZINC000217938058 IK On-Demand Unstable KCNK3 75 42 COc1ccccc1NC(=O)c1ccc(NC(=O)c2cc(C(C)C)nc3onc(C)c23)cc1 ZINC000217938058 IK On-Demand Unstable KCNK9 55 42 C[C@H](NCl)C(=O)NCC(=O)O ZINC000217938096 AB For-Sale Unstable ECE1 36 50 C[C@H](NCl)C(=O)NCC(=O)O ZINC000217938096 AB For-Sale Unstable ACE2 19 48 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cc(Br)ccc1Cl ZINC000217938108 JI For-Sale Unstable HCRTR2 40 38 COc1cccc(/C=C/NC(=O)Nc2nccs2)c1 ZINC000217938114 CF For-Sale Unstable MAP1 114 41 COc1cc(C(=O)CCN)ccc1Br ZINC000217938116 CD For-Sale Unstable THRA 29 42 Cn1cccc1[C@H](O)CCNC(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217938117 EF In-Stock Unstable GCGR 58 48 Cn1cccc1[C@H](O)CCNC(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217938117 EF In-Stock Unstable TRPV1 0 53 Cn1cccc1[C@H](O)CCNC(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217938117 EF In-Stock Unstable SCN9A 0 45 Cn1cccc1[C@H](O)CCNC(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217938117 EF In-Stock Unstable GIPR 50 40 Cn1cccc1[C@H](O)CCNC(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217938117 EF In-Stock Unstable SHH 43 34 CCO[C@@H]1C[C@H](NC(=O)NC2CCCCC2)C1(C)C ZINC000217938126 CF For-Sale Unstable EPHX2 20 47 COc1ccc([N+](=O)[O-])cc1N[C@H]1C[C@H](C)N(C)C[C@@H]1C ZINC000217938127 CF For-Sale Unstable KCNMA1 20 44 CCOc1ccc(NC(=O)c2ccc(NC(=O)c3cc(C(C)C)nc4onc(C)c34)cc2)cc1 ZINC000217938151 JK On-Demand Unstable PRNP 33 45 CCOc1ccc(NC(=O)c2ccc(NC(=O)c3cc(C(C)C)nc4onc(C)c34)cc2)cc1 ZINC000217938151 JK On-Demand Unstable P4HTM 0 46 CCOc1ccc(NC(=O)c2ccc(NC(=O)c3cc(C(C)C)nc4onc(C)c34)cc2)cc1 ZINC000217938151 JK On-Demand Unstable SHH 41 32 C[C@@H](NCl)C(=O)NCC(=O)O ZINC000217938166 AB For-Sale Unstable ECE1 36 50 C[C@@H](NCl)C(=O)NCC(=O)O ZINC000217938166 AB For-Sale Unstable ACE2 19 48 CC(C)c1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217938170 DJ In-Stock Unstable ADRB1 17 43 CC(C)c1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217938170 DJ In-Stock Unstable ADRB3 21 43 CC(C)c1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217938170 DJ In-Stock Unstable SCN2A 32 41 CC(C)c1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217938170 DJ In-Stock Unstable MMP3 20 43 CC(C)c1ccc(CCCNC(=S)Nc2ccccc2)cc1 ZINC000217938170 DJ In-Stock Unstable AMP1_PLAFQ 24 41 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cc(Br)ccc1Cl ZINC000217938173 JI For-Sale Unstable HCRTR2 40 38 Cn1cccc1[C@@H](O)CCNC(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217938192 EF In-Stock Unstable GCGR 58 48 Cn1cccc1[C@@H](O)CCNC(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217938192 EF In-Stock Unstable TRPV1 0 53 Cn1cccc1[C@@H](O)CCNC(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217938192 EF In-Stock Unstable SCN9A 0 45 Cn1cccc1[C@@H](O)CCNC(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217938192 EF In-Stock Unstable GIPR 50 40 Cn1cccc1[C@@H](O)CCNC(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217938192 EF In-Stock Unstable SHH 43 34 CCO[C@H]1C[C@H](NC(=O)NC2CCCCC2)C1(C)C ZINC000217938193 CF For-Sale Unstable EPHX2 20 47 CC[C@@H](CCO)NC(=O)CCCN ZINC000217938195 AC For-Sale Unstable PLA2G2C 0 40 CC[C@@H](CCO)NC(=O)CCCN ZINC000217938195 AC For-Sale Unstable NOD1 61 42 COc1cccc(/C=C/NC(=O)Nc2cccc(SC)c2)c1 ZINC000217938228 DI For-Sale Unstable MTNR1A 25 44 COc1cccc(/C=C/NC(=O)Nc2cccc(SC)c2)c1 ZINC000217938228 DI For-Sale Unstable MTNR1B 31 44 COc1cccc(/C=C/NC(=O)Nc2cccc(SC)c2)c1 ZINC000217938228 DI For-Sale Unstable TAAR1 29 41 Cc1ccccc1N1CCCN(C(=O)c2cc(CC(C)C)nc(N)n2)CC1 ZINC000217938248 FF In-Stock Unstable KCNQ2 46 31 CC[C@H](CCO)NC(=O)CCCN ZINC000217938266 AC For-Sale Unstable PLA2G2C 0 40 CC[C@H](CCO)NC(=O)CCCN ZINC000217938266 AC For-Sale Unstable NOD1 61 42 S=C(NCCCN1CCCc2ccccc21)Nc1ccccc1 ZINC000217938275 EH In-Stock Unstable AVPR2 23 42 S=C(NCCCN1CCCc2ccccc21)Nc1ccccc1 ZINC000217938275 EH In-Stock Unstable QPCT 53 39 S=C(NCCCN1CCCc2ccccc21)Nc1ccccc1 ZINC000217938275 EH In-Stock Unstable NAMPT 0 43 Cn1cccc1[C@H](O)CCNC(=O)c1cc(-c2ccc(F)cc2)nn1C ZINC000217938299 FE In-Stock Unstable HMGCR 52 38 Cn1cccc1[C@H](O)CCNC(=O)c1cc(-c2ccc(F)cc2)nn1C ZINC000217938299 FE In-Stock Unstable EPHX2 0 40 CC1(C)C[C@H]2C[C@](C)(CN2[C@@H](C(=O)O)c2c[nH]c3cc(NC(=O)c4ccccc4)ccc23)C1 ZINC000217938312 IK In-Stock Unstable AVPR2 16 43 CC1(C)C[C@H]2C[C@](C)(CN2[C@@H](C(=O)O)c2c[nH]c3cc(NC(=O)c4ccccc4)ccc23)C1 ZINC000217938312 IK In-Stock Unstable AVPR1A 33 43 CN(Cc1ccoc1)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217938315 CG For-Sale Unstable AKR1C3 40 39 C[C@H]1Cc2ccccc2N(S(=O)(=O)[C@H](C)C(=O)O)C1 ZINC000217938341 CD For-Sale Unstable ACE 21 43 C[C@H]1Cc2ccccc2N(S(=O)(=O)[C@H](C)C(=O)O)C1 ZINC000217938341 CD For-Sale Unstable TPP2 48 33 COc1ccc(/C=C\c2csc(N)n2)c(F)c1 ZINC000217938342 CG For-Sale Unstable CYP1B1 41 40 COc1ccc(/C=C\c2csc(N)n2)c(F)c1 ZINC000217938342 CG For-Sale Unstable CYP1A1 37 40 COc1cccc(/C=C/NC(=O)Nc2cc(S(=O)(=O)N3CCOCC3)ccc2Cl)c1 ZINC000217938343 JG For-Sale Unstable LPL 47 40 COc1cccc(/C=C/NC(=O)Nc2cc(S(=O)(=O)N3CCOCC3)ccc2Cl)c1 ZINC000217938343 JG For-Sale Unstable PKM 23 44 COc1cccc(/C=C/NC(=O)Nc2cc(S(=O)(=O)N3CCOCC3)ccc2Cl)c1 ZINC000217938343 JG For-Sale Unstable LIPG 19 40 CC[C@@H](CCO)NC(=O)CCCCCN ZINC000217938369 BC For-Sale Unstable PLA2G2C 0 45 CC[C@@H](CCO)NC(=O)CCCCCN ZINC000217938369 BC For-Sale Unstable NMT1 33 44 CC[C@@H](CCO)NC(=O)CCCCCN ZINC000217938369 BC For-Sale Unstable Q6UB75_PIG 0 42 CC[C@@H](CCO)NC(=O)CCCCCN ZINC000217938369 BC For-Sale Unstable NOD1 76 50 CC[C@@H](CCO)NC(=O)CCCCCN ZINC000217938369 BC For-Sale Unstable CQSS 40 32 Cn1cccc1[C@@H](O)CCNC(=O)c1cc(-c2ccc(F)cc2)nn1C ZINC000217938380 FE In-Stock Unstable HMGCR 52 38 Cn1cccc1[C@@H](O)CCNC(=O)c1cc(-c2ccc(F)cc2)nn1C ZINC000217938380 FE In-Stock Unstable EPHX2 0 40 COc1cccc(C(=O)NCCCc2ccccc2OC)c1 ZINC000217938397 CG In-Stock Unstable HTR1A 20 60 COc1cccc(C(=O)NCCCc2ccccc2OC)c1 ZINC000217938397 CG In-Stock Unstable DRD2 29 48 COc1cccc(C(=O)NCCCc2ccccc2OC)c1 ZINC000217938397 CG In-Stock Unstable DRD1 0 49 COc1cccc(C(=O)NCCCc2ccccc2OC)c1 ZINC000217938397 CG In-Stock Unstable DRD4 62 48 COc1cccc(C(=O)NCCCc2ccccc2OC)c1 ZINC000217938397 CG In-Stock Unstable ACHE 0 45 COc1cccc(C(=O)NCCCc2ccccc2OC)c1 ZINC000217938397 CG In-Stock Unstable ADRA1D 16 40 COc1cccc(C(=O)NCCCc2ccccc2OC)c1 ZINC000217938397 CG In-Stock Unstable DRD3 43 51 COc1cccc(C(=O)NCCCc2ccccc2OC)c1 ZINC000217938397 CG In-Stock Unstable PTAFR 15 45 COc1cccc(C(=O)NCCCc2ccccc2OC)c1 ZINC000217938397 CG In-Stock Unstable NQO2 33 55 COc1cccc(C(=O)NCCCc2ccccc2OC)c1 ZINC000217938397 CG In-Stock Unstable TRPV1 0 44 COc1cccc(C(=O)NCCCc2ccccc2OC)c1 ZINC000217938397 CG In-Stock Unstable ECR 18 43 COc1cccc(C(=O)NCCCc2ccccc2OC)c1 ZINC000217938397 CG In-Stock Unstable MTNR1A 105 50 COc1cccc(C(=O)NCCCc2ccccc2OC)c1 ZINC000217938397 CG In-Stock Unstable MTNR1B 93 55 COc1cccc(C(=O)NCCCc2ccccc2OC)c1 ZINC000217938397 CG In-Stock Unstable ABCB1 26 40 COc1cccc(C(=O)NCCCc2ccccc2OC)c1 ZINC000217938397 CG In-Stock Unstable MT-ND1 16 41 COc1cccc(C(=O)NCCCc2ccccc2OC)c1 ZINC000217938397 CG In-Stock Unstable TAAR1 26 41 COc1cccc(C(=O)NCCCc2ccccc2OC)c1 ZINC000217938397 CG In-Stock Unstable CRTM 42 37 COc1cccc(C(=O)NCCCc2ccccc2OC)c1 ZINC000217938397 CG In-Stock Unstable KCNK3 44 38 COc1cccc(C(=O)NCCCc2ccccc2OC)c1 ZINC000217938397 CG In-Stock Unstable KCNK9 42 38 COc1ccc(/C=C\c2csc(N)n2)c(Cl)c1 ZINC000217938426 CH For-Sale Unstable CYP1B1 41 40 COc1ccc(/C=C\c2csc(N)n2)c(Cl)c1 ZINC000217938426 CH For-Sale Unstable CYP1A1 37 40 CC[C@H](CCO)NC(=O)CCCCCN ZINC000217938440 BC For-Sale Unstable PLA2G2C 0 45 CC[C@H](CCO)NC(=O)CCCCCN ZINC000217938440 BC For-Sale Unstable NMT1 33 44 CC[C@H](CCO)NC(=O)CCCCCN ZINC000217938440 BC For-Sale Unstable Q6UB75_PIG 0 42 CC[C@H](CCO)NC(=O)CCCCCN ZINC000217938440 BC For-Sale Unstable NOD1 76 50 CC[C@H](CCO)NC(=O)CCCCCN ZINC000217938440 BC For-Sale Unstable CQSS 40 32 COc1cccc(/C=C/NC(=O)NCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217938441 FD For-Sale Unstable CA2 98 54 COc1cccc(/C=C/NC(=O)NCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217938441 FD For-Sale Unstable CA1 80 54 COc1cccc(/C=C/NC(=O)NCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217938441 FD For-Sale Unstable CA7 51 50 COc1cccc(/C=C/NC(=O)NCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217938441 FD For-Sale Unstable MMP13 23 40 COc1cccc(/C=C/NC(=O)NCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217938441 FD For-Sale Unstable CA5B 41 44 COc1cccc(/C=C/NC(=O)NCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217938441 FD For-Sale Unstable CA4 59 47 COc1cccc(/C=C/NC(=O)NCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217938441 FD For-Sale Unstable CA5A 43 44 COc1cccc(/C=C/NC(=O)NCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217938441 FD For-Sale Unstable CA14 49 50 COc1cccc(/C=C/NC(=O)NCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217938441 FD For-Sale Unstable MTNR1A 41 40 COc1cccc(/C=C/NC(=O)NCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217938441 FD For-Sale Unstable MTNR1B 41 40 COc1cccc(/C=C/NC(=O)NCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217938441 FD For-Sale Unstable CA12 68 54 COc1cccc(/C=C/NC(=O)NCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217938441 FD For-Sale Unstable CA9 77 54 COc1cccc(/C=C/NC(=O)NCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217938441 FD For-Sale Unstable UREA_CANEN 21 43 COc1cccc(/C=C/NC(=O)NCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217938441 FD For-Sale Unstable CYNT 19 41 COc1cccc(/C=C/NC(=O)NCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217938441 FD For-Sale Unstable MTCA1 36 45 COc1cccc(/C=C/NC(=O)NCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217938441 FD For-Sale Unstable P96878_MYCTU 45 45 COc1cccc(/C=C/NC(=O)NCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217938441 FD For-Sale Unstable NAMPT 32 40 COCCCn1c(C)cc(C)c(C(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)c1=O ZINC000217938465 HD In-Stock Unstable CHRNA4 27 46 CCOc1ccc(CCCNC(=O)c2cccc(OC)c2)cc1 ZINC000217938501 DG In-Stock Unstable DRD4 59 45 CCOc1ccc(CCCNC(=O)c2cccc(OC)c2)cc1 ZINC000217938501 DG In-Stock Unstable DRD3 19 47 CCOc1ccc(CCCNC(=O)c2cccc(OC)c2)cc1 ZINC000217938501 DG In-Stock Unstable PTAFR 22 48 CCOc1ccc(CCCNC(=O)c2cccc(OC)c2)cc1 ZINC000217938501 DG In-Stock Unstable NQO2 24 47 CCOc1ccc(CCCNC(=O)c2cccc(OC)c2)cc1 ZINC000217938501 DG In-Stock Unstable SCN2A 23 47 CCOc1ccc(CCCNC(=O)c2cccc(OC)c2)cc1 ZINC000217938501 DG In-Stock Unstable MTNR1A 94 48 CCOc1ccc(CCCNC(=O)c2cccc(OC)c2)cc1 ZINC000217938501 DG In-Stock Unstable MTNR1B 74 55 CCOc1ccc(CCCNC(=O)c2cccc(OC)c2)cc1 ZINC000217938501 DG In-Stock Unstable SLC6A5 27 42 CCOc1ccc(CCCNC(=O)c2cccc(OC)c2)cc1 ZINC000217938501 DG In-Stock Unstable CRTM 62 38 CCOc1ccc(CCCNC(=O)c2cccc(OC)c2)cc1 ZINC000217938501 DG In-Stock Unstable ALPHA-1A 0 44 CCOc1ccc(CCCNC(=O)c2cccc(OC)c2)cc1 ZINC000217938501 DG In-Stock Unstable PDS 42 40 COc1ccc(/C=C\c2csc(N)n2)c(OC)c1OC ZINC000217938513 CF For-Sale Unstable CYP1B1 31 45 COc1cccc(/C=C/NC(=O)Nc2cccnc2Cl)c1 ZINC000217938540 DH For-Sale Unstable G2YM83_BOTF4 66 34 COCCN(C)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217938563 CD For-Sale Unstable TUBB1 42 38 COCCN(C)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217938563 CD For-Sale Unstable AKR1C3 23 42 COCCN(C)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217938563 CD For-Sale Unstable ABCG2 15 43 CC(C)NC(=O)c1ccccc1NC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217938577 GF In-Stock Unstable CHRNA4 29 45 CC(C)NC(=O)c1ccccc1NC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217938577 GF In-Stock Unstable RBP4 61 39 O=C1C/C(=C2/CCN(Cc3ccccc3)C2)C(=O)N1 ZINC000217938596 CD For-Sale Unstable DRD4 15 43 O=C1C/C(=C2/CCN(Cc3ccccc3)C2)C(=O)N1 ZINC000217938596 CD For-Sale Unstable SIGMAR1 35 41 CCCOc1ccccc1CCCNC(=O)c1cccc(OC)c1 ZINC000217938600 EH In-Stock Unstable DRD2 18 47 CCCOc1ccccc1CCCNC(=O)c1cccc(OC)c1 ZINC000217938600 EH In-Stock Unstable DRD1 0 47 CCCOc1ccccc1CCCNC(=O)c1cccc(OC)c1 ZINC000217938600 EH In-Stock Unstable DRD4 57 44 CCCOc1ccccc1CCCNC(=O)c1cccc(OC)c1 ZINC000217938600 EH In-Stock Unstable DRD3 30 47 CCCOc1ccccc1CCCNC(=O)c1cccc(OC)c1 ZINC000217938600 EH In-Stock Unstable PTAFR 16 41 CCCOc1ccccc1CCCNC(=O)c1cccc(OC)c1 ZINC000217938600 EH In-Stock Unstable NQO2 23 49 CCCOc1ccccc1CCCNC(=O)c1cccc(OC)c1 ZINC000217938600 EH In-Stock Unstable MTNR1A 98 49 CCCOc1ccccc1CCCNC(=O)c1cccc(OC)c1 ZINC000217938600 EH In-Stock Unstable MTNR1B 85 51 CCCOc1ccccc1CCCNC(=O)c1cccc(OC)c1 ZINC000217938600 EH In-Stock Unstable ABCB1 22 43 CCCOc1ccccc1CCCNC(=O)c1cccc(OC)c1 ZINC000217938600 EH In-Stock Unstable ALPHA-1A 0 47 COc1cccc(/C=C/NC(=O)N2C[C@@H](C)C[C@@H](C)C2)c1 ZINC000217938652 CG For-Sale Unstable DRD4 40 30 COc1cccc(/C=C/NC(=O)N2C[C@@H](C)C[C@@H](C)C2)c1 ZINC000217938652 CG For-Sale Unstable MTNR1A 27 40 COc1cccc(/C=C/NC(=O)N2C[C@@H](C)C[C@@H](C)C2)c1 ZINC000217938652 CG For-Sale Unstable MTNR1B 37 40 COc1cccc(/C=C/NC(=O)N2C[C@@H](C)C[C@@H](C)C2)c1 ZINC000217938652 CG For-Sale Unstable RORC 37 44 COCCN(C)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217938674 CD For-Sale Unstable PTGER2 35 46 COCCN(C)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217938674 CD For-Sale Unstable PTGER4 19 46 COCCN(C)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217938674 CD For-Sale Unstable PTGER3 18 40 COCCN(C)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217938674 CD For-Sale Unstable AKR1B10 29 40 Cn1cccc1[C@H](O)CCNC(=O)Cc1c(F)cccc1Cl ZINC000217938695 DF In-Stock Unstable P2RX7 37 45 COc1cccc(C(=O)N[C@@H](C)c2ccc(N3CCC(C)CC3)cc2)c1 ZINC000217938707 FI In-Stock Unstable DRD4 58 48 COc1cccc(C(=O)N[C@@H](C)c2ccc(N3CCC(C)CC3)cc2)c1 ZINC000217938707 FI In-Stock Unstable PRKD1 31 41 COc1cccc(C(=O)N[C@@H](C)c2ccc(N3CCC(C)CC3)cc2)c1 ZINC000217938707 FI In-Stock Unstable BRPF1 0 42 COc1cccc(/C=C/NC(=O)N2C[C@H](C)C[C@@H](C)C2)c1 ZINC000217938739 CG For-Sale Unstable DRD4 40 30 COc1cccc(/C=C/NC(=O)N2C[C@H](C)C[C@@H](C)C2)c1 ZINC000217938739 CG For-Sale Unstable MTNR1A 27 40 COc1cccc(/C=C/NC(=O)N2C[C@H](C)C[C@@H](C)C2)c1 ZINC000217938739 CG For-Sale Unstable MTNR1B 37 40 COc1cccc(/C=C/NC(=O)N2C[C@H](C)C[C@@H](C)C2)c1 ZINC000217938739 CG For-Sale Unstable RORC 37 44 Cn1cccc1[C@@H](O)CCNC(=O)Cc1c(F)cccc1Cl ZINC000217938759 DF In-Stock Unstable P2RX7 37 45 Cc1n[nH]c(C)c1CCNC(=O)CSCc1ccccc1Cl ZINC000217938768 EG In-Stock Unstable P2RX7 31 59 COc1cccc(C(=O)N[C@H](C)c2ccc(N3CCC(C)CC3)cc2)c1 ZINC000217938784 FI In-Stock Unstable DRD4 58 48 COc1cccc(C(=O)N[C@H](C)c2ccc(N3CCC(C)CC3)cc2)c1 ZINC000217938784 FI In-Stock Unstable PRKD1 31 41 COc1cccc(C(=O)N[C@H](C)c2ccc(N3CCC(C)CC3)cc2)c1 ZINC000217938784 FI In-Stock Unstable BRPF1 0 42 O=C(O)/C=C\c1ccccc1CN1CCN(C2CC2)CC1 ZINC000217938787 CE For-Sale Unstable PTGER2 34 46 O=C(O)/C=C\c1ccccc1CN1CCN(C2CC2)CC1 ZINC000217938787 CE For-Sale Unstable PTGER4 17 46 O=C(O)/C=C\c1ccccc1CN1CCN(C2CC2)CC1 ZINC000217938787 CE For-Sale Unstable PTGER3 18 46 O=C(O)/C=C\c1ccccc1CN1CCN(C2CC2)CC1 ZINC000217938787 CE For-Sale Unstable PTGDR 16 42 COc1cccc(/C=C/NC(=O)N2C[C@@H](C)C[C@H](C)C2)c1 ZINC000217938821 CG For-Sale Unstable DRD4 40 30 COc1cccc(/C=C/NC(=O)N2C[C@@H](C)C[C@H](C)C2)c1 ZINC000217938821 CG For-Sale Unstable MTNR1A 27 40 COc1cccc(/C=C/NC(=O)N2C[C@@H](C)C[C@H](C)C2)c1 ZINC000217938821 CG For-Sale Unstable MTNR1B 37 40 COc1cccc(/C=C/NC(=O)N2C[C@@H](C)C[C@H](C)C2)c1 ZINC000217938821 CG For-Sale Unstable RORC 37 44 CC[C@@H](CCO)NC(=O)CCCCCCN ZINC000217938858 BD For-Sale Unstable PLA2G2C 0 45 CC[C@@H](CCO)NC(=O)CCCCCCN ZINC000217938858 BD For-Sale Unstable NMT1 33 44 CC[C@@H](CCO)NC(=O)CCCCCCN ZINC000217938858 BD For-Sale Unstable Q6UB75_PIG 0 42 CC[C@@H](CCO)NC(=O)CCCCCCN ZINC000217938858 BD For-Sale Unstable NOD1 76 50 CC[C@@H](CCO)NC(=O)CCCCCCN ZINC000217938858 BD For-Sale Unstable CQSS 40 32 O=C(O)/C=C\c1ccc(CN2CCN(C3CC3)CC2)cc1 ZINC000217938891 CE For-Sale Unstable SIGMAR1 42 48 O=C(O)/C=C\c1ccc(CN2CCN(C3CC3)CC2)cc1 ZINC000217938891 CE For-Sale Unstable L3MBTL3 49 46 COc1cccc(C(=O)N[C@@H](C)c2ccc(N3CCC[C@@H](C)C3)cc2)c1 ZINC000217938895 FI In-Stock Unstable DRD4 54 44 COc1cccc(C(=O)N[C@@H](C)c2ccc(N3CCC[C@@H](C)C3)cc2)c1 ZINC000217938895 FI In-Stock Unstable CTSL 15 40 COc1cccc(C(=O)N[C@@H](C)c2ccc(N3CCC[C@@H](C)C3)cc2)c1 ZINC000217938895 FI In-Stock Unstable PRKD1 34 41 COc1cccc(C(=O)N[C@@H](C)c2ccc(N3CCC[C@@H](C)C3)cc2)c1 ZINC000217938895 FI In-Stock Unstable MTNR1B 19 40 COc1cccc(C(=O)N[C@@H](C)c2ccc(N3CCC[C@@H](C)C3)cc2)c1 ZINC000217938895 FI In-Stock Unstable RORC 45 39 COc1cccc(C(=O)N[C@@H](C)c2ccc(N3CCC[C@@H](C)C3)cc2)c1 ZINC000217938895 FI In-Stock Unstable BRPF1 0 44 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccccc1Oc1ccccc1 ZINC000217938901 II For-Sale Unstable CFTR 21 42 CNCCc1c(Cl)cccc1Br ZINC000217938903 BF For-Sale Unstable TAAR1 22 52 COc1cccc(/C=C/NC(=O)Nc2ncccn2)c1 ZINC000217938932 CE For-Sale Unstable CYP1B1 15 40 COc1cccc(/C=C/NC(=O)Nc2ncccn2)c1 ZINC000217938932 CE For-Sale Unstable MTNR1A 29 42 COc1cccc(/C=C/NC(=O)Nc2ncccn2)c1 ZINC000217938932 CE For-Sale Unstable MTNR1B 33 42 CC[C@H](CCO)NC(=O)CCCCCCN ZINC000217938950 BD For-Sale Unstable PLA2G2C 0 45 CC[C@H](CCO)NC(=O)CCCCCCN ZINC000217938950 BD For-Sale Unstable NMT1 33 44 CC[C@H](CCO)NC(=O)CCCCCCN ZINC000217938950 BD For-Sale Unstable Q6UB75_PIG 0 42 CC[C@H](CCO)NC(=O)CCCCCCN ZINC000217938950 BD For-Sale Unstable NOD1 76 50 CC[C@H](CCO)NC(=O)CCCCCCN ZINC000217938950 BD For-Sale Unstable CQSS 40 32 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccccc1Oc1ccccc1 ZINC000217938965 II For-Sale Unstable CFTR 21 42 COc1cccc(C(=O)N[C@H](C)c2ccc(N3CCC[C@@H](C)C3)cc2)c1 ZINC000217938969 FI In-Stock Unstable DRD4 54 44 COc1cccc(C(=O)N[C@H](C)c2ccc(N3CCC[C@@H](C)C3)cc2)c1 ZINC000217938969 FI In-Stock Unstable CTSL 15 40 COc1cccc(C(=O)N[C@H](C)c2ccc(N3CCC[C@@H](C)C3)cc2)c1 ZINC000217938969 FI In-Stock Unstable PRKD1 34 41 COc1cccc(C(=O)N[C@H](C)c2ccc(N3CCC[C@@H](C)C3)cc2)c1 ZINC000217938969 FI In-Stock Unstable MTNR1B 19 40 COc1cccc(C(=O)N[C@H](C)c2ccc(N3CCC[C@@H](C)C3)cc2)c1 ZINC000217938969 FI In-Stock Unstable RORC 45 39 COc1cccc(C(=O)N[C@H](C)c2ccc(N3CCC[C@@H](C)C3)cc2)c1 ZINC000217938969 FI In-Stock Unstable BRPF1 0 44 O=C(O)/C=C\c1cccc(CN2CCN(C3CC3)CC2)c1 ZINC000217938993 CE For-Sale Unstable DRD2 21 40 O=C(O)/C=C\c1cccc(CN2CCN(C3CC3)CC2)c1 ZINC000217938993 CE For-Sale Unstable DRD4 41 39 O=C(O)/C=C\c1cccc(CN2CCN(C3CC3)CC2)c1 ZINC000217938993 CE For-Sale Unstable ACHE 27 43 O=C(O)/C=C\c1cccc(CN2CCN(C3CC3)CC2)c1 ZINC000217938993 CE For-Sale Unstable SIGMAR1 52 49 O=C(O)/C=C\c1cccc(CN2CCN(C3CC3)CC2)c1 ZINC000217938993 CE For-Sale Unstable CCR3 18 40 O=C(O)/C=C\c1cccc(CN2CCN(C3CC3)CC2)c1 ZINC000217938993 CE For-Sale Unstable L3MBTL3 30 44 COc1cccc(/C=C/NC(=O)Nc2ccccc2F)c1 ZINC000217939038 CH For-Sale Unstable MTNR1A 27 41 COc1cccc(/C=C/NC(=O)Nc2ccccc2F)c1 ZINC000217939038 CH For-Sale Unstable MTNR1B 30 41 COc1cccc(/C=C/NC(=O)Nc2ccccc2F)c1 ZINC000217939038 CH For-Sale Unstable TAAR1 21 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccccc1Oc1ccccc1 ZINC000217939044 II For-Sale Unstable CFTR 21 42 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1cccc([N+](=O)[O-])c1 ZINC000217939059 CI For-Sale Unstable TRPM8 25 43 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1cccc([N+](=O)[O-])c1 ZINC000217939059 CI For-Sale Unstable OSIGBA0132E09-OSIGBA0108L24.11 0 40 O=C1C/C(=C2/CCCN(Cc3ccccc3)C2)C(=O)N1 ZINC000217939074 CD For-Sale Unstable NOX1 41 35 O=C(CCCC(=O)c1ccccc1)N[C@@H]1CCOC1 ZINC000217939088 CD In-Stock Unstable HDAC8 31 41 O=C(CCCC(=O)c1ccccc1)N[C@@H]1CCOC1 ZINC000217939088 CD In-Stock Unstable CYP2J2 53 38 COc1cccc(C(=O)N[C@@H]2CC(C)(C)Oc3ccc(C)cc32)c1 ZINC000217939093 EI In-Stock Unstable DRD4 46 39 COc1cccc(C(=O)N[C@@H]2CC(C)(C)Oc3ccc(C)cc32)c1 ZINC000217939093 EI In-Stock Unstable KCNK3 23 45 COc1ccc(CN2CCN(C)CC2)cc1/C=C\C(=O)O ZINC000217939107 CD For-Sale Unstable DRD2 27 40 COc1ccc(CN2CCN(C)CC2)cc1/C=C\C(=O)O ZINC000217939107 CD For-Sale Unstable ACHE 21 45 COc1ccc(CN2CCN(C)CC2)cc1/C=C\C(=O)O ZINC000217939107 CD For-Sale Unstable DRD3 25 40 COc1ccc(CN2CCN(C)CC2)cc1/C=C\C(=O)O ZINC000217939107 CD For-Sale Unstable PTGER2 35 43 COc1ccc(CN2CCN(C)CC2)cc1/C=C\C(=O)O ZINC000217939107 CD For-Sale Unstable PTGER4 22 43 COc1ccc(CN2CCN(C)CC2)cc1/C=C\C(=O)O ZINC000217939107 CD For-Sale Unstable PTGER3 19 43 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccccc1Oc1ccccc1 ZINC000217939114 II For-Sale Unstable CFTR 21 42 COc1cccc(/C=C/NC(=O)N(C)c2ccccc2)c1 ZINC000217939132 CH For-Sale Unstable CYP1B1 22 40 COc1cccc(/C=C/NC(=O)N(C)c2ccccc2)c1 ZINC000217939132 CH For-Sale Unstable MTNR1A 36 51 COc1cccc(/C=C/NC(=O)N(C)c2ccccc2)c1 ZINC000217939132 CH For-Sale Unstable MTNR1B 40 51 COc1cccc(/C=C/NC(=O)N(C)c2ccccc2)c1 ZINC000217939132 CH For-Sale Unstable CYP1A1 15 40 COc1cccc(/C=C/NC(=O)N(C)c2ccccc2)c1 ZINC000217939132 CH For-Sale Unstable HSD17B2 24 43 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1cccc([N+](=O)[O-])c1 ZINC000217939139 CI For-Sale Unstable TRPM8 25 43 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1cccc([N+](=O)[O-])c1 ZINC000217939139 CI For-Sale Unstable OSIGBA0132E09-OSIGBA0108L24.11 0 40 O=C(CCCC(=O)c1ccccc1)N[C@H]1CCOC1 ZINC000217939156 CD In-Stock Unstable HDAC8 31 41 O=C(CCCC(=O)c1ccccc1)N[C@H]1CCOC1 ZINC000217939156 CD In-Stock Unstable CYP2J2 53 38 COc1cccc(C(=O)N[C@H]2CC(C)(C)Oc3ccc(C)cc32)c1 ZINC000217939172 EI In-Stock Unstable DRD4 46 39 COc1cccc(C(=O)N[C@H]2CC(C)(C)Oc3ccc(C)cc32)c1 ZINC000217939172 EI In-Stock Unstable KCNK3 23 45 COc1cccc2c(O)c(C(=O)NCCCCCc3nc4ccccc4n3C)cnc12 ZINC000217939197 HH In-Stock Unstable DRD2 19 41 COc1cccc2c(O)c(C(=O)NCCCCCc3nc4ccccc4n3C)cnc12 ZINC000217939197 HH In-Stock Unstable DRD3 35 42 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCCCc1ccccc1 ZINC000217939211 GH For-Sale Unstable FKBP1A 41 38 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCCCc1ccccc1 ZINC000217939211 GH For-Sale Unstable PREP 46 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCCCc1ccccc1 ZINC000217939211 GH For-Sale Unstable FAAH 71 42 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCCCc1ccccc1 ZINC000217939211 GH For-Sale Unstable CES1 68 39 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCCCc1ccccc1 ZINC000217939211 GH For-Sale Unstable CES1D 45 35 CN1CCN(Cc2ccc(/C=C\C(=O)O)cc2F)CC1 ZINC000217939214 CD For-Sale Unstable GPR183 0 43 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1cccc([N+](=O)[O-])c1 ZINC000217939215 CI For-Sale Unstable TRPM8 25 43 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1cccc([N+](=O)[O-])c1 ZINC000217939215 CI For-Sale Unstable OSIGBA0132E09-OSIGBA0108L24.11 0 40 COc1ccc(C(=O)NCC[C@@H](O)c2cccn2C)cc1F ZINC000217939224 DE In-Stock Unstable DRD4 43 33 COc1ccc(C(=O)NCC[C@@H](O)c2cccn2C)cc1F ZINC000217939224 DE In-Stock Unstable COLA 60 35 COc1ccc(C(=O)NCC[C@@H](O)c2cccn2C)cc1F ZINC000217939224 DE In-Stock Unstable CPT1A 57 34 COc1ccc(C(=O)NCC[C@@H](O)c2cccn2C)cc1F ZINC000217939224 DE In-Stock Unstable CPT1B 45 33 COc1cccc(/C=C/NC(=O)N2CCCC2)c1 ZINC000217939227 BE For-Sale Unstable DRD4 44 34 COc1cccc(/C=C/NC(=O)N2CCCC2)c1 ZINC000217939227 BE For-Sale Unstable CYP1B1 20 41 COc1cccc(/C=C/NC(=O)N2CCCC2)c1 ZINC000217939227 BE For-Sale Unstable MTNR1A 38 43 COc1cccc(/C=C/NC(=O)N2CCCC2)c1 ZINC000217939227 BE For-Sale Unstable MTNR1B 46 43 COc1cccc(/C=C/NC(=O)N2CCCC2)c1 ZINC000217939227 BE For-Sale Unstable CYP1A1 19 41 COc1cccc(C(=O)N[C@@H]2CC(C)(C)Oc3cc(C)ccc32)c1 ZINC000217939281 EI In-Stock Unstable DRD4 47 40 COc1cccc(C(=O)N[C@@H]2CC(C)(C)Oc3cc(C)ccc32)c1 ZINC000217939281 EI In-Stock Unstable LGALS1 0 40 COc1cccc(C(=O)N[C@@H]2CC(C)(C)Oc3cc(C)ccc32)c1 ZINC000217939281 EI In-Stock Unstable KCNK3 35 40 CN1CCN(C)[C@@H](CC(=O)NCCc2ccccc2OC(F)(F)F)C1 ZINC000217939287 FD In-Stock Unstable SCN9A 0 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCCCc1ccccc1 ZINC000217939291 GH For-Sale Unstable FKBP1A 41 38 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCCCc1ccccc1 ZINC000217939291 GH For-Sale Unstable PREP 46 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCCCc1ccccc1 ZINC000217939291 GH For-Sale Unstable FAAH 71 42 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCCCc1ccccc1 ZINC000217939291 GH For-Sale Unstable CES1 68 39 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CCCCc1ccccc1 ZINC000217939291 GH For-Sale Unstable CES1D 45 35 Cc1nc(-c2ccccc2)sc1C(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217939292 GH In-Stock Unstable CHRNA4 37 48 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1cccc([N+](=O)[O-])c1 ZINC000217939300 CI For-Sale Unstable TRPM8 25 43 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1cccc([N+](=O)[O-])c1 ZINC000217939300 CI For-Sale Unstable OSIGBA0132E09-OSIGBA0108L24.11 0 40 C[C@@H](S)C(=O)NCc1ccccc1 ZINC000217939306 AD For-Sale Unstable CAPNS1 44 32 COc1cccc(/C=C/NC(=O)N2CCCCCC2)c1 ZINC000217939313 CG For-Sale Unstable DRD4 43 33 COc1cccc(/C=C/NC(=O)N2CCCCCC2)c1 ZINC000217939313 CG For-Sale Unstable MTNR1A 35 42 COc1cccc(/C=C/NC(=O)N2CCCCCC2)c1 ZINC000217939313 CG For-Sale Unstable MTNR1B 44 42 O=C(O)/C=C\c1ccccc1CN1CCc2sccc2C1 ZINC000217939314 CG For-Sale Unstable PTGER2 43 42 O=C(O)/C=C\c1ccccc1CN1CCc2sccc2C1 ZINC000217939314 CG For-Sale Unstable PTGER4 22 42 O=C(O)/C=C\c1ccccc1CN1CCc2sccc2C1 ZINC000217939314 CG For-Sale Unstable PTGER3 19 42 O=C(O)/C=C\c1ccccc1CN1CCc2sccc2C1 ZINC000217939314 CG For-Sale Unstable CYP2B6 15 57 COc1ccc(C(=O)NCC[C@H](O)c2cccn2C)cc1F ZINC000217939321 DE In-Stock Unstable DRD4 43 33 COc1ccc(C(=O)NCC[C@H](O)c2cccn2C)cc1F ZINC000217939321 DE In-Stock Unstable COLA 60 35 COc1ccc(C(=O)NCC[C@H](O)c2cccn2C)cc1F ZINC000217939321 DE In-Stock Unstable CPT1A 57 34 COc1ccc(C(=O)NCC[C@H](O)c2cccn2C)cc1F ZINC000217939321 DE In-Stock Unstable CPT1B 45 33 CCCCOc1ccc(/C=C2/CC(=O)NC2=O)cc1 ZINC000217939334 CE For-Sale Unstable PLA2G4B 66 33 CCCCOc1ccc(/C=C2/CC(=O)NC2=O)cc1 ZINC000217939334 CE For-Sale Unstable HPGD 88 44 C[C@@H](O)C1CCN(C(=O)NC2CCC2)CC1 ZINC000217939347 BD On-Demand Unstable EPHX2 17 45 COc1ccc(/C=C\C(=O)O)c(CS[C@@H](C)CCO)c1 ZINC000217939355 CF For-Sale Unstable PTGER2 27 43 COc1cccc(C(=O)N[C@H]2CC(C)(C)Oc3cc(C)ccc32)c1 ZINC000217939368 EI In-Stock Unstable DRD4 47 40 COc1cccc(C(=O)N[C@H]2CC(C)(C)Oc3cc(C)ccc32)c1 ZINC000217939368 EI In-Stock Unstable LGALS1 0 40 COc1cccc(C(=O)N[C@H]2CC(C)(C)Oc3cc(C)ccc32)c1 ZINC000217939368 EI In-Stock Unstable KCNK3 35 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCCCc1ccccc1 ZINC000217939371 GH For-Sale Unstable FKBP1A 41 38 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCCCc1ccccc1 ZINC000217939371 GH For-Sale Unstable PREP 46 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCCCc1ccccc1 ZINC000217939371 GH For-Sale Unstable FAAH 71 42 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCCCc1ccccc1 ZINC000217939371 GH For-Sale Unstable CES1 68 39 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCCCc1ccccc1 ZINC000217939371 GH For-Sale Unstable CES1D 45 35 C[C@H](S)C(=O)NCc1ccccc1 ZINC000217939385 AD For-Sale Unstable CAPNS1 44 32 O=C(O)c1ccc(N2CCC[C@@H]3CCCC[C@H]32)c(Cl)c1 ZINC000217939409 CI For-Sale Unstable NR3C2 26 43 COc1cccc(/C=C/NC(=O)NC[C@@H](C)O)c1 ZINC000217939426 CD For-Sale Unstable MTNR1A 65 49 COc1cccc(/C=C/NC(=O)NC[C@@H](C)O)c1 ZINC000217939426 CD For-Sale Unstable MTNR1B 62 49 C[C@H](O)C1CCN(C(=O)NC2CCC2)CC1 ZINC000217939429 BD On-Demand Unstable EPHX2 17 45 O=C(O)/C=C\c1ccc(CN2CCc3sccc3C2)cc1 ZINC000217939445 CG For-Sale Unstable SIGMAR1 25 42 O=C(O)/C=C\c1ccc(CN2CCc3sccc3C2)cc1 ZINC000217939445 CG For-Sale Unstable NOD2 40 33 COc1ccc(/C=C\C(=O)O)c(CS[C@H](C)CCO)c1 ZINC000217939452 CF For-Sale Unstable PTGER2 27 43 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCCCc1ccccc1 ZINC000217939457 GH For-Sale Unstable FKBP1A 41 38 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCCCc1ccccc1 ZINC000217939457 GH For-Sale Unstable PREP 46 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCCCc1ccccc1 ZINC000217939457 GH For-Sale Unstable FAAH 71 42 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCCCc1ccccc1 ZINC000217939457 GH For-Sale Unstable CES1 68 39 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CCCCc1ccccc1 ZINC000217939457 GH For-Sale Unstable CES1D 45 35 COc1cccc(C(=O)N[C@@H]2CC(C)(C)Oc3ccc(OC)cc32)c1 ZINC000217939481 EH In-Stock Unstable ABCC9 38 40 COc1cccc(C(=O)N[C@@H]2CC(C)(C)Oc3ccc(OC)cc32)c1 ZINC000217939481 EH In-Stock Unstable DRD4 46 35 COc1cccc(C(=O)N[C@@H]2CC(C)(C)Oc3ccc(OC)cc32)c1 ZINC000217939481 EH In-Stock Unstable CSNK1E 16 43 COc1cccc(C(=O)N[C@@H]2CC(C)(C)Oc3ccc(OC)cc32)c1 ZINC000217939481 EH In-Stock Unstable NAAA 15 45 COc1cccc(C(=O)N[C@@H]2CC(C)(C)Oc3ccc(OC)cc32)c1 ZINC000217939481 EH In-Stock Unstable LGALS1 0 41 O=C(O)c1ccc(N2CCC[C@H]3CCCC[C@H]32)c(Cl)c1 ZINC000217939492 CI For-Sale Unstable NR3C2 26 43 COc1cccc(/C=C/NC(=O)NC[C@H](C)O)c1 ZINC000217939501 CD For-Sale Unstable MTNR1A 65 49 COc1cccc(/C=C/NC(=O)NC[C@H](C)O)c1 ZINC000217939501 CD For-Sale Unstable MTNR1B 62 49 O=C(Cc1n[nH]c(=O)c2ccccc12)N1CCCC[C@H]1c1cccnc1 ZINC000217939527 EF In-Stock Unstable CHRNA2 39 40 O=C(Cc1n[nH]c(=O)c2ccccc12)N1CCCC[C@H]1c1cccnc1 ZINC000217939527 EF In-Stock Unstable COLA 119 42 O=C(Cc1n[nH]c(=O)c2ccccc12)N1CCCC[C@H]1c1cccnc1 ZINC000217939527 EF In-Stock Unstable CPT1A 106 42 O=C(Cc1n[nH]c(=O)c2ccccc12)N1CCCC[C@H]1c1cccnc1 ZINC000217939527 EF In-Stock Unstable PARP1 38 44 O=C(Cc1n[nH]c(=O)c2ccccc12)N1CCCC[C@H]1c1cccnc1 ZINC000217939527 EF In-Stock Unstable CRTY 0 40 O=C(O)/C=C\c1cccc(CN2CCc3sccc3C2)c1 ZINC000217939552 CG For-Sale Unstable SIGMAR1 23 41 O=C(O)/C=C\c1cccc(CN2CCc3sccc3C2)c1 ZINC000217939552 CG For-Sale Unstable AKR1C3 25 42 COc1cccc(C(=O)N[C@H]2CC(C)(C)Oc3ccc(OC)cc32)c1 ZINC000217939572 EH In-Stock Unstable ABCC9 38 40 COc1cccc(C(=O)N[C@H]2CC(C)(C)Oc3ccc(OC)cc32)c1 ZINC000217939572 EH In-Stock Unstable DRD4 46 35 COc1cccc(C(=O)N[C@H]2CC(C)(C)Oc3ccc(OC)cc32)c1 ZINC000217939572 EH In-Stock Unstable CSNK1E 16 43 COc1cccc(C(=O)N[C@H]2CC(C)(C)Oc3ccc(OC)cc32)c1 ZINC000217939572 EH In-Stock Unstable NAAA 15 45 COc1cccc(C(=O)N[C@H]2CC(C)(C)Oc3ccc(OC)cc32)c1 ZINC000217939572 EH In-Stock Unstable LGALS1 0 41 CCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217939610 BD For-Sale Unstable DRD4 42 32 CCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217939610 BD For-Sale Unstable CYP1B1 45 47 CCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217939610 BD For-Sale Unstable MTNR1A 73 46 CCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217939610 BD For-Sale Unstable MTNR1B 66 47 NC(=O)C1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217939657 CD For-Sale Unstable DRD2 17 43 NC(=O)C1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217939657 CD For-Sale Unstable DRD4 34 43 NC(=O)C1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217939657 CD For-Sale Unstable ACHE 38 42 NC(=O)C1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217939657 CD For-Sale Unstable DRD3 0 43 NC(=O)C1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217939657 CD For-Sale Unstable CHRM3 22 40 NC(=O)C1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217939657 CD For-Sale Unstable SIGMAR1 50 51 NC(=O)C1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217939657 CD For-Sale Unstable CCR3 17 42 COc1cccc(C(=O)N[C@@H]2CC(C)(C)Oc3cc(OC)ccc32)c1 ZINC000217939677 EH In-Stock Unstable DRD4 47 36 COc1cccc(C(=O)N[C@@H]2CC(C)(C)Oc3cc(OC)ccc32)c1 ZINC000217939677 EH In-Stock Unstable NAAA 19 46 COc1cccc(C(=O)N[C@@H]2CC(C)(C)Oc3cc(OC)ccc32)c1 ZINC000217939677 EH In-Stock Unstable LGALS1 0 42 COc1cccc(C(=O)N[C@@H]2CC(C)(C)Oc3cc(OC)ccc32)c1 ZINC000217939677 EH In-Stock Unstable LGALS9 0 42 COc1cccc(C(=O)N[C@@H]2CC(C)(C)Oc3cc(OC)ccc32)c1 ZINC000217939677 EH In-Stock Unstable BRPF1 0 40 C[C@@H](S)C(=O)Nc1ccc(F)cc1Cl ZINC000217939684 BF For-Sale Unstable PYGL 27 47 CCCCN(CCC)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217939715 CH For-Sale Unstable MTNR1A 43 44 CCCCN(CCC)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217939715 CH For-Sale Unstable MTNR1B 43 44 Cc1noc2nc(C(C)C)cc(C(=O)Nc3cc(C(F)(F)F)ccc3N3CCOCC3)c12 ZINC000217939727 IJ On-Demand Unstable TEK 22 40 CNC(=O)[C@@H]1CC[C@@H](CNC(=O)CCCN2Cc3ccccc3C2)CC1 ZINC000217939745 FE In-Stock Unstable HTR7 42 38 C[C@H]1C[C@H](C)CCN1c1ccc(C(F)(F)F)cc1C(=O)O ZINC000217939747 DI For-Sale Unstable LIPC 0 46 C[C@H]1C[C@H](C)CCN1c1ccc(C(F)(F)F)cc1C(=O)O ZINC000217939747 DI For-Sale Unstable LIPG 71 49 COc1cccc(C(=O)N[C@H]2CC(C)(C)Oc3cc(OC)ccc32)c1 ZINC000217939751 EH In-Stock Unstable DRD4 47 36 COc1cccc(C(=O)N[C@H]2CC(C)(C)Oc3cc(OC)ccc32)c1 ZINC000217939751 EH In-Stock Unstable NAAA 19 46 COc1cccc(C(=O)N[C@H]2CC(C)(C)Oc3cc(OC)ccc32)c1 ZINC000217939751 EH In-Stock Unstable LGALS1 0 42 COc1cccc(C(=O)N[C@H]2CC(C)(C)Oc3cc(OC)ccc32)c1 ZINC000217939751 EH In-Stock Unstable LGALS9 0 42 COc1cccc(C(=O)N[C@H]2CC(C)(C)Oc3cc(OC)ccc32)c1 ZINC000217939751 EH In-Stock Unstable BRPF1 0 40 C[C@H](S)C(=O)Nc1ccc(F)cc1Cl ZINC000217939757 BF For-Sale Unstable PYGL 27 47 CN(Cc1ccccc1/C=C\C(=O)O)C1CCCCC1 ZINC000217939778 CH For-Sale Unstable PTGER2 49 50 CN(Cc1ccccc1/C=C\C(=O)O)C1CCCCC1 ZINC000217939778 CH For-Sale Unstable PTGER4 23 50 CN(Cc1ccccc1/C=C\C(=O)O)C1CCCCC1 ZINC000217939778 CH For-Sale Unstable PTGER3 18 50 CN(Cc1ccccc1/C=C\C(=O)O)C1CCCCC1 ZINC000217939778 CH For-Sale Unstable AMY2 44 31 CN(Cc1ccccc1/C=C\C(=O)O)C1CCCCC1 ZINC000217939778 CH For-Sale Unstable PTGDR 0 48 O=C([C@H]1CC(=O)N(c2ccccc2)C1)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217939781 GD In-Stock Unstable CHRNA4 30 50 C[C@H]1CCN(c2ccc(C(F)(F)F)cc2C(=O)O)[C@@H](C)C1 ZINC000217939821 DI For-Sale Unstable LIPC 0 46 C[C@H]1CCN(c2ccc(C(F)(F)F)cc2C(=O)O)[C@@H](C)C1 ZINC000217939821 DI For-Sale Unstable LIPG 71 49 CCCCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217939835 CG For-Sale Unstable DRD4 41 31 CCCCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217939835 CG For-Sale Unstable HRH2 21 40 CCCCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217939835 CG For-Sale Unstable AHR 19 41 CCCCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217939835 CG For-Sale Unstable MTNR1A 99 50 CCCCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217939835 CG For-Sale Unstable MTNR1B 92 50 CCCCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217939835 CG For-Sale Unstable PA2A1_NAJMO 0 44 CCCCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217939835 CG For-Sale Unstable ACAT 0 48 CC[C@@H](NC(=O)c1cccc(OC)c1)c1ccc(C)c(C)c1 ZINC000217939854 CI In-Stock Unstable DRD4 53 42 CC[C@@H](NC(=O)c1cccc(OC)c1)c1ccc(C)c(C)c1 ZINC000217939854 CI In-Stock Unstable KCNA5 0 45 CC[C@@H](NC(=O)c1cccc(OC)c1)c1ccc(C)c(C)c1 ZINC000217939854 CI In-Stock Unstable PTGER3 40 39 CC[C@@H](NC(=O)c1cccc(OC)c1)c1ccc(C)c(C)c1 ZINC000217939854 CI In-Stock Unstable CTSK 15 47 CC[C@@H](NC(=O)c1cccc(OC)c1)c1ccc(C)c(C)c1 ZINC000217939854 CI In-Stock Unstable CTSL 28 42 CC[C@@H](NC(=O)c1cccc(OC)c1)c1ccc(C)c(C)c1 ZINC000217939854 CI In-Stock Unstable MTNR1B 38 40 CC[C@@H](NC(=O)c1cccc(OC)c1)c1ccc(C)c(C)c1 ZINC000217939854 CI In-Stock Unstable CTSS 21 42 CC[C@@H](NC(=O)c1cccc(OC)c1)c1ccc(C)c(C)c1 ZINC000217939854 CI In-Stock Unstable UTS2 67 46 CC[C@@H](NC(=O)c1cccc(OC)c1)c1ccc(C)c(C)c1 ZINC000217939854 CI In-Stock Unstable BRPF1 0 45 O=C([C@@H]1CC(=O)N(c2ccccc2)C1)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217939859 GD In-Stock Unstable CHRNA4 30 50 C[C@@H](S)C(=O)Nc1ccc2c(c1)OCCO2 ZINC000217939866 BD For-Sale Unstable TRPV1 0 54 CN(Cc1ccc(/C=C\C(=O)O)cc1)C1CCCCC1 ZINC000217939888 CH For-Sale Unstable NR1H4 32 44 CC[C@H](NC(=O)c1cccc(OC)c1)c1ccc(C)c(C)c1 ZINC000217939924 CI In-Stock Unstable DRD4 53 42 CC[C@H](NC(=O)c1cccc(OC)c1)c1ccc(C)c(C)c1 ZINC000217939924 CI In-Stock Unstable KCNA5 0 45 CC[C@H](NC(=O)c1cccc(OC)c1)c1ccc(C)c(C)c1 ZINC000217939924 CI In-Stock Unstable PTGER3 40 39 CC[C@H](NC(=O)c1cccc(OC)c1)c1ccc(C)c(C)c1 ZINC000217939924 CI In-Stock Unstable CTSK 15 47 CC[C@H](NC(=O)c1cccc(OC)c1)c1ccc(C)c(C)c1 ZINC000217939924 CI In-Stock Unstable CTSL 32 42 CC[C@H](NC(=O)c1cccc(OC)c1)c1ccc(C)c(C)c1 ZINC000217939924 CI In-Stock Unstable MTNR1A 45 42 CC[C@H](NC(=O)c1cccc(OC)c1)c1ccc(C)c(C)c1 ZINC000217939924 CI In-Stock Unstable MTNR1B 45 42 CC[C@H](NC(=O)c1cccc(OC)c1)c1ccc(C)c(C)c1 ZINC000217939924 CI In-Stock Unstable CTSS 24 47 CC[C@H](NC(=O)c1cccc(OC)c1)c1ccc(C)c(C)c1 ZINC000217939924 CI In-Stock Unstable UTS2 73 46 CC[C@H](NC(=O)c1cccc(OC)c1)c1ccc(C)c(C)c1 ZINC000217939924 CI In-Stock Unstable KCNK3 38 46 CC[C@H](NC(=O)c1cccc(OC)c1)c1ccc(C)c(C)c1 ZINC000217939924 CI In-Stock Unstable BRPF1 0 45 Cc1cc(N2CCCN(C(=O)Cn3nnnc3N)CC2)ccn1 ZINC000217939933 DB In-Stock Unstable CCR1 41 41 COc1cccc(/C=C/NC(=O)Nc2ccccc2)c1 ZINC000217939936 CG For-Sale Unstable LPL 44 35 COc1cccc(/C=C/NC(=O)Nc2ccccc2)c1 ZINC000217939936 CG For-Sale Unstable CYP1B1 35 42 COc1cccc(/C=C/NC(=O)Nc2ccccc2)c1 ZINC000217939936 CG For-Sale Unstable MTNR1A 43 53 COc1cccc(/C=C/NC(=O)Nc2ccccc2)c1 ZINC000217939936 CG For-Sale Unstable MTNR1B 46 53 COc1cccc(/C=C/NC(=O)Nc2ccccc2)c1 ZINC000217939936 CG For-Sale Unstable CYP1A1 23 42 COc1cccc(/C=C/NC(=O)Nc2ccccc2)c1 ZINC000217939936 CG For-Sale Unstable TAAR1 31 40 COc1cccc(/C=C/NC(=O)Nc2ccccc2)c1 ZINC000217939936 CG For-Sale Unstable AKR1C3 35 47 COc1cccc(/C=C/NC(=O)Nc2ccccc2)c1 ZINC000217939936 CG For-Sale Unstable AKR1C2 54 39 COc1cccc(/C=C/NC(=O)Nc2ccccc2)c1 ZINC000217939936 CG For-Sale Unstable P95276_MYCTO 0 41 COc1cccc(/C=C/NC(=O)Nc2ccccc2)c1 ZINC000217939936 CG For-Sale Unstable KCNK3 43 48 C[C@H](S)C(=O)Nc1ccc2c(c1)OCCO2 ZINC000217939944 BD For-Sale Unstable TRPV1 0 54 O=C(OC(=O)c1ccc(OCCCO)cc1)c1ccccc1 ZINC000217939954 DE For-Sale Unstable SRD5A2 32 44 O=C(OC(=O)c1ccc(OCCCO)cc1)c1ccccc1 ZINC000217939954 DE For-Sale Unstable PPARG 15 44 O=C(OC(=O)c1ccc(OCCCO)cc1)c1ccccc1 ZINC000217939954 DE For-Sale Unstable PPARA 17 44 O=C(OC(=O)c1ccc(OCCCO)cc1)c1ccccc1 ZINC000217939954 DE For-Sale Unstable LTA4H 40 39 O=C(OC(=O)c1ccc(OCCCO)cc1)c1ccccc1 ZINC000217939954 DE For-Sale Unstable CYSLTR2 47 33 O=C(OC(=O)c1ccc(OCCCO)cc1)c1ccccc1 ZINC000217939954 DE For-Sale Unstable PLA2G4B 91 47 O=C(OC(=O)c1ccc(OCCCO)cc1)c1ccccc1 ZINC000217939954 DE For-Sale Unstable ESRRG 53 43 O=C(OC(=O)c1ccc(OCCCO)cc1)c1ccccc1 ZINC000217939954 DE For-Sale Unstable ACR 40 46 O=C(OC(=O)c1ccc(OCCCO)cc1)c1ccccc1 ZINC000217939954 DE For-Sale Unstable CYP3A5 21 40 O=C(OC(=O)c1ccc(OCCCO)cc1)c1ccccc1 ZINC000217939954 DE For-Sale Unstable PSMB1 27 40 CC(C)Cn1nc(CC(=O)N2CCCC[C@H]2c2cccnc2)c2ccccc2c1=O ZINC000217939961 HH In-Stock Unstable COLA 76 38 CC(C)Cn1nc(CC(=O)N2CCCC[C@H]2c2cccnc2)c2ccccc2c1=O ZINC000217939961 HH In-Stock Unstable CPT1A 73 38 CC(C)Cn1nc(CC(=O)N2CCCC[C@H]2c2cccnc2)c2ccccc2c1=O ZINC000217939961 HH In-Stock Unstable Q7YY07_CRYPV 80 33 CCC[C@@H](C)N(C)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217939987 CG For-Sale Unstable TUBB1 47 39 CCC[C@@H](C)N(C)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217939987 CG For-Sale Unstable AKR1C3 30 41 CC[C@@H](NC(=O)c1cccc(OC)c1)c1ccc(C)cc1C ZINC000217940018 CI In-Stock Unstable DRD4 50 43 CC[C@@H](NC(=O)c1cccc(OC)c1)c1ccc(C)cc1C ZINC000217940018 CI In-Stock Unstable CTSK 16 45 CC[C@@H](NC(=O)c1cccc(OC)c1)c1ccc(C)cc1C ZINC000217940018 CI In-Stock Unstable CTSL 35 46 CC[C@@H](NC(=O)c1cccc(OC)c1)c1ccc(C)cc1C ZINC000217940018 CI In-Stock Unstable MTNR1A 31 40 CC[C@@H](NC(=O)c1cccc(OC)c1)c1ccc(C)cc1C ZINC000217940018 CI In-Stock Unstable MTNR1B 33 40 CC[C@@H](NC(=O)c1cccc(OC)c1)c1ccc(C)cc1C ZINC000217940018 CI In-Stock Unstable CTSS 27 46 CC[C@@H](NC(=O)c1cccc(OC)c1)c1ccc(C)cc1C ZINC000217940018 CI In-Stock Unstable CTSV 32 41 CC[C@@H](NC(=O)c1cccc(OC)c1)c1ccc(C)cc1C ZINC000217940018 CI In-Stock Unstable UTS2 56 40 CC[C@@H](NC(=O)c1cccc(OC)c1)c1ccc(C)cc1C ZINC000217940018 CI In-Stock Unstable KCNK3 68 50 CC[C@@H](NC(=O)c1cccc(OC)c1)c1ccc(C)cc1C ZINC000217940018 CI In-Stock Unstable KCNK9 55 37 CC[C@@H](NC(=O)c1cccc(OC)c1)c1ccc(C)cc1C ZINC000217940018 CI In-Stock Unstable BRPF1 0 43 C[C@@H](S)C(=O)Nc1ccccc1-c1ccccc1 ZINC000217940031 CH For-Sale Unstable ACE 25 45 C[C@@H](S)C(=O)Nc1ccccc1-c1ccccc1 ZINC000217940031 CH For-Sale Unstable MME 50 45 C[C@@H](S)C(=O)Nc1ccccc1-c1ccccc1 ZINC000217940031 CH For-Sale Unstable ACE2 69 45 CCOC(=O)[C@@H]1CCCN(C(=O)N/C=C/c2cccc(OC)c2)C1 ZINC000217940036 EF For-Sale Unstable FDFT1 28 41 CCC[C@H](C)N(C)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217940075 CG For-Sale Unstable TUBB1 47 39 CCC[C@H](C)N(C)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217940075 CG For-Sale Unstable AKR1C3 30 41 CC[C@H](NC(=O)c1cccc(OC)c1)c1ccc(C)cc1C ZINC000217940100 CI In-Stock Unstable DRD4 50 43 CC[C@H](NC(=O)c1cccc(OC)c1)c1ccc(C)cc1C ZINC000217940100 CI In-Stock Unstable CTSK 16 45 CC[C@H](NC(=O)c1cccc(OC)c1)c1ccc(C)cc1C ZINC000217940100 CI In-Stock Unstable CTSL 35 46 CC[C@H](NC(=O)c1cccc(OC)c1)c1ccc(C)cc1C ZINC000217940100 CI In-Stock Unstable MTNR1A 31 40 CC[C@H](NC(=O)c1cccc(OC)c1)c1ccc(C)cc1C ZINC000217940100 CI In-Stock Unstable MTNR1B 33 40 CC[C@H](NC(=O)c1cccc(OC)c1)c1ccc(C)cc1C ZINC000217940100 CI In-Stock Unstable CTSS 27 46 CC[C@H](NC(=O)c1cccc(OC)c1)c1ccc(C)cc1C ZINC000217940100 CI In-Stock Unstable CTSV 32 41 CC[C@H](NC(=O)c1cccc(OC)c1)c1ccc(C)cc1C ZINC000217940100 CI In-Stock Unstable UTS2 56 40 CC[C@H](NC(=O)c1cccc(OC)c1)c1ccc(C)cc1C ZINC000217940100 CI In-Stock Unstable KCNK3 68 50 CC[C@H](NC(=O)c1cccc(OC)c1)c1ccc(C)cc1C ZINC000217940100 CI In-Stock Unstable KCNK9 55 37 CC[C@H](NC(=O)c1cccc(OC)c1)c1ccc(C)cc1C ZINC000217940100 CI In-Stock Unstable BRPF1 0 43 C[C@H](S)C(=O)Nc1ccccc1-c1ccccc1 ZINC000217940103 CH For-Sale Unstable ACE 25 45 C[C@H](S)C(=O)Nc1ccccc1-c1ccccc1 ZINC000217940103 CH For-Sale Unstable MME 50 45 C[C@H](S)C(=O)Nc1ccccc1-c1ccccc1 ZINC000217940103 CH For-Sale Unstable ACE2 69 45 CCOC(=O)[C@H]1CCCN(C(=O)N/C=C/c2cccc(OC)c2)C1 ZINC000217940106 EF For-Sale Unstable FDFT1 28 41 CCC[C@@H](C)N(C)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217940173 CG For-Sale Unstable PTGER2 24 41 CCC[C@@H](C)N(C)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217940173 CG For-Sale Unstable PTGER4 0 41 CC[C@@H](NC(=O)c1cccc(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217940208 EH In-Stock Unstable DRD4 50 38 CC[C@@H](NC(=O)c1cccc(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217940208 EH In-Stock Unstable KCNA5 0 42 CC[C@@H](NC(=O)c1cccc(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217940208 EH In-Stock Unstable PTGER3 19 42 CC[C@@H](NC(=O)c1cccc(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217940208 EH In-Stock Unstable MTNR1B 44 40 CC[C@@H](NC(=O)c1cccc(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217940208 EH In-Stock Unstable UTS2 70 47 CC[C@@H](NC(=O)c1cccc(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217940208 EH In-Stock Unstable BRPF1 0 40 COc1cccc(/C=C/NC(=O)Nc2ccc(CC(=O)O)cc2)c1 ZINC000217940213 EG For-Sale Unstable MTNR1A 44 46 COc1cccc(/C=C/NC(=O)Nc2ccc(CC(=O)O)cc2)c1 ZINC000217940213 EG For-Sale Unstable MTNR1B 47 46 COc1cccc(/C=C/NC(=O)Nc2ccc(CC(=O)O)cc2)c1 ZINC000217940213 EG For-Sale Unstable AKR1C2 40 32 C[C@@H](S)C(=O)NCc1ccc2c(c1)OCO2 ZINC000217940243 BD For-Sale Unstable PDE5A 0 44 C[C@@H](S)C(=O)NCc1ccc2c(c1)OCO2 ZINC000217940243 BD For-Sale Unstable EDNRB 41 39 C[C@@H](S)C(=O)NCc1ccc2c(c1)OCO2 ZINC000217940243 BD For-Sale Unstable BMP1 53 39 C[C@@H](S)C(=O)NCc1ccc2c(c1)OCO2 ZINC000217940243 BD For-Sale Unstable NOS2 99 40 C[C@@H](S)C(=O)NCc1ccc2c(c1)OCO2 ZINC000217940243 BD For-Sale Unstable SSTR3 79 31 CCC[C@H](C)N(C)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217940253 CG For-Sale Unstable PTGER2 24 41 CCC[C@H](C)N(C)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217940253 CG For-Sale Unstable PTGER4 0 41 CCCCCCCCOc1ccc([C@H](CC(=O)OC)C2=C(O)C(=O)C([C@H](CC(=O)OC)c3ccc(OCCCCCCCC)cc3)=C(O)C2=O)cc1 ZINC000217940254 KK In-Stock Unstable THRA 43 39 CCCCCCCCOc1ccc([C@H](CC(=O)OC)C2=C(O)C(=O)C([C@H](CC(=O)OC)c3ccc(OCCCCCCCC)cc3)=C(O)C2=O)cc1 ZINC000217940254 KK In-Stock Unstable KCNQ1 0 40 CCCCCCCCOc1ccc([C@H](CC(=O)OC)C2=C(O)C(=O)C([C@H](CC(=O)OC)c3ccc(OCCCCCCCC)cc3)=C(O)C2=O)cc1 ZINC000217940254 KK In-Stock Unstable PLA2G4B 104 43 CCCCCCCCOc1ccc([C@H](CC(=O)OC)C2=C(O)C(=O)C([C@H](CC(=O)OC)c3ccc(OCCCCCCCC)cc3)=C(O)C2=O)cc1 ZINC000217940254 KK In-Stock Unstable FAAH 23 43 CCOC(=O)c1cnn(-c2ccc(Cl)c(Cl)c2)c1O ZINC000217940272 DG For-Sale Unstable HPD 39 41 CCOC(=O)c1cnn(-c2ccc(Cl)c(Cl)c2)c1O ZINC000217940272 DG For-Sale Unstable MURB 0 40 CCOC(=O)c1cnn(-c2ccc(Cl)c(Cl)c2)c1O ZINC000217940272 DG For-Sale Unstable RPA1 63 38 CCOC(=O)c1cnn(-c2ccc(Cl)c(Cl)c2)c1O ZINC000217940272 DG For-Sale Unstable Q9FYV8_MAIZE 31 46 CC[C@H](NC(=O)c1cccc(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217940285 EH In-Stock Unstable DRD4 50 38 CC[C@H](NC(=O)c1cccc(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217940285 EH In-Stock Unstable KCNA5 0 42 CC[C@H](NC(=O)c1cccc(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217940285 EH In-Stock Unstable PTGER3 19 42 CC[C@H](NC(=O)c1cccc(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217940285 EH In-Stock Unstable MTNR1B 44 40 CC[C@H](NC(=O)c1cccc(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217940285 EH In-Stock Unstable UTS2 70 47 CC[C@H](NC(=O)c1cccc(OC)c1)c1ccc(OC)c(OC)c1 ZINC000217940285 EH In-Stock Unstable BRPF1 0 40 C[C@H](S)C(=O)NCc1ccc2c(c1)OCO2 ZINC000217940326 BD For-Sale Unstable PDE5A 0 44 C[C@H](S)C(=O)NCc1ccc2c(c1)OCO2 ZINC000217940326 BD For-Sale Unstable EDNRB 41 39 C[C@H](S)C(=O)NCc1ccc2c(c1)OCO2 ZINC000217940326 BD For-Sale Unstable BMP1 53 39 C[C@H](S)C(=O)NCc1ccc2c(c1)OCO2 ZINC000217940326 BD For-Sale Unstable NOS2 99 40 C[C@H](S)C(=O)NCc1ccc2c(c1)OCO2 ZINC000217940326 BD For-Sale Unstable SSTR3 79 31 COc1cccc(/C=C/NC(=O)NCc2ccc(C(=O)O)cc2)c1 ZINC000217940331 EF For-Sale Unstable DRD4 42 32 COc1cccc(/C=C/NC(=O)NCc2ccc(C(=O)O)cc2)c1 ZINC000217940331 EF For-Sale Unstable MTNR1A 40 42 COc1cccc(/C=C/NC(=O)NCc2ccc(C(=O)O)cc2)c1 ZINC000217940331 EF For-Sale Unstable MTNR1B 38 42 COc1cccc(/C=C/NC(=O)NCc2ccc(C(=O)O)cc2)c1 ZINC000217940331 EF For-Sale Unstable PDS 42 32 CCCCCCCCOc1ccc([C@@H](CC(=O)OC)C2=C(O)C(=O)C([C@H](CC(=O)OC)c3ccc(OCCCCCCCC)cc3)=C(O)C2=O)cc1 ZINC000217940340 KK In-Stock Unstable THRA 43 39 CCCCCCCCOc1ccc([C@@H](CC(=O)OC)C2=C(O)C(=O)C([C@H](CC(=O)OC)c3ccc(OCCCCCCCC)cc3)=C(O)C2=O)cc1 ZINC000217940340 KK In-Stock Unstable KCNQ1 0 40 CCCCCCCCOc1ccc([C@@H](CC(=O)OC)C2=C(O)C(=O)C([C@H](CC(=O)OC)c3ccc(OCCCCCCCC)cc3)=C(O)C2=O)cc1 ZINC000217940340 KK In-Stock Unstable PLA2G4B 104 43 CCCCCCCCOc1ccc([C@@H](CC(=O)OC)C2=C(O)C(=O)C([C@H](CC(=O)OC)c3ccc(OCCCCCCCC)cc3)=C(O)C2=O)cc1 ZINC000217940340 KK In-Stock Unstable FAAH 23 43 Cn1cccc1[C@H](O)CCNC(=O)c1ccc(C(F)(F)F)nc1 ZINC000217940342 EE In-Stock Unstable EPHX2 25 48 CCC[C@@H](NC(=O)NCc1ccc(F)cc1)C(=O)N1CCN(c2ccc(O)cc2)CC1 ZINC000217940367 IF On-Demand Unstable P2RY12 46 33 CC(C)CN(Cc1cccc(/C=C\C(=O)O)c1)CC(C)C ZINC000217940370 CH For-Sale Unstable PTGER2 23 41 CC(C)CN(Cc1cccc(/C=C\C(=O)O)c1)CC(C)C ZINC000217940370 CH For-Sale Unstable NR1H4 39 40 CC(C)CN(Cc1cccc(/C=C\C(=O)O)c1)CC(C)C ZINC000217940370 CH For-Sale Unstable AKR1C3 33 49 CC[C@@H](NC(=O)c1cccc(OC)c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217940396 EF In-Stock Unstable DRD4 47 36 CC[C@@H](NC(=O)c1cccc(OC)c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217940396 EF In-Stock Unstable PTGS2 19 40 CC[C@@H](NC(=O)c1cccc(OC)c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217940396 EF In-Stock Unstable KCNA5 0 50 CC[C@@H](NC(=O)c1cccc(OC)c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217940396 EF In-Stock Unstable MMP13 16 43 CC[C@@H](NC(=O)c1cccc(OC)c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217940396 EF In-Stock Unstable UTS2 65 44 Cn1cccc1[C@@H](O)CCNC(=O)c1ccc(C(F)(F)F)nc1 ZINC000217940427 EE In-Stock Unstable EPHX2 25 48 CCCCCCCCOc1ccc([C@H](CC(=O)OC)C2=C(O)C(=O)C([C@@H](CC(=O)OC)c3ccc(OCCCCCCCC)cc3)=C(O)C2=O)cc1 ZINC000217940429 KK In-Stock Unstable THRA 43 39 CCCCCCCCOc1ccc([C@H](CC(=O)OC)C2=C(O)C(=O)C([C@@H](CC(=O)OC)c3ccc(OCCCCCCCC)cc3)=C(O)C2=O)cc1 ZINC000217940429 KK In-Stock Unstable KCNQ1 0 40 CCCCCCCCOc1ccc([C@H](CC(=O)OC)C2=C(O)C(=O)C([C@@H](CC(=O)OC)c3ccc(OCCCCCCCC)cc3)=C(O)C2=O)cc1 ZINC000217940429 KK In-Stock Unstable PLA2G4B 104 43 CCCCCCCCOc1ccc([C@H](CC(=O)OC)C2=C(O)C(=O)C([C@@H](CC(=O)OC)c3ccc(OCCCCCCCC)cc3)=C(O)C2=O)cc1 ZINC000217940429 KK In-Stock Unstable FAAH 23 43 COc1cccc(/C=C/NC(=O)Nc2c(F)cccc2F)c1 ZINC000217940434 DH For-Sale Unstable DHODH 16 40 COc1cccc(/C=C/NC(=O)Nc2c(F)cccc2F)c1 ZINC000217940434 DH For-Sale Unstable CYP1B1 15 43 COc1cccc(/C=C/NC(=O)Nc2c(F)cccc2F)c1 ZINC000217940434 DH For-Sale Unstable AHR 19 42 COc1cccc(/C=C/NC(=O)Nc2c(F)cccc2F)c1 ZINC000217940434 DH For-Sale Unstable MTNR1A 28 42 COc1cccc(/C=C/NC(=O)Nc2c(F)cccc2F)c1 ZINC000217940434 DH For-Sale Unstable MTNR1B 31 42 COc1cccc(/C=C/NC(=O)Nc2c(F)cccc2F)c1 ZINC000217940434 DH For-Sale Unstable TAAR1 18 41 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1ccccc1[N+](=O)[O-] ZINC000217940437 CI For-Sale Unstable SERPINE1 42 44 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1ccccc1[N+](=O)[O-] ZINC000217940437 CI For-Sale Unstable TRPM8 17 49 CCC[C@H](NC(=O)NCc1ccc(F)cc1)C(=O)N1CCN(c2ccc(O)cc2)CC1 ZINC000217940443 IF On-Demand Unstable P2RY12 46 33 CN(Cc1ccccc1/C=C\C(=O)O)C[C@@H]1CCCCO1 ZINC000217940477 CF For-Sale Unstable OXTR 26 41 CN(Cc1ccccc1/C=C\C(=O)O)C[C@@H]1CCCCO1 ZINC000217940477 CF For-Sale Unstable PTGER2 34 40 CN(Cc1ccccc1/C=C\C(=O)O)C[C@@H]1CCCCO1 ZINC000217940477 CF For-Sale Unstable PTGER4 0 40 CC[C@H](NC(=O)c1cccc(OC)c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217940482 EF In-Stock Unstable DRD4 47 36 CC[C@H](NC(=O)c1cccc(OC)c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217940482 EF In-Stock Unstable PTGS2 19 40 CC[C@H](NC(=O)c1cccc(OC)c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217940482 EF In-Stock Unstable KCNA5 0 50 CC[C@H](NC(=O)c1cccc(OC)c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217940482 EF In-Stock Unstable MMP13 16 43 CC[C@H](NC(=O)c1cccc(OC)c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217940482 EF In-Stock Unstable UTS2 65 44 C[C@@H](CC(=O)O)c1cc(Cl)ccc1C(F)F ZINC000217940516 BH For-Sale Unstable OXER1 40 34 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1ccccc1[N+](=O)[O-] ZINC000217940518 CI For-Sale Unstable SERPINE1 42 44 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1ccccc1[N+](=O)[O-] ZINC000217940518 CI For-Sale Unstable TRPM8 17 49 CCOC(=O)c1cnn(-c2ccccc2F)c1O ZINC000217940528 CD For-Sale Unstable HPD 23 41 CCN(CC)CCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217940534 CE For-Sale Unstable DRD4 42 32 CCN(CC)CCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217940534 CE For-Sale Unstable MTNR1A 75 44 CCN(CC)CCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217940534 CE For-Sale Unstable MTNR1B 67 44 COC(=O)C[C@@H](C1=C(O)C(=O)C([C@H](CC(=O)OC)c2cccnc2)=C(O)C1=O)c1cccnc1 ZINC000217940543 JE In-Stock Unstable TBXAS1 0 47 COC(=O)C[C@@H](C1=C(O)C(=O)C([C@H](CC(=O)OC)c2cccnc2)=C(O)C1=O)c1cccnc1 ZINC000217940543 JE In-Stock Unstable KCNA5 29 56 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1ccccc1[N+](=O)[O-] ZINC000217940577 CI For-Sale Unstable SERPINE1 42 44 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1ccccc1[N+](=O)[O-] ZINC000217940577 CI For-Sale Unstable TRPM8 17 49 C[C@H](CC(=O)O)c1cc(Cl)ccc1C(F)F ZINC000217940601 BH For-Sale Unstable OXER1 40 34 COC(=O)C[C@H](C1=C(O)C(=O)C([C@H](CC(=O)OC)c2cccnc2)=C(O)C1=O)c1cccnc1 ZINC000217940613 JE In-Stock Unstable TBXAS1 25 47 COC(=O)C[C@H](C1=C(O)C(=O)C([C@H](CC(=O)OC)c2cccnc2)=C(O)C1=O)c1cccnc1 ZINC000217940613 JE In-Stock Unstable KCNA5 29 56 COc1cccc(C(=O)NCc2nc(-c3ccc(OC)cc3OC)no2)c1 ZINC000217940623 FF In-Stock Unstable DRD4 50 38 COc1cccc(C(=O)NCc2nc(-c3ccc(OC)cc3OC)no2)c1 ZINC000217940623 FF In-Stock Unstable GRIN2B 25 41 COc1cccc(C(=O)NCc2nc(-c3ccc(OC)cc3OC)no2)c1 ZINC000217940623 FF In-Stock Unstable CYP1B1 15 40 COc1cccc(C(=O)NCc2nc(-c3ccc(OC)cc3OC)no2)c1 ZINC000217940623 FF In-Stock Unstable NQO2 20 41 COc1cccc(C(=O)NCc2nc(-c3ccc(OC)cc3OC)no2)c1 ZINC000217940623 FF In-Stock Unstable HRH3 15 43 COc1cccc(C(=O)NCc2nc(-c3ccc(OC)cc3OC)no2)c1 ZINC000217940623 FF In-Stock Unstable RAF1 19 40 COc1cccc(C(=O)NCc2nc(-c3ccc(OC)cc3OC)no2)c1 ZINC000217940623 FF In-Stock Unstable MT-ND1 16 41 COc1cccc(C(=O)NCc2nc(-c3ccc(OC)cc3OC)no2)c1 ZINC000217940623 FF In-Stock Unstable Q8MMZ8_EIMTE 16 40 COc1cccc(C(=O)NCc2nc(-c3ccc(OC)cc3OC)no2)c1 ZINC000217940623 FF In-Stock Unstable KCNK3 19 42 COc1ccc(/C=C\C(=O)O)cc1CS[C@@H](C)CCO ZINC000217940626 CF For-Sale Unstable AKR1C3 39 41 CCc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217940645 CI For-Sale Unstable MTNR1A 40 48 CCc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217940645 CI For-Sale Unstable MTNR1B 44 48 CCc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217940645 CI For-Sale Unstable ROCK2 19 43 CCc1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217940645 CI For-Sale Unstable ACR 28 42 O=C(O)c1cnn(-c2ccc([N+](=O)[O-])cc2)c1O ZINC000217940658 BD For-Sale Bother AKR1C2 15 43 C=C1CCC(CNC(=O)OCc2ccccc2)CC1 ZINC000217940670 CH For-Sale Unstable GRIN2B 38 44 C=C1CCC(CNC(=O)OCc2ccccc2)CC1 ZINC000217940670 CH For-Sale Unstable CTSB 45 43 C=C1CCC(CNC(=O)OCc2ccccc2)CC1 ZINC000217940670 CH For-Sale Unstable CTSK 34 43 C=C1CCC(CNC(=O)OCc2ccccc2)CC1 ZINC000217940670 CH For-Sale Unstable CTSL 39 43 C=C1CCC(CNC(=O)OCc2ccccc2)CC1 ZINC000217940670 CH For-Sale Unstable PREP 22 45 C=C1CCC(CNC(=O)OCc2ccccc2)CC1 ZINC000217940670 CH For-Sale Unstable CAPNS1 60 35 C=C1CCC(CNC(=O)OCc2ccccc2)CC1 ZINC000217940670 CH For-Sale Unstable CTSS 22 42 C=C1CCC(CNC(=O)OCc2ccccc2)CC1 ZINC000217940670 CH For-Sale Unstable CAPN1 60 44 C=C1CCC(CNC(=O)OCc2ccccc2)CC1 ZINC000217940670 CH For-Sale Unstable CASP1 22 41 C=C1CCC(CNC(=O)OCc2ccccc2)CC1 ZINC000217940670 CH For-Sale Unstable CAPN2 103 44 C=C1CCC(CNC(=O)OCc2ccccc2)CC1 ZINC000217940670 CH For-Sale Unstable TGM2 34 51 C=C1CCC(CNC(=O)OCc2ccccc2)CC1 ZINC000217940670 CH For-Sale Unstable NPR 67 40 C=C1CCC(CNC(=O)OCc2ccccc2)CC1 ZINC000217940670 CH For-Sale Unstable F13A1 27 51 C=C1CCC(CNC(=O)OCc2ccccc2)CC1 ZINC000217940670 CH For-Sale Unstable NAAA 38 45 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1ccccc1[N+](=O)[O-] ZINC000217940673 CI For-Sale Unstable SERPINE1 42 44 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1ccccc1[N+](=O)[O-] ZINC000217940673 CI For-Sale Unstable TRPM8 17 49 Cc1noc2nc(C(C)C)cc(C(=O)Nc3cccc(S(=O)(=O)N(C)c4ccccc4)c3)c12 ZINC000217940681 JJ On-Demand Unstable KCNK3 41 35 COC(=O)C[C@H](C1=C(O)C(=O)C([C@@H](CC(=O)OC)c2cccnc2)=C(O)C1=O)c1cccnc1 ZINC000217940691 JE In-Stock Unstable TBXAS1 25 47 COC(=O)C[C@H](C1=C(O)C(=O)C([C@@H](CC(=O)OC)c2cccnc2)=C(O)C1=O)c1cccnc1 ZINC000217940691 JE In-Stock Unstable KCNA5 29 56 COc1ccc(/C=C\C(=O)O)cc1CS[C@H](C)CCO ZINC000217940718 CF For-Sale Unstable AKR1C3 39 41 CCCN(CCO)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217940719 CD For-Sale Unstable PLA2G4B 65 33 CCc1ccc(/C=C2/CC(=O)NC2=O)cc1 ZINC000217940721 BD For-Sale Unstable HPGD 46 38 COc1cccc(C(=O)N(C)Cc2nc(-c3cccc(OC)c3)no2)c1 ZINC000217940730 FG In-Stock Unstable DRD4 41 31 COc1cccc(C(=O)N(C)Cc2nc(-c3cccc(OC)c3)no2)c1 ZINC000217940730 FG In-Stock Unstable HSD17B2 34 53 Cn1cccc1[C@H](O)CCNS(=O)(=O)c1cccnc1 ZINC000217940740 CC In-Stock Unstable ADRB3 43 34 Cn1cccc1[C@H](O)CCNS(=O)(=O)c1cccnc1 ZINC000217940740 CC In-Stock Unstable TBXAS1 42 39 O=C(c1cccnc1)N1CCC(N2CCn3nc(CO)cc3C2)CC1 ZINC000217940777 EC In-Stock Unstable L3MBTL1 0 43 O=C(c1cccnc1)N1CCC(N2CCn3nc(CO)cc3C2)CC1 ZINC000217940777 EC In-Stock Unstable L3MBTL3 69 41 CCOC(=O)c1cnn(-c2ccccc2[N+](=O)[O-])c1O ZINC000217940782 CD For-Sale Unstable CACNA1D 34 41 COC(=O)C[C@H](c1c(O)cc(C)oc1=O)c1coc2ccccc2c1=O ZINC000217940798 FE In-Stock Unstable ALDH2 51 32 Cn1cccc1[C@@H](O)CCNS(=O)(=O)c1cccnc1 ZINC000217940806 CC In-Stock Unstable ADRB3 43 34 Cn1cccc1[C@@H](O)CCNS(=O)(=O)c1cccnc1 ZINC000217940806 CC In-Stock Unstable TBXAS1 42 39 O=C1C/C(=C/c2ccc(OC(F)(F)F)cc2)C(=O)N1 ZINC000217940809 CE For-Sale Unstable HPGD 50 35 C[C@@H](S)C(=O)NC1CCCC1 ZINC000217940824 AD For-Sale Unstable HDAC4 15 40 C[C@@H](S)C(=O)NC1CCCC1 ZINC000217940824 AD For-Sale Unstable EPHX2 16 40 COc1ccc(CS[C@@H](C)CCO)cc1/C=C\C(=O)O ZINC000217940836 CF For-Sale Unstable PTGER2 22 41 COc1cccc(C(=O)N(C)Cc2nc(-c3ccc(OC)cc3OC)no2)c1 ZINC000217940844 GG In-Stock Unstable GYS1 22 40 COc1cccc(C(=O)N(C)Cc2nc(-c3ccc(OC)cc3OC)no2)c1 ZINC000217940844 GG In-Stock Unstable HSD17B2 22 42 COc1cccc(/C=C/NC(=O)NC2CC(C)(C)NC(C)(C)C2)c1 ZINC000217940864 EG For-Sale Unstable EZH2 52 37 COC(=O)C[C@@H](c1c(O)cc(C)oc1=O)c1coc2ccccc2c1=O ZINC000217940873 FE In-Stock Unstable ALDH2 51 32 C[C@H](S)C(=O)NC1CCCC1 ZINC000217940914 AD For-Sale Unstable HDAC4 15 40 C[C@H](S)C(=O)NC1CCCC1 ZINC000217940914 AD For-Sale Unstable EPHX2 16 40 CCN(CC(=O)Nc1cccc(OC)c1)c1ncnc2c1cnn2C ZINC000217940934 ED On-Demand Unstable PDGFRB 38 44 CCN(CC(=O)Nc1cccc(OC)c1)c1ncnc2c1cnn2C ZINC000217940934 ED On-Demand Unstable GSK3B 16 42 CCN(CC(=O)Nc1cccc(OC)c1)c1ncnc2c1cnn2C ZINC000217940934 ED On-Demand Unstable MTNR1A 21 42 CCN(CC(=O)Nc1cccc(OC)c1)c1ncnc2c1cnn2C ZINC000217940934 ED On-Demand Unstable MTNR1B 24 41 CCN(CC(=O)Nc1cccc(OC)c1)c1ncnc2c1cnn2C ZINC000217940934 ED On-Demand Unstable FLT4 25 44 CCN(CC(=O)Nc1cccc(OC)c1)c1ncnc2c1cnn2C ZINC000217940934 ED On-Demand Unstable FLT3 20 44 CCN(CC(=O)Nc1cccc(OC)c1)c1ncnc2c1cnn2C ZINC000217940934 ED On-Demand Unstable PANK1 0 41 CCN(CC(=O)Nc1cccc(OC)c1)c1ncnc2c1cnn2C ZINC000217940934 ED On-Demand Unstable PANK3 0 41 COc1ccc(CS[C@H](C)CCO)cc1/C=C\C(=O)O ZINC000217940935 CF For-Sale Unstable PTGER2 22 41 COc1cccc(C(=O)NCCCc2ccc(C(C)C)cc2)c1 ZINC000217940956 DI In-Stock Unstable DRD2 15 50 COc1cccc(C(=O)NCCCc2ccc(C(C)C)cc2)c1 ZINC000217940956 DI In-Stock Unstable DRD4 62 47 COc1cccc(C(=O)NCCCc2ccc(C(C)C)cc2)c1 ZINC000217940956 DI In-Stock Unstable DRD3 32 50 COc1cccc(C(=O)NCCCc2ccc(C(C)C)cc2)c1 ZINC000217940956 DI In-Stock Unstable PTAFR 26 51 COc1cccc(C(=O)NCCCc2ccc(C(C)C)cc2)c1 ZINC000217940956 DI In-Stock Unstable NQO2 25 45 COc1cccc(C(=O)NCCCc2ccc(C(C)C)cc2)c1 ZINC000217940956 DI In-Stock Unstable TRPV1 0 43 COc1cccc(C(=O)NCCCc2ccc(C(C)C)cc2)c1 ZINC000217940956 DI In-Stock Unstable PTGER3 40 38 COc1cccc(C(=O)NCCCc2ccc(C(C)C)cc2)c1 ZINC000217940956 DI In-Stock Unstable C3AR1 17 40 COc1cccc(C(=O)NCCCc2ccc(C(C)C)cc2)c1 ZINC000217940956 DI In-Stock Unstable MTNR1A 87 54 COc1cccc(C(=O)NCCCc2ccc(C(C)C)cc2)c1 ZINC000217940956 DI In-Stock Unstable MTNR1B 84 54 COc1cccc(C(=O)NCCCc2ccc(C(C)C)cc2)c1 ZINC000217940956 DI In-Stock Unstable CTSS 20 45 COc1cccc(C(=O)NCCCc2ccc(C(C)C)cc2)c1 ZINC000217940956 DI In-Stock Unstable SLC6A5 23 40 COc1cccc(C(=O)NCCCc2ccc(C(C)C)cc2)c1 ZINC000217940956 DI In-Stock Unstable AMP1_PLAFQ 20 40 COc1cccc(C(=O)NCCCc2ccc(C(C)C)cc2)c1 ZINC000217940956 DI In-Stock Unstable CRTM 50 38 COc1cccc(C(=O)NCCCc2ccc(C(C)C)cc2)c1 ZINC000217940956 DI In-Stock Unstable CAN2 0 43 COc1cccc(C(=O)NCCCc2ccc(C(C)C)cc2)c1 ZINC000217940956 DI In-Stock Unstable ALPHA-1A 0 41 COc1cccc(C(=O)NCCCc2ccc(C(C)C)cc2)c1 ZINC000217940956 DI In-Stock Unstable KCNK3 18 43 CCN(Cc1cccs1)Cc1ccccc1/C=C\C(=O)O ZINC000217940965 DH For-Sale Unstable PTGER3 20 44 CCN(Cc1cccs1)Cc1ccccc1/C=C\C(=O)O ZINC000217940965 DH For-Sale Unstable PTGDR 0 43 O=C(O)C[C@@H]1CCCN1C[C@@H]1COc2ccccc2O1 ZINC000217940979 CD For-Sale Unstable HTR1A 15 49 O=C(O)C[C@@H]1CCCN1C[C@@H]1COc2ccccc2O1 ZINC000217940979 CD For-Sale Unstable DRD2 15 49 O=C(O)C[C@@H]1CCCN1C[C@@H]1COc2ccccc2O1 ZINC000217940979 CD For-Sale Unstable ADRA2B 24 43 O=C1C/C(=C\c2ccc(-n3ccnc3)cc2)C(=O)N1 ZINC000217940986 CD For-Sale Unstable GRM2 20 40 C[C@@H](S)C(=O)NC12CC3CC(CC(C3)C1)C2 ZINC000217941052 BE For-Sale Unstable EPHX2 95 55 C[C@@H](S)C(=O)NC12CC3CC(CC(C3)C1)C2 ZINC000217941052 BE For-Sale Unstable P95276_MYCTO 0 42 O=C(NC1CCC1)N1CCc2ccc(F)cc21 ZINC000217941065 BE On-Demand Unstable CCR3 33 43 O=C(NC1CCC1)N1CCc2ccc(F)cc21 ZINC000217941065 BE On-Demand Unstable SCD1 29 42 COc1cccc(C(=O)NCCCN2CCCc3ccccc32)c1 ZINC000217941070 DG In-Stock Unstable HTR1A 35 61 COc1cccc(C(=O)NCCCN2CCCc3ccccc32)c1 ZINC000217941070 DG In-Stock Unstable ADRA2A 15 48 COc1cccc(C(=O)NCCCN2CCCc3ccccc32)c1 ZINC000217941070 DG In-Stock Unstable DRD2 48 55 COc1cccc(C(=O)NCCCN2CCCc3ccccc32)c1 ZINC000217941070 DG In-Stock Unstable DRD1 28 51 COc1cccc(C(=O)NCCCN2CCCc3ccccc32)c1 ZINC000217941070 DG In-Stock Unstable DRD4 72 58 COc1cccc(C(=O)NCCCN2CCCc3ccccc32)c1 ZINC000217941070 DG In-Stock Unstable ADRA1D 21 42 COc1cccc(C(=O)NCCCN2CCCc3ccccc32)c1 ZINC000217941070 DG In-Stock Unstable HTR2A 37 44 COc1cccc(C(=O)NCCCN2CCCc3ccccc32)c1 ZINC000217941070 DG In-Stock Unstable HTR2C 35 44 COc1cccc(C(=O)NCCCN2CCCc3ccccc32)c1 ZINC000217941070 DG In-Stock Unstable AVPR2 35 57 COc1cccc(C(=O)NCCCN2CCCc3ccccc32)c1 ZINC000217941070 DG In-Stock Unstable ADRA1B 16 42 COc1cccc(C(=O)NCCCN2CCCc3ccccc32)c1 ZINC000217941070 DG In-Stock Unstable DRD3 72 58 COc1cccc(C(=O)NCCCN2CCCc3ccccc32)c1 ZINC000217941070 DG In-Stock Unstable HTR7 28 43 COc1cccc(C(=O)NCCCN2CCCc3ccccc32)c1 ZINC000217941070 DG In-Stock Unstable MTNR1A 45 39 COc1cccc(C(=O)NCCCN2CCCc3ccccc32)c1 ZINC000217941070 DG In-Stock Unstable CTSS 15 42 COc1cccc(C(=O)NCCCN2CCCc3ccccc32)c1 ZINC000217941070 DG In-Stock Unstable NAMPT 0 40 COc1cccc(C(=O)NCCCN2CCCc3ccccc32)c1 ZINC000217941070 DG In-Stock Unstable ALPHA-1A 0 51 COc1cccc(C(=O)NCCCN2CCCc3ccccc32)c1 ZINC000217941070 DG In-Stock Unstable BRPF1 0 45 COc1cccc(/C=C/NC(=O)N2CCN(CCO)CC2)c1 ZINC000217941091 DC For-Sale Unstable HTR1A 17 42 COc1cccc(/C=C/NC(=O)N2CCN(CCO)CC2)c1 ZINC000217941091 DC For-Sale Unstable DRD4 51 39 COc1cccc(/C=C/NC(=O)N2CCN(CCO)CC2)c1 ZINC000217941091 DC For-Sale Unstable DRD3 22 42 COc1cccc(/C=C/NC(=O)N2CCN(CCO)CC2)c1 ZINC000217941091 DC For-Sale Unstable MTNR1A 28 40 COc1cccc(/C=C/NC(=O)N2CCN(CCO)CC2)c1 ZINC000217941091 DC For-Sale Unstable MTNR1B 37 40 C[C@@H](Cc1ccc(C(F)F)cc1Cl)C(=O)O ZINC000217941103 BH For-Sale Unstable PTGS1 17 40 C[C@H](S)C(=O)NC12CC3CC(CC(C3)C1)C2 ZINC000217941131 BE For-Sale Unstable EPHX2 95 55 C[C@H](S)C(=O)NC12CC3CC(CC(C3)C1)C2 ZINC000217941131 BE For-Sale Unstable P95276_MYCTO 0 42 CCOC(=O)c1cnn(-c2cccc([N+](=O)[O-])c2)c1O ZINC000217941134 CD For-Sale Unstable CACNA1C 72 44 CCOC(=O)c1cnn(-c2cccc([N+](=O)[O-])c2)c1O ZINC000217941134 CD For-Sale Unstable CACNA1D 101 43 CCOC(=O)c1cnn(-c2cccc([N+](=O)[O-])c2)c1O ZINC000217941134 CD For-Sale Unstable CTRB1 28 42 Cc1noc2nc(C(C)C)cc(C(=O)Nc3cccc(S(=O)(=O)Nc4ccccc4Cl)c3)c12 ZINC000217941151 JK On-Demand Unstable GRM4 34 43 Cc1noc2nc(C(C)C)cc(C(=O)Nc3cccc(S(=O)(=O)Nc4ccccc4Cl)c3)c12 ZINC000217941151 JK On-Demand Unstable NR2E3 52 33 C[C@H](Cc1ccc(C(F)F)cc1Cl)C(=O)O ZINC000217941190 BH For-Sale Unstable PTGS1 17 40 COc1ccc(CNC(=O)c2ccc(C)c([N+](=O)[O-])c2)c(OC)c1OC ZINC000217941191 FF In-Stock Unstable TPPP 0 40 CC[C@@H]1CCCN1CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217941193 CG For-Sale Unstable LTA4H 16 41 CC[C@@H]1CCCN1CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217941193 CG For-Sale Unstable HRH3 18 41 CC[C@@H]1CCCN1CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217941193 CG For-Sale Unstable CHRNA10 65 38 CC[C@@H]1CCCN1CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217941193 CG For-Sale Unstable ACKR3 72 38 COc1cccc(/C=C/NC(=O)N2CCC[C@@H](C)C2)c1 ZINC000217941206 CG For-Sale Unstable EBP 18 41 COc1cccc(/C=C/NC(=O)N2CCC[C@@H](C)C2)c1 ZINC000217941206 CG For-Sale Unstable RORC 47 41 COc1cccc(/C=C/NC(=O)N2CCC[C@@H](C)C2)c1 ZINC000217941206 CG For-Sale Unstable ACKR3 48 33 O=C(O)c1cnn(-c2cccc([N+](=O)[O-])c2)c1O ZINC000217941250 BD For-Sale Bother AKR1C2 17 43 CN(C/C(=C\C#N)c1ccccc1)C(=O)OC(C)(C)C ZINC000217941260 CG For-Sale Unstable CTSB 32 45 CN(C/C(=C\C#N)c1ccccc1)C(=O)OC(C)(C)C ZINC000217941260 CG For-Sale Unstable PAPA1_CARPA 44 39 O=C(O)C[C@@H]1CCCN1C/C=C\c1ccccc1 ZINC000217941279 BF On-Demand Unstable SLC6A1 33 58 O=C(O)C[C@@H]1CCCN1C/C=C\c1ccccc1 ZINC000217941279 BF On-Demand Unstable ACKR3 40 39 CC[C@H]1CCCN1CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217941281 CG For-Sale Unstable LTA4H 16 41 CC[C@H]1CCCN1CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217941281 CG For-Sale Unstable HRH3 18 41 CC[C@H]1CCCN1CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217941281 CG For-Sale Unstable CHRNA10 65 38 CC[C@H]1CCCN1CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217941281 CG For-Sale Unstable ACKR3 72 38 COc1cccc(/C=C/NC(=O)N2CCC[C@H](C)C2)c1 ZINC000217941289 CG For-Sale Unstable EBP 18 41 COc1cccc(/C=C/NC(=O)N2CCC[C@H](C)C2)c1 ZINC000217941289 CG For-Sale Unstable RORC 47 41 COc1cccc(/C=C/NC(=O)N2CCC[C@H](C)C2)c1 ZINC000217941289 CG For-Sale Unstable ACKR3 48 33 CCOc1ccc(CNC(=O)c2ccc(C)c([N+](=O)[O-])c2)cc1OCC ZINC000217941298 FH In-Stock Unstable MT-ND1 15 40 Cc1ccc(N[C@H]2C[C@H](C)CC[C@H]2C(C)C)cc1[N+](=O)[O-] ZINC000217941316 CJ For-Sale Unstable TRPM8 15 41 O=C1C/C(=C\c2c[nH]c3ccccc23)C(=O)N1 ZINC000217941328 BD For-Sale Unstable PRKCB 0 43 COc1cccc(/C=C/NC(=O)Nc2ccc(C)c(C)c2)c1 ZINC000217941392 CI For-Sale Unstable CYP1B1 22 41 COc1cccc(/C=C/NC(=O)Nc2ccc(C)c(C)c2)c1 ZINC000217941392 CI For-Sale Unstable MTNR1A 34 46 COc1cccc(/C=C/NC(=O)Nc2ccc(C)c(C)c2)c1 ZINC000217941392 CI For-Sale Unstable MTNR1B 39 46 COc1cccc(/C=C/NC(=O)Nc2ccc(C)c(C)c2)c1 ZINC000217941392 CI For-Sale Unstable CYP1A1 18 41 COc1cccc(/C=C/NC(=O)Nc2ccc(C)c(C)c2)c1 ZINC000217941392 CI For-Sale Unstable IMPDH2 0 41 CC(F)(F)c1c(Cl)cccc1CCC(=O)O ZINC000217941397 BG For-Sale Unstable CXCL8 44 36 CC(F)(F)c1c(Cl)cccc1CCC(=O)O ZINC000217941397 BG For-Sale Unstable FFAR1 46 38 CC(F)(F)c1c(Cl)cccc1CCC(=O)O ZINC000217941397 BG For-Sale Unstable FFAR4 48 33 CC[C@@H]1CCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217941405 CG For-Sale Unstable LTA4H 33 46 CC[C@@H]1CCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217941405 CG For-Sale Unstable HRH3 39 44 CC[C@@H]1CCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217941405 CG For-Sale Unstable CHRNA10 44 37 CC[C@@H]1CCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217941405 CG For-Sale Unstable PSMB2 45 34 Cc1ccc(N[C@H]2C[C@@H](C)CC[C@H]2C(C)C)cc1[N+](=O)[O-] ZINC000217941407 CJ For-Sale Unstable TRPM8 15 41 COc1ccccc1CCCNC(=O)c1ccc(C)c([N+](=O)[O-])c1 ZINC000217941409 EG In-Stock Unstable DRD2 17 41 COc1ccccc1CCCNC(=O)c1ccc(C)c([N+](=O)[O-])c1 ZINC000217941409 EG In-Stock Unstable DRD3 25 41 COc1ccccc1CCCNC(=O)c1ccc(C)c([N+](=O)[O-])c1 ZINC000217941409 EG In-Stock Unstable COLA 42 32 COc1ccccc1CCCNC(=O)c1ccc(C)c([N+](=O)[O-])c1 ZINC000217941409 EG In-Stock Unstable MTNR1B 36 41 COc1ccccc1CCCNC(=O)c1ccc(C)c([N+](=O)[O-])c1 ZINC000217941409 EG In-Stock Unstable TAAR1 19 41 CC[C@H]1CCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217941484 CG For-Sale Unstable LTA4H 33 46 CC[C@H]1CCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217941484 CG For-Sale Unstable HRH3 39 44 CC[C@H]1CCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217941484 CG For-Sale Unstable CHRNA10 44 37 CC[C@H]1CCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217941484 CG For-Sale Unstable PSMB2 45 34 O=C(O)c1cnn(-c2ncc(C(F)(F)F)cc2Cl)c1O ZINC000217941488 DE For-Sale Anodyne TRPM8 40 35 C[C@@H](CC(=O)O)c1cccc(Cl)c1C(F)F ZINC000217941498 BH For-Sale Unstable CXCL8 53 35 Cc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1[N+](=O)[O-] ZINC000217941505 FI In-Stock Unstable PYGL 24 41 Cc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1[N+](=O)[O-] ZINC000217941505 FI In-Stock Unstable PPARD 0 41 Cc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1[N+](=O)[O-] ZINC000217941505 FI In-Stock Unstable NR1H4 24 44 Cc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1[N+](=O)[O-] ZINC000217941505 FI In-Stock Unstable KCNMA1 29 42 Cc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1[N+](=O)[O-] ZINC000217941505 FI In-Stock Unstable FABH 0 43 Cc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1[N+](=O)[O-] ZINC000217941505 FI In-Stock Unstable TAAR1 20 44 Cc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1[N+](=O)[O-] ZINC000217941505 FI In-Stock Unstable SIRT2 17 47 Cc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1[N+](=O)[O-] ZINC000217941505 FI In-Stock Unstable MCL1 0 40 Cc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1[N+](=O)[O-] ZINC000217941505 FI In-Stock Unstable AKR1C3 19 45 Cc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1[N+](=O)[O-] ZINC000217941505 FI In-Stock Unstable PAGA 0 42 Cc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1[N+](=O)[O-] ZINC000217941505 FI In-Stock Unstable KCNK3 60 34 Cc1ccc(C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1[N+](=O)[O-] ZINC000217941505 FI In-Stock Unstable KLF10 0 44 CCN(Cc1ccccc1)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217941516 DH For-Sale Unstable TSPO 50 34 CCN(Cc1ccccc1)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217941516 DH For-Sale Unstable G6PC 28 49 CCN(Cc1ccccc1)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217941516 DH For-Sale Unstable MTNR1A 46 42 CCN(Cc1ccccc1)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217941516 DH For-Sale Unstable MTNR1B 48 42 CCN(Cc1ccccc1)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217941516 DH For-Sale Unstable ROCK2 30 46 CCN(Cc1ccccc1)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217941516 DH For-Sale Unstable NR1H4 44 37 CCN(Cc1ccccc1)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217941516 DH For-Sale Unstable PTGES 22 48 CCN(Cc1ccccc1)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217941516 DH For-Sale Unstable PDS 35 43 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)NCCn3c(=O)c(O)nc4ccccc43)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217941562 KF In-Stock Unstable TUBA1A 15 57 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)NCCn3c(=O)c(O)nc4ccccc43)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217941562 KF In-Stock Unstable TPPP 0 54 C[C@H](CC(=O)O)c1cccc(Cl)c1C(F)F ZINC000217941576 BH For-Sale Unstable CXCL8 53 35 COc1ccc(CN2CCC(C)CC2)cc1/C=C\C(=O)O ZINC000217941620 CG For-Sale Unstable DRD2 20 40 COc1ccc(CN2CCC(C)CC2)cc1/C=C\C(=O)O ZINC000217941620 CG For-Sale Unstable DRD4 38 40 COc1ccc(CN2CCC(C)CC2)cc1/C=C\C(=O)O ZINC000217941620 CG For-Sale Unstable ACHE 28 44 COc1ccc(CN2CCC(C)CC2)cc1/C=C\C(=O)O ZINC000217941620 CG For-Sale Unstable PTGER2 28 41 COc1ccc(CN2CCC(C)CC2)cc1/C=C\C(=O)O ZINC000217941620 CG For-Sale Unstable PTGER4 0 41 COc1ccc(CN2CCC(C)CC2)cc1/C=C\C(=O)O ZINC000217941620 CG For-Sale Unstable SIGMAR1 37 42 COc1ccc(CN2CCC(C)CC2)cc1/C=C\C(=O)O ZINC000217941620 CG For-Sale Unstable SSTR5 64 39 COc1ccc(CN2CCC(C)CC2)cc1/C=C\C(=O)O ZINC000217941620 CG For-Sale Unstable CCR3 18 40 COc1ccc(CN2CCC(C)CC2)cc1/C=C\C(=O)O ZINC000217941620 CG For-Sale Unstable MCHR1 27 45 COc1ccc(CN2CCC(C)CC2)cc1/C=C\C(=O)O ZINC000217941620 CG For-Sale Unstable CCR8 19 41 CCOc1ccc(CCCNC(=O)c2ccc(C)c([N+](=O)[O-])c2)cc1 ZINC000217941627 EH In-Stock Unstable SCN2A 21 44 COc1cccc(/C=C/NC(=O)N2CCCC[C@@H]2C)c1 ZINC000217941633 CG For-Sale Unstable FKBP1A 22 44 COc1cccc(/C=C/NC(=O)N2CCCC[C@@H]2C)c1 ZINC000217941633 CG For-Sale Unstable DRD4 40 32 COc1cccc(/C=C/NC(=O)N2CCCC[C@@H]2C)c1 ZINC000217941633 CG For-Sale Unstable COLA 50 38 COc1cccc(/C=C/NC(=O)N2CCCC[C@@H]2C)c1 ZINC000217941633 CG For-Sale Unstable CPT1A 48 38 COc1cccc(/C=C/NC(=O)N2CCCC[C@@H]2C)c1 ZINC000217941633 CG For-Sale Unstable MTNR1A 41 36 COc1cccc(/C=C/NC(=O)N2CCCC[C@@H]2C)c1 ZINC000217941633 CG For-Sale Unstable MTNR1B 48 40 C[C@@H](Cc1cccc(Cl)c1C(F)F)C(=O)O ZINC000217941678 BH For-Sale Unstable CXCL8 54 33 Cc1cc(S(=O)(=O)NCC[C@H](O)c2cccn2C)ccc1F ZINC000217941683 ED In-Stock Unstable LEF 69 43 COc1cccc(/C=C/NC(=O)N2CCCC[C@H]2C)c1 ZINC000217941715 CG For-Sale Unstable FKBP1A 22 44 COc1cccc(/C=C/NC(=O)N2CCCC[C@H]2C)c1 ZINC000217941715 CG For-Sale Unstable DRD4 40 32 COc1cccc(/C=C/NC(=O)N2CCCC[C@H]2C)c1 ZINC000217941715 CG For-Sale Unstable COLA 50 38 COc1cccc(/C=C/NC(=O)N2CCCC[C@H]2C)c1 ZINC000217941715 CG For-Sale Unstable CPT1A 48 38 COc1cccc(/C=C/NC(=O)N2CCCC[C@H]2C)c1 ZINC000217941715 CG For-Sale Unstable MTNR1A 41 36 COc1cccc(/C=C/NC(=O)N2CCCC[C@H]2C)c1 ZINC000217941715 CG For-Sale Unstable MTNR1B 48 40 CCCOc1ccccc1CCCNC(=O)c1ccc(C)c([N+](=O)[O-])c1 ZINC000217941734 FI In-Stock Unstable ACAT 0 40 CNC(=O)[C@@H]1CCCN(C(=O)NC2CCC2)C1 ZINC000217941746 BC On-Demand Unstable NMUR2 0 40 CNC(=O)[C@@H]1CCCN(C(=O)NC2CCC2)C1 ZINC000217941746 BC On-Demand Unstable NMUR1 0 40 C[C@H](Cc1cccc(Cl)c1C(F)F)C(=O)O ZINC000217941753 BH For-Sale Unstable CXCL8 54 33 Cc1cc(S(=O)(=O)NCC[C@@H](O)c2cccn2C)ccc1F ZINC000217941758 ED In-Stock Unstable LEF 69 43 Cc1ccc(C(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)c(-n2cnnn2)c1C ZINC000217941784 GD In-Stock Unstable CHRNA4 26 41 C[C@@H](S)C(=O)NC1CCCCC1 ZINC000217941797 AD For-Sale Unstable MMP2 0 45 Cc1ccccc1OC[C@@H](C)NC(=O)c1ccc(C)c([N+](=O)[O-])c1 ZINC000217941820 EG In-Stock Unstable COLA 43 32 Cc1ccccc1OC[C@@H](C)NC(=O)c1ccc(C)c([N+](=O)[O-])c1 ZINC000217941820 EG In-Stock Unstable TAAR1 18 41 CNC(=O)[C@H]1CCCN(C(=O)NC2CCC2)C1 ZINC000217941826 BC On-Demand Unstable NMUR2 0 40 CNC(=O)[C@H]1CCCN(C(=O)NC2CCC2)C1 ZINC000217941826 BC On-Demand Unstable NMUR1 0 40 O=C(N[C@@H]1CCC[C@@H]1CO)c1ccc([N+](=O)[O-])o1 ZINC000217941827 CD For-Sale Unstable DDIT3 0 47 CC[C@@H]1CCCCN1C(=O)N/C=C/c1cccc(OC)c1 ZINC000217941834 CH For-Sale Unstable FKBP1A 34 44 CC[C@@H]1CCCCN1C(=O)N/C=C/c1cccc(OC)c1 ZINC000217941834 CH For-Sale Unstable DRD4 40 31 CC[C@@H]1CCCCN1C(=O)N/C=C/c1cccc(OC)c1 ZINC000217941834 CH For-Sale Unstable COLA 66 38 CC[C@@H]1CCCCN1C(=O)N/C=C/c1cccc(OC)c1 ZINC000217941834 CH For-Sale Unstable CPT1A 61 38 CC[C@@H]1CCCCN1C(=O)N/C=C/c1cccc(OC)c1 ZINC000217941834 CH For-Sale Unstable MTNR1A 40 38 CC[C@@H]1CCCCN1C(=O)N/C=C/c1cccc(OC)c1 ZINC000217941834 CH For-Sale Unstable MTNR1B 50 38 CC[C@@H]1CCCCN1C(=O)N/C=C/c1cccc(OC)c1 ZINC000217941834 CH For-Sale Unstable CHRNA10 34 41 CC[C@@H]1CCCCN1C(=O)N/C=C/c1cccc(OC)c1 ZINC000217941834 CH For-Sale Unstable ACKR3 59 35 CN1CCN(Cc2ccc(F)c(/C=C\C(=O)O)c2)CC1 ZINC000217941843 CD For-Sale Unstable SIGMAR1 19 40 Cc1cc(Cl)c(F)c([C@@H](C)CC(=O)O)c1F ZINC000217941863 BH For-Sale Unstable HMGCR 45 36 CCOC(=O)c1cnn(-c2ccccc2Cl)c1O ZINC000217941867 CE For-Sale Unstable HPD 41 41 C[C@H](S)C(=O)NC1CCCCC1 ZINC000217941871 AD For-Sale Unstable MMP2 0 45 Cn1cccc1[C@H](O)CCNS(=O)(=O)c1ccc(F)c(F)c1 ZINC000217941881 ED In-Stock Unstable TBXA2R 42 33 Cn1cccc1[C@H](O)CCNS(=O)(=O)c1ccc(F)c(F)c1 ZINC000217941881 ED In-Stock Unstable LEF 40 33 O=C(N[C@H]1CCC[C@@H]1CO)c1ccc([N+](=O)[O-])o1 ZINC000217941907 CD For-Sale Unstable DDIT3 0 47 CC[C@H]1CCCCN1C(=O)N/C=C/c1cccc(OC)c1 ZINC000217941917 CH For-Sale Unstable FKBP1A 34 44 CC[C@H]1CCCCN1C(=O)N/C=C/c1cccc(OC)c1 ZINC000217941917 CH For-Sale Unstable DRD4 40 31 CC[C@H]1CCCCN1C(=O)N/C=C/c1cccc(OC)c1 ZINC000217941917 CH For-Sale Unstable COLA 66 38 CC[C@H]1CCCCN1C(=O)N/C=C/c1cccc(OC)c1 ZINC000217941917 CH For-Sale Unstable CPT1A 61 38 CC[C@H]1CCCCN1C(=O)N/C=C/c1cccc(OC)c1 ZINC000217941917 CH For-Sale Unstable MTNR1A 40 38 CC[C@H]1CCCCN1C(=O)N/C=C/c1cccc(OC)c1 ZINC000217941917 CH For-Sale Unstable MTNR1B 50 38 CC[C@H]1CCCCN1C(=O)N/C=C/c1cccc(OC)c1 ZINC000217941917 CH For-Sale Unstable CHRNA10 34 41 CC[C@H]1CCCCN1C(=O)N/C=C/c1cccc(OC)c1 ZINC000217941917 CH For-Sale Unstable ACKR3 59 35 Cc1cc(Cl)c(F)c([C@H](C)CC(=O)O)c1F ZINC000217941933 BH For-Sale Unstable HMGCR 45 36 Cn1cccc1[C@@H](O)CCNS(=O)(=O)c1ccc(F)c(F)c1 ZINC000217941967 ED In-Stock Unstable TBXA2R 42 33 Cn1cccc1[C@@H](O)CCNS(=O)(=O)c1ccc(F)c(F)c1 ZINC000217941967 ED In-Stock Unstable LEF 40 33 C[C@@H](S)C(=O)Nc1cccc(Oc2ccccc2)c1 ZINC000217941980 CH For-Sale Unstable MME 18 47 C[C@@H](S)C(=O)Nc1cccc(Oc2ccccc2)c1 ZINC000217941980 CH For-Sale Unstable LTA4H 30 42 C[C@@H](S)C(=O)Nc1cccc(Oc2ccccc2)c1 ZINC000217941980 CH For-Sale Unstable CA1 26 50 C[C@@H](S)C(=O)Nc1cccc(Oc2ccccc2)c1 ZINC000217941980 CH For-Sale Unstable ACACA 15 45 C[C@@H](S)C(=O)Nc1cccc(Oc2ccccc2)c1 ZINC000217941980 CH For-Sale Unstable ACACB 17 45 C[C@@H](S)C(=O)Nc1cccc(Oc2ccccc2)c1 ZINC000217941980 CH For-Sale Unstable RAF1 22 45 C[C@@H](S)C(=O)Nc1cccc(Oc2ccccc2)c1 ZINC000217941980 CH For-Sale Unstable MTNR1B 19 53 C[C@@H](S)C(=O)Nc1cccc(Oc2ccccc2)c1 ZINC000217941980 CH For-Sale Unstable NPY5R 29 40 C[C@@H](S)C(=O)Nc1cccc(Oc2ccccc2)c1 ZINC000217941980 CH For-Sale Unstable ACE2 50 47 C[C@@H](S)C(=O)Nc1cccc(Oc2ccccc2)c1 ZINC000217941980 CH For-Sale Unstable AMP1_PLAFQ 23 43 C[C@@H](S)C(=O)Nc1cccc(Oc2ccccc2)c1 ZINC000217941980 CH For-Sale Unstable F13A1 18 50 C[C@@H](S)C(=O)Nc1cccc(Oc2ccccc2)c1 ZINC000217941980 CH For-Sale Unstable TAAR1 42 41 C[C@@H](S)C(=O)Nc1cccc(Oc2ccccc2)c1 ZINC000217941980 CH For-Sale Unstable KCNK3 105 43 C[C@@H](S)C(=O)Nc1cccc(Oc2ccccc2)c1 ZINC000217941980 CH For-Sale Unstable KCNK9 77 40 O=C(N[C@@H]1CCC[C@H]1CO)c1ccc([N+](=O)[O-])o1 ZINC000217941983 CD For-Sale Unstable DDIT3 0 47 O=C(/C=C\c1cc(Cl)ccc1Cl)CCl ZINC000217941993 BH For-Sale Unstable BOTA 17 45 O=C(/C=C\c1cc(Cl)ccc1Cl)CCl ZINC000217941993 BH For-Sale Unstable CYSP_PLAFA 28 46 CCOC(=O)c1cnn(-c2ccc(C)cc2C)c1O ZINC000217941995 CE For-Sale Unstable HPD 34 41 COc1cccc(/C=C/NC(=O)N(Cc2ccccc2)Cc2ccccc2)c1 ZINC000217942025 FK For-Sale Unstable TSPO 45 36 COc1cccc(/C=C/NC(=O)N(Cc2ccccc2)Cc2ccccc2)c1 ZINC000217942025 FK For-Sale Unstable G6PC 30 52 COc1cccc(/C=C/NC(=O)N(Cc2ccccc2)Cc2ccccc2)c1 ZINC000217942025 FK For-Sale Unstable MTNR1A 53 44 COc1cccc(/C=C/NC(=O)N(Cc2ccccc2)Cc2ccccc2)c1 ZINC000217942025 FK For-Sale Unstable MTNR1B 55 44 COc1cccc(/C=C/NC(=O)N(Cc2ccccc2)Cc2ccccc2)c1 ZINC000217942025 FK For-Sale Unstable NR1H4 47 39 COc1cccc(/C=C/NC(=O)N(Cc2ccccc2)Cc2ccccc2)c1 ZINC000217942025 FK For-Sale Unstable CRTM 40 34 COc1cccc(/C=C/NC(=O)N(Cc2ccccc2)Cc2ccccc2)c1 ZINC000217942025 FK For-Sale Unstable PTGES 28 53 O=C(N[C@H]1CCC[C@H]1CO)c1ccc([N+](=O)[O-])o1 ZINC000217942044 CD On-Demand Unstable GSR 40 41 O=C(N[C@H]1CCC[C@H]1CO)c1ccc([N+](=O)[O-])o1 ZINC000217942044 CD On-Demand Unstable DDIT3 0 47 CC1(C)[C@H]2CC[C@@]1(C)[C@@H](NC(=O)Cn1c3ccccc3c(=O)c3ccccc31)C2 ZINC000217942045 GI On-Demand Unstable AVPR2 40 37 CC1(C)[C@H]2CC[C@@]1(C)[C@@H](NC(=O)Cn1c3ccccc3c(=O)c3ccccc31)C2 ZINC000217942045 GI On-Demand Unstable CNR2 15 43 C[C@H](S)C(=O)Nc1cccc(Oc2ccccc2)c1 ZINC000217942055 CH For-Sale Unstable MME 18 47 C[C@H](S)C(=O)Nc1cccc(Oc2ccccc2)c1 ZINC000217942055 CH For-Sale Unstable LTA4H 30 42 C[C@H](S)C(=O)Nc1cccc(Oc2ccccc2)c1 ZINC000217942055 CH For-Sale Unstable CA1 26 50 C[C@H](S)C(=O)Nc1cccc(Oc2ccccc2)c1 ZINC000217942055 CH For-Sale Unstable ACACA 15 45 C[C@H](S)C(=O)Nc1cccc(Oc2ccccc2)c1 ZINC000217942055 CH For-Sale Unstable ACACB 17 45 C[C@H](S)C(=O)Nc1cccc(Oc2ccccc2)c1 ZINC000217942055 CH For-Sale Unstable RAF1 22 45 C[C@H](S)C(=O)Nc1cccc(Oc2ccccc2)c1 ZINC000217942055 CH For-Sale Unstable MTNR1B 19 53 C[C@H](S)C(=O)Nc1cccc(Oc2ccccc2)c1 ZINC000217942055 CH For-Sale Unstable NPY5R 29 40 C[C@H](S)C(=O)Nc1cccc(Oc2ccccc2)c1 ZINC000217942055 CH For-Sale Unstable ACE2 50 47 C[C@H](S)C(=O)Nc1cccc(Oc2ccccc2)c1 ZINC000217942055 CH For-Sale Unstable AMP1_PLAFQ 23 43 C[C@H](S)C(=O)Nc1cccc(Oc2ccccc2)c1 ZINC000217942055 CH For-Sale Unstable F13A1 18 50 C[C@H](S)C(=O)Nc1cccc(Oc2ccccc2)c1 ZINC000217942055 CH For-Sale Unstable TAAR1 42 41 C[C@H](S)C(=O)Nc1cccc(Oc2ccccc2)c1 ZINC000217942055 CH For-Sale Unstable KCNK3 105 43 C[C@H](S)C(=O)Nc1cccc(Oc2ccccc2)c1 ZINC000217942055 CH For-Sale Unstable KCNK9 77 40 CN(Cc1cccc(/C=C\C(=O)O)c1)C1CCCCC1 ZINC000217942078 CH For-Sale Unstable ACE 41 36 CN(Cc1cccc(/C=C\C(=O)O)c1)C1CCCCC1 ZINC000217942078 CH For-Sale Unstable PTGER2 24 42 CN(Cc1cccc(/C=C\C(=O)O)c1)C1CCCCC1 ZINC000217942078 CH For-Sale Unstable NR1H4 47 42 CC(C)CCn1cnc2ccc(NC(=O)c3cccnc3)cc2c1=O ZINC000217942088 EG In-Stock Unstable TBXAS1 32 43 CC(C)CCn1cnc2ccc(NC(=O)c3cccnc3)cc2c1=O ZINC000217942088 EG In-Stock Unstable CSF1R 0 40 CC(C)CCn1cnc2ccc(NC(=O)c3cccnc3)cc2c1=O ZINC000217942088 EG In-Stock Unstable SCD1 0 45 CCOC(=O)c1cnn(Cc2ccc(C)cc2)c1O ZINC000217942119 CE For-Sale Unstable F2RL3 18 40 COc1cccc(/C=C/NC(=O)N(CCO)Cc2ccccc2)c1 ZINC000217942136 EF For-Sale Unstable TSPO 42 33 COc1cccc(/C=C/NC(=O)N(CCO)Cc2ccccc2)c1 ZINC000217942136 EF For-Sale Unstable G6PC 27 47 COc1cccc(/C=C/NC(=O)N(CCO)Cc2ccccc2)c1 ZINC000217942136 EF For-Sale Unstable MTNR1A 32 40 COc1cccc(/C=C/NC(=O)N(CCO)Cc2ccccc2)c1 ZINC000217942136 EF For-Sale Unstable MTNR1B 27 40 COc1cccc(/C=C/NC(=O)N(CCO)Cc2ccccc2)c1 ZINC000217942136 EF For-Sale Unstable ROCK2 29 48 COc1cccc(/C=C/NC(=O)N(CCO)Cc2ccccc2)c1 ZINC000217942136 EF For-Sale Unstable CDC42BPA 0 48 COc1cccc(/C=C/NC(=O)N(CCO)Cc2ccccc2)c1 ZINC000217942136 EF For-Sale Unstable PTGES 22 46 Cc1ccc([N+](=O)[O-])cc1N[C@H]1C[C@H](C)CC[C@H]1C(C)C ZINC000217942137 CJ For-Sale Unstable TRPM8 15 41 C[C@@H](S)C(=O)N(Cc1ccccc1)Cc1ccccc1 ZINC000217942173 CH For-Sale Unstable ACE 55 46 C[C@@H](S)C(=O)N(Cc1ccccc1)Cc1ccccc1 ZINC000217942173 CH For-Sale Unstable MME 76 43 C[C@@H](S)C(=O)N(Cc1ccccc1)Cc1ccccc1 ZINC000217942173 CH For-Sale Unstable CPA1 64 39 C[C@@H](S)C(=O)N(Cc1ccccc1)Cc1ccccc1 ZINC000217942173 CH For-Sale Unstable ACE2 57 39 C[C@@H](S)C(=O)N(Cc1ccccc1)Cc1ccccc1 ZINC000217942173 CH For-Sale Unstable PTGES 25 43 C[C@@H](S)C(=O)N(Cc1ccccc1)Cc1ccccc1 ZINC000217942173 CH For-Sale Unstable BLAIMP-1 0 44 O=C(O)C[C@@H]1CCCN1C[C@@H](O)c1ccccc1 ZINC000217942176 BD On-Demand Unstable SLC18A2 50 47 O=C(O)C[C@@H]1CCCN1C[C@@H](O)c1ccccc1 ZINC000217942176 BD On-Demand Unstable SLC18A3 24 45 O=C(O)C[C@@H]1CCCN1C[C@@H](O)c1ccccc1 ZINC000217942176 BD On-Demand Unstable Q8WSF8_APLCA 33 44 Cc1ccc([C@H](N)C(=O)O)c(C)c1Br ZINC000217942206 CE For-Sale Unstable CACNA2D1 23 53 Cc1ccc([N+](=O)[O-])cc1N[C@H]1C[C@@H](C)CC[C@H]1C(C)C ZINC000217942222 CJ For-Sale Unstable TRPM8 15 41 C[C@H](S)C(=O)N(Cc1ccccc1)Cc1ccccc1 ZINC000217942251 CH For-Sale Unstable ACE 55 46 C[C@H](S)C(=O)N(Cc1ccccc1)Cc1ccccc1 ZINC000217942251 CH For-Sale Unstable MME 76 43 C[C@H](S)C(=O)N(Cc1ccccc1)Cc1ccccc1 ZINC000217942251 CH For-Sale Unstable CPA1 64 39 C[C@H](S)C(=O)N(Cc1ccccc1)Cc1ccccc1 ZINC000217942251 CH For-Sale Unstable ACE2 57 39 C[C@H](S)C(=O)N(Cc1ccccc1)Cc1ccccc1 ZINC000217942251 CH For-Sale Unstable PTGES 25 43 C[C@H](S)C(=O)N(Cc1ccccc1)Cc1ccccc1 ZINC000217942251 CH For-Sale Unstable BLAIMP-1 0 44 COc1cccc(/C=C/NC(=O)Nc2ccc(OC)cc2OC)c1 ZINC000217942261 EH For-Sale Unstable CYP1B1 67 49 COc1cccc(/C=C/NC(=O)Nc2ccc(OC)cc2OC)c1 ZINC000217942261 EH For-Sale Unstable MTNR1A 43 45 COc1cccc(/C=C/NC(=O)Nc2ccc(OC)cc2OC)c1 ZINC000217942261 EH For-Sale Unstable MTNR1B 45 45 COc1cccc(/C=C/NC(=O)Nc2ccc(OC)cc2OC)c1 ZINC000217942261 EH For-Sale Unstable CYP1A1 45 51 COc1cccc(/C=C/NC(=O)Nc2ccc(OC)cc2OC)c1 ZINC000217942261 EH For-Sale Unstable ROCK2 21 42 COc1cccc(/C=C/NC(=O)Nc2ccc(OC)cc2OC)c1 ZINC000217942261 EH For-Sale Unstable ABCG2 18 48 COc1cccc(/C=C/NC(=O)Nc2ccc(OC)cc2OC)c1 ZINC000217942261 EH For-Sale Unstable AKR1C2 45 34 Cc1ccc([C@@H](N)C(=O)O)c(C)c1Br ZINC000217942294 CE For-Sale Unstable CACNA2D1 23 53 COc1cccc(/C=C/NC(=O)Nc2cc(C)on2)c1 ZINC000217942360 CF For-Sale Unstable CYP1B1 24 42 COc1cccc(/C=C/NC(=O)Nc2cc(C)on2)c1 ZINC000217942360 CF For-Sale Unstable MTNR1A 29 41 COc1cccc(/C=C/NC(=O)Nc2cc(C)on2)c1 ZINC000217942360 CF For-Sale Unstable MTNR1B 32 41 COc1cccc(/C=C/NC(=O)Nc2cc(C)on2)c1 ZINC000217942360 CF For-Sale Unstable CYP1A1 20 42 COc1cccc(/C=C/NC(=O)Nc2cc(C)on2)c1 ZINC000217942360 CF For-Sale Unstable Q8MMZ8_EIMTE 0 45 Cc1c(Br)ccc([C@H](N)C(=O)O)c1C ZINC000217942417 CE For-Sale Unstable CACNA2D1 23 50 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cc2C)c1 ZINC000217942474 DI For-Sale Unstable S1PR4 24 44 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cc2C)c1 ZINC000217942474 DI For-Sale Unstable TAAR1 19 40 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cc2C)c1 ZINC000217942474 DI For-Sale Unstable H9CNL0_SPOEX 0 41 CCOC(=O)c1cnn(-c2cccc(Br)c2)c1O ZINC000217942476 DF For-Sale Unstable HPD 51 43 CCOC(=O)c1cnn(-c2cccc(Br)c2)c1O ZINC000217942476 DF For-Sale Unstable ELANE 17 40 Cc1c(Br)ccc([C@@H](N)C(=O)O)c1C ZINC000217942505 CE For-Sale Unstable CACNA2D1 23 50 COc1ccc(C)cc1S(=O)(=O)NCC[C@H](O)c1cccn1C ZINC000217942514 ED In-Stock Unstable CPT1A 44 31 C[C@@H](S)C(=O)N[C@@H]1CCCc2ccccc21 ZINC000217942563 BE For-Sale Unstable ACE 40 51 C[C@@H](S)C(=O)N[C@@H]1CCCc2ccccc21 ZINC000217942563 BE For-Sale Unstable MME 35 41 C[C@@H](S)C(=O)N[C@@H]1CCCc2ccccc21 ZINC000217942563 BE For-Sale Unstable BDKRB1 33 40 C[C@@H](S)C(=O)N[C@@H]1CCCc2ccccc21 ZINC000217942563 BE For-Sale Unstable KCNN3 16 40 C[C@@H](S)C(=O)N[C@@H]1CCCc2ccccc21 ZINC000217942563 BE For-Sale Unstable XIAP 48 60 C[C@@H](S)C(=O)N[C@@H]1CCCc2ccccc21 ZINC000217942563 BE For-Sale Unstable BIRC3 64 52 C[C@@H](S)C(=O)N[C@@H]1CCCc2ccccc21 ZINC000217942563 BE For-Sale Unstable BIRC2 66 52 C[C@@H](S)C(=O)N[C@@H]1CCCc2ccccc21 ZINC000217942563 BE For-Sale Unstable ACAT 0 59 COc1cccc(/C=C/NC(=O)NCCCO)c1 ZINC000217942575 CD For-Sale Unstable DRD4 42 32 COc1cccc(/C=C/NC(=O)NCCCO)c1 ZINC000217942575 CD For-Sale Unstable AHR 18 42 COc1cccc(/C=C/NC(=O)NCCCO)c1 ZINC000217942575 CD For-Sale Unstable MTNR1A 89 51 COc1cccc(/C=C/NC(=O)NCCCO)c1 ZINC000217942575 CD For-Sale Unstable MTNR1B 83 51 CCOC(=O)c1cnn(-c2ccccc2Br)c1O ZINC000217942583 DF For-Sale Unstable HPD 26 43 CCOC(=O)c1cnn(-c2ccccc2Br)c1O ZINC000217942583 DF For-Sale Unstable SLC5A1 15 49 CCOC(=O)c1cnn(-c2ccccc2Br)c1O ZINC000217942583 DF For-Sale Unstable SLC5A2 16 49 COc1ccc(C)cc1S(=O)(=O)NCC[C@@H](O)c1cccn1C ZINC000217942588 ED In-Stock Unstable CPT1A 44 31 O=Cc1cc(Cl)c(=O)n(Cc2ccccc2)n1 ZINC000217942594 BD For-Sale Unstable CXCR2 20 43 O=Cc1cc(Cl)c(=O)n(Cc2ccccc2)n1 ZINC000217942594 BD For-Sale Unstable NPBWR1 29 42 Cc1cc([C@H](N)C(=O)O)c(C)cc1Br ZINC000217942628 CE For-Sale Unstable CACNA2D1 21 50 C[C@H](S)C(=O)N[C@@H]1CCCc2ccccc21 ZINC000217942653 BE For-Sale Unstable ACE 40 51 C[C@H](S)C(=O)N[C@@H]1CCCc2ccccc21 ZINC000217942653 BE For-Sale Unstable MME 35 41 C[C@H](S)C(=O)N[C@@H]1CCCc2ccccc21 ZINC000217942653 BE For-Sale Unstable BDKRB1 33 40 C[C@H](S)C(=O)N[C@@H]1CCCc2ccccc21 ZINC000217942653 BE For-Sale Unstable KCNN3 16 40 C[C@H](S)C(=O)N[C@@H]1CCCc2ccccc21 ZINC000217942653 BE For-Sale Unstable XIAP 48 60 C[C@H](S)C(=O)N[C@@H]1CCCc2ccccc21 ZINC000217942653 BE For-Sale Unstable BIRC3 64 52 C[C@H](S)C(=O)N[C@@H]1CCCc2ccccc21 ZINC000217942653 BE For-Sale Unstable BIRC2 66 52 C[C@H](S)C(=O)N[C@@H]1CCCc2ccccc21 ZINC000217942653 BE For-Sale Unstable ACAT 0 59 CN(Cc1cccc(/C=C\C(=O)O)c1)C[C@@H]1CCCCO1 ZINC000217942696 CF For-Sale Unstable OXTR 26 42 CN(Cc1cccc(/C=C\C(=O)O)c1)C[C@@H]1CCCCO1 ZINC000217942696 CF For-Sale Unstable AVPR1A 0 42 COc1cccc(/C=C/NC(=O)NCCOCCO)c1 ZINC000217942699 CC For-Sale Unstable DRD4 40 30 COc1cccc(/C=C/NC(=O)NCCOCCO)c1 ZINC000217942699 CC For-Sale Unstable MTNR1A 69 47 COc1cccc(/C=C/NC(=O)NCCOCCO)c1 ZINC000217942699 CC For-Sale Unstable MTNR1B 67 47 CCOC(=O)c1cnn(-c2cccc(C#N)c2)c1O ZINC000217942715 CD For-Sale Unstable P2RY12 36 41 Cc1cc([C@@H](N)C(=O)O)c(C)cc1Br ZINC000217942718 CE For-Sale Unstable CACNA2D1 21 50 C[C@@H](S)C(=O)N[C@H]1CCCc2ccccc21 ZINC000217942736 BE For-Sale Unstable ACE 40 51 C[C@@H](S)C(=O)N[C@H]1CCCc2ccccc21 ZINC000217942736 BE For-Sale Unstable MME 35 41 C[C@@H](S)C(=O)N[C@H]1CCCc2ccccc21 ZINC000217942736 BE For-Sale Unstable BDKRB1 33 40 C[C@@H](S)C(=O)N[C@H]1CCCc2ccccc21 ZINC000217942736 BE For-Sale Unstable KCNN3 16 40 C[C@@H](S)C(=O)N[C@H]1CCCc2ccccc21 ZINC000217942736 BE For-Sale Unstable XIAP 48 60 C[C@@H](S)C(=O)N[C@H]1CCCc2ccccc21 ZINC000217942736 BE For-Sale Unstable BIRC3 64 52 C[C@@H](S)C(=O)N[C@H]1CCCc2ccccc21 ZINC000217942736 BE For-Sale Unstable BIRC2 66 52 C[C@@H](S)C(=O)N[C@H]1CCCc2ccccc21 ZINC000217942736 BE For-Sale Unstable ACAT 0 59 CCN(CC(=O)NC)Cc1ccccc1/C=C\C(=O)O ZINC000217942802 CD For-Sale Unstable PTGER2 42 46 CCN(CC(=O)NC)Cc1ccccc1/C=C\C(=O)O ZINC000217942802 CD For-Sale Unstable PTGER4 0 46 CCN(CC(=O)NC)Cc1ccccc1/C=C\C(=O)O ZINC000217942802 CD For-Sale Unstable PTGER3 18 47 Cc1noc2nc(C(C)C)cc(C(=O)Nc3nc(-c4ccc(F)c(F)c4)cs3)c12 ZINC000217942806 HK On-Demand Unstable MPL 40 45 C[C@H](S)C(=O)N[C@H]1CCCc2ccccc21 ZINC000217942814 BE For-Sale Unstable ACE 40 51 C[C@H](S)C(=O)N[C@H]1CCCc2ccccc21 ZINC000217942814 BE For-Sale Unstable MME 35 41 C[C@H](S)C(=O)N[C@H]1CCCc2ccccc21 ZINC000217942814 BE For-Sale Unstable BDKRB1 33 40 C[C@H](S)C(=O)N[C@H]1CCCc2ccccc21 ZINC000217942814 BE For-Sale Unstable KCNN3 16 40 C[C@H](S)C(=O)N[C@H]1CCCc2ccccc21 ZINC000217942814 BE For-Sale Unstable XIAP 48 60 C[C@H](S)C(=O)N[C@H]1CCCc2ccccc21 ZINC000217942814 BE For-Sale Unstable BIRC3 64 52 C[C@H](S)C(=O)N[C@H]1CCCc2ccccc21 ZINC000217942814 BE For-Sale Unstable BIRC2 66 52 C[C@H](S)C(=O)N[C@H]1CCCc2ccccc21 ZINC000217942814 BE For-Sale Unstable ACAT 0 59 Cc1cc(C)c([C@H](N)C(=O)O)c(Br)c1 ZINC000217942823 CE For-Sale Unstable CACNA2D1 20 47 COc1ccc2c(c1)[C@@H](NC(=O)c1ccc(C)c([N+](=O)[O-])c1)CC(C)(C)O2 ZINC000217942832 FH In-Stock Unstable TAAR1 18 40 COc1ccc(F)cc1S(=O)(=O)NCC[C@@H](O)c1cccn1C ZINC000217942883 ED In-Stock Unstable CPT1A 44 31 COc1ccc2c(c1)[C@H](NC(=O)c1ccc(C)c([N+](=O)[O-])c1)CC(C)(C)O2 ZINC000217942909 FH In-Stock Unstable TAAR1 18 40 Cc1cc(C)c([C@@H](N)C(=O)O)c(Br)c1 ZINC000217942913 CE For-Sale Unstable CACNA2D1 20 47 CCCCN(CCCC)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217942916 DI For-Sale Unstable AHR 19 41 CCCCN(CCCC)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217942916 DI For-Sale Unstable MTNR1A 49 45 CCCCN(CCCC)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217942916 DI For-Sale Unstable MTNR1B 49 45 O=C(NC[C@@H]1CCCNC1)c1cc(Cl)ccn1 ZINC000217942920 CD On-Demand Unstable CACNA1I 44 35 COc1ccc(/C=C\c2csc(N)n2)c(Br)c1 ZINC000217942928 DH For-Sale Unstable CYP1B1 41 40 COc1ccc(/C=C\c2csc(N)n2)c(Br)c1 ZINC000217942928 DH For-Sale Unstable CYP1A1 38 40 C[C@@H](S)C(=O)Nc1ccc2ccccc2c1 ZINC000217942939 BG For-Sale Unstable MME 20 41 C[C@@H](S)C(=O)Nc1ccc2ccccc2c1 ZINC000217942939 BG For-Sale Unstable CMA1 32 52 C[C@@H](S)C(=O)Nc1ccc2ccccc2c1 ZINC000217942939 BG For-Sale Unstable CA1 15 44 C[C@@H](S)C(=O)Nc1ccc2ccccc2c1 ZINC000217942939 BG For-Sale Unstable ACE2 40 41 C[C@@H](S)C(=O)Nc1ccc2ccccc2c1 ZINC000217942939 BG For-Sale Unstable IMDH_CRYPV 52 44 C[C@@H](S)C(=O)Nc1ccc2ccccc2c1 ZINC000217942939 BG For-Sale Unstable Q25615_ONCVO 15 43 COc1ccc(F)cc1S(=O)(=O)NCC[C@H](O)c1cccn1C ZINC000217942966 ED In-Stock Unstable CPT1A 44 31 C[C@H](S)C(=O)Nc1ccc2ccccc2c1 ZINC000217943005 BG For-Sale Unstable MME 20 41 C[C@H](S)C(=O)Nc1ccc2ccccc2c1 ZINC000217943005 BG For-Sale Unstable CMA1 32 52 C[C@H](S)C(=O)Nc1ccc2ccccc2c1 ZINC000217943005 BG For-Sale Unstable CA1 15 44 C[C@H](S)C(=O)Nc1ccc2ccccc2c1 ZINC000217943005 BG For-Sale Unstable ACE2 40 41 C[C@H](S)C(=O)Nc1ccc2ccccc2c1 ZINC000217943005 BG For-Sale Unstable IMDH_CRYPV 52 44 C[C@H](S)C(=O)Nc1ccc2ccccc2c1 ZINC000217943005 BG For-Sale Unstable Q25615_ONCVO 15 43 Cc1ccc(C)c([C@H](N)C(=O)O)c1Br ZINC000217943020 CE For-Sale Unstable CACNA2D1 26 50 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1ccc(C)c([N+](=O)[O-])c1 ZINC000217943025 FH In-Stock Unstable CACNA1D 45 34 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)c1ccc(C)c([N+](=O)[O-])c1 ZINC000217943025 FH In-Stock Unstable TAAR1 25 44 CCN(CC)CCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217943030 DF For-Sale Unstable MTNR1A 68 46 CCN(CC)CCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217943030 DF For-Sale Unstable MTNR1B 63 46 CCCN(CCO)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217943041 CD For-Sale Unstable AKR1C3 38 40 CC[C@@H](CCO)NC(=O)CCCNC(C)C ZINC000217943060 BD For-Sale Unstable Q6UB75_PIG 0 41 CC[C@@H](CCO)NC(=O)CCCNC(C)C ZINC000217943060 BD For-Sale Unstable NOD1 55 35 CCCCCCCCOc1ccc([C@H](CC(=O)OC)c2oc(CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)cc(=O)c2O)cc1 ZINC000217943082 KK In-Stock Unstable CHRNA4 25 40 Cc1ccc(C)c([C@@H](N)C(=O)O)c1Br ZINC000217943097 CE For-Sale Unstable CACNA2D1 26 50 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1ccc(C)c([N+](=O)[O-])c1 ZINC000217943105 FH In-Stock Unstable CACNA1D 45 34 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)c1ccc(C)c([N+](=O)[O-])c1 ZINC000217943105 FH In-Stock Unstable TAAR1 25 44 COc1cccc(/C=C/NC(=O)NCCCN(C)C)c1 ZINC000217943136 CD For-Sale Unstable DRD4 40 30 COc1cccc(/C=C/NC(=O)NCCCN(C)C)c1 ZINC000217943136 CD For-Sale Unstable CYP1B1 15 40 COc1cccc(/C=C/NC(=O)NCCCN(C)C)c1 ZINC000217943136 CD For-Sale Unstable MTNR1A 73 48 COc1cccc(/C=C/NC(=O)NCCCN(C)C)c1 ZINC000217943136 CD For-Sale Unstable MTNR1B 70 48 CC[C@H](CCO)NC(=O)CCCNC(C)C ZINC000217943137 BD For-Sale Unstable Q6UB75_PIG 0 41 CC[C@H](CCO)NC(=O)CCCNC(C)C ZINC000217943137 BD For-Sale Unstable NOD1 55 35 CCCN(CCO)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217943145 CD For-Sale Unstable PTGER2 28 41 CCCN(CCO)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217943145 CD For-Sale Unstable PTGER4 15 41 CCCCCCCCOc1ccc([C@@H](CC(=O)OC)c2oc(CN3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)cc(=O)c2O)cc1 ZINC000217943158 KK In-Stock Unstable CHRNA4 25 40 Cc1cc([C@H](N)C(=O)O)cc(C)c1Br ZINC000217943209 CE For-Sale Unstable CACNA2D1 27 57 CS(=O)(=O)c1cc(Cl)cc(CC(=O)O)c1 ZINC000217943213 BD For-Sale Unstable PTGDR2 31 42 CC[C@@H](NC(=O)c1ccc(C)c([N+](=O)[O-])c1)c1ccc(C)c(C)c1 ZINC000217943218 EI In-Stock Unstable UTS2 47 32 O=C(N[C@@H]1CCC[C@@H]1CO)c1ccc2[nH]ccc2c1 ZINC000217943228 CE For-Sale Unstable SSTR3 29 40 Cn1cccc1[C@H](O)CCNS(=O)(=O)c1ccc(F)c(Cl)c1 ZINC000217943244 EE In-Stock Unstable TBXA2R 44 35 COc1cccc(/C=C/NC(=O)N2[C@@H](C)CCC[C@@H]2C)c1 ZINC000217943254 CH For-Sale Unstable MTNR1A 35 42 COc1cccc(/C=C/NC(=O)N2[C@@H](C)CCC[C@@H]2C)c1 ZINC000217943254 CH For-Sale Unstable MTNR1B 37 42 CN1CCN(c2ccc(C(=O)N[C@@]34C[C@@H]5C[C@@](C)(C[C@@](C)(C5)C3)C4)cc2[N+](=O)[O-])CC1 ZINC000217943269 IH In-Stock Unstable WDR5 38 44 CC[C@H](C)[C@H](C(=O)N1CCCC[C@H]1c1cccnc1)N1Cc2ccccc2C1=O ZINC000217943283 GI In-Stock Unstable GPBAR1 0 40 Cc1cc([C@@H](N)C(=O)O)cc(C)c1Br ZINC000217943294 CE For-Sale Unstable CACNA2D1 27 57 CC[C@H](NC(=O)c1ccc(C)c([N+](=O)[O-])c1)c1ccc(C)c(C)c1 ZINC000217943303 EI In-Stock Unstable UTS2 47 32 O=C(N[C@H]1CCC[C@@H]1CO)c1ccc2[nH]ccc2c1 ZINC000217943306 CE For-Sale Unstable SSTR3 29 40 Cn1cccc1[C@@H](O)CCNS(=O)(=O)c1ccc(F)c(Cl)c1 ZINC000217943320 EE In-Stock Unstable TBXA2R 44 35 Cc1ccc(N[C@H]2C[C@H](C)CC[C@H]2C(C)C)c([N+](=O)[O-])c1 ZINC000217943350 CJ For-Sale Unstable SERPINE1 40 41 Cc1ccc(N[C@H]2C[C@H](C)CC[C@H]2C(C)C)c([N+](=O)[O-])c1 ZINC000217943350 CJ For-Sale Unstable TRPM8 15 46 COc1cccc(/C=C/NC(=O)N2[C@@H](C)CCC[C@H]2C)c1 ZINC000217943352 CH For-Sale Unstable MTNR1A 35 42 COc1cccc(/C=C/NC(=O)N2[C@@H](C)CCC[C@H]2C)c1 ZINC000217943352 CH For-Sale Unstable MTNR1B 37 42 Cc1cccc(N2CCN(CC(=O)N[C@@H](C)Cc3cccnc3)CC2)c1 ZINC000217943356 FE In-Stock Unstable HTR1A 16 45 CCN(Cc1cccc(/C=C\C(=O)O)c1)Cc1cccs1 ZINC000217943362 DH For-Sale Unstable HCAR2 0 41 O=C(N[C@@H]1CCC[C@H]1CO)c1ccc2[nH]ccc2c1 ZINC000217943388 CE For-Sale Unstable SSTR3 29 40 COc1cccc(/C=C/NC(=O)N2[C@H](C)CCC[C@H]2C)c1 ZINC000217943431 CH For-Sale Unstable MTNR1A 35 42 COc1cccc(/C=C/NC(=O)N2[C@H](C)CCC[C@H]2C)c1 ZINC000217943431 CH For-Sale Unstable MTNR1B 37 42 Cc1ccc(N[C@H]2C[C@@H](C)CC[C@H]2C(C)C)c([N+](=O)[O-])c1 ZINC000217943437 CJ For-Sale Unstable SERPINE1 40 41 Cc1ccc(N[C@H]2C[C@@H](C)CC[C@H]2C(C)C)c([N+](=O)[O-])c1 ZINC000217943437 CJ For-Sale Unstable TRPM8 15 46 Cc1cccc(N2CCN(CC(=O)N[C@H](C)Cc3cccnc3)CC2)c1 ZINC000217943440 FE In-Stock Unstable HTR1A 16 45 O=C(N[C@H]1CCC[C@H]1CO)c1ccc2[nH]ccc2c1 ZINC000217943456 CE On-Demand Unstable SSTR3 28 40 CC1CCC(N(C)Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217943486 CH For-Sale Unstable PTGER2 47 49 CC1CCC(N(C)Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217943486 CH For-Sale Unstable PTGER4 23 49 CC1CCC(N(C)Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217943486 CH For-Sale Unstable PTGER3 17 49 CC1CCC(N(C)Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217943486 CH For-Sale Unstable PTGDR 0 45 Cc1noc2nc(C(C)C)cc(C(=O)Nc3ccc(S(=O)(=O)N4CCC(C)CC4)cc3)c12 ZINC000217943493 JI On-Demand Unstable TGM2 40 38 Cc1noc2nc(C(C)C)cc(C(=O)Nc3ccc(S(=O)(=O)N4CCC(C)CC4)cc3)c12 ZINC000217943493 JI On-Demand Unstable F13A1 58 38 Cc1noc2nc(C(C)C)cc(C(=O)Nc3ccc(S(=O)(=O)N4CCC(C)CC4)cc3)c12 ZINC000217943493 JI On-Demand Unstable MERTK 28 41 Cc1noc2nc(C(C)C)cc(C(=O)Nc3ccc(S(=O)(=O)N4CCC(C)CC4)cc3)c12 ZINC000217943493 JI On-Demand Unstable NAMPT 24 42 Cc1noc2nc(C(C)C)cc(C(=O)Nc3ccc(S(=O)(=O)N4CCC(C)CC4)cc3)c12 ZINC000217943493 JI On-Demand Unstable DDIT3 0 47 CCOc1ccc(/C=C2/CC(=O)NC2=O)cc1 ZINC000217943597 BD For-Sale Unstable HPGD 59 43 CCC(=O)c1ccc(OCc2cnn(-c3ccccc3)c2)cc1 ZINC000217943611 DI On-Demand Unstable SRD5A2 0 42 CCC(=O)c1ccc(OCc2cnn(-c3ccccc3)c2)cc1 ZINC000217943611 DI On-Demand Unstable GRM4 28 47 CC[C@@H](NC(=O)c1ccc(C)c([N+](=O)[O-])c1)c1ccc(OC)c(OC)c1 ZINC000217943622 FH In-Stock Unstable TAAR1 18 40 CC[C@@H](NC(=O)c1ccc(C)c([N+](=O)[O-])c1)c1ccc(OC)c(OC)c1 ZINC000217943622 FH In-Stock Unstable UTS2 43 34 O=C(c1ccncc1O)N1CCC(N2CCC(O)CC2)CC1 ZINC000217943681 DC In-Stock Unstable L3MBTL1 0 48 O=C(c1ccncc1O)N1CCC(N2CCC(O)CC2)CC1 ZINC000217943681 DC In-Stock Unstable L3MBTL3 81 48 O=C(c1ccncc1O)N1CCC(N2CCC(O)CC2)CC1 ZINC000217943681 DC In-Stock Unstable L3MBTL4 0 41 O=C(c1ccncc1O)N1CCC(N2CCC(O)CC2)CC1 ZINC000217943681 DC In-Stock Unstable MBTD1 0 45 O=C(c1ccncc1O)N1CCC(N2CCC(O)CC2)CC1 ZINC000217943681 DC In-Stock Unstable TP53BP1 0 48 CC(C)(C)OC(=O)N1CCCC[C@@H]1CNc1nccc(C(F)(F)F)n1 ZINC000217943690 FH On-Demand Unstable HCRTR1 15 41 CC[C@@H]1CCCN1Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217943712 CG For-Sale Unstable DRD2 40 40 CC[C@@H]1CCCN1Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217943712 CG For-Sale Unstable ACKR3 73 38 CC[C@H](NC(=O)c1ccc(C)c([N+](=O)[O-])c1)c1ccc(OC)c(OC)c1 ZINC000217943714 FH In-Stock Unstable TAAR1 18 40 CC[C@H](NC(=O)c1ccc(C)c([N+](=O)[O-])c1)c1ccc(OC)c(OC)c1 ZINC000217943714 FH In-Stock Unstable UTS2 43 34 NCNC(=O)Nc1ccccc1 ZINC000217943753 AC For-Sale Unstable CA2 24 49 NCNC(=O)Nc1ccccc1 ZINC000217943753 AC For-Sale Unstable LTA4H 15 40 NCNC(=O)Nc1ccccc1 ZINC000217943753 AC For-Sale Unstable CA1 61 43 NCNC(=O)Nc1ccccc1 ZINC000217943753 AC For-Sale Unstable CA4 19 53 NCNC(=O)Nc1ccccc1 ZINC000217943753 AC For-Sale Unstable EPHX2 20 64 NCNC(=O)Nc1ccccc1 ZINC000217943753 AC For-Sale Unstable F7 21 40 NCNC(=O)Nc1ccccc1 ZINC000217943753 AC For-Sale Unstable CA12 36 49 NCNC(=O)Nc1ccccc1 ZINC000217943753 AC For-Sale Unstable CA9 36 49 NCNC(=O)Nc1ccccc1 ZINC000217943753 AC For-Sale Unstable NCE103 47 49 NCNC(=O)Nc1ccccc1 ZINC000217943753 AC For-Sale Unstable MTCA1 41 50 NCNC(=O)Nc1ccccc1 ZINC000217943753 AC For-Sale Unstable P96878_MYCTU 52 50 NCNC(=O)Nc1ccccc1 ZINC000217943753 AC For-Sale Unstable NAMPT 30 41 NCNC(=O)Nc1ccccc1 ZINC000217943753 AC For-Sale Unstable KCNK3 42 33 CC(C)(C)OC(=O)N1CCCC[C@H]1CNc1nccc(C(F)(F)F)n1 ZINC000217943754 FH On-Demand Unstable HCRTR1 15 41 COc1ccc(OC)c(/C=C2/CC(=O)NC2=O)c1 ZINC000217943762 BD For-Sale Unstable CYP1B1 36 44 COc1ccc(OC)c(/C=C2/CC(=O)NC2=O)c1 ZINC000217943762 BD For-Sale Unstable CYP1A1 37 44 CCOC(=O)c1cnn(-c2cccc(F)c2)c1O ZINC000217943792 CD For-Sale Unstable HPD 36 42 CC[C@H]1CCCN1Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217943801 CG For-Sale Unstable DRD2 40 40 CC[C@H]1CCCN1Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217943801 CG For-Sale Unstable ACKR3 73 38 CC[C@@H](NC(=O)c1ccc(C)c([N+](=O)[O-])c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217943816 GG In-Stock Unstable COLA 55 32 CC[C@@H](NC(=O)c1ccc(C)c([N+](=O)[O-])c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217943816 GG In-Stock Unstable UTS2 41 32 CCN(CCO)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217943859 CD For-Sale Unstable MTNR1A 39 43 CCN(CCO)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217943859 CD For-Sale Unstable MTNR1B 40 43 CCN(CCO)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217943859 CD For-Sale Unstable ROCK2 16 40 CC[C@@H]1CCCN1Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217943903 CG For-Sale Unstable DRD2 44 42 CC[C@@H]1CCCN1Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217943903 CG For-Sale Unstable ACKR3 66 35 CC[C@H](NC(=O)c1ccc(C)c([N+](=O)[O-])c1)c1ccc(S(C)(=O)=O)cc1 ZINC000217943904 GG In-Stock Unstable COLA 53 32 NS(=O)(=O)c1cc(Cl)c(Cl)c(C(=O)OCCC2CC2)c1 ZINC000217943940 EF On-Demand Unstable CA2 15 43 NS(=O)(=O)c1cc(Cl)c(Cl)c(C(=O)OCCC2CC2)c1 ZINC000217943940 EF On-Demand Unstable CA4 17 43 NS(=O)(=O)c1cc(Cl)c(Cl)c(C(=O)OCCC2CC2)c1 ZINC000217943940 EF On-Demand Unstable Q5TU56_ANOGA 0 43 COc1cccc(/C=C/NC(=O)NCCCOC(C)C)c1 ZINC000217943971 CF For-Sale Unstable HRH2 25 41 COc1cccc(/C=C/NC(=O)NCCCOC(C)C)c1 ZINC000217943971 CF For-Sale Unstable MTNR1A 75 47 COc1cccc(/C=C/NC(=O)NCCCOC(C)C)c1 ZINC000217943971 CF For-Sale Unstable MTNR1B 73 47 CC[C@H]1CCCN1Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217943978 CG For-Sale Unstable DRD2 44 42 CC[C@H]1CCCN1Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217943978 CG For-Sale Unstable ACKR3 66 35 COc1cccc(-c2noc(CNC(=O)c3ccc(C)c([N+](=O)[O-])c3)n2)c1 ZINC000217944012 FF In-Stock Unstable DRD4 43 34 COc1cccc(-c2noc(CNC(=O)c3ccc(C)c([N+](=O)[O-])c3)n2)c1 ZINC000217944012 FF In-Stock Unstable TAAR1 27 44 O=C1C/C(=C\c2ccc(-c3cccnc3)o2)C(=O)N1 ZINC000217944035 CD For-Sale Unstable CYP11B2 15 44 O=C1C/C(=C\c2ccc(-c3cccnc3)o2)C(=O)N1 ZINC000217944035 CD For-Sale Unstable CYP2E1 38 42 O=C1C/C(=C\c2ccc(-c3cccnc3)o2)C(=O)N1 ZINC000217944035 CD For-Sale Unstable CYP2A6 31 49 COC(=O)C[C@H](c1ccc(OC)cc1)c1c(O)cc(C)oc1=O ZINC000217944064 DE In-Stock Unstable RORC 47 42 COc1cccc(/C=C/NC(=O)N(c2ccccc2)c2ccc(N)cc2)c1 ZINC000217944090 FJ For-Sale Unstable MTNR1A 22 46 COc1cccc(/C=C/NC(=O)N(c2ccccc2)c2ccc(N)cc2)c1 ZINC000217944090 FJ For-Sale Unstable MTNR1B 29 46 CC1CCN(Cc2ccc(/C=C\C(=O)O)cc2F)CC1 ZINC000217944102 CG For-Sale Unstable CCR2 40 42 CC1CCN(Cc2ccc(/C=C\C(=O)O)cc2F)CC1 ZINC000217944102 CG For-Sale Unstable GPR183 0 42 CNCCc1ccc(Br)cc1C(=O)O ZINC000217944116 CD For-Sale Unstable PRS 41 35 COc1ccc(-c2noc(CNC(=O)c3ccc(C)c([N+](=O)[O-])c3)n2)c(OC)c1 ZINC000217944120 GF In-Stock Unstable TAAR1 22 41 O=C(CNC(=O)c1cccc(Cl)c1)N[C@H]1CCC[C@H]1CO ZINC000217944153 DD On-Demand Unstable CCKBR 0 41 O=C(CNC(=O)c1cccc(Cl)c1)N[C@H]1CCC[C@H]1CO ZINC000217944153 DD On-Demand Unstable CACNA1I 41 33 COC(=O)C[C@@H](c1ccc(OC)cc1)c1c(O)cc(C)oc1=O ZINC000217944154 DE In-Stock Unstable RORC 47 42 COc1cccc(/C=C/NC(=O)Nc2ccc(Nc3ccccc3)cc2)c1 ZINC000217944190 FK For-Sale Unstable LPL 42 33 COc1cccc(/C=C/NC(=O)Nc2ccc(Nc3ccccc3)cc2)c1 ZINC000217944190 FK For-Sale Unstable MTNR1A 30 62 COc1cccc(/C=C/NC(=O)Nc2ccc(Nc3ccccc3)cc2)c1 ZINC000217944190 FK For-Sale Unstable MTNR1B 38 62 COc1cccc(/C=C/NC(=O)Nc2ccc(Nc3ccccc3)cc2)c1 ZINC000217944190 FK For-Sale Unstable TAAR1 28 40 COc1cccc(/C=C/NC(=O)Nc2ccc(Nc3ccccc3)cc2)c1 ZINC000217944190 FK For-Sale Unstable AKR1C3 47 48 COc1cccc(/C=C/NC(=O)Nc2ccc(Nc3ccccc3)cc2)c1 ZINC000217944190 FK For-Sale Unstable AKR1C2 66 39 Cn1cccc1[C@H](O)CCNS(=O)(=O)c1cc2c3c(c1)CCN3C(=O)CC2 ZINC000217944196 GD In-Stock Unstable CYP11B1 29 40 Cn1cccc1[C@H](O)CCNS(=O)(=O)c1cc2c3c(c1)CCN3C(=O)CC2 ZINC000217944196 GD In-Stock Unstable CYP11B2 29 40 CC1CCN(Cc2ccc(F)cc2/C=C\C(=O)O)CC1 ZINC000217944219 CG For-Sale Unstable SIGMAR1 24 42 CC1CCN(Cc2ccc(F)cc2/C=C\C(=O)O)CC1 ZINC000217944219 CG For-Sale Unstable CCR3 26 44 C[C@H](N)Cc1ccc(Br)cc1C(=O)O ZINC000217944232 CE For-Sale Unstable PRS 50 35 COc1ccc2[nH]c(=O)c([C@@H]3CC(=O)Oc4cc(OC)c(OC)c(OC)c43)cc2c1 ZINC000217944275 HG In-Stock Unstable TUBB2B 43 43 Cn1cccc1[C@@H](O)CCNS(=O)(=O)c1cc2c3c(c1)CCN3C(=O)CC2 ZINC000217944286 GD In-Stock Unstable CYP11B1 29 40 Cn1cccc1[C@@H](O)CCNS(=O)(=O)c1cc2c3c(c1)CCN3C(=O)CC2 ZINC000217944286 GD In-Stock Unstable CYP11B2 29 40 COc1cccc(/C=C/NC(=O)N2CCc3ccccc3C2)c1 ZINC000217944294 DG For-Sale Unstable DRD4 44 34 COc1cccc(/C=C/NC(=O)N2CCc3ccccc3C2)c1 ZINC000217944294 DG For-Sale Unstable MTNR1B 45 42 COc1cccc(/C=C/NC(=O)N2CCc3ccccc3C2)c1 ZINC000217944294 DG For-Sale Unstable HDAC6 33 43 CN(Cc1ccccc1/C=C\C(=O)O)c1ccccc1 ZINC000217944311 CG For-Sale Unstable PTGER2 52 52 CN(Cc1ccccc1/C=C\C(=O)O)c1ccccc1 ZINC000217944311 CG For-Sale Unstable PTGER4 22 43 CN(Cc1ccccc1/C=C\C(=O)O)c1ccccc1 ZINC000217944311 CG For-Sale Unstable PTGER3 19 52 C[C@@H](N)Cc1ccc(Br)cc1C(=O)O ZINC000217944326 CE For-Sale Unstable PRS 50 35 COc1ccc2[nH]c(=O)c([C@H]3CC(=O)Oc4cc(OC)c(OC)c(OC)c43)cc2c1 ZINC000217944349 HG In-Stock Unstable TUBB2B 43 43 N#Cc1cc(B(O)O)ccc1O ZINC000217944350 AA In-Stock Reactive AMPC 0 40 CN(Cc1ccc(/C=C\C(=O)O)cc1)c1ccccc1 ZINC000217944394 CG For-Sale Unstable PTGER2 31 40 CN(Cc1ccc(/C=C\C(=O)O)cc1)c1ccccc1 ZINC000217944394 CG For-Sale Unstable F3 23 41 CN(Cc1ccc(/C=C\C(=O)O)cc1)c1ccccc1 ZINC000217944394 CG For-Sale Unstable NR1H4 45 42 CN(Cc1ccc(/C=C\C(=O)O)cc1)c1ccccc1 ZINC000217944394 CG For-Sale Unstable HDAC1 15 40 COc1cccc(/C=C/NC(=O)Nc2cccc(C)n2)c1 ZINC000217944401 CG For-Sale Unstable CYP1B1 30 40 COc1cccc(/C=C/NC(=O)Nc2cccc(C)n2)c1 ZINC000217944401 CG For-Sale Unstable MTNR1A 28 42 COc1cccc(/C=C/NC(=O)Nc2cccc(C)n2)c1 ZINC000217944401 CG For-Sale Unstable MTNR1B 30 42 COc1cccc(/C=C/NC(=O)Nc2cccc(C)n2)c1 ZINC000217944401 CG For-Sale Unstable CYP1A1 17 40 COc1cccc(/C=C/NC(=O)Nc2cccc(C)n2)c1 ZINC000217944401 CG For-Sale Unstable GRM5 23 43 CC[C@@H](CO)Nc1ccc([N+](=O)[O-])cc1C(=O)O ZINC000217944426 CD For-Sale Unstable AKR1C3 15 47 CC[C@@H](CO)Nc1ccc([N+](=O)[O-])cc1C(=O)O ZINC000217944426 CD For-Sale Unstable AKR1C2 24 40 CN[C@@H](C)c1ccc(Br)cc1C(=O)O ZINC000217944441 CE For-Sale Unstable PRS 64 39 COc1cccc(-c2noc(CN(C)C(=O)c3ccc(C)c([N+](=O)[O-])c3)n2)c1 ZINC000217944471 GG In-Stock Unstable HSD17B2 22 46 CCOc1ccccc1/C(C)=C1/CC(=O)NC1=O ZINC000217944497 BD For-Sale Unstable HCN1 45 35 CCOc1ccccc1/C(C)=C1/CC(=O)NC1=O ZINC000217944497 BD For-Sale Unstable HCN4 45 35 CC[C@H](CO)Nc1ccc([N+](=O)[O-])cc1C(=O)O ZINC000217944514 CD For-Sale Unstable AKR1C3 15 47 CC[C@H](CO)Nc1ccc([N+](=O)[O-])cc1C(=O)O ZINC000217944514 CD For-Sale Unstable AKR1C2 24 40 COc1cccc(/C=C/NC(=O)NCCCCCO)c1 ZINC000217944519 CE For-Sale Unstable DRD4 41 31 COc1cccc(/C=C/NC(=O)NCCCCCO)c1 ZINC000217944519 CE For-Sale Unstable MTNR1A 81 49 COc1cccc(/C=C/NC(=O)NCCCCCO)c1 ZINC000217944519 CE For-Sale Unstable MTNR1B 76 49 CN[C@H](C)c1ccc(Br)cc1C(=O)O ZINC000217944524 CE For-Sale Unstable PRS 64 39 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1cc([N+](=O)[O-])ccc1Cl ZINC000217944562 DK For-Sale Unstable TRPM8 15 45 O=C1C/C(=C/c2cccc(Cl)c2)C(=O)N1 ZINC000217944582 BD For-Sale Unstable AKR1B1 15 40 CCCN(CCC)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217944585 CG For-Sale Unstable PTGER2 39 44 CCCN(CCC)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217944585 CG For-Sale Unstable PTGER4 22 44 CCCN(CCC)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217944585 CG For-Sale Unstable PTGER3 17 44 CCCN(CCC)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217944585 CG For-Sale Unstable AKR1B10 30 40 COc1cccc(/C=C/NC(=O)Nc2ccccn2)c1 ZINC000217944620 CF For-Sale Unstable CYP1B1 19 40 COc1cccc(/C=C/NC(=O)Nc2ccccn2)c1 ZINC000217944620 CF For-Sale Unstable KDR 15 40 COc1cccc(/C=C/NC(=O)Nc2ccccn2)c1 ZINC000217944620 CF For-Sale Unstable MTNR1A 26 43 COc1cccc(/C=C/NC(=O)Nc2ccccn2)c1 ZINC000217944620 CF For-Sale Unstable MTNR1B 33 43 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1cc([N+](=O)[O-])ccc1Cl ZINC000217944636 DK For-Sale Unstable TRPM8 15 45 O=C(CCCc1c[nH]c2ccccc12)N1CCCC[C@H]1c1cccnc1 ZINC000217944672 EJ In-Stock Unstable HTR1D 43 39 O=C(CCCc1c[nH]c2ccccc12)N1CCCC[C@H]1c1cccnc1 ZINC000217944672 EJ In-Stock Unstable PTAFR 21 41 O=C(CCCc1c[nH]c2ccccc12)N1CCCC[C@H]1c1cccnc1 ZINC000217944672 EJ In-Stock Unstable MC4R 42 42 O=C(CCCc1c[nH]c2ccccc12)N1CCCC[C@H]1c1cccnc1 ZINC000217944672 EJ In-Stock Unstable CCKAR 21 46 O=C(CCCc1c[nH]c2ccccc12)N1CCCC[C@H]1c1cccnc1 ZINC000217944672 EJ In-Stock Unstable COLA 114 41 O=C(CCCc1c[nH]c2ccccc12)N1CCCC[C@H]1c1cccnc1 ZINC000217944672 EJ In-Stock Unstable CPT1A 97 38 O=C(CCCc1c[nH]c2ccccc12)N1CCCC[C@H]1c1cccnc1 ZINC000217944672 EJ In-Stock Unstable PREP 46 36 O=C(CCCc1c[nH]c2ccccc12)N1CCCC[C@H]1c1cccnc1 ZINC000217944672 EJ In-Stock Unstable MC5R 30 43 O=C(CCCc1c[nH]c2ccccc12)N1CCCC[C@H]1c1cccnc1 ZINC000217944672 EJ In-Stock Unstable Q7YY07_CRYPV 54 34 O=C(CCCc1c[nH]c2ccccc12)N1CCCC[C@H]1c1cccnc1 ZINC000217944672 EJ In-Stock Unstable GPBAR1 0 41 Cc1ccc(C(=O)N(C)Cc2nc(-c3ccccc3Cl)no2)cc1[N+](=O)[O-] ZINC000217944707 GH In-Stock Unstable GPBAR1 24 41 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1cc([N+](=O)[O-])ccc1Cl ZINC000217944714 DK For-Sale Unstable TRPM8 15 45 COc1cccc(/C=C/NC(=O)Nc2cccnc2)c1 ZINC000217944738 CF For-Sale Unstable MTNR1A 24 45 COc1cccc(/C=C/NC(=O)Nc2cccnc2)c1 ZINC000217944738 CF For-Sale Unstable MTNR1B 29 45 C[C@H](N)Cc1ccc(C(=O)O)cc1Br ZINC000217944757 CE For-Sale Unstable HTR2B 17 45 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1cc([N+](=O)[O-])ccc1Cl ZINC000217944796 DK For-Sale Unstable TRPM8 15 45 CCOC(=O)c1sc(NS(=O)(=O)C2CCCC2)cc1C ZINC000217944819 DF For-Sale Unstable DHODH 18 41 CCOC(=O)c1sc(NS(=O)(=O)C2CCCC2)cc1C ZINC000217944819 DF For-Sale Unstable TLR4 15 40 CCCOc1ccc(/C=C2/CC(=O)NC2=O)cc1OC ZINC000217944829 CD For-Sale Unstable ESRRA 51 40 CCCOc1ccc(/C=C2/CC(=O)NC2=O)cc1OC ZINC000217944829 CD For-Sale Unstable HPGD 55 50 C[C@@H](N)Cc1ccc(C(=O)O)cc1Br ZINC000217944843 CE For-Sale Unstable HTR2B 17 45 CCN(CC)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217944853 BF For-Sale Unstable CYP1B1 34 43 CCN(CC)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217944853 BF For-Sale Unstable AHR 24 44 CCN(CC)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217944853 BF For-Sale Unstable MTNR1A 63 47 CCN(CC)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217944853 BF For-Sale Unstable MTNR1B 60 47 CCN(CC)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217944853 BF For-Sale Unstable CYP1A1 24 43 CCN(CC)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217944853 BF For-Sale Unstable ROCK2 18 40 Cc1ccc(C(=O)NCCCc2ccc(C(C)C)cc2)cc1[N+](=O)[O-] ZINC000217944927 EI In-Stock Unstable PTAFR 15 42 C[C@@H](O)CNc1ccc(C(=O)O)cc1[N+](=O)[O-] ZINC000217944944 BD For-Sale Unstable BDKRB1 0 43 C[C@@H](O)CNc1ccc(C(=O)O)cc1[N+](=O)[O-] ZINC000217944944 BD For-Sale Unstable COLA 40 31 C[C@@H](O)CNc1ccc(C(=O)O)cc1[N+](=O)[O-] ZINC000217944944 BD For-Sale Unstable AKR1C4 0 44 CC1(C)CN(Cc2ccccc2/C=C\C(=O)O)CCO1 ZINC000217944948 CE For-Sale Unstable PTGER2 38 42 CC1(C)CN(Cc2ccccc2/C=C\C(=O)O)CCO1 ZINC000217944948 CE For-Sale Unstable PTGER4 18 42 CC1(C)CN(Cc2ccccc2/C=C\C(=O)O)CCO1 ZINC000217944948 CE For-Sale Unstable PTGER3 18 42 CC1(C)CN(Cc2ccccc2/C=C\C(=O)O)CCO1 ZINC000217944948 CE For-Sale Unstable PTGDR 15 41 CNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217944962 BD For-Sale Unstable CYP1B1 49 45 CNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217944962 BD For-Sale Unstable AHR 26 48 CNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217944962 BD For-Sale Unstable MTNR1A 44 47 CNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217944962 BD For-Sale Unstable MTNR1B 34 54 C[C@H](O)CNc1ccc(C(=O)O)cc1[N+](=O)[O-] ZINC000217945026 BD For-Sale Unstable BDKRB1 0 43 C[C@H](O)CNc1ccc(C(=O)O)cc1[N+](=O)[O-] ZINC000217945026 BD For-Sale Unstable COLA 40 31 C[C@H](O)CNc1ccc(C(=O)O)cc1[N+](=O)[O-] ZINC000217945026 BD For-Sale Unstable AKR1C4 0 44 Cc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1[N+](=O)[O-] ZINC000217945043 FG In-Stock Unstable DRD4 43 35 Cc1ccc(C(=O)NCCCN2CCCc3ccccc32)cc1[N+](=O)[O-] ZINC000217945043 FG In-Stock Unstable AVPR2 39 44 COc1cccc(/C=C/NC(=O)NC(C)(C)CC(C)(C)C)c1 ZINC000217945089 DI For-Sale Unstable CYP1B1 19 41 COc1cccc(/C=C/NC(=O)NC(C)(C)CC(C)(C)C)c1 ZINC000217945089 DI For-Sale Unstable MTNR1A 42 43 COc1cccc(/C=C/NC(=O)NC(C)(C)CC(C)(C)C)c1 ZINC000217945089 DI For-Sale Unstable MTNR1B 44 43 COc1cccc(/C=C/NC(=O)NC(C)(C)CC(C)(C)C)c1 ZINC000217945089 DI For-Sale Unstable CYP1A1 18 41 C[C@@H](O)CNc1ccc([N+](=O)[O-])cc1C(=O)O ZINC000217945131 BD For-Sale Unstable AKR1C2 28 41 CC[C@H](C(=O)OC)[C@H](NC(=O)OC(C)(C)C)C(C)C ZINC000217945137 CF For-Sale Unstable PAPA1_CARPA 34 42 CC[C@H](C(=O)OC)[C@H](NC(=O)OC(C)(C)C)C(C)C ZINC000217945137 CF For-Sale Unstable CTSK 18 49 CC[C@H](C(=O)OC)[C@H](NC(=O)OC(C)(C)C)C(C)C ZINC000217945137 CF For-Sale Unstable PGA5 23 40 CCCOC(=O)c1ccc(NC(=O)c2cc(C(C)C)nc3onc(C)c23)cc1 ZINC000217945145 GI On-Demand Unstable F3 57 33 CN(CC(=O)N1CC(c2nc3ccccc3[nH]2)C1)Cc1cccnc1 ZINC000217945147 EE In-Stock Unstable SMO 30 40 COc1ccccc1OCC(=O)NCc1ccc(OC)c(OC)c1OC ZINC000217945157 FE In-Stock Unstable PDE4D 0 50 COc1ccccc1OCC(=O)NCc1ccc(OC)c(OC)c1OC ZINC000217945157 FE In-Stock Unstable SLC9A1 59 33 O=C(CCc1ccc(-n2cnnc2)cc1)N1CCCC[C@H]1c1cccnc1 ZINC000217945158 FG In-Stock Unstable CHRNA2 40 41 O=C(CCc1ccc(-n2cnnc2)cc1)N1CCCC[C@H]1c1cccnc1 ZINC000217945158 FG In-Stock Unstable PRCP 16 41 O=C(CCc1ccc(-n2cnnc2)cc1)N1CCCC[C@H]1c1cccnc1 ZINC000217945158 FG In-Stock Unstable CHRNA7 18 41 O=C(CCc1ccc(-n2cnnc2)cc1)N1CCCC[C@H]1c1cccnc1 ZINC000217945158 FG In-Stock Unstable COLA 111 42 O=C(CCc1ccc(-n2cnnc2)cc1)N1CCCC[C@H]1c1cccnc1 ZINC000217945158 FG In-Stock Unstable CPT1A 99 38 O=C(CCc1ccc(-n2cnnc2)cc1)N1CCCC[C@H]1c1cccnc1 ZINC000217945158 FG In-Stock Unstable C3AR1 43 40 O=C(CCc1ccc(-n2cnnc2)cc1)N1CCCC[C@H]1c1cccnc1 ZINC000217945158 FG In-Stock Unstable PREP 43 36 O=C(CCc1ccc(-n2cnnc2)cc1)N1CCCC[C@H]1c1cccnc1 ZINC000217945158 FG In-Stock Unstable CRTY 0 41 COc1ccc(CN2CC[C@@H](N)[C@@H](C)C2)cn1 ZINC000217945169 BD On-Demand Unstable PDE1C 17 44 C[C@H]1CN(C)[C@@H](C)C[C@@H]1NCCCn1ccnc1 ZINC000217945183 CD For-Sale Unstable TBXAS1 25 40 CC[C@@H](CO)NC(=O)N/C=C/c1cccc(OC)c1 ZINC000217945189 CD For-Sale Unstable MTNR1A 39 42 CC[C@@H](CO)NC(=O)N/C=C/c1cccc(OC)c1 ZINC000217945189 CD For-Sale Unstable MTNR1B 40 42 C[C@H](O)CNc1ccc([N+](=O)[O-])cc1C(=O)O ZINC000217945211 BD For-Sale Unstable AKR1C2 28 41 CC[C@@H](C(=O)OC)[C@H](NC(=O)OC(C)(C)C)C(C)C ZINC000217945214 CF For-Sale Unstable PAPA1_CARPA 34 42 CC[C@@H](C(=O)OC)[C@H](NC(=O)OC(C)(C)C)C(C)C ZINC000217945214 CF For-Sale Unstable CTSK 18 49 CC[C@@H](C(=O)OC)[C@H](NC(=O)OC(C)(C)C)C(C)C ZINC000217945214 CF For-Sale Unstable PGA5 23 40 COC(=O)c1ccccc1C(=O)N1C[C@H](Oc2ccccc2F)C[C@@H]1C(=O)OC ZINC000217945223 HE For-Sale Unstable HCRTR1 50 40 COC(=O)c1ccccc1C(=O)N1C[C@H](Oc2ccccc2F)C[C@@H]1C(=O)OC ZINC000217945223 HE For-Sale Unstable PLA2G4A 42 36 COC(=O)c1ccccc1C(=O)N1C[C@H](Oc2ccccc2F)C[C@@H]1C(=O)OC ZINC000217945223 HE For-Sale Unstable HCRTR2 55 40 CN[C@@H]1CCN(Cc2ccc(OC)nc2)C[C@@H]1C ZINC000217945236 BD For-Sale Unstable PDE1C 21 45 COc1ccc(N2C(=O)N[C@@H](CCC(=O)NCCc3c[nH]c4ccccc34)C2=O)cc1 ZINC000217945255 HF In-Stock Unstable ACHE 29 40 COc1ccc(N2C(=O)N[C@@H](CCC(=O)NCCc3c[nH]c4ccccc34)C2=O)cc1 ZINC000217945255 HF In-Stock Unstable MC4R 52 40 COc1ccc(N2C(=O)N[C@@H](CCC(=O)NCCc3c[nH]c4ccccc34)C2=O)cc1 ZINC000217945255 HF In-Stock Unstable NQO2 26 45 COc1ccc(N2C(=O)N[C@@H](CCC(=O)NCCc3c[nH]c4ccccc34)C2=O)cc1 ZINC000217945255 HF In-Stock Unstable CCKAR 47 44 COc1ccc(N2C(=O)N[C@@H](CCC(=O)NCCc3c[nH]c4ccccc34)C2=O)cc1 ZINC000217945255 HF In-Stock Unstable BCHE 16 45 COc1ccc(N2C(=O)N[C@@H](CCC(=O)NCCc3c[nH]c4ccccc34)C2=O)cc1 ZINC000217945255 HF In-Stock Unstable NMBR 25 40 COc1ccc(N2C(=O)N[C@@H](CCC(=O)NCCc3c[nH]c4ccccc34)C2=O)cc1 ZINC000217945255 HF In-Stock Unstable MC5R 35 43 COc1ccc(N2C(=O)N[C@@H](CCC(=O)NCCc3c[nH]c4ccccc34)C2=O)cc1 ZINC000217945255 HF In-Stock Unstable MTNR1A 65 52 COc1ccc(N2C(=O)N[C@@H](CCC(=O)NCCc3c[nH]c4ccccc34)C2=O)cc1 ZINC000217945255 HF In-Stock Unstable MTNR1B 49 45 COc1ccc(N2C(=O)N[C@@H](CCC(=O)NCCc3c[nH]c4ccccc34)C2=O)cc1 ZINC000217945255 HF In-Stock Unstable CCKBR 42 40 COc1ccc(N2C(=O)N[C@@H](CCC(=O)NCCc3c[nH]c4ccccc34)C2=O)cc1 ZINC000217945255 HF In-Stock Unstable GHSR 44 39 COc1ccc(N2C(=O)N[C@@H](CCC(=O)NCCc3c[nH]c4ccccc34)C2=O)cc1 ZINC000217945255 HF In-Stock Unstable AANAT 45 32 COc1ccccc1OCC(=O)NCc1ccc(OC(C)C)c(OC)c1 ZINC000217945258 FG In-Stock Unstable HCRTR1 18 42 COc1ccccc1OCC(=O)NCc1ccc(OC(C)C)c(OC)c1 ZINC000217945258 FG In-Stock Unstable TRPV1 27 45 COc1ccccc1OCC(=O)NCc1ccc(OC(C)C)c(OC)c1 ZINC000217945258 FG In-Stock Unstable PDE6A 42 32 COc1ccccc1OCC(=O)NCc1ccc(OC(C)C)c(OC)c1 ZINC000217945258 FG In-Stock Unstable ABCB1 24 41 COc1ccccc1OCC(=O)NCc1ccc(OC(C)C)c(OC)c1 ZINC000217945258 FG In-Stock Unstable MT-ND1 25 42 COc1ccccc1OCC(=O)NCc1ccc(OC(C)C)c(OC)c1 ZINC000217945258 FG In-Stock Unstable ABCG2 24 41 COc1ccccc1OCC(=O)NCc1ccc(OC(C)C)c(OC)c1 ZINC000217945258 FG In-Stock Unstable ENPP1 40 31 COc1ccccc1OCC(=O)NCc1ccc(OC(C)C)c(OC)c1 ZINC000217945258 FG In-Stock Unstable DRTS_TRYCR 48 33 COc1ccccc1OCC(=O)NCc1ccc(OC(C)C)c(OC)c1 ZINC000217945258 FG In-Stock Unstable CAN2 0 40 COc1ccccc1OCC(=O)NCc1ccc(OC(C)C)c(OC)c1 ZINC000217945258 FG In-Stock Unstable KCNK3 41 34 CC[C@H](CO)NC(=O)N/C=C/c1cccc(OC)c1 ZINC000217945261 CD For-Sale Unstable MTNR1A 39 42 CC[C@H](CO)NC(=O)N/C=C/c1cccc(OC)c1 ZINC000217945261 CD For-Sale Unstable MTNR1B 40 42 COC(=O)c1ccccc1C(=O)N1C[C@@H](Oc2ccccc2F)C[C@@H]1C(=O)OC ZINC000217945309 HE For-Sale Unstable HCRTR1 50 40 COC(=O)c1ccccc1C(=O)N1C[C@@H](Oc2ccccc2F)C[C@@H]1C(=O)OC ZINC000217945309 HE For-Sale Unstable PLA2G4A 42 36 COC(=O)c1ccccc1C(=O)N1C[C@@H](Oc2ccccc2F)C[C@@H]1C(=O)OC ZINC000217945309 HE For-Sale Unstable HCRTR2 55 40 C[C@@H](O)CNc1ccc([N+](=O)[O-])c(C(=O)O)c1 ZINC000217945310 BD On-Demand Unstable COLA 54 31 C[C@@H](O)CNc1ccc([N+](=O)[O-])c(C(=O)O)c1 ZINC000217945310 BD On-Demand Unstable AADAC 0 42 C[C@@H]1NCc2ccccc2[C@@H](c2ccccc2)[C@@H]1C ZINC000217945313 CH For-Sale Unstable PRCP 0 42 C[C@]1(CF)C[C@H](O)c2ccc(Cl)cc2O1 ZINC000217945356 BF For-Sale Unstable ABCC9 42 32 N#C[C@@H]1CNCCN1C[C@@H]1COc2ccccc2O1 ZINC000217945365 CC For-Sale Unstable ADRA2B 20 43 C=CCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217945376 BE For-Sale Unstable DRD4 40 30 C=CCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217945376 BE For-Sale Unstable CYP1B1 20 41 C=CCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217945376 BE For-Sale Unstable MTNR1A 70 45 C=CCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217945376 BE For-Sale Unstable MTNR1B 67 45 C=CCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217945376 BE For-Sale Unstable CYP1A1 18 41 COc1ccccc1OCC(=O)NCCCc1ccc(Cl)cc1 ZINC000217945391 EG In-Stock Unstable DRD2 18 42 COc1ccccc1OCC(=O)NCCCc1ccc(Cl)cc1 ZINC000217945391 EG In-Stock Unstable DRD3 27 42 COc1ccccc1OCC(=O)NCCCc1ccc(Cl)cc1 ZINC000217945391 EG In-Stock Unstable SCNN1A 64 36 COc1ccccc1OCC(=O)NCCCc1ccc(Cl)cc1 ZINC000217945391 EG In-Stock Unstable CYSP_TRYCR 0 40 COc1ccccc1OCC(=O)NCCCc1ccc(Cl)cc1 ZINC000217945391 EG In-Stock Unstable MTNR1B 25 49 COc1ccccc1OCC(=O)NCCCc1ccc(Cl)cc1 ZINC000217945391 EG In-Stock Unstable SCN5A 0 43 COc1ccccc1OCC(=O)NCCCc1ccc(Cl)cc1 ZINC000217945391 EG In-Stock Unstable NCE103 20 42 COc1ccccc1OCC(=O)NCCCc1ccc(Cl)cc1 ZINC000217945391 EG In-Stock Unstable CRTM 46 44 COc1ccccc1OCC(=O)NCCCc1ccc(Cl)cc1 ZINC000217945391 EG In-Stock Unstable P96878_MYCTU 17 42 COc1ccccc1OCC(=O)NCCCc1ccc(Cl)cc1 ZINC000217945391 EG In-Stock Unstable CAN2 0 42 COC(=O)c1ccccc1C(=O)N1C[C@H](Oc2ccccc2F)C[C@H]1C(=O)OC ZINC000217945392 HE For-Sale Unstable HCRTR1 50 40 COC(=O)c1ccccc1C(=O)N1C[C@H](Oc2ccccc2F)C[C@H]1C(=O)OC ZINC000217945392 HE For-Sale Unstable PLA2G4A 42 36 COC(=O)c1ccccc1C(=O)N1C[C@H](Oc2ccccc2F)C[C@H]1C(=O)OC ZINC000217945392 HE For-Sale Unstable HCRTR2 55 40 C[C@H](O)CNc1ccc([N+](=O)[O-])c(C(=O)O)c1 ZINC000217945394 BD On-Demand Unstable COLA 54 31 C[C@H](O)CNc1ccc([N+](=O)[O-])c(C(=O)O)c1 ZINC000217945394 BD On-Demand Unstable AADAC 0 42 C[C@@H]1[C@@H](C)NCc2ccccc2[C@H]1c1ccccc1 ZINC000217945401 CH For-Sale Unstable PRCP 0 42 O=C(NC[C@@H](c1cccnc1)N1CCOCC1)c1ncccc1O ZINC000217945411 EC In-Stock Unstable KCNA5 37 42 Cc1ccc(/C=C\C(=O)CCl)cc1 ZINC000217945421 AF For-Sale Unstable 17HSDCL 41 33 Cc1ccc(/C=C\C(=O)CCl)cc1 ZINC000217945421 AF For-Sale Unstable SSSIM 16 50 Cc1ccc(/C=C\C(=O)CCl)cc1 ZINC000217945421 AF For-Sale Unstable GPR183 0 43 O=C(O)C[C@@H]1CCCN1C(=O)[C@@H]1C[C@@H](O)CN1 ZINC000217945435 BB For-Sale Unstable DPP4 25 42 COC(=O)c1ccccc1C(=O)N1C[C@@H](Oc2ccccc2F)C[C@H]1C(=O)OC ZINC000217945472 HE For-Sale Unstable HCRTR1 50 40 COC(=O)c1ccccc1C(=O)N1C[C@@H](Oc2ccccc2F)C[C@H]1C(=O)OC ZINC000217945472 HE For-Sale Unstable PLA2G4A 42 36 COC(=O)c1ccccc1C(=O)N1C[C@@H](Oc2ccccc2F)C[C@H]1C(=O)OC ZINC000217945472 HE For-Sale Unstable HCRTR2 55 40 COc1cccc(/C=C/NC(=O)N(C(C)=O)c2cccc(N)c2)c1 ZINC000217945486 EG For-Sale Unstable MTNR1A 21 44 COc1cccc(/C=C/NC(=O)N(C(C)=O)c2cccc(N)c2)c1 ZINC000217945486 EG For-Sale Unstable MTNR1B 26 44 O=C(NC[C@H](c1cccnc1)N1CCOCC1)c1ncccc1O ZINC000217945490 EC In-Stock Unstable KCNA5 37 42 COc1ccc2nc(C)cc(OCc3cccc(C#N)c3)c2c1 ZINC000217945491 DI On-Demand Unstable MAOB 20 46 COc1ccc2nc(C)cc(OCc3cccc(C#N)c3)c2c1 ZINC000217945491 DI On-Demand Unstable CYP2C8 15 40 COc1ccc2nc(C)cc(OCc3cccc(C#N)c3)c2c1 ZINC000217945491 DI On-Demand Unstable GRM5 16 40 COc1ccc(/C=C\C(=O)CCl)cc1OC ZINC000217945497 BF For-Sale Unstable CYP1B1 49 50 COc1ccc(/C=C\C(=O)CCl)cc1OC ZINC000217945497 BF For-Sale Unstable CA7 0 51 COc1ccc(/C=C\C(=O)CCl)cc1OC ZINC000217945497 BF For-Sale Unstable APP 22 44 COc1ccc(/C=C\C(=O)CCl)cc1OC ZINC000217945497 BF For-Sale Unstable CA14 0 51 COc1ccc(/C=C\C(=O)CCl)cc1OC ZINC000217945497 BF For-Sale Unstable CYP1A1 44 50 COc1ccc(/C=C\C(=O)CCl)cc1OC ZINC000217945497 BF For-Sale Unstable TUBB1 64 45 COc1ccc(/C=C\C(=O)CCl)cc1OC ZINC000217945497 BF For-Sale Unstable PTPA 0 49 COc1ccc(/C=C\C(=O)CCl)cc1OC ZINC000217945497 BF For-Sale Unstable ABCG2 23 55 COc1ccc(/C=C\C(=O)CCl)cc1OC ZINC000217945497 BF For-Sale Unstable NFE2L2 0 48 COc1ccc(/C=C\C(=O)CCl)cc1OC ZINC000217945497 BF For-Sale Unstable CYSP_PLAFA 50 49 COc1ccccc1OCC(=O)NCCCc1ccc(F)cc1 ZINC000217945503 DF In-Stock Unstable HTR1A 15 44 COc1ccccc1OCC(=O)NCCCc1ccc(F)cc1 ZINC000217945503 DF In-Stock Unstable DRD2 21 43 COc1ccccc1OCC(=O)NCCCc1ccc(F)cc1 ZINC000217945503 DF In-Stock Unstable DRD1 0 41 COc1ccccc1OCC(=O)NCCCc1ccc(F)cc1 ZINC000217945503 DF In-Stock Unstable CYSP_TRYCR 0 43 COc1ccccc1OCC(=O)NCCCc1ccc(F)cc1 ZINC000217945503 DF In-Stock Unstable MTNR1B 29 50 COc1ccccc1OCC(=O)NCCCc1ccc(F)cc1 ZINC000217945503 DF In-Stock Unstable SCN5A 0 44 COc1ccccc1OCC(=O)NCCCc1ccc(F)cc1 ZINC000217945503 DF In-Stock Unstable CRTM 44 45 COc1ccccc1OCC(=O)NCCCc1ccc(F)cc1 ZINC000217945503 DF In-Stock Unstable AP2S1 0 40 O=C(O)C[C@H]1CCCN1C(=O)[C@@H]1C[C@@H](O)CN1 ZINC000217945525 BB For-Sale Unstable DPP4 25 42 O=C(O)C[C@@H]1CCCN1C(=O)[C@H]1C[C@@H](O)CN1 ZINC000217945577 BB For-Sale Unstable DPP4 25 42 COc1cccc(/C=C/NC(=O)Nc2cccc(NC(C)=O)c2)c1 ZINC000217945605 EG For-Sale Unstable CYP1B1 26 41 COc1cccc(/C=C/NC(=O)Nc2cccc(NC(C)=O)c2)c1 ZINC000217945605 EG For-Sale Unstable MTNR1A 40 56 COc1cccc(/C=C/NC(=O)Nc2cccc(NC(C)=O)c2)c1 ZINC000217945605 EG For-Sale Unstable MTNR1B 42 56 COc1cccc(/C=C/NC(=O)Nc2cccc(NC(C)=O)c2)c1 ZINC000217945605 EG For-Sale Unstable CYP1A1 18 41 COc1cccc(/C=C/NC(=O)Nc2cccc(NC(C)=O)c2)c1 ZINC000217945605 EG For-Sale Unstable TAAR1 31 44 COc1cccc(/C=C/NC(=O)Nc2cccc(NC(C)=O)c2)c1 ZINC000217945605 EG For-Sale Unstable AKR1C3 17 40 COc1cccc(/C=C/NC(=O)Nc2cccc(NC(C)=O)c2)c1 ZINC000217945605 EG For-Sale Unstable KCNK3 53 47 COc1cccc(/C=C/NC(=O)Nc2cccc(NC(C)=O)c2)c1 ZINC000217945605 EG For-Sale Unstable KCNK9 41 38 COc1ccc2nc(C)cc(OCC(=O)N[C@@H](C)c3ccc(Cl)cc3)c2c1 ZINC000217945610 GI On-Demand Unstable PTGS1 20 48 COc1ccc2nc(C)cc(OCC(=O)N[C@@H](C)c3ccc(Cl)cc3)c2c1 ZINC000217945610 GI On-Demand Unstable PTGS2 43 48 COc1ccc2nc(C)cc(OCC(=O)N[C@@H](C)c3ccc(Cl)cc3)c2c1 ZINC000217945610 GI On-Demand Unstable ACACA 48 38 COc1ccccc1CCCNC(=O)COc1ccccc1OC ZINC000217945623 EF In-Stock Unstable HTR1A 15 42 COc1ccccc1CCCNC(=O)COc1ccccc1OC ZINC000217945623 EF In-Stock Unstable DRD2 20 41 COc1ccccc1CCCNC(=O)COc1ccccc1OC ZINC000217945623 EF In-Stock Unstable ADRA1D 15 40 COc1ccccc1CCCNC(=O)COc1ccccc1OC ZINC000217945623 EF In-Stock Unstable CYSP_TRYCR 0 40 COc1ccccc1CCCNC(=O)COc1ccccc1OC ZINC000217945623 EF In-Stock Unstable MTNR1A 60 43 COc1ccccc1CCCNC(=O)COc1ccccc1OC ZINC000217945623 EF In-Stock Unstable MTNR1B 55 48 COc1ccccc1CCCNC(=O)COc1ccccc1OC ZINC000217945623 EF In-Stock Unstable GPM3 0 54 COc1ccccc1CCCNC(=O)COc1ccccc1OC ZINC000217945623 EF In-Stock Unstable CRTM 40 37 COc1ccccc1CCCNC(=O)COc1ccccc1OC ZINC000217945623 EF In-Stock Unstable MBTPS1 41 35 O=C(O)C[C@H]1CCCN1C(=O)[C@H]1C[C@@H](O)CN1 ZINC000217945645 BB For-Sale Unstable DPP4 25 42 COc1ccc2nc(C)cc(OCC(=O)N[C@H](C)c3ccc(Cl)cc3)c2c1 ZINC000217945688 GI On-Demand Unstable PTGS1 20 48 COc1ccc2nc(C)cc(OCC(=O)N[C@H](C)c3ccc(Cl)cc3)c2c1 ZINC000217945688 GI On-Demand Unstable PTGS2 43 48 COc1ccc2nc(C)cc(OCC(=O)N[C@H](C)c3ccc(Cl)cc3)c2c1 ZINC000217945688 GI On-Demand Unstable ACACA 48 38 COc1cccc(/C=C/NC(=O)N(C)CCO)c1 ZINC000217945710 CD For-Sale Unstable MTNR1A 42 44 COc1cccc(/C=C/NC(=O)N(C)CCO)c1 ZINC000217945710 CD For-Sale Unstable MTNR1B 42 44 COc1ccc(/C=C\C(=O)O)cc1CN1CCC[C@@H]1CO ZINC000217945718 CD For-Sale Unstable DRD2 39 40 COc1ccc(/C=C\C(=O)O)cc1CN1CCC[C@@H]1CO ZINC000217945718 CD For-Sale Unstable ACKR3 73 38 O=S(=O)(Cl)c1ccc2c(c1)CC[C@H](F)C2 ZINC000217945719 BE For-Sale Unstable CA7 27 43 O=S(=O)(Cl)c1ccc2c(c1)CC[C@H](F)C2 ZINC000217945719 BE For-Sale Unstable CA14 15 43 COc1ccc(OC[C@@H](C)NC(=O)COc2ccccc2OC)cc1 ZINC000217945738 EF In-Stock Unstable SDH1 0 43 COc1ccc(OC[C@@H](C)NC(=O)COc2ccccc2OC)cc1 ZINC000217945738 EF In-Stock Unstable CAPN2 33 41 COc1ccc2nc(C)cc(OCC(=O)NC3CCC(C)CC3)c2c1 ZINC000217945784 EH On-Demand Unstable AVPR1B 21 42 COc1ccc2nc(C)cc(OCC(=O)NC3CCC(C)CC3)c2c1 ZINC000217945784 EH On-Demand Unstable ADAM17 57 35 COc1ccc2nc(C)cc(OCC(=O)NC3CCC(C)CC3)c2c1 ZINC000217945784 EH On-Demand Unstable MTNR1A 39 40 COc1ccc2nc(C)cc(OCC(=O)NC3CCC(C)CC3)c2c1 ZINC000217945784 EH On-Demand Unstable MTNR1B 28 40 COc1ccc2nc(C)cc(OCC(=O)NC3CCC(C)CC3)c2c1 ZINC000217945784 EH On-Demand Unstable TNKS 46 32 O=S(=O)(Cl)c1ccc2c(c1)CC[C@@H](F)C2 ZINC000217945788 BE For-Sale Unstable CA7 27 43 O=S(=O)(Cl)c1ccc2c(c1)CC[C@@H](F)C2 ZINC000217945788 BE For-Sale Unstable CA14 15 43 COc1ccc(OC[C@H](C)NC(=O)COc2ccccc2OC)cc1 ZINC000217945817 EF In-Stock Unstable SDH1 0 43 COc1ccc(OC[C@H](C)NC(=O)COc2ccccc2OC)cc1 ZINC000217945817 EF In-Stock Unstable CAPN2 33 41 CC1CCC(N(C)Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217945829 CH For-Sale Unstable PTGER2 24 41 CC(C)C[C@H](NC(=O)CCc1cn(C)c2ccccc12)c1nc2ccccc2[nH]1 ZINC000217945850 GJ In-Stock Unstable EDNRA 29 46 COc1ccc2nc(C)cc(OCC(=O)N(C)Cc3ccc(F)cc3)c2c1 ZINC000217945875 FH On-Demand Unstable MTTP 41 34 COc1ccc2nc(C)cc(OCC(=O)N(C)Cc3ccc(F)cc3)c2c1 ZINC000217945875 FH On-Demand Unstable ACAT 54 42 O=S(=O)(Cl)c1ccc2c(c1)C[C@H](F)CC2 ZINC000217945900 BE For-Sale Unstable CA7 27 43 O=S(=O)(Cl)c1ccc2c(c1)C[C@H](F)CC2 ZINC000217945900 BE For-Sale Unstable CA14 15 43 CC1(C)COCCN1Cc1ccccc1/C=C\C(=O)O ZINC000217945918 CE For-Sale Unstable PTGER2 42 42 CC1(C)COCCN1Cc1ccccc1/C=C\C(=O)O ZINC000217945918 CE For-Sale Unstable PTGER4 19 42 CC1(C)COCCN1Cc1ccccc1/C=C\C(=O)O ZINC000217945918 CE For-Sale Unstable PTGER3 18 42 CC1(C)COCCN1Cc1ccccc1/C=C\C(=O)O ZINC000217945918 CE For-Sale Unstable PTGDR 15 41 CC[C@@H]1NCc2ccccc2[C@H](c2ccccc2)[C@@H]1C ZINC000217945920 CI For-Sale Unstable PRCP 50 38 COc1ccccc1OCC(=O)Nc1ccccc1C(=O)c1ccccc1 ZINC000217945924 FH In-Stock Unstable KCNA3 22 41 COc1ccccc1OCC(=O)Nc1ccccc1C(=O)c1ccccc1 ZINC000217945924 FH In-Stock Unstable ABCB1 0 42 COc1ccccc1OCC(=O)Nc1ccccc1C(=O)c1ccccc1 ZINC000217945924 FH In-Stock Unstable KCNK3 45 38 COc1ccccc1OCC(=O)Nc1ccccc1C(=O)c1ccccc1 ZINC000217945924 FH In-Stock Unstable FAS 29 42 COC(=O)C[C@@H]1c2cccnc2Oc2cc(O)c3c(=O)cc(-c4ccc(OC)c(O)c4)oc3c21 ZINC000217945958 JI In-Stock Unstable AKR1B1 0 43 COC(=O)C[C@@H]1c2cccnc2Oc2cc(O)c3c(=O)cc(-c4ccc(OC)c(O)c4)oc3c21 ZINC000217945958 JI In-Stock Unstable CYP1B1 54 43 COC(=O)C[C@@H]1c2cccnc2Oc2cc(O)c3c(=O)cc(-c4ccc(OC)c(O)c4)oc3c21 ZINC000217945958 JI In-Stock Unstable CYP1A1 44 43 O=C(/C=C\c1c[nH]c2cc([N+](=O)[O-])ccc12)CCl ZINC000217945975 CF For-Sale Unstable TDO2 0 48 O=S(=O)(Cl)c1ccc2c(c1)C[C@@H](F)CC2 ZINC000217945988 BE For-Sale Unstable CA7 27 43 O=S(=O)(Cl)c1ccc2c(c1)C[C@@H](F)CC2 ZINC000217945988 BE For-Sale Unstable CA14 15 43 COc1ccc2nc(C)cc(OCC(=O)N[C@@H](C)c3ccccc3OC)c2c1 ZINC000217945997 GH On-Demand Unstable ADAM17 55 35 COc1ccc2nc(C)cc(OCC(=O)N[C@@H](C)c3ccccc3OC)c2c1 ZINC000217945997 GH On-Demand Unstable MTNR1A 46 39 COc1ccc2nc(C)cc(OCC(=O)N[C@@H](C)c3ccccc3OC)c2c1 ZINC000217945997 GH On-Demand Unstable MTNR1B 44 39 COc1ccc2nc(C)cc(OCC(=O)N[C@@H](C)c3ccccc3OC)c2c1 ZINC000217945997 GH On-Demand Unstable PDE10A 17 44 COc1ccc2nc(C)cc(OCC(=O)N[C@@H](C)c3ccccc3OC)c2c1 ZINC000217945997 GH On-Demand Unstable ISPD 0 40 CC[C@H]1NCc2ccccc2[C@H](c2ccccc2)[C@@H]1C ZINC000217946014 CI For-Sale Unstable PRCP 50 38 COc1ccccc1OCC(=O)NCCCc1cccc(OC(C)C)c1 ZINC000217946026 FH In-Stock Unstable HRH2 26 41 COc1ccccc1OCC(=O)NCCCc1cccc(OC(C)C)c1 ZINC000217946026 FH In-Stock Unstable FDFT1 19 50 COc1ccccc1OCC(=O)NCCCc1cccc(OC(C)C)c1 ZINC000217946026 FH In-Stock Unstable MTNR1A 51 48 COc1ccccc1OCC(=O)NCCCc1cccc(OC(C)C)c1 ZINC000217946026 FH In-Stock Unstable MTNR1B 45 49 COc1ccccc1OCC(=O)NCCCc1cccc(OC(C)C)c1 ZINC000217946026 FH In-Stock Unstable AMP1_PLAFQ 24 43 COc1ccccc1OCC(=O)NCCCc1cccc(OC(C)C)c1 ZINC000217946026 FH In-Stock Unstable POLG_WNV 47 37 COc1ccccc1OCC(=O)NCCCc1cccc(OC(C)C)c1 ZINC000217946026 FH In-Stock Unstable CRTM 79 50 COc1ccccc1OCC(=O)NCCCc1cccc(OC(C)C)c1 ZINC000217946026 FH In-Stock Unstable PDS 45 38 COC(=O)C[C@H]1c2cccnc2Oc2cc(O)c3c(=O)cc(-c4ccc(OC)c(O)c4)oc3c21 ZINC000217946039 JI In-Stock Unstable AKR1B1 0 43 COC(=O)C[C@H]1c2cccnc2Oc2cc(O)c3c(=O)cc(-c4ccc(OC)c(O)c4)oc3c21 ZINC000217946039 JI In-Stock Unstable CYP1B1 54 43 COC(=O)C[C@H]1c2cccnc2Oc2cc(O)c3c(=O)cc(-c4ccc(OC)c(O)c4)oc3c21 ZINC000217946039 JI In-Stock Unstable CYP1A1 44 43 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1cc([N+](=O)[O-])ccc1F ZINC000217946048 CJ For-Sale Unstable TRPM8 16 45 COc1ccc2nc(C)cc(OCC(=O)N[C@H](C)c3ccccc3OC)c2c1 ZINC000217946092 GH On-Demand Unstable ADAM17 55 35 COc1ccc2nc(C)cc(OCC(=O)N[C@H](C)c3ccccc3OC)c2c1 ZINC000217946092 GH On-Demand Unstable MTNR1A 46 39 COc1ccc2nc(C)cc(OCC(=O)N[C@H](C)c3ccccc3OC)c2c1 ZINC000217946092 GH On-Demand Unstable MTNR1B 44 39 COc1ccc2nc(C)cc(OCC(=O)N[C@H](C)c3ccccc3OC)c2c1 ZINC000217946092 GH On-Demand Unstable PDE10A 17 44 COc1ccc2nc(C)cc(OCC(=O)N[C@H](C)c3ccccc3OC)c2c1 ZINC000217946092 GH On-Demand Unstable ISPD 0 40 O=S(=O)(Cl)c1ccc2c(c1)[C@H](F)CCC2 ZINC000217946095 BF For-Sale Unstable HTR6 42 36 COC(=O)c1ccc(N[C@@H]2C[C@@H](C)N(C)C[C@@H]2C)cc1 ZINC000217946102 CF For-Sale Unstable BRD2 19 40 COC(=O)c1ccc(N[C@@H]2C[C@@H](C)N(C)C[C@@H]2C)cc1 ZINC000217946102 CF For-Sale Unstable BRD3 23 41 CC[C@@H]1CCCN1Cc1ccc(/C=C\C(=O)O)cc1F ZINC000217946116 CG For-Sale Unstable ACKR3 55 31 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1cc([N+](=O)[O-])ccc1F ZINC000217946129 CJ For-Sale Unstable TRPM8 16 45 COc1ccccc1OCC(=O)NCCCc1ccc(OC(C)C)cc1 ZINC000217946131 FH In-Stock Unstable SCN2A 15 40 COc1ccccc1OCC(=O)NCCCc1ccc(OC(C)C)cc1 ZINC000217946131 FH In-Stock Unstable MTNR1A 37 40 COc1ccccc1OCC(=O)NCCCc1ccc(OC(C)C)cc1 ZINC000217946131 FH In-Stock Unstable MTNR1B 29 46 COc1ccccc1OCC(=O)NCCCc1ccc(OC(C)C)cc1 ZINC000217946131 FH In-Stock Unstable CRTM 44 41 COc1ccc(/C=C\c2csc(N)n2)cc1OC ZINC000217946155 CF For-Sale Unstable CYP1B1 42 50 COc1ccc(/C=C\c2csc(N)n2)cc1OC ZINC000217946155 CF For-Sale Unstable CYP1A1 42 50 COc1ccc(/C=C\c2csc(N)n2)cc1OC ZINC000217946155 CF For-Sale Unstable TUBB1 40 39 COc1ccc(/C=C\c2csc(N)n2)cc1OC ZINC000217946155 CF For-Sale Unstable CAMK2A 15 40 COC(=O)c1ccc(N[C@H]2C[C@@H](C)N(C)C[C@@H]2C)cc1 ZINC000217946174 CF For-Sale Unstable BRD2 19 40 COC(=O)c1ccc(N[C@H]2C[C@@H](C)N(C)C[C@@H]2C)cc1 ZINC000217946174 CF For-Sale Unstable BRD3 23 41 O=S(=O)(Cl)c1ccc2c(c1)[C@@H](F)CCC2 ZINC000217946178 BF For-Sale Unstable HTR6 42 36 CC[C@H]1CCCN1Cc1ccc(/C=C\C(=O)O)cc1F ZINC000217946189 CG For-Sale Unstable ACKR3 55 31 CCOC(=O)c1cnn(-c2ccccc2OC)c1O ZINC000217946200 CD For-Sale Unstable HPD 32 44 CCOC(=O)c1cnn(-c2ccccc2OC)c1O ZINC000217946200 CD For-Sale Unstable DHFR-TS 0 40 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1cc([N+](=O)[O-])ccc1F ZINC000217946205 CJ For-Sale Unstable TRPM8 16 45 COC(=O)c1ccc(N[C@@H]2C[C@H](C)N(C)C[C@@H]2C)cc1 ZINC000217946251 CF For-Sale Unstable BRD2 19 40 COC(=O)c1ccc(N[C@@H]2C[C@H](C)N(C)C[C@@H]2C)cc1 ZINC000217946251 CF For-Sale Unstable BRD3 23 41 CCOc1ccc(CCCNC(=O)COc2ccccc2OC)cc1 ZINC000217946266 EG In-Stock Unstable DRD2 15 41 CCOc1ccc(CCCNC(=O)COc2ccccc2OC)cc1 ZINC000217946266 EG In-Stock Unstable SCN2A 24 50 CCOc1ccc(CCCNC(=O)COc2ccccc2OC)cc1 ZINC000217946266 EG In-Stock Unstable MTNR1A 60 44 CCOc1ccc(CCCNC(=O)COc2ccccc2OC)cc1 ZINC000217946266 EG In-Stock Unstable MTNR1B 41 47 CCOc1ccc(CCCNC(=O)COc2ccccc2OC)cc1 ZINC000217946266 EG In-Stock Unstable CRTM 45 43 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1cc([N+](=O)[O-])ccc1F ZINC000217946278 CJ For-Sale Unstable TRPM8 16 45 CC[C@@H]1CCCN1Cc1ccc(F)cc1/C=C\C(=O)O ZINC000217946315 CG For-Sale Unstable ACKR3 45 32 COC(=O)c1ccc(N[C@H]2C[C@H](C)N(C)C[C@@H]2C)cc1 ZINC000217946336 CF For-Sale Unstable BRD2 19 40 COC(=O)c1ccc(N[C@H]2C[C@H](C)N(C)C[C@@H]2C)cc1 ZINC000217946336 CF For-Sale Unstable BRD3 23 41 CC[C@@H](CCO)NC(=O)[C@H](N)C(C)C ZINC000217946338 BC For-Sale Unstable SLC15A2 0 44 CCOC(=O)c1cnn(CCCc2ccccc2)c1O ZINC000217946353 CE For-Sale Unstable HPD 49 33 CCOC(=O)c1cnn(CCCc2ccccc2)c1O ZINC000217946353 CE For-Sale Unstable CACNA1C 42 39 CCOC(=O)c1cnn(CCCc2ccccc2)c1O ZINC000217946353 CE For-Sale Unstable FAAH 46 37 CCOC(=O)c1cnn(CCCc2ccccc2)c1O ZINC000217946353 CE For-Sale Unstable CES1 42 34 CCCOc1ccccc1CCCNC(=O)COc1ccccc1OC ZINC000217946385 FH In-Stock Unstable MTNR1A 55 44 CCCOc1ccccc1CCCNC(=O)COc1ccccc1OC ZINC000217946385 FH In-Stock Unstable MTNR1B 50 45 CCCOc1ccccc1CCCNC(=O)COc1ccccc1OC ZINC000217946385 FH In-Stock Unstable ACAT 0 40 Nc1nc(/C=C\c2c[nH]c3ccccc23)cs1 ZINC000217946404 BG For-Sale Unstable TDO2 0 57 CC[C@H]1CCCN1Cc1ccc(F)cc1/C=C\C(=O)O ZINC000217946408 CG For-Sale Unstable ACKR3 45 32 CC[C@H](CCO)NC(=O)[C@H](N)C(C)C ZINC000217946414 BC For-Sale Unstable SLC15A2 0 44 CC(C)n1cc(CC(=O)N2CCCC3=C[C@H]4C[C@H](CN5CCCC[C@@H]45)[C@H]32)c2ccccc21 ZINC000217946425 IK In-Stock Unstable Q7YY07_CRYPV 43 32 Cn1c(=O)n(CCC(=O)N(Cc2ccccc2)Cc2ccccc2)c2ccccc21 ZINC000217946451 GH On-Demand Unstable CMA1 20 41 Cn1c(=O)n(CCC(=O)N(Cc2ccccc2)Cc2ccccc2)c2ccccc21 ZINC000217946451 GH On-Demand Unstable TSPO 24 47 Cn1c(=O)n(CCC(=O)N(Cc2ccccc2)Cc2ccccc2)c2ccccc21 ZINC000217946451 GH On-Demand Unstable CTSG 35 40 C[C@H]1CN(C)[C@@H](C)C[C@@H]1Nc1ccc(C(=O)O)cc1 ZINC000217946452 CF For-Sale Unstable BRD4 15 40 C[C@H]1CN(C)[C@@H](C)C[C@@H]1Nc1ccc(C(=O)O)cc1 ZINC000217946452 CF For-Sale Unstable BRD2 34 40 C[C@H]1CN(C)[C@@H](C)C[C@@H]1Nc1ccc(C(=O)O)cc1 ZINC000217946452 CF For-Sale Unstable BRD3 29 40 O=C(O)c1cnn(CCCc2ccccc2)c1O ZINC000217946458 BD For-Sale Unstable SIGMAR1 28 44 O=C(O)c1cnn(CCCc2ccccc2)c1O ZINC000217946458 BD For-Sale Unstable PREP 40 36 O=C(O)c1cnn(CCCc2ccccc2)c1O ZINC000217946458 BD For-Sale Unstable CES1D 44 32 Nc1nc(/C=C\c2c[nH]c3ncccc23)cs1 ZINC000217946494 BF For-Sale Unstable TDO2 0 44 Nc1nc(/C=C\c2c[nH]c3ncccc23)cs1 ZINC000217946494 BF For-Sale Unstable CDC7 47 38 CC(C)n1cc(CC(=O)N2CCCC3=C[C@H]4C[C@H](CN5CCCC[C@@H]45)[C@@H]32)c2ccccc21 ZINC000217946501 IK In-Stock Unstable Q7YY07_CRYPV 43 32 CC1CCN(Cc2ccc(F)c(/C=C\C(=O)O)c2)CC1 ZINC000217946524 CG For-Sale Unstable ACHE 15 46 CC1CCN(Cc2ccc(F)c(/C=C\C(=O)O)c2)CC1 ZINC000217946524 CG For-Sale Unstable SIGMAR1 38 46 CC1CCN(Cc2ccc(F)c(/C=C\C(=O)O)c2)CC1 ZINC000217946524 CG For-Sale Unstable CCR1 24 40 CC1CCN(Cc2ccc(F)c(/C=C\C(=O)O)c2)CC1 ZINC000217946524 CG For-Sale Unstable CCR3 31 46 CC1CCN(Cc2ccc(F)c(/C=C\C(=O)O)c2)CC1 ZINC000217946524 CG For-Sale Unstable MLNR 40 35 CC1CCN(Cc2ccc(F)c(/C=C\C(=O)O)c2)CC1 ZINC000217946524 CG For-Sale Unstable MCHR1 31 41 CCC[C@@H](NC(=O)NCc1ccc(F)cc1)C(=O)N(C)C1CCCCC1 ZINC000217946555 FH On-Demand Unstable ANPEP 15 47 CCC[C@@H](NC(=O)NCc1ccc(F)cc1)C(=O)N(C)C1CCCCC1 ZINC000217946555 FH On-Demand Unstable CCR3 45 31 CCOC(=O)c1cnn(CCCOc2ccccc2)c1O ZINC000217946571 CE For-Sale Unstable PLA2G4B 77 34 NC(=S)N/N=C/C1=C(Cl)CCC1 ZINC000217946602 BD For-Sale Unstable UREA_CANEN 32 45 NC(=S)N/N=C/C1=C(Cl)CCC1 ZINC000217946602 BD For-Sale Unstable GAG 0 46 CN(Cc1cccc(/C=C\C(=O)O)c1)c1ccccc1 ZINC000217946611 CG For-Sale Unstable PTGER2 31 45 CN(Cc1cccc(/C=C\C(=O)O)c1)c1ccccc1 ZINC000217946611 CG For-Sale Unstable PTGER3 15 40 CN(Cc1cccc(/C=C\C(=O)O)c1)c1ccccc1 ZINC000217946611 CG For-Sale Unstable NR1H4 50 40 CN(Cc1cccc(/C=C\C(=O)O)c1)c1ccccc1 ZINC000217946611 CG For-Sale Unstable HSD17B2 26 40 CN(Cc1cccc(/C=C\C(=O)O)c1)c1ccccc1 ZINC000217946611 CG For-Sale Unstable 17HSDCL 0 40 CN(Cc1cccc(/C=C\C(=O)O)c1)c1ccccc1 ZINC000217946611 CG For-Sale Unstable AKR1C3 35 45 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CNC(=O)c1ccccc1 ZINC000217946619 HD For-Sale Unstable PLA2G4A 20 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CNC(=O)c1ccccc1 ZINC000217946619 HD For-Sale Unstable PREP 17 44 CCC[C@H](NC(=O)NCc1ccc(F)cc1)C(=O)N(C)C1CCCCC1 ZINC000217946627 FH On-Demand Unstable ANPEP 15 47 CCC[C@H](NC(=O)NCc1ccc(F)cc1)C(=O)N(C)C1CCCCC1 ZINC000217946627 FH On-Demand Unstable CCR3 45 31 COC(=O)C[C@@H](C1=C(O)C(=O)C([C@H](CC(=O)OC)c2ccc(O)c(OC)c2)=C(O)C1=O)c1ccc(O)c(OC)c1 ZINC000217946628 KF In-Stock Unstable PNLIP 0 47 COC(=O)C[C@@H](C1=C(O)C(=O)C([C@H](CC(=O)OC)c2ccc(O)c(OC)c2)=C(O)C1=O)c1ccc(O)c(OC)c1 ZINC000217946628 KF In-Stock Unstable FOLH1 35 44 COC(=O)C[C@@H](C1=C(O)C(=O)C([C@H](CC(=O)OC)c2ccc(O)c(OC)c2)=C(O)C1=O)c1ccc(O)c(OC)c1 ZINC000217946628 KF In-Stock Unstable TNF 21 42 COC(=O)C[C@@H](C1=C(O)C(=O)C([C@H](CC(=O)OC)c2ccc(O)c(OC)c2)=C(O)C1=O)c1ccc(O)c(OC)c1 ZINC000217946628 KF In-Stock Unstable TRPV1 0 44 COC(=O)C[C@@H](C1=C(O)C(=O)C([C@H](CC(=O)OC)c2ccc(O)c(OC)c2)=C(O)C1=O)c1ccc(O)c(OC)c1 ZINC000217946628 KF In-Stock Unstable SLC22A3 0 44 O=C(O)c1cnn(CCCOc2ccccc2)c1O ZINC000217946683 CD For-Sale Unstable HRH3 29 41 O=C(O)c1cnn(CCCOc2ccccc2)c1O ZINC000217946683 CD For-Sale Unstable PLA2G4B 74 36 CN(Cc1ccc(F)cc1/C=C\C(=O)O)c1ccccc1 ZINC000217946700 CH For-Sale Unstable PTGER2 39 40 CN(Cc1ccc(F)cc1/C=C\C(=O)O)c1ccccc1 ZINC000217946700 CH For-Sale Unstable PTGER3 15 40 CN(Cc1ccc(F)cc1/C=C\C(=O)O)c1ccccc1 ZINC000217946700 CH For-Sale Unstable PTGDR 0 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CNC(=O)c1ccccc1 ZINC000217946705 HD For-Sale Unstable PLA2G4A 20 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CNC(=O)c1ccccc1 ZINC000217946705 HD For-Sale Unstable PREP 17 44 COc1ccccc1OCC(=O)N[C@@H](C)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217946712 GI In-Stock Unstable RORC 46 40 COC(=O)C[C@H](C1=C(O)C(=O)C([C@H](CC(=O)OC)c2ccc(O)c(OC)c2)=C(O)C1=O)c1ccc(O)c(OC)c1 ZINC000217946729 KF In-Stock Unstable PNLIP 0 47 COC(=O)C[C@H](C1=C(O)C(=O)C([C@H](CC(=O)OC)c2ccc(O)c(OC)c2)=C(O)C1=O)c1ccc(O)c(OC)c1 ZINC000217946729 KF In-Stock Unstable FOLH1 35 44 COC(=O)C[C@H](C1=C(O)C(=O)C([C@H](CC(=O)OC)c2ccc(O)c(OC)c2)=C(O)C1=O)c1ccc(O)c(OC)c1 ZINC000217946729 KF In-Stock Unstable TNF 21 42 COC(=O)C[C@H](C1=C(O)C(=O)C([C@H](CC(=O)OC)c2ccc(O)c(OC)c2)=C(O)C1=O)c1ccc(O)c(OC)c1 ZINC000217946729 KF In-Stock Unstable TRPV1 0 44 COC(=O)C[C@H](C1=C(O)C(=O)C([C@H](CC(=O)OC)c2ccc(O)c(OC)c2)=C(O)C1=O)c1ccc(O)c(OC)c1 ZINC000217946729 KF In-Stock Unstable SLC22A3 0 44 C[C@H](Nc1ncnc(N)c1C#Cc1ccccc1)c1nc2cccc(Cl)c2c(=O)n1-c1ccccc1 ZINC000217946766 JJ Annotated Unstable PIK3CD 28 52 C[C@H](Nc1ncnc(N)c1C#Cc1ccccc1)c1nc2cccc(Cl)c2c(=O)n1-c1ccccc1 ZINC000217946766 JJ Annotated Unstable PIK3CG 15 45 CCCC[C@@H](CC)CNCC(=O)Nc1cccc(C)c1 ZINC000217946773 CH For-Sale Unstable KCNK3 58 39 CCCC[C@@H](CC)CNCC(=O)Nc1cccc(C)c1 ZINC000217946773 CH For-Sale Unstable KCNK9 43 39 CN(Cc1ccc(F)c(/C=C\C(=O)O)c1)c1ccccc1 ZINC000217946784 CH For-Sale Unstable PTGER2 34 40 CN(Cc1ccc(F)c(/C=C\C(=O)O)c1)c1ccccc1 ZINC000217946784 CH For-Sale Unstable PTGER4 0 40 CN(Cc1ccc(F)c(/C=C\C(=O)O)c1)c1ccccc1 ZINC000217946784 CH For-Sale Unstable PTGER3 19 42 CN(Cc1ccc(F)c(/C=C\C(=O)O)c1)c1ccccc1 ZINC000217946784 CH For-Sale Unstable PTGDR 0 42 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CNC(=O)c1ccccc1 ZINC000217946788 HD For-Sale Unstable PLA2G4A 20 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CNC(=O)c1ccccc1 ZINC000217946788 HD For-Sale Unstable PREP 17 44 COC(=O)C[C@H](C1=C(O)C(=O)C([C@@H](CC(=O)OC)c2ccc(O)c(OC)c2)=C(O)C1=O)c1ccc(O)c(OC)c1 ZINC000217946799 KF In-Stock Unstable PNLIP 0 47 COC(=O)C[C@H](C1=C(O)C(=O)C([C@@H](CC(=O)OC)c2ccc(O)c(OC)c2)=C(O)C1=O)c1ccc(O)c(OC)c1 ZINC000217946799 KF In-Stock Unstable FOLH1 35 44 COC(=O)C[C@H](C1=C(O)C(=O)C([C@@H](CC(=O)OC)c2ccc(O)c(OC)c2)=C(O)C1=O)c1ccc(O)c(OC)c1 ZINC000217946799 KF In-Stock Unstable TNF 21 42 COC(=O)C[C@H](C1=C(O)C(=O)C([C@@H](CC(=O)OC)c2ccc(O)c(OC)c2)=C(O)C1=O)c1ccc(O)c(OC)c1 ZINC000217946799 KF In-Stock Unstable TRPV1 0 44 COC(=O)C[C@H](C1=C(O)C(=O)C([C@@H](CC(=O)OC)c2ccc(O)c(OC)c2)=C(O)C1=O)c1ccc(O)c(OC)c1 ZINC000217946799 KF In-Stock Unstable SLC22A3 0 44 COc1ccccc1OCC(=O)N[C@H](C)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217946800 GI In-Stock Unstable RORC 46 40 CCOC(=O)c1cnn(Cc2ccccc2C)c1O ZINC000217946801 CE For-Sale Unstable NPBWR1 30 43 CC(=O)N[C@@H](C(=O)N[C@@H]1CCC[C@@H]1CO)C(C)C ZINC000217946825 CC For-Sale Unstable CASP2 42 37 CCCCCCCCC/C=C\C(F)(F)F ZINC000217946844 BK For-Sale Unstable CES2 48 35 CCCCCCCCC/C=C\C(F)(F)F ZINC000217946844 BK For-Sale Unstable CES1 45 31 CCCCCCCCC/C=C\C(F)(F)F ZINC000217946844 BK For-Sale Unstable EST1_PIG 53 35 CCCCCCCCC/C=C\C(F)(F)F ZINC000217946844 BK For-Sale Unstable CES2C 56 34 CCCCCCCCC/C=C\C(F)(F)F ZINC000217946844 BK For-Sale Unstable FABP3 24 42 CCCC[C@H](CC)CNCC(=O)Nc1cccc(C)c1 ZINC000217946847 CH For-Sale Unstable KCNK3 58 39 CCCC[C@H](CC)CNCC(=O)Nc1cccc(C)c1 ZINC000217946847 CH For-Sale Unstable KCNK9 43 39 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CNC(=O)c1ccccc1 ZINC000217946856 HD For-Sale Unstable PLA2G4A 20 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CNC(=O)c1ccccc1 ZINC000217946856 HD For-Sale Unstable PREP 17 44 CC(=O)N[C@H](C(=O)N[C@@H]1CCC[C@@H]1CO)C(C)C ZINC000217946902 CC For-Sale Unstable CASP2 42 37 COC(=O)C[C@@H](C1=C(O)C(=O)C([C@H](CC(=O)OC)c2ccc(C(C)C)cc2)=C(O)C1=O)c1ccc(C(C)C)cc1 ZINC000217946905 KK In-Stock Unstable KCNA5 29 40 COc1cccc(/C=C/NC(=O)Nc2ccccc2N2CCOCC2)c1 ZINC000217946912 FG For-Sale Unstable DRD4 43 36 COc1cccc(/C=C/NC(=O)Nc2ccccc2N2CCOCC2)c1 ZINC000217946912 FG For-Sale Unstable KCNQ2 82 50 COc1cccc(/C=C/NC(=O)Nc2ccccc2N2CCOCC2)c1 ZINC000217946912 FG For-Sale Unstable CSF1R 0 44 COc1cccc(/C=C/NC(=O)Nc2ccccc2N2CCOCC2)c1 ZINC000217946912 FG For-Sale Unstable BRPF1 0 48 Cn1cccc1[C@H](O)CCNC(=O)C(=O)NCCc1ccccc1 ZINC000217946915 EC In-Stock Unstable DNPEP 0 40 Cn1cccc1[C@H](O)CCNC(=O)C(=O)NCCc1ccccc1 ZINC000217946915 EC In-Stock Unstable AMP1_PLAFQ 31 45 Cc1ccccc1Cn1ncc(C(=O)O)c1O ZINC000217946919 BD For-Sale Unstable NPBWR1 27 43 C[C@H]1CN(C)[C@@H](C)C[C@@H]1Nc1cccc(C(=O)O)c1 ZINC000217946940 CF For-Sale Unstable AKR1C3 50 43 C[C@H]1CN(C)[C@@H](C)C[C@@H]1Nc1cccc(C(=O)O)c1 ZINC000217946940 CF For-Sale Unstable KCNK3 57 32 Fc1ccc2c(c1)N(c1ccc(CBr)cn1)CC2 ZINC000217946943 DH For-Sale Unstable SCD1 25 40 Fc1ccc2c(c1)N(c1ccc(CBr)cn1)CC2 ZINC000217946943 DH For-Sale Unstable SCD 25 40 CC(=O)N[C@@H](C(=O)N[C@H]1CCC[C@@H]1CO)C(C)C ZINC000217946971 CC For-Sale Unstable CASP2 42 37 NC[C@H](c1ccc(Br)s1)N1CCC[C@@H]1c1cccnc1 ZINC000217946972 FH For-Sale Unstable CHRNA2 45 46 NC[C@H](c1ccc(Br)s1)N1CCC[C@@H]1c1cccnc1 ZINC000217946972 FH For-Sale Unstable CRTY 0 46 CCS(=O)(=O)[C@@H]1CCC(CN)(CN)C1 ZINC000217946977 BB In-Stock Unstable CACNA2D1 40 41 COC(=O)C[C@H](C1=C(O)C(=O)C([C@H](CC(=O)OC)c2ccc(C(C)C)cc2)=C(O)C1=O)c1ccc(C(C)C)cc1 ZINC000217946990 KK In-Stock Unstable KCNA5 29 40 Cn1cccc1[C@@H](O)CCNC(=O)C(=O)NCCc1ccccc1 ZINC000217947008 EC In-Stock Unstable DNPEP 0 40 Cn1cccc1[C@@H](O)CCNC(=O)C(=O)NCCc1ccccc1 ZINC000217947008 EC In-Stock Unstable AMP1_PLAFQ 31 45 COc1cccc(/C=C/NC(=O)Nc2ccc(N3CCN(C)CC3)cc2)c1 ZINC000217947020 FG For-Sale Unstable DRD4 49 41 COc1cccc(/C=C/NC(=O)Nc2ccc(N3CCN(C)CC3)cc2)c1 ZINC000217947020 FG For-Sale Unstable HTR1B 18 48 COc1cccc(/C=C/NC(=O)Nc2ccc(N3CCN(C)CC3)cc2)c1 ZINC000217947020 FG For-Sale Unstable LCK 26 41 COc1cccc(/C=C/NC(=O)Nc2ccc(N3CCN(C)CC3)cc2)c1 ZINC000217947020 FG For-Sale Unstable PRNP 37 43 COc1cccc(/C=C/NC(=O)Nc2ccc(N3CCN(C)CC3)cc2)c1 ZINC000217947020 FG For-Sale Unstable MTNR1A 17 43 COc1cccc(/C=C/NC(=O)Nc2ccc(N3CCN(C)CC3)cc2)c1 ZINC000217947020 FG For-Sale Unstable MTNR1B 24 43 COc1cccc(/C=C/NC(=O)Nc2ccc(N3CCN(C)CC3)cc2)c1 ZINC000217947020 FG For-Sale Unstable FLT3 15 40 COc1cccc(/C=C/NC(=O)Nc2ccc(N3CCN(C)CC3)cc2)c1 ZINC000217947020 FG For-Sale Unstable TAAR1 16 41 O=C(CCn1ccc(=O)[nH]c1=O)N1CCC[C@@H]1c1nccs1 ZINC000217947047 DC In-Stock Unstable COLA 58 39 O=C(CCn1ccc(=O)[nH]c1=O)N1CCC[C@@H]1c1nccs1 ZINC000217947047 DC In-Stock Unstable CPT1A 56 37 O=C(CCn1ccc(=O)[nH]c1=O)N1CCC[C@@H]1c1nccs1 ZINC000217947047 DC In-Stock Unstable DUT 74 49 CCS(=O)(=O)[C@H]1CCC(CN)(CN)C1 ZINC000217947054 BB In-Stock Unstable CACNA2D1 40 41 CC(=O)N[C@H](C(=O)N[C@H]1CCC[C@@H]1CO)C(C)C ZINC000217947063 CC For-Sale Unstable CASP2 42 37 COC(=O)C[C@H](C1=C(O)C(=O)C([C@@H](CC(=O)OC)c2ccc(C(C)C)cc2)=C(O)C1=O)c1ccc(C(C)C)cc1 ZINC000217947072 KK In-Stock Unstable KCNA5 29 40 Cc1ccc(C(=O)O)c(O[C@H]2C[C@H](C)CC[C@H]2C(C)C)n1 ZINC000217947073 CH For-Sale Unstable TRPM8 0 40 CCCCN(C(=O)c1cc(C(C)C)nc2onc(C)c12)c1ccccc1 ZINC000217947097 FK On-Demand Unstable TSPO 18 41 O=C(CCn1ccc(=O)[nH]c1=O)N1CCC[C@H]1c1nccs1 ZINC000217947127 DC In-Stock Unstable COLA 58 39 O=C(CCn1ccc(=O)[nH]c1=O)N1CCC[C@H]1c1nccs1 ZINC000217947127 DC In-Stock Unstable CPT1A 56 37 O=C(CCn1ccc(=O)[nH]c1=O)N1CCC[C@H]1c1nccs1 ZINC000217947127 DC In-Stock Unstable DUT 74 49 COc1cccc(/C=C/NC(=O)Nc2ccc(N3CCCCC3)cc2)c1 ZINC000217947131 FI For-Sale Unstable DRD4 46 38 COc1cccc(/C=C/NC(=O)Nc2ccc(N3CCCCC3)cc2)c1 ZINC000217947131 FI For-Sale Unstable HRH2 22 43 COc1cccc(/C=C/NC(=O)Nc2ccc(N3CCCCC3)cc2)c1 ZINC000217947131 FI For-Sale Unstable LPL 20 40 COc1cccc(/C=C/NC(=O)Nc2ccc(N3CCCCC3)cc2)c1 ZINC000217947131 FI For-Sale Unstable MTNR1A 19 44 COc1cccc(/C=C/NC(=O)Nc2ccc(N3CCCCC3)cc2)c1 ZINC000217947131 FI For-Sale Unstable MTNR1B 27 44 COc1cccc(/C=C/NC(=O)Nc2ccc(N3CCCCC3)cc2)c1 ZINC000217947131 FI For-Sale Unstable GALR2 43 40 COc1cccc(/C=C/NC(=O)Nc2ccc(N3CCCCC3)cc2)c1 ZINC000217947131 FI For-Sale Unstable TAAR1 30 40 COc1cccc(/C=C/NC(=O)Nc2ccc(N3CCCCC3)cc2)c1 ZINC000217947131 FI For-Sale Unstable BRPF1 0 41 C#CCNC(=O)N1[C@H](C(=O)O)C[C@@H]2CCCC[C@@H]21 ZINC000217947141 CD For-Sale Unstable ACE 20 57 Cc1ccc(C(=O)O)c(O[C@H]2C[C@@H](C)CC[C@H]2C(C)C)n1 ZINC000217947155 CH For-Sale Unstable TRPM8 0 40 CCS(=O)(=O)[C@@H]1CC[C@@](CN)(CO)C1 ZINC000217947162 BB In-Stock Unstable CACNA2D1 48 44 COC(=O)C[C@H](c1ccc(O)c(Cl)c1)c1oc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c1O ZINC000217947169 KG In-Stock Unstable CHRNA4 26 45 C#CCNC(=O)N1[C@H](C(=O)O)C[C@H]2CCCC[C@@H]21 ZINC000217947230 CD For-Sale Unstable ACE 20 57 COc1cccc(/C=C/NC(=O)Nc2ccc(SC#N)cc2)c1 ZINC000217947246 EI For-Sale Unstable MTNR1B 23 44 Cc1ccc(C(=O)O)c(O[C@H]2C[C@H](C)CC[C@H]2C(C)C)c1 ZINC000217947248 CJ For-Sale Unstable SERPINE1 41 40 Cc1ccc(C(=O)O)c(O[C@H]2C[C@H](C)CC[C@H]2C(C)C)c1 ZINC000217947248 CJ For-Sale Unstable TRPM8 15 44 CCOC(=O)c1cnn(Cc2ccc(F)cc2)c1O ZINC000217947249 CD For-Sale Unstable Q76353_9HIV1 0 44 CCS(=O)(=O)[C@H]1CC[C@@](CN)(CO)C1 ZINC000217947251 BB In-Stock Unstable CACNA2D1 48 44 COC(=O)C[C@@H](c1ccc(O)c(Cl)c1)c1oc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c1O ZINC000217947258 KG In-Stock Unstable CHRNA4 26 45 Cn1cccc1[C@H](O)CCNC(=O)C(=O)NCc1ccc(F)cc1 ZINC000217947308 ED In-Stock Unstable HMGCR 35 40 CCS(=O)(=O)[C@@H]1CC[C@](CN)(CO)C1 ZINC000217947330 BB In-Stock Unstable CACNA2D1 48 44 Cc1ccc(C(=O)O)c(O[C@H]2C[C@@H](C)CC[C@H]2C(C)C)c1 ZINC000217947334 CJ For-Sale Unstable SERPINE1 41 40 Cc1ccc(C(=O)O)c(O[C@H]2C[C@@H](C)CC[C@H]2C(C)C)c1 ZINC000217947334 CJ For-Sale Unstable TRPM8 15 44 COc1cccc(/C=C/NC(=O)Nc2ccc(N(C)C)cc2)c1 ZINC000217947355 DH For-Sale Unstable CA1 15 43 COc1cccc(/C=C/NC(=O)Nc2ccc(N(C)C)cc2)c1 ZINC000217947355 DH For-Sale Unstable MTNR1A 28 60 COc1cccc(/C=C/NC(=O)Nc2ccc(N(C)C)cc2)c1 ZINC000217947355 DH For-Sale Unstable MTNR1B 34 60 CC(C)C[C@H](CC(=O)NCc1ccccc1)c1c(O)cc(O)c2c(=O)cc(-c3ccccc3)oc12 ZINC000217947373 JK In-Stock Unstable CYP1A1 24 45 CC(C)C[C@H](CC(=O)NCc1ccccc1)c1c(O)cc(O)c2c(=O)cc(-c3ccccc3)oc12 ZINC000217947373 JK In-Stock Unstable ABCB1 15 45 CC(C)C[C@H](CC(=O)NCc1ccccc1)c1c(O)cc(O)c2c(=O)cc(-c3ccccc3)oc12 ZINC000217947373 JK In-Stock Unstable CYP1A2 19 45 Cn1cccc1[C@@H](O)CCNC(=O)C(=O)NCc1ccc(F)cc1 ZINC000217947390 ED In-Stock Unstable HMGCR 35 40 C[C@H]1CN(C)[C@@H](C)C[C@@H]1Nc1ccccc1C(=O)O ZINC000217947405 CF For-Sale Unstable AKR1C2 42 39 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Oc1ccc(C(=O)O)cc1Cl ZINC000217947411 DJ For-Sale Unstable SERPINE1 43 45 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Oc1ccc(C(=O)O)cc1Cl ZINC000217947411 DJ For-Sale Unstable TRPM8 15 48 CCS(=O)(=O)[C@H]1CC[C@](CN)(CO)C1 ZINC000217947419 BB In-Stock Unstable CACNA2D1 48 44 COc1cccc(/C=C/NC(=O)NCCO)c1 ZINC000217947460 BC For-Sale Unstable DRD4 43 33 COc1cccc(/C=C/NC(=O)NCCO)c1 ZINC000217947460 BC For-Sale Unstable CYP1B1 29 42 COc1cccc(/C=C/NC(=O)NCCO)c1 ZINC000217947460 BC For-Sale Unstable AHR 28 47 COc1cccc(/C=C/NC(=O)NCCO)c1 ZINC000217947460 BC For-Sale Unstable MTNR1A 93 47 COc1cccc(/C=C/NC(=O)NCCO)c1 ZINC000217947460 BC For-Sale Unstable MTNR1B 84 47 COc1cccc(/C=C/NC(=O)NCCO)c1 ZINC000217947460 BC For-Sale Unstable CYP1A1 21 42 CC(C)C[C@@H](CC(=O)NCc1ccccc1)c1c(O)cc(O)c2c(=O)cc(-c3ccccc3)oc12 ZINC000217947461 JK In-Stock Unstable CYP1A1 24 45 CC(C)C[C@@H](CC(=O)NCc1ccccc1)c1c(O)cc(O)c2c(=O)cc(-c3ccccc3)oc12 ZINC000217947461 JK In-Stock Unstable ABCB1 15 45 CC(C)C[C@@H](CC(=O)NCc1ccccc1)c1c(O)cc(O)c2c(=O)cc(-c3ccccc3)oc12 ZINC000217947461 JK In-Stock Unstable CYP1A2 19 45 CCOC(=O)c1cnn(Cc2cccc(F)c2)c1O ZINC000217947474 CD For-Sale Unstable EGFR 17 40 CCOC(=O)c1cnn(Cc2cccc(F)c2)c1O ZINC000217947474 CD For-Sale Unstable P2RY12 22 41 CCOC(=O)c1cnn(Cc2cccc(F)c2)c1O ZINC000217947474 CD For-Sale Unstable ERBB2 32 40 CN(Cc1ccc(Cl)s1)Cc1ccccc1/C=C\C(=O)O ZINC000217947487 DI For-Sale Unstable PTGER2 40 44 CN(Cc1ccc(Cl)s1)Cc1ccccc1/C=C\C(=O)O ZINC000217947487 DI For-Sale Unstable PTGER4 0 44 CN(Cc1ccc(Cl)s1)Cc1ccccc1/C=C\C(=O)O ZINC000217947487 DI For-Sale Unstable PTGER3 17 44 CN(Cc1ccc(Cl)s1)Cc1ccccc1/C=C\C(=O)O ZINC000217947487 DI For-Sale Unstable PTGDR 0 42 Cc1ccc(NC(=O)C(=O)NCC[C@H](O)c2cccn2C)cc1F ZINC000217947495 ED In-Stock Unstable FPR2 19 42 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Oc1ccc(C(=O)O)cc1Cl ZINC000217947503 DJ For-Sale Unstable SERPINE1 43 45 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Oc1ccc(C(=O)O)cc1Cl ZINC000217947503 DJ For-Sale Unstable TRPM8 15 48 CCS(=O)(=O)[C@@H]1CC[C@](CN)(C(=O)O)C1 ZINC000217947537 BC In-Stock Unstable CACNA2D1 40 36 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1ccc(F)c([N+](=O)[O-])c1 ZINC000217947539 CJ For-Sale Unstable TRPM8 15 45 Cc1ccc(NC(=O)C(=O)NCC[C@@H](O)c2cccn2C)cc1F ZINC000217947571 ED In-Stock Unstable FPR2 19 42 COc1cccc(/C=C/NC(=O)Nc2cccc3ccccc23)c1 ZINC000217947576 DJ For-Sale Unstable TRPV1 27 50 COc1cccc(/C=C/NC(=O)Nc2cccc3ccccc23)c1 ZINC000217947576 DJ For-Sale Unstable MTNR1A 67 50 COc1cccc(/C=C/NC(=O)Nc2cccc3ccccc23)c1 ZINC000217947576 DJ For-Sale Unstable MTNR1B 62 50 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Oc1ccc(C(=O)O)cc1Cl ZINC000217947587 DJ For-Sale Unstable SERPINE1 43 45 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Oc1ccc(C(=O)O)cc1Cl ZINC000217947587 DJ For-Sale Unstable TRPM8 15 48 O=C(O)c1cnn(Cc2cccc(F)c2)c1O ZINC000217947591 BD For-Sale Unstable FABP4 26 44 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1ccc(F)c([N+](=O)[O-])c1 ZINC000217947615 CJ For-Sale Unstable TRPM8 15 45 CCS(=O)(=O)[C@H]1CC[C@](CN)(C(=O)O)C1 ZINC000217947616 BC In-Stock Unstable CACNA2D1 40 36 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Oc1ccc(C(=O)O)cc1Cl ZINC000217947660 DJ For-Sale Unstable SERPINE1 43 45 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Oc1ccc(C(=O)O)cc1Cl ZINC000217947660 DJ For-Sale Unstable TRPM8 15 48 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc(Cl)cc1Cl ZINC000217947685 HH For-Sale Unstable HCRTR1 42 35 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc(Cl)cc1Cl ZINC000217947685 HH For-Sale Unstable HCRTR2 44 35 COC(=O)c1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217947691 EG For-Sale Unstable VDR 0 41 COC(=O)c1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217947691 EG For-Sale Unstable MTNR1A 29 49 COC(=O)c1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217947691 EG For-Sale Unstable MTNR1B 34 49 COC(=O)c1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217947691 EG For-Sale Unstable ACR 62 48 COC(=O)c1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217947691 EG For-Sale Unstable Q8MMZ8_EIMTE 0 44 COC(=O)c1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217947691 EG For-Sale Unstable TAAR1 29 40 COC(=O)c1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217947691 EG For-Sale Unstable SENP1 0 42 CCS(=O)(=O)[C@@H]1CC[C@@](CN)(C(=O)O)C1 ZINC000217947700 BC In-Stock Unstable CACNA2D1 40 36 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1ccc(F)c([N+](=O)[O-])c1 ZINC000217947712 CJ For-Sale Unstable TRPM8 15 45 CCOC(=O)c1cnn(Cc2ccc(Cl)cc2)c1O ZINC000217947713 CE For-Sale Unstable NPBWR1 15 41 CCC(CC)CN(CC)Cc1ccccc1/C=C\C(=O)O ZINC000217947742 CI For-Sale Unstable PTGER2 42 47 CCC(CC)CN(CC)Cc1ccccc1/C=C\C(=O)O ZINC000217947742 CI For-Sale Unstable PTGER4 0 47 CCC(CC)CN(CC)Cc1ccccc1/C=C\C(=O)O ZINC000217947742 CI For-Sale Unstable PTGER3 16 47 CCC(CC)CN(CC)Cc1ccccc1/C=C\C(=O)O ZINC000217947742 CI For-Sale Unstable PTGDR 0 45 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Oc1ccc(C(=O)O)c(Cl)c1 ZINC000217947746 DJ For-Sale Unstable SERPINE1 42 43 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Oc1ccc(C(=O)O)c(Cl)c1 ZINC000217947746 DJ For-Sale Unstable TRPM8 15 45 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc(Cl)cc1Cl ZINC000217947770 HH For-Sale Unstable HCRTR1 42 35 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc(Cl)cc1Cl ZINC000217947770 HH For-Sale Unstable HCRTR2 44 35 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1ccc(F)c([N+](=O)[O-])c1 ZINC000217947788 CJ For-Sale Unstable TRPM8 15 45 CCS(=O)(=O)[C@H]1CC[C@@](CN)(C(=O)O)C1 ZINC000217947794 BC In-Stock Unstable CACNA2D1 40 36 COc1cccc(/C=C/NC(=O)N(Cc2ccccc2)c2ccccc2)c1 ZINC000217947803 FK For-Sale Unstable TSPO 45 36 COc1cccc(/C=C/NC(=O)N(Cc2ccccc2)c2ccccc2)c1 ZINC000217947803 FK For-Sale Unstable G6PC 28 48 COc1cccc(/C=C/NC(=O)N(Cc2ccccc2)c2ccccc2)c1 ZINC000217947803 FK For-Sale Unstable MTNR1A 43 44 COc1cccc(/C=C/NC(=O)N(Cc2ccccc2)c2ccccc2)c1 ZINC000217947803 FK For-Sale Unstable MTNR1B 47 44 COc1cccc(/C=C/NC(=O)N(Cc2ccccc2)c2ccccc2)c1 ZINC000217947803 FK For-Sale Unstable NR1H4 57 44 COc1cccc(/C=C/NC(=O)N(Cc2ccccc2)c2ccccc2)c1 ZINC000217947803 FK For-Sale Unstable HSD17B2 17 40 COc1cccc(/C=C/NC(=O)N(Cc2ccccc2)c2ccccc2)c1 ZINC000217947803 FK For-Sale Unstable PTGES 16 44 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Oc1ccc(C(=O)O)c(Cl)c1 ZINC000217947827 DJ For-Sale Unstable SERPINE1 42 43 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Oc1ccc(C(=O)O)c(Cl)c1 ZINC000217947827 DJ For-Sale Unstable TRPM8 15 45 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc(Cl)cc1Cl ZINC000217947850 HH For-Sale Unstable HCRTR1 42 35 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc(Cl)cc1Cl ZINC000217947850 HH For-Sale Unstable HCRTR2 44 35 COc1cccc(/C=C/NC(=O)Nc2ccc3ccccc3c2)c1 ZINC000217947903 DJ For-Sale Unstable CA1 17 43 COc1cccc(/C=C/NC(=O)Nc2ccc3ccccc3c2)c1 ZINC000217947903 DJ For-Sale Unstable UL80 28 48 COc1cccc(/C=C/NC(=O)Nc2ccc3ccccc3c2)c1 ZINC000217947903 DJ For-Sale Unstable MTNR1A 38 48 COc1cccc(/C=C/NC(=O)Nc2ccc3ccccc3c2)c1 ZINC000217947903 DJ For-Sale Unstable MTNR1B 38 48 COc1cccc(/C=C/NC(=O)Nc2ccc3ccccc3c2)c1 ZINC000217947903 DJ For-Sale Unstable IMPDH2 0 40 COc1cccc(/C=C/NC(=O)Nc2ccc3ccccc3c2)c1 ZINC000217947903 DJ For-Sale Unstable PTPA 0 45 COc1cccc(/C=C/NC(=O)Nc2ccc3ccccc3c2)c1 ZINC000217947903 DJ For-Sale Unstable IMDH_CRYPV 32 43 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Oc1ccc(C(=O)O)c(Cl)c1 ZINC000217947915 DJ For-Sale Unstable SERPINE1 42 43 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Oc1ccc(C(=O)O)c(Cl)c1 ZINC000217947915 DJ For-Sale Unstable TRPM8 15 45 CCOC(=O)c1cnn(Cc2cccc(Cl)c2)c1O ZINC000217947946 CE For-Sale Unstable P2RY12 34 41 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc(Cl)cc1Cl ZINC000217947949 HH For-Sale Unstable HCRTR1 42 35 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc(Cl)cc1Cl ZINC000217947949 HH For-Sale Unstable HCRTR2 44 35 CC(C)Oc1ccc(/C=C2/CC(=O)NC2=O)cc1 ZINC000217947968 BD For-Sale Unstable HPGD 53 38 COc1cccc(/C=C2\Oc3c(ccc4c3[C@H](c3cc(OC)c(OC)c(OC)c3)CC(=O)O4)C2=O)c1OC ZINC000217947972 KJ In-Stock Unstable MT-ND4 49 30 N#C[C@@H]1CNCCN1CC(=O)N1CCC[C@@H](C(N)=O)C1 ZINC000217947976 CA For-Sale Unstable DPP4 28 44 N#C[C@@H]1CNCCN1CC(=O)N1CCC[C@@H](C(N)=O)C1 ZINC000217947976 CA For-Sale Unstable PREP 21 42 CCC(CC)CN(CC)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217947994 CI For-Sale Unstable AKR1C3 32 43 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Oc1ccc(C(=O)O)c(Cl)c1 ZINC000217947995 DJ For-Sale Unstable SERPINE1 42 43 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Oc1ccc(C(=O)O)c(Cl)c1 ZINC000217947995 DJ For-Sale Unstable TRPM8 15 45 CC[C@@H](NC(=O)COc1ccccc1OC)c1ccc(OC)c(OC)c1 ZINC000217948013 FG In-Stock Unstable MTNR1B 26 41 CC[C@@H](NC(=O)COc1ccccc1OC)c1ccc(OC)c(OC)c1 ZINC000217948013 FG In-Stock Unstable ENPP1 58 34 CC[C@@H](NC(=O)COc1ccccc1OC)c1ccc(OC)c(OC)c1 ZINC000217948013 FG In-Stock Unstable PDS 40 33 COc1cccc(/C=C/NC(=O)N(C)c2ccc(O)cc2)c1 ZINC000217948016 CG For-Sale Unstable MTNR1A 26 49 COc1cccc(/C=C/NC(=O)N(C)c2ccc(O)cc2)c1 ZINC000217948016 CG For-Sale Unstable MTNR1B 31 49 COc1cccc(/C=C/NC(=O)N(C)c2ccc(O)cc2)c1 ZINC000217948016 CG For-Sale Unstable HSD17B2 21 40 COc1cccc(/C=C2\Oc3c(ccc4c3[C@@H](c3cc(OC)c(OC)c(OC)c3)CC(=O)O4)C2=O)c1OC ZINC000217948043 KJ In-Stock Unstable MT-ND4 49 30 Cn1cccc1[C@H](O)CCNC(=O)C(=O)Nc1ccc2c(c1)OCO2 ZINC000217948045 EC In-Stock Unstable DYRK2 40 34 O=C(O)c1cnn(Cc2cccc(Cl)c2)c1O ZINC000217948063 CD For-Sale Unstable CCR2 0 45 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc(Cl)c(Cl)c1 ZINC000217948065 HH For-Sale Unstable HCRTR2 41 34 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Oc1cc(Cl)ccc1C(=O)O ZINC000217948081 DJ For-Sale Unstable SERPINE1 40 39 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Oc1cc(Cl)ccc1C(=O)O ZINC000217948081 DJ For-Sale Unstable TRPM8 15 47 CC[C@H](NC(=O)COc1ccccc1OC)c1ccc(OC)c(OC)c1 ZINC000217948096 FG In-Stock Unstable MTNR1B 26 41 CC[C@H](NC(=O)COc1ccccc1OC)c1ccc(OC)c(OC)c1 ZINC000217948096 FG In-Stock Unstable ENPP1 58 34 CC[C@H](NC(=O)COc1ccccc1OC)c1ccc(OC)c(OC)c1 ZINC000217948096 FG In-Stock Unstable PDS 40 33 COc1ccc(CN2CCC[C@@H]2CO)cc1/C=C\C(=O)O ZINC000217948121 CD For-Sale Unstable DRD2 43 42 COc1ccc(CN2CCC[C@@H]2CO)cc1/C=C\C(=O)O ZINC000217948121 CD For-Sale Unstable SPHK1 19 43 COc1ccc(CN2CCC[C@@H]2CO)cc1/C=C\C(=O)O ZINC000217948121 CD For-Sale Unstable ACKR3 66 36 CCCCN(C)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217948134 CG For-Sale Unstable MTNR1A 45 44 CCCCN(C)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217948134 CG For-Sale Unstable MTNR1B 45 44 Cn1cccc1[C@@H](O)CCNC(=O)C(=O)Nc1ccc2c(c1)OCO2 ZINC000217948138 EC In-Stock Unstable DYRK2 40 34 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc(Cl)c(Cl)c1 ZINC000217948145 HH For-Sale Unstable HCRTR2 41 34 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Oc1cc(Cl)ccc1C(=O)O ZINC000217948152 DJ For-Sale Unstable SERPINE1 40 39 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Oc1cc(Cl)ccc1C(=O)O ZINC000217948152 DJ For-Sale Unstable TRPM8 15 47 Cc1ncc(C(=O)NCc2ccc3nc(C)[nH]c3c2)c(=O)[nH]1 ZINC000217948159 CD In-Stock Unstable TYMS 78 45 CCOC(=O)c1cnn(Cc2ccccc2Cl)c1O ZINC000217948167 CE For-Sale Unstable NPBWR1 54 41 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc(Cl)c(Cl)c1 ZINC000217948209 HH For-Sale Unstable HCRTR2 41 34 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Oc1cc(Cl)ccc1C(=O)O ZINC000217948223 DJ For-Sale Unstable SERPINE1 40 39 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Oc1cc(Cl)ccc1C(=O)O ZINC000217948223 DJ For-Sale Unstable TRPM8 15 47 O=S(=O)(Cl)Cc1ccc2nnsc2c1 ZINC000217948246 BD For-Sale Unstable PRMT3 69 43 COCCN(CCOC)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217948252 DD For-Sale Unstable DRD4 42 32 COCCN(CCOC)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217948252 DD For-Sale Unstable CYP1B1 24 41 COCCN(CCOC)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217948252 DD For-Sale Unstable AHR 19 43 COCCN(CCOC)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217948252 DD For-Sale Unstable MTNR1A 48 45 COCCN(CCOC)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217948252 DD For-Sale Unstable MTNR1B 46 45 COCCN(CCOC)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217948252 DD For-Sale Unstable CYP1A1 18 41 O=C(O)c1cnn(Cc2ccccc2Cl)c1O ZINC000217948258 CD For-Sale Unstable NPBWR1 42 38 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Oc1cc(Cl)ccc1C(=O)O ZINC000217948303 DJ For-Sale Unstable SERPINE1 40 39 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Oc1cc(Cl)ccc1C(=O)O ZINC000217948303 DJ For-Sale Unstable TRPM8 15 47 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc(Cl)c(Cl)c1 ZINC000217948310 HH For-Sale Unstable HCRTR2 41 34 CC1(C)COCCN1Cc1cccc(/C=C\C(=O)O)c1 ZINC000217948313 CE For-Sale Unstable HDAC8 23 40 COc1ccc([C@@H]2Nc3ccccc3C(=O)N2CCCC(=O)Nc2ccccc2O)cc1 ZINC000217948317 II In-Stock Unstable TSHR 65 51 CCCC[C@@H](CC)CNCC(=O)Nc1ccccc1 ZINC000217948349 CG For-Sale Unstable SOAT1 21 49 CCCN(CCC)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217948360 CG For-Sale Unstable DRD4 40 30 CCCN(CCC)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217948360 CG For-Sale Unstable CYP1B1 20 41 CCCN(CCC)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217948360 CG For-Sale Unstable AHR 19 43 CCCN(CCC)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217948360 CG For-Sale Unstable MTNR1A 53 45 CCCN(CCC)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217948360 CG For-Sale Unstable MTNR1B 49 45 CCCN(CCC)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217948360 CG For-Sale Unstable CYP1A1 18 41 COc1ccc(-c2noc(CNC(=O)COc3ccccc3OC)n2)c(OC)c1 ZINC000217948383 GE In-Stock Unstable MTNR1A 61 39 COc1ccc(-c2noc(CNC(=O)COc3ccccc3OC)n2)c(OC)c1 ZINC000217948383 GE In-Stock Unstable MTNR1B 50 39 COc1ccc([C@H]2Nc3ccccc3C(=O)N2CCCC(=O)Nc2ccccc2O)cc1 ZINC000217948393 II In-Stock Unstable TSHR 65 51 CCCC[C@H](CC)CNCC(=O)Nc1ccccc1 ZINC000217948420 CG For-Sale Unstable SOAT1 21 49 O=C(O)c1cnn(Cc2ccc(Br)cc2)c1O ZINC000217948466 CE For-Sale Unstable PRS 56 33 COc1cccc(/C=C/NC(=O)N(C=O)CCCN)c1 ZINC000217948476 CD For-Sale Unstable MTNR1A 32 40 COc1cccc(/C=C/NC(=O)N(C=O)CCCN)c1 ZINC000217948476 CD For-Sale Unstable MTNR1B 34 40 COc1cccc(/C=C2\Oc3c(ccc4c3[C@H](c3cc5ccccc5[nH]c3=O)CC(=O)O4)C2=O)c1OC ZINC000217948512 JJ In-Stock Unstable MT-ND4 40 31 COc1cccc(/C=C2\Oc3c(ccc4c3[C@@H](c3cc5ccccc5[nH]c3=O)CC(=O)O4)C2=O)c1OC ZINC000217948584 JJ In-Stock Unstable MT-ND4 40 31 COc1cccc(/C=C/NC(=O)NCCCNC=O)c1 ZINC000217948588 CD For-Sale Unstable DRD4 40 30 COc1cccc(/C=C/NC(=O)NCCCNC=O)c1 ZINC000217948588 CD For-Sale Unstable MTNR1A 71 48 COc1cccc(/C=C/NC(=O)NCCCNC=O)c1 ZINC000217948588 CD For-Sale Unstable MTNR1B 67 48 CCN(CC)S(=O)(=O)c1cc(NC(=O)c2cc(C(C)C)nc3onc(C)c23)ccc1Cl ZINC000217948596 JJ On-Demand Unstable SMG1 22 40 N#C[C@@H]1CNCCN1CC(=O)N1CCC[C@@H]1c1cccs1 ZINC000217948656 DD For-Sale Unstable COLA 42 38 N#C[C@@H]1CNCCN1CC(=O)N1CCC[C@@H]1c1cccs1 ZINC000217948656 DD For-Sale Unstable CPT1A 43 37 N#C[C@@H]1CNCCN1CC(=O)N1CCC[C@@H]1c1cccs1 ZINC000217948656 DD For-Sale Unstable DPP4 62 40 N#C[C@@H]1CNCCN1CC(=O)N1CCC[C@@H]1c1cccs1 ZINC000217948656 DD For-Sale Unstable PREP 57 41 N#C[C@@H]1CNCCN1CC(=O)N1CCC[C@@H]1c1cccs1 ZINC000217948656 DD For-Sale Unstable FAP 0 46 O=C(Cc1ccc(Br)cc1)NCC1C[C@@H]2CC[C@H](C1)N2 ZINC000217948710 EF For-Sale Unstable LUXR 15 43 O=C(Cc1ccc(Br)cc1)NCC1C[C@@H]2CC[C@H](C1)N2 ZINC000217948710 EF For-Sale Unstable TRAR 23 43 C[C@@H]1CCC[C@H]([C@@H](N)Cc2cc(Br)ccc2F)C1 ZINC000217948725 DI For-Sale Unstable DPP4 25 44 COc1ccccc1OCC(=O)NCCCc1ccc(C(C)C)cc1 ZINC000217948737 EH In-Stock Unstable DRD2 20 43 COc1ccccc1OCC(=O)NCCCc1ccc(C(C)C)cc1 ZINC000217948737 EH In-Stock Unstable MTNR1B 28 47 COc1ccccc1OCC(=O)NCCCc1ccc(C(C)C)cc1 ZINC000217948737 EH In-Stock Unstable CRTM 43 43 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc(Cl)c1 ZINC000217948748 GG For-Sale Unstable CFTR 45 39 C[C@@H]1CCCN1CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217948755 CF For-Sale Unstable HTR3A 15 43 C[C@@H]1CCCN1CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217948755 CF For-Sale Unstable LTA4H 15 42 C[C@@H]1CCCN1CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217948755 CF For-Sale Unstable HRH3 68 45 C[C@@H]1CCCN1CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217948755 CF For-Sale Unstable CHRNA10 50 35 C[C@@H]1CCCN1CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217948755 CF For-Sale Unstable ACKR3 60 41 C=CCNC(=O)N1[C@H](C(=O)O)C[C@@H]2CCCC[C@@H]21 ZINC000217948785 CD For-Sale Unstable ACE 16 57 C[C@H]1CCC[C@H]([C@@H](N)Cc2cc(Br)ccc2F)C1 ZINC000217948808 DI For-Sale Unstable DPP4 25 44 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc(Cl)c1 ZINC000217948830 GG For-Sale Unstable CFTR 45 39 C[C@H]1CCCN1CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217948832 CF For-Sale Unstable HTR3A 15 43 C[C@H]1CCCN1CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217948832 CF For-Sale Unstable LTA4H 15 42 C[C@H]1CCCN1CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217948832 CF For-Sale Unstable HRH3 68 45 C[C@H]1CCCN1CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217948832 CF For-Sale Unstable CHRNA10 50 35 C[C@H]1CCCN1CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217948832 CF For-Sale Unstable ACKR3 60 41 COc1ccccc1OCC(=O)NCCCN1CCCc2ccccc21 ZINC000217948843 FG In-Stock Unstable HTR1A 49 44 COc1ccccc1OCC(=O)NCCCN1CCCc2ccccc21 ZINC000217948843 FG In-Stock Unstable DRD2 45 46 COc1ccccc1OCC(=O)NCCCN1CCCc2ccccc21 ZINC000217948843 FG In-Stock Unstable DRD4 25 46 COc1ccccc1OCC(=O)NCCCN1CCCc2ccccc21 ZINC000217948843 FG In-Stock Unstable ADRA1D 38 42 COc1ccccc1OCC(=O)NCCCN1CCCc2ccccc21 ZINC000217948843 FG In-Stock Unstable HTR2A 29 42 COc1ccccc1OCC(=O)NCCCN1CCCc2ccccc21 ZINC000217948843 FG In-Stock Unstable ADRA1A 31 50 COc1ccccc1OCC(=O)NCCCN1CCCc2ccccc21 ZINC000217948843 FG In-Stock Unstable ADRA1B 19 41 COc1ccccc1OCC(=O)NCCCN1CCCc2ccccc21 ZINC000217948843 FG In-Stock Unstable DRD3 53 45 COc1ccccc1OCC(=O)NCCCN1CCCc2ccccc21 ZINC000217948843 FG In-Stock Unstable HTR7 45 41 COc1ccccc1OCC(=O)NCCCN1CCCc2ccccc21 ZINC000217948843 FG In-Stock Unstable MTNR1C 0 40 COc1ccccc1OCC(=O)NCCCN1CCCc2ccccc21 ZINC000217948843 FG In-Stock Unstable TYRO3 24 41 COc1cccc(/C=C/NC(=O)N2C[C@@]3(C)C[C@H]2CC(C)(C)C3)c1 ZINC000217948844 EI For-Sale Unstable AVPR2 17 47 COc1cccc(/C=C/NC(=O)N2C[C@@]3(C)C[C@H]2CC(C)(C)C3)c1 ZINC000217948844 EI For-Sale Unstable AVPR1A 36 41 C=CCNC(=O)N1[C@H](C(=O)O)C[C@H]2CCCC[C@@H]21 ZINC000217948869 CD For-Sale Unstable ACE 16 57 C[C@@H]1CCC[C@@H]([C@@H](N)Cc2cc(Br)ccc2F)C1 ZINC000217948883 DI For-Sale Unstable DPP4 25 44 COCCn1ccc2ccc(C(=O)NCCn3ccc4cc(OC)ccc43)cc21 ZINC000217948886 GH In-Stock Unstable DRD4 50 38 COCCn1ccc2ccc(C(=O)NCCn3ccc4cc(OC)ccc43)cc21 ZINC000217948886 GH In-Stock Unstable NQO2 17 40 COCCn1ccc2ccc(C(=O)NCCn3ccc4cc(OC)ccc43)cc21 ZINC000217948886 GH In-Stock Unstable MTNR1A 41 44 COCCn1ccc2ccc(C(=O)NCCn3ccc4cc(OC)ccc43)cc21 ZINC000217948886 GH In-Stock Unstable MTNR1B 28 44 COc1cc(Br)c(/C=C\C(=O)CCl)cc1OC ZINC000217948888 DG For-Sale Unstable CYSP_PLAFA 46 33 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc(Cl)c1 ZINC000217948917 GG For-Sale Unstable CFTR 45 39 C[C@@H]1CCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217948937 CF On-Demand Unstable ESR1 16 43 C[C@@H]1CCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217948937 CF On-Demand Unstable HTR3A 16 46 C[C@@H]1CCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217948937 CF On-Demand Unstable KCNH2 0 44 C[C@@H]1CCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217948937 CF On-Demand Unstable LTA4H 35 47 C[C@@H]1CCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217948937 CF On-Demand Unstable HRH3 88 49 C[C@@H]1CCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217948937 CF On-Demand Unstable PSMB1 40 35 C[C@H]1CCC[C@@H]([C@@H](N)Cc2cc(Br)ccc2F)C1 ZINC000217948955 DI For-Sale Unstable DPP4 25 44 COc1ccc(CN(C)C(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1 ZINC000217948964 EJ In-Stock Unstable TRPV1 0 45 COc1ccc(CN(C)C(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1 ZINC000217948964 EJ In-Stock Unstable CYP24A1 19 43 COc1ccc(CN(C)C(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1 ZINC000217948964 EJ In-Stock Unstable CYP27B1 25 43 COc1ccc(CN(C)C(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1 ZINC000217948964 EJ In-Stock Unstable GPR183 0 40 O=C(/C=C\c1ccc(N2CCCC2=O)cc1)CCl ZINC000217948965 CF For-Sale Unstable AKR1C3 0 41 Cn1cccc1[C@H](O)CCNC(=O)C(=O)Nc1ccc(OC(F)(F)F)cc1 ZINC000217948994 GE In-Stock Unstable P2RY1 59 38 Cn1cccc1[C@H](O)CCNC(=O)C(=O)Nc1ccc(OC(F)(F)F)cc1 ZINC000217948994 GE In-Stock Unstable EPHX2 49 39 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc(Cl)c1 ZINC000217949010 GG For-Sale Unstable CFTR 45 39 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217949014 DK For-Sale Unstable TRPM8 15 45 C[C@H]1CCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217949025 CF On-Demand Unstable ESR1 16 43 C[C@H]1CCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217949025 CF On-Demand Unstable HTR3A 16 46 C[C@H]1CCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217949025 CF On-Demand Unstable KCNH2 0 44 C[C@H]1CCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217949025 CF On-Demand Unstable LTA4H 35 47 C[C@H]1CCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217949025 CF On-Demand Unstable HRH3 88 49 C[C@H]1CCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217949025 CF On-Demand Unstable PSMB1 40 35 CCOC(=O)c1cnn(-c2ccc(F)cc2C)c1O ZINC000217949028 CE For-Sale Unstable HPD 29 43 CCOC(=O)c1cnn(-c2ccc(F)cc2C)c1O ZINC000217949028 CE For-Sale Unstable GABRA4 23 41 CCOC(=O)c1cnn(-c2ccc(F)cc2C)c1O ZINC000217949028 CE For-Sale Unstable GABRA5 27 41 COc1cccc(/C=C/NC(=O)Nc2cccc(N(C)C)c2)c1 ZINC000217949055 DH For-Sale Unstable MTNR1A 32 53 COc1cccc(/C=C/NC(=O)Nc2cccc(N(C)C)c2)c1 ZINC000217949055 DH For-Sale Unstable MTNR1B 34 53 COc1cccc(/C=C/NC(=O)Nc2cccc(N(C)C)c2)c1 ZINC000217949055 DH For-Sale Unstable KCNK3 28 40 CS(=O)(=O)Nc1ccc(/C=C\C(=O)CCl)cc1 ZINC000217949058 CD For-Sale Unstable TRPV1 17 40 CS(=O)(=O)Nc1ccc(/C=C\C(=O)CCl)cc1 ZINC000217949058 CD For-Sale Unstable HDAC8 16 44 CS(=O)(=O)Nc1ccc(/C=C\C(=O)CCl)cc1 ZINC000217949058 CD For-Sale Unstable HDAC1 0 44 CS(=O)(=O)Nc1ccc(/C=C\C(=O)CCl)cc1 ZINC000217949058 CD For-Sale Unstable SSSIM 15 45 Cn1cccc1[C@@H](O)CCNC(=O)C(=O)Nc1ccc(OC(F)(F)F)cc1 ZINC000217949064 GE In-Stock Unstable P2RY1 59 38 Cn1cccc1[C@@H](O)CCNC(=O)C(=O)Nc1ccc(OC(F)(F)F)cc1 ZINC000217949064 GE In-Stock Unstable EPHX2 49 39 COc1ccc(N2CCN(C(=O)/C=C/c3ccc(C(C)(C)C)cc3)CC2)cc1 ZINC000217949078 GI In-Stock Unstable PDK1 22 41 COc1ccc(N2CCN(C(=O)/C=C/c3ccc(C(C)(C)C)cc3)CC2)cc1 ZINC000217949078 GI In-Stock Unstable GPR183 0 63 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217949086 DK For-Sale Unstable TRPM8 15 45 C[C@H]1CN(Cc2ccccc2/C=C\C(=O)O)C[C@@H](C)O1 ZINC000217949105 CE For-Sale Unstable PTGER2 43 46 C[C@H]1CN(Cc2ccccc2/C=C\C(=O)O)C[C@@H](C)O1 ZINC000217949105 CE For-Sale Unstable PTGER4 20 46 C[C@H]1CN(Cc2ccccc2/C=C\C(=O)O)C[C@@H](C)O1 ZINC000217949105 CE For-Sale Unstable PTGER3 18 46 C[C@H]1CN(Cc2ccccc2/C=C\C(=O)O)C[C@@H](C)O1 ZINC000217949105 CE For-Sale Unstable PTGDR 17 44 COc1ccc(/C=C\C(=O)CCl)cc1C ZINC000217949127 BF For-Sale Unstable APP 20 40 COc1ccc(/C=C\C(=O)CCl)cc1C ZINC000217949127 BF For-Sale Unstable CA14 0 45 COc1ccc(/C=C\C(=O)CCl)cc1C ZINC000217949127 BF For-Sale Unstable CYP1A1 18 40 COc1ccc(/C=C\C(=O)CCl)cc1C ZINC000217949127 BF For-Sale Unstable TUBB1 67 45 COc1ccc(/C=C\C(=O)CCl)cc1C ZINC000217949127 BF For-Sale Unstable PTPA 0 41 COc1ccc(/C=C\C(=O)CCl)cc1C ZINC000217949127 BF For-Sale Unstable ABCG2 19 45 COc1ccc(/C=C\C(=O)CCl)cc1C ZINC000217949127 BF For-Sale Unstable NFE2L2 0 43 Cc1cc(F)ccc1-n1ncc(C(=O)O)c1O ZINC000217949132 BD For-Sale Unstable HPD 22 47 CC[C@@H](CCO)NC(=O)CCCCN ZINC000217949157 BC For-Sale Unstable PLA2G2C 0 43 CC[C@@H](CCO)NC(=O)CCCCN ZINC000217949157 BC For-Sale Unstable NMT1 31 42 CC[C@@H](CCO)NC(=O)CCCCN ZINC000217949157 BC For-Sale Unstable Q6UB75_PIG 0 40 CC[C@@H](CCO)NC(=O)CCCCN ZINC000217949157 BC For-Sale Unstable NOD1 65 48 CC(C)C1CCN(c2ccccc2CBr)CC1 ZINC000217949162 CI For-Sale Unstable KCNQ2 41 33 COc1cccc(/C=C/NC(=O)Nc2nc3c(s2)CN(C)CC3)c1 ZINC000217949165 EF For-Sale Unstable F10 24 41 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217949172 DK For-Sale Unstable TRPM8 15 45 CC(C)(C)c1ccc(/C=C/C(=O)Nc2ccc(CSc3ccccc3)cc2)cc1 ZINC000217949178 HK In-Stock Unstable TRPV1 27 69 CC(C)(C)c1ccc(/C=C/C(=O)Nc2ccc(CSc3ccccc3)cc2)cc1 ZINC000217949178 HK In-Stock Unstable HDAC8 25 49 CC(C)(C)c1ccc(/C=C/C(=O)Nc2ccc(CSc3ccccc3)cc2)cc1 ZINC000217949178 HK In-Stock Unstable MMP2 23 51 CC(C)(C)c1ccc(/C=C/C(=O)Nc2ccc(CSc3ccccc3)cc2)cc1 ZINC000217949178 HK In-Stock Unstable HDAC1 25 46 CC(C)(C)c1ccc(/C=C/C(=O)Nc2ccc(CSc3ccccc3)cc2)cc1 ZINC000217949178 HK In-Stock Unstable HDAC6 20 40 CC(C)(C)c1ccc(/C=C/C(=O)Nc2ccc(CSc3ccccc3)cc2)cc1 ZINC000217949178 HK In-Stock Unstable MMP9 19 51 CC(C)(C)c1ccc(/C=C/C(=O)Nc2ccc(CSc3ccccc3)cc2)cc1 ZINC000217949178 HK In-Stock Unstable IMPDH2 0 48 CC(C)(C)c1ccc(/C=C/C(=O)Nc2ccc(CSc3ccccc3)cc2)cc1 ZINC000217949178 HK In-Stock Unstable MMP1 25 49 CC(C)(C)c1ccc(/C=C/C(=O)Nc2ccc(CSc3ccccc3)cc2)cc1 ZINC000217949178 HK In-Stock Unstable MCHR1 0 46 CC[C@H](CCO)NC(=O)CCCCN ZINC000217949231 BC For-Sale Unstable PLA2G2C 0 43 CC[C@H](CCO)NC(=O)CCCCN ZINC000217949231 BC For-Sale Unstable NMT1 31 42 CC[C@H](CCO)NC(=O)CCCCN ZINC000217949231 BC For-Sale Unstable Q6UB75_PIG 0 40 CC[C@H](CCO)NC(=O)CCCCN ZINC000217949231 BC For-Sale Unstable NOD1 65 48 O=C(Cc1ccccc1Br)NCC1C[C@@H]2CC[C@H](C1)N2 ZINC000217949238 EF For-Sale Unstable CA9 18 43 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217949253 DK For-Sale Unstable TRPM8 15 45 C=CCN(CC=C)C(=O)N1[C@H](C(=O)O)C[C@@H]2CCCC[C@@H]21 ZINC000217949278 CE For-Sale Unstable ACE 15 53 COc1cccc(/C=C/NC(=O)Nc2ccc3nc[nH]c3c2)c1 ZINC000217949282 DG For-Sale Unstable MTNR1A 18 40 COc1cccc(/C=C/NC(=O)Nc2ccc3nc[nH]c3c2)c1 ZINC000217949282 DG For-Sale Unstable MTNR1B 22 40 Cc1cccc(CSCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)c1 ZINC000217949288 FK In-Stock Unstable HDAC8 32 41 O=C(/C=C\c1cc2c(cc1F)NC(=O)CC2)CCl ZINC000217949289 CF For-Sale Unstable PKM 35 41 Cn1cccc1[C@H](O)CCNC(=O)Nc1ccccc1 ZINC000217949333 CE In-Stock Unstable CCR3 17 41 Cn1cccc1[C@H](O)CCNC(=O)Nc1ccccc1 ZINC000217949333 CE In-Stock Unstable ACAT 0 43 Cn1cccc1[C@H](O)CCNC(=O)Nc1ccccc1 ZINC000217949333 CE In-Stock Unstable P95276_MYCTO 0 41 CCOC(=O)c1cnn(-c2cc(F)c(F)cc2F)c1O ZINC000217949353 CE For-Sale Unstable Q9FYV8_MAIZE 17 40 C[C@@H]1CCC[C@H]([C@@H](N)Cc2ccc(F)cc2Cl)C1 ZINC000217949354 CI For-Sale Unstable DPP4 19 40 C=CCN(CC=C)C(=O)N1[C@H](C(=O)O)C[C@H]2CCCC[C@@H]21 ZINC000217949369 CE For-Sale Unstable ACE 15 53 COc1ccc(/C=C\C(=O)CCl)cc1F ZINC000217949370 BF For-Sale Unstable TUBB1 66 52 COc1ccc(/C=C\C(=O)CCl)cc1F ZINC000217949370 BF For-Sale Unstable PTPA 0 40 COc1ccc(/C=C\C(=O)CCl)cc1F ZINC000217949370 BF For-Sale Unstable ABCG2 18 44 COc1ccc(/C=C\C(=O)CCl)cc1F ZINC000217949370 BF For-Sale Unstable NFE2L2 0 55 COc1ccc(/C=C\C(=O)CCl)cc1F ZINC000217949370 BF For-Sale Unstable CYSP_PLAFA 43 39 CC(C)C1CCN(c2ccc(CBr)cc2F)CC1 ZINC000217949380 DJ For-Sale Unstable NPY2R 42 37 CC(C)(C)c1ccc(/C=C/C(=O)NCCSCc2ccc(Cl)cc2Cl)cc1 ZINC000217949389 HK In-Stock Unstable PYGL 25 54 Cn1cccc1[C@@H](O)CCNC(=O)Nc1ccccc1 ZINC000217949425 CE In-Stock Unstable CCR3 17 41 Cn1cccc1[C@@H](O)CCNC(=O)Nc1ccccc1 ZINC000217949425 CE In-Stock Unstable ACAT 0 43 Cn1cccc1[C@@H](O)CCNC(=O)Nc1ccccc1 ZINC000217949425 CE In-Stock Unstable P95276_MYCTO 0 41 C[C@H]1CCC[C@H]([C@@H](N)Cc2ccc(F)cc2Cl)C1 ZINC000217949452 CI For-Sale Unstable DPP4 19 40 COc1cccc(/C=C/NC(=O)Nc2ccccc2C(N)=O)c1 ZINC000217949504 DF For-Sale Unstable MAPK10 16 42 COc1cccc(/C=C/NC(=O)Nc2ccccc2C(N)=O)c1 ZINC000217949504 DF For-Sale Unstable AKR1C3 15 44 COC(=O)c1ccc(C)c(NC(=O)/C=C/c2ccc(C(C)(C)C)cc2)c1 ZINC000217949505 FJ In-Stock Unstable TRPV1 15 57 COC(=O)c1ccc(C)c(NC(=O)/C=C/c2ccc(C(C)(C)C)cc2)c1 ZINC000217949505 FJ In-Stock Unstable MMP2 18 47 COC(=O)c1ccc(C)c(NC(=O)/C=C/c2ccc(C(C)(C)C)cc2)c1 ZINC000217949505 FJ In-Stock Unstable MMP9 15 47 COC(=O)c1ccc(C)c(NC(=O)/C=C/c2ccc(C(C)(C)C)cc2)c1 ZINC000217949505 FJ In-Stock Unstable IMPDH2 0 45 COc1cccc(S(=O)(=O)Br)c1 ZINC000217949519 CD For-Sale Unstable MTNR1B 26 43 C[C@@H]1CCC[C@@H]([C@@H](N)Cc2ccc(F)cc2Cl)C1 ZINC000217949530 CI For-Sale Unstable DPP4 19 40 C[C@H]1CCC[C@@H]([C@@H](N)Cc2ccc(F)cc2Cl)C1 ZINC000217949602 CI For-Sale Unstable DPP4 19 40 CC(C)(C)c1ccc(/C=C/C(=O)NCCSCc2ccc(Cl)c(Cl)c2)cc1 ZINC000217949613 HK In-Stock Unstable TRPV1 21 46 CC(C)(C)c1ccc(/C=C/C(=O)NCCSCc2ccc(Cl)c(Cl)c2)cc1 ZINC000217949613 HK In-Stock Unstable PYGL 29 64 COc1cccc(/C=C/NC(=O)NCCN(C)C)c1 ZINC000217949618 CD For-Sale Unstable DRD4 41 31 COc1cccc(/C=C/NC(=O)NCCN(C)C)c1 ZINC000217949618 CD For-Sale Unstable MTNR1A 82 45 COc1cccc(/C=C/NC(=O)NCCN(C)C)c1 ZINC000217949618 CD For-Sale Unstable MTNR1B 72 45 Cn1cc(/C=C\c2csc(N)n2)c2ccccc21 ZINC000217949714 CG For-Sale Unstable IMPDH2 21 47 CN(Cc1ccccc1)Cc1ccccc1/C=C\C(=O)O ZINC000217949738 CG For-Sale Unstable PTGER2 61 51 CN(Cc1ccccc1)Cc1ccccc1/C=C\C(=O)O ZINC000217949738 CG For-Sale Unstable PTGER4 28 46 CN(Cc1ccccc1)Cc1ccccc1/C=C\C(=O)O ZINC000217949738 CG For-Sale Unstable PTGER3 24 52 COc1cccc(/C=C/NC(=O)Nc2cccc(Br)c2)c1 ZINC000217949742 EI For-Sale Unstable MTNR1A 25 46 COc1cccc(/C=C/NC(=O)Nc2cccc(Br)c2)c1 ZINC000217949742 EI For-Sale Unstable MTNR1B 31 46 COc1cccc(/C=C/NC(=O)Nc2cccc(Br)c2)c1 ZINC000217949742 EI For-Sale Unstable TAAR1 31 43 C[C@H](C(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)c1ccc(C[C@@H]2CCCC2=O)cc1 ZINC000217949744 HH In-Stock Unstable CHRNA4 36 46 Cn1cccc1[C@H](O)CCNC(=O)NC1CCCCC1 ZINC000217949750 CE In-Stock Unstable CNR1 16 40 Cn1cccc1[C@H](O)CCNC(=O)NC1CCCCC1 ZINC000217949750 CE In-Stock Unstable EPHX2 34 45 CCOC(=O)c1cnn(-c2ccc(Cl)c(F)c2)c1O ZINC000217949801 CF For-Sale Unstable Q9FYV8_MAIZE 44 44 CC(C)(C)SCCNC(=O)/C=C/c1ccc(C(C)(C)C)cc1 ZINC000217949832 DJ In-Stock Unstable PYGL 0 48 CC(C)(C)SCCNC(=O)/C=C/c1ccc(C(C)(C)C)cc1 ZINC000217949832 DJ In-Stock Unstable HDAC8 0 45 CC(C)(C)SCCNC(=O)/C=C/c1ccc(C(C)(C)C)cc1 ZINC000217949832 DJ In-Stock Unstable HDAC1 0 45 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CSc1nc2ccccc2o1 ZINC000217949834 IG For-Sale Unstable HCRTR1 21 43 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CSc1nc2ccccc2o1 ZINC000217949834 IG For-Sale Unstable HCRTR2 23 43 Cn1cccc1[C@@H](O)CCNC(=O)NC1CCCCC1 ZINC000217949838 CE In-Stock Unstable CNR1 16 40 Cn1cccc1[C@@H](O)CCNC(=O)NC1CCCCC1 ZINC000217949838 CE In-Stock Unstable EPHX2 34 45 CN(Cc1ccccc1)Cc1ccc(/C=C\C(=O)O)cc1 ZINC000217949842 CG For-Sale Unstable ACHE 0 49 CN(Cc1ccccc1)Cc1ccc(/C=C\C(=O)O)cc1 ZINC000217949842 CG For-Sale Unstable PTGER2 32 44 CN(Cc1ccccc1)Cc1ccc(/C=C\C(=O)O)cc1 ZINC000217949842 CG For-Sale Unstable PTGER4 0 44 CN(Cc1ccccc1)Cc1ccc(/C=C\C(=O)O)cc1 ZINC000217949842 CG For-Sale Unstable G6PC 42 34 CN(Cc1ccccc1)Cc1ccc(/C=C\C(=O)O)cc1 ZINC000217949842 CG For-Sale Unstable F3 24 43 CN(Cc1ccccc1)Cc1ccc(/C=C\C(=O)O)cc1 ZINC000217949842 CG For-Sale Unstable NR1H4 30 41 CN(Cc1ccccc1)Cc1ccc(/C=C\C(=O)O)cc1 ZINC000217949842 CG For-Sale Unstable HDAC1 22 45 CN(Cc1ccccc1)Cc1ccc(/C=C\C(=O)O)cc1 ZINC000217949842 CG For-Sale Unstable HDAC4 15 42 CN(Cc1ccccc1)Cc1ccc(/C=C\C(=O)O)cc1 ZINC000217949842 CG For-Sale Unstable HDAC6 23 42 CN(Cc1ccccc1)Cc1ccc(/C=C\C(=O)O)cc1 ZINC000217949842 CG For-Sale Unstable 17HSDCL 0 44 CN(Cc1ccccc1)Cc1ccc(/C=C\C(=O)O)cc1 ZINC000217949842 CG For-Sale Unstable AKR1C3 32 42 CN(Cc1ccccc1)Cc1ccc(/C=C\C(=O)O)cc1 ZINC000217949842 CG For-Sale Unstable LGB 0 40 CN(Cc1ccccc1)Cc1ccc(/C=C\C(=O)O)cc1 ZINC000217949842 CG For-Sale Unstable AKR1B10 18 44 CN(Cc1ccccc1)Cc1ccc(/C=C\C(=O)O)cc1 ZINC000217949842 CG For-Sale Unstable GPR183 0 42 COC(=O)C[C@H](c1ccc(C)o1)c1oc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c1O ZINC000217949844 JF In-Stock Unstable CHRNA4 27 45 Cc1ccc(CN2CC[C@@H](C)NC[C@@H](C)C2)cn1 ZINC000217949851 BE For-Sale Unstable MLNR 44 35 CCN1CCN(C(=O)N/C=C/c2cccc(OC)c2)CC1 ZINC000217949858 CE For-Sale Unstable DRD4 47 36 CCN1CCN(C(=O)N/C=C/c2cccc(OC)c2)CC1 ZINC000217949858 CE For-Sale Unstable MTNR1A 38 41 CCN1CCN(C(=O)N/C=C/c2cccc(OC)c2)CC1 ZINC000217949858 CE For-Sale Unstable MTNR1B 44 41 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CSc1nc2ccccc2o1 ZINC000217949911 IG For-Sale Unstable HCRTR1 21 43 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CSc1nc2ccccc2o1 ZINC000217949911 IG For-Sale Unstable HCRTR2 23 43 O=C(O)c1cnn(-c2ccc(Cl)c(F)c2)c1O ZINC000217949916 CE For-Sale Anodyne AKR1C1 41 33 O=C(O)c1cnn(-c2ccc(Cl)c(F)c2)c1O ZINC000217949916 CE For-Sale Anodyne RPA1 48 38 COC(=O)C[C@@H](c1ccc(C)o1)c1oc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c1O ZINC000217949919 JF In-Stock Unstable CHRNA4 27 45 Cc1ccc(CN2CC[C@H](C)NC[C@@H](C)C2)cn1 ZINC000217949932 BE For-Sale Unstable MLNR 44 35 Cc1ccccc1NC(=O)NCC[C@H](O)c1cccn1C ZINC000217949949 CF In-Stock Unstable ACAT 0 43 CCOc1ccc(CCNC(=O)N/C=C/c2cccc(OC)c2)cc1OCC ZINC000217949968 GI For-Sale Unstable MTNR1A 89 46 CCOc1ccc(CCNC(=O)N/C=C/c2cccc(OC)c2)cc1OCC ZINC000217949968 GI For-Sale Unstable MTNR1B 81 46 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CSc1nc2ccccc2o1 ZINC000217949988 IG For-Sale Unstable HCRTR1 21 43 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CSc1nc2ccccc2o1 ZINC000217949988 IG For-Sale Unstable HCRTR2 23 43 CC(C)C1CCN(c2ccc(CBr)cc2)CC1 ZINC000217950007 CI For-Sale Unstable L3MBTL3 41 42 Cc1cc(C(=O)NCCc2ccncc2)cc(=O)[nH]1 ZINC000217950020 CD In-Stock Unstable CNR2 23 45 Cc1cc(C(=O)NCCc2ccncc2)cc(=O)[nH]1 ZINC000217950020 CD In-Stock Unstable KDM4E 21 42 Cc1ccccc1NC(=O)NCC[C@@H](O)c1cccn1C ZINC000217950028 CF In-Stock Unstable ACAT 0 43 CCOC(=O)c1cnn(-c2cc(F)c(F)c(F)c2)c1O ZINC000217950034 CE For-Sale Unstable HPD 45 34 CC[C@@H]1CCN(Cc2ccnc(OC)c2)CC[C@@H](C)N1 ZINC000217950037 CE For-Sale Unstable SSTR5 65 36 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)c1 ZINC000217950056 FK In-Stock Unstable TRPV1 29 52 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)c1 ZINC000217950056 FK In-Stock Unstable HDAC8 33 41 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)c1 ZINC000217950056 FK In-Stock Unstable HDAC1 0 40 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)c1 ZINC000217950056 FK In-Stock Unstable PDS 50 36 COc1cccc(/C=C/NC(=O)Nc2ccc(C(C)(C)C)cc2)c1 ZINC000217950065 DJ For-Sale Unstable TRPV1 19 55 COc1cccc(/C=C/NC(=O)Nc2ccc(C(C)(C)C)cc2)c1 ZINC000217950065 DJ For-Sale Unstable RAF1 29 44 COc1cccc(/C=C/NC(=O)Nc2ccc(C(C)(C)C)cc2)c1 ZINC000217950065 DJ For-Sale Unstable MTNR1A 26 49 COc1cccc(/C=C/NC(=O)Nc2ccc(C(C)(C)C)cc2)c1 ZINC000217950065 DJ For-Sale Unstable MTNR1B 32 49 COc1cccc(/C=C/NC(=O)Nc2ccc(C(C)(C)C)cc2)c1 ZINC000217950065 DJ For-Sale Unstable Q8MMZ8_EIMTE 36 44 COc1cccc(/C=C/NC(=O)Nc2ccc(C(C)(C)C)cc2)c1 ZINC000217950065 DJ For-Sale Unstable AKR1C3 20 42 COc1cccc(/C=C/NC(=O)Nc2ccc(C(C)(C)C)cc2)c1 ZINC000217950065 DJ For-Sale Unstable AKR1C2 38 42 COc1cccc(/C=C/NC(=O)Nc2ccc(C(C)(C)C)cc2)c1 ZINC000217950065 DJ For-Sale Unstable IMDH_CRYPV 48 44 CN(Cc1ccccc1/C=C\C(=O)O)C1CCOCC1 ZINC000217950081 CE For-Sale Unstable PTGER2 43 48 CN(Cc1ccccc1/C=C\C(=O)O)C1CCOCC1 ZINC000217950081 CE For-Sale Unstable PTGER4 21 48 CN(Cc1ccccc1/C=C\C(=O)O)C1CCOCC1 ZINC000217950081 CE For-Sale Unstable PTGER3 18 48 CN(Cc1ccccc1/C=C\C(=O)O)C1CCOCC1 ZINC000217950081 CE For-Sale Unstable PTGDR 17 44 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CSc1nc2ccccc2o1 ZINC000217950082 IG For-Sale Unstable HCRTR1 21 43 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CSc1nc2ccccc2o1 ZINC000217950082 IG For-Sale Unstable HCRTR2 23 43 CC[C@H]1CCN(Cc2ccnc(OC)c2)CC[C@@H](C)N1 ZINC000217950131 CE For-Sale Unstable SSTR5 65 36 COc1ccc(CNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)c(OC)c1OC ZINC000217950152 GI In-Stock Unstable TRPV1 33 55 COc1ccc(CNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)c(OC)c1OC ZINC000217950152 GI In-Stock Unstable HDAC8 0 40 COc1ccc(CNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)c(OC)c1OC ZINC000217950152 GI In-Stock Unstable TUBB1 42 40 COc1ccc(CNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)c(OC)c1OC ZINC000217950152 GI In-Stock Unstable MT-ND1 24 42 COc1cccc(/C=C/NC(=O)Nc2nc[nH]n2)c1 ZINC000217950183 CD For-Sale Unstable MTNR1A 23 41 COc1cccc(/C=C/NC(=O)Nc2nc[nH]n2)c1 ZINC000217950183 CD For-Sale Unstable MTNR1B 27 41 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)NCc3cccnc3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217950216 KF In-Stock Unstable NPY2R 44 34 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)NCc3cccnc3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217950216 KF In-Stock Unstable HSD17B1 0 40 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)NCc3cccnc3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217950216 KF In-Stock Unstable TUBA1A 19 65 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)NCc3cccnc3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217950216 KF In-Stock Unstable TPPP 0 62 CCOc1ccc(CNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1OCC ZINC000217950252 GK In-Stock Unstable TRPV1 39 56 CCOc1ccc(CNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1OCC ZINC000217950252 GK In-Stock Unstable HDAC8 0 44 CCOc1ccc(CNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1OCC ZINC000217950252 GK In-Stock Unstable HDAC1 0 41 CCOc1ccc(CNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1OCC ZINC000217950252 GK In-Stock Unstable MT-ND1 26 44 CCOc1ccc(CNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1OCC ZINC000217950252 GK In-Stock Unstable AKR1C3 15 40 Cn1cccc1[C@H](O)CCNC(=O)NCCc1ccccc1 ZINC000217950291 DD In-Stock Unstable AMP1_PLAFQ 27 42 COc1cccc(/C=C/NC(=O)Nc2nc(C)c(C)s2)c1 ZINC000217950294 DH For-Sale Unstable MTNR1A 20 40 COc1cccc(/C=C/NC(=O)Nc2nc(C)c(C)s2)c1 ZINC000217950294 DH For-Sale Unstable MTNR1B 24 40 C[C@@H]1CCC[C@H]([C@@H](N)Cc2ccc(F)cc2Br)C1 ZINC000217950322 DI For-Sale Unstable DPP4 18 40 COc1ccc2cc(/C=C\c3csc(N)n3)ccc2c1 ZINC000217950324 CI For-Sale Unstable CYP1B1 58 43 COc1ccc2cc(/C=C\c3csc(N)n3)ccc2c1 ZINC000217950324 CI For-Sale Unstable AHR 37 43 COc1ccc2cc(/C=C\c3csc(N)n3)ccc2c1 ZINC000217950324 CI For-Sale Unstable CYP1A1 41 43 COc1cc(C)c(CS(=O)(=O)Cl)c(C)c1 ZINC000217950351 BE For-Sale Unstable FFAR4 17 42 Cn1cccc1[C@@H](O)CCNC(=O)NCCc1ccccc1 ZINC000217950369 DD In-Stock Unstable AMP1_PLAFQ 27 42 COc1cc(CNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)ccc1OC(C)C ZINC000217950375 GK In-Stock Unstable TRPV1 43 55 COc1cc(CNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)ccc1OC(C)C ZINC000217950375 GK In-Stock Unstable MT-ND1 30 51 Cc1noc2nc(C(C)C)cc(C(=O)Nc3ccc(Cl)c(S(=O)(=O)N4CCCCC4)c3)c12 ZINC000217950386 JJ On-Demand Unstable NR1H4 18 41 Cc1noc2nc(C(C)C)cc(C(=O)Nc3ccc(Cl)c(S(=O)(=O)N4CCCCC4)c3)c12 ZINC000217950386 JJ On-Demand Unstable NR2E3 44 32 CN(CCOc1ccc(/C=C\C(=O)O)cc1)CC1CC1 ZINC000217950387 CF On-Demand Unstable LSS 29 50 COc1cccc(/C=C/NC(=O)NCC(OC)OC)c1 ZINC000217950389 CD For-Sale Unstable MTNR1A 63 46 COc1cccc(/C=C/NC(=O)NCC(OC)OC)c1 ZINC000217950389 CD For-Sale Unstable MTNR1B 60 46 C[C@H]1CCC[C@H]([C@@H](N)Cc2ccc(F)cc2Br)C1 ZINC000217950403 DI For-Sale Unstable DPP4 18 40 CC[C@@H]1CCN(Cc2ccc(OC)nc2)CC[C@@H](C)N1 ZINC000217950436 CE For-Sale Unstable SSTR5 47 35 Cc1c(N[C@H]2C[C@H](C)CC[C@H]2C(C)C)cccc1[N+](=O)[O-] ZINC000217950465 CJ For-Sale Unstable SERPINE1 40 41 Cc1c(N[C@H]2C[C@H](C)CC[C@H]2C(C)C)cccc1[N+](=O)[O-] ZINC000217950465 CJ For-Sale Unstable TRPM8 16 41 Cn1cccc1[C@H](O)CCNC(=O)Nc1ccccc1Cl ZINC000217950475 DF In-Stock Unstable CXCL8 45 37 Cn1cccc1[C@H](O)CCNC(=O)Nc1ccccc1Cl ZINC000217950475 DF In-Stock Unstable PTGER3 16 43 CC(C)(C)c1ccc(/C=C/C(=O)NCCCc2ccccc2Cl)cc1 ZINC000217950479 FK In-Stock Unstable DRD3 15 41 CC(C)(C)c1ccc(/C=C/C(=O)NCCCc2ccccc2Cl)cc1 ZINC000217950479 FK In-Stock Unstable PYGL 27 50 CC(C)(C)c1ccc(/C=C/C(=O)NCCCc2ccccc2Cl)cc1 ZINC000217950479 FK In-Stock Unstable HDAC8 23 40 CC(C)(C)c1ccc(/C=C/C(=O)NCCCc2ccccc2Cl)cc1 ZINC000217950479 FK In-Stock Unstable HDAC1 23 40 CC(C)(C)c1ccc(/C=C/C(=O)NCCCc2ccccc2Cl)cc1 ZINC000217950479 FK In-Stock Unstable HDAC9 40 38 CC(C)(C)c1ccc(/C=C/C(=O)NCCCc2ccccc2Cl)cc1 ZINC000217950479 FK In-Stock Unstable HDAC7 51 38 C[C@@H]1CCC[C@@H]([C@@H](N)Cc2ccc(F)cc2Br)C1 ZINC000217950483 DI For-Sale Unstable DPP4 18 40 COc1cccc(/C=C/NC(=O)Nc2ccc3cn[nH]c3c2)c1 ZINC000217950495 DG For-Sale Unstable MTNR1A 22 40 COc1cccc(/C=C/NC(=O)Nc2ccc3cn[nH]c3c2)c1 ZINC000217950495 DG For-Sale Unstable MTNR1B 24 40 COc1cccc(/C=C/NC(=O)Nc2ccc3cn[nH]c3c2)c1 ZINC000217950495 DG For-Sale Unstable ROCK2 28 41 CC[C@H]1CCN(Cc2ccc(OC)nc2)CC[C@@H](C)N1 ZINC000217950521 CE For-Sale Unstable SSTR5 47 35 Cc1c(N[C@H]2C[C@@H](C)CC[C@H]2C(C)C)cccc1[N+](=O)[O-] ZINC000217950537 CJ For-Sale Unstable SERPINE1 40 41 Cc1c(N[C@H]2C[C@@H](C)CC[C@H]2C(C)C)cccc1[N+](=O)[O-] ZINC000217950537 CJ For-Sale Unstable TRPM8 16 41 Cn1cccc1[C@@H](O)CCNC(=O)Nc1ccccc1Cl ZINC000217950545 DF In-Stock Unstable CXCL8 45 37 Cn1cccc1[C@@H](O)CCNC(=O)Nc1ccccc1Cl ZINC000217950545 DF In-Stock Unstable PTGER3 16 43 C[C@H]1CCC[C@@H]([C@@H](N)Cc2ccc(F)cc2Br)C1 ZINC000217950547 DI For-Sale Unstable DPP4 18 40 CO[C@@H]1CCN(c2ccc(F)cc2CBr)C1 ZINC000217950570 CF For-Sale Unstable LIPG 52 39 CC(C)(C)c1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217950578 FK In-Stock Unstable TRPV1 25 51 CC(C)(C)c1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217950578 FK In-Stock Unstable PYGL 26 49 CC(C)(C)c1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217950578 FK In-Stock Unstable HDAC8 22 46 CC(C)(C)c1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217950578 FK In-Stock Unstable HDAC1 22 43 CC(C)(C)c1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217950578 FK In-Stock Unstable HDAC2 0 41 CC(C)(C)c1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217950578 FK In-Stock Unstable HDAC4 19 41 CC(C)(C)c1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217950578 FK In-Stock Unstable HDAC9 28 41 CC(C)(C)c1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217950578 FK In-Stock Unstable HDAC7 43 41 CC(C)(C)c1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217950578 FK In-Stock Unstable MMP1 0 41 CC(C)(C)c1ccc(/C=C/C(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217950578 FK In-Stock Unstable TRPM2 0 40 CN1CCC(=O)c2ccc(C(F)(F)F)cc21 ZINC000217950591 BF For-Sale Unstable SRD5A1 22 42 CCN(Cc1ccccc1/C=C\C(=O)O)C[C@@H]1CCCO1 ZINC000217950619 CF For-Sale Unstable OXTR 26 41 CCN(Cc1ccccc1/C=C\C(=O)O)C[C@@H]1CCCO1 ZINC000217950619 CF For-Sale Unstable AVPR1A 0 40 CCN(Cc1ccccc1/C=C\C(=O)O)C[C@@H]1CCCO1 ZINC000217950619 CF For-Sale Unstable PTGER2 33 40 CCN(Cc1ccccc1/C=C\C(=O)O)C[C@@H]1CCCO1 ZINC000217950619 CF For-Sale Unstable PTGER4 0 40 O=C(CCn1ccc2ccccc21)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217950620 FF In-Stock Unstable CHRNA4 42 55 CO[C@H]1CCN(c2ccc(F)cc2CBr)C1 ZINC000217950645 CF For-Sale Unstable LIPG 52 39 Cn1cccc1[C@H](O)CCNC(=O)Nc1ccc2c(c1)OCO2 ZINC000217950648 DD In-Stock Unstable NOS2 44 31 Cn1cccc1[C@H](O)CCNC(=O)Nc1ccc2c(c1)OCO2 ZINC000217950648 DD In-Stock Unstable CCR2 0 40 C[C@H](NC(=O)N[C@@H](C(=O)O)[C@H](C)O)c1ccccc1 ZINC000217950683 CC For-Sale Unstable MME 27 47 C[C@H](NC(=O)N[C@@H](C(=O)O)[C@H](C)O)c1ccccc1 ZINC000217950683 CC For-Sale Unstable ACACA 24 40 C[C@H](NC(=O)N[C@@H](C(=O)O)[C@H](C)O)c1ccccc1 ZINC000217950683 CC For-Sale Unstable MENB 0 40 CC(C)(C)c1ccc(/C=C/C(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217950692 EJ In-Stock Unstable TRPV1 22 53 CC(C)(C)c1ccc(/C=C/C(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217950692 EJ In-Stock Unstable PYGL 22 43 CC(C)(C)c1ccc(/C=C/C(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217950692 EJ In-Stock Unstable HDAC8 20 46 CC(C)(C)c1ccc(/C=C/C(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217950692 EJ In-Stock Unstable HDAC1 26 41 CC(C)(C)c1ccc(/C=C/C(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217950692 EJ In-Stock Unstable HDAC4 0 41 CC(C)(C)c1ccc(/C=C/C(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217950692 EJ In-Stock Unstable HDAC7 51 36 CC(C)(C)c1ccc(/C=C/C(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217950692 EJ In-Stock Unstable LEF 40 38 CC(C)(C)c1ccc(/C=C/C(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217950692 EJ In-Stock Unstable TRPM2 0 40 C[C@@H]1Cc2ccccc2[C@@H](c2ccccc2)[C@@H](C)N1 ZINC000217950725 CH For-Sale Unstable PRCP 47 38 Cn1cccc1[C@@H](O)CCNC(=O)Nc1ccc2c(c1)OCO2 ZINC000217950727 DD In-Stock Unstable NOS2 44 31 Cn1cccc1[C@@H](O)CCNC(=O)Nc1ccc2c(c1)OCO2 ZINC000217950727 DD In-Stock Unstable CCR2 0 40 COc1ccc(CN2C(=O)N[C@@H](CCC(=O)N3CCCC[C@H]3c3cccnc3)C2=O)cc1 ZINC000217950728 IG In-Stock Unstable COLA 117 41 COc1ccc(CN2C(=O)N[C@@H](CCC(=O)N3CCCC[C@H]3c3cccnc3)C2=O)cc1 ZINC000217950728 IG In-Stock Unstable CPT1A 109 41 COc1ccc(CN2C(=O)N[C@@H](CCC(=O)N3CCCC[C@H]3c3cccnc3)C2=O)cc1 ZINC000217950728 IG In-Stock Unstable GPBAR1 0 45 COc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217950729 GD For-Sale Unstable CA2 93 59 COc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217950729 GD For-Sale Unstable NQO2 28 40 COc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217950729 GD For-Sale Unstable CA1 80 59 COc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217950729 GD For-Sale Unstable CA7 53 59 COc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217950729 GD For-Sale Unstable CA5B 42 46 COc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217950729 GD For-Sale Unstable CA4 55 49 COc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217950729 GD For-Sale Unstable CA5A 43 46 COc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217950729 GD For-Sale Unstable CA14 49 47 COc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217950729 GD For-Sale Unstable MTNR1A 82 43 COc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217950729 GD For-Sale Unstable MTNR1B 72 43 COc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217950729 GD For-Sale Unstable CA12 65 55 COc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217950729 GD For-Sale Unstable CA9 75 59 COc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217950729 GD For-Sale Unstable UREA_CANEN 17 42 COc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217950729 GD For-Sale Unstable CYNT 25 43 COc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217950729 GD For-Sale Unstable NCE103 40 47 COc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217950729 GD For-Sale Unstable LIG1 0 41 COc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217950729 GD For-Sale Unstable P96878_MYCTU 47 42 COc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217950729 GD For-Sale Unstable CAN2 0 42 COc1cccc(/C=C/NC(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1 ZINC000217950729 GD For-Sale Unstable A6YCJ1_9METZ 17 45 CCN(Cc1ccc(/C=C\C(=O)O)cc1)C[C@@H]1CCCO1 ZINC000217950730 CF For-Sale Unstable OXTR 25 41 CCN(Cc1ccc(/C=C\C(=O)O)cc1)C[C@@H]1CCCO1 ZINC000217950730 CF For-Sale Unstable AVPR1A 0 41 O=C(c1ccc(N2CCCC2)cc1)N1CCC[C@@H](c2nnc[nH]2)C1 ZINC000217950770 EE In-Stock Unstable PREP 15 40 O=C(c1ccc(N2CCCC2)cc1)N1CCC[C@@H](c2nnc[nH]2)C1 ZINC000217950770 EE In-Stock Unstable L3MBTL1 0 46 O=C(c1ccc(N2CCCC2)cc1)N1CCC[C@@H](c2nnc[nH]2)C1 ZINC000217950770 EE In-Stock Unstable L3MBTL3 61 46 O=C(c1ccc(N2CCCC2)cc1)N1CCC[C@@H](c2nnc[nH]2)C1 ZINC000217950770 EE In-Stock Unstable L3MBTL4 0 46 O=C(c1ccc(N2CCCC2)cc1)N1CCC[C@@H](c2nnc[nH]2)C1 ZINC000217950770 EE In-Stock Unstable MBTD1 0 46 O=C(c1ccc(N2CCCC2)cc1)N1CCC[C@@H](c2nnc[nH]2)C1 ZINC000217950770 EE In-Stock Unstable TP53BP1 0 46 C[C@H](NC(=O)N[C@H](C(=O)O)[C@H](C)O)c1ccccc1 ZINC000217950782 CC For-Sale Unstable MME 27 47 C[C@H](NC(=O)N[C@H](C(=O)O)[C@H](C)O)c1ccccc1 ZINC000217950782 CC For-Sale Unstable ACACA 24 40 C[C@H](NC(=O)N[C@H](C(=O)O)[C@H](C)O)c1ccccc1 ZINC000217950782 CC For-Sale Unstable MENB 0 40 COc1ccccc1CCCNC(=O)/C=C/c1ccc(C(C)(C)C)cc1 ZINC000217950796 FJ In-Stock Unstable DRD3 27 51 COc1ccccc1CCCNC(=O)/C=C/c1ccc(C(C)(C)C)cc1 ZINC000217950796 FJ In-Stock Unstable TRPV1 18 60 COc1ccccc1CCCNC(=O)/C=C/c1ccc(C(C)(C)C)cc1 ZINC000217950796 FJ In-Stock Unstable LTB4R 0 40 COc1ccccc1CCCNC(=O)/C=C/c1ccc(C(C)(C)C)cc1 ZINC000217950796 FJ In-Stock Unstable MTNR1B 31 40 COc1ccccc1CCCNC(=O)/C=C/c1ccc(C(C)(C)C)cc1 ZINC000217950796 FJ In-Stock Unstable MMP2 15 45 C[C@H]1Cc2ccccc2[C@@H](c2ccccc2)[C@@H](C)N1 ZINC000217950806 CH For-Sale Unstable PRCP 47 38 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CC(c1ccccc1)c1ccccc1 ZINC000217950811 IJ For-Sale Unstable AGTR2 58 37 CN(Cc1ccccc1/C=C\C(=O)O)C[C@@H]1CCCO1 ZINC000217950840 CE For-Sale Unstable OXTR 28 44 CN(Cc1ccccc1/C=C\C(=O)O)C[C@@H]1CCCO1 ZINC000217950840 CE For-Sale Unstable AVPR1A 18 42 CN(Cc1ccccc1/C=C\C(=O)O)C[C@@H]1CCCO1 ZINC000217950840 CE For-Sale Unstable PTGER2 38 41 CN(Cc1ccccc1/C=C\C(=O)O)C[C@@H]1CCCO1 ZINC000217950840 CE For-Sale Unstable PTGER4 18 41 CN(Cc1ccccc1/C=C\C(=O)O)C[C@@H]1CCCO1 ZINC000217950840 CE For-Sale Unstable PTGER3 16 41 CN(Cc1ccccc1/C=C\C(=O)O)C[C@@H]1CCCO1 ZINC000217950840 CE For-Sale Unstable PTGDR 15 40 COc1cccc(/C=C/NC(=O)Nc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1 ZINC000217950848 HK For-Sale Unstable UL80 17 44 COc1cccc(/C=C/NC(=O)Nc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1 ZINC000217950848 HK For-Sale Unstable MTNR1A 22 42 COc1cccc(/C=C/NC(=O)Nc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1 ZINC000217950848 HK For-Sale Unstable MTNR1B 28 42 COc1cccc(/C=C/NC(=O)Nc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1 ZINC000217950848 HK For-Sale Unstable AKR1C2 17 44 O=C(c1ccc(N2CCCC2)cc1)N1CCC[C@H](c2nnc[nH]2)C1 ZINC000217950865 EE In-Stock Unstable PREP 15 40 O=C(c1ccc(N2CCCC2)cc1)N1CCC[C@H](c2nnc[nH]2)C1 ZINC000217950865 EE In-Stock Unstable L3MBTL1 0 46 O=C(c1ccc(N2CCCC2)cc1)N1CCC[C@H](c2nnc[nH]2)C1 ZINC000217950865 EE In-Stock Unstable L3MBTL3 61 46 O=C(c1ccc(N2CCCC2)cc1)N1CCC[C@H](c2nnc[nH]2)C1 ZINC000217950865 EE In-Stock Unstable L3MBTL4 0 46 O=C(c1ccc(N2CCCC2)cc1)N1CCC[C@H](c2nnc[nH]2)C1 ZINC000217950865 EE In-Stock Unstable MBTD1 0 46 O=C(c1ccc(N2CCCC2)cc1)N1CCC[C@H](c2nnc[nH]2)C1 ZINC000217950865 EE In-Stock Unstable TP53BP1 0 46 C[C@@H]1Cc2ccccc2[C@H](c2ccccc2)[C@@H](C)N1 ZINC000217950876 CH For-Sale Unstable PRCP 47 38 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CC(c1ccccc1)c1ccccc1 ZINC000217950894 IJ For-Sale Unstable AGTR2 58 37 COc1cccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)c1 ZINC000217950896 FJ In-Stock Unstable DRD3 17 43 COc1cccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)c1 ZINC000217950896 FJ In-Stock Unstable PTAFR 20 43 COc1cccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)c1 ZINC000217950896 FJ In-Stock Unstable TRPV1 17 51 COc1cccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)c1 ZINC000217950896 FJ In-Stock Unstable HDAC8 28 40 COc1cccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)c1 ZINC000217950896 FJ In-Stock Unstable MTNR1A 48 59 COc1cccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)c1 ZINC000217950896 FJ In-Stock Unstable MTNR1B 41 59 COc1cccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)c1 ZINC000217950896 FJ In-Stock Unstable HDAC1 19 41 COc1cccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)c1 ZINC000217950896 FJ In-Stock Unstable HDAC6 20 40 COc1cccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)c1 ZINC000217950896 FJ In-Stock Unstable AMP1_PLAFQ 19 40 COc1cccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)c1 ZINC000217950896 FJ In-Stock Unstable CRTM 59 47 CCS(=O)(=O)[C@@H]1CC[C@](N)(C(=O)O)C1 ZINC000217950897 BB In-Stock Unstable GRM1 0 50 CCCOc1ccc(/C=C2/CC(=O)NC2=O)cc1 ZINC000217950925 BD For-Sale Unstable HPGD 63 44 O=C(c1cc(-c2cccnc2)[nH]n1)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217950941 FD In-Stock Unstable CHRNA4 28 48 CO[C@@H]1C[C@@H](C(=O)O)N(C(=O)N[C@@H](C)c2ccccc2)C1 ZINC000217950945 CD On-Demand Unstable ACE 44 49 CO[C@@H]1C[C@@H](C(=O)O)N(C(=O)N[C@@H](C)c2ccccc2)C1 ZINC000217950945 CD On-Demand Unstable AGTR2 99 36 CN(Cc1ccc(/C=C\C(=O)O)cc1)C[C@@H]1CCCO1 ZINC000217950950 CE For-Sale Unstable OXTR 27 42 CN(Cc1ccc(/C=C\C(=O)O)cc1)C[C@@H]1CCCO1 ZINC000217950950 CE For-Sale Unstable AVPR1A 18 42 CCc1ccccc1NC(=O)N/C=C/c1cccc(OC)c1 ZINC000217950952 CI For-Sale Unstable MTNR1A 52 43 CCc1ccccc1NC(=O)N/C=C/c1cccc(OC)c1 ZINC000217950952 CI For-Sale Unstable MTNR1B 49 43 C[C@H]1Cc2ccccc2[C@H](c2ccccc2)[C@@H](C)N1 ZINC000217950970 CH For-Sale Unstable PRCP 47 38 CCS(=O)(=O)[C@H]1CC[C@](N)(C(=O)O)C1 ZINC000217950977 BB In-Stock Unstable GRM1 0 50 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CC(c1ccccc1)c1ccccc1 ZINC000217950982 IJ For-Sale Unstable AGTR2 58 37 COc1ccc(CCNC(=O)NCC[C@@H](O)c2cccn2C)cc1 ZINC000217950990 ED In-Stock Unstable MTNR1A 41 39 COc1ccc(CCNC(=O)NCC[C@@H](O)c2cccn2C)cc1 ZINC000217950990 ED In-Stock Unstable MTNR1B 40 36 O=C1C/C(=C\c2ccc(-n3cccn3)cc2)C(=O)N1 ZINC000217951000 CD For-Sale Unstable AMP1_PLAFQ 49 36 COc1ccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1 ZINC000217951004 FJ In-Stock Unstable DRD3 15 48 COc1ccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1 ZINC000217951004 FJ In-Stock Unstable PTAFR 15 42 COc1ccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1 ZINC000217951004 FJ In-Stock Unstable TRPV1 29 61 COc1ccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1 ZINC000217951004 FJ In-Stock Unstable HDAC8 33 49 COc1ccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1 ZINC000217951004 FJ In-Stock Unstable MTNR1A 23 40 COc1ccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1 ZINC000217951004 FJ In-Stock Unstable HDAC6 21 49 COc1ccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1 ZINC000217951004 FJ In-Stock Unstable HDAC7 40 36 COc1ccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1 ZINC000217951004 FJ In-Stock Unstable CYP24A1 26 43 COc1ccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1 ZINC000217951004 FJ In-Stock Unstable HDA106 0 41 COc1ccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1 ZINC000217951004 FJ In-Stock Unstable PROKR1 43 31 COc1ccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1 ZINC000217951004 FJ In-Stock Unstable CYP27B1 26 43 CO[C@H]1C[C@@H](C(=O)O)N(C(=O)N[C@@H](C)c2ccccc2)C1 ZINC000217951038 CD On-Demand Unstable ACE 44 49 CO[C@H]1C[C@@H](C(=O)O)N(C(=O)N[C@@H](C)c2ccccc2)C1 ZINC000217951038 CD On-Demand Unstable AGTR2 99 36 COc1ccc(/C=C2\Oc3c(ccc4c3[C@H](c3cccc(OCCc5ccc(OC)cc5)c3)CC(=O)O4)C2=O)cc1 ZINC000217951039 KK In-Stock Unstable ACHE 15 44 CCS(=O)(=O)[C@@H]1CC[C@@](N)(C(=O)O)C1 ZINC000217951040 BB In-Stock Unstable GRM1 0 50 COc1cccc(/C=C/NC(=O)NC(=O)c2ccc(N)cc2)c1 ZINC000217951048 DE For-Sale Unstable MTNR1A 22 40 COc1cccc(/C=C/NC(=O)NC(=O)c2ccc(N)cc2)c1 ZINC000217951048 DE For-Sale Unstable MTNR1B 27 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CC(c1ccccc1)c1ccccc1 ZINC000217951059 IJ For-Sale Unstable AGTR2 58 37 COc1ccc(CCNC(=O)NCC[C@H](O)c2cccn2C)cc1 ZINC000217951078 ED In-Stock Unstable MTNR1A 41 39 COc1ccc(CCNC(=O)NCC[C@H](O)c2cccn2C)cc1 ZINC000217951078 ED In-Stock Unstable MTNR1B 40 36 CO[C@@H]1CCN(c2ncc(CBr)cc2C)C1 ZINC000217951100 CF For-Sale Unstable CACNA2D1 15 40 CO[C@@H]1CCN(c2ncc(CBr)cc2C)C1 ZINC000217951100 CF For-Sale Unstable PDE3B 43 36 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1 ZINC000217951105 FJ In-Stock Unstable SDH1 0 40 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1 ZINC000217951105 FJ In-Stock Unstable HDAC8 16 49 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1 ZINC000217951105 FJ In-Stock Unstable HDAC2 15 45 CCS(=O)(=O)[C@H]1CC[C@@](N)(C(=O)O)C1 ZINC000217951110 BB In-Stock Unstable GRM1 0 50 COc1ccc(/C=C2\Oc3c(ccc4c3[C@@H](c3cccc(OCCc5ccc(OC)cc5)c3)CC(=O)O4)C2=O)cc1 ZINC000217951118 KK In-Stock Unstable ACHE 15 44 COc1cccc(/C=C/NC(=O)Nc2ccc(C(N)=O)cc2)c1 ZINC000217951155 DF For-Sale Unstable CYP1B1 18 40 COc1cccc(/C=C/NC(=O)Nc2ccc(C(N)=O)cc2)c1 ZINC000217951155 DF For-Sale Unstable RAF1 17 45 COc1cccc(/C=C/NC(=O)Nc2ccc(C(N)=O)cc2)c1 ZINC000217951155 DF For-Sale Unstable MTNR1A 26 51 COc1cccc(/C=C/NC(=O)Nc2ccc(C(N)=O)cc2)c1 ZINC000217951155 DF For-Sale Unstable MTNR1B 32 51 COc1cccc(/C=C/NC(=O)Nc2ccc(C(N)=O)cc2)c1 ZINC000217951155 DF For-Sale Unstable F7 16 44 COc1cccc(/C=C/NC(=O)Nc2ccc(C(N)=O)cc2)c1 ZINC000217951155 DF For-Sale Unstable ACR 57 47 COc1cccc(/C=C/NC(=O)Nc2ccc(C(N)=O)cc2)c1 ZINC000217951155 DF For-Sale Unstable PDGFRA 33 40 COc1cccc(/C=C/NC(=O)Nc2ccc(C(N)=O)cc2)c1 ZINC000217951155 DF For-Sale Unstable Q8MMZ8_EIMTE 15 45 COc1cccc(/C=C/NC(=O)Nc2ccc(C(N)=O)cc2)c1 ZINC000217951155 DF For-Sale Unstable TAAR1 31 41 COc1cccc(/C=C/NC(=O)Nc2ccc(C(N)=O)cc2)c1 ZINC000217951155 DF For-Sale Unstable KCNK3 18 41 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc(C)cc1C ZINC000217951165 FG For-Sale Unstable HCRTR1 49 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc(C)cc1C ZINC000217951165 FG For-Sale Unstable HCRTR2 51 40 CO[C@H]1CCN(c2ncc(CBr)cc2C)C1 ZINC000217951180 CF For-Sale Unstable CACNA2D1 15 40 CO[C@H]1CCN(c2ncc(CBr)cc2C)C1 ZINC000217951180 CF For-Sale Unstable PDE3B 43 36 Cn1cccc1[C@H](O)CCNC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217951183 EG In-Stock Unstable CCR3 28 46 Cn1cccc1[C@H](O)CCNC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217951183 EG In-Stock Unstable RAF1 19 44 Cn1cccc1[C@H](O)CCNC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217951183 EG In-Stock Unstable KDR 15 42 Cn1cccc1[C@H](O)CCNC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217951183 EG In-Stock Unstable EPHX2 21 44 Cn1cccc1[C@H](O)CCNC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217951183 EG In-Stock Unstable Q8MMZ8_EIMTE 0 44 O=C(O)/C=C\c1ccccc1CN1CCCC[C@@H]1CO ZINC000217951186 CE For-Sale Unstable PTGER2 34 43 O=C(O)/C=C\c1ccccc1CN1CCCC[C@@H]1CO ZINC000217951186 CE For-Sale Unstable PTGER4 17 43 O=C(O)/C=C\c1ccccc1CN1CCCC[C@@H]1CO ZINC000217951186 CE For-Sale Unstable PTGER3 17 43 O=C(O)/C=C\c1ccccc1CN1CCCC[C@@H]1CO ZINC000217951186 CE For-Sale Unstable PTGDR 15 40 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1 ZINC000217951188 FJ In-Stock Unstable SDH1 0 40 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1 ZINC000217951188 FJ In-Stock Unstable HDAC8 16 49 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1 ZINC000217951188 FJ In-Stock Unstable HDAC2 15 45 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc(C)cc1C ZINC000217951242 FG For-Sale Unstable HCRTR1 49 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc(C)cc1C ZINC000217951242 FG For-Sale Unstable HCRTR2 51 40 Cn1cc(C(=O)N[C@@H]2CCC[C@@H]2CO)c2ccccc21 ZINC000217951254 CE On-Demand Unstable CNR1 22 44 COc1cccc(/C=C/NC(=O)Nc2ccc(F)c(Cl)c2)c1 ZINC000217951257 DI For-Sale Unstable UL80 19 40 COc1cccc(/C=C/NC(=O)Nc2ccc(F)c(Cl)c2)c1 ZINC000217951257 DI For-Sale Unstable AHR 15 45 COc1cccc(/C=C/NC(=O)Nc2ccc(F)c(Cl)c2)c1 ZINC000217951257 DI For-Sale Unstable MTNR1A 18 43 COc1cccc(/C=C/NC(=O)Nc2ccc(F)c(Cl)c2)c1 ZINC000217951257 DI For-Sale Unstable MTNR1B 24 43 COc1cccc(/C=C/NC(=O)Nc2ccc(F)c(Cl)c2)c1 ZINC000217951257 DI For-Sale Unstable Q8MMZ8_EIMTE 0 41 COc1cccc(/C=C/NC(=O)Nc2ccc(F)c(Cl)c2)c1 ZINC000217951257 DI For-Sale Unstable TAAR1 25 55 Cn1cccc1[C@@H](O)CCNC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217951261 EG In-Stock Unstable CCR3 28 46 Cn1cccc1[C@@H](O)CCNC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217951261 EG In-Stock Unstable RAF1 19 44 Cn1cccc1[C@@H](O)CCNC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217951261 EG In-Stock Unstable KDR 15 42 Cn1cccc1[C@@H](O)CCNC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217951261 EG In-Stock Unstable EPHX2 21 44 Cn1cccc1[C@@H](O)CCNC(=O)Nc1cccc(C(F)(F)F)c1 ZINC000217951261 EG In-Stock Unstable Q8MMZ8_EIMTE 0 44 C[C@@H]1CCC[C@H]([C@@H](N)Cc2cc(F)ccc2Br)C1 ZINC000217951272 DI For-Sale Unstable DPP4 20 43 COc1c(C(C)C)cccc1S(=O)(=O)Cl ZINC000217951287 BF For-Sale Unstable SOAT1 18 41 Cc1ccc(NC(=O)c2cc(C(C)C)nc3onc(C)c23)cc1S(=O)(=O)Nc1ccccc1Cl ZINC000217951334 JK On-Demand Unstable GRM4 33 47 Cc1ccc(NC(=O)c2cc(C(C)C)nc3onc(C)c23)cc1S(=O)(=O)Nc1ccccc1Cl ZINC000217951334 JK On-Demand Unstable NR2E3 61 35 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc(C)cc1C ZINC000217951335 FG For-Sale Unstable HCRTR1 49 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc(C)cc1C ZINC000217951335 FG For-Sale Unstable HCRTR2 51 40 Cn1cc(C(=O)N[C@H]2CCC[C@@H]2CO)c2ccccc21 ZINC000217951340 CE For-Sale Unstable CNR1 24 44 Cn1cc(C(=O)N[C@H]2CCC[C@@H]2CO)c2ccccc21 ZINC000217951340 CE For-Sale Unstable HTR4 20 40 C[C@H]1CCC[C@H]([C@@H](N)Cc2cc(F)ccc2Br)C1 ZINC000217951361 DI For-Sale Unstable DPP4 20 43 CCN(CC)c1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217951366 EI For-Sale Unstable MTNR1A 35 55 CCN(CC)c1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217951366 EI For-Sale Unstable MTNR1B 38 55 CCN(CC)c1ccc(NC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217951366 EI For-Sale Unstable ROCK2 15 40 CC(C)CCN(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217951382 CG For-Sale Unstable FDPS 16 40 CC(C)CCN(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217951382 CG For-Sale Unstable AKR1C3 28 41 Cn1cccc1[C@H](O)CCNC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217951384 EH In-Stock Unstable P95276_MYCTO 0 42 CC(C)(C)c1ccc(/C=C/C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217951415 GK In-Stock Unstable TRPV1 15 64 CC(C)(C)c1ccc(/C=C/C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217951415 GK In-Stock Unstable LTB4R 0 57 CC(C)(C)c1ccc(/C=C/C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217951415 GK In-Stock Unstable MMP2 24 52 CC(C)(C)c1ccc(/C=C/C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217951415 GK In-Stock Unstable NR1H4 15 47 CC(C)(C)c1ccc(/C=C/C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217951415 GK In-Stock Unstable HDAC1 23 52 CC(C)(C)c1ccc(/C=C/C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217951415 GK In-Stock Unstable HDAC2 16 41 CC(C)(C)c1ccc(/C=C/C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217951415 GK In-Stock Unstable MMP9 20 52 CC(C)(C)c1ccc(/C=C/C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217951415 GK In-Stock Unstable IMPDH2 0 44 CC(C)(C)c1ccc(/C=C/C(=O)Nc2ccccc2C(=O)c2ccccc2)cc1 ZINC000217951415 GK In-Stock Unstable MMP1 26 52 Cn1cc(C(=O)N[C@@H]2CCC[C@H]2CO)c2ccccc21 ZINC000217951422 CE For-Sale Unstable CNR1 24 44 Cn1cc(C(=O)N[C@@H]2CCC[C@H]2CO)c2ccccc21 ZINC000217951422 CE For-Sale Unstable HTR4 20 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc(C)cc1C ZINC000217951424 FG For-Sale Unstable HCRTR1 49 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc(C)cc1C ZINC000217951424 FG For-Sale Unstable HCRTR2 51 40 COc1cccc(/C(C)=C2/CC(=O)NC2=O)c1 ZINC000217951434 BD For-Sale Unstable DRD4 44 34 C[C@@H]1CCC[C@@H]([C@@H](N)Cc2cc(F)ccc2Br)C1 ZINC000217951440 DI For-Sale Unstable DPP4 20 43 COC(=O)C[C@@H](c1oc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c1O)C1CCCCC1 ZINC000217951443 JG In-Stock Unstable CHRNA4 27 44 Cn1cccc1[C@@H](O)CCNC(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217951464 EH In-Stock Unstable P95276_MYCTO 0 42 COc1cccc(/C=C/NC(=O)NCc2ccc(F)cc2)c1 ZINC000217951469 DG For-Sale Unstable CCR3 18 41 COc1cccc(/C=C/NC(=O)NCc2ccc(F)cc2)c1 ZINC000217951469 DG For-Sale Unstable MTNR1A 54 43 COc1cccc(/C=C/NC(=O)NCc2ccc(F)cc2)c1 ZINC000217951469 DG For-Sale Unstable MTNR1B 54 43 COc1cccc(/C=C/NC(=O)NCc2ccc(F)cc2)c1 ZINC000217951469 DG For-Sale Unstable ROCK2 30 42 COc1cccc(/C=C/NC(=O)NCc2ccc(F)cc2)c1 ZINC000217951469 DG For-Sale Unstable AMP1_PLAFQ 17 40 COc1cccc(/C=C/NC(=O)NCc2ccc(F)cc2)c1 ZINC000217951469 DG For-Sale Unstable PDS 42 39 CC(C)CCN(C)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217951481 CG On-Demand Unstable FDPS 24 41 CC(C)CCN(C)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217951481 CG On-Demand Unstable LTA4H 18 40 CO[C@@H]1CCN(c2ccc(CBr)c(C(F)(F)F)c2)C1 ZINC000217951487 EH For-Sale Unstable LIPG 46 34 Cn1cc(C(=O)N[C@H]2CCC[C@H]2CO)c2ccccc21 ZINC000217951504 CE For-Sale Unstable CNR1 24 44 Cn1cc(C(=O)N[C@H]2CCC[C@H]2CO)c2ccccc21 ZINC000217951504 CE For-Sale Unstable HTR4 20 40 COC(=O)C[C@H](c1oc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c1O)C1CCCCC1 ZINC000217951513 JG In-Stock Unstable CHRNA4 27 44 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)c1 ZINC000217951517 GK In-Stock Unstable PYGL 0 40 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)c1 ZINC000217951517 GK In-Stock Unstable AMP1_PLAFQ 23 41 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)c1 ZINC000217951517 GK In-Stock Unstable CRTM 53 48 C[C@H]1CCC[C@@H]([C@@H](N)Cc2cc(F)ccc2Br)C1 ZINC000217951521 DI For-Sale Unstable DPP4 20 43 O=C(Nc1ccn2nccc2c1)c1csc(-c2ccccc2)n1 ZINC000217951566 DH In-Stock Anodyne CHEK1 0 47 CO[C@H]1CCN(c2ccc(CBr)c(C(F)(F)F)c2)C1 ZINC000217951576 EH For-Sale Unstable LIPG 46 34 COc1cccc(/C=C/NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000217951584 FG For-Sale Unstable HTR1A 98 51 COc1cccc(/C=C/NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000217951584 FG For-Sale Unstable DRD2 71 51 COc1cccc(/C=C/NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000217951584 FG For-Sale Unstable DRD1 28 41 COc1cccc(/C=C/NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000217951584 FG For-Sale Unstable DRD4 46 39 COc1cccc(/C=C/NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000217951584 FG For-Sale Unstable ADRA1D 74 45 COc1cccc(/C=C/NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000217951584 FG For-Sale Unstable HTR1D 22 43 COc1cccc(/C=C/NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000217951584 FG For-Sale Unstable HTR1B 20 51 COc1cccc(/C=C/NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000217951584 FG For-Sale Unstable HTR2A 37 41 COc1cccc(/C=C/NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000217951584 FG For-Sale Unstable ADRA1A 66 45 COc1cccc(/C=C/NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000217951584 FG For-Sale Unstable ADRA1B 60 45 COc1cccc(/C=C/NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000217951584 FG For-Sale Unstable DRD3 77 51 COc1cccc(/C=C/NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000217951584 FG For-Sale Unstable PDGFRB 34 42 COc1cccc(/C=C/NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000217951584 FG For-Sale Unstable HTR7 61 48 COc1cccc(/C=C/NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000217951584 FG For-Sale Unstable TACR3 22 44 COc1cccc(/C=C/NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000217951584 FG For-Sale Unstable MTNR1B 28 40 COc1cccc(/C=C/NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000217951584 FG For-Sale Unstable ABCB1 0 41 COc1cccc(/C=C/NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000217951584 FG For-Sale Unstable RBP4 15 44 COc1cccc(/C=C/NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000217951584 FG For-Sale Unstable ALPHA-1A 0 41 COc1ccc(/C=C\C(=O)O)cc1CN1CCC[C@H]1C ZINC000217951589 CF For-Sale Unstable HRH3 25 45 COc1ccc(/C=C\C(=O)O)cc1CN1CCC[C@H]1C ZINC000217951589 CF For-Sale Unstable ACKR3 65 36 CC(C)Oc1ccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1 ZINC000217951632 GK In-Stock Unstable HDAC8 0 43 CCc1ncnc(NCCc2ccccc2)c1F ZINC000217951648 BF On-Demand Unstable HTT 0 40 COc1ccc(/C=C\C(=O)O)cc1CN1CCC[C@@H]1C ZINC000217951678 CF For-Sale Unstable HRH3 25 45 COc1ccc(/C=C\C(=O)O)cc1CN1CCC[C@@H]1C ZINC000217951678 CF For-Sale Unstable ACKR3 65 36 CCCC[C@@H](CC)CN[C@@H](C)C(=O)Nc1ccccc1 ZINC000217951680 CH For-Sale Unstable MMP2 16 46 CCCC[C@@H](CC)CN[C@@H](C)C(=O)Nc1ccccc1 ZINC000217951680 CH For-Sale Unstable MMP3 34 46 CCCC[C@@H](CC)CN[C@@H](C)C(=O)Nc1ccccc1 ZINC000217951680 CH For-Sale Unstable HDAC2 17 40 COc1cccc(/C=C/NC(=O)NC2=NCCS2)c1 ZINC000217951684 CE For-Sale Unstable MTNR1A 17 40 COc1cccc(/C=C/NC(=O)NC2=NCCS2)c1 ZINC000217951684 CE For-Sale Unstable MTNR1B 23 40 CO[C@@H]1CCN(c2nc3ccccc3cc2CBr)C1 ZINC000217951692 DG For-Sale Unstable PDE3A 49 40 CO[C@@H]1CCN(c2nc3ccccc3cc2CBr)C1 ZINC000217951692 DG For-Sale Unstable PDE1B 0 41 CO[C@@H]1CCN(c2nc3ccccc3cc2CBr)C1 ZINC000217951692 DG For-Sale Unstable PDE3B 73 40 O=C(O)[C@@H]1C[C@@H]2CCCC[C@@H]2N1C(=O)N1CCCC1 ZINC000217951705 CD For-Sale Unstable ACE 16 62 O=C(O)[C@@H]1C[C@@H]2CCCC[C@@H]2N1C(=O)N1CCCC1 ZINC000217951705 CD For-Sale Unstable PREP 32 51 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1ccc([N+](=O)[O-])cc1 ZINC000217951708 CI For-Sale Unstable TRPM8 16 44 O=Cc1ccc(-c2cc(C(=O)O)ncn2)cc1Cl ZINC000217951718 CE For-Sale Anodyne RPA1 42 33 CN(CCNC(=O)/C=C/c1ccc(C(C)(C)C)cc1)c1ccccc1 ZINC000217951750 EI In-Stock Unstable HDAC8 22 42 CN(CCNC(=O)/C=C/c1ccc(C(C)(C)C)cc1)c1ccccc1 ZINC000217951750 EI In-Stock Unstable HDAC1 22 43 CN(CCNC(=O)/C=C/c1ccc(C(C)(C)C)cc1)c1ccccc1 ZINC000217951750 EI In-Stock Unstable HDAC6 23 41 CN(CCNC(=O)/C=C/c1ccc(C(C)(C)C)cc1)c1ccccc1 ZINC000217951750 EI In-Stock Unstable HDAC7 48 38 C[C@H]1CN(Cc2cccc(/C=C\C(=O)O)c2)C[C@@H](C)O1 ZINC000217951758 CE For-Sale Unstable SIGMAR1 17 43 CO[C@H]1CCN(c2nc3ccccc3cc2CBr)C1 ZINC000217951768 DG For-Sale Unstable PDE3A 49 40 CO[C@H]1CCN(c2nc3ccccc3cc2CBr)C1 ZINC000217951768 DG For-Sale Unstable PDE1B 0 41 CO[C@H]1CCN(c2nc3ccccc3cc2CBr)C1 ZINC000217951768 DG For-Sale Unstable PDE3B 73 40 C[C@@H]1CCC[C@H]([C@@H](N)Cc2ccc(Br)cc2F)C1 ZINC000217951770 DI For-Sale Unstable DPP4 20 43 Cn1cccc(C(=O)Nc2ccn3nccc3c2)c1=O ZINC000217951771 CD In-Stock Unstable KCNK3 43 33 Cn1cccc(C(=O)Nc2ccn3nccc3c2)c1=O ZINC000217951771 CD In-Stock Unstable KCNK9 45 34 CCCC[C@H](CC)CN[C@@H](C)C(=O)Nc1ccccc1 ZINC000217951777 CH For-Sale Unstable MMP2 16 46 CCCC[C@H](CC)CN[C@@H](C)C(=O)Nc1ccccc1 ZINC000217951777 CH For-Sale Unstable MMP3 34 46 CCCC[C@H](CC)CN[C@@H](C)C(=O)Nc1ccccc1 ZINC000217951777 CH For-Sale Unstable HDAC2 17 40 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1ccc([N+](=O)[O-])cc1 ZINC000217951781 CI For-Sale Unstable TRPM8 16 44 O=C(O)[C@@H]1C[C@H]2CCCC[C@@H]2N1C(=O)N1CCCC1 ZINC000217951784 CD For-Sale Unstable ACE 16 62 O=C(O)[C@@H]1C[C@H]2CCCC[C@@H]2N1C(=O)N1CCCC1 ZINC000217951784 CD For-Sale Unstable PREP 32 51 COc1cccc(/C=C/NC(=O)N(CC(C)C)CC(C)C)c1 ZINC000217951791 DH For-Sale Unstable MTNR1A 45 44 COc1cccc(/C=C/NC(=O)N(CC(C)C)CC(C)C)c1 ZINC000217951791 DH For-Sale Unstable MTNR1B 46 44 COc1cccc(/C=C/NC(=O)N(CC(C)C)CC(C)C)c1 ZINC000217951791 DH For-Sale Unstable NR1H4 26 40 COc1cc2c(=O)[nH]ccc2cc1F ZINC000217951806 AD In-Stock Unstable CDC42 44 33 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1ccc([N+](=O)[O-])cc1 ZINC000217951850 CI For-Sale Unstable TRPM8 16 44 C[C@H]1CCC[C@H]([C@@H](N)Cc2ccc(Br)cc2F)C1 ZINC000217951852 DI For-Sale Unstable DPP4 20 43 CCCC[C@@H](CC)CN[C@H](C)C(=O)Nc1ccccc1 ZINC000217951857 CH For-Sale Unstable MMP2 16 46 CCCC[C@@H](CC)CN[C@H](C)C(=O)Nc1ccccc1 ZINC000217951857 CH For-Sale Unstable MMP3 34 46 CCCC[C@@H](CC)CN[C@H](C)C(=O)Nc1ccccc1 ZINC000217951857 CH For-Sale Unstable HDAC2 17 40 CO[C@@H]1CCN(c2nc3ccccn3c2CBr)C1 ZINC000217951867 DE For-Sale Unstable PDE3B 50 35 CC(C)(C)c1ccc(/C=C/C(=O)Nc2ccc(OC3CCCC3)cc2)cc1 ZINC000217951868 FK In-Stock Unstable TRPV1 20 68 CC(C)(C)c1ccc(/C=C/C(=O)Nc2ccc(OC3CCCC3)cc2)cc1 ZINC000217951868 FK In-Stock Unstable HDAC8 0 42 CC(C)(C)c1ccc(/C=C/C(=O)Nc2ccc(OC3CCCC3)cc2)cc1 ZINC000217951868 FK In-Stock Unstable MMP2 19 51 CC(C)(C)c1ccc(/C=C/C(=O)Nc2ccc(OC3CCCC3)cc2)cc1 ZINC000217951868 FK In-Stock Unstable HDAC1 25 47 CC(C)(C)c1ccc(/C=C/C(=O)Nc2ccc(OC3CCCC3)cc2)cc1 ZINC000217951868 FK In-Stock Unstable MMP9 15 51 CC(C)(C)c1ccc(/C=C/C(=O)Nc2ccc(OC3CCCC3)cc2)cc1 ZINC000217951868 FK In-Stock Unstable IMPDH2 0 49 CC(C)(C)c1ccc(/C=C/C(=O)Nc2ccc(OC3CCCC3)cc2)cc1 ZINC000217951868 FK In-Stock Unstable MMP1 24 47 CC(C)(C)c1ccc(/C=C/C(=O)Nc2ccc(OC3CCCC3)cc2)cc1 ZINC000217951868 FK In-Stock Unstable MCHR1 16 44 Cc1noc2nc(C(C)C)cc(C(=O)Nc3ccc(Cl)c(S(=O)(=O)N4CCCC4)c3)c12 ZINC000217951870 JI On-Demand Unstable NR1H4 18 41 Cc1noc2nc(C(C)C)cc(C(=O)Nc3ccc(Cl)c(S(=O)(=O)N4CCCC4)c3)c12 ZINC000217951870 JI On-Demand Unstable NR2E3 51 32 O=C(/C=C/c1ccccc1Cl)Nc1ccn2nccc2c1 ZINC000217951878 CH In-Stock Anodyne KCNQ2 20 40 O=C(/C=C/c1ccccc1Cl)Nc1ccn2nccc2c1 ZINC000217951878 CH In-Stock Anodyne MMP1 0 41 COc1cccc(/C=C/NC(=O)N2CCN(C=O)CC2)c1 ZINC000217951895 CD For-Sale Unstable DRD4 41 32 COc1cccc(/C=C/NC(=O)N2CCN(C=O)CC2)c1 ZINC000217951895 CD For-Sale Unstable MTNR1A 27 40 COc1cccc(/C=C/NC(=O)N2CCN(C=O)CC2)c1 ZINC000217951895 CD For-Sale Unstable MTNR1B 38 40 COc1cc2c(cc1F)CCNC2=O ZINC000217951915 AD For-Sale Unstable CSNK1D 30 43 COc1cc2c(cc1F)CCNC2=O ZINC000217951915 AD For-Sale Unstable CSNK1G2 73 43 COC(=O)C[C@H](c1cccc(Oc2ncccn2)c1)c1oc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c1O ZINC000217951921 KG In-Stock Unstable CHRNA4 25 41 CCCC[C@H](CC)CN[C@H](C)C(=O)Nc1ccccc1 ZINC000217951933 CH For-Sale Unstable MMP2 16 46 CCCC[C@H](CC)CN[C@H](C)C(=O)Nc1ccccc1 ZINC000217951933 CH For-Sale Unstable MMP3 34 46 CCCC[C@H](CC)CN[C@H](C)C(=O)Nc1ccccc1 ZINC000217951933 CH For-Sale Unstable HDAC2 17 40 N#C[C@@H]1CNCCN1CC(=O)N1CCC[C@@H]2CCCC[C@@H]21 ZINC000217951935 CC For-Sale Unstable DPP4 58 44 N#C[C@@H]1CNCCN1CC(=O)N1CCC[C@@H]2CCCC[C@@H]21 ZINC000217951935 CC For-Sale Unstable DPP9 18 40 N#C[C@@H]1CNCCN1CC(=O)N1CCC[C@@H]2CCCC[C@@H]21 ZINC000217951935 CC For-Sale Unstable FAP 0 40 C[C@@H]1CCC[C@@H]([C@@H](N)Cc2ccc(Br)cc2F)C1 ZINC000217951936 DI For-Sale Unstable DPP4 20 43 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1ccc([N+](=O)[O-])cc1 ZINC000217951937 CI For-Sale Unstable TRPM8 16 44 CO[C@H]1CCN(c2nc3ccccn3c2CBr)C1 ZINC000217951952 DE For-Sale Unstable PDE3B 50 35 COc1cccc(/C=C/NC(=O)NC2CCCCCC2)c1 ZINC000217951983 CH For-Sale Unstable MTNR1A 37 40 COc1cccc(/C=C/NC(=O)NC2CCCCCC2)c1 ZINC000217951983 CH For-Sale Unstable MTNR1B 40 40 COc1cccc(/C=C/NC(=O)NC2CCCCCC2)c1 ZINC000217951983 CH For-Sale Unstable NR1H4 22 40 COc1cccc(/C=C/NC(=O)NC2CCCCCC2)c1 ZINC000217951983 CH For-Sale Unstable FAAH 26 46 COc1cccc(/C=C/NC(=O)NC2CCCCCC2)c1 ZINC000217951983 CH For-Sale Unstable EPHX2 28 50 COC(=O)C[C@@H](c1cccc(Oc2ncccn2)c1)c1oc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c1O ZINC000217952016 KG In-Stock Unstable CHRNA4 25 41 C[C@H]1CCC[C@@H]([C@@H](N)Cc2ccc(Br)cc2F)C1 ZINC000217952021 DI For-Sale Unstable DPP4 20 43 CCS(=O)(=O)Nc1ccc(/C=C\C(=O)CCl)cc1 ZINC000217952025 CE For-Sale Unstable HDAC8 15 47 COc1cccc(/C=C/NC(=O)Nc2cc(C)ccc2C)c1 ZINC000217952083 CI For-Sale Unstable MTNR1A 28 40 COc1cccc(/C=C/NC(=O)Nc2cc(C)ccc2C)c1 ZINC000217952083 CI For-Sale Unstable MTNR1B 29 40 COc1ccc(Br)c(C(=O)Nc2ccn3nccc3c2)c1 ZINC000217952087 EG In-Stock Unstable TAAR1 23 41 COc1ccc(Br)c(C(=O)Nc2ccn3nccc3c2)c1 ZINC000217952087 EG In-Stock Unstable AKR1C2 41 34 CCCS(=O)(=O)Nc1ccc(/C=C\C(=O)CCl)cc1 ZINC000217952098 DF For-Sale Unstable HDAC8 0 45 C[C@H]1CN(Cc2ccc(F)c(/C=C\C(=O)O)c2)C[C@@H](C)O1 ZINC000217952099 CF For-Sale Unstable CCR1 0 41 COc1ccc2c(c1)CCc1c(C(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)n[nH]c1-2 ZINC000217952117 HF In-Stock Unstable CHRNA4 25 40 COC(=O)c1ccc(C(=O)Nc2ccn3nccc3c2)cc1 ZINC000217952174 CE In-Stock Unstable TRPV1 15 40 COC(=O)c1ccc(C(=O)Nc2ccn3nccc3c2)cc1 ZINC000217952174 CE In-Stock Unstable PRNP 55 35 COC(=O)c1ccc(C(=O)Nc2ccn3nccc3c2)cc1 ZINC000217952174 CE In-Stock Unstable DDR1 43 36 COC(=O)c1ccc(C(=O)Nc2ccn3nccc3c2)cc1 ZINC000217952174 CE In-Stock Unstable KCNK3 84 40 COC(=O)c1ccc(C(=O)Nc2ccn3nccc3c2)cc1 ZINC000217952174 CE In-Stock Unstable KCNK9 62 35 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1 ZINC000217952175 FK In-Stock Unstable TRPV1 15 47 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1 ZINC000217952175 FK In-Stock Unstable SCN2A 15 41 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1 ZINC000217952175 FK In-Stock Unstable PYGL 0 40 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1 ZINC000217952175 FK In-Stock Unstable HDAC8 15 46 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1 ZINC000217952175 FK In-Stock Unstable TRPM2 0 40 COc1cccc(/C=C/NC(=O)Nc2cc(Cl)cc(Cl)c2)c1 ZINC000217952187 EJ For-Sale Unstable AHR 22 57 COc1cccc(/C=C/NC(=O)Nc2cc(Cl)cc(Cl)c2)c1 ZINC000217952187 EJ For-Sale Unstable MTNR1A 28 44 COc1cccc(/C=C/NC(=O)Nc2cc(Cl)cc(Cl)c2)c1 ZINC000217952187 EJ For-Sale Unstable MTNR1B 33 44 COc1cccc(/C=C/NC(=O)Nc2cc(Cl)cc(Cl)c2)c1 ZINC000217952187 EJ For-Sale Unstable TAAR1 23 40 COc1cccc(/C=C/NC(=O)Nc2cc(Cl)cc(Cl)c2)c1 ZINC000217952187 EJ For-Sale Unstable AKR1C2 28 41 CCc1cc(C)nc(OCc2ccccc2)c1C#N ZINC000217952228 CG For-Sale Unstable MAOB 15 40 CCc1cc(C)nc(OCc2ccccc2)c1C#N ZINC000217952228 CG For-Sale Unstable MAPK9 24 46 CCc1cc(C)nc(OCc2ccccc2)c1C#N ZINC000217952228 CG For-Sale Unstable MAPK8 16 46 CCc1cc(C)nc(OCc2ccccc2)c1C#N ZINC000217952228 CG For-Sale Unstable RPS27 48 42 CN(Cc1ccccc1)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217952256 CG For-Sale Unstable ACHE 22 46 CN(Cc1ccccc1)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217952256 CG For-Sale Unstable PTGER2 38 46 CN(Cc1ccccc1)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217952256 CG For-Sale Unstable PTGER4 0 42 CN(Cc1ccccc1)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217952256 CG For-Sale Unstable NR1H4 48 39 CN(Cc1ccccc1)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217952256 CG For-Sale Unstable HDAC6 22 40 CN(Cc1ccccc1)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217952256 CG For-Sale Unstable HSD17B2 25 41 CN(Cc1ccccc1)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217952256 CG For-Sale Unstable 17HSDCL 0 42 CN(Cc1ccccc1)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217952256 CG For-Sale Unstable AKR1C3 36 46 COc1ccc(/C=C\C(=O)CCl)c(F)c1 ZINC000217952279 BF For-Sale Unstable CYP1B1 42 39 COc1ccc(/C=C\C(=O)CCl)c(F)c1 ZINC000217952279 BF For-Sale Unstable CYSP_PLAFA 56 44 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccc(C(C)(C)C)cc1 ZINC000217952283 GK In-Stock Unstable DRD3 15 42 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccc(C(C)(C)C)cc1 ZINC000217952283 GK In-Stock Unstable MTNR1A 25 43 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccc(C(C)(C)C)cc1 ZINC000217952283 GK In-Stock Unstable MTNR1B 25 43 CCOc1ccccc1NC(=O)N/C=C/c1cccc(OC)c1 ZINC000217952287 DH For-Sale Unstable TSPO 40 33 CCOc1ccccc1NC(=O)N/C=C/c1cccc(OC)c1 ZINC000217952287 DH For-Sale Unstable MTNR1A 36 40 CCOc1ccccc1NC(=O)N/C=C/c1cccc(OC)c1 ZINC000217952287 DH For-Sale Unstable MTNR1B 38 47 CCOc1ccccc1NC(=O)N/C=C/c1cccc(OC)c1 ZINC000217952287 DH For-Sale Unstable KCNK3 31 41 CCOc1ccccc1NC(=O)N/C=C/c1cccc(OC)c1 ZINC000217952287 DH For-Sale Unstable KCNK9 24 41 C[C@H]1CN(C)[C@@H](C)C[C@@H]1Nc1ccc([N+](=O)[O-])cc1 ZINC000217952308 CF For-Sale Unstable KCNJ1 18 42 CCc1cc(C)nc(OCc2ccccc2)c1CO ZINC000217952332 CG For-Sale Unstable AGTR1 15 40 COc1ccc(/C=C\C(=O)CCl)c(Cl)c1 ZINC000217952358 BG For-Sale Unstable CYP1B1 46 40 COc1ccc(/C=C\C(=O)CCl)c(Cl)c1 ZINC000217952358 BG For-Sale Unstable CYP1A1 37 40 COc1ccc(/C=C\C(=O)CCl)c(Cl)c1 ZINC000217952358 BG For-Sale Unstable CYP1A2 0 40 COc1ccc(/C=C\C(=O)CCl)c(Cl)c1 ZINC000217952358 BG For-Sale Unstable BOTA 28 40 COc1ccc(/C=C\C(=O)CCl)c(Cl)c1 ZINC000217952358 BG For-Sale Unstable CYSP_PLAFA 53 48 COc1ccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1OC ZINC000217952387 GJ In-Stock Unstable DRD3 15 42 COc1ccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1OC ZINC000217952387 GJ In-Stock Unstable TRPV1 34 60 COc1ccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1OC ZINC000217952387 GJ In-Stock Unstable PYGL 0 42 COc1ccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1OC ZINC000217952387 GJ In-Stock Unstable HDAC1 18 45 COc1ccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1OC ZINC000217952387 GJ In-Stock Unstable MT-ND1 30 47 COc1ccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1OC ZINC000217952387 GJ In-Stock Unstable ABCG2 17 43 COc1cccc(/C=C/NC(=O)Nc2cc(C)cc(C)c2)c1 ZINC000217952400 CI For-Sale Unstable MTNR1A 30 45 COc1cccc(/C=C/NC(=O)Nc2cc(C)cc(C)c2)c1 ZINC000217952400 CI For-Sale Unstable MTNR1B 33 45 COc1cccc(/C=C/NC(=O)Nc2cc(C)cc(C)c2)c1 ZINC000217952400 CI For-Sale Unstable AKR1C2 28 40 COc1cccc(/C=C/NC(=O)Nc2cc(C)cc(C)c2)c1 ZINC000217952400 CI For-Sale Unstable KCNK3 19 42 O=C(Nc1ccn2nccc2c1)C1CC1 ZINC000217952401 BD In-Stock Unstable ADORA2B 0 43 O=C(Nc1ccn2nccc2c1)C1CC1 ZINC000217952401 BD In-Stock Unstable JAK1 0 42 O=C(Nc1ccn2nccc2c1)C1CC1 ZINC000217952401 BD In-Stock Unstable MAPK10 15 41 O=C(Nc1ccn2nccc2c1)C1CC1 ZINC000217952401 BD In-Stock Unstable TYK2 60 42 COc1ccc(/C=C\C(=O)CCl)c(OC)c1OC ZINC000217952435 CF For-Sale Unstable CYP1B1 28 44 COc1ccc(/C=C\C(=O)CCl)c(OC)c1OC ZINC000217952435 CF For-Sale Unstable TUBB1 45 40 COc1ccc(/C=C\C(=O)CCl)c(OC)c1OC ZINC000217952435 CF For-Sale Unstable CYSP_PLAFA 54 55 CO[C@@H]1CCN(c2ccc(CBr)cc2C)C1 ZINC000217952464 CG For-Sale Unstable LIPG 42 35 CCc1ncnc(NCc2ccncc2)c1F ZINC000217952492 BE On-Demand Unstable USP10 0 40 CCc1ncnc(NCc2ccncc2)c1F ZINC000217952492 BE On-Demand Unstable USP13 0 40 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccc(C(C)(C)C)cc1 ZINC000217952497 FJ In-Stock Unstable SDH1 0 40 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccc(C(C)(C)C)cc1 ZINC000217952497 FJ In-Stock Unstable MMP2 18 42 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccc(C(C)(C)C)cc1 ZINC000217952497 FJ In-Stock Unstable MMP9 15 42 O=C(Nc1ccn2nccc2c1)C1CCCC1 ZINC000217952508 BE In-Stock Unstable TYK2 54 38 COc1ccc(OCCNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217952510 EG For-Sale Unstable DRD4 41 31 COc1ccc(OCCNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217952510 EG For-Sale Unstable HRH2 26 45 COc1ccc(OCCNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217952510 EG For-Sale Unstable CYP1B1 23 41 COc1ccc(OCCNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217952510 EG For-Sale Unstable AHR 29 40 COc1ccc(OCCNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217952510 EG For-Sale Unstable MTNR1A 120 57 COc1ccc(OCCNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217952510 EG For-Sale Unstable MTNR1B 104 57 COc1ccc(OCCNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217952510 EG For-Sale Unstable CYP1A1 21 41 CC(C)c1ccc(/C=C\C(=O)CCl)cc1 ZINC000217952527 BH For-Sale Unstable SSSIM 15 46 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc2nccnc2c1 ZINC000217952531 GF For-Sale Unstable HCRTR1 47 35 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc2nccnc2c1 ZINC000217952531 GF For-Sale Unstable HCRTR2 50 35 CN1CCC(N(C)Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217952537 CE For-Sale Unstable PTGER2 46 48 CN1CCC(N(C)Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217952537 CE For-Sale Unstable PTGER4 22 48 CN1CCC(N(C)Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217952537 CE For-Sale Unstable PTGER3 19 48 CN1CCC(N(C)Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217952537 CE For-Sale Unstable NOS3 15 42 CN1CCC(N(C)Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217952537 CE For-Sale Unstable PTGDR 17 44 CO[C@H]1CCN(c2ccc(CBr)cc2C)C1 ZINC000217952547 CG For-Sale Unstable LIPG 42 35 C[C@H]1CN(C)[C@@H](C)C[C@@H]1NCCc1cccc(F)c1 ZINC000217952560 CF For-Sale Unstable HRH2 0 47 C[C@H]1CN(C)[C@@H](C)C[C@@H]1NCCc1cccc(F)c1 ZINC000217952560 CF For-Sale Unstable CHRM4 0 47 Cc1ccccc1OC[C@H](C)NC(=O)/C=C/c1ccc(C(C)(C)C)cc1 ZINC000217952577 FJ In-Stock Unstable SDH1 0 40 Cc1ccccc1OC[C@H](C)NC(=O)/C=C/c1ccc(C(C)(C)C)cc1 ZINC000217952577 FJ In-Stock Unstable MMP2 18 42 Cc1ccccc1OC[C@H](C)NC(=O)/C=C/c1ccc(C(C)(C)C)cc1 ZINC000217952577 FJ In-Stock Unstable MMP9 15 42 Cc1cc([N+](=O)[O-])ccc1N[C@H]1C[C@H](C)CC[C@H]1C(C)C ZINC000217952593 CJ For-Sale Unstable TRPM8 15 41 CCc1ncnc(NCCCN2CCOCC2)c1F ZINC000217952594 CD On-Demand Unstable EGFR 20 43 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc2nccnc2c1 ZINC000217952609 GF For-Sale Unstable HCRTR1 47 35 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc2nccnc2c1 ZINC000217952609 GF For-Sale Unstable HCRTR2 50 35 COc1cccc(/C=C/NC(=O)N(CCN)C(C)=O)c1 ZINC000217952623 CD For-Sale Unstable MTNR1A 35 42 COc1cccc(/C=C/NC(=O)N(CCN)C(C)=O)c1 ZINC000217952623 CD For-Sale Unstable MTNR1B 36 42 O=C(O)[C@@H]1C[C@@H]2CCCC[C@@H]2N1C(=O)Nc1nccs1 ZINC000217952667 CE On-Demand Unstable MAP1 88 42 Cc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1 ZINC000217952672 FJ In-Stock Unstable SDH1 0 40 Cc1cc([N+](=O)[O-])ccc1N[C@H]1C[C@@H](C)CC[C@H]1C(C)C ZINC000217952694 CJ For-Sale Unstable TRPM8 15 41 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc2nccnc2c1 ZINC000217952695 GF For-Sale Unstable HCRTR1 47 35 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc2nccnc2c1 ZINC000217952695 GF For-Sale Unstable HCRTR2 50 35 COc1cccc(/C=C/NC(=O)NCCNC(C)=O)c1 ZINC000217952718 CD For-Sale Unstable DRD4 44 33 COc1cccc(/C=C/NC(=O)NCCNC(C)=O)c1 ZINC000217952718 CD For-Sale Unstable CYP1B1 29 42 COc1cccc(/C=C/NC(=O)NCCNC(C)=O)c1 ZINC000217952718 CD For-Sale Unstable NQO2 48 40 COc1cccc(/C=C/NC(=O)NCCNC(C)=O)c1 ZINC000217952718 CD For-Sale Unstable MTR1B_CHICK 0 40 COc1cccc(/C=C/NC(=O)NCCNC(C)=O)c1 ZINC000217952718 CD For-Sale Unstable AHR 23 43 COc1cccc(/C=C/NC(=O)NCCNC(C)=O)c1 ZINC000217952718 CD For-Sale Unstable MTNR1A 141 57 COc1cccc(/C=C/NC(=O)NCCNC(C)=O)c1 ZINC000217952718 CD For-Sale Unstable MTNR1B 127 57 COc1cccc(/C=C/NC(=O)NCCNC(C)=O)c1 ZINC000217952718 CD For-Sale Unstable CYP1A1 21 42 Cc1ccccc1C(=O)Nc1ccn2nccc2c1 ZINC000217952734 CF In-Stock Unstable AVPR2 30 40 Cc1ccccc1C(=O)Nc1ccn2nccc2c1 ZINC000217952734 CF In-Stock Unstable AVPR1A 27 40 Cc1ccccc1C(=O)Nc1ccn2nccc2c1 ZINC000217952734 CF In-Stock Unstable GRM4 31 48 Cc1ccccc1C(=O)Nc1ccn2nccc2c1 ZINC000217952734 CF In-Stock Unstable CCR8 40 31 Cc1ccccc1C(=O)Nc1ccn2nccc2c1 ZINC000217952734 CF In-Stock Unstable NR2E3 31 41 Cc1ccccc1C(=O)Nc1ccn2nccc2c1 ZINC000217952734 CF In-Stock Unstable KCNK3 81 52 Cc1ccccc1C(=O)Nc1ccn2nccc2c1 ZINC000217952734 CF In-Stock Unstable KCNK9 73 49 O=C(O)[C@@H]1C[C@H]2CCCC[C@@H]2N1C(=O)Nc1nccs1 ZINC000217952750 CE On-Demand Unstable MAP1 88 42 Cc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1 ZINC000217952752 FJ In-Stock Unstable SDH1 0 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc2nccnc2c1 ZINC000217952768 GF For-Sale Unstable HCRTR1 47 35 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc2nccnc2c1 ZINC000217952768 GF For-Sale Unstable HCRTR2 50 35 CCN(C(=O)N/C=C/c1cccc(OC)c1)C(C)(C)C ZINC000217952822 CG For-Sale Unstable MTNR1A 41 43 CCN(C(=O)N/C=C/c1cccc(OC)c1)C(C)(C)C ZINC000217952822 CG For-Sale Unstable MTNR1B 41 43 COc1ccc(OC2CCN(C(=O)CCC3=NNC(=O)CC3)CC2)cc1 ZINC000217952843 FE In-Stock Unstable PRSS2 51 34 CC(C)(C)c1ccc(C(=O)Nc2ccn3nccc3c2)cc1 ZINC000217952848 CH In-Stock Unstable KIT 18 41 CC(C)(C)c1ccc(C(=O)Nc2ccn3nccc3c2)cc1 ZINC000217952848 CH In-Stock Unstable TRPV1 34 52 CC(C)(C)c1ccc(C(=O)Nc2ccn3nccc3c2)cc1 ZINC000217952848 CH In-Stock Unstable PRNP 56 35 CC(C)(C)c1ccc(C(=O)Nc2ccn3nccc3c2)cc1 ZINC000217952848 CH In-Stock Unstable FLT1 25 45 CC(C)(C)c1ccc(C(=O)Nc2ccn3nccc3c2)cc1 ZINC000217952848 CH In-Stock Unstable NR1H4 19 44 CC(C)(C)c1ccc(C(=O)Nc2ccn3nccc3c2)cc1 ZINC000217952848 CH In-Stock Unstable MAP3K5 64 42 CC(C)(C)c1ccc(C(=O)Nc2ccn3nccc3c2)cc1 ZINC000217952848 CH In-Stock Unstable BTK 22 43 CC(C)(C)c1ccc(C(=O)Nc2ccn3nccc3c2)cc1 ZINC000217952848 CH In-Stock Unstable CYNT 25 43 CC(C)(C)c1ccc(C(=O)Nc2ccn3nccc3c2)cc1 ZINC000217952848 CH In-Stock Unstable DDR1 54 37 CC(C)(C)c1ccc(C(=O)Nc2ccn3nccc3c2)cc1 ZINC000217952848 CH In-Stock Unstable NAMPT 17 50 CC(C)(C)c1ccc(C(=O)Nc2ccn3nccc3c2)cc1 ZINC000217952848 CH In-Stock Unstable KCNK3 92 50 CC(C)(C)c1ccc(C(=O)Nc2ccn3nccc3c2)cc1 ZINC000217952848 CH In-Stock Unstable KCNK9 44 36 CC1CCN(c2ccc([C@@H](C)NC(=O)/C=C/c3ccc(C(C)(C)C)cc3)cc2)CC1 ZINC000217952853 HK In-Stock Unstable KCNQ2 46 35 COc1cccc(/C=C/NC(=O)NC23CC4CC(CC(C4)C2)C3)c1 ZINC000217952944 EH For-Sale Unstable MTNR1A 26 40 COc1cccc(/C=C/NC(=O)NC23CC4CC(CC(C4)C2)C3)c1 ZINC000217952944 EH For-Sale Unstable MTNR1B 29 40 COc1cccc(/C=C/NC(=O)NC23CC4CC(CC(C4)C2)C3)c1 ZINC000217952944 EH For-Sale Unstable EPHX2 109 63 CC1CCN(c2ccc([C@H](C)NC(=O)/C=C/c3ccc(C(C)(C)C)cc3)cc2)CC1 ZINC000217952948 HK In-Stock Unstable KCNQ2 46 35 O=C(c1cccc(-c2ccccc2)c1)N1CCC[C@@H](N2CCCC2=O)C1 ZINC000217952967 EH In-Stock Unstable INHA 26 41 O=C(c1cccc(-c2ccccc2)c1)N1CCC[C@@H](N2CCCC2=O)C1 ZINC000217952967 EH In-Stock Unstable HSD11B1 15 46 O=C(c1cccc(-c2ccccc2)c1)N1CCC[C@@H](N2CCCC2=O)C1 ZINC000217952967 EH In-Stock Unstable ABHD6 0 42 O=C(c1cccc(-c2ccccc2)c1)N1CCC[C@@H](N2CCCC2=O)C1 ZINC000217952967 EH In-Stock Unstable RHOA 0 43 O=C(c1cccc(-c2ccccc2)c1)N1CCC[C@@H](N2CCCC2=O)C1 ZINC000217952967 EH In-Stock Unstable L3MBTL1 0 41 O=C(c1cccc(-c2ccccc2)c1)N1CCC[C@@H](N2CCCC2=O)C1 ZINC000217952967 EH In-Stock Unstable L3MBTL3 43 39 O=C(c1cccc(-c2ccccc2)c1)N1CCC[C@@H](N2CCCC2=O)C1 ZINC000217952967 EH In-Stock Unstable SLC6A7 0 44 CCCCOc1ccc(C(=O)Nc2ccn3nccc3c2)cc1 ZINC000217952970 DH In-Stock Unstable CYSLTR1 17 42 CCCCOc1ccc(C(=O)Nc2ccn3nccc3c2)cc1 ZINC000217952970 DH In-Stock Unstable KCNQ1 0 43 CCCCOc1ccc(C(=O)Nc2ccn3nccc3c2)cc1 ZINC000217952970 DH In-Stock Unstable CYSLTR2 52 34 CCCCOc1ccc(C(=O)Nc2ccn3nccc3c2)cc1 ZINC000217952970 DH In-Stock Unstable TRPV1 18 44 CCCCOc1ccc(C(=O)Nc2ccn3nccc3c2)cc1 ZINC000217952970 DH In-Stock Unstable SCN2A 18 40 CCCCOc1ccc(C(=O)Nc2ccn3nccc3c2)cc1 ZINC000217952970 DH In-Stock Unstable PRNP 61 35 CCCCOc1ccc(C(=O)Nc2ccn3nccc3c2)cc1 ZINC000217952970 DH In-Stock Unstable PLA2G4B 92 38 CCCCOc1ccc(C(=O)Nc2ccn3nccc3c2)cc1 ZINC000217952970 DH In-Stock Unstable FAAH 23 40 CCCCOc1ccc(C(=O)Nc2ccn3nccc3c2)cc1 ZINC000217952970 DH In-Stock Unstable DDR1 59 39 CCCCOc1ccc(C(=O)Nc2ccn3nccc3c2)cc1 ZINC000217952970 DH In-Stock Unstable KCNK3 69 36 CO[C@@H]1CCN(c2ccc(CBr)cc2F)C1 ZINC000217953017 CF For-Sale Unstable LIPG 51 39 O=C(c1cccc(-c2ccccc2)c1)N1CCC[C@H](N2CCCC2=O)C1 ZINC000217953050 EH In-Stock Unstable INHA 26 41 O=C(c1cccc(-c2ccccc2)c1)N1CCC[C@H](N2CCCC2=O)C1 ZINC000217953050 EH In-Stock Unstable HSD11B1 15 46 O=C(c1cccc(-c2ccccc2)c1)N1CCC[C@H](N2CCCC2=O)C1 ZINC000217953050 EH In-Stock Unstable ABHD6 0 42 O=C(c1cccc(-c2ccccc2)c1)N1CCC[C@H](N2CCCC2=O)C1 ZINC000217953050 EH In-Stock Unstable RHOA 0 43 O=C(c1cccc(-c2ccccc2)c1)N1CCC[C@H](N2CCCC2=O)C1 ZINC000217953050 EH In-Stock Unstable L3MBTL1 0 41 O=C(c1cccc(-c2ccccc2)c1)N1CCC[C@H](N2CCCC2=O)C1 ZINC000217953050 EH In-Stock Unstable L3MBTL3 43 39 O=C(c1cccc(-c2ccccc2)c1)N1CCC[C@H](N2CCCC2=O)C1 ZINC000217953050 EH In-Stock Unstable SLC6A7 0 44 COc1cccc(/C=C/NC(=O)Nc2cccc3cccnc23)c1 ZINC000217953054 DI For-Sale Unstable TRPV1 0 40 COc1cccc(/C=C/NC(=O)Nc2cccc3cccnc23)c1 ZINC000217953054 DI For-Sale Unstable P2RY1 19 41 COc1cccc(/C=C/NC(=O)Nc2cccc3cccnc23)c1 ZINC000217953054 DI For-Sale Unstable MTNR1A 25 42 COc1cccc(/C=C/NC(=O)Nc2cccc3cccnc23)c1 ZINC000217953054 DI For-Sale Unstable MTNR1B 25 42 COc1ccc(C(=O)Nc2ccn3nccc3c2)c(OC)c1 ZINC000217953076 CF In-Stock Unstable BRPF1 0 40 O=C(CCCc1nc(-c2ccco2)no1)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217953080 GE In-Stock Unstable CHRNA4 28 49 CO[C@H]1CCN(c2ccc(CBr)cc2F)C1 ZINC000217953093 CF For-Sale Unstable LIPG 51 39 Nc1nc(/C=C\c2c[nH]c3cc(Br)ccc23)cs1 ZINC000217953094 DI For-Sale Unstable TDO2 0 41 Cc1c(OC(C)C)cccc1C(=O)OC(C)C ZINC000217953097 BG For-Sale Unstable KCNK3 42 40 Cc1c(OC(C)C)cccc1C(=O)OC(C)C ZINC000217953097 BG For-Sale Unstable KCNK9 41 40 CN(Cc1cccc(/C=C\C(=O)O)c1)C1CCOCC1 ZINC000217953104 CE For-Sale Unstable PTGER2 21 40 C[C@@H](CNC1CCN(C(=O)OC(C)(C)C)CC1)CN1CCCC1 ZINC000217953150 EF On-Demand Unstable GPR119 30 41 COc1cccc(/C=C/NC(=O)NCc2ccccc2F)c1 ZINC000217953157 DG For-Sale Unstable DRD4 41 31 COc1cccc(/C=C/NC(=O)NCc2ccccc2F)c1 ZINC000217953157 DG For-Sale Unstable MTNR1A 57 41 COc1cccc(/C=C/NC(=O)NCc2ccccc2F)c1 ZINC000217953157 DG For-Sale Unstable MTNR1B 54 41 C[C@@H]1CCC[C@H]([C@@H](N)CCCc2ccccc2)C1 ZINC000217953160 BI For-Sale Unstable SLC18A2 41 44 C[C@@H]1CCC[C@H]([C@@H](N)CCCc2ccccc2)C1 ZINC000217953160 BI For-Sale Unstable SIGMAR1 19 40 O=C(Cn1ccc2ccccc21)N1CCCC[C@H]1c1cccnc1 ZINC000217953176 DH In-Stock Unstable PTAFR 20 43 O=C(Cn1ccc2ccccc21)N1CCCC[C@H]1c1cccnc1 ZINC000217953176 DH In-Stock Unstable CHRNA2 41 43 O=C(Cn1ccc2ccccc21)N1CCCC[C@H]1c1cccnc1 ZINC000217953176 DH In-Stock Unstable CHRNA7 20 43 O=C(Cn1ccc2ccccc21)N1CCCC[C@H]1c1cccnc1 ZINC000217953176 DH In-Stock Unstable COLA 118 45 O=C(Cn1ccc2ccccc21)N1CCCC[C@H]1c1cccnc1 ZINC000217953176 DH In-Stock Unstable CPT1A 112 45 O=C(Cn1ccc2ccccc21)N1CCCC[C@H]1c1cccnc1 ZINC000217953176 DH In-Stock Unstable GPBAR1 0 43 O=C(Cn1ccc2ccccc21)N1CCCC[C@H]1c1cccnc1 ZINC000217953176 DH In-Stock Unstable CRTY 0 43 O=C(O)[C@@H]1C[C@@H]2CCCC[C@@H]2N1C(=O)N1CCOCC1 ZINC000217953181 CD On-Demand Unstable AKR1C3 30 40 O=C(Nc1ccn2nccc2c1)c1ccc2c(c1)OCO2 ZINC000217953187 CE In-Stock Unstable KCNK3 51 35 C[C@H](CNC1CCN(C(=O)OC(C)(C)C)CC1)CN1CCCC1 ZINC000217953231 EF On-Demand Unstable GPR119 30 41 C[C@H]1CCC[C@H]([C@@H](N)CCCc2ccccc2)C1 ZINC000217953246 BI For-Sale Unstable SLC18A2 41 44 C[C@H]1CCC[C@H]([C@@H](N)CCCc2ccccc2)C1 ZINC000217953246 BI For-Sale Unstable SIGMAR1 19 40 O=C(O)[C@@H]1C[C@H]2CCCC[C@@H]2N1C(=O)N1CCOCC1 ZINC000217953267 CD On-Demand Unstable AKR1C3 30 40 COc1cccc(/C=C/NC(=O)N2c3ccccc3C[C@@H]2C)c1 ZINC000217953272 DH For-Sale Unstable DRD4 30 46 CC(C)CCn1cnc2ccc(NC(=O)CCCC[C@@H]3SC[C@@H]4NC(=O)N[C@H]34)cc2c1=O ZINC000217953289 JG In-Stock Unstable AGAL_COFAR 0 46 CC(C)CCn1cnc2ccc(NC(=O)CCCC[C@@H]3SC[C@@H]4NC(=O)N[C@H]34)cc2c1=O ZINC000217953289 JG In-Stock Unstable BIRA 0 40 O=C(Nc1ccn2nccc2c1)c1ccc(F)cc1 ZINC000217953294 CF In-Stock Anodyne HTR1F 39 42 O=C(Nc1ccn2nccc2c1)c1ccc(F)cc1 ZINC000217953294 CF In-Stock Anodyne CXCR2 15 40 O=C(Nc1ccn2nccc2c1)c1ccc(F)cc1 ZINC000217953294 CF In-Stock Anodyne PRNP 50 36 O=C(Nc1ccn2nccc2c1)c1ccc(F)cc1 ZINC000217953294 CF In-Stock Anodyne SHH 25 41 O=C(Nc1ccn2nccc2c1)c1ccc(F)cc1 ZINC000217953294 CF In-Stock Anodyne KCNK3 76 43 O=C(Nc1ccn2nccc2c1)c1ccc(F)cc1 ZINC000217953294 CF In-Stock Anodyne KCNK9 40 37 C[C@@H]1CCC[C@@H]([C@@H](N)CCCc2ccccc2)C1 ZINC000217953322 BI For-Sale Unstable SLC18A2 41 44 C[C@@H]1CCC[C@@H]([C@@H](N)CCCc2ccccc2)C1 ZINC000217953322 BI For-Sale Unstable SIGMAR1 19 40 COc1ccc(/C=C\C(=O)O)cc1CN(C)CC1CC1 ZINC000217953325 CF For-Sale Unstable AKR1C3 37 40 COc1cccc(/C=C/NC(=O)N2c3ccccc3C[C@H]2C)c1 ZINC000217953362 DH For-Sale Unstable DRD4 30 46 COc1cc2c(cc1OC)[C@@H](c1ccccc1)N(C(=O)c1cc(C(C)C)nc3onc(C)c13)CC2 ZINC000217953382 JK On-Demand Unstable MTNR1B 20 42 O=C(Nc1ccn2nccc2c1)c1ccccc1Cl ZINC000217953399 CG In-Stock Anodyne JAK1 0 45 O=C(Nc1ccn2nccc2c1)c1ccccc1Cl ZINC000217953399 CG In-Stock Anodyne FLT1 29 41 O=C(Nc1ccn2nccc2c1)c1ccccc1Cl ZINC000217953399 CG In-Stock Anodyne GRM4 62 50 O=C(Nc1ccn2nccc2c1)c1ccccc1Cl ZINC000217953399 CG In-Stock Anodyne TYK2 59 39 O=C(Nc1ccn2nccc2c1)c1ccccc1Cl ZINC000217953399 CG In-Stock Anodyne EPHB3 46 44 O=C(Nc1ccn2nccc2c1)c1ccccc1Cl ZINC000217953399 CG In-Stock Anodyne NR2E3 74 40 O=C(Nc1ccn2nccc2c1)c1ccccc1Cl ZINC000217953399 CG In-Stock Anodyne SHH 49 50 O=C(Nc1ccn2nccc2c1)c1ccccc1Cl ZINC000217953399 CG In-Stock Anodyne SMO 30 48 O=C(Nc1ccn2nccc2c1)c1ccccc1Cl ZINC000217953399 CG In-Stock Anodyne KCNK3 65 46 O=C(Nc1ccn2nccc2c1)c1ccccc1Cl ZINC000217953399 CG In-Stock Anodyne KCNK9 58 37 CO[C@@H]1CCN(c2ccc(CBr)cc2C(F)(F)F)C1 ZINC000217953404 EH For-Sale Unstable LIPG 59 41 COCCn1cc(C(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)c2cc(Cl)ccc21 ZINC000217953405 IG In-Stock Unstable CHRNA4 26 42 C[C@H]1CCC[C@@H]([C@@H](N)CCCc2ccccc2)C1 ZINC000217953406 BI For-Sale Unstable SLC18A2 41 44 C[C@H]1CCC[C@@H]([C@@H](N)CCCc2ccccc2)C1 ZINC000217953406 BI For-Sale Unstable SIGMAR1 19 40 C[C@H](Oc1ccc(Cl)cc1)C(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217953424 CE On-Demand Unstable GUAB 0 44 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)C[C@@H]1CCCN1 ZINC000217953429 CF For-Sale Unstable TRPM8 17 47 CCN(Cc1cccc(/C=C\C(=O)O)c1)C[C@@H]1CCCO1 ZINC000217953430 CF For-Sale Unstable OXTR 26 43 CCN(Cc1cccc(/C=C\C(=O)O)c1)C[C@@H]1CCCO1 ZINC000217953430 CF For-Sale Unstable AVPR1A 0 43 COc1ccc(CC/C(C)=C2\CC(=O)NC2=O)cc1 ZINC000217953432 CD For-Sale Unstable SLC18A2 15 41 COc1cc2c(cc1OC)[C@H](c1ccccc1)N(C(=O)c1cc(C(C)C)nc3onc(C)c13)CC2 ZINC000217953466 JK On-Demand Unstable MTNR1B 30 42 COc1cccc(/C=C/NC(=O)NC2CC2)c1 ZINC000217953467 BE For-Sale Unstable CYP1B1 24 41 COc1cccc(/C=C/NC(=O)NC2CC2)c1 ZINC000217953467 BE For-Sale Unstable MTNR1A 40 43 COc1cccc(/C=C/NC(=O)NC2CC2)c1 ZINC000217953467 BE For-Sale Unstable MTNR1B 38 43 COc1cccc(/C=C/NC(=O)NC2CC2)c1 ZINC000217953467 BE For-Sale Unstable CYP1A1 18 41 CO[C@H]1CCN(c2ccc(CBr)cc2C(F)(F)F)C1 ZINC000217953485 EH For-Sale Unstable LIPG 59 41 O=C(Nc1ccn2nccc2c1)c1cccc(Cl)c1 ZINC000217953507 CG In-Stock Anodyne PPIA 18 48 O=C(Nc1ccn2nccc2c1)c1cccc(Cl)c1 ZINC000217953507 CG In-Stock Anodyne CPT1A 45 38 O=C(Nc1ccn2nccc2c1)c1cccc(Cl)c1 ZINC000217953507 CG In-Stock Anodyne GRM5 16 54 O=C(Nc1ccn2nccc2c1)c1cccc(Cl)c1 ZINC000217953507 CG In-Stock Anodyne CSF1R 19 50 O=C(Nc1ccn2nccc2c1)c1cccc(Cl)c1 ZINC000217953507 CG In-Stock Anodyne BRAF 25 41 O=C(Nc1ccn2nccc2c1)c1cccc(Cl)c1 ZINC000217953507 CG In-Stock Anodyne LUCI_LUCLA 16 43 O=C(Nc1ccn2nccc2c1)c1cccc(Cl)c1 ZINC000217953507 CG In-Stock Anodyne TAAR1 25 52 O=C(Nc1ccn2nccc2c1)c1cccc(Cl)c1 ZINC000217953507 CG In-Stock Anodyne DDR1 37 44 O=C(Nc1ccn2nccc2c1)c1cccc(Cl)c1 ZINC000217953507 CG In-Stock Anodyne KCNK3 89 43 O=C(Nc1ccn2nccc2c1)c1cccc(Cl)c1 ZINC000217953507 CG In-Stock Anodyne KCNK9 52 53 COc1ccc2c(c1Cl)C(=O)NCC2 ZINC000217953512 BD For-Sale Unstable CSNK1G2 51 30 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)C[C@@H]1CCCN1 ZINC000217953523 CF On-Demand Unstable TRPM8 19 47 COC(=O)C[C@H](c1ccc(O)c(OC)c1)c1cc2c(cc1O)OCO2 ZINC000217953526 EF In-Stock Unstable FOLH1 23 40 COC(=O)C[C@H](c1ccc(O)c(OC)c1)c1cc2c(cc1O)OCO2 ZINC000217953526 EF In-Stock Unstable RORC 54 42 COC[C@H](C)N(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217953530 CE For-Sale Unstable NR1H4 41 40 COC[C@H](C)N(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217953530 CE For-Sale Unstable AKR1C3 28 40 COc1cccc(/C=C/NC(=O)NCc2ccccc2OC)c1 ZINC000217953565 DG For-Sale Unstable CYP1B1 43 38 COc1cccc(/C=C/NC(=O)NCc2ccccc2OC)c1 ZINC000217953565 DG For-Sale Unstable MTNR1A 62 43 COc1cccc(/C=C/NC(=O)NCc2ccccc2OC)c1 ZINC000217953565 DG For-Sale Unstable MTNR1B 61 43 COc1cccc(/C=C/NC(=O)NCc2ccccc2OC)c1 ZINC000217953565 DG For-Sale Unstable CYP1A1 28 43 COc1cccc(/C=C/NC(=O)NCc2ccccc2OC)c1 ZINC000217953565 DG For-Sale Unstable ABCG2 17 44 C[C@H](Oc1ccc(Cl)cc1)C(=O)N[C@H]1CCC[C@@H]1CO ZINC000217953570 CE For-Sale Unstable AVPR1A 19 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1c[nH]c2ccccc12 ZINC000217953598 GG For-Sale Unstable HCRTR1 42 38 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1c[nH]c2ccccc12 ZINC000217953598 GG For-Sale Unstable HCRTR2 48 38 COC(=O)C[C@@H](c1ccc(O)c(OC)c1)c1cc2c(cc1O)OCO2 ZINC000217953606 EF In-Stock Unstable FOLH1 23 40 COC(=O)C[C@@H](c1ccc(O)c(OC)c1)c1cc2c(cc1O)OCO2 ZINC000217953606 EF In-Stock Unstable RORC 54 42 COC[C@@H](C)N(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217953614 CE For-Sale Unstable NR1H4 41 40 COC[C@@H](C)N(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217953614 CE For-Sale Unstable AKR1C3 28 40 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)C[C@@H]1CCCN1 ZINC000217953618 CF For-Sale Unstable TRPM8 17 47 O=C(Nc1ccn2nccc2c1)c1cccc(Br)c1 ZINC000217953634 DG In-Stock Anodyne TAAR1 25 40 O=C(Nc1ccn2nccc2c1)c1cccc(Br)c1 ZINC000217953634 DG In-Stock Anodyne KCNK3 87 43 O=C(Nc1ccn2nccc2c1)c1cccc(Br)c1 ZINC000217953634 DG In-Stock Anodyne KCNK9 50 40 COc1cccc(/C=C/NC(=O)N2CCN(c3ncccn3)CC2)c1 ZINC000217953660 ED For-Sale Unstable DRD4 43 32 COc1cccc(/C=C/NC(=O)N2CCN(c3ncccn3)CC2)c1 ZINC000217953660 ED For-Sale Unstable PDGFRB 39 41 COc1cccc(/C=C/NC(=O)N2CCN(c3ncccn3)CC2)c1 ZINC000217953660 ED For-Sale Unstable SLC6A7 0 48 CCOC(=O)N1CCN(c2cc(Cl)nc(C3CC3)n2)CC1 ZINC000217953670 DE On-Demand Unstable P2RY12 41 33 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1c[nH]c2ccccc12 ZINC000217953682 GG For-Sale Unstable HCRTR1 42 38 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1c[nH]c2ccccc12 ZINC000217953682 GG For-Sale Unstable HCRTR2 48 38 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)C[C@@H]1CCCN1 ZINC000217953700 CF For-Sale Unstable TRPM8 17 47 COc1ccc(Cl)cc1C(=O)Nc1ccn2nccc2c1 ZINC000217953736 DG In-Stock Unstable HTR2A 38 46 COc1ccc(Cl)cc1C(=O)Nc1ccn2nccc2c1 ZINC000217953736 DG In-Stock Unstable F10 50 35 COc1ccc(Cl)cc1C(=O)Nc1ccn2nccc2c1 ZINC000217953736 DG In-Stock Unstable COLA 85 37 COc1ccc(Cl)cc1C(=O)Nc1ccn2nccc2c1 ZINC000217953736 DG In-Stock Unstable CPT1A 71 37 COc1ccc(Cl)cc1C(=O)Nc1ccn2nccc2c1 ZINC000217953736 DG In-Stock Unstable CPT2 48 36 COc1ccc(Cl)cc1C(=O)Nc1ccn2nccc2c1 ZINC000217953736 DG In-Stock Unstable GRM4 30 46 COc1ccc(Cl)cc1C(=O)Nc1ccn2nccc2c1 ZINC000217953736 DG In-Stock Unstable KCNMA1 35 48 COc1ccc(Cl)cc1C(=O)Nc1ccn2nccc2c1 ZINC000217953736 DG In-Stock Unstable CPT1B 56 36 COc1ccc(Cl)cc1C(=O)Nc1ccn2nccc2c1 ZINC000217953736 DG In-Stock Unstable TYK2 15 44 COc1ccc(Cl)cc1C(=O)Nc1ccn2nccc2c1 ZINC000217953736 DG In-Stock Unstable EPHB3 32 41 COc1ccc(Cl)cc1C(=O)Nc1ccn2nccc2c1 ZINC000217953736 DG In-Stock Unstable SHH 28 40 COc1ccc(Cl)cc1C(=O)Nc1ccn2nccc2c1 ZINC000217953736 DG In-Stock Unstable ENPP1 49 31 COc1ccc(Cl)cc1C(=O)Nc1ccn2nccc2c1 ZINC000217953736 DG In-Stock Unstable KCNK3 49 44 COc1ccc(Cl)cc1C(=O)Nc1ccn2nccc2c1 ZINC000217953736 DG In-Stock Unstable KCNK9 41 44 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1c[nH]c2ccccc12 ZINC000217953761 GG For-Sale Unstable HCRTR1 42 38 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1c[nH]c2ccccc12 ZINC000217953761 GG For-Sale Unstable HCRTR2 48 38 CCc1ncnc(NCc2cccc(Cl)c2)c1F ZINC000217953770 CG On-Demand Unstable ABL1 22 45 COc1cccc(/C=C/NC(=O)N2CCN(c3cccc(C)c3)CC2)c1 ZINC000217953788 FH For-Sale Unstable DRD4 46 40 COc1cccc(/C=C/NC(=O)N2CCN(c3cccc(C)c3)CC2)c1 ZINC000217953788 FH For-Sale Unstable CCKAR 35 42 COc1cccc(/C=C/NC(=O)N2CCN(c3cccc(C)c3)CC2)c1 ZINC000217953788 FH For-Sale Unstable CCR1 0 40 COc1cccc(/C=C/NC(=O)N2CCN(c3cccc(C)c3)CC2)c1 ZINC000217953788 FH For-Sale Unstable GPR183 0 44 CCCOc1ccc([C@@H](N)[C@@H]2CCC[C@@H](C)C2)cc1 ZINC000217953809 CI For-Sale Unstable ACACA 30 40 COc1ccc(/C=C2/CC(=O)NC2=O)cc1Br ZINC000217953815 CD For-Sale Unstable ESRRA 52 46 COc1ccc(/C=C2/CC(=O)NC2=O)cc1Br ZINC000217953815 CD For-Sale Unstable HPGD 44 42 O=C(C[C@H]1CCCN1)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000217953818 CD On-Demand Unstable DRD2 0 49 O=C(C[C@H]1CCCN1)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000217953818 CD On-Demand Unstable DRD4 35 55 O=C(C[C@H]1CCCN1)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000217953818 CD On-Demand Unstable ACHE 29 42 O=C(C[C@H]1CCCN1)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000217953818 CD On-Demand Unstable DRD3 30 47 O=C(C[C@H]1CCCN1)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000217953818 CD On-Demand Unstable LTA4H 26 40 O=C(C[C@H]1CCCN1)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000217953818 CD On-Demand Unstable SIGMAR1 52 57 O=C(C[C@H]1CCCN1)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000217953818 CD On-Demand Unstable CCR3 37 53 O=C(C[C@H]1CCCN1)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000217953818 CD On-Demand Unstable MLNR 42 35 O=C(C[C@H]1CCCN1)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000217953818 CD On-Demand Unstable MCHR1 28 57 O=C(C[C@H]1CCCN1)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000217953818 CD On-Demand Unstable BIRC2 42 37 O=C(C[C@H]1CCCN1)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000217953818 CD On-Demand Unstable ADIPOR1 0 45 O=C(C[C@H]1CCCN1)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000217953818 CD On-Demand Unstable ADIPOR2 0 45 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1c[nH]c2ccccc12 ZINC000217953847 GG For-Sale Unstable HCRTR1 42 38 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1c[nH]c2ccccc12 ZINC000217953847 GG For-Sale Unstable HCRTR2 48 38 O=C(Nc1ccn2nccc2c1)c1ccccc1C(F)(F)F ZINC000217953858 DH In-Stock Anodyne FLT1 31 41 O=C(Nc1ccn2nccc2c1)c1ccccc1C(F)(F)F ZINC000217953858 DH In-Stock Anodyne GRM4 20 42 O=C(Nc1ccn2nccc2c1)c1ccccc1C(F)(F)F ZINC000217953858 DH In-Stock Anodyne RBP4 59 34 O=C(Nc1ccn2nccc2c1)c1ccccc1C(F)(F)F ZINC000217953858 DH In-Stock Anodyne NR2E3 43 31 O=C(Nc1ccn2nccc2c1)c1ccccc1C(F)(F)F ZINC000217953858 DH In-Stock Anodyne KCNK3 67 55 O=C(Nc1ccn2nccc2c1)c1ccccc1C(F)(F)F ZINC000217953858 DH In-Stock Anodyne KCNK9 53 48 O=C1C/C(=C/c2ccc(-c3ccc(F)cc3)s2)C(=O)N1 ZINC000217953896 CF For-Sale Unstable PRF1 46 39 CCOC(=O)N1CCC(NC(=O)N/C=C/c2cccc(OC)c2)CC1 ZINC000217953898 EF For-Sale Unstable MTNR1B 35 44 CCOC(=O)N1CCC(NC(=O)N/C=C/c2cccc(OC)c2)CC1 ZINC000217953898 EF For-Sale Unstable EPHX2 30 42 CCCOc1ccc([C@H](N)[C@@H]2CCC[C@@H](C)C2)cc1 ZINC000217953901 CI For-Sale Unstable ACACA 30 40 O=C(C[C@H]1CCCN1)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000217953904 CD On-Demand Unstable DRD2 0 49 O=C(C[C@H]1CCCN1)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000217953904 CD On-Demand Unstable DRD4 35 55 O=C(C[C@H]1CCCN1)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000217953904 CD On-Demand Unstable ACHE 29 42 O=C(C[C@H]1CCCN1)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000217953904 CD On-Demand Unstable DRD3 30 47 O=C(C[C@H]1CCCN1)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000217953904 CD On-Demand Unstable LTA4H 26 40 O=C(C[C@H]1CCCN1)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000217953904 CD On-Demand Unstable SIGMAR1 52 57 O=C(C[C@H]1CCCN1)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000217953904 CD On-Demand Unstable CCR3 37 53 O=C(C[C@H]1CCCN1)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000217953904 CD On-Demand Unstable MLNR 42 35 O=C(C[C@H]1CCCN1)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000217953904 CD On-Demand Unstable MCHR1 28 57 O=C(C[C@H]1CCCN1)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000217953904 CD On-Demand Unstable BIRC2 42 37 O=C(C[C@H]1CCCN1)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000217953904 CD On-Demand Unstable ADIPOR1 0 45 O=C(C[C@H]1CCCN1)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000217953904 CD On-Demand Unstable ADIPOR2 0 45 CN(Cc1cccc(/C=C\C(=O)O)c1)C[C@@H]1CCCO1 ZINC000217953908 CE For-Sale Unstable OXTR 28 45 CN(Cc1cccc(/C=C\C(=O)O)c1)C[C@@H]1CCCO1 ZINC000217953908 CE For-Sale Unstable AVPR1A 18 45 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)C(C)C ZINC000217953947 DE For-Sale Unstable ACE 15 43 O=C(CCC(=O)N1CCCCCC1)NCc1nc2cc(F)ccc2[nH]1 ZINC000217953956 EF In-Stock Unstable FABK 0 43 Cc1noc2nc(C(C)C)cc(C(=O)Nc3cc(Cl)ccc3N3CCN(C)CC3)c12 ZINC000217953967 II On-Demand Unstable DRD1 49 35 Cc1noc2nc(C(C)C)cc(C(=O)Nc3cc(Cl)ccc3N3CCN(C)CC3)c12 ZINC000217953967 II On-Demand Unstable WDR5 37 45 O=C(Nc1ccn2nccc2c1)c1cccc(C(F)(F)F)c1 ZINC000217953975 DH In-Stock Anodyne ABL1 23 46 O=C(Nc1ccn2nccc2c1)c1cccc(C(F)(F)F)c1 ZINC000217953975 DH In-Stock Anodyne INSR 22 41 O=C(Nc1ccn2nccc2c1)c1cccc(C(F)(F)F)c1 ZINC000217953975 DH In-Stock Anodyne KIT 25 52 O=C(Nc1ccn2nccc2c1)c1cccc(C(F)(F)F)c1 ZINC000217953975 DH In-Stock Anodyne KCNJ11 20 42 O=C(Nc1ccn2nccc2c1)c1cccc(C(F)(F)F)c1 ZINC000217953975 DH In-Stock Anodyne LCK 33 44 O=C(Nc1ccn2nccc2c1)c1cccc(C(F)(F)F)c1 ZINC000217953975 DH In-Stock Anodyne TRPV1 15 50 O=C(Nc1ccn2nccc2c1)c1cccc(C(F)(F)F)c1 ZINC000217953975 DH In-Stock Anodyne RAF1 18 43 O=C(Nc1ccn2nccc2c1)c1cccc(C(F)(F)F)c1 ZINC000217953975 DH In-Stock Anodyne FLT1 22 43 O=C(Nc1ccn2nccc2c1)c1cccc(C(F)(F)F)c1 ZINC000217953975 DH In-Stock Anodyne KDR 27 52 O=C(Nc1ccn2nccc2c1)c1cccc(C(F)(F)F)c1 ZINC000217953975 DH In-Stock Anodyne NPY5R 16 40 O=C(Nc1ccn2nccc2c1)c1cccc(C(F)(F)F)c1 ZINC000217953975 DH In-Stock Anodyne EPHB2 20 41 O=C(Nc1ccn2nccc2c1)c1cccc(C(F)(F)F)c1 ZINC000217953975 DH In-Stock Anodyne CCR2 68 39 O=C(Nc1ccn2nccc2c1)c1cccc(C(F)(F)F)c1 ZINC000217953975 DH In-Stock Anodyne BLK 19 40 O=C(Nc1ccn2nccc2c1)c1cccc(C(F)(F)F)c1 ZINC000217953975 DH In-Stock Anodyne EPHX2 15 47 O=C(Nc1ccn2nccc2c1)c1cccc(C(F)(F)F)c1 ZINC000217953975 DH In-Stock Anodyne HCK 23 41 O=C(Nc1ccn2nccc2c1)c1cccc(C(F)(F)F)c1 ZINC000217953975 DH In-Stock Anodyne LYN 33 41 O=C(Nc1ccn2nccc2c1)c1cccc(C(F)(F)F)c1 ZINC000217953975 DH In-Stock Anodyne TYK2 17 40 O=C(Nc1ccn2nccc2c1)c1cccc(C(F)(F)F)c1 ZINC000217953975 DH In-Stock Anodyne CSF1R 17 51 O=C(Nc1ccn2nccc2c1)c1cccc(C(F)(F)F)c1 ZINC000217953975 DH In-Stock Anodyne TEK 38 47 O=C(Nc1ccn2nccc2c1)c1cccc(C(F)(F)F)c1 ZINC000217953975 DH In-Stock Anodyne Q8MMZ8_EIMTE 0 43 O=C(Nc1ccn2nccc2c1)c1cccc(C(F)(F)F)c1 ZINC000217953975 DH In-Stock Anodyne EPHA3 18 42 O=C(Nc1ccn2nccc2c1)c1cccc(C(F)(F)F)c1 ZINC000217953975 DH In-Stock Anodyne BMX 32 42 O=C(Nc1ccn2nccc2c1)c1cccc(C(F)(F)F)c1 ZINC000217953975 DH In-Stock Anodyne BTK 27 46 O=C(Nc1ccn2nccc2c1)c1cccc(C(F)(F)F)c1 ZINC000217953975 DH In-Stock Anodyne BRAF 51 48 O=C(Nc1ccn2nccc2c1)c1cccc(C(F)(F)F)c1 ZINC000217953975 DH In-Stock Anodyne EPHB4 28 45 O=C(Nc1ccn2nccc2c1)c1cccc(C(F)(F)F)c1 ZINC000217953975 DH In-Stock Anodyne TEC 15 40 O=C(Nc1ccn2nccc2c1)c1cccc(C(F)(F)F)c1 ZINC000217953975 DH In-Stock Anodyne TXK 26 40 O=C(Nc1ccn2nccc2c1)c1cccc(C(F)(F)F)c1 ZINC000217953975 DH In-Stock Anodyne DDR1 50 46 O=C(Nc1ccn2nccc2c1)c1cccc(C(F)(F)F)c1 ZINC000217953975 DH In-Stock Anodyne SHH 29 45 O=C(Nc1ccn2nccc2c1)c1cccc(C(F)(F)F)c1 ZINC000217953975 DH In-Stock Anodyne DDR2 21 46 O=C(Nc1ccn2nccc2c1)c1cccc(C(F)(F)F)c1 ZINC000217953975 DH In-Stock Anodyne KCNK3 111 60 O=C(Nc1ccn2nccc2c1)c1cccc(C(F)(F)F)c1 ZINC000217953975 DH In-Stock Anodyne KCNK9 64 38 CCCOc1ccc([C@@H](N)[C@H]2CCC[C@@H](C)C2)cc1 ZINC000217953990 CI For-Sale Unstable ACACA 30 40 C[C@@H](C(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)N1Cc2ccccc2C1=O ZINC000217953991 GD In-Stock Unstable CHRNA4 36 48 COc1cccc(/C=C/NC(=O)N2CCN(c3cccc(Cl)c3)CC2)c1 ZINC000217953997 FH For-Sale Unstable DRD4 49 41 COc1cccc(/C=C/NC(=O)N2CCN(c3cccc(Cl)c3)CC2)c1 ZINC000217953997 FH For-Sale Unstable CCKAR 27 49 COc1cc([N+](=O)[O-])ccc1N[C@@H]1C[C@@H](C)N(C)C[C@@H]1C ZINC000217954007 CF For-Sale Unstable KCNMA1 21 45 CN(Cc1ccc(F)cc1/C=C\C(=O)O)C[C@@H]1CCCO1 ZINC000217954012 CF For-Sale Unstable OXTR 26 45 CN(Cc1ccc(F)cc1/C=C\C(=O)O)C[C@@H]1CCCO1 ZINC000217954012 CF For-Sale Unstable AVPR1A 0 45 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)C(C)C ZINC000217954034 DE For-Sale Unstable ACE 15 43 CC[C@@H](NC(=O)/C=C/c1ccc(C(C)(C)C)cc1)c1ccc(C)c(C)c1 ZINC000217954038 EK In-Stock Unstable HDAC1 15 40 CC(=O)NN1Cc2ccccc2C1 ZINC000217954041 AD For-Sale Unstable HSD17B3 26 46 CC(=O)NN1Cc2ccccc2C1 ZINC000217954041 AD For-Sale Unstable ADAM9 47 33 CCCOc1ccc([C@H](N)[C@H]2CCC[C@@H](C)C2)cc1 ZINC000217954060 CI For-Sale Unstable ACACA 30 40 CCc1ncnc(NCc2ccc(S(N)(=O)=O)cc2)c1F ZINC000217954068 DD On-Demand Unstable CA2 72 54 CCc1ncnc(NCc2ccc(S(N)(=O)=O)cc2)c1F ZINC000217954068 DD On-Demand Unstable CA1 59 51 CCc1ncnc(NCc2ccc(S(N)(=O)=O)cc2)c1F ZINC000217954068 DD On-Demand Unstable CA7 47 42 CCc1ncnc(NCc2ccc(S(N)(=O)=O)cc2)c1F ZINC000217954068 DD On-Demand Unstable CA13 36 53 CCc1ncnc(NCc2ccc(S(N)(=O)=O)cc2)c1F ZINC000217954068 DD On-Demand Unstable CA4 40 45 CCc1ncnc(NCc2ccc(S(N)(=O)=O)cc2)c1F ZINC000217954068 DD On-Demand Unstable CA14 29 45 CCc1ncnc(NCc2ccc(S(N)(=O)=O)cc2)c1F ZINC000217954068 DD On-Demand Unstable CA12 38 43 CCc1ncnc(NCc2ccc(S(N)(=O)=O)cc2)c1F ZINC000217954068 DD On-Demand Unstable CA9 49 51 CCc1ncnc(NCc2ccc(S(N)(=O)=O)cc2)c1F ZINC000217954068 DD On-Demand Unstable CYNT 45 39 COc1cc([N+](=O)[O-])ccc1N[C@H]1C[C@@H](C)N(C)C[C@@H]1C ZINC000217954071 CF For-Sale Unstable KCNMA1 21 45 O=C(Nc1ccn2nccc2c1)c1cccc2ccccc12 ZINC000217954080 CH In-Stock Anodyne KCNK3 67 36 O=C(Nc1ccn2nccc2c1)c1cccc2ccccc12 ZINC000217954080 CH In-Stock Anodyne KCNK9 64 37 O=C(Nc1ccn2nccc2c1)c1cccc2ccccc12 ZINC000217954080 CH In-Stock Anodyne POLR1A 43 30 COc1cccc(/C=C/NC(=O)Nc2ccc(-c3nc4ccc(C)cc4s3)cc2)c1 ZINC000217954104 HK For-Sale Unstable KIT 19 40 COc1cccc(/C=C/NC(=O)Nc2ccc(-c3nc4ccc(C)cc4s3)cc2)c1 ZINC000217954104 HK For-Sale Unstable CSNK1D 28 41 COc1cccc(/C=C/NC(=O)Nc2ccc(-c3nc4ccc(C)cc4s3)cc2)c1 ZINC000217954104 HK For-Sale Unstable PIK3CA 0 40 COc1cccc(/C=C/NC(=O)Nc2ccc(-c3nc4ccc(C)cc4s3)cc2)c1 ZINC000217954104 HK For-Sale Unstable APP 25 48 COc1cccc(/C=C/NC(=O)Nc2ccc(-c3nc4ccc(C)cc4s3)cc2)c1 ZINC000217954104 HK For-Sale Unstable KDR 16 40 COc1cccc(/C=C/NC(=O)Nc2ccc(-c3nc4ccc(C)cc4s3)cc2)c1 ZINC000217954104 HK For-Sale Unstable TEK 29 40 COc1cccc(/C=C/NC(=O)Nc2ccc(-c3nc4ccc(C)cc4s3)cc2)c1 ZINC000217954104 HK For-Sale Unstable LUCI_PHOPE 34 48 COc1cccc(/C=C/NC(=O)Nc2ccc(-c3nc4ccc(C)cc4s3)cc2)c1 ZINC000217954104 HK For-Sale Unstable ETHR 20 51 COc1cc2c(c(OC)c1OC)-c1ccc(NCCCCCC(=O)NCc3ccccc3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217954107 KK In-Stock Unstable TUBA1A 18 65 CC[C@H](NC(=O)/C=C/c1ccc(C(C)(C)C)cc1)c1ccc(C)c(C)c1 ZINC000217954114 EK In-Stock Unstable HDAC1 15 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)C(C)C ZINC000217954117 DE For-Sale Unstable ACE 15 43 CN(Cc1ccc(F)c(/C=C\C(=O)O)c1)C[C@@H]1CCCO1 ZINC000217954118 CF For-Sale Unstable OXTR 26 42 CN(Cc1ccc(F)c(/C=C\C(=O)O)c1)C[C@@H]1CCCO1 ZINC000217954118 CF For-Sale Unstable AVPR1A 0 42 COc1cc([N+](=O)[O-])ccc1N[C@@H]1C[C@H](C)N(C)C[C@@H]1C ZINC000217954145 CF For-Sale Unstable KCNMA1 21 45 COc1ccc2c(c1I)C(=O)NCC2 ZINC000217954173 DD For-Sale Unstable CSNK1G2 51 30 CCOC(=O)[C@@H]1CCCN(c2ncnc(CC)c2F)C1 ZINC000217954177 CD On-Demand Unstable SLC6A1 48 33 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)C(C)C ZINC000217954185 DE For-Sale Unstable ACE 15 43 O=C(/C=C/c1ccccc1)Nc1ccn2nccc2c1 ZINC000217954192 CF In-Stock Anodyne MMP2 24 56 O=C(/C=C/c1ccccc1)Nc1ccn2nccc2c1 ZINC000217954192 CF In-Stock Anodyne MMP9 22 51 O=C(/C=C/c1ccccc1)Nc1ccn2nccc2c1 ZINC000217954192 CF In-Stock Anodyne IMPDH2 0 44 O=C(/C=C/c1ccccc1)Nc1ccn2nccc2c1 ZINC000217954192 CF In-Stock Anodyne MMP1 26 54 O=C(/C=C/c1ccccc1)Nc1ccn2nccc2c1 ZINC000217954192 CF In-Stock Anodyne MCHR1 0 48 O=C(/C=C/c1ccccc1)Nc1ccn2nccc2c1 ZINC000217954192 CF In-Stock Anodyne HDA106 0 40 COc1cccc(/C=C/NC(=O)Nc2ccc3c(c2)OCO3)c1 ZINC000217954223 DG For-Sale Unstable EDNRB 58 40 COc1cccc(/C=C/NC(=O)Nc2ccc3c(c2)OCO3)c1 ZINC000217954223 DG For-Sale Unstable EDNRA 57 40 COc1cccc(/C=C/NC(=O)Nc2ccc3c(c2)OCO3)c1 ZINC000217954223 DG For-Sale Unstable MTNR1A 26 43 COc1cccc(/C=C/NC(=O)Nc2ccc3c(c2)OCO3)c1 ZINC000217954223 DG For-Sale Unstable MTNR1B 28 45 COc1cccc(/C=C/NC(=O)Nc2ccc3c(c2)OCO3)c1 ZINC000217954223 DG For-Sale Unstable CCR2 0 46 COc1cccc(/C=C/NC(=O)Nc2ccc3c(c2)OCO3)c1 ZINC000217954223 DG For-Sale Unstable IMPDH2 0 44 COc1cccc(/C=C/NC(=O)Nc2ccc3c(c2)OCO3)c1 ZINC000217954223 DG For-Sale Unstable DYRK2 47 38 O=C(O)/C=C\c1ccc(CN2CCCC[C@@H]2CO)cc1 ZINC000217954231 CE For-Sale Unstable SPHK1 23 42 COc1cc([N+](=O)[O-])ccc1N[C@H]1C[C@H](C)N(C)C[C@@H]1C ZINC000217954232 CF For-Sale Unstable KCNMA1 21 45 CCOC(=O)[C@H]1CCCN(c2ncnc(CC)c2F)C1 ZINC000217954251 CD On-Demand Unstable SLC6A1 48 33 Nc1cc(C(=O)N2CCC(Oc3ccccc3F)CC2)n[nH]1 ZINC000217954269 DD In-Stock Unstable GRIN2B 26 41 Nc1cc(C(=O)N2CCC(Oc3ccccc3F)CC2)n[nH]1 ZINC000217954269 DD In-Stock Unstable TACR3 18 40 Nc1cc(C(=O)N2CCC(Oc3ccccc3F)CC2)n[nH]1 ZINC000217954269 DD In-Stock Unstable SCD1 53 38 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc2ccccc12 ZINC000217954292 GH For-Sale Unstable HCRTR1 60 43 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc2ccccc12 ZINC000217954292 GH For-Sale Unstable HCRTR2 66 43 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc2ccccc12 ZINC000217954292 GH For-Sale Unstable NR1D1 40 42 O=C(COc1ccc(Cl)cc1)Nc1ccn2nccc2c1 ZINC000217954298 DG In-Stock Unstable CETP 24 48 O=C(COc1ccc(Cl)cc1)Nc1ccn2nccc2c1 ZINC000217954298 DG In-Stock Unstable MCHR1 17 49 CC[C@@H](CCO)NC(=O)CC[C@@H](C)N ZINC000217954302 BC For-Sale Unstable NOD1 79 36 COc1cccc(/C=C/NC(=O)Nc2ccccc2Br)c1 ZINC000217954319 EI For-Sale Unstable MTNR1A 27 41 COc1cccc(/C=C/NC(=O)Nc2ccccc2Br)c1 ZINC000217954319 EI For-Sale Unstable MTNR1B 30 41 CCOC(=O)[C@@H](NC(C)(C)C)c1ccccc1 ZINC000217954329 BF For-Sale Unstable CTSK 17 41 CCOC(=O)[C@@H](NC(C)(C)C)c1ccccc1 ZINC000217954329 BF For-Sale Unstable AMY2 57 36 CCOC(=O)[C@@H](NC(C)(C)C)c1ccccc1 ZINC000217954329 BF For-Sale Unstable SOAT1 31 43 CCOC(=O)[C@@H](NC(C)(C)C)c1ccccc1 ZINC000217954329 BF For-Sale Unstable CAPN2 26 40 CCc1ncnc(N[C@@H]2CCCc3ccccc32)c1F ZINC000217954359 CH On-Demand Unstable KCNN3 30 45 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc2ccccc12 ZINC000217954371 GH For-Sale Unstable HCRTR1 60 43 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc2ccccc12 ZINC000217954371 GH For-Sale Unstable HCRTR2 66 43 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc2ccccc12 ZINC000217954371 GH For-Sale Unstable NR1D1 40 42 CC[C@@H](NC(=O)/C=C/c1ccc(C(C)(C)C)cc1)c1ccc(OC)c(OC)c1 ZINC000217954391 GK In-Stock Unstable TRPV1 32 62 CC[C@H](CCO)NC(=O)CC[C@@H](C)N ZINC000217954408 BC For-Sale Unstable NOD1 79 36 CCOC(=O)[C@H](NC(C)(C)C)c1ccccc1 ZINC000217954414 BF For-Sale Unstable CTSK 17 41 CCOC(=O)[C@H](NC(C)(C)C)c1ccccc1 ZINC000217954414 BF For-Sale Unstable AMY2 57 36 CCOC(=O)[C@H](NC(C)(C)C)c1ccccc1 ZINC000217954414 BF For-Sale Unstable SOAT1 31 43 CCOC(=O)[C@H](NC(C)(C)C)c1ccccc1 ZINC000217954414 BF For-Sale Unstable CAPN2 26 40 COc1cccc(/C=C/NC(=O)Nc2cccc(F)c2)c1 ZINC000217954420 CH For-Sale Unstable AHR 15 40 COc1cccc(/C=C/NC(=O)Nc2cccc(F)c2)c1 ZINC000217954420 CH For-Sale Unstable MTNR1A 26 46 COc1cccc(/C=C/NC(=O)Nc2cccc(F)c2)c1 ZINC000217954420 CH For-Sale Unstable MTNR1B 31 46 COc1cccc(/C=C/NC(=O)Nc2cccc(F)c2)c1 ZINC000217954420 CH For-Sale Unstable PDGFRA 17 42 COc1cccc(/C=C/NC(=O)Nc2cccc(F)c2)c1 ZINC000217954420 CH For-Sale Unstable TAAR1 32 45 COc1cccc(/C=C/NC(=O)Nc2cccc(F)c2)c1 ZINC000217954420 CH For-Sale Unstable KCNK3 34 42 CCc1ncnc(N[C@H]2CCCc3ccccc32)c1F ZINC000217954451 CH On-Demand Unstable KCNN3 30 45 O=C(O)/C=C\c1cccc(CN2CCCC[C@@H]2CO)c1 ZINC000217954452 CE For-Sale Unstable SPHK1 19 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc2ccccc12 ZINC000217954458 GH For-Sale Unstable HCRTR1 60 43 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc2ccccc12 ZINC000217954458 GH For-Sale Unstable HCRTR2 66 43 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc2ccccc12 ZINC000217954458 GH For-Sale Unstable NR1D1 40 42 CC[C@H](NC(=O)/C=C/c1ccc(C(C)(C)C)cc1)c1ccc(OC)c(OC)c1 ZINC000217954474 GK In-Stock Unstable TRPV1 32 62 CC[C@@H](CCO)NC(=O)CC[C@H](C)N ZINC000217954485 BC For-Sale Unstable NOD1 79 36 COc1ccccc1OCC(=O)Nc1ccn2nccc2c1 ZINC000217954519 CE In-Stock Unstable CETP 0 47 COc1ccccc1OCC(=O)Nc1ccn2nccc2c1 ZINC000217954519 CE In-Stock Unstable ENPP1 63 38 COc1ccccc1OCC(=O)Nc1ccn2nccc2c1 ZINC000217954519 CE In-Stock Unstable KCNK3 43 37 COc1cccc(/C=C/NC(=O)NCCc2ccc(F)cc2)c1 ZINC000217954522 DG For-Sale Unstable CCR3 24 43 COc1cccc(/C=C/NC(=O)NCCc2ccc(F)cc2)c1 ZINC000217954522 DG For-Sale Unstable MTNR1A 102 46 COc1cccc(/C=C/NC(=O)NCCc2ccc(F)cc2)c1 ZINC000217954522 DG For-Sale Unstable MTNR1B 93 46 COc1cccc(/C=C/NC(=O)NCCc2ccc(F)cc2)c1 ZINC000217954522 DG For-Sale Unstable ABCG2 17 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc2ccccc12 ZINC000217954542 GH For-Sale Unstable HCRTR1 60 43 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc2ccccc12 ZINC000217954542 GH For-Sale Unstable HCRTR2 66 43 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc2ccccc12 ZINC000217954542 GH For-Sale Unstable NR1D1 40 42 CC[C@H](CCO)NC(=O)CC[C@H](C)N ZINC000217954553 BC For-Sale Unstable NOD1 79 36 COc1ccc(/C=C\C(=O)O)cc1CN(C)CCC(C)C ZINC000217954564 CG For-Sale Unstable AKR1C3 30 42 CC[C@@H](NC(=O)/C=C/c1ccc(C(C)(C)C)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217954569 GJ In-Stock Unstable CTSF 45 34 Cc1ccccc1OCC(=O)Nc1ccn2nccc2c1 ZINC000217954612 CF In-Stock Unstable CETP 0 48 COc1cccc(/C=C/NC(=O)N2CCc3ccccc32)c1 ZINC000217954613 CG For-Sale Unstable DRD4 44 36 COc1cccc(/C=C/NC(=O)N2CCc3ccccc32)c1 ZINC000217954613 CG For-Sale Unstable AVPR2 26 46 CC1(NC(=O)N2[C@H](C(=O)O)C[C@@H]3CCCC[C@@H]32)CCCC1 ZINC000217954620 CF For-Sale Unstable ACE 18 55 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1cccnc1 ZINC000217954639 FD For-Sale Unstable COLA 84 38 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1cccnc1 ZINC000217954639 FD For-Sale Unstable CPT1A 79 38 CC[C@H](NC(=O)/C=C/c1ccc(C(C)(C)C)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217954645 GJ In-Stock Unstable CTSF 45 34 COc1ccc(CN2CCC[C@H]2C)cc1/C=C\C(=O)O ZINC000217954669 CF For-Sale Unstable DRD2 42 37 COc1ccc(CN2CCC[C@H]2C)cc1/C=C\C(=O)O ZINC000217954669 CF For-Sale Unstable PTGER2 23 40 COc1ccc(CN2CCC[C@H]2C)cc1/C=C\C(=O)O ZINC000217954669 CF For-Sale Unstable PTGER4 15 40 COc1ccc(CN2CCC[C@H]2C)cc1/C=C\C(=O)O ZINC000217954669 CF For-Sale Unstable HRH3 54 42 COc1ccc(CN2CCC[C@H]2C)cc1/C=C\C(=O)O ZINC000217954669 CF For-Sale Unstable ACKR3 53 36 CC[C@@H](CCO)NC(=O)CCCNC ZINC000217954678 BC For-Sale Unstable PLA2G2C 0 43 CC[C@@H](CCO)NC(=O)CCCNC ZINC000217954678 BC For-Sale Unstable Q6UB75_PIG 0 42 CC1(NC(=O)N2[C@H](C(=O)O)C[C@H]3CCCC[C@@H]32)CCCC1 ZINC000217954697 CF For-Sale Unstable ACE 18 55 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1cccnc1 ZINC000217954712 FD For-Sale Unstable COLA 84 38 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1cccnc1 ZINC000217954712 FD For-Sale Unstable CPT1A 79 38 O=C(COc1ccc(F)cc1)Nc1ccn2nccc2c1 ZINC000217954720 CE In-Stock Unstable ADORA2A 0 42 O=C(COc1ccc(F)cc1)Nc1ccn2nccc2c1 ZINC000217954720 CE In-Stock Unstable ADORA2B 47 42 O=C(COc1ccc(F)cc1)Nc1ccn2nccc2c1 ZINC000217954720 CE In-Stock Unstable CETP 0 45 COc1cccc(/C=C/NC(=O)Nc2ccc(I)cc2)c1 ZINC000217954724 GI For-Sale Unstable MTNR1A 31 50 COc1cccc(/C=C/NC(=O)Nc2ccc(I)cc2)c1 ZINC000217954724 GI For-Sale Unstable MTNR1B 37 50 COc1cccc(/C=C/NC(=O)Nc2ccc(I)cc2)c1 ZINC000217954724 GI For-Sale Unstable Q8MMZ8_EIMTE 0 44 Cc1nc(N2CC[C@H](N3CCCC3)C2)sc1[C@H](C)O ZINC000217954740 CE For-Sale Unstable HRH3 25 42 COc1ccc(CN2CCC[C@@H]2C)cc1/C=C\C(=O)O ZINC000217954749 CF For-Sale Unstable DRD2 42 37 COc1ccc(CN2CCC[C@@H]2C)cc1/C=C\C(=O)O ZINC000217954749 CF For-Sale Unstable PTGER2 23 40 COc1ccc(CN2CCC[C@@H]2C)cc1/C=C\C(=O)O ZINC000217954749 CF For-Sale Unstable PTGER4 0 40 COc1ccc(CN2CCC[C@@H]2C)cc1/C=C\C(=O)O ZINC000217954749 CF For-Sale Unstable HRH3 54 42 COc1ccc(CN2CCC[C@@H]2C)cc1/C=C\C(=O)O ZINC000217954749 CF For-Sale Unstable ACKR3 53 36 CC(C)(C)c1ccc(/C=C/C(=O)NCc2nc(-c3ccccc3)no2)cc1 ZINC000217954756 FI In-Stock Unstable HDAC8 53 38 CC(C)(C)c1ccc(/C=C/C(=O)NCc2nc(-c3ccccc3)no2)cc1 ZINC000217954756 FI In-Stock Unstable HDAC1 22 42 CC(C)(C)c1ccc(/C=C/C(=O)NCc2nc(-c3ccccc3)no2)cc1 ZINC000217954756 FI In-Stock Unstable HDAC2 17 42 CC(C)(C)c1ccc(/C=C/C(=O)NCc2nc(-c3ccccc3)no2)cc1 ZINC000217954756 FI In-Stock Unstable HDAC6 43 36 CC[C@H](CCO)NC(=O)CCCNC ZINC000217954760 BC For-Sale Unstable PLA2G2C 0 43 CC[C@H](CCO)NC(=O)CCCNC ZINC000217954760 BC For-Sale Unstable Q6UB75_PIG 0 42 Cc1[nH]c2ccccc2c1/C=C\C(=O)CCl ZINC000217954785 BG For-Sale Unstable TSPO 16 43 CCCCCCN[C@@H](C(=O)OCC)c1ccccc1 ZINC000217954793 CG On-Demand Unstable PLA2G4B 44 31 CCCCCCN[C@@H](C(=O)OCC)c1ccccc1 ZINC000217954793 CG On-Demand Unstable SOAT1 63 45 CCCCCCN[C@@H](C(=O)OCC)c1ccccc1 ZINC000217954793 CG On-Demand Unstable FAAH 24 44 CCCCCCN[C@@H](C(=O)OCC)c1ccccc1 ZINC000217954793 CG On-Demand Unstable S1PR2 43 34 CCCCCCN[C@@H](C(=O)OCC)c1ccccc1 ZINC000217954793 CG On-Demand Unstable EST1_RABIT 0 44 CCCCCCN[C@@H](C(=O)OCC)c1ccccc1 ZINC000217954793 CG On-Demand Unstable ASAH1 83 44 CCCCCCN[C@@H](C(=O)OCC)c1ccccc1 ZINC000217954793 CG On-Demand Unstable ACAT 0 43 CCCCCCN[C@@H](C(=O)OCC)c1ccccc1 ZINC000217954793 CG On-Demand Unstable ACER2 0 44 CCCCCCN[C@@H](C(=O)OCC)c1ccccc1 ZINC000217954793 CG On-Demand Unstable COL4A3BP 0 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1cccnc1 ZINC000217954799 FD For-Sale Unstable COLA 84 38 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1cccnc1 ZINC000217954799 FD For-Sale Unstable CPT1A 79 38 O[C@H]1CCCc2nc(N3CC[C@H](N4CCCC4)C3)sc21 ZINC000217954819 CE For-Sale Unstable HRH3 22 44 COc1cccc(/C=C/NC(=O)NCCc2c[nH]c3ccccc23)c1 ZINC000217954841 EH For-Sale Unstable HTR1D 15 43 COc1cccc(/C=C/NC(=O)NCCc2c[nH]c3ccccc23)c1 ZINC000217954841 EH For-Sale Unstable HTR1B 15 43 COc1cccc(/C=C/NC(=O)NCCc2c[nH]c3ccccc23)c1 ZINC000217954841 EH For-Sale Unstable TACR1 36 43 COc1cccc(/C=C/NC(=O)NCCc2c[nH]c3ccccc23)c1 ZINC000217954841 EH For-Sale Unstable MC4R 34 42 COc1cccc(/C=C/NC(=O)NCCc2c[nH]c3ccccc23)c1 ZINC000217954841 EH For-Sale Unstable NQO2 44 55 COc1cccc(/C=C/NC(=O)NCCc2c[nH]c3ccccc23)c1 ZINC000217954841 EH For-Sale Unstable CCKAR 52 42 COc1cccc(/C=C/NC(=O)NCCc2c[nH]c3ccccc23)c1 ZINC000217954841 EH For-Sale Unstable NMBR 33 44 COc1cccc(/C=C/NC(=O)NCCc2c[nH]c3ccccc23)c1 ZINC000217954841 EH For-Sale Unstable MTNR1A 121 59 COc1cccc(/C=C/NC(=O)NCCc2c[nH]c3ccccc23)c1 ZINC000217954841 EH For-Sale Unstable MTNR1B 102 55 COc1cccc(/C=C/NC(=O)NCCc2c[nH]c3ccccc23)c1 ZINC000217954841 EH For-Sale Unstable MMP14 42 34 COc1cccc(/C=C/NC(=O)NCCc2c[nH]c3ccccc23)c1 ZINC000217954841 EH For-Sale Unstable CCKBR 47 44 COc1cccc(/C=C/NC(=O)NCCc2c[nH]c3ccccc23)c1 ZINC000217954841 EH For-Sale Unstable GHSR 43 42 COc1cccc(/C=C/NC(=O)NCCc2c[nH]c3ccccc23)c1 ZINC000217954841 EH For-Sale Unstable MMP9 15 48 Cc1cccc(-c2noc(CNC(=O)/C=C/c3ccc(C(C)(C)C)cc3)n2)c1 ZINC000217954855 GJ In-Stock Unstable HDAC8 53 35 Cc1cccc(-c2noc(CNC(=O)/C=C/c3ccc(C(C)(C)C)cc3)n2)c1 ZINC000217954855 GJ In-Stock Unstable HDAC6 40 34 C[C@@H]1CCCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217954860 CF For-Sale Unstable ESR1 44 40 C[C@@H]1CCCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217954860 CF For-Sale Unstable HRH2 40 37 C[C@@H]1CCCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217954860 CF For-Sale Unstable SLC6A1 139 38 C[C@@H]1CCCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217954860 CF For-Sale Unstable ESR2 33 41 C[C@@H]1CCCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217954860 CF For-Sale Unstable LTA4H 33 42 C[C@@H]1CCCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217954860 CF For-Sale Unstable HRH3 36 53 C[C@@H]1CCCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217954860 CF For-Sale Unstable CHRNA10 46 34 C[C@@H]1CCCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217954860 CF For-Sale Unstable PSMB1 40 38 C[C@@H]1CCCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217954860 CF For-Sale Unstable ACKR3 50 34 O=C(/C=C\c1c[nH]c2ccccc12)CCl ZINC000217954868 BF For-Sale Unstable TDO2 0 47 O=C(/C=C\c1c[nH]c2ccccc12)CCl ZINC000217954868 BF For-Sale Unstable CCR2 29 41 CCCCCCN[C@H](C(=O)OCC)c1ccccc1 ZINC000217954870 CG On-Demand Unstable PLA2G4B 44 31 CCCCCCN[C@H](C(=O)OCC)c1ccccc1 ZINC000217954870 CG On-Demand Unstable SOAT1 63 45 CCCCCCN[C@H](C(=O)OCC)c1ccccc1 ZINC000217954870 CG On-Demand Unstable FAAH 24 44 CCCCCCN[C@H](C(=O)OCC)c1ccccc1 ZINC000217954870 CG On-Demand Unstable S1PR2 43 34 CCCCCCN[C@H](C(=O)OCC)c1ccccc1 ZINC000217954870 CG On-Demand Unstable EST1_RABIT 0 44 CCCCCCN[C@H](C(=O)OCC)c1ccccc1 ZINC000217954870 CG On-Demand Unstable ASAH1 83 44 CCCCCCN[C@H](C(=O)OCC)c1ccccc1 ZINC000217954870 CG On-Demand Unstable ACAT 0 43 CCCCCCN[C@H](C(=O)OCC)c1ccccc1 ZINC000217954870 CG On-Demand Unstable ACER2 0 44 CCCCCCN[C@H](C(=O)OCC)c1ccccc1 ZINC000217954870 CG On-Demand Unstable COL4A3BP 0 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1cccnc1 ZINC000217954883 FD For-Sale Unstable COLA 84 38 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1cccnc1 ZINC000217954883 FD For-Sale Unstable CPT1A 79 38 Cc1nc(N2CC[C@H](N3CCCCC3)C2)sc1[C@H](C)O ZINC000217954900 CF For-Sale Unstable HRH3 27 44 CC[C@H](C(=O)Nc1ccn2nccc2c1)c1ccccc1 ZINC000217954936 CG In-Stock Unstable KCNQ2 52 50 COc1cccc(/C=C/NC(=O)N2CCC(C(N)=O)CC2)c1 ZINC000217954947 DD For-Sale Unstable MTNR1A 26 41 COc1cccc(/C=C/NC(=O)N2CCC(C(N)=O)CC2)c1 ZINC000217954947 DD For-Sale Unstable MTNR1B 34 41 CSCC[C@H](NC(=O)c1cn(Cc2ccccc2)c2ccccc12)C(=O)O ZINC000217954948 GH In-Stock Unstable ACE 27 48 CSCC[C@H](NC(=O)c1cn(Cc2ccccc2)c2ccccc12)C(=O)O ZINC000217954948 GH In-Stock Unstable CNR1 28 51 CSCC[C@H](NC(=O)c1cn(Cc2ccccc2)c2ccccc12)C(=O)O ZINC000217954948 GH In-Stock Unstable MME 40 48 CSCC[C@H](NC(=O)c1cn(Cc2ccccc2)c2ccccc12)C(=O)O ZINC000217954948 GH In-Stock Unstable ANPEP 26 40 CSCC[C@H](NC(=O)c1cn(Cc2ccccc2)c2ccccc12)C(=O)O ZINC000217954948 GH In-Stock Unstable CNR2 27 51 CSCC[C@H](NC(=O)c1cn(Cc2ccccc2)c2ccccc12)C(=O)O ZINC000217954948 GH In-Stock Unstable CCKAR 32 51 CSCC[C@H](NC(=O)c1cn(Cc2ccccc2)c2ccccc12)C(=O)O ZINC000217954948 GH In-Stock Unstable FPR1 42 42 C[C@H]1CCCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217954949 CF For-Sale Unstable ESR1 44 40 C[C@H]1CCCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217954949 CF For-Sale Unstable HRH2 40 37 C[C@H]1CCCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217954949 CF For-Sale Unstable SLC6A1 139 38 C[C@H]1CCCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217954949 CF For-Sale Unstable ESR2 33 41 C[C@H]1CCCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217954949 CF For-Sale Unstable LTA4H 33 42 C[C@H]1CCCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217954949 CF For-Sale Unstable HRH3 36 53 C[C@H]1CCCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217954949 CF For-Sale Unstable CHRNA10 46 34 C[C@H]1CCCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217954949 CF For-Sale Unstable PSMB1 40 38 C[C@H]1CCCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217954949 CF For-Sale Unstable ACKR3 50 34 Cc1ccc(-c2noc(CNC(=O)/C=C/c3ccc(C(C)(C)C)cc3)n2)cc1 ZINC000217954952 GJ In-Stock Unstable HDAC8 0 51 O[C@H]1CCCc2nc(N3CC[C@H](N4CCCCC4)C3)sc21 ZINC000217954970 DF For-Sale Unstable HRH3 24 46 CCOC(CNC(=O)c1cccc(OC)c1[N+](=O)[O-])OCC ZINC000217955017 DD For-Sale Unstable HCN1 43 32 CCOC(CNC(=O)c1cccc(OC)c1[N+](=O)[O-])OCC ZINC000217955017 DD For-Sale Unstable KCNK3 44 39 CC[C@@H](C(=O)Nc1ccn2nccc2c1)c1ccccc1 ZINC000217955019 CG In-Stock Unstable KCNQ2 52 50 CC[C@@H](C(=O)Nc1ccn2nccc2c1)c1ccccc1 ZINC000217955019 CG In-Stock Unstable KCNQ4 0 45 O=C(/C=C\c1c[nH]c2ncccc12)CCl ZINC000217955023 BE For-Sale Unstable CDC7 53 46 CCOC(=O)[C@@H](NC(C)(C)CO)c1ccccc1 ZINC000217955032 CD On-Demand Unstable SOAT1 19 40 O=C(O)[C@@H]1C[C@@H]2CCCC[C@@H]2N1C(=O)NCc1ccco1 ZINC000217955048 CE On-Demand Unstable ACE 18 50 COc1cccc(/C=C/NC(=O)NC(=O)C2CCNCC2)c1 ZINC000217955058 DD For-Sale Unstable MTNR1A 33 44 COc1cccc(/C=C/NC(=O)NC(=O)C2CCNCC2)c1 ZINC000217955058 DD For-Sale Unstable MTNR1B 36 44 COc1cccc(-c2noc(CNC(=O)/C=C/c3ccc(C(C)(C)C)cc3)n2)c1 ZINC000217955060 GI In-Stock Unstable HDAC8 41 39 C[C@@H]1CCCN(CCOc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217955069 CF On-Demand Unstable ESR1 80 42 C[C@@H]1CCCN(CCOc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217955069 CF On-Demand Unstable SLC6A1 128 38 C[C@@H]1CCCN(CCOc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217955069 CF On-Demand Unstable ESR2 53 42 C[C@@H]1CCCN(CCOc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217955069 CF On-Demand Unstable LTA4H 58 42 C[C@@H]1CCCN(CCOc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217955069 CF On-Demand Unstable HRH3 63 52 C[C@@H]1CCCN(CCOc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217955069 CF On-Demand Unstable EBP 19 43 C[C@@H]1CCCN(CCOc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217955069 CF On-Demand Unstable PSMB2 43 41 C[C@@H]1CCCN(CCOc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217955069 CF On-Demand Unstable PSMB1 47 41 CCC[C@H](NC(=O)NCc1ccc(F)cc1)C(=O)N[C@@H]1CCC[C@@H](C)[C@@H]1C ZINC000217955082 GH On-Demand Unstable ANPEP 15 47 COc1ccc(C)cc1/C=C\C(=O)CCl ZINC000217955108 BF For-Sale Unstable TNFRSF1A 27 42 COc1ccc(C)cc1/C=C\C(=O)CCl ZINC000217955108 BF For-Sale Unstable ABCG2 19 47 COc1ccc(C)cc1/C=C\C(=O)CCl ZINC000217955108 BF For-Sale Unstable CYSP_PLAFA 53 42 CCOC(=O)[C@H](NC(C)(C)CO)c1ccccc1 ZINC000217955109 CD On-Demand Unstable SOAT1 19 40 O=C(O)[C@@H]1C[C@H]2CCCC[C@@H]2N1C(=O)NCc1ccco1 ZINC000217955127 CE On-Demand Unstable ACE 18 50 O=C(Cc1cccs1)Nc1ccn2nccc2c1 ZINC000217955141 CF In-Stock Unstable CA5B 44 49 O=C(Cc1cccs1)Nc1ccn2nccc2c1 ZINC000217955141 CF In-Stock Unstable CA5A 45 49 C[C@H]1CCCN(CCOc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217955164 CF On-Demand Unstable ESR1 80 42 C[C@H]1CCCN(CCOc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217955164 CF On-Demand Unstable SLC6A1 128 38 C[C@H]1CCCN(CCOc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217955164 CF On-Demand Unstable ESR2 53 42 C[C@H]1CCCN(CCOc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217955164 CF On-Demand Unstable LTA4H 58 42 C[C@H]1CCCN(CCOc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217955164 CF On-Demand Unstable HRH3 63 52 C[C@H]1CCCN(CCOc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217955164 CF On-Demand Unstable EBP 19 43 C[C@H]1CCCN(CCOc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217955164 CF On-Demand Unstable PSMB2 43 41 C[C@H]1CCCN(CCOc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217955164 CF On-Demand Unstable PSMB1 47 41 O=C([C@@H]1CC[C@@H](Cn2cnnn2)CC1)N1CCC(Cc2ccccc2)CC1 ZINC000217955172 FF In-Stock Unstable GRIN2B 44 42 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccc(C(C)(C)C)cc3)n2)c(OC)c1 ZINC000217955186 HI In-Stock Unstable TRPV1 0 45 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccc(C(C)(C)C)cc3)n2)c(OC)c1 ZINC000217955186 HI In-Stock Unstable MT-ND1 23 43 COc1cc(C)c(/C=C\C(=O)CCl)cc1OC ZINC000217955197 CF For-Sale Unstable CYSP_PLAFA 47 33 COc1ccc2c(c1N)C(=O)NCC2 ZINC000217955231 AC For-Sale Unstable CSNK1G2 51 30 COc1ccc(/C=C\C(=O)O)cc1CN(CC#N)CC#N ZINC000217955243 CD For-Sale Unstable PTGER2 0 44 COc1ccc(/C=C\C(=O)O)cc1CN(CC#N)CC#N ZINC000217955243 CD For-Sale Unstable TUBB1 42 38 COc1ccc(/C=C\C(=O)O)cc1CN(CC#N)CC#N ZINC000217955243 CD For-Sale Unstable AKR1C3 23 42 COc1ccc(/C=C\C(=O)O)cc1CN(CC#N)CC#N ZINC000217955243 CD For-Sale Unstable ABCG2 15 40 O=C(CCc1ccccc1)Nc1ccn2nccc2c1 ZINC000217955259 CF In-Stock Unstable CES1 40 33 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cc2C(F)(F)F)c1 ZINC000217955272 FK For-Sale Unstable AHR 15 45 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cc2C(F)(F)F)c1 ZINC000217955272 FK For-Sale Unstable TAAR1 15 43 COc1ccc(/C=C\C(=O)CCl)c(Br)c1 ZINC000217955352 CG For-Sale Unstable CYP1B1 49 41 COc1ccc(/C=C\C(=O)CCl)c(Br)c1 ZINC000217955352 CG For-Sale Unstable CYP1A1 38 41 COc1ccc(/C=C\C(=O)CCl)c(Br)c1 ZINC000217955352 CG For-Sale Unstable CYP1A2 18 41 COc1ccc(/C=C\C(=O)CCl)c(Br)c1 ZINC000217955352 CG For-Sale Unstable ABCG2 15 44 COc1ccc(/C=C\C(=O)CCl)c(Br)c1 ZINC000217955352 CG For-Sale Unstable CYSP_PLAFA 44 43 CN(C)S(=O)(=O)c1ccc(C(=O)Nc2ccn3nccc3c2)cc1 ZINC000217955364 ED In-Stock Unstable KCNK3 62 38 CC(C)(C)c1ccc(/C=C/C(=O)NCc2nc(-c3ccc(Cl)cc3)no2)cc1 ZINC000217955405 GK In-Stock Unstable HDAC8 0 51 CC(C)(C)c1ccc(/C=C/C(=O)NCc2nc(-c3ccc(Cl)cc3)no2)cc1 ZINC000217955405 GK In-Stock Unstable HDAC2 15 43 COc1cc(CCC(=O)N2CCCC[C@H]2c2cccnc2)on1 ZINC000217955420 DF In-Stock Unstable CHRNA2 40 41 COc1cc(CCC(=O)N2CCCC[C@H]2c2cccnc2)on1 ZINC000217955420 DF In-Stock Unstable CPT1A 111 40 COc1cc(CCC(=O)N2CCCC[C@H]2c2cccnc2)on1 ZINC000217955420 DF In-Stock Unstable GPBAR1 0 47 COc1cc(CCC(=O)N2CCCC[C@H]2c2cccnc2)on1 ZINC000217955420 DF In-Stock Unstable CRTY 0 41 CCOC(=O)[C@@H](NC(C)(C)CC)c1ccccc1 ZINC000217955442 BG For-Sale Unstable AMY2 58 35 CCOC(=O)[C@@H](NC(C)(C)CC)c1ccccc1 ZINC000217955442 BG For-Sale Unstable SOAT1 21 41 COc1cc(Cl)c2c(c1Cl)C(=O)NCC2 ZINC000217955443 BE For-Sale Unstable CSNK1G2 51 30 O=C(Nc1ccn2nccc2c1)c1ccco1 ZINC000217955467 BE In-Stock Anodyne KISS1R 48 32 O=C(Nc1ccn2nccc2c1)c1ccco1 ZINC000217955467 BE In-Stock Anodyne KCNK3 19 48 CN1CCC(N(C)Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217955477 CE For-Sale Unstable HDAC8 39 40 CN1CCC(N(C)Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217955477 CE For-Sale Unstable HDAC1 17 40 CN1CCC(N(C)Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217955477 CE For-Sale Unstable HDAC6 31 40 COc1cccc(/C=C/NC(=O)Nc2cc(OC)c(Cl)cc2OC)c1 ZINC000217955504 FI For-Sale Unstable CYP1B1 23 42 COc1cccc(/C=C/NC(=O)Nc2cc(OC)c(Cl)cc2OC)c1 ZINC000217955504 FI For-Sale Unstable CYP1A1 19 42 CCOC(=O)[C@H](NC(C)(C)CC)c1ccccc1 ZINC000217955523 BG For-Sale Unstable AMY2 58 35 CCOC(=O)[C@H](NC(C)(C)CC)c1ccccc1 ZINC000217955523 BG For-Sale Unstable SOAT1 21 41 COc1ccc(N2C(=O)N[C@@H](CC(=O)N3CCc4cc(OC)c(OC)cc4C3)C2=O)cc1 ZINC000217955525 IE In-Stock Unstable ABCB1B 52 33 COc1ccc(N2C(=O)N[C@@H](CC(=O)N3CCc4cc(OC)c(OC)cc4C3)C2=O)cc1 ZINC000217955525 IE In-Stock Unstable ABCB1 23 56 COc1ccc(N2C(=O)N[C@@H](CC(=O)N3CCc4cc(OC)c(OC)cc4C3)C2=O)cc1 ZINC000217955525 IE In-Stock Unstable HCRTR2 15 42 Cc1c(F)cc(Br)c(O)c1C(=O)O ZINC000217955539 BE For-Sale Unstable AKR1C2 22 40 Cc1c(F)cc(Br)c(O)c1C(=O)O ZINC000217955539 BE For-Sale Unstable AKR1C1 24 40 CCN(Cc1ccccc1/C=C\C(=O)O)C1CCCCC1 ZINC000217955595 CH For-Sale Unstable PTGER2 43 47 CCN(Cc1ccccc1/C=C\C(=O)O)C1CCCCC1 ZINC000217955595 CH For-Sale Unstable PTGER4 0 47 CCN(Cc1ccccc1/C=C\C(=O)O)C1CCCCC1 ZINC000217955595 CH For-Sale Unstable PTGER3 16 47 CCN(Cc1ccccc1/C=C\C(=O)O)C1CCCCC1 ZINC000217955595 CH For-Sale Unstable PTGDR 0 45 COc1cccc(/C=C/NC(=O)Nc2c(Cl)cccc2Cl)c1 ZINC000217955603 EJ For-Sale Unstable CYP1B1 17 40 COc1cccc(/C=C/NC(=O)Nc2c(Cl)cccc2Cl)c1 ZINC000217955603 EJ For-Sale Unstable AHR 15 48 COc1cccc(/C=C/NC(=O)Nc2c(Cl)cccc2Cl)c1 ZINC000217955603 EJ For-Sale Unstable MTNR1A 30 42 COc1cccc(/C=C/NC(=O)Nc2c(Cl)cccc2Cl)c1 ZINC000217955603 EJ For-Sale Unstable MTNR1B 32 42 COc1cccc(/C=C/NC(=O)Nc2c(Cl)cccc2Cl)c1 ZINC000217955603 EJ For-Sale Unstable TAAR1 17 41 Cc1cccc(-c2noc(CN(C)C(=O)/C=C/c3ccc(C(C)(C)C)cc3)n2)c1 ZINC000217955625 GK In-Stock Unstable FABI 43 33 CCOC(=O)[C@@H](c1ccccc1)N1CCCC[C@@H]1C ZINC000217955677 CG For-Sale Unstable CHRM1 33 46 CCOC(=O)[C@@H](c1ccccc1)N1CCCC[C@@H]1C ZINC000217955677 CG For-Sale Unstable ACE 29 41 CCOC(=O)[C@@H](c1ccccc1)N1CCCC[C@@H]1C ZINC000217955677 CG For-Sale Unstable FKBP1A 44 40 CCOC(=O)[C@@H](c1ccccc1)N1CCCC[C@@H]1C ZINC000217955677 CG For-Sale Unstable SLC6A1 59 40 CCOC(=O)[C@@H](c1ccccc1)N1CCCC[C@@H]1C ZINC000217955677 CG For-Sale Unstable OPRM1 0 40 CCOC(=O)[C@@H](c1ccccc1)N1CCCC[C@@H]1C ZINC000217955677 CG For-Sale Unstable SLC6A3 26 51 CCOC(=O)[C@@H](c1ccccc1)N1CCCC[C@@H]1C ZINC000217955677 CG For-Sale Unstable CHRM3 33 46 CCOC(=O)[C@@H](c1ccccc1)N1CCCC[C@@H]1C ZINC000217955677 CG For-Sale Unstable KCNQ2 50 39 CCOC(=O)[C@@H](c1ccccc1)N1CCCC[C@@H]1C ZINC000217955677 CG For-Sale Unstable CCR5 43 39 CCOC(=O)[C@@H](c1ccccc1)N1CCCC[C@@H]1C ZINC000217955677 CG For-Sale Unstable AMY2 48 34 CCOC(=O)[C@@H](c1ccccc1)N1CCCC[C@@H]1C ZINC000217955677 CG For-Sale Unstable FKBP12.6 0 40 CCOC(=O)[C@@H](c1ccccc1)N1CCCC[C@@H]1C ZINC000217955677 CG For-Sale Unstable XIAP 42 38 Cc1noc2nc(C(C)C)cc(C(=O)Nc3ccc(S(=O)(=O)N4CCC[C@@H](C)C4)cc3)c12 ZINC000217955679 JI On-Demand Unstable NAMPT 19 44 COc1cccc(/C=C/NC(=O)N2CCN(c3cccc(C)c3C)CC2)c1 ZINC000217955737 FH For-Sale Unstable DRD4 46 37 COc1cccc(/C=C/NC(=O)N2CCN(c3cccc(C)c3C)CC2)c1 ZINC000217955737 FH For-Sale Unstable ABCB1 0 43 Cc1noc2nc(C(C)C)cc(C(=O)Nc3ccc(S(=O)(=O)N4CCC[C@H](C)C4)cc3)c12 ZINC000217955761 JI On-Demand Unstable NAMPT 19 44 CCOC(=O)[C@H](c1ccccc1)N1CCCC[C@@H]1C ZINC000217955762 CG For-Sale Unstable CHRM1 33 46 CCOC(=O)[C@H](c1ccccc1)N1CCCC[C@@H]1C ZINC000217955762 CG For-Sale Unstable ACE 29 41 CCOC(=O)[C@H](c1ccccc1)N1CCCC[C@@H]1C ZINC000217955762 CG For-Sale Unstable FKBP1A 44 40 CCOC(=O)[C@H](c1ccccc1)N1CCCC[C@@H]1C ZINC000217955762 CG For-Sale Unstable SLC6A1 59 40 CCOC(=O)[C@H](c1ccccc1)N1CCCC[C@@H]1C ZINC000217955762 CG For-Sale Unstable OPRM1 0 40 CCOC(=O)[C@H](c1ccccc1)N1CCCC[C@@H]1C ZINC000217955762 CG For-Sale Unstable SLC6A3 26 51 CCOC(=O)[C@H](c1ccccc1)N1CCCC[C@@H]1C ZINC000217955762 CG For-Sale Unstable CHRM3 33 46 CCOC(=O)[C@H](c1ccccc1)N1CCCC[C@@H]1C ZINC000217955762 CG For-Sale Unstable KCNQ2 50 39 CCOC(=O)[C@H](c1ccccc1)N1CCCC[C@@H]1C ZINC000217955762 CG For-Sale Unstable CCR5 43 39 CCOC(=O)[C@H](c1ccccc1)N1CCCC[C@@H]1C ZINC000217955762 CG For-Sale Unstable AMY2 48 34 CCOC(=O)[C@H](c1ccccc1)N1CCCC[C@@H]1C ZINC000217955762 CG For-Sale Unstable FKBP12.6 0 40 CCOC(=O)[C@H](c1ccccc1)N1CCCC[C@@H]1C ZINC000217955762 CG For-Sale Unstable XIAP 42 38 COc1cc(CCCN)c(Br)cc1C ZINC000217955765 CF For-Sale Unstable HTR2C 15 51 COc1ccc(CCC(=O)Nc2ccn3nccc3c2)cc1 ZINC000217955796 CF In-Stock Unstable PANK1 0 41 COc1ccc(CCC(=O)Nc2ccn3nccc3c2)cc1 ZINC000217955796 CF In-Stock Unstable PANK3 0 40 COc1cccc(/C=C/NC(=O)N2CCN(c3ccccc3)CC2)c1 ZINC000217955842 EG For-Sale Unstable HTR1A 18 48 COc1cccc(/C=C/NC(=O)N2CCN(c3ccccc3)CC2)c1 ZINC000217955842 EG For-Sale Unstable DRD4 49 39 COc1cccc(/C=C/NC(=O)N2CCN(c3ccccc3)CC2)c1 ZINC000217955842 EG For-Sale Unstable DRD3 15 48 COc1cccc(/C=C/NC(=O)N2CCN(c3ccccc3)CC2)c1 ZINC000217955842 EG For-Sale Unstable PDGFRB 24 41 COc1cccc(/C=C/NC(=O)N2CCN(c3ccccc3)CC2)c1 ZINC000217955842 EG For-Sale Unstable HTR7 15 41 COc1cccc(/C=C/NC(=O)N2CCN(c3ccccc3)CC2)c1 ZINC000217955842 EG For-Sale Unstable MMP2 0 41 Cc1cc(C(=O)N[C@@H](C)Cc2cccnc2)cc(=O)[nH]1 ZINC000217955917 CD In-Stock Unstable PTAFR 28 41 CC[C@@H](C#N)N1CCN(C(=O)c2cnccn2)CC1 ZINC000217955921 CC For-Sale Unstable PTAFR 33 41 CCN(CC)c1ccc(NC(=O)N/C=C/c2cccc(OC)c2)c(C)c1 ZINC000217955950 FJ For-Sale Unstable MTNR1A 23 43 CCN(CC)c1ccc(NC(=O)N/C=C/c2cccc(OC)c2)c(C)c1 ZINC000217955950 FJ For-Sale Unstable MTNR1B 25 43 CC[C@H](C#N)N1CCN(C(=O)c2cnccn2)CC1 ZINC000217955989 CC For-Sale Unstable PTAFR 33 41 Cc1cc(C(=O)N[C@H](C)Cc2cccnc2)cc(=O)[nH]1 ZINC000217955996 CD In-Stock Unstable PTAFR 28 41 O=C(CSc1ccc(F)cc1)Nc1ccn2nccc2c1 ZINC000217956011 DG In-Stock Unstable ENPP1 51 32 O=C(CSc1ccc(F)cc1)Nc1ccn2nccc2c1 ZINC000217956011 DG In-Stock Unstable FAS 60 33 CN(C)Cc1ccc(C(=O)N[C@@H]2CCC[C@@H]2CO)cc1 ZINC000217956032 CD On-Demand Unstable SSTR3 31 45 CN(Cc1nc(-c2ccccc2Cl)no1)C(=O)/C=C/c1ccc(C(C)(C)C)cc1 ZINC000217956042 HK In-Stock Unstable FABI 40 31 COc1cccc(/C=C/NC(=O)Nc2c(C)cccc2C)c1 ZINC000217956044 CI For-Sale Unstable CYP1B1 24 41 COc1cccc(/C=C/NC(=O)Nc2c(C)cccc2C)c1 ZINC000217956044 CI For-Sale Unstable MTNR1A 31 43 COc1cccc(/C=C/NC(=O)Nc2c(C)cccc2C)c1 ZINC000217956044 CI For-Sale Unstable MTNR1B 34 43 COc1cccc(/C=C/NC(=O)Nc2c(C)cccc2C)c1 ZINC000217956044 CI For-Sale Unstable CYP1A1 18 41 CCOc1ccc(C)cc1/C=C\c1csc(N)n1 ZINC000217956092 CH For-Sale Unstable FOLA 15 40 COc1cc(CCCN)c(C)cc1Br ZINC000217956107 CF For-Sale Unstable HTR2A 15 60 COc1cc(CCCN)c(C)cc1Br ZINC000217956107 CF For-Sale Unstable HTR2C 16 60 COc1cccc(/C=C/NC(=O)Nc2cc([N+](=O)[O-])ccc2OC)c1 ZINC000217956140 EG For-Sale Unstable KCNMA1 22 51 COc1cccc(/C=C/NC(=O)Nc2cc([N+](=O)[O-])ccc2OC)c1 ZINC000217956140 EG For-Sale Unstable TAAR1 21 44 COc1cccc(/C=C/NC(=O)Nc2cc([N+](=O)[O-])ccc2OC)c1 ZINC000217956140 EG For-Sale Unstable ABCG2 18 40 COc1cccc(/C=C/NC(=O)Nc2cc([N+](=O)[O-])ccc2OC)c1 ZINC000217956140 EG For-Sale Unstable TRPM8 0 52 COc1cccc(/C=C/NC(=O)Nc2cc([N+](=O)[O-])ccc2OC)c1 ZINC000217956140 EG For-Sale Unstable AKR1C2 23 42 O=C1C/C(=C/c2cccc(C(F)(F)F)c2)C(=O)N1 ZINC000217956158 CE For-Sale Unstable PRKCA 28 46 CCOC(=O)c1c(Cl)ccc(Cl)c1C ZINC000217956193 BG For-Sale Unstable PRKCZ 28 40 CCOC(=O)c1c(Cl)ccc(Cl)c1C ZINC000217956193 BG For-Sale Unstable Q9FYV8_MAIZE 17 40 O=C(Nc1ccn(Cc2ccncc2)n1)c1ccccc1 ZINC000217956203 CF On-Demand Unstable KCNK3 51 47 Cc1ccc2[nH]c(C(=O)N3CCCn4nc([C@@H](O)CO)cc4C3)nc2c1 ZINC000217956240 FD In-Stock Unstable GRIN2B 22 41 COc1ccc(/C=C2/CC(=O)NC2=O)cc1OC(F)F ZINC000217956247 CD For-Sale Unstable ESRRA 54 40 COc1ccc(/C=C2/CC(=O)NC2=O)cc1OC(F)F ZINC000217956247 CD For-Sale Unstable HPGD 43 38 CC[C@H](C)[C@@H](NC(=O)N[C@H](C)CC)C(=O)O ZINC000217956249 BD For-Sale Unstable ENPEP 65 41 CC[C@H](C)[C@@H](NC(=O)N[C@H](C)CC)C(=O)O ZINC000217956249 BD For-Sale Unstable ACE2 25 41 O=C(Nc1ccn2nccc2c1)c1ccsc1 ZINC000217956315 BF In-Stock Anodyne KCNK3 53 54 Cc1ccc2[nH]c(C(=O)N3CCCn4nc([C@H](O)CO)cc4C3)nc2c1 ZINC000217956333 FD In-Stock Unstable GRIN2B 22 41 O=C(O)COc1c(F)cccc1Br ZINC000217956348 BE For-Sale Unstable PTPN1 20 42 O=C1CC[C@@H](C(=O)N[C@@H]2CCC[C@@H]2CO)N1 ZINC000217956361 BB For-Sale Unstable TRHR 40 36 O=C(Nc1ccn2nccc2c1)c1ccc(Oc2ccccc2)cc1 ZINC000217956420 EI In-Stock Anodyne FABH 0 41 CCN(C(=O)N/C=C/c1cccc(OC)c1)c1cccc(C)c1 ZINC000217956425 DI For-Sale Unstable MTNR1A 30 43 CCN(C(=O)N/C=C/c1cccc(OC)c1)c1cccc(C)c1 ZINC000217956425 DI For-Sale Unstable MTNR1B 33 43 CCN(C(=O)N/C=C/c1cccc(OC)c1)c1cccc(C)c1 ZINC000217956425 DI For-Sale Unstable NR1H4 51 41 O=C1CC[C@@H](C(=O)N[C@H]2CCC[C@@H]2CO)N1 ZINC000217956446 BB For-Sale Unstable TRHR 40 36 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1 ZINC000217956479 FK In-Stock Unstable TRPV1 22 47 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1 ZINC000217956479 FK In-Stock Unstable PYGL 23 44 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1 ZINC000217956479 FK In-Stock Unstable HDAC8 15 45 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccc(C(C)(C)C)cc2)cc1 ZINC000217956479 FK In-Stock Unstable HDAC1 0 40 O=C1CC[C@@H](C(=O)N[C@@H]2CCC[C@H]2CO)N1 ZINC000217956521 BB For-Sale Unstable TRHR 40 36 COc1cccc(/C=C/NC(=O)NCCC(C)C)c1 ZINC000217956525 CG For-Sale Unstable DRD4 41 31 COc1cccc(/C=C/NC(=O)NCCC(C)C)c1 ZINC000217956525 CG For-Sale Unstable MTNR1A 78 46 COc1cccc(/C=C/NC(=O)NCCC(C)C)c1 ZINC000217956525 CG For-Sale Unstable MTNR1B 74 46 O=C(CCSc1ccccc1)Nc1ccn2nccc2c1 ZINC000217956544 CG In-Stock Unstable FAS 51 41 CN(CCCNC(=O)/C=C/c1ccc(C(C)(C)C)cc1)c1ccccc1 ZINC000217956575 FJ In-Stock Unstable DRD3 15 40 CN(CCCNC(=O)/C=C/c1ccc(C(C)(C)C)cc1)c1ccccc1 ZINC000217956575 FJ In-Stock Unstable HDAC8 17 41 CN(CCCNC(=O)/C=C/c1ccc(C(C)(C)C)cc1)c1ccccc1 ZINC000217956575 FJ In-Stock Unstable MMP2 15 47 CN(CCCNC(=O)/C=C/c1ccc(C(C)(C)C)cc1)c1ccccc1 ZINC000217956575 FJ In-Stock Unstable HDAC1 21 41 CN(CCCNC(=O)/C=C/c1ccc(C(C)(C)C)cc1)c1ccccc1 ZINC000217956575 FJ In-Stock Unstable HDAC2 20 41 CN(CCCNC(=O)/C=C/c1ccc(C(C)(C)C)cc1)c1ccccc1 ZINC000217956575 FJ In-Stock Unstable HDAC4 24 41 CN(CCCNC(=O)/C=C/c1ccc(C(C)(C)C)cc1)c1ccccc1 ZINC000217956575 FJ In-Stock Unstable HDAC9 40 41 CN(CCCNC(=O)/C=C/c1ccc(C(C)(C)C)cc1)c1ccccc1 ZINC000217956575 FJ In-Stock Unstable HDAC7 51 41 CCOc1cccc(/C=C2/CC(=O)NC2=O)c1 ZINC000217956602 BD For-Sale Unstable AKR1B1 21 42 O=C1CC[C@@H](C(=O)N[C@H]2CCC[C@H]2CO)N1 ZINC000217956609 BB On-Demand Unstable TRHR 40 36 COc1cccc(/C=C/NC(=O)NC[C@@H]2COc3ccccc3O2)c1 ZINC000217956624 EF For-Sale Unstable ADRA2B 24 42 COc1cccc(/C=C/NC(=O)NC[C@@H]2COc3ccccc3O2)c1 ZINC000217956624 EF For-Sale Unstable ADRA2C 29 42 COc1cccc(/C=C/NC(=O)NC[C@@H]2COc3ccccc3O2)c1 ZINC000217956624 EF For-Sale Unstable MTNR1A 29 42 CCC[C@@H](O)CNC(=O)[C@@H](N)CCOC ZINC000217956655 BB On-Demand Unstable DPP7 30 43 CC(C)(C)c1ccc(/C=C/C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217956694 GJ In-Stock Unstable DRD3 26 46 CC(C)(C)c1ccc(/C=C/C(=O)NCCCN2CCCc3ccccc32)cc1 ZINC000217956694 GJ In-Stock Unstable HDAC1 25 40 COc1cccc(/C=C/NC(=O)NC[C@H]2COc3ccccc3O2)c1 ZINC000217956705 EF For-Sale Unstable ADRA2B 24 42 COc1cccc(/C=C/NC(=O)NC[C@H]2COc3ccccc3O2)c1 ZINC000217956705 EF For-Sale Unstable ADRA2C 29 42 COc1cccc(/C=C/NC(=O)NC[C@H]2COc3ccccc3O2)c1 ZINC000217956705 EF For-Sale Unstable MTNR1A 29 42 CCC[C@H](O)CNC(=O)[C@@H](N)CCOC ZINC000217956722 BB On-Demand Unstable DPP7 30 43 CC(C)COC[C@@H](O)Cn1c(CC(=O)NCc2ccc(Cl)cc2)nc2ccccc21 ZINC000217956729 IH On-Demand Unstable TBXA2R 0 44 O=C(Nc1ccn2nccc2c1)c1ccc2nsnc2c1 ZINC000217956742 CF In-Stock Anodyne KCNK3 71 37 O=C(NC[C@@H]1C[C@H]2C=C[C@@H]1C2)c1ccc(NC(=O)N2CCOCC2)cc1 ZINC000217956787 FE In-Stock Unstable EPHX2 15 41 O=C(/C=C/c1ccc(Cl)cc1)Nc1ccc(CSc2ccccc2)cc1 ZINC000217956794 GK In-Stock Unstable HDAC8 21 42 O=C(/C=C/c1ccc(Cl)cc1)Nc1ccc(CSc2ccccc2)cc1 ZINC000217956794 GK In-Stock Unstable MMP2 25 67 O=C(/C=C/c1ccc(Cl)cc1)Nc1ccc(CSc2ccccc2)cc1 ZINC000217956794 GK In-Stock Unstable HDAC1 29 42 O=C(/C=C/c1ccc(Cl)cc1)Nc1ccc(CSc2ccccc2)cc1 ZINC000217956794 GK In-Stock Unstable HDAC2 24 41 O=C(/C=C/c1ccc(Cl)cc1)Nc1ccc(CSc2ccccc2)cc1 ZINC000217956794 GK In-Stock Unstable HDAC3 15 40 O=C(/C=C/c1ccc(Cl)cc1)Nc1ccc(CSc2ccccc2)cc1 ZINC000217956794 GK In-Stock Unstable MMP9 23 67 O=C(/C=C/c1ccc(Cl)cc1)Nc1ccc(CSc2ccccc2)cc1 ZINC000217956794 GK In-Stock Unstable HPSE 60 37 O=C(/C=C/c1ccc(Cl)cc1)Nc1ccc(CSc2ccccc2)cc1 ZINC000217956794 GK In-Stock Unstable MMP1 27 67 CC(C)COC[C@H](O)Cn1c(CC(=O)NCc2ccc(Cl)cc2)nc2ccccc21 ZINC000217956799 IH On-Demand Unstable TBXA2R 0 44 COc1cccc(/C=C/NC(=O)N2CCN(c3ccccc3F)CC2)c1 ZINC000217956804 FG For-Sale Unstable HTR1A 27 49 COc1cccc(/C=C/NC(=O)N2CCN(c3ccccc3F)CC2)c1 ZINC000217956804 FG For-Sale Unstable DRD2 23 41 COc1cccc(/C=C/NC(=O)N2CCN(c3ccccc3F)CC2)c1 ZINC000217956804 FG For-Sale Unstable DRD4 49 41 COc1cccc(/C=C/NC(=O)N2CCN(c3ccccc3F)CC2)c1 ZINC000217956804 FG For-Sale Unstable HTR1B 15 49 COc1cccc(/C=C/NC(=O)N2CCN(c3ccccc3F)CC2)c1 ZINC000217956804 FG For-Sale Unstable NPY2R 41 41 CCC[C@@H](O)CNC(=O)[C@H](N)CCOC ZINC000217956812 BB On-Demand Unstable DPP7 30 43 Cn1nc(-c2ccc(F)cc2)cc1C(=O)Nc1ccn2nccc2c1 ZINC000217956854 EG In-Stock Unstable AGER 0 45 CC[C@@H]1COCCN1Cc1ccccc1/C=C\C(=O)O ZINC000217956856 CE For-Sale Unstable PTGER2 31 41 CC[C@@H]1COCCN1Cc1ccccc1/C=C\C(=O)O ZINC000217956856 CE For-Sale Unstable PTGER4 15 41 CC[C@@H]1COCCN1Cc1ccccc1/C=C\C(=O)O ZINC000217956856 CE For-Sale Unstable PTGER3 16 41 CC[C@@H]1COCCN1Cc1ccccc1/C=C\C(=O)O ZINC000217956856 CE For-Sale Unstable PTGDR 15 40 O=C(NC[C@@H]1C[C@@H]2C=C[C@@H]1C2)c1ccc(NC(=O)N2CCOCC2)cc1 ZINC000217956869 FE In-Stock Unstable EPHX2 17 44 COc1cc2c(cc1OC)-c1[nH]nc(C(=O)NC[C@@H]3CCCN4CCCC[C@H]34)c1C2 ZINC000217956880 HF In-Stock Unstable CHEK1 45 43 COc1cc2c(cc1OC)-c1[nH]nc(C(=O)NC[C@@H]3CCCN4CCCC[C@H]34)c1C2 ZINC000217956880 HF In-Stock Unstable EIF2AK1 45 39 CCC[C@H](O)CNC(=O)[C@H](N)CCOC ZINC000217956889 BB On-Demand Unstable DPP7 30 43 Cc1cccc(CSCCNC(=O)/C=C/c2ccc(Cl)cc2)c1 ZINC000217956907 EJ In-Stock Unstable PYGL 24 55 Cc1cccc(CSCCNC(=O)/C=C/c2ccc(Cl)cc2)c1 ZINC000217956907 EJ In-Stock Unstable MMP2 16 45 Cc1cccc(CSCCNC(=O)/C=C/c2ccc(Cl)cc2)c1 ZINC000217956907 EJ In-Stock Unstable MMP9 15 45 Cc1cccc(CSCCNC(=O)/C=C/c2ccc(Cl)cc2)c1 ZINC000217956907 EJ In-Stock Unstable MMP1 0 42 O=C(O)[C@@H]1C[C@@H]2CCCC[C@@H]2N1C(=O)NC1CC1 ZINC000217956924 CD For-Sale Unstable ACE 17 60 CC[C@H]1COCCN1Cc1ccccc1/C=C\C(=O)O ZINC000217956933 CE For-Sale Unstable PTGER2 31 41 CC[C@H]1COCCN1Cc1ccccc1/C=C\C(=O)O ZINC000217956933 CE For-Sale Unstable PTGER4 15 41 CC[C@H]1COCCN1Cc1ccccc1/C=C\C(=O)O ZINC000217956933 CE For-Sale Unstable PTGER3 16 41 CC[C@H]1COCCN1Cc1ccccc1/C=C\C(=O)O ZINC000217956933 CE For-Sale Unstable PTGDR 15 40 O=C(Nc1ccn2nccc2c1)c1ccc(Cl)s1 ZINC000217956960 CG In-Stock Anodyne TYK2 45 34 O=C(O)[C@@H]1C[C@H]2CCCC[C@@H]2N1C(=O)NC1CC1 ZINC000217957004 CD For-Sale Unstable ACE 17 60 O=C(/C=C/c1ccc(Cl)cc1)NCCSCc1ccc(Cl)cc1Cl ZINC000217957027 HK In-Stock Unstable PYGL 27 60 O=C(/C=C/c1ccc(Cl)cc1)NCCSCc1ccc(Cl)cc1Cl ZINC000217957027 HK In-Stock Unstable HDAC9 20 40 O=C(/C=C/c1ccc(Cl)cc1)NCCSCc1ccc(Cl)cc1Cl ZINC000217957027 HK In-Stock Unstable HDAC7 30 40 Cc1noc(C)c1CC(=O)Nc1ccn2nccc2c1 ZINC000217957072 CE In-Stock Unstable P2RX7 15 47 O=C(N[C@@H]1CCC[C@@H]1CO)c1cncc(F)c1 ZINC000217957077 BD For-Sale Unstable SSTR3 24 40 O=C(/C=C/c1ccc(Cl)cc1)NCCSCc1ccc(Cl)c(Cl)c1 ZINC000217957129 HK In-Stock Unstable PYGL 31 70 O=C(N[C@H]1CCC[C@@H]1CO)c1cncc(F)c1 ZINC000217957161 BD For-Sale Unstable SSTR3 24 40 COc1cccc2c1ccn2CCC(=O)N1CCCC[C@H]1c1cccnc1 ZINC000217957175 FI In-Stock Unstable PTAFR 18 40 COc1cccc2c1ccn2CCC(=O)N1CCCC[C@H]1c1cccnc1 ZINC000217957175 FI In-Stock Unstable CHRNA2 41 42 COc1cccc2c1ccn2CCC(=O)N1CCCC[C@H]1c1cccnc1 ZINC000217957175 FI In-Stock Unstable COLA 90 38 COc1cccc2c1ccn2CCC(=O)N1CCCC[C@H]1c1cccnc1 ZINC000217957175 FI In-Stock Unstable CPT1A 85 35 COc1cccc2c1ccn2CCC(=O)N1CCCC[C@H]1c1cccnc1 ZINC000217957175 FI In-Stock Unstable GPBAR1 0 49 COc1cccc2c1ccn2CCC(=O)N1CCCC[C@H]1c1cccnc1 ZINC000217957175 FI In-Stock Unstable CRTY 0 42 COc1cccc(/C=C/NC(=O)Nc2ccc(Br)c(C)c2)c1 ZINC000217957207 FJ For-Sale Unstable MTNR1A 21 44 COc1cccc(/C=C/NC(=O)Nc2ccc(Br)c(C)c2)c1 ZINC000217957207 FJ For-Sale Unstable MTNR1B 28 44 COc1cccc(/C=C/NC(=O)Nc2ccc(Br)c(C)c2)c1 ZINC000217957207 FJ For-Sale Unstable TAAR1 22 41 COc1ccc(CN(C)CC2CC2)cc1/C=C\C(=O)O ZINC000217957209 CF For-Sale Unstable PTGER2 30 41 COc1ccc(CN(C)CC2CC2)cc1/C=C\C(=O)O ZINC000217957209 CF For-Sale Unstable PTGER4 0 41 O=C(/C=C/c1ccc(Cl)cc1)NCCSCc1ccco1 ZINC000217957229 DH In-Stock Unstable PYGL 0 52 Cc1nc([C@@H](C)NC(=O)c2cccc(N3Cc4ccccc4C3)c2)n[nH]1 ZINC000217957256 EG In-Stock Unstable PRKD1 29 40 O=C(N[C@@H]1CCC[C@H]1CO)c1cncc(F)c1 ZINC000217957257 BD For-Sale Unstable SSTR3 24 40 COc1ccc(/C(N)=C/O)cc1 ZINC000217957261 AD For-Sale Unstable KLK14 0 40 COc1ccc(N2C(=O)N[C@@H](CC(=O)N3CCc4ccccc4C3)C2=O)cc1 ZINC000217957278 GE In-Stock Unstable NOD1 16 41 COc1ccc(N2C(=O)N[C@@H](CC(=O)N3CCc4ccccc4C3)C2=O)cc1 ZINC000217957278 GE In-Stock Unstable NOD2 32 41 CC[C@@H](C)c1ccccc1NC(=O)N/C=C/c1cccc(OC)c1 ZINC000217957311 DK For-Sale Unstable KCNQ2 18 41 COC[C@H](C)N(C)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217957325 CE For-Sale Unstable TUBB1 52 39 COC[C@H](C)N(C)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217957325 CE For-Sale Unstable AKR1C3 30 41 CC(C)(C)SCCNC(=O)/C=C/c1ccc(Cl)cc1 ZINC000217957331 CI In-Stock Unstable PYGL 26 53 CC(C)(C)SCCNC(=O)/C=C/c1ccc(Cl)cc1 ZINC000217957331 CI In-Stock Unstable HDAC8 0 45 CC(C)(C)SCCNC(=O)/C=C/c1ccc(Cl)cc1 ZINC000217957331 CI In-Stock Unstable HDAC1 0 40 CC(C)(C)SCCNC(=O)/C=C/c1ccc(Cl)cc1 ZINC000217957331 CI In-Stock Unstable HDAC7 41 39 O=C(N[C@H]1CCC[C@H]1CO)c1cncc(F)c1 ZINC000217957342 BD On-Demand Unstable SSTR3 0 40 Cc1nc([C@H](C)NC(=O)c2cccc(N3Cc4ccccc4C3)c2)n[nH]1 ZINC000217957347 EG In-Stock Unstable PRKD1 29 40 O=C(Nc1ccn2nccc2c1)c1noc2c1CCCC2 ZINC000217957377 CE In-Stock Unstable PANC 59 38 CC[C@H](C)c1ccccc1NC(=O)N/C=C/c1cccc(OC)c1 ZINC000217957393 DK For-Sale Unstable KCNQ2 18 41 COC[C@@H](C)N(C)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217957411 CE For-Sale Unstable TUBB1 52 39 COC[C@@H](C)N(C)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217957411 CE For-Sale Unstable AKR1C3 30 41 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccc(Cl)cc2)c1 ZINC000217957441 EI In-Stock Unstable BDKRB2 50 32 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccc(Cl)cc2)c1 ZINC000217957441 EI In-Stock Unstable MMP2 0 46 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccc(Cl)cc2)c1 ZINC000217957441 EI In-Stock Unstable HDAC1 25 40 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccc(Cl)cc2)c1 ZINC000217957441 EI In-Stock Unstable HDAC2 0 41 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccc(Cl)cc2)c1 ZINC000217957441 EI In-Stock Unstable MMP9 0 41 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccc(Cl)cc2)c1 ZINC000217957441 EI In-Stock Unstable MMP1 0 41 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccc(Cl)cc2)c1 ZINC000217957441 EI In-Stock Unstable AMP1_PLAFQ 30 43 CC(C)Oc1cccc(CNC(=O)/C=C/c2ccc(Cl)cc2)c1 ZINC000217957441 EI In-Stock Unstable PDS 70 38 O=C(Nc1ccn2nccc2c1)c1ccc(C(F)(F)F)nc1 ZINC000217957472 DG In-Stock Anodyne KIT 15 40 O=C(Nc1ccn2nccc2c1)c1ccc(C(F)(F)F)nc1 ZINC000217957472 DG In-Stock Anodyne TRPV1 15 48 O=C(Nc1ccn2nccc2c1)c1ccc(C(F)(F)F)nc1 ZINC000217957472 DG In-Stock Anodyne DDR1 46 39 COc1cccc(/C=C/NC(=O)NCCN2C(=O)CSC2=O)c1 ZINC000217957509 ED For-Sale Unstable DRD4 46 35 CCCNC(=O)CN(C)Cc1ccccc1/C=C\C(=O)O ZINC000217957530 CD For-Sale Unstable PTGER2 35 43 CCCNC(=O)CN(C)Cc1ccccc1/C=C\C(=O)O ZINC000217957530 CD For-Sale Unstable PTGER4 0 43 CCCNC(=O)CN(C)Cc1ccccc1/C=C\C(=O)O ZINC000217957530 CD For-Sale Unstable PTGER3 17 43 C[C@@H]1CCCC[C@@H]1NC(=O)c1c[nH]nc1-c1ccc(F)cc1 ZINC000217957540 DH On-Demand Unstable SSTR3 0 40 CCOc1ccc(CNC(=O)/C=C/c2ccc(Cl)cc2)cc1OCC ZINC000217957549 FI In-Stock Unstable BDKRB2 86 38 CCOc1ccc(CNC(=O)/C=C/c2ccc(Cl)cc2)cc1OCC ZINC000217957549 FI In-Stock Unstable HDAC8 0 40 CCOc1ccc(CNC(=O)/C=C/c2ccc(Cl)cc2)cc1OCC ZINC000217957549 FI In-Stock Unstable AKR1C3 19 40 O=C(Cc1ccc(C(F)(F)F)cc1)Nc1ccn2nccc2c1 ZINC000217957569 DH In-Stock Unstable CSNK1D 29 40 O=C(Cc1ccc(C(F)(F)F)cc1)Nc1ccn2nccc2c1 ZINC000217957569 DH In-Stock Unstable FLT1 30 44 O=C(Cc1ccc(C(F)(F)F)cc1)Nc1ccn2nccc2c1 ZINC000217957569 DH In-Stock Unstable MCHR1 22 48 O=C(Cc1ccc(C(F)(F)F)cc1)Nc1ccn2nccc2c1 ZINC000217957569 DH In-Stock Unstable RORC 42 45 CN(C)C[C@H]1[C@@H]2CN(Cc3ccc(F)c(Cl)c3)C[C@H]12 ZINC000217957606 CF In-Stock Unstable SLC6A9 38 47 C[C@H]1CCCC[C@@H]1NC(=O)c1c[nH]nc1-c1ccc(F)cc1 ZINC000217957620 DH On-Demand Unstable SSTR3 0 40 COc1cccc(/C=C/NC(=O)NC2CCN(Cc3ccccc3)CC2)c1 ZINC000217957629 FH For-Sale Unstable DRD2 0 47 COc1cccc(/C=C/NC(=O)NC2CCN(Cc3ccccc3)CC2)c1 ZINC000217957629 FH For-Sale Unstable DRD3 41 52 COc1cccc(/C=C/NC(=O)NC2CCN(Cc3ccccc3)CC2)c1 ZINC000217957629 FH For-Sale Unstable BCHE 0 48 COc1cccc(/C=C/NC(=O)NC2CCN(Cc3ccccc3)CC2)c1 ZINC000217957629 FH For-Sale Unstable ADIPOR1 0 45 COc1cccc(/C=C/NC(=O)NC2CCN(Cc3ccccc3)CC2)c1 ZINC000217957629 FH For-Sale Unstable ADIPOR2 0 45 COc1cc(CNC(=O)/C=C/c2ccc(Cl)cc2)ccc1OC(C)C ZINC000217957651 FI In-Stock Unstable TRPV1 24 46 COc1cc(CNC(=O)/C=C/c2ccc(Cl)cc2)ccc1OC(C)C ZINC000217957651 FI In-Stock Unstable HDAC8 0 46 COc1cc(CNC(=O)/C=C/c2ccc(Cl)cc2)ccc1OC(C)C ZINC000217957651 FI In-Stock Unstable U38 0 41 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccc(C)cc1 ZINC000217957681 GF For-Sale Unstable COLA 79 37 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccc(C)cc1 ZINC000217957681 GF For-Sale Unstable CPT1A 68 37 CC(=O)c1cc(Br)ccc1C(F)F ZINC000217957691 BH For-Sale Unstable PYK 51 32 C[C@@H]1CCCC[C@H]1NC(=O)c1c[nH]nc1-c1ccc(F)cc1 ZINC000217957695 DH On-Demand Unstable SSTR3 0 40 COc1ccccc1CCNc1cc(Cl)nc(C2CC2)n1 ZINC000217957738 DH On-Demand Unstable PTGDR 31 43 O=C(/C=C/c1ccc(Cl)cc1)NCCCc1ccccc1Cl ZINC000217957754 EJ In-Stock Unstable DRD3 15 48 O=C(/C=C/c1ccc(Cl)cc1)NCCCc1ccccc1Cl ZINC000217957754 EJ In-Stock Unstable PYGL 29 54 O=C(/C=C/c1ccc(Cl)cc1)NCCCc1ccccc1Cl ZINC000217957754 EJ In-Stock Unstable MMP2 17 50 O=C(/C=C/c1ccc(Cl)cc1)NCCCc1ccccc1Cl ZINC000217957754 EJ In-Stock Unstable HDAC2 21 42 O=C(/C=C/c1ccc(Cl)cc1)NCCCc1ccccc1Cl ZINC000217957754 EJ In-Stock Unstable HDAC4 22 42 O=C(/C=C/c1ccc(Cl)cc1)NCCCc1ccccc1Cl ZINC000217957754 EJ In-Stock Unstable MMP9 15 50 O=C(/C=C/c1ccc(Cl)cc1)NCCCc1ccccc1Cl ZINC000217957754 EJ In-Stock Unstable HDAC9 42 42 O=C(/C=C/c1ccc(Cl)cc1)NCCCc1ccccc1Cl ZINC000217957754 EJ In-Stock Unstable HDAC7 54 42 O=C(/C=C/c1ccc(Cl)cc1)NCCCc1ccccc1Cl ZINC000217957754 EJ In-Stock Unstable MMP1 0 47 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccc(C)cc1 ZINC000217957756 GF For-Sale Unstable COLA 79 37 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccc(C)cc1 ZINC000217957756 GF For-Sale Unstable CPT1A 68 37 C[C@H]1CCCC[C@H]1NC(=O)c1c[nH]nc1-c1ccc(F)cc1 ZINC000217957767 DH On-Demand Unstable SSTR3 0 40 O=C(O)[C@@H]1C[C@@H]2CCCC[C@@H]2N1C(=O)NC1CCCC1 ZINC000217957770 CE On-Demand Unstable ACE 15 60 O=C(O)[C@@H]1C[C@H]2CCCC[C@@H]2N1C(=O)NC1CCCC1 ZINC000217957822 CE On-Demand Unstable ACE 15 60 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccc(C)cc1 ZINC000217957836 GF For-Sale Unstable COLA 79 37 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccc(C)cc1 ZINC000217957836 GF For-Sale Unstable CPT1A 68 37 COc1cccc(/C=C/NC(=O)Nc2ccc(F)c(F)c2F)c1 ZINC000217957845 DH For-Sale Unstable TAAR1 18 41 COC(=O)C[C@@H](C1=C(O)C(=O)C([C@@H](CC(=O)OC)c2coc3ccc(OC)cc3c2=O)=C(O)C1=O)c1coc2ccc(OC)cc2c1=O ZINC000217957849 KH In-Stock Unstable ALDH2 63 33 COC(=O)C[C@@H](C1=C(O)C(=O)C([C@@H](CC(=O)OC)c2coc3ccc(OC)cc3c2=O)=C(O)C1=O)c1coc2ccc(OC)cc2c1=O ZINC000217957849 KH In-Stock Unstable NQO2 21 45 COC(=O)C[C@@H](C1=C(O)C(=O)C([C@@H](CC(=O)OC)c2coc3ccc(OC)cc3c2=O)=C(O)C1=O)c1coc2ccc(OC)cc2c1=O ZINC000217957849 KH In-Stock Unstable MTNR1A 45 45 COC(=O)C[C@@H](C1=C(O)C(=O)C([C@@H](CC(=O)OC)c2coc3ccc(OC)cc3c2=O)=C(O)C1=O)c1coc2ccc(OC)cc2c1=O ZINC000217957849 KH In-Stock Unstable MTNR1B 31 45 O=C(/C=C/c1ccc(Cl)cc1)NCCCc1ccc(Cl)cc1 ZINC000217957866 EJ In-Stock Unstable PYGL 29 57 O=C(/C=C/c1ccc(Cl)cc1)NCCCc1ccc(Cl)cc1 ZINC000217957866 EJ In-Stock Unstable HDAC8 34 43 O=C(/C=C/c1ccc(Cl)cc1)NCCCc1ccc(Cl)cc1 ZINC000217957866 EJ In-Stock Unstable HDAC2 22 46 O=C(/C=C/c1ccc(Cl)cc1)NCCCc1ccc(Cl)cc1 ZINC000217957866 EJ In-Stock Unstable HDAC4 34 46 O=C(/C=C/c1ccc(Cl)cc1)NCCCc1ccc(Cl)cc1 ZINC000217957866 EJ In-Stock Unstable HDAC5 31 40 O=C(/C=C/c1ccc(Cl)cc1)NCCCc1ccc(Cl)cc1 ZINC000217957866 EJ In-Stock Unstable HDAC9 55 46 O=C(/C=C/c1ccc(Cl)cc1)NCCCc1ccc(Cl)cc1 ZINC000217957866 EJ In-Stock Unstable HDAC7 56 46 O=C(/C=C/c1ccc(Cl)cc1)NCCCc1ccc(Cl)cc1 ZINC000217957866 EJ In-Stock Unstable MMP1 0 48 O=C(/C=C/c1ccc(Cl)cc1)NCCCc1ccc(Cl)cc1 ZINC000217957866 EJ In-Stock Unstable TRPM2 0 43 Cc1cnc(C)c(NCC2(c3ccccc3)CCC2)n1 ZINC000217957910 CH On-Demand Unstable ICMT 55 33 Cc1cnc(C)c(NCC2(c3ccccc3)CCC2)n1 ZINC000217957910 CH On-Demand Unstable ACAT 0 40 COc1cc(F)c(/C=C\C(=O)CCl)c(F)c1 ZINC000217957918 BF For-Sale Unstable NFE2L2 0 42 Cc1nccc(N2CCN(C3CCOCC3)C[C@@H](O)C2)n1 ZINC000217957919 CC In-Stock Unstable SORD 54 35 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccc(C)cc1 ZINC000217957924 GF For-Sale Unstable COLA 79 37 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccc(C)cc1 ZINC000217957924 GF For-Sale Unstable CPT1A 68 37 O=C(/C=C/c1ccc(Cl)cc1)NCCCc1ccc(F)cc1 ZINC000217957932 DI In-Stock Unstable PYGL 27 51 O=C(/C=C/c1ccc(Cl)cc1)NCCCc1ccc(F)cc1 ZINC000217957932 DI In-Stock Unstable HDAC8 15 43 O=C(/C=C/c1ccc(Cl)cc1)NCCCc1ccc(F)cc1 ZINC000217957932 DI In-Stock Unstable HDAC1 20 47 O=C(/C=C/c1ccc(Cl)cc1)NCCCc1ccc(F)cc1 ZINC000217957932 DI In-Stock Unstable HDAC2 18 47 O=C(/C=C/c1ccc(Cl)cc1)NCCCc1ccc(F)cc1 ZINC000217957932 DI In-Stock Unstable HDAC4 17 47 O=C(/C=C/c1ccc(Cl)cc1)NCCCc1ccc(F)cc1 ZINC000217957932 DI In-Stock Unstable HDAC9 36 47 O=C(/C=C/c1ccc(Cl)cc1)NCCCc1ccc(F)cc1 ZINC000217957932 DI In-Stock Unstable HDAC7 54 47 O=C(/C=C/c1ccc(Cl)cc1)NCCCc1ccc(F)cc1 ZINC000217957932 DI In-Stock Unstable MMP1 0 43 O=C(/C=C/c1ccc(Cl)cc1)NCCCc1ccc(F)cc1 ZINC000217957932 DI In-Stock Unstable LEF 47 36 COC(=O)C[C@@H](C1=C(O)C(=O)C([C@H](CC(=O)OC)c2coc3ccc(OC)cc3c2=O)=C(O)C1=O)c1coc2ccc(OC)cc2c1=O ZINC000217957933 KH In-Stock Unstable ALDH2 63 33 COC(=O)C[C@@H](C1=C(O)C(=O)C([C@H](CC(=O)OC)c2coc3ccc(OC)cc3c2=O)=C(O)C1=O)c1coc2ccc(OC)cc2c1=O ZINC000217957933 KH In-Stock Unstable NQO2 21 45 COC(=O)C[C@@H](C1=C(O)C(=O)C([C@H](CC(=O)OC)c2coc3ccc(OC)cc3c2=O)=C(O)C1=O)c1coc2ccc(OC)cc2c1=O ZINC000217957933 KH In-Stock Unstable MTNR1A 45 45 COC(=O)C[C@@H](C1=C(O)C(=O)C([C@H](CC(=O)OC)c2coc3ccc(OC)cc3c2=O)=C(O)C1=O)c1coc2ccc(OC)cc2c1=O ZINC000217957933 KH In-Stock Unstable MTNR1B 31 45 COc1cccc(/C=C/NC(=O)N2CCN(Cc3ccc4c(c3)OCO4)CC2)c1 ZINC000217957955 GF For-Sale Unstable DRD4 42 32 COc1cccc(/C=C/NC(=O)N2CCN(Cc3ccc4c(c3)OCO4)CC2)c1 ZINC000217957955 GF For-Sale Unstable HRH2 22 42 COc1cccc(/C=C/NC(=O)N2CCN(Cc3ccc4c(c3)OCO4)CC2)c1 ZINC000217957955 GF For-Sale Unstable EDNRB 60 45 COc1cccc(/C=C/NC(=O)N2CCN(Cc3ccc4c(c3)OCO4)CC2)c1 ZINC000217957955 GF For-Sale Unstable EDNRA 59 45 COc1cccc(/C=C/NC(=O)N2CCN(Cc3ccc4c(c3)OCO4)CC2)c1 ZINC000217957955 GF For-Sale Unstable BMP1 65 45 COc1cccc(/C=C/NC(=O)N2CCN(Cc3ccc4c(c3)OCO4)CC2)c1 ZINC000217957955 GF For-Sale Unstable CCR3 15 41 COc1cccc(/C=C/NC(=O)N2CCN(Cc3ccc4c(c3)OCO4)CC2)c1 ZINC000217957955 GF For-Sale Unstable SSTR3 53 31 COc1cccc(/C=C/NC(=O)N2CCN(Cc3ccc4c(c3)OCO4)CC2)c1 ZINC000217957955 GF For-Sale Unstable FAAH 21 45 COc1cccc(/C=C/NC(=O)N2CCN(Cc3ccc4c(c3)OCO4)CC2)c1 ZINC000217957955 GF For-Sale Unstable MCHR1 38 55 COC(=O)C[C@H](C1=C(O)C(=O)C([C@@H](CC(=O)OC)c2coc3ccc(OC)cc3c2=O)=C(O)C1=O)c1coc2ccc(OC)cc2c1=O ZINC000217958012 KH In-Stock Unstable ALDH2 63 33 COC(=O)C[C@H](C1=C(O)C(=O)C([C@@H](CC(=O)OC)c2coc3ccc(OC)cc3c2=O)=C(O)C1=O)c1coc2ccc(OC)cc2c1=O ZINC000217958012 KH In-Stock Unstable NQO2 21 45 COC(=O)C[C@H](C1=C(O)C(=O)C([C@@H](CC(=O)OC)c2coc3ccc(OC)cc3c2=O)=C(O)C1=O)c1coc2ccc(OC)cc2c1=O ZINC000217958012 KH In-Stock Unstable MTNR1A 45 45 COC(=O)C[C@H](C1=C(O)C(=O)C([C@@H](CC(=O)OC)c2coc3ccc(OC)cc3c2=O)=C(O)C1=O)c1coc2ccc(OC)cc2c1=O ZINC000217958012 KH In-Stock Unstable MTNR1B 31 45 COc1ccccc1CCCNC(=O)/C=C/c1ccc(Cl)cc1 ZINC000217958043 EI In-Stock Unstable DRD3 26 62 COc1ccccc1CCCNC(=O)/C=C/c1ccc(Cl)cc1 ZINC000217958043 EI In-Stock Unstable BDKRB2 54 33 COc1ccccc1CCCNC(=O)/C=C/c1ccc(Cl)cc1 ZINC000217958043 EI In-Stock Unstable LTB4R 0 41 COc1ccccc1CCCNC(=O)/C=C/c1ccc(Cl)cc1 ZINC000217958043 EI In-Stock Unstable PYGL 25 46 COc1ccccc1CCCNC(=O)/C=C/c1ccc(Cl)cc1 ZINC000217958043 EI In-Stock Unstable MTNR1B 33 41 COc1ccccc1CCCNC(=O)/C=C/c1ccc(Cl)cc1 ZINC000217958043 EI In-Stock Unstable MMP2 0 45 COc1ccccc1CCCNC(=O)/C=C/c1ccc(Cl)cc1 ZINC000217958043 EI In-Stock Unstable HDAC9 40 39 COc1ccccc1CCCNC(=O)/C=C/c1ccc(Cl)cc1 ZINC000217958043 EI In-Stock Unstable HDAC7 51 39 COc1ccccc1CCCNC(=O)/C=C/c1ccc(Cl)cc1 ZINC000217958043 EI In-Stock Unstable MMP1 0 42 COc1ccccc1CCCNC(=O)/C=C/c1ccc(Cl)cc1 ZINC000217958043 EI In-Stock Unstable CYSP_PLAFA 36 40 O=C(O)/C=C\c1cccc(OCCN2CCC[C@H](O)C2)c1 ZINC000217958049 CD For-Sale Unstable HRH2 42 36 O=C(O)/C=C\c1cccc(OCCN2CCC[C@H](O)C2)c1 ZINC000217958049 CD For-Sale Unstable SLC6A1 138 39 O=C(O)/C=C\c1cccc(OCCN2CCC[C@H](O)C2)c1 ZINC000217958049 CD For-Sale Unstable ESR2 0 42 O=C(O)/C=C\c1cccc(OCCN2CCC[C@H](O)C2)c1 ZINC000217958049 CD For-Sale Unstable LTA4H 36 43 O=C(O)/C=C\c1cccc(OCCN2CCC[C@H](O)C2)c1 ZINC000217958049 CD For-Sale Unstable HRH3 26 40 O=C(O)/C=C\c1cccc(OCCN2CCC[C@H](O)C2)c1 ZINC000217958049 CD For-Sale Unstable SIGMAR1 16 46 O=C(O)/C=C\c1cccc(OCCN2CCC[C@H](O)C2)c1 ZINC000217958049 CD For-Sale Unstable PSMB2 46 39 O=C(O)/C=C\c1cccc(OCCN2CCC[C@H](O)C2)c1 ZINC000217958049 CD For-Sale Unstable PSMB1 40 39 CCOC(=O)N1CCN(C(=O)N/C=C/c2cccc(OC)c2)CC1 ZINC000217958060 EE For-Sale Unstable DRD4 42 33 CCOC(=O)N1CCN(C(=O)N/C=C/c2cccc(OC)c2)CC1 ZINC000217958060 EE For-Sale Unstable P2RY12 53 44 CCOC(=O)N1CCN(C(=O)N/C=C/c2cccc(OC)c2)CC1 ZINC000217958060 EE For-Sale Unstable MTNR1A 42 42 CCOC(=O)N1CCN(C(=O)N/C=C/c2cccc(OC)c2)CC1 ZINC000217958060 EE For-Sale Unstable MTNR1B 46 42 CNC1C[C@@H]2CC[C@@H](C1)N2[C@@H](C)Cc1ccc(F)cc1 ZINC000217958130 CF For-Sale Unstable SLC6A3 22 43 Cc1cc(Cl)cc(C(=O)N[C@@H]2CCC[C@@H]2CO)c1 ZINC000217958133 CF On-Demand Unstable CACNA1I 40 37 COc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)c1 ZINC000217958148 EI In-Stock Unstable DRD4 44 38 COc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)c1 ZINC000217958148 EI In-Stock Unstable MAOB 0 46 COc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)c1 ZINC000217958148 EI In-Stock Unstable PTGS2 21 47 COc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)c1 ZINC000217958148 EI In-Stock Unstable PYGL 26 47 COc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)c1 ZINC000217958148 EI In-Stock Unstable HDAC8 33 41 COc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)c1 ZINC000217958148 EI In-Stock Unstable MTNR1B 47 60 COc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)c1 ZINC000217958148 EI In-Stock Unstable MMP2 0 47 COc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)c1 ZINC000217958148 EI In-Stock Unstable HDAC1 21 40 COc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)c1 ZINC000217958148 EI In-Stock Unstable HDAC2 22 40 COc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)c1 ZINC000217958148 EI In-Stock Unstable HDAC6 22 41 COc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)c1 ZINC000217958148 EI In-Stock Unstable HDAC9 28 40 COc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)c1 ZINC000217958148 EI In-Stock Unstable HDAC7 42 40 COc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)c1 ZINC000217958148 EI In-Stock Unstable MMP1 0 40 COc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)c1 ZINC000217958148 EI In-Stock Unstable AMP1_PLAFQ 26 41 COc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)c1 ZINC000217958148 EI In-Stock Unstable AKR1C3 24 40 COc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)c1 ZINC000217958148 EI In-Stock Unstable FOXO1 0 40 COc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)c1 ZINC000217958148 EI In-Stock Unstable CRTM 68 49 C[C@H](Oc1ccc(Cl)cc1Cl)C(=O)Nc1ccn2nccc2c1 ZINC000217958152 FI In-Stock Unstable GUAB 0 46 C[C@H](Oc1ccc(Cl)cc1Cl)C(=O)Nc1ccn2nccc2c1 ZINC000217958152 FI In-Stock Unstable IMDH_CRYPV 36 55 COc1ccc(CN(C)CCC(C)C)cc1/C=C\C(=O)O ZINC000217958157 CG For-Sale Unstable PTGER2 24 42 COc1ccc(CN(C)CCC(C)C)cc1/C=C\C(=O)O ZINC000217958157 CG For-Sale Unstable PTGER4 0 42 O=C(/C=C\c1ccc(Cl)cc1Cl)CCl ZINC000217958159 BH For-Sale Unstable ALPL 43 35 O=C(/C=C\c1ccc(Cl)cc1Cl)CCl ZINC000217958159 BH For-Sale Unstable BOTA 33 61 O=C(/C=C\c1ccc(Cl)cc1Cl)CCl ZINC000217958159 BH For-Sale Unstable CYSP_PLAFA 35 41 Cc1cc(Cl)cc(C(=O)N[C@H]2CCC[C@@H]2CO)c1 ZINC000217958209 CF For-Sale Unstable CACNA1I 49 37 COc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217958234 EI In-Stock Unstable PTGS2 26 53 COc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217958234 EI In-Stock Unstable SCNN1A 53 42 COc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217958234 EI In-Stock Unstable PYGL 26 48 COc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217958234 EI In-Stock Unstable HDAC8 37 50 COc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217958234 EI In-Stock Unstable HDAC1 29 42 COc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217958234 EI In-Stock Unstable HDAC2 24 42 COc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217958234 EI In-Stock Unstable HDAC4 24 40 COc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217958234 EI In-Stock Unstable HDAC6 22 50 COc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217958234 EI In-Stock Unstable CCR2 0 48 COc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217958234 EI In-Stock Unstable HDAC9 40 40 COc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217958234 EI In-Stock Unstable HDAC7 43 40 COc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217958234 EI In-Stock Unstable U38 0 42 COc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217958234 EI In-Stock Unstable PROKR1 54 38 C[C@@H](Oc1ccc(Cl)cc1Cl)C(=O)Nc1ccn2nccc2c1 ZINC000217958240 FI In-Stock Unstable GUAB 0 46 C[C@@H](Oc1ccc(Cl)cc1Cl)C(=O)Nc1ccn2nccc2c1 ZINC000217958240 FI In-Stock Unstable IMDH_CRYPV 36 55 COc1ccc(OC)c(/C=C\c2csc(N)n2)c1 ZINC000217958243 CF For-Sale Unstable CYP1B1 55 54 COc1ccc(OC)c(/C=C\c2csc(N)n2)c1 ZINC000217958243 CF For-Sale Unstable CYP1A1 44 54 COc1ccc(OC)c(/C=C\c2csc(N)n2)c1 ZINC000217958243 CF For-Sale Unstable CYP1A2 16 54 CCCCCCCCOc1ccc(F)cc1CO ZINC000217958263 CI For-Sale Unstable INHA 58 35 CCCCCCCCOc1ccc(F)cc1CO ZINC000217958263 CI For-Sale Unstable LTB4R 26 41 CCCCCCCCOc1ccc(F)cc1CO ZINC000217958263 CI For-Sale Unstable LPAR2 39 40 CCCCCCCCOc1ccc(F)cc1CO ZINC000217958263 CI For-Sale Unstable S1PR3 20 40 CCCCCCCCOc1ccc(F)cc1CO ZINC000217958263 CI For-Sale Unstable PLA2G4B 80 38 CCCCCCCCOc1ccc(F)cc1CO ZINC000217958263 CI For-Sale Unstable S1PR2 42 40 Cc1cc(Cl)cc(C(=O)N[C@@H]2CCC[C@H]2CO)c1 ZINC000217958290 CF For-Sale Unstable CACNA1I 49 37 Cc1nc(Br)oc1C[C@H](N)C(=O)O ZINC000217958294 BC For-Sale Unstable GRIA3 48 40 Cc1nc(Br)oc1C[C@H](N)C(=O)O ZINC000217958294 BC For-Sale Unstable GRIA1 38 40 Cc1nc(Br)oc1C[C@H](N)C(=O)O ZINC000217958294 BC For-Sale Unstable GRIA2 39 40 Cc1nc(Br)oc1C[C@H](N)C(=O)O ZINC000217958294 BC For-Sale Unstable GRIA4 47 40 Cc1nc(Br)oc1C[C@H](N)C(=O)O ZINC000217958294 BC For-Sale Unstable GRIK1 31 40 CO[C@@H]1CC[C@@H](NC(=O)c2ccc(Cl)c(F)c2)CC1 ZINC000217958309 CG In-Stock Unstable MAPK11 35 40 CO[C@@H]1CC[C@@H](NC(=O)c2ccc(Cl)c(F)c2)CC1 ZINC000217958309 CG In-Stock Unstable MAPK14 61 46 CO[C@@H]1CC[C@@H](NC(=O)c2ccc(Cl)c(F)c2)CC1 ZINC000217958309 CG In-Stock Unstable SSTR5 40 37 CO[C@@H]1CC[C@@H](NC(=O)c2ccc(Cl)c(F)c2)CC1 ZINC000217958309 CG In-Stock Unstable MAPK13 88 43 CO[C@@H]1CC[C@@H](NC(=O)c2ccc(Cl)c(F)c2)CC1 ZINC000217958309 CG In-Stock Unstable SSTR3 0 45 CO[C@@H]1CC[C@@H](NC(=O)c2ccc(Cl)c(F)c2)CC1 ZINC000217958309 CG In-Stock Unstable EPHX2 29 42 CO[C@@H]1CC[C@@H](NC(=O)c2ccc(Cl)c(F)c2)CC1 ZINC000217958309 CG In-Stock Unstable ENV 50 40 CO[C@@H]1CC[C@@H](NC(=O)c2ccc(Cl)c(F)c2)CC1 ZINC000217958309 CG In-Stock Unstable EZH2 43 36 O=C(Nc1ccc(-c2nc3ccccc3s2)cn1)C1CCN(c2nc3ccccc3o2)CC1 ZINC000217958321 JK On-Demand Unstable APEX1 0 40 CC(C)n1ccc2ccc(C(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)cc21 ZINC000217958324 GH In-Stock Unstable CHRNA4 35 46 CCc1ncnc(-n2cnc3ccccc32)c1F ZINC000217958326 BF For-Sale Unstable PDGFRB 0 45 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217958339 EH In-Stock Unstable PTGS2 25 50 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217958339 EH In-Stock Unstable SDH1 0 40 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217958339 EH In-Stock Unstable AHR 21 40 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217958339 EH In-Stock Unstable HDAC8 20 50 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217958339 EH In-Stock Unstable CDC25B 0 43 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217958339 EH In-Stock Unstable MMP2 16 46 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217958339 EH In-Stock Unstable HDAC2 20 44 O=C(/C=C/c1cc(F)ccc1F)Nc1ccn2nccc2c1 ZINC000217958342 CG In-Stock Anodyne KCNQ2 30 42 O=C(/C=C/c1cc(F)ccc1F)Nc1ccn2nccc2c1 ZINC000217958342 CG In-Stock Anodyne MMP1 0 43 CN(CCC#N)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217958363 CE For-Sale Unstable FDPS 15 40 Cc1cc(Cl)cc(C(=O)N[C@H]2CCC[C@H]2CO)c1 ZINC000217958365 CF For-Sale Unstable CACNA1I 49 37 C#CCCCCOC(=O)c1ccc(CN2CCC(N)CC2)cc1 ZINC000217958371 DF For-Sale Unstable ACHE 19 42 C#CCCCCOC(=O)c1ccc(CN2CCC(N)CC2)cc1 ZINC000217958371 DF For-Sale Unstable SIGMAR1 30 41 Cc1nc(Br)oc1C[C@@H](N)C(=O)O ZINC000217958380 BC For-Sale Unstable GRIA3 48 40 Cc1nc(Br)oc1C[C@@H](N)C(=O)O ZINC000217958380 BC For-Sale Unstable GRIA1 38 40 Cc1nc(Br)oc1C[C@@H](N)C(=O)O ZINC000217958380 BC For-Sale Unstable GRIA2 39 40 Cc1nc(Br)oc1C[C@@H](N)C(=O)O ZINC000217958380 BC For-Sale Unstable GRIA4 47 40 Cc1nc(Br)oc1C[C@@H](N)C(=O)O ZINC000217958380 BC For-Sale Unstable GRIK1 31 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccc(Cl)cc1Cl ZINC000217958385 IH For-Sale Unstable CCR1 34 41 COc1cccc(/C=C/NC(=O)Nc2ccc(C(F)(F)F)cc2)c1 ZINC000217958407 EJ For-Sale Unstable TRPV1 16 45 COc1cccc(/C=C/NC(=O)Nc2ccc(C(F)(F)F)cc2)c1 ZINC000217958407 EJ For-Sale Unstable UL80 25 46 COc1cccc(/C=C/NC(=O)Nc2ccc(C(F)(F)F)cc2)c1 ZINC000217958407 EJ For-Sale Unstable P2RY1 24 47 COc1cccc(/C=C/NC(=O)Nc2ccc(C(F)(F)F)cc2)c1 ZINC000217958407 EJ For-Sale Unstable RAF1 35 45 COc1cccc(/C=C/NC(=O)Nc2ccc(C(F)(F)F)cc2)c1 ZINC000217958407 EJ For-Sale Unstable MTNR1A 23 47 COc1cccc(/C=C/NC(=O)Nc2ccc(C(F)(F)F)cc2)c1 ZINC000217958407 EJ For-Sale Unstable MTNR1B 31 47 COc1cccc(/C=C/NC(=O)Nc2ccc(C(F)(F)F)cc2)c1 ZINC000217958407 EJ For-Sale Unstable EPHX2 34 40 COc1cccc(/C=C/NC(=O)Nc2ccc(C(F)(F)F)cc2)c1 ZINC000217958407 EJ For-Sale Unstable AKR1C3 19 42 COc1cccc(/C=C/NC(=O)Nc2ccc(C(F)(F)F)cc2)c1 ZINC000217958407 EJ For-Sale Unstable AKR1C2 31 42 COc1cccc(/C=C/NC(=O)Nc2ccc(C(F)(F)F)cc2)c1 ZINC000217958407 EJ For-Sale Unstable IMDH_CRYPV 30 40 Cc1ncccc1OCCOc1cccc(Cl)c1 ZINC000217958411 CH On-Demand Unstable S1PR4 30 49 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217958412 EH In-Stock Unstable PTGS2 25 50 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217958412 EH In-Stock Unstable SDH1 0 40 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217958412 EH In-Stock Unstable AHR 21 40 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217958412 EH In-Stock Unstable HDAC8 20 50 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217958412 EH In-Stock Unstable CDC25B 0 43 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217958412 EH In-Stock Unstable MMP2 16 46 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217958412 EH In-Stock Unstable HDAC2 20 44 O=C(NCC(=O)N1CCCC[C@H]1c1cccnc1)c1ccccc1 ZINC000217958430 DF In-Stock Unstable CHRNA2 45 46 O=C(NCC(=O)N1CCCC[C@H]1c1cccnc1)c1ccccc1 ZINC000217958430 DF In-Stock Unstable CHRNA7 27 41 O=C(NCC(=O)N1CCCC[C@H]1c1cccnc1)c1ccccc1 ZINC000217958430 DF In-Stock Unstable CPT1A 118 43 O=C(NCC(=O)N1CCCC[C@H]1c1cccnc1)c1ccccc1 ZINC000217958430 DF In-Stock Unstable CPT2 43 32 O=C(NCC(=O)N1CCCC[C@H]1c1cccnc1)c1ccccc1 ZINC000217958430 DF In-Stock Unstable DPP4 17 42 O=C(NCC(=O)N1CCCC[C@H]1c1cccnc1)c1ccccc1 ZINC000217958430 DF In-Stock Unstable PREP 54 42 O=C(NCC(=O)N1CCCC[C@H]1c1cccnc1)c1ccccc1 ZINC000217958430 DF In-Stock Unstable FAP 0 59 O=C(NCC(=O)N1CCCC[C@H]1c1cccnc1)c1ccccc1 ZINC000217958430 DF In-Stock Unstable GPBAR1 0 41 O=C(NCC(=O)N1CCCC[C@H]1c1cccnc1)c1ccccc1 ZINC000217958430 DF In-Stock Unstable ACHP_LYMST 17 46 O=C(NCC(=O)N1CCCC[C@H]1c1cccnc1)c1ccccc1 ZINC000217958430 DF In-Stock Unstable NAMPT 42 40 O=C(NCC(=O)N1CCCC[C@H]1c1cccnc1)c1ccccc1 ZINC000217958430 DF In-Stock Unstable CRTY 0 46 COc1ccc(CN2CCOCC2)cc1/C=C\C(=O)O ZINC000217958438 CD For-Sale Unstable ACHE 15 44 COc1ccc(CN2CCOCC2)cc1/C=C\C(=O)O ZINC000217958438 CD For-Sale Unstable PTGER2 31 42 COc1ccc(CN2CCOCC2)cc1/C=C\C(=O)O ZINC000217958438 CD For-Sale Unstable PTGER4 17 42 COc1ccc(CN2CCOCC2)cc1/C=C\C(=O)O ZINC000217958438 CD For-Sale Unstable PTGER3 15 42 O=C(Nc1ccn2nccc2c1)NC1CCCCC1 ZINC000217958442 CF In-Stock Unstable CCKBR 47 40 O=C(Nc1ccn2nccc2c1)NC1CCCCC1 ZINC000217958442 CF In-Stock Unstable EPHX2 49 49 CCCCCCCOc1ccc(F)cc1CNC ZINC000217958444 CH For-Sale Unstable SLC6A4 15 51 CCCCCCCOc1ccc(F)cc1CNC ZINC000217958444 CH For-Sale Unstable LPAR2 55 46 CCCCCCCOc1ccc(F)cc1CNC ZINC000217958444 CH For-Sale Unstable S1PR3 19 46 CCCCCCCOc1ccc(F)cc1CNC ZINC000217958444 CH For-Sale Unstable PLA2G4B 43 34 CCCCCCCOc1ccc(F)cc1CNC ZINC000217958444 CH For-Sale Unstable S1PR2 53 46 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)COc1ccc(Cl)cc1Cl ZINC000217958459 IH For-Sale Unstable CCR1 34 41 COC(=O)c1cc(CN2CCC(NC(=O)OC(C)(C)C)CC2)cc(C(=O)NCCOCCO)c1 ZINC000217958473 JD For-Sale Unstable DRD4 18 40 COC(=O)c1cc(CN2CCC(NC(=O)OC(C)(C)C)CC2)cc(C(=O)NCCOCCO)c1 ZINC000217958473 JD For-Sale Unstable SSTR5 47 39 COC(=O)c1cc(CN2CCC(NC(=O)OC(C)(C)C)CC2)cc(C(=O)NCCOCCO)c1 ZINC000217958473 JD For-Sale Unstable MCHR1 25 43 COC(=O)c1cc(CN2CCC(NC(=O)OC(C)(C)C)CC2)cc(C(=O)NCCOCCO)c1 ZINC000217958473 JD For-Sale Unstable CACNA1I 57 35 COc1cccc(/C=C/NC(=O)Nc2ccc(F)cc2F)c1 ZINC000217958526 DH For-Sale Unstable MTNR1A 24 42 COc1cccc(/C=C/NC(=O)Nc2ccc(F)cc2F)c1 ZINC000217958526 DH For-Sale Unstable MTNR1B 27 42 COc1cccc(/C=C/NC(=O)Nc2ccc(F)cc2F)c1 ZINC000217958526 DH For-Sale Unstable SOAT1 18 42 COc1cccc(/C=C/NC(=O)Nc2ccc(F)cc2F)c1 ZINC000217958526 DH For-Sale Unstable TAAR1 27 41 O=C(/C=C/c1ccc(Cl)cc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217958535 FK In-Stock Anodyne MAOB 0 49 O=C(/C=C/c1ccc(Cl)cc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217958535 FK In-Stock Anodyne LTB4R 0 60 O=C(/C=C/c1ccc(Cl)cc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217958535 FK In-Stock Anodyne HDAC8 15 42 O=C(/C=C/c1ccc(Cl)cc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217958535 FK In-Stock Anodyne MMP2 25 58 O=C(/C=C/c1ccc(Cl)cc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217958535 FK In-Stock Anodyne HDAC1 27 43 O=C(/C=C/c1ccc(Cl)cc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217958535 FK In-Stock Anodyne HDAC2 23 43 O=C(/C=C/c1ccc(Cl)cc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217958535 FK In-Stock Anodyne MMP9 23 58 O=C(/C=C/c1ccc(Cl)cc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217958535 FK In-Stock Anodyne MMP1 28 58 O=C(/C=C/c1ccc(Cl)cc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217958535 FK In-Stock Anodyne HDA106 0 46 O=C(/C=C/c1ccc(Cl)cc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217958535 FK In-Stock Anodyne TRPM2 0 50 O=C(/C=C/c1ccc(Cl)cc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217958535 FK In-Stock Anodyne A0A060INS8_CAPHI 0 44 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccc(Cl)cc1Cl ZINC000217958539 IH For-Sale Unstable CCR1 34 41 COc1ccc(CN2CCC[C@@H](C)C2)cc1/C=C\C(=O)O ZINC000217958555 CG For-Sale Unstable DRD4 26 40 COc1ccc(CN2CCC[C@@H](C)C2)cc1/C=C\C(=O)O ZINC000217958555 CG For-Sale Unstable SLC6A1 59 38 COc1ccc(CN2CCC[C@@H](C)C2)cc1/C=C\C(=O)O ZINC000217958555 CG For-Sale Unstable DRD3 0 40 COc1ccc(CN2CCC[C@@H](C)C2)cc1/C=C\C(=O)O ZINC000217958555 CG For-Sale Unstable ACKR3 42 31 O=C(Nc1ccc(Cl)c(Cl)c1)Nc1ccn2nccc2c1 ZINC000217958564 DI In-Stock Anodyne FLT1 15 45 O=C(Nc1ccc(Cl)c(Cl)c1)Nc1ccn2nccc2c1 ZINC000217958564 DI In-Stock Anodyne GRM4 42 38 O=C(Nc1ccc(Cl)c(Cl)c1)Nc1ccn2nccc2c1 ZINC000217958564 DI In-Stock Anodyne Q8MMZ8_EIMTE 32 41 O=C(Nc1ccc(Cl)c(Cl)c1)Nc1ccn2nccc2c1 ZINC000217958564 DI In-Stock Anodyne BLM 0 47 O=C(Nc1ccc(Cl)c(Cl)c1)Nc1ccn2nccc2c1 ZINC000217958564 DI In-Stock Anodyne P95276_MYCTO 0 55 O=C(Nc1ccc(Cl)c(Cl)c1)Nc1ccn2nccc2c1 ZINC000217958564 DI In-Stock Anodyne WRN 0 45 O=C(Nc1ccc(Cl)c(Cl)c1)Nc1ccn2nccc2c1 ZINC000217958564 DI In-Stock Anodyne PPX1 0 43 Nc1cccc(S(=O)(=O)N2CCC[C@@H]3CCCC[C@H]32)c1 ZINC000217958576 CF On-Demand Unstable CASP3 50 34 Nc1cccc(S(=O)(=O)N2CCC[C@@H]3CCCC[C@H]32)c1 ZINC000217958576 CF On-Demand Unstable AKR1C3 55 35 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)COc1ccc(Cl)cc1Cl ZINC000217958630 IH For-Sale Unstable CCR1 34 41 COc1ccc(CN2CCC[C@H](C)C2)cc1/C=C\C(=O)O ZINC000217958641 CG For-Sale Unstable DRD4 26 40 COc1ccc(CN2CCC[C@H](C)C2)cc1/C=C\C(=O)O ZINC000217958641 CG For-Sale Unstable SLC6A1 59 38 COc1ccc(CN2CCC[C@H](C)C2)cc1/C=C\C(=O)O ZINC000217958641 CG For-Sale Unstable DRD3 19 40 COc1ccc(CN2CCC[C@H](C)C2)cc1/C=C\C(=O)O ZINC000217958641 CG For-Sale Unstable MCHR1 16 44 COc1ccc(CN2CCC[C@H](C)C2)cc1/C=C\C(=O)O ZINC000217958641 CG For-Sale Unstable ACKR3 42 31 COc1cccc(/C=C/NC(=O)Nc2cc(F)ccc2F)c1 ZINC000217958648 DH For-Sale Unstable AHR 15 41 COc1cccc(/C=C/NC(=O)Nc2cc(F)ccc2F)c1 ZINC000217958648 DH For-Sale Unstable MTNR1A 25 42 COc1cccc(/C=C/NC(=O)Nc2cc(F)ccc2F)c1 ZINC000217958648 DH For-Sale Unstable MTNR1B 28 42 COc1cccc(/C=C/NC(=O)Nc2cc(F)ccc2F)c1 ZINC000217958648 DH For-Sale Unstable TAAR1 22 43 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)c1 ZINC000217958659 FJ In-Stock Unstable PTAFR 16 41 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)c1 ZINC000217958659 FJ In-Stock Unstable HDAC7 41 38 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)c1 ZINC000217958659 FJ In-Stock Unstable AMP1_PLAFQ 34 42 CC(C)Oc1cccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)c1 ZINC000217958659 FJ In-Stock Unstable CRTM 66 48 Nc1cccc(S(=O)(=O)N2CCC[C@H]3CCCC[C@H]32)c1 ZINC000217958660 CF On-Demand Unstable CASP3 50 34 Nc1cccc(S(=O)(=O)N2CCC[C@H]3CCCC[C@H]32)c1 ZINC000217958660 CF On-Demand Unstable AKR1C3 55 35 Nc1nc(/C=C\c2c[nH]c3ccc([N+](=O)[O-])cc23)cs1 ZINC000217958663 CG For-Sale Unstable TDO2 0 40 O=C(Nc1ccc(F)cc1)Nc1ccn2nccc2c1 ZINC000217958668 CG In-Stock Anodyne HTR2A 34 44 COc1ccc(CN(CC#N)CC#N)cc1/C=C\C(=O)O ZINC000217958718 CD For-Sale Unstable PTGER2 31 43 COc1ccc(CN(CC#N)CC#N)cc1/C=C\C(=O)O ZINC000217958718 CD For-Sale Unstable PTGER4 0 43 COc1ccc(CN(CC#N)CC#N)cc1/C=C\C(=O)O ZINC000217958718 CD For-Sale Unstable PTGER3 15 43 O=C(Nc1ccc(-c2nc3ccccc3s2)cn1)c1ccc(Cl)cc1F ZINC000217958726 GK On-Demand Anodyne F10 45 43 O=C(Nc1ccc(-c2nc3ccccc3s2)cn1)c1ccc(Cl)cc1F ZINC000217958726 GK On-Demand Anodyne CSNK1D 15 40 O=C(Nc1ccc(-c2nc3ccccc3s2)cn1)c1ccc(Cl)cc1F ZINC000217958726 GK On-Demand Anodyne HSD17B1 0 41 O=C(Nc1ccc(-c2nc3ccccc3s2)cn1)c1ccc(Cl)cc1F ZINC000217958726 GK On-Demand Anodyne EPHB4 0 46 O=C(Nc1ccc(-c2nc3ccccc3s2)cn1)c1ccc(Cl)cc1F ZINC000217958726 GK On-Demand Anodyne LUCI_LUCLA 45 47 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)N3CCc4ccccc4C3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217958735 KH In-Stock Unstable TUBA1A 18 66 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)N3CCc4ccccc4C3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217958735 KH In-Stock Unstable TPPP 0 63 COc1cccc(/C=C/NC(=O)N2CCCC[C@@H]2CCO)c1 ZINC000217958746 DF For-Sale Unstable FKBP1A 23 43 COc1cccc(/C=C/NC(=O)N2CCCC[C@@H]2CCO)c1 ZINC000217958746 DF For-Sale Unstable SLC18A2 28 40 COc1cccc(/C=C/NC(=O)N2CCCC[C@@H]2CCO)c1 ZINC000217958746 DF For-Sale Unstable COLA 50 35 COc1cccc(/C=C/NC(=O)N2CCCC[C@@H]2CCO)c1 ZINC000217958746 DF For-Sale Unstable CPT1A 47 35 COc1cccc(/C=C/NC(=O)N2CCCC[C@@H]2CCO)c1 ZINC000217958746 DF For-Sale Unstable ACKR3 69 35 CC(C)Oc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217958751 FJ In-Stock Unstable HDAC7 41 38 COc1ccccc1NC(=O)Nc1ccn2nccc2c1 ZINC000217958774 CF In-Stock Unstable PTGER3 0 46 C[C@H](C(=O)NN)c1ccc(CN2CCC[C@@H]2C)cc1 ZINC000217958817 CD For-Sale Unstable HRH3 64 48 COc1cccc(/C=C/NC(=O)N2CCCC[C@H]2CCO)c1 ZINC000217958847 DF For-Sale Unstable FKBP1A 23 43 COc1cccc(/C=C/NC(=O)N2CCCC[C@H]2CCO)c1 ZINC000217958847 DF For-Sale Unstable SLC18A2 28 40 COc1cccc(/C=C/NC(=O)N2CCCC[C@H]2CCO)c1 ZINC000217958847 DF For-Sale Unstable COLA 50 35 COc1cccc(/C=C/NC(=O)N2CCCC[C@H]2CCO)c1 ZINC000217958847 DF For-Sale Unstable CPT1A 47 35 COc1cccc(/C=C/NC(=O)N2CCCC[C@H]2CCO)c1 ZINC000217958847 DF For-Sale Unstable ACKR3 69 35 O=C(/C=C/c1ccc(Cl)cc1)Nc1ccc(OC2CCCC2)cc1 ZINC000217958865 EK In-Stock Unstable HDAC8 17 53 O=C(/C=C/c1ccc(Cl)cc1)Nc1ccc(OC2CCCC2)cc1 ZINC000217958865 EK In-Stock Unstable MMP2 20 60 O=C(/C=C/c1ccc(Cl)cc1)Nc1ccc(OC2CCCC2)cc1 ZINC000217958865 EK In-Stock Unstable HDAC1 21 45 O=C(/C=C/c1ccc(Cl)cc1)Nc1ccc(OC2CCCC2)cc1 ZINC000217958865 EK In-Stock Unstable HDAC2 15 41 O=C(/C=C/c1ccc(Cl)cc1)Nc1ccc(OC2CCCC2)cc1 ZINC000217958865 EK In-Stock Unstable MMP9 22 60 O=C(/C=C/c1ccc(Cl)cc1)Nc1ccc(OC2CCCC2)cc1 ZINC000217958865 EK In-Stock Unstable EPHX2 18 49 O=C(/C=C/c1ccc(Cl)cc1)Nc1ccc(OC2CCCC2)cc1 ZINC000217958865 EK In-Stock Unstable MMP1 27 60 O=C(/C=C/c1ccc(Cl)cc1)Nc1ccc(OC2CCCC2)cc1 ZINC000217958865 EK In-Stock Unstable MCHR1 16 49 CCOc1ccc(NC(=O)Nc2ccn3nccc3c2)cc1 ZINC000217958892 CG In-Stock Unstable HTR2A 36 40 CCOc1ccc(NC(=O)Nc2ccn3nccc3c2)cc1 ZINC000217958892 CG In-Stock Unstable CA1 50 40 CCOc1ccc(NC(=O)Nc2ccn3nccc3c2)cc1 ZINC000217958892 CG In-Stock Unstable P2RY1 44 39 CCOc1ccc(NC(=O)Nc2ccn3nccc3c2)cc1 ZINC000217958892 CG In-Stock Unstable RAF1 35 41 CCOc1ccc(NC(=O)Nc2ccn3nccc3c2)cc1 ZINC000217958892 CG In-Stock Unstable CA12 24 42 CCOc1ccc(NC(=O)Nc2ccn3nccc3c2)cc1 ZINC000217958892 CG In-Stock Unstable PDGFRA 48 37 CCOc1ccc(NC(=O)Nc2ccn3nccc3c2)cc1 ZINC000217958892 CG In-Stock Unstable CA9 23 42 CCOc1ccc(NC(=O)Nc2ccn3nccc3c2)cc1 ZINC000217958892 CG In-Stock Unstable Q8MMZ8_EIMTE 59 41 CCOc1ccc(NC(=O)Nc2ccn3nccc3c2)cc1 ZINC000217958892 CG In-Stock Unstable NCE103 24 42 C[C@@H](CNC(=O)c1cc(N)cc(Cl)c1)N(C)C1CC1 ZINC000217958911 CE For-Sale Unstable CACNA1I 63 42 CCN(Cc1ccc(/C=C\C(=O)O)cc1)C1CCCCC1 ZINC000217958920 CH For-Sale Unstable NR1H4 26 42 C[C@@H](C(=O)NN)c1ccc(CN2CCC[C@@H](CO)C2)cc1 ZINC000217958932 CC For-Sale Unstable BIRC2 42 36 COc1cccc(/C=C/NC(=O)NC(C)(C)CO)c1 ZINC000217958966 CD For-Sale Unstable MTNR1A 43 44 COc1cccc(/C=C/NC(=O)NC(C)(C)CO)c1 ZINC000217958966 CD For-Sale Unstable MTNR1B 46 44 C[C@H](CNC(=O)c1cc(N)cc(Cl)c1)N(C)C1CC1 ZINC000217958982 CE For-Sale Unstable CACNA1I 63 42 O=C(Nc1ccc2c(c1)OCO2)Nc1ccn2nccc2c1 ZINC000217959009 CF In-Stock Unstable NOS2 73 32 O=C(Nc1ccc2c(c1)OCO2)Nc1ccn2nccc2c1 ZINC000217959009 CF In-Stock Unstable CCR2 16 45 C[C@H](C(=O)NN)c1ccc(CN2CCC[C@@H](CO)C2)cc1 ZINC000217959020 CC For-Sale Unstable BIRC2 42 36 CCN(Cc1cccc(/C=C\C(=O)O)c1)C1CCCCC1 ZINC000217959034 CH For-Sale Unstable PTGER2 0 40 CCN(Cc1cccc(/C=C\C(=O)O)c1)C1CCCCC1 ZINC000217959034 CH For-Sale Unstable NR1H4 40 40 COc1cccc(/C=C/NC(=O)N2CCN(c3ccccn3)CC2)c1 ZINC000217959077 EF For-Sale Unstable DRD4 41 32 COc1cccc(/C=C/NC(=O)N2CCN(c3ccccn3)CC2)c1 ZINC000217959077 EF For-Sale Unstable PDGFRB 29 42 COc1cccc(/C=C/NC(=O)N2CCN(c3ccccn3)CC2)c1 ZINC000217959077 EF For-Sale Unstable EBP 29 46 COc1cccc(/C=C/NC(=O)N2CCN(c3ccccn3)CC2)c1 ZINC000217959077 EF For-Sale Unstable SLC6A7 0 41 Nc1cc(S(=O)(=O)N2CCC[C@@H]3CCCC[C@H]32)ccc1O ZINC000217959094 DE For-Sale Unstable CASP3 56 35 Nc1cc(S(=O)(=O)N2CCC[C@@H]3CCCC[C@H]32)ccc1O ZINC000217959094 DE For-Sale Unstable CASP7 60 35 CCC[C@@H](O)CNC(=O)[C@@H](N)CCC(=O)O ZINC000217959101 BB For-Sale Unstable GRIK3 19 44 O=C(O)[C@@H]1C[C@H]2CCCC[C@@H]2N1C(=O)C[C@@H]1CCCN1 ZINC000217959102 CD For-Sale Unstable ACE 15 57 COc1cccc2c1CCc1c(C(=O)NC[C@@H]3CCCN4CCCC[C@H]34)n[nH]c1-2 ZINC000217959115 GG In-Stock Unstable DRD2 15 40 CC(=O)N1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217959116 CD For-Sale Unstable PTGER2 48 49 CC(=O)N1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217959116 CD For-Sale Unstable PTGER4 24 49 CC(=O)N1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217959116 CD For-Sale Unstable PTGER3 22 49 C[C@H]1C[C@@H](C)CN(Cc2ccc([C@H](C)C(=O)NN)cc2)C1 ZINC000217959155 CE For-Sale Unstable MLNR 17 42 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217959158 EJ In-Stock Unstable SCN2A 15 41 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217959158 EJ In-Stock Unstable PYGL 25 46 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217959158 EJ In-Stock Unstable HDAC7 42 39 CCOc1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217959158 EJ In-Stock Unstable TRPM2 0 40 Nc1cc(S(=O)(=O)N2CCC[C@H]3CCCC[C@H]32)ccc1O ZINC000217959176 DE For-Sale Unstable CASP3 56 35 Nc1cc(S(=O)(=O)N2CCC[C@H]3CCCC[C@H]32)ccc1O ZINC000217959176 DE For-Sale Unstable CASP7 60 35 CC[C@@H](C)[C@@H]1NCC[C@@H]1c1ccccc1 ZINC000217959185 BG For-Sale Unstable GALR1 46 37 COC(=O)CCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217959189 CD For-Sale Unstable DRD4 42 32 COC(=O)CCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217959189 CD For-Sale Unstable CYP1B1 15 40 COC(=O)CCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217959189 CD For-Sale Unstable MTNR1A 84 45 COC(=O)CCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217959189 CD For-Sale Unstable MTNR1B 78 45 COC(=O)CCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217959189 CD For-Sale Unstable CYP1A1 15 40 CCC[C@H](O)CNC(=O)[C@@H](N)CCC(=O)O ZINC000217959208 BB For-Sale Unstable GRIK3 19 44 C[C@H](C(=O)NN)c1ccc(CN2C[C@H](C)C[C@@H](C)C2)cc1 ZINC000217959241 CE For-Sale Unstable MLNR 17 42 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccc(Cl)cc1 ZINC000217959266 FJ In-Stock Unstable DRD3 16 51 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccc(Cl)cc1 ZINC000217959266 FJ In-Stock Unstable BDKRB2 45 38 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccc(Cl)cc1 ZINC000217959266 FJ In-Stock Unstable MTNR1A 21 44 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccc(Cl)cc1 ZINC000217959266 FJ In-Stock Unstable HDAC7 41 36 C[C@@H](CNC(=O)c1cccc(Cl)c1N)N(C)C1CC1 ZINC000217959267 CE For-Sale Unstable ECR 41 33 Nc1cc(S(=O)(=O)N2CCC[C@@H]3CCCC[C@H]32)ccc1F ZINC000217959269 DF For-Sale Unstable CASP3 64 39 Nc1cc(S(=O)(=O)N2CCC[C@@H]3CCCC[C@H]32)ccc1F ZINC000217959269 DF For-Sale Unstable CASP7 73 39 CC[C@H](C)[C@@H]1NCC[C@@H]1c1ccccc1 ZINC000217959279 BG For-Sale Unstable GALR1 46 37 CCC[C@@H](O)CNC(=O)[C@H](N)CCC(=O)O ZINC000217959282 BB For-Sale Unstable GRIK3 19 44 CCOC(=O)CCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217959309 CD For-Sale Unstable DRD4 41 32 CCOC(=O)CCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217959309 CD For-Sale Unstable MTNR1A 76 43 CCOC(=O)CCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217959309 CD For-Sale Unstable MTNR1B 69 43 CC(C)(C)c1ccc(NC(=O)Nc2ccn3nccc3c2)cc1 ZINC000217959324 DI In-Stock Unstable MAPK14 26 44 CC(C)(C)c1ccc(NC(=O)Nc2ccn3nccc3c2)cc1 ZINC000217959324 DI In-Stock Unstable TRPV1 31 43 CC(C)(C)c1ccc(NC(=O)Nc2ccn3nccc3c2)cc1 ZINC000217959324 DI In-Stock Unstable P2RY1 22 41 CC(C)(C)c1ccc(NC(=O)Nc2ccn3nccc3c2)cc1 ZINC000217959324 DI In-Stock Unstable RAF1 26 46 CC(C)(C)c1ccc(NC(=O)Nc2ccn3nccc3c2)cc1 ZINC000217959324 DI In-Stock Unstable FLT1 20 45 CC(C)(C)c1ccc(NC(=O)Nc2ccn3nccc3c2)cc1 ZINC000217959324 DI In-Stock Unstable KDR 30 45 CC(C)(C)c1ccc(NC(=O)Nc2ccn3nccc3c2)cc1 ZINC000217959324 DI In-Stock Unstable EPHX2 18 40 CC(C)(C)c1ccc(NC(=O)Nc2ccn3nccc3c2)cc1 ZINC000217959324 DI In-Stock Unstable FLT3 36 42 CC(C)(C)c1ccc(NC(=O)Nc2ccn3nccc3c2)cc1 ZINC000217959324 DI In-Stock Unstable Q8MMZ8_EIMTE 46 46 CC(C)(C)c1ccc(NC(=O)Nc2ccn3nccc3c2)cc1 ZINC000217959324 DI In-Stock Unstable IMDH_CRYPV 41 33 O=C(CN1CCN(C[C@@H](O)COc2ccccc2Cl)CC1)NCc1ccccc1 ZINC000217959325 HE On-Demand Unstable ADRB2 46 44 O=C(CN1CCN(C[C@@H](O)COc2ccccc2Cl)CC1)NCc1ccccc1 ZINC000217959325 HE On-Demand Unstable ADRB1 18 45 O=C(CN1CCN(C[C@@H](O)COc2ccccc2Cl)CC1)NCc1ccccc1 ZINC000217959325 HE On-Demand Unstable DRD4 18 48 O=C(CN1CCN(C[C@@H](O)COc2ccccc2Cl)CC1)NCc1ccccc1 ZINC000217959325 HE On-Demand Unstable ADRB3 48 44 O=C(CN1CCN(C[C@@H](O)COc2ccccc2Cl)CC1)NCc1ccccc1 ZINC000217959325 HE On-Demand Unstable HTR7 15 40 O=C(CN1CCN(C[C@@H](O)COc2ccccc2Cl)CC1)NCc1ccccc1 ZINC000217959325 HE On-Demand Unstable ACOX1 64 42 O=C(CN1CCN(C[C@@H](O)COc2ccccc2Cl)CC1)NCc1ccccc1 ZINC000217959325 HE On-Demand Unstable CCR1 41 39 O=C(CN1CCN(C[C@@H](O)COc2ccccc2Cl)CC1)NCc1ccccc1 ZINC000217959325 HE On-Demand Unstable CYP2D6 31 51 O=C(CN1CCN(C[C@@H](O)COc2ccccc2Cl)CC1)NCc1ccccc1 ZINC000217959325 HE On-Demand Unstable ABCB1 129 53 O=C(CN1CCN(C[C@@H](O)COc2ccccc2Cl)CC1)NCc1ccccc1 ZINC000217959325 HE On-Demand Unstable PDS 46 51 Nc1cc(S(=O)(=O)N2CCC[C@H]3CCCC[C@H]32)ccc1F ZINC000217959334 DF For-Sale Unstable CASP3 64 39 Nc1cc(S(=O)(=O)N2CCC[C@H]3CCCC[C@H]32)ccc1F ZINC000217959334 DF For-Sale Unstable CASP7 73 39 C[C@H](CNC(=O)c1cccc(Cl)c1N)N(C)C1CC1 ZINC000217959346 CE For-Sale Unstable ECR 41 33 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccc(Cl)cc1 ZINC000217959358 EI In-Stock Unstable BDKRB2 57 36 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccc(Cl)cc1 ZINC000217959358 EI In-Stock Unstable SDH1 0 42 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccc(Cl)cc1 ZINC000217959358 EI In-Stock Unstable CDC25B 0 40 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccc(Cl)cc1 ZINC000217959358 EI In-Stock Unstable MMP2 0 45 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccc(Cl)cc1 ZINC000217959358 EI In-Stock Unstable HDAC1 0 41 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccc(Cl)cc1 ZINC000217959358 EI In-Stock Unstable MMP9 0 45 Cc1ccccc1OC[C@@H](C)NC(=O)/C=C/c1ccc(Cl)cc1 ZINC000217959358 EI In-Stock Unstable MMP1 0 45 CC[C@@H](C)[C@H]1NCC[C@@H]1c1ccccc1 ZINC000217959360 BG For-Sale Unstable GALR1 46 37 N#Cc1cc2c(Br)cccc2c(=O)[nH]1 ZINC000217959361 BE For-Sale Mild PARP2 47 37 N#Cc1cc2c(Br)cccc2c(=O)[nH]1 ZINC000217959361 BE For-Sale Mild PARP1 17 46 CCC[C@H](O)CNC(=O)[C@H](N)CCC(=O)O ZINC000217959368 BB For-Sale Unstable GRIK3 19 44 O=C(CN1CCN(C[C@H](O)COc2ccccc2Cl)CC1)NCc1ccccc1 ZINC000217959411 HE On-Demand Unstable ADRB2 46 44 O=C(CN1CCN(C[C@H](O)COc2ccccc2Cl)CC1)NCc1ccccc1 ZINC000217959411 HE On-Demand Unstable ADRB1 18 45 O=C(CN1CCN(C[C@H](O)COc2ccccc2Cl)CC1)NCc1ccccc1 ZINC000217959411 HE On-Demand Unstable DRD4 18 48 O=C(CN1CCN(C[C@H](O)COc2ccccc2Cl)CC1)NCc1ccccc1 ZINC000217959411 HE On-Demand Unstable ADRB3 48 44 O=C(CN1CCN(C[C@H](O)COc2ccccc2Cl)CC1)NCc1ccccc1 ZINC000217959411 HE On-Demand Unstable HTR7 15 40 O=C(CN1CCN(C[C@H](O)COc2ccccc2Cl)CC1)NCc1ccccc1 ZINC000217959411 HE On-Demand Unstable ACOX1 64 42 O=C(CN1CCN(C[C@H](O)COc2ccccc2Cl)CC1)NCc1ccccc1 ZINC000217959411 HE On-Demand Unstable CCR1 41 39 O=C(CN1CCN(C[C@H](O)COc2ccccc2Cl)CC1)NCc1ccccc1 ZINC000217959411 HE On-Demand Unstable CYP2D6 31 51 O=C(CN1CCN(C[C@H](O)COc2ccccc2Cl)CC1)NCc1ccccc1 ZINC000217959411 HE On-Demand Unstable ABCB1 129 53 O=C(CN1CCN(C[C@H](O)COc2ccccc2Cl)CC1)NCc1ccccc1 ZINC000217959411 HE On-Demand Unstable PDS 46 51 CCOC(=O)CNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217959415 CD For-Sale Unstable AHR 19 41 CCOC(=O)CNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217959415 CD For-Sale Unstable MTNR1A 62 46 CCOC(=O)CNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217959415 CD For-Sale Unstable MTNR1B 60 46 C[C@H](C(=O)NN)c1ccc(CN2CCCC[C@@H]2C)cc1 ZINC000217959421 CE For-Sale Unstable HRH3 47 47 O=C(Nc1ccn2nccc2c1)Nc1ccccc1Cl ZINC000217959425 CH In-Stock Anodyne LPL 52 41 O=C(Nc1ccn2nccc2c1)Nc1ccccc1Cl ZINC000217959425 CH In-Stock Anodyne PTGER3 32 46 O=C(Nc1ccn2nccc2c1)Nc1ccccc1Cl ZINC000217959425 CH In-Stock Anodyne GRM4 41 38 O=C(Nc1ccn2nccc2c1)Nc1ccccc1Cl ZINC000217959425 CH In-Stock Anodyne MAPK10 18 45 O=C(Nc1ccn2nccc2c1)Nc1ccccc1Cl ZINC000217959425 CH In-Stock Anodyne EPHB4 0 43 O=C(Nc1ccn2nccc2c1)Nc1ccccc1Cl ZINC000217959425 CH In-Stock Anodyne EPHB3 67 45 O=C(Nc1ccn2nccc2c1)Nc1ccccc1Cl ZINC000217959425 CH In-Stock Anodyne LIPG 21 41 Cc1ccccc1OC[C@H](C)NC(=O)/C=C/c1ccc(Cl)cc1 ZINC000217959429 EI In-Stock Unstable BDKRB2 57 36 Cc1ccccc1OC[C@H](C)NC(=O)/C=C/c1ccc(Cl)cc1 ZINC000217959429 EI In-Stock Unstable SDH1 0 42 Cc1ccccc1OC[C@H](C)NC(=O)/C=C/c1ccc(Cl)cc1 ZINC000217959429 EI In-Stock Unstable CDC25B 0 40 Cc1ccccc1OC[C@H](C)NC(=O)/C=C/c1ccc(Cl)cc1 ZINC000217959429 EI In-Stock Unstable MMP2 0 45 Cc1ccccc1OC[C@H](C)NC(=O)/C=C/c1ccc(Cl)cc1 ZINC000217959429 EI In-Stock Unstable HDAC1 0 41 Cc1ccccc1OC[C@H](C)NC(=O)/C=C/c1ccc(Cl)cc1 ZINC000217959429 EI In-Stock Unstable MMP9 0 45 Cc1ccccc1OC[C@H](C)NC(=O)/C=C/c1ccc(Cl)cc1 ZINC000217959429 EI In-Stock Unstable MMP1 0 45 CC[C@H](C)[C@H]1NCC[C@@H]1c1ccccc1 ZINC000217959438 BG For-Sale Unstable GALR1 46 37 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc(C)c1 ZINC000217959450 FF For-Sale Unstable KCNK3 42 35 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1cccc(OCC#N)c1 ZINC000217959469 CI For-Sale Unstable TRPM8 17 44 O=C(N[C@@H]1CCC[C@@H]1CO)c1cccc2ncccc12 ZINC000217959504 CE For-Sale Unstable PREP 15 40 O=C(N[C@@H]1CCC[C@@H]1CO)c1cccc2ncccc12 ZINC000217959504 CE For-Sale Unstable SSTR3 17 41 COC(=O)CNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217959511 CD For-Sale Unstable DRD4 40 31 COC(=O)CNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217959511 CD For-Sale Unstable CYP1B1 29 42 COC(=O)CNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217959511 CD For-Sale Unstable AHR 23 43 COC(=O)CNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217959511 CD For-Sale Unstable MTNR1A 74 49 COC(=O)CNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217959511 CD For-Sale Unstable MTNR1B 70 49 COC(=O)CNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217959511 CD For-Sale Unstable CYP1A1 22 42 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc(C)c1 ZINC000217959521 FF For-Sale Unstable KCNK3 42 35 CNC(=O)[C@@H]1Cc2ccccc2CN1C(=O)c1c(C)cc(C)n(CCOC)c1=O ZINC000217959534 GD In-Stock Unstable OPRM1 29 46 CNC(=O)[C@@H]1Cc2ccccc2CN1C(=O)c1c(C)cc(C)n(CCOC)c1=O ZINC000217959534 GD In-Stock Unstable OPRD1 69 42 CNC(=O)[C@@H]1Cc2ccccc2CN1C(=O)c1c(C)cc(C)n(CCOC)c1=O ZINC000217959534 GD In-Stock Unstable CFTR 72 40 CNC(=O)[C@@H]1Cc2ccccc2CN1C(=O)c1c(C)cc(C)n(CCOC)c1=O ZINC000217959534 GD In-Stock Unstable ADAM9 63 35 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1cccc(OCC#N)c1 ZINC000217959545 CI For-Sale Unstable TRPM8 17 44 Cc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217959554 EI In-Stock Unstable SDH1 0 40 Cc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217959554 EI In-Stock Unstable HDAC8 0 44 Cc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217959554 EI In-Stock Unstable CDC25B 0 41 CCCCCCCOc1ccc(CNC)cc1F ZINC000217959571 CH For-Sale Unstable INHA 77 35 CCCCCCCOc1ccc(CNC)cc1F ZINC000217959571 CH For-Sale Unstable S1PR4 22 42 CCCCCCCOc1ccc(CNC)cc1F ZINC000217959571 CH For-Sale Unstable LPAR2 68 68 CCCCCCCOc1ccc(CNC)cc1F ZINC000217959571 CH For-Sale Unstable S1PR3 30 68 CCCCCCCOc1ccc(CNC)cc1F ZINC000217959571 CH For-Sale Unstable PLA2G4B 52 33 CCCCCCCOc1ccc(CNC)cc1F ZINC000217959571 CH For-Sale Unstable S1PR2 71 68 CCCCCCCOc1ccc(CNC)cc1F ZINC000217959571 CH For-Sale Unstable S1PR1 17 68 CCCCCCCOc1ccc(CNC)cc1F ZINC000217959571 CH For-Sale Unstable S1PR5 18 42 O=C(N[C@H]1CCC[C@@H]1CO)c1cccc2ncccc12 ZINC000217959593 CE For-Sale Unstable PREP 15 40 O=C(N[C@H]1CCC[C@@H]1CO)c1cccc2ncccc12 ZINC000217959593 CE For-Sale Unstable SSTR3 17 41 Cc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217959610 EI In-Stock Unstable SDH1 0 40 Cc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217959610 EI In-Stock Unstable HDAC8 0 44 Cc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217959610 EI In-Stock Unstable CDC25B 0 41 CCn1c(SCCC(=O)NC[C@@H]2CCS(=O)(=O)C2)nc2ccccc21 ZINC000217959611 GE In-Stock Unstable PTGDR2 16 40 CCn1c(SCCC(=O)NC[C@@H]2CCS(=O)(=O)C2)nc2ccccc21 ZINC000217959611 GE In-Stock Unstable TNKS 40 31 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cccc(C)c1 ZINC000217959613 FF For-Sale Unstable KCNK3 42 35 COC(=O)c1cccc(NC(=O)N/C=C/c2cccc(OC)c2)c1 ZINC000217959624 EG For-Sale Unstable CYP1B1 18 40 COC(=O)c1cccc(NC(=O)N/C=C/c2cccc(OC)c2)c1 ZINC000217959624 EG For-Sale Unstable MTNR1A 26 45 COC(=O)c1cccc(NC(=O)N/C=C/c2cccc(OC)c2)c1 ZINC000217959624 EG For-Sale Unstable MTNR1B 32 45 COC(=O)c1cccc(NC(=O)N/C=C/c2cccc(OC)c2)c1 ZINC000217959624 EG For-Sale Unstable TAAR1 31 41 COC(=O)c1cccc(NC(=O)N/C=C/c2cccc(OC)c2)c1 ZINC000217959624 EG For-Sale Unstable AKR1C3 28 42 COC(=O)c1cccc(NC(=O)N/C=C/c2cccc(OC)c2)c1 ZINC000217959624 EG For-Sale Unstable KCNK3 56 46 O=C(c1cc(-c2ccccc2)n[nH]1)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217959636 FE In-Stock Unstable CHRNA4 30 48 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1cccc(OCC#N)c1 ZINC000217959640 CI For-Sale Unstable TRPM8 17 44 C[C@H](C(=O)NN)c1ccc(CN2CCC[C@@H](C)C2)cc1 ZINC000217959669 CE For-Sale Unstable SIGMAR1 15 40 C[C@H](C(=O)NN)c1ccc(CN2CCC[C@@H](C)C2)cc1 ZINC000217959669 CE For-Sale Unstable MLNR 38 41 C[C@H](C(=O)NN)c1ccc(CN2CCC[C@@H](C)C2)cc1 ZINC000217959669 CE For-Sale Unstable BIRC2 48 37 O=C(N[C@@H]1CCC[C@H]1CO)c1cccc2ncccc12 ZINC000217959676 CE For-Sale Unstable PREP 15 40 O=C(N[C@@H]1CCC[C@H]1CO)c1cccc2ncccc12 ZINC000217959676 CE For-Sale Unstable SSTR3 17 41 COc1ccc(CCNC(=O)Nc2ccn3nccc3c2)cc1 ZINC000217959678 DF In-Stock Unstable HRH2 16 40 COc1ccc(CCNC(=O)Nc2ccn3nccc3c2)cc1 ZINC000217959678 DF In-Stock Unstable PTGER3 15 41 COc1ccc(CCNC(=O)Nc2ccn3nccc3c2)cc1 ZINC000217959678 DF In-Stock Unstable RAF1 42 39 COc1ccc(CCNC(=O)Nc2ccn3nccc3c2)cc1 ZINC000217959678 DF In-Stock Unstable MTNR1A 56 39 COc1ccc(CCNC(=O)Nc2ccn3nccc3c2)cc1 ZINC000217959678 DF In-Stock Unstable MTNR1B 50 36 COc1ccc(CCNC(=O)Nc2ccn3nccc3c2)cc1 ZINC000217959678 DF In-Stock Unstable ROCK2 20 56 COc1ccc(CCNC(=O)Nc2ccn3nccc3c2)cc1 ZINC000217959678 DF In-Stock Unstable PTGDR 23 47 COc1ccc(CCNC(=O)Nc2ccn3nccc3c2)cc1 ZINC000217959678 DF In-Stock Unstable CA9 15 40 COc1ccc(CCNC(=O)Nc2ccn3nccc3c2)cc1 ZINC000217959678 DF In-Stock Unstable QPCT 16 40 COc1ccc(CCNC(=O)Nc2ccn3nccc3c2)cc1 ZINC000217959678 DF In-Stock Unstable NCE103 20 42 COc1cc(/C=C2/CC(=O)NC2=O)ccc1OC(F)F ZINC000217959690 CD For-Sale Unstable ESRRA 56 42 COc1cc(/C=C2/CC(=O)NC2=O)ccc1OC(F)F ZINC000217959690 CD For-Sale Unstable HPGD 42 39 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cccc(C)c1 ZINC000217959704 FF For-Sale Unstable KCNK3 42 35 CCn1c(SCCC(=O)NC[C@H]2CCS(=O)(=O)C2)nc2ccccc21 ZINC000217959705 GE In-Stock Unstable PTGDR2 16 40 CCn1c(SCCC(=O)NC[C@H]2CCS(=O)(=O)C2)nc2ccccc21 ZINC000217959705 GE In-Stock Unstable TNKS 40 31 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1cccc(OCC#N)c1 ZINC000217959726 CI For-Sale Unstable TRPM8 17 44 CC1CCN(c2ccc([C@@H](C)NC(=O)/C=C/c3ccc(Cl)cc3)cc2)CC1 ZINC000217959745 GK In-Stock Unstable SDH1 0 42 CC1CCN(c2ccc([C@@H](C)NC(=O)/C=C/c3ccc(Cl)cc3)cc2)CC1 ZINC000217959745 GK In-Stock Unstable KCNQ2 48 38 CCOC(=O)c1ccc(CNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217959751 FG For-Sale Unstable MTNR1A 37 40 CCOC(=O)c1ccc(CNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217959751 FG For-Sale Unstable MTNR1B 37 40 CCOC(=O)c1ccc(CNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217959751 FG For-Sale Unstable PDS 37 41 O=C(N[C@H]1CCC[C@H]1CO)c1cccc2ncccc12 ZINC000217959761 CE On-Demand Unstable PREP 25 40 O=C(N[C@H]1CCC[C@H]1CO)c1cccc2ncccc12 ZINC000217959761 CE On-Demand Unstable FAP 0 47 COc1ccc(CNC(=O)Nc2ccn3nccc3c2)cc1 ZINC000217959793 CF In-Stock Unstable TRPV1 26 51 CC1CCN(c2ccc([C@H](C)NC(=O)/C=C/c3ccc(Cl)cc3)cc2)CC1 ZINC000217959820 GK In-Stock Unstable SDH1 0 42 CC1CCN(c2ccc([C@H](C)NC(=O)/C=C/c3ccc(Cl)cc3)cc2)CC1 ZINC000217959820 GK In-Stock Unstable KCNQ2 48 38 C[C@@H]1CCc2ccccc2N1C(=O)Cn1c2ccccc2c(=O)c2ccccc21 ZINC000217959847 GJ On-Demand Unstable ACE 25 42 C[C@@H]1CCc2ccccc2N1C(=O)Cn1c2ccccc2c(=O)c2ccccc21 ZINC000217959847 GJ On-Demand Unstable DRD4 28 41 CCC[C@@H](O)CNC(=O)CCC[C@@H](C)N ZINC000217959848 BC For-Sale Unstable NOD1 71 36 COC(=O)c1ccc(CNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217959867 EF For-Sale Unstable MTNR1A 38 42 COC(=O)c1ccc(CNC(=O)N/C=C/c2cccc(OC)c2)cc1 ZINC000217959867 EF For-Sale Unstable MTNR1B 37 40 CCC[C@H](O)CNC(=O)CCC[C@@H](C)N ZINC000217959908 BC For-Sale Unstable NOD1 71 36 C[C@H]1CCc2ccccc2N1C(=O)Cn1c2ccccc2c(=O)c2ccccc21 ZINC000217959910 GJ On-Demand Unstable ACE 25 42 C[C@H]1CCc2ccccc2N1C(=O)Cn1c2ccccc2c(=O)c2ccccc21 ZINC000217959910 GJ On-Demand Unstable DRD4 28 41 COc1cccc(/C=C/NC(=O)NCc2ccc(CO)cc2)c1 ZINC000217959940 DF For-Sale Unstable ANPEP 16 42 COc1cccc(/C=C/NC(=O)NCc2ccc(CO)cc2)c1 ZINC000217959940 DF For-Sale Unstable MTNR1A 56 43 COc1cccc(/C=C/NC(=O)NCc2ccc(CO)cc2)c1 ZINC000217959940 DF For-Sale Unstable MTNR1B 57 43 COc1cccc(/C=C/NC(=O)NCc2ccc(CO)cc2)c1 ZINC000217959940 DF For-Sale Unstable ROCK2 24 42 CCCC[C@@H](NC(=O)N1C[C@H](C)O[C@@H](C)C1)C(=O)O ZINC000217959971 CD For-Sale Unstable NOD1 89 44 CCC[C@@H](O)CNC(=O)CCC[C@H](C)N ZINC000217959979 BC For-Sale Unstable NOD1 71 36 COc1cccc(/C=C/NC(=O)NCc2ccccc2C)c1 ZINC000217960038 CG For-Sale Unstable MTNR1A 61 42 COc1cccc(/C=C/NC(=O)NCc2ccccc2C)c1 ZINC000217960038 CG For-Sale Unstable MTNR1B 56 42 CCCC[C@H](NC(=O)N1C[C@H](C)O[C@@H](C)C1)C(=O)O ZINC000217960044 CD For-Sale Unstable NOD1 89 44 CCCC[C@H](NC(=O)N1C[C@H](C)O[C@@H](C)C1)C(=O)O ZINC000217960044 CD For-Sale Unstable ZM.86993 0 40 CCC[C@H](O)CNC(=O)CCC[C@H](C)N ZINC000217960060 BC For-Sale Unstable NOD1 71 36 COc1cccc(/C=C/NC(=O)NCc2ccccc2Br)c1 ZINC000217960129 FH For-Sale Unstable MTNR1A 44 39 COc1cccc(/C=C/NC(=O)NCc2ccccc2Br)c1 ZINC000217960129 FH For-Sale Unstable MTNR1B 41 40 Cc1ccc(-c2cc(C(=O)N3CCN(c4ccccc4C)CC3)c3c(C)noc3n2)cc1 ZINC000217960136 IJ On-Demand Unstable TACR3 24 48 COc1cccc(/C=C/NC(=O)NCc2cccc(C)c2)c1 ZINC000217960229 CG For-Sale Unstable ROCK1 29 42 COc1cccc(/C=C/NC(=O)NCc2cccc(C)c2)c1 ZINC000217960229 CG For-Sale Unstable MTNR1A 58 46 COc1cccc(/C=C/NC(=O)NCc2cccc(C)c2)c1 ZINC000217960229 CG For-Sale Unstable MTNR1B 58 46 COc1cccc(/C=C/NC(=O)NCc2cccc(C)c2)c1 ZINC000217960229 CG For-Sale Unstable ROCK2 36 41 COc1cccc(/C=C/NC(=O)NCc2cccc(C)c2)c1 ZINC000217960229 CG For-Sale Unstable HSD17B2 15 42 COc1cccc(/C=C/NC(=O)NCc2cccc(C)c2)c1 ZINC000217960229 CG For-Sale Unstable PDS 40 39 O=C1CCNc2ccccc2CCN1 ZINC000217960291 AD For-Sale Unstable PRCP 40 32 CCC[C@@H](NC(=O)N1C[C@H](C)O[C@@H](C)C1)C(=O)O ZINC000217960293 CD For-Sale Unstable NOD1 51 37 COc1cccc(/C=C/NC(=O)NCc2cccc(OC)c2)c1 ZINC000217960311 DG For-Sale Unstable DRD4 40 30 COc1cccc(/C=C/NC(=O)NCc2cccc(OC)c2)c1 ZINC000217960311 DG For-Sale Unstable CYP1B1 20 41 COc1cccc(/C=C/NC(=O)NCc2cccc(OC)c2)c1 ZINC000217960311 DG For-Sale Unstable ROCK1 42 47 COc1cccc(/C=C/NC(=O)NCc2cccc(OC)c2)c1 ZINC000217960311 DG For-Sale Unstable MTNR1A 74 52 COc1cccc(/C=C/NC(=O)NCc2cccc(OC)c2)c1 ZINC000217960311 DG For-Sale Unstable MTNR1B 71 52 COc1cccc(/C=C/NC(=O)NCc2cccc(OC)c2)c1 ZINC000217960311 DG For-Sale Unstable CYP1A1 18 41 COc1cccc(/C=C/NC(=O)NCc2cccc(OC)c2)c1 ZINC000217960311 DG For-Sale Unstable ROCK2 53 52 COc1cccc(/C=C/NC(=O)NCc2cccc(OC)c2)c1 ZINC000217960311 DG For-Sale Unstable PDS 44 41 CCC[C@H](NC(=O)N1C[C@H](C)O[C@@H](C)C1)C(=O)O ZINC000217960345 CD For-Sale Unstable NOD1 51 37 C[C@@H]1CN(CC[C@H]2CCCN2)C[C@@H](C)O1 ZINC000217960381 BD For-Sale Unstable ZM.86993 0 43 COc1cccc(/C=C/NC(=O)NCc2cccc(F)c2)c1 ZINC000217960395 DG For-Sale Unstable GRIN2B 15 41 COc1cccc(/C=C/NC(=O)NCc2cccc(F)c2)c1 ZINC000217960395 DG For-Sale Unstable ROCK1 27 41 COc1cccc(/C=C/NC(=O)NCc2cccc(F)c2)c1 ZINC000217960395 DG For-Sale Unstable MTNR1A 47 44 COc1cccc(/C=C/NC(=O)NCc2cccc(F)c2)c1 ZINC000217960395 DG For-Sale Unstable MTNR1B 48 44 COc1cccc(/C=C/NC(=O)NCc2cccc(F)c2)c1 ZINC000217960395 DG For-Sale Unstable ROCK2 33 45 COc1cccc(/C=C/NC(=O)NCc2cccc(F)c2)c1 ZINC000217960395 DG For-Sale Unstable PDS 34 40 COc1ccc(CN2CCN(Cc3csc(-c4ccccn4)n3)CC2)c(OC)c1OC ZINC000217960404 IH On-Demand Unstable SLC9A1 62 36 O=C(c1ncccc1O)N1CCC[C@@H]1c1ccc(F)cc1 ZINC000217960421 CF On-Demand Unstable KCNA5 15 45 O=C(c1ncccc1O)N1CCC[C@H]1c1ccc(F)cc1 ZINC000217960484 CF On-Demand Unstable KCNA5 15 45 COc1cccc(/C=C/NC(=O)NCc2cccc(Cl)c2)c1 ZINC000217960496 DH For-Sale Unstable DRD4 41 33 COc1cccc(/C=C/NC(=O)NCc2cccc(Cl)c2)c1 ZINC000217960496 DH For-Sale Unstable ROCK1 26 41 COc1cccc(/C=C/NC(=O)NCc2cccc(Cl)c2)c1 ZINC000217960496 DH For-Sale Unstable MTNR1A 47 44 COc1cccc(/C=C/NC(=O)NCc2cccc(Cl)c2)c1 ZINC000217960496 DH For-Sale Unstable MTNR1B 49 44 COc1cccc(/C=C/NC(=O)NCc2cccc(Cl)c2)c1 ZINC000217960496 DH For-Sale Unstable ROCK2 33 43 COc1cccc(/C=C/NC(=O)NCc2cccc(Cl)c2)c1 ZINC000217960496 DH For-Sale Unstable PDS 74 40 O=C(N[C@@H]1CCC[C@@H]1CO)c1cnc(Cl)c(Cl)c1 ZINC000217960498 CE For-Sale Unstable SSTR3 30 40 CCC(=O)CCc1ccc(OCOC)cc1 ZINC000217960506 BF For-Sale Unstable PLA2G4B 59 35 CCC(=O)CCc1ccc(OCOC)cc1 ZINC000217960506 BF For-Sale Unstable FFAR1 58 43 CCC(=O)CCc1ccc(OCOC)cc1 ZINC000217960506 BF For-Sale Unstable FFAR4 49 39 O=C(N[C@H]1CCC[C@@H]1CO)c1cnc(Cl)c(Cl)c1 ZINC000217960569 CE For-Sale Unstable SSTR3 30 40 COc1cccc(/C=C/NC(=O)NCc2cccc(Br)c2)c1 ZINC000217960599 FH For-Sale Unstable ROCK2 32 40 COc1cccc(/C=C/NC(=O)NCc2cccc(Br)c2)c1 ZINC000217960599 FH For-Sale Unstable PDS 38 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217960614 JE For-Sale Unstable PKM 22 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217960614 JE For-Sale Unstable TGM2 44 35 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217960614 JE For-Sale Unstable F13A1 49 32 CCOC1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217960617 CF For-Sale Unstable PTGER2 46 42 CCOC1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217960617 CF For-Sale Unstable PTGER4 23 42 CCOC1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217960617 CF For-Sale Unstable SIGMAR1 29 40 CCOC1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217960617 CF For-Sale Unstable PTGER3 18 42 CCOC1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217960617 CF For-Sale Unstable TIMP3 69 33 O=C(N[C@@H]1CCC[C@H]1CO)c1cnc(Cl)c(Cl)c1 ZINC000217960638 CE For-Sale Unstable SSTR3 30 40 COc1cccc(/C=C/NC(=O)NCc2ccc(Br)cc2)c1 ZINC000217960675 FH For-Sale Unstable ANPEP 21 44 COc1cccc(/C=C/NC(=O)NCc2ccc(Br)cc2)c1 ZINC000217960675 FH For-Sale Unstable MTNR1A 41 43 COc1cccc(/C=C/NC(=O)NCc2ccc(Br)cc2)c1 ZINC000217960675 FH For-Sale Unstable PDS 41 37 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217960677 JE For-Sale Unstable PKM 22 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217960677 JE For-Sale Unstable TGM2 44 35 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217960677 JE For-Sale Unstable F13A1 49 32 COc1ccc([C@@H](C)NCC(=O)N2CCc3sccc3C2)cc1Br ZINC000217960679 HH On-Demand Unstable MTNR1B 19 40 CC[C@@H](NC(=O)/C=C/c1ccc(Cl)cc1)c1ccc(C)c(C)c1 ZINC000217960680 EK In-Stock Unstable BOTA 23 40 O=C(N[C@H]1CCC[C@H]1CO)c1cnc(Cl)c(Cl)c1 ZINC000217960694 CE For-Sale Unstable SSTR3 30 40 C[C@H]1CO[C@H](C)CN1Cc1ccc(CC(=O)NN)cc1 ZINC000217960699 CC For-Sale Unstable AOC2 0 40 COC[C@H](C)N(C)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217960707 CE For-Sale Unstable PTGER2 28 41 COC[C@H](C)N(C)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217960707 CE For-Sale Unstable PTGER4 17 41 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217960731 JE For-Sale Unstable PKM 22 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217960731 JE For-Sale Unstable TGM2 44 35 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217960731 JE For-Sale Unstable F13A1 49 32 Cc1ccc(/C=C2/CC(=O)NC2=O)cc1 ZINC000217960746 BD For-Sale Unstable HPGD 29 43 CC[C@H](NC(=O)/C=C/c1ccc(Cl)cc1)c1ccc(C)c(C)c1 ZINC000217960749 EK In-Stock Unstable BOTA 23 40 O=C(NCc1ccc(F)cc1)Nc1ccn2nccc2c1 ZINC000217960754 CF In-Stock Unstable CCR3 48 37 O=C(NCc1ccc(F)cc1)Nc1ccn2nccc2c1 ZINC000217960754 CF In-Stock Unstable ROCK2 22 45 O=C(NCc1ccc(F)cc1)Nc1ccn2nccc2c1 ZINC000217960754 CF In-Stock Unstable NAMPT 47 41 COc1ccc([C@H](C)NCC(=O)N2CCc3sccc3C2)cc1Br ZINC000217960761 HH On-Demand Unstable MTNR1B 19 40 COc1cccc(/C=C/NC(=O)NCCc2ccccc2C)c1 ZINC000217960780 DH For-Sale Unstable DRD4 40 31 COc1cccc(/C=C/NC(=O)NCCc2ccccc2C)c1 ZINC000217960780 DH For-Sale Unstable NQO2 44 44 COc1cccc(/C=C/NC(=O)NCCc2ccccc2C)c1 ZINC000217960780 DH For-Sale Unstable MTNR1A 131 47 COc1cccc(/C=C/NC(=O)NCCc2ccccc2C)c1 ZINC000217960780 DH For-Sale Unstable MTNR1B 109 46 C[C@H]1CN(Cc2ccc(CC(=O)NN)cc2)[C@@H](C)CO1 ZINC000217960784 CC For-Sale Unstable AOC2 0 40 COC[C@@H](C)N(C)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217960790 CE For-Sale Unstable PTGER2 28 41 COC[C@@H](C)N(C)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217960790 CE For-Sale Unstable PTGER4 17 41 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217960802 JE For-Sale Unstable PKM 22 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217960802 JE For-Sale Unstable TGM2 44 35 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000217960802 JE For-Sale Unstable F13A1 49 32 FC(F)(F)Oc1ccc(-c2cc(Cl)ncn2)cc1Cl ZINC000217960827 DI For-Sale Anodyne GRIN2B 15 45 CC(C)CCn1cnc2ccc(NC(=O)CCn3cnc4ccccc4c3=O)cc2c1=O ZINC000217960837 IG In-Stock Unstable SCD1 0 49 CC(C)CCn1cnc2ccc(NC(=O)CCn3cnc4ccccc4c3=O)cc2c1=O ZINC000217960837 IG In-Stock Unstable SCD 0 44 CC(C)CCn1cnc2ccc(NC(=O)CCn3cnc4ccccc4c3=O)cc2c1=O ZINC000217960837 IG In-Stock Unstable IMDH_CRYPV 44 39 CC[C@@H](NC(=O)/C=C/c1ccc(Cl)cc1)c1ccc(C)cc1C ZINC000217960867 EK In-Stock Unstable BOTA 16 40 CS(=O)(=O)[C@@H]1C[C@@]1(N)C(=O)O ZINC000217960871 AA In-Stock Unstable GRM2 0 42 CS(=O)(=O)[C@@H]1C[C@@]1(N)C(=O)O ZINC000217960871 AA In-Stock Unstable GRM1 0 42 COc1cccc(/C=C/NC(=O)NCCc2ccccc2OC)c1 ZINC000217960876 EG For-Sale Unstable CYP1B1 26 42 COc1cccc(/C=C/NC(=O)NCCc2ccccc2OC)c1 ZINC000217960876 EG For-Sale Unstable NQO2 47 44 COc1cccc(/C=C/NC(=O)NCCc2ccccc2OC)c1 ZINC000217960876 EG For-Sale Unstable MTNR1A 137 48 COc1cccc(/C=C/NC(=O)NCCc2ccccc2OC)c1 ZINC000217960876 EG For-Sale Unstable MTNR1B 118 48 COc1cccc(/C=C/NC(=O)NCCc2ccccc2OC)c1 ZINC000217960876 EG For-Sale Unstable CYP1A1 22 42 COc1cccc(/C=C/NC(=O)NCCc2ccccc2OC)c1 ZINC000217960876 EG For-Sale Unstable ABCG2 28 42 COc1cccc(/C=C/NC(=O)NCCc2ccccc2OC)c1 ZINC000217960876 EG For-Sale Unstable ACKR3 46 31 CCCC[C@@H](CC)COC(=O)OC(C)(C)C ZINC000217960900 BI For-Sale Unstable CTSK 20 45 COc1ccc(OC)c(/C=C\C(=O)CCl)c1 ZINC000217960903 BF For-Sale Unstable PTGS2 0 45 COc1ccc(OC)c(/C=C\C(=O)CCl)c1 ZINC000217960903 BF For-Sale Unstable CYP1B1 58 54 COc1ccc(OC)c(/C=C\C(=O)CCl)c1 ZINC000217960903 BF For-Sale Unstable TNFRSF1A 28 42 COc1ccc(OC)c(/C=C\C(=O)CCl)c1 ZINC000217960903 BF For-Sale Unstable MTNR1A 44 44 COc1ccc(OC)c(/C=C\C(=O)CCl)c1 ZINC000217960903 BF For-Sale Unstable MTNR1B 38 44 COc1ccc(OC)c(/C=C\C(=O)CCl)c1 ZINC000217960903 BF For-Sale Unstable CYP1A1 43 54 COc1ccc(OC)c(/C=C\C(=O)CCl)c1 ZINC000217960903 BF For-Sale Unstable CYP1A2 18 54 COc1ccc(OC)c(/C=C\C(=O)CCl)c1 ZINC000217960903 BF For-Sale Unstable ABCG2 23 65 COc1ccc(OC)c(/C=C\C(=O)CCl)c1 ZINC000217960903 BF For-Sale Unstable CYSP_PLAFA 64 57 CC[C@H](NC(=O)/C=C/c1ccc(Cl)cc1)c1ccc(C)cc1C ZINC000217960944 EK In-Stock Unstable BOTA 16 40 CS(=O)(=O)[C@H]1C[C@@]1(N)C(=O)O ZINC000217960945 AA In-Stock Unstable GRM2 0 42 CS(=O)(=O)[C@H]1C[C@@]1(N)C(=O)O ZINC000217960945 AA In-Stock Unstable GRM1 0 42 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1ccc(Cl)c(F)c1 ZINC000217960967 CK For-Sale Unstable ENV 44 33 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1ccc(Cl)c(F)c1 ZINC000217960967 CK For-Sale Unstable TRPM8 16 49 O=C(NCCCc1ccccc1)Nc1ccn2nccc2c1 ZINC000217960975 CG In-Stock Unstable CES1 40 33 O=C(NCCCc1ccccc1)Nc1ccn2nccc2c1 ZINC000217960975 CG In-Stock Unstable NCE103 18 42 O=C(NCCCc1ccccc1)Nc1ccn2nccc2c1 ZINC000217960975 CG In-Stock Unstable CRTM 42 38 O=C(NCCCc1ccccc1)Nc1ccn2nccc2c1 ZINC000217960975 CG In-Stock Unstable ACAT 0 46 COc1cccc(/C=C/NC(=O)NCCc2ccccc2F)c1 ZINC000217960978 DG For-Sale Unstable DRD4 42 32 COc1cccc(/C=C/NC(=O)NCCc2ccccc2F)c1 ZINC000217960978 DG For-Sale Unstable NQO2 47 47 COc1cccc(/C=C/NC(=O)NCCc2ccccc2F)c1 ZINC000217960978 DG For-Sale Unstable MTNR1A 139 49 COc1cccc(/C=C/NC(=O)NCCc2ccccc2F)c1 ZINC000217960978 DG For-Sale Unstable MTNR1B 114 48 CCCC[C@H](CC)COC(=O)OC(C)(C)C ZINC000217960980 BI For-Sale Unstable CTSK 20 45 CS(=O)(=O)[C@@H]1C[C@]1(N)C(=O)O ZINC000217961028 AA In-Stock Unstable GRM2 0 42 CS(=O)(=O)[C@@H]1C[C@]1(N)C(=O)O ZINC000217961028 AA In-Stock Unstable GRM1 0 42 COc1cc2c(cc1OC)-c1[nH]nc(C(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)c1C2 ZINC000217961037 IE In-Stock Unstable CHRNA4 25 41 COc1cc2c(cc1OC)-c1[nH]nc(C(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)c1C2 ZINC000217961037 IE In-Stock Unstable CHEK1 40 38 COc1cc2c(cc1OC)-c1[nH]nc(C(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)c1C2 ZINC000217961037 IE In-Stock Unstable EIF2AK1 43 39 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1ccc(Cl)c(F)c1 ZINC000217961050 CK For-Sale Unstable ENV 44 33 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1ccc(Cl)c(F)c1 ZINC000217961050 CK For-Sale Unstable TRPM8 16 49 C[C@@H](C(=O)NN)c1ccc(CN2CC[C@@H](N)C2)cc1 ZINC000217961056 CC For-Sale Unstable MLNR 30 40 CC[C@@H](NC(=O)/C=C/c1ccc(Cl)cc1)c1ccc(OC)c(OC)c1 ZINC000217961062 FJ In-Stock Unstable UTS2 41 33 CC[C@@H](NC(=O)/C=C/c1ccc(Cl)cc1)c1ccc(OC)c(OC)c1 ZINC000217961062 FJ In-Stock Unstable CYSP_PLAFA 38 40 COCCNC(=O)Nc1ccn2nccc2c1 ZINC000217961075 BD In-Stock Unstable PRMT3 45 32 COc1cccc(/C=C/NC(=O)NCCc2ccccc2Cl)c1 ZINC000217961078 EH For-Sale Unstable DRD4 45 38 COc1cccc(/C=C/NC(=O)NCCc2ccccc2Cl)c1 ZINC000217961078 EH For-Sale Unstable NQO2 43 43 COc1cccc(/C=C/NC(=O)NCCc2ccccc2Cl)c1 ZINC000217961078 EH For-Sale Unstable MTNR1A 126 47 COc1cccc(/C=C/NC(=O)NCCc2ccccc2Cl)c1 ZINC000217961078 EH For-Sale Unstable MTNR1B 105 46 COc1cccc(/C=C/NC(=O)NCCc2ccccc2Cl)c1 ZINC000217961078 EH For-Sale Unstable CAN2 0 44 CCCN1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217961083 CE For-Sale Unstable PTGER2 45 47 CCCN1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217961083 CE For-Sale Unstable PTGER4 21 47 CCCN1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217961083 CE For-Sale Unstable SIGMAR1 20 43 CCCN1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217961083 CE For-Sale Unstable PTGER3 19 47 CCCN1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217961083 CE For-Sale Unstable PTGDR 17 45 COc1ccc(-c2cccc([N+](=O)[O-])c2O)cc1 ZINC000217961099 BF For-Sale Unstable HDAC2 23 50 CS(=O)(=O)[C@H]1C[C@]1(N)C(=O)O ZINC000217961107 AA In-Stock Unstable GRM2 0 42 CS(=O)(=O)[C@H]1C[C@]1(N)C(=O)O ZINC000217961107 AA In-Stock Unstable GRM1 0 42 CC[C@@H](C)[C@@H](NC(=O)N1CCC[C@@H](C)C1)C(=O)O ZINC000217961110 CD For-Sale Unstable RIR1_HHV11 48 32 CC[C@@H](C)[C@@H](NC(=O)N1CCC[C@@H](C)C1)C(=O)O ZINC000217961110 CD For-Sale Unstable NTSR1 56 33 CC[C@@H](C)[C@@H](NC(=O)N1CCC[C@@H](C)C1)C(=O)O ZINC000217961110 CD For-Sale Unstable ENPEP 60 36 CC[C@@H](C)[C@@H](NC(=O)N1CCC[C@@H](C)C1)C(=O)O ZINC000217961110 CD For-Sale Unstable TPP2 20 50 O=C(CN1CCC(c2ccccc2)CC1)N1CCC[C@@](O)(CO)CC1 ZINC000217961133 ED In-Stock Unstable DRD4 0 42 O=C(CN1CCC(c2ccccc2)CC1)N1CCC[C@@](O)(CO)CC1 ZINC000217961133 ED In-Stock Unstable CCR5 19 42 O=C(CN1CCC(c2ccccc2)CC1)N1CCC[C@@](O)(CO)CC1 ZINC000217961133 ED In-Stock Unstable SLC18A3 46 33 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1ccc(Cl)c(F)c1 ZINC000217961141 CK For-Sale Unstable ENV 44 33 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1ccc(Cl)c(F)c1 ZINC000217961141 CK For-Sale Unstable TRPM8 16 49 COc1ccc(F)cc1/C=C\C(=O)CCl ZINC000217961146 BF For-Sale Unstable TNFRSF1A 27 42 COc1ccc(F)cc1/C=C\C(=O)CCl ZINC000217961146 BF For-Sale Unstable ABCG2 16 47 COc1ccc(F)cc1/C=C\C(=O)CCl ZINC000217961146 BF For-Sale Unstable NFE2L2 0 43 COc1ccc(F)cc1/C=C\C(=O)CCl ZINC000217961146 BF For-Sale Unstable CYSP_PLAFA 59 42 CC[C@H](NC(=O)/C=C/c1ccc(Cl)cc1)c1ccc(OC)c(OC)c1 ZINC000217961147 FJ In-Stock Unstable UTS2 41 33 CC[C@H](NC(=O)/C=C/c1ccc(Cl)cc1)c1ccc(OC)c(OC)c1 ZINC000217961147 FJ In-Stock Unstable CYSP_PLAFA 38 40 C[C@H](C(=O)NN)c1ccc(CN2CC[C@@H](N)C2)cc1 ZINC000217961153 CC For-Sale Unstable MLNR 30 40 Cc1ncccc1C(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217961157 BD For-Sale Unstable G2YM83_BOTF4 52 35 CC(C)C[C@@H](C(=O)N1CCCC[C@H]1c1cccnc1)N1Cc2ccccc2C1=O ZINC000217961166 GI In-Stock Unstable COLA 49 37 CC(C)C[C@@H](C(=O)N1CCCC[C@H]1c1cccnc1)N1Cc2ccccc2C1=O ZINC000217961166 GI In-Stock Unstable CPT1A 52 34 CC(C)C[C@@H](C(=O)N1CCCC[C@H]1c1cccnc1)N1Cc2ccccc2C1=O ZINC000217961166 GI In-Stock Unstable GPBAR1 0 41 COc1cccc(/C=C/NC(=O)NCCc2ccccc2Br)c1 ZINC000217961185 GH For-Sale Unstable NQO2 45 43 COc1cccc(/C=C/NC(=O)NCCc2ccccc2Br)c1 ZINC000217961185 GH For-Sale Unstable MTNR1A 124 47 COc1cccc(/C=C/NC(=O)NCCc2ccccc2Br)c1 ZINC000217961185 GH For-Sale Unstable MTNR1B 103 46 CC[C@H](C)[C@@H](NC(=O)N1CCC[C@@H](C)C1)C(=O)O ZINC000217961187 CD For-Sale Unstable RIR1_HHV11 48 32 CC[C@H](C)[C@@H](NC(=O)N1CCC[C@@H](C)C1)C(=O)O ZINC000217961187 CD For-Sale Unstable NTSR1 56 33 CC[C@H](C)[C@@H](NC(=O)N1CCC[C@@H](C)C1)C(=O)O ZINC000217961187 CD For-Sale Unstable ENPEP 60 36 CC[C@H](C)[C@@H](NC(=O)N1CCC[C@@H](C)C1)C(=O)O ZINC000217961187 CD For-Sale Unstable TPP2 20 50 CCCN1CCN(Cc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217961192 CE For-Sale Unstable DRD4 29 40 CCCN1CCN(Cc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217961192 CE For-Sale Unstable SIGMAR1 34 46 CCCN1CCN(Cc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217961192 CE For-Sale Unstable CACNA1G 20 43 c1ccc2c(c1)CCNCCCN2 ZINC000217961216 AD For-Sale Unstable PRCP 42 34 COc1ccc(I)cc1/C=C\C(=O)CCl ZINC000217961225 EG For-Sale Unstable TNFRSF1A 23 41 COc1ccc(I)cc1/C=C\C(=O)CCl ZINC000217961225 EG For-Sale Unstable ABCG2 16 46 COc1ccc(I)cc1/C=C\C(=O)CCl ZINC000217961225 EG For-Sale Unstable CYSP_PLAFA 52 42 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1ccc(Cl)c(F)c1 ZINC000217961227 CK For-Sale Unstable ENV 44 33 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1ccc(Cl)c(F)c1 ZINC000217961227 CK For-Sale Unstable TRPM8 16 49 Cc1ncccc1C(=O)N[C@H]1CCC[C@@H]1CO ZINC000217961229 BD For-Sale Unstable G2YM83_BOTF4 52 35 O=C(CN1CCC(c2ccccc2)CC1)N1CCC[C@](O)(CO)CC1 ZINC000217961239 ED In-Stock Unstable DRD4 0 42 O=C(CN1CCC(c2ccccc2)CC1)N1CCC[C@](O)(CO)CC1 ZINC000217961239 ED In-Stock Unstable CCR5 19 42 O=C(CN1CCC(c2ccccc2)CC1)N1CCC[C@](O)(CO)CC1 ZINC000217961239 ED In-Stock Unstable SLC18A3 46 33 CC[C@@H](NC(=O)/C=C/c1ccc(Cl)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217961264 GI In-Stock Unstable PTGS2 17 42 CC[C@@H](NC(=O)/C=C/c1ccc(Cl)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217961264 GI In-Stock Unstable HDAC8 0 46 O=C1C[C@H](C(=O)N2CCCC[C@H]2c2cccnc2)CN1c1ccccc1 ZINC000217961271 EG In-Stock Unstable CHRNA2 43 44 O=C1C[C@H](C(=O)N2CCCC[C@H]2c2cccnc2)CN1c1ccccc1 ZINC000217961271 EG In-Stock Unstable CHRNA4 16 44 O=C1C[C@H](C(=O)N2CCCC[C@H]2c2cccnc2)CN1c1ccccc1 ZINC000217961271 EG In-Stock Unstable COLA 87 41 O=C1C[C@H](C(=O)N2CCCC[C@H]2c2cccnc2)CN1c1ccccc1 ZINC000217961271 EG In-Stock Unstable CPT1A 83 36 O=C1C[C@H](C(=O)N2CCCC[C@H]2c2cccnc2)CN1c1ccccc1 ZINC000217961271 EG In-Stock Unstable GPBAR1 0 44 O=C1C[C@H](C(=O)N2CCCC[C@H]2c2cccnc2)CN1c1ccccc1 ZINC000217961271 EG In-Stock Unstable CRTY 0 44 CCC[C@@H](O)CNC(=O)[C@@H](N)CC(=O)O ZINC000217961278 BB For-Sale Unstable DPP7 37 41 CCC[C@@H](O)CNC(=O)[C@@H](N)CC(=O)O ZINC000217961278 BB For-Sale Unstable DPP8 32 40 CCC[C@@H](O)CNC(=O)[C@@H](N)CC(=O)O ZINC000217961278 BB For-Sale Unstable DPP9 27 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000217961281 JF For-Sale Unstable NAMPT 16 40 COc1cccc(/C=C/NC(=O)NCCc2cccc(C)c2)c1 ZINC000217961291 DH For-Sale Unstable DRD4 41 34 COc1cccc(/C=C/NC(=O)NCCc2cccc(C)c2)c1 ZINC000217961291 DH For-Sale Unstable MTNR1A 99 53 COc1cccc(/C=C/NC(=O)NCCc2cccc(C)c2)c1 ZINC000217961291 DH For-Sale Unstable MTNR1B 89 53 COc1cccc(/C=C/NC(=O)NCCc2cccc(C)c2)c1 ZINC000217961291 DH For-Sale Unstable ABCG2 17 41 COc1ccc(/C=C\C(=O)CCl)cc1Cl ZINC000217961296 BG For-Sale Unstable PYGL 19 44 COc1ccc(/C=C\C(=O)CCl)cc1Cl ZINC000217961296 BG For-Sale Unstable CA14 17 45 COc1ccc(/C=C\C(=O)CCl)cc1Cl ZINC000217961296 BG For-Sale Unstable CYP1A1 18 40 COc1ccc(/C=C\C(=O)CCl)cc1Cl ZINC000217961296 BG For-Sale Unstable TUBB1 60 43 COc1ccc(/C=C\C(=O)CCl)cc1Cl ZINC000217961296 BG For-Sale Unstable ABCG2 19 45 COc1ccc(/C=C\C(=O)CCl)cc1Cl ZINC000217961296 BG For-Sale Unstable CYSP_PLAFA 53 42 Fc1cc(N[C@@H]2C[C@@H]3C[C@@H]2[C@@H]2CCC[C@@H]32)ccc1Cl ZINC000217961299 CJ For-Sale Unstable ENV 43 35 O=S(=O)(Cc1ccccc1)Nc1ccn2nccc2c1 ZINC000217961300 CE In-Stock Unstable NR1I2 41 31 Cc1ncccc1C(=O)N[C@@H]1CCC[C@H]1CO ZINC000217961309 BD For-Sale Unstable G2YM83_BOTF4 52 35 CCCN1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217961311 CE For-Sale Unstable HTR1A 19 40 CCCN1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217961311 CE For-Sale Unstable DRD2 30 40 CCCN1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217961311 CE For-Sale Unstable SIGMAR1 50 46 CCCN1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217961311 CE For-Sale Unstable HDAC1 17 41 CCCN1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217961311 CE For-Sale Unstable CACNA1G 29 41 CCCN1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217961311 CE For-Sale Unstable AKR1C3 33 41 CC(C)Oc1cc2c(cn1)CCNC2=O ZINC000217961325 BD For-Sale Unstable CSNK1G2 55 30 COC(=O)CCSc1nc2cc(C)ccc2o1 ZINC000217961332 CF On-Demand Unstable CETP 16 40 COC(=O)CCSc1nc2cc(C)ccc2o1 ZINC000217961332 CF On-Demand Unstable AGPAT2 22 42 CCC[C@H](O)CNC(=O)[C@@H](N)CC(=O)O ZINC000217961341 BB For-Sale Unstable DPP7 37 41 CCC[C@H](O)CNC(=O)[C@@H](N)CC(=O)O ZINC000217961341 BB For-Sale Unstable DPP8 32 40 CCC[C@H](O)CNC(=O)[C@@H](N)CC(=O)O ZINC000217961341 BB For-Sale Unstable DPP9 27 40 CC[C@H](NC(=O)/C=C/c1ccc(Cl)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217961346 GI In-Stock Unstable PTGS2 17 42 CC[C@H](NC(=O)/C=C/c1ccc(Cl)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217961346 GI In-Stock Unstable HDAC8 0 46 O=C1C[C@@H](C(=O)N2CCCC[C@H]2c2cccnc2)CN1c1ccccc1 ZINC000217961347 EG In-Stock Unstable CHRNA2 43 44 O=C1C[C@@H](C(=O)N2CCCC[C@H]2c2cccnc2)CN1c1ccccc1 ZINC000217961347 EG In-Stock Unstable CHRNA4 16 44 O=C1C[C@@H](C(=O)N2CCCC[C@H]2c2cccnc2)CN1c1ccccc1 ZINC000217961347 EG In-Stock Unstable COLA 87 41 O=C1C[C@@H](C(=O)N2CCCC[C@H]2c2cccnc2)CN1c1ccccc1 ZINC000217961347 EG In-Stock Unstable CPT1A 83 36 O=C1C[C@@H](C(=O)N2CCCC[C@H]2c2cccnc2)CN1c1ccccc1 ZINC000217961347 EG In-Stock Unstable GPBAR1 0 44 O=C1C[C@@H](C(=O)N2CCCC[C@H]2c2cccnc2)CN1c1ccccc1 ZINC000217961347 EG In-Stock Unstable CRTY 0 44 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000217961356 JF For-Sale Unstable NAMPT 16 40 COc1ccc(/C=C\C(=O)CCl)cc1Br ZINC000217961377 CG For-Sale Unstable APP 48 39 COc1ccc(/C=C\C(=O)CCl)cc1Br ZINC000217961377 CG For-Sale Unstable TUBB1 60 42 COc1ccc(/C=C\C(=O)CCl)cc1Br ZINC000217961377 CG For-Sale Unstable PTPA 0 40 COc1ccc(/C=C\C(=O)CCl)cc1Br ZINC000217961377 CG For-Sale Unstable ABCG2 18 44 COc1ccc(/C=C\C(=O)CCl)cc1Br ZINC000217961377 CG For-Sale Unstable NFE2L2 0 42 Cc1ncccc1C(=O)N[C@H]1CCC[C@H]1CO ZINC000217961384 BD For-Sale Unstable G2YM83_BOTF4 52 35 Fc1cc(N[C@H]2C[C@@H]3C[C@@H]2[C@@H]2CCC[C@@H]32)ccc1Cl ZINC000217961393 CJ For-Sale Unstable ENV 43 35 COc1cccc(/C=C/NC(=O)NCCc2cccc(OC)c2)c1 ZINC000217961402 EG For-Sale Unstable DRD4 41 31 COc1cccc(/C=C/NC(=O)NCCc2cccc(OC)c2)c1 ZINC000217961402 EG For-Sale Unstable HRH2 26 41 COc1cccc(/C=C/NC(=O)NCCc2cccc(OC)c2)c1 ZINC000217961402 EG For-Sale Unstable MTNR1A 117 60 COc1cccc(/C=C/NC(=O)NCCc2cccc(OC)c2)c1 ZINC000217961402 EG For-Sale Unstable MTNR1B 105 60 COc1cccc(/C=C/NC(=O)NCCc2cccc(OC)c2)c1 ZINC000217961402 EG For-Sale Unstable ROCK2 36 40 COc1cccc(/C=C/NC(=O)NCCc2cccc(OC)c2)c1 ZINC000217961402 EG For-Sale Unstable ABCG2 18 40 COc1cccc(/C=C/NC(=O)NCCc2cccc(OC)c2)c1 ZINC000217961402 EG For-Sale Unstable CRTM 55 39 O=C(O)/C=C\c1ccc(OCCN2CCC[C@H](O)C2)cc1 ZINC000217961421 CD For-Sale Unstable ESR1 70 38 O=C(O)/C=C\c1ccc(OCCN2CCC[C@H](O)C2)cc1 ZINC000217961421 CD For-Sale Unstable SLC6A1 122 39 O=C(O)/C=C\c1ccc(OCCN2CCC[C@H](O)C2)cc1 ZINC000217961421 CD For-Sale Unstable ESR2 47 38 O=C(O)/C=C\c1ccc(OCCN2CCC[C@H](O)C2)cc1 ZINC000217961421 CD For-Sale Unstable LTA4H 60 52 O=C(O)/C=C\c1ccc(OCCN2CCC[C@H](O)C2)cc1 ZINC000217961421 CD For-Sale Unstable HRH3 52 50 O=C(O)/C=C\c1ccc(OCCN2CCC[C@H](O)C2)cc1 ZINC000217961421 CD For-Sale Unstable PSMB2 53 41 O=C(O)/C=C\c1ccc(OCCN2CCC[C@H](O)C2)cc1 ZINC000217961421 CD For-Sale Unstable PSMB5 18 41 O=C(O)/C=C\c1ccc(OCCN2CCC[C@H](O)C2)cc1 ZINC000217961421 CD For-Sale Unstable PSMB1 47 41 CCC[C@@H](O)CNC(=O)[C@H](N)CC(=O)O ZINC000217961424 BB For-Sale Unstable DPP7 37 41 CCC[C@@H](O)CNC(=O)[C@H](N)CC(=O)O ZINC000217961424 BB For-Sale Unstable DPP8 32 40 CCC[C@@H](O)CNC(=O)[C@H](N)CC(=O)O ZINC000217961424 BB For-Sale Unstable DPP9 27 40 Nc1cc(S(=O)(=O)N2CCC[C@@H]3CCCC[C@H]32)ccc1Cl ZINC000217961431 EG For-Sale Unstable CASP3 67 37 Nc1cc(S(=O)(=O)N2CCC[C@@H]3CCCC[C@H]32)ccc1Cl ZINC000217961431 EG For-Sale Unstable CASP7 74 37 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000217961438 JF For-Sale Unstable NAMPT 16 40 O=C(CCc1c[nH]c2ccccc12)N1CCCC[C@H]1c1cccnc1 ZINC000217961453 EI In-Stock Unstable TACR2 29 44 O=C(CCc1c[nH]c2ccccc12)N1CCCC[C@H]1c1cccnc1 ZINC000217961453 EI In-Stock Unstable COLA 115 42 O=C(CCc1c[nH]c2ccccc12)N1CCCC[C@H]1c1cccnc1 ZINC000217961453 EI In-Stock Unstable GPBAR1 0 42 Fc1cc(N[C@@H]2C[C@H]3C[C@@H]2[C@@H]2CCC[C@@H]32)ccc1Cl ZINC000217961478 CJ For-Sale Unstable ENV 43 35 Cc1cc(C(=O)Nc2ccccc2Nc2ccccc2)c2c(C)noc2n1 ZINC000217961486 FJ On-Demand Unstable AKR1C2 42 37 Cc1cccc(-c2noc(CNC(=O)/C=C/c3ccc(Cl)cc3)n2)c1 ZINC000217961489 FI In-Stock Unstable BDKRB2 65 35 Cc1cccc(-c2noc(CNC(=O)/C=C/c3ccc(Cl)cc3)n2)c1 ZINC000217961489 FI In-Stock Unstable HDAC8 53 40 Cc1cccc(-c2noc(CNC(=O)/C=C/c3ccc(Cl)cc3)n2)c1 ZINC000217961489 FI In-Stock Unstable HDAC1 24 40 Cc1cccc(-c2noc(CNC(=O)/C=C/c3ccc(Cl)cc3)n2)c1 ZINC000217961489 FI In-Stock Unstable HDAC6 41 40 Cc1cccc(-c2noc(CNC(=O)/C=C/c3ccc(Cl)cc3)n2)c1 ZINC000217961489 FI In-Stock Unstable GRM5 17 41 CC(=O)c1ccc2c(c1)CCN2C=O ZINC000217961493 AD For-Sale Unstable SRD5A1 41 37 CC(=O)c1ccc2c(c1)CCN2C=O ZINC000217961493 AD For-Sale Unstable SRD5A2 40 37 CCC[C@H](O)CNC(=O)[C@H](N)CC(=O)O ZINC000217961505 BB For-Sale Unstable DPP7 37 41 CCC[C@H](O)CNC(=O)[C@H](N)CC(=O)O ZINC000217961505 BB For-Sale Unstable DPP8 32 40 CCC[C@H](O)CNC(=O)[C@H](N)CC(=O)O ZINC000217961505 BB For-Sale Unstable DPP9 27 40 Nc1cc(S(=O)(=O)N2CCC[C@H]3CCCC[C@H]32)ccc1Cl ZINC000217961508 EG For-Sale Unstable CASP3 67 37 Nc1cc(S(=O)(=O)N2CCC[C@H]3CCCC[C@H]32)ccc1Cl ZINC000217961508 EG For-Sale Unstable CASP7 74 37 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000217961514 JF For-Sale Unstable NAMPT 16 40 COc1cccc(/C=C/NC(=O)NCCc2cccc(F)c2)c1 ZINC000217961518 DG For-Sale Unstable MTNR1A 93 51 COc1cccc(/C=C/NC(=O)NCCc2cccc(F)c2)c1 ZINC000217961518 DG For-Sale Unstable MTNR1B 85 51 O=S(=O)(Nc1ccn2nccc2c1)c1ccccc1F ZINC000217961519 CE In-Stock Anodyne NR1I2 27 46 O=S(=O)(Nc1ccn2nccc2c1)c1ccccc1F ZINC000217961519 CE In-Stock Anodyne SGK1 33 41 COc1ccc2cc(/C=C\C(=O)CCl)ccc2c1 ZINC000217961542 CH For-Sale Unstable CYP1B1 55 43 COc1ccc2cc(/C=C\C(=O)CCl)ccc2c1 ZINC000217961542 CH For-Sale Unstable NQO2 31 43 COc1ccc2cc(/C=C\C(=O)CCl)ccc2c1 ZINC000217961542 CH For-Sale Unstable AHR 37 41 COc1ccc2cc(/C=C\C(=O)CCl)ccc2c1 ZINC000217961542 CH For-Sale Unstable MTNR1A 74 42 COc1ccc2cc(/C=C\C(=O)CCl)ccc2c1 ZINC000217961542 CH For-Sale Unstable MTNR1B 60 42 COc1ccc2cc(/C=C\C(=O)CCl)ccc2c1 ZINC000217961542 CH For-Sale Unstable CYP1A1 36 43 COc1ccc2cc(/C=C\C(=O)CCl)ccc2c1 ZINC000217961542 CH For-Sale Unstable AKR1C3 23 41 COc1ccc2cc(/C=C\C(=O)CCl)ccc2c1 ZINC000217961542 CH For-Sale Unstable PTPA 0 53 COc1ccc2cc(/C=C\C(=O)CCl)ccc2c1 ZINC000217961542 CH For-Sale Unstable ABCG2 18 48 COc1ccc2cc(/C=C\C(=O)CCl)ccc2c1 ZINC000217961542 CH For-Sale Unstable GPR183 0 41 Fc1cc(N[C@H]2C[C@H]3C[C@@H]2[C@@H]2CCC[C@@H]32)ccc1Cl ZINC000217961543 CJ For-Sale Unstable ENV 43 35 Cc1nnnn1-c1ccc(C(=O)N2CCCC[C@H]2c2cccnc2)cc1 ZINC000217961565 EF In-Stock Unstable CHRNA2 42 43 Cc1nnnn1-c1ccc(C(=O)N2CCCC[C@H]2c2cccnc2)cc1 ZINC000217961565 EF In-Stock Unstable CRTY 0 43 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccc(Cl)cc3)n2)cc1 ZINC000217961579 FH In-Stock Unstable PTGS2 0 40 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccc(Cl)cc3)n2)cc1 ZINC000217961579 FH In-Stock Unstable HDAC8 0 52 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccc(Cl)cc3)n2)cc1 ZINC000217961579 FH In-Stock Unstable HDAC1 0 41 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccc(Cl)cc3)n2)cc1 ZINC000217961579 FH In-Stock Unstable HDAC2 20 45 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccc(Cl)cc3)n2)cc1 ZINC000217961579 FH In-Stock Unstable PDK1 34 40 Nc1cccc(OCCN2CCC[C@@H]3CCCC[C@H]32)c1 ZINC000217961606 CG For-Sale Unstable LTA4H 19 51 Nc1cccc(OCCN2CCC[C@@H]3CCCC[C@H]32)c1 ZINC000217961606 CG For-Sale Unstable HRH3 29 41 Nc1cccc(OCCN2CCC[C@@H]3CCCC[C@H]32)c1 ZINC000217961606 CG For-Sale Unstable CHRNA10 78 38 O=C(/C=C\c1c[nH]c2cc(Br)ccc12)CCl ZINC000217961607 CH For-Sale Unstable TDO2 0 50 COc1cccc(/C=C/NC(=O)NCCc2cccc(Cl)c2)c1 ZINC000217961627 EH For-Sale Unstable DRD4 43 34 COc1cccc(/C=C/NC(=O)NCCc2cccc(Cl)c2)c1 ZINC000217961627 EH For-Sale Unstable MTNR1A 90 51 COc1cccc(/C=C/NC(=O)NCCc2cccc(Cl)c2)c1 ZINC000217961627 EH For-Sale Unstable MTNR1B 82 51 COc1cccc(/C=C/NC(=O)NCCc2cccc(Cl)c2)c1 ZINC000217961627 EH For-Sale Unstable LMGT2 0 42 CCC[C@@H](O)CNC(=O)[C@@H](N)CCCOC ZINC000217961628 BC For-Sale Unstable DPP7 35 48 O=S(=O)(Nc1ccn2nccc2c1)c1ccc(F)c(Cl)c1 ZINC000217961633 EF In-Stock Anodyne SCN9A 0 41 O=S(=O)(Nc1ccn2nccc2c1)c1ccc(F)c(Cl)c1 ZINC000217961633 EF In-Stock Anodyne PKM 15 43 CCc1ncnc(NCCCN2CCCC2)c1F ZINC000217961643 CE On-Demand Unstable HNMT 47 38 Nc1cccc(OCCN2CCC[C@H]3CCCC[C@H]32)c1 ZINC000217961679 CG For-Sale Unstable LTA4H 19 51 Nc1cccc(OCCN2CCC[C@H]3CCCC[C@H]32)c1 ZINC000217961679 CG For-Sale Unstable HRH3 29 41 Nc1cccc(OCCN2CCC[C@H]3CCCC[C@H]32)c1 ZINC000217961679 CG For-Sale Unstable CHRNA10 78 38 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccc(Cl)cc3)n2)c(OC)c1 ZINC000217961685 GH In-Stock Unstable PTGS2 29 44 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccc(Cl)cc3)n2)c(OC)c1 ZINC000217961685 GH In-Stock Unstable BDKRB2 49 34 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccc(Cl)cc3)n2)c(OC)c1 ZINC000217961685 GH In-Stock Unstable CYSP_PLAFA 42 36 COCOc1ccc([C@@H]2C[C@@H]2C(=O)O)cc1 ZINC000217961701 BD For-Sale Unstable FFAR1 19 51 CCC[C@H](O)CNC(=O)[C@@H](N)CCCOC ZINC000217961715 BC For-Sale Unstable DPP7 35 48 N#Cc1c(CN2CCN(Cc3cc(=O)n4ccsc4n3)CC2)cn2ccccc12 ZINC000217961718 HE On-Demand Unstable PKM 19 52 COc1cccc(/C=C/NC(=O)NCCc2cccc(Br)c2)c1 ZINC000217961731 GH For-Sale Unstable MTNR1A 90 51 COc1cccc(/C=C/NC(=O)NCCc2cccc(Br)c2)c1 ZINC000217961731 GH For-Sale Unstable MTNR1B 83 51 Cc1ccc(S(=O)(=O)N2CCC[C@@H]3CCCC[C@H]32)cc1N ZINC000217961772 DF For-Sale Unstable CASP3 71 38 Cc1ccc(S(=O)(=O)N2CCC[C@@H]3CCCC[C@H]32)cc1N ZINC000217961772 DF For-Sale Unstable CASP7 75 38 CN(Cc1ccccc1/C=C\C(=O)O)CC1CCCCC1 ZINC000217961780 CH For-Sale Unstable PTGER2 43 44 CN(Cc1ccccc1/C=C\C(=O)O)CC1CCCCC1 ZINC000217961780 CH For-Sale Unstable PTGER4 0 44 CN(Cc1ccccc1/C=C\C(=O)O)CC1CCCCC1 ZINC000217961780 CH For-Sale Unstable PTGER3 18 44 CN(Cc1ccccc1/C=C\C(=O)O)CC1CCCCC1 ZINC000217961780 CH For-Sale Unstable PTGDR 0 43 O=C(/C=C/c1ccc(Cl)cc1)NCc1nc(-c2ccccc2Cl)no1 ZINC000217961782 FI In-Stock Unstable HDAC8 0 41 O=C(/C=C/c1ccc(Cl)cc1)NCc1nc(-c2ccccc2Cl)no1 ZINC000217961782 FI In-Stock Unstable HDAC1 0 48 O=C(/C=C/c1ccc(Cl)cc1)NCc1nc(-c2ccccc2Cl)no1 ZINC000217961782 FI In-Stock Unstable HDAC2 16 48 CCC[C@@H](O)CNC(=O)[C@H](N)CCCOC ZINC000217961787 BC For-Sale Unstable DPP7 35 48 COCOc1ccc([C@H]2C[C@@H]2C(=O)O)cc1 ZINC000217961791 BD For-Sale Unstable FFAR1 19 51 COc1cccc(/C=C/NC(=O)NCCc2ccc(C)cc2)c1 ZINC000217961830 DH For-Sale Unstable DRD4 42 38 COc1cccc(/C=C/NC(=O)NCCc2ccc(C)cc2)c1 ZINC000217961830 DH For-Sale Unstable MTNR1A 98 47 COc1cccc(/C=C/NC(=O)NCCc2ccc(C)cc2)c1 ZINC000217961830 DH For-Sale Unstable MTNR1B 89 47 Cc1ccc(S(=O)(=O)N2CCC[C@H]3CCCC[C@H]32)cc1N ZINC000217961850 DF For-Sale Unstable CASP3 71 38 Cc1ccc(S(=O)(=O)N2CCC[C@H]3CCCC[C@H]32)cc1N ZINC000217961850 DF For-Sale Unstable CASP7 75 38 COCOc1ccc([C@@H]2C[C@H]2C(=O)O)cc1 ZINC000217961856 BD For-Sale Unstable FFAR1 19 51 CN(CCC#N)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217961862 CE For-Sale Unstable FDPS 23 40 CCC[C@H](O)CNC(=O)[C@H](N)CCCOC ZINC000217961872 BC For-Sale Unstable DPP7 35 48 O=C(/C=C/c1ccc(Cl)cc1)NCc1nc(-c2ccc(Cl)cc2)no1 ZINC000217961880 FI In-Stock Unstable PYGL 0 40 O=C(/C=C/c1ccc(Cl)cc1)NCc1nc(-c2ccc(Cl)cc2)no1 ZINC000217961880 FI In-Stock Unstable HDAC8 0 55 O=C(/C=C/c1ccc(Cl)cc1)NCc1nc(-c2ccc(Cl)cc2)no1 ZINC000217961880 FI In-Stock Unstable HDAC2 19 45 C[C@H]1C[C@H](C)CCN1Cc1ccc(CC(=O)NN)cc1 ZINC000217961886 CD For-Sale Unstable SIGMAR1 18 41 C[C@H]1C[C@H](C)CCN1Cc1ccc(CC(=O)NN)cc1 ZINC000217961886 CD For-Sale Unstable AOC2 0 40 COc1cccc(/C=C/NC(=O)NCCc2ccc(Cl)cc2)c1 ZINC000217961924 EH For-Sale Unstable DRD4 45 39 COc1cccc(/C=C/NC(=O)NCCc2ccc(Cl)cc2)c1 ZINC000217961924 EH For-Sale Unstable PTGS2 0 40 COc1cccc(/C=C/NC(=O)NCCc2ccc(Cl)cc2)c1 ZINC000217961924 EH For-Sale Unstable MTNR1A 93 46 COc1cccc(/C=C/NC(=O)NCCc2ccc(Cl)cc2)c1 ZINC000217961924 EH For-Sale Unstable MTNR1B 85 46 COc1cccc(/C=C/NC(=O)NCCc2ccc(Cl)cc2)c1 ZINC000217961924 EH For-Sale Unstable U38 0 40 COc1cccc(/C=C/NC(=O)NCCc2ccc(Cl)cc2)c1 ZINC000217961924 EH For-Sale Unstable NCE103 22 47 COc1cccc(/C=C/NC(=O)NCCc2ccc(Cl)cc2)c1 ZINC000217961924 EH For-Sale Unstable CAN2 0 47 CCCc1ccc(S(=O)(=O)Nc2ccn3nccc3c2)cc1 ZINC000217961925 DG In-Stock Unstable ADRB2 41 36 CCCc1ccc(S(=O)(=O)Nc2ccn3nccc3c2)cc1 ZINC000217961925 DG In-Stock Unstable ADRB3 51 36 CCCc1ccc(S(=O)(=O)Nc2ccn3nccc3c2)cc1 ZINC000217961925 DG In-Stock Unstable NR1I2 31 50 CCCc1ccc(S(=O)(=O)Nc2ccn3nccc3c2)cc1 ZINC000217961925 DG In-Stock Unstable LIMK2 40 37 COCOc1ccc([C@H]2C[C@H]2C(=O)O)cc1 ZINC000217961933 BD For-Sale Unstable FFAR1 19 51 O=C(CCc1ccc2c(c1)CCO2)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217961952 FE In-Stock Unstable CHRNA4 28 44 Nc1cccc(CN2CCC[C@@H]3CCCC[C@H]32)c1 ZINC000217961970 BG For-Sale Unstable SLC18A3 16 43 CCN1CCC(Nc2cc(Cl)nc(C3CC3)n2)CC1 ZINC000217961975 CF On-Demand Unstable CHRM3 17 47 CCN1CCC(Nc2cc(Cl)nc(C3CC3)n2)CC1 ZINC000217961975 CF On-Demand Unstable SSTR5 54 35 O=C(/C=C/c1ccc(Cl)cc1)NCc1nc(-c2cccc(Br)c2)no1 ZINC000217961978 HI In-Stock Unstable HDAC8 52 39 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cc(-c2ccc(F)cc2)n[nH]1 ZINC000217961980 IG For-Sale Unstable TACR3 23 48 C[C@H]1CCN(Cc2ccc(CC(=O)NN)cc2)[C@@H](C)C1 ZINC000217961983 CD For-Sale Unstable SIGMAR1 18 41 C[C@H]1CCN(Cc2ccc(CC(=O)NN)cc2)[C@@H](C)C1 ZINC000217961983 CD For-Sale Unstable AOC2 0 40 C[C@@H]1CCCN(Cc2ccc(/C=C\C(=O)O)cc2F)C1 ZINC000217961990 CG For-Sale Unstable SLC6A1 79 35 COC(=O)c1ccc(S(=O)(=O)Nc2ccn3nccc3c2)cc1 ZINC000217962026 ED In-Stock Unstable LIMK2 45 35 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cc(-c2ccc(F)cc2)n[nH]1 ZINC000217962045 IG For-Sale Unstable TACR3 23 48 O=C(O)c1csc(Nc2ccc3c(c2)CCCC3)n1 ZINC000217962048 CG For-Sale Unstable SPHK1 41 33 O=C(O)c1csc(Nc2ccc3c(c2)CCCC3)n1 ZINC000217962048 CG For-Sale Unstable TRPC6 83 47 O=C(O)c1csc(Nc2ccc3c(c2)CCCC3)n1 ZINC000217962048 CG For-Sale Unstable TRPC3 71 47 Nc1cccc(CN2CCC[C@H]3CCCC[C@H]32)c1 ZINC000217962049 BG For-Sale Unstable SLC18A3 16 43 COc1cccc(/C=C/NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217962059 GH For-Sale Unstable MTNR1A 95 46 COc1cccc(/C=C/NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217962059 GH For-Sale Unstable MTNR1B 86 46 COc1cccc(/C=C/NC(=O)NCCc2ccc(Br)cc2)c1 ZINC000217962059 GH For-Sale Unstable NCE103 15 42 CNC[C@@H](C)S(=O)(=O)NCc1ccc(C)cc1 ZINC000217962062 CD For-Sale Unstable GRIA4 18 42 C[C@@H](O)c1cc2n(n1)CCN(C(=O)CCn1c(=O)[nH]c3ccccc31)C2 ZINC000217962070 FD In-Stock Unstable PLD1 41 31 O=C(/C=C/c1ccc(Cl)cc1)NCc1nc(-c2cccs2)no1 ZINC000217962078 EH In-Stock Unstable ETHR 30 40 C[C@H]1CCCN(Cc2ccc(/C=C\C(=O)O)cc2F)C1 ZINC000217962093 CG For-Sale Unstable SLC6A1 79 35 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cc(-c2ccc(F)cc2)n[nH]1 ZINC000217962128 IG For-Sale Unstable TACR3 23 48 C[C@@H](C(=O)NN)c1ccc(CN2CC[C@@H](O)C2)cc1 ZINC000217962139 CC For-Sale Unstable MLNR 33 40 CNC[C@H](C)S(=O)(=O)NCc1ccc(C)cc1 ZINC000217962149 CD For-Sale Unstable GRIA4 18 42 C[C@H](O)c1cc2n(n1)CCN(C(=O)CCn1c(=O)[nH]c3ccccc31)C2 ZINC000217962158 FD In-Stock Unstable PLD1 41 31 COc1cccc(/C=C/NC(=O)Nc2ccc(C)nc2)c1 ZINC000217962162 CG For-Sale Unstable MTNR1A 22 46 COc1cccc(/C=C/NC(=O)Nc2ccc(C)nc2)c1 ZINC000217962162 CG For-Sale Unstable MTNR1B 29 46 CN(Cc1nc(-c2ccccc2)no1)C(=O)/C=C/c1ccc(Cl)cc1 ZINC000217962188 FI In-Stock Unstable FABI 41 31 CN(Cc1nc(-c2ccccc2)no1)C(=O)/C=C/c1ccc(Cl)cc1 ZINC000217962188 FI In-Stock Unstable TSPO 21 45 CN(Cc1nc(-c2ccccc2)no1)C(=O)/C=C/c1ccc(Cl)cc1 ZINC000217962188 FI In-Stock Unstable GPBAR1 19 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cc(-c2ccc(F)cc2)n[nH]1 ZINC000217962206 IG For-Sale Unstable TACR3 23 48 C[C@@H]1CCCN(Cc2ccc(F)cc2/C=C\C(=O)O)C1 ZINC000217962223 CG For-Sale Unstable SLC6A1 117 44 C[C@H](C(=O)NN)c1ccc(CN2CC[C@@H](O)C2)cc1 ZINC000217962229 CC For-Sale Unstable MLNR 33 40 CCOc1ccc(S(=O)(=O)Nc2ccn3nccc3c2)cc1F ZINC000217962236 EF In-Stock Unstable SCN9A 0 41 O=C(O)Cc1csc(Nc2ccc3c(c2)CCCC3)n1 ZINC000217962256 CG For-Sale Unstable COLA 17 41 O=C(O)Cc1csc(Nc2ccc3c(c2)CCCC3)n1 ZINC000217962256 CG For-Sale Unstable CPT1A 27 41 O=C(O)Cc1csc(Nc2ccc3c(c2)CCCC3)n1 ZINC000217962256 CG For-Sale Unstable CPT1B 36 41 O=C(O)Cc1csc(Nc2ccc3c(c2)CCCC3)n1 ZINC000217962256 CG For-Sale Unstable TRPC6 57 38 O=C(O)Cc1csc(Nc2ccc3c(c2)CCCC3)n1 ZINC000217962256 CG For-Sale Unstable TRPC3 56 38 COc1cccc(/C=C/NC(=O)Nc2ccc(C)cn2)c1 ZINC000217962267 CG For-Sale Unstable MTNR1A 19 41 COc1cccc(/C=C/NC(=O)Nc2ccc(C)cn2)c1 ZINC000217962267 CG For-Sale Unstable MTNR1B 26 41 COc1cccc(/C=C/NC(=O)Nc2ccc(C)cn2)c1 ZINC000217962267 CG For-Sale Unstable LUCI_LUCLA 20 54 C[C@H]1CCCN(Cc2ccc(F)cc2/C=C\C(=O)O)C1 ZINC000217962291 CG For-Sale Unstable SLC6A1 117 44 Cc1cccc(-c2noc(CN(C)C(=O)/C=C/c3ccc(Cl)cc3)n2)c1 ZINC000217962311 FI In-Stock Unstable FABI 41 31 Cc1cccc(-c2noc(CN(C)C(=O)/C=C/c3ccc(Cl)cc3)n2)c1 ZINC000217962311 FI In-Stock Unstable GRM5 17 41 Cc1cccc(-c2noc(CN(C)C(=O)/C=C/c3ccc(Cl)cc3)n2)c1 ZINC000217962311 FI In-Stock Unstable GPBAR1 15 46 C[C@H]1CN(C)[C@@H](C)C[C@@H]1Nc1ccc(Cl)c(F)c1 ZINC000217962324 CH For-Sale Unstable ENV 44 37 Cc1nc(Nc2ccc3c(c2)CCCC3)sc1C(=O)O ZINC000217962357 CH For-Sale Unstable DHODH 28 53 Cc1nc(Nc2ccc3c(c2)CCCC3)sc1C(=O)O ZINC000217962357 CH For-Sale Unstable TRPC6 57 36 Cc1nc(Nc2ccc3c(c2)CCCC3)sc1C(=O)O ZINC000217962357 CH For-Sale Unstable TRPC3 57 36 C[C@H](C(=O)NN)c1ccc(CN2CC[C@@H](C)C2)cc1 ZINC000217962412 CD For-Sale Unstable MLNR 44 42 Cc1ccc(-c2noc(CN(C)C(=O)/C=C/c3ccc(Cl)cc3)n2)cc1 ZINC000217962424 FI In-Stock Unstable TSPO 15 50 CCc1nc(C)ccc1OCC(=O)NCc1nnnn1-c1ccccc1 ZINC000217962484 FD In-Stock Unstable PLA2G2D 49 32 COc1cccc(/C=C/NC(=O)Nc2ccc(Br)cn2)c1 ZINC000217962488 EH For-Sale Unstable MTNR1A 17 40 COc1cccc(/C=C/NC(=O)Nc2ccc(Br)cn2)c1 ZINC000217962488 EH For-Sale Unstable MTNR1B 24 40 COc1cccc(/C=C/NC(=O)Nc2ccc(Br)cn2)c1 ZINC000217962488 EH For-Sale Unstable LUCI_LUCLA 17 40 COc1ccc2cc(/C=C3/CC(=O)NC3=O)ccc2c1 ZINC000217962521 CE For-Sale Unstable ESRRA 46 37 COc1ccc2cc(/C=C3/CC(=O)NC3=O)ccc2c1 ZINC000217962521 CE For-Sale Unstable CYP1B1 40 38 COc1ccc2cc(/C=C3/CC(=O)NC3=O)ccc2c1 ZINC000217962521 CE For-Sale Unstable HPGD 40 42 COc1cc2c(cc1OC)CN(C(=O)[C@@H]1CC[C@@H](Cn3cnnn3)CC1)CC2 ZINC000217962523 GE In-Stock Unstable ABCB1 0 41 CCCCN(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217962576 CF For-Sale Unstable THRA 46 44 CCCCN(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217962576 CF For-Sale Unstable FDPS 28 44 CCCCN(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217962576 CF For-Sale Unstable ACHE 0 45 CCCCN(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217962576 CF For-Sale Unstable PPARA 15 40 CCCCN(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217962576 CF For-Sale Unstable THRB 23 44 CCCCN(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217962576 CF For-Sale Unstable LTB4R 19 44 CCCCN(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217962576 CF For-Sale Unstable MTNR1A 16 40 CCCCN(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217962576 CF For-Sale Unstable PLA2G4B 62 40 CCCCN(C)CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217962576 CF For-Sale Unstable AKR1C3 35 43 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cn2)c1 ZINC000217962593 DH For-Sale Unstable F10 54 37 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cn2)c1 ZINC000217962593 DH For-Sale Unstable MTNR1A 17 40 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cn2)c1 ZINC000217962593 DH For-Sale Unstable MTNR1B 23 40 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cn2)c1 ZINC000217962593 DH For-Sale Unstable LUCI_LUCLA 32 40 COc1cccc(/C=C/NC(=O)Nc2ccc(Cl)cn2)c1 ZINC000217962593 DH For-Sale Unstable CYSP_PLAFA 42 34 CCc1ncnc(NCCCOc2ccccc2)c1F ZINC000217962621 CG On-Demand Unstable FOLP 0 43 O=C(Cc1ccc(O)c(Cl)c1)NCCc1cnccn1 ZINC000217962642 CD In-Stock Unstable NCE103 41 62 O=C(Cc1ccc(O)c(Cl)c1)NCCc1cnccn1 ZINC000217962642 CD In-Stock Unstable P96878_MYCTU 28 62 O=C(Cc1ccc(O)c(Cl)c1)NCCc1cnccn1 ZINC000217962642 CD In-Stock Unstable CAN2 0 62 COc1ccc(-c2noc(CN(C)C(=O)/C=C/c3ccc(Cl)cc3)n2)c(OC)c1 ZINC000217962646 HI In-Stock Unstable PTGS2 0 41 COc1ccc(-c2noc(CN(C)C(=O)/C=C/c3ccc(Cl)cc3)n2)c(OC)c1 ZINC000217962646 HI In-Stock Unstable CYSP_PLAFA 42 35 CC(=O)N1CCN(Cc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217962663 CD For-Sale Unstable DRD4 24 41 CC(=O)N1CCN(Cc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217962663 CD For-Sale Unstable ITGAL 16 41 CC(=O)N1CCN(Cc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217962663 CD For-Sale Unstable SIGMAR1 30 47 CC(=O)N1CCN(Cc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217962663 CD For-Sale Unstable FAAH 15 42 CC(=O)N1CCN(Cc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217962663 CD For-Sale Unstable MGLL 0 40 CC(=O)N1CCN(Cc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217962663 CD For-Sale Unstable AKR1C3 31 42 CC(=O)N1CCN(Cc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217962663 CD For-Sale Unstable GPR183 0 44 COc1cccc(/C=C2\Oc3c(ccc4c3[C@H](c3cc(OC)c(OC(C)=O)c(OC)c3)CC(=O)O4)C2=O)c1OC ZINC000217962710 KJ In-Stock Unstable MT-ND4 41 31 COc1cccc(/C=C/NC(=O)Nc2cc(Cl)ccn2)c1 ZINC000217962721 DH For-Sale Unstable TYK2 41 38 CN(Cc1nc(-c2ccccc2Cl)no1)C(=O)/C=C/c1ccc(Cl)cc1 ZINC000217962757 GJ In-Stock Unstable GPBAR1 33 42 CC(=O)N1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217962764 CD For-Sale Unstable ACHE 19 40 CC(=O)N1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217962764 CD For-Sale Unstable PTGER2 27 43 CC(=O)N1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217962764 CD For-Sale Unstable CHRM3 16 46 CC(=O)N1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217962764 CD For-Sale Unstable SIGMAR1 45 48 CC(=O)N1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217962764 CD For-Sale Unstable HDAC8 40 37 CC(=O)N1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217962764 CD For-Sale Unstable HDAC1 16 43 CC(=O)N1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217962764 CD For-Sale Unstable FAAH 27 45 CC(=O)N1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217962764 CD For-Sale Unstable MGLL 0 41 CC(=O)N1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217962764 CD For-Sale Unstable AKR1C3 33 41 CC(=O)N1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217962764 CD For-Sale Unstable GPR183 0 43 COc1cccc(/C=C2\Oc3c(ccc4c3[C@@H](c3cc(OC)c(OC(C)=O)c(OC)c3)CC(=O)O4)C2=O)c1OC ZINC000217962797 KJ In-Stock Unstable MT-ND4 41 31 COc1cccc(/C=C/NC(=O)Nc2cc(Br)ccn2)c1 ZINC000217962835 EH For-Sale Unstable MTNR1A 20 41 COc1cccc(/C=C/NC(=O)Nc2cc(Br)ccn2)c1 ZINC000217962835 EH For-Sale Unstable MTNR1B 27 41 O=C(O)/C=C\c1ccccc1CN1CCc2ccccc21 ZINC000217962844 CG For-Sale Unstable PTGER2 41 56 O=C(O)/C=C\c1ccccc1CN1CCc2ccccc21 ZINC000217962844 CG For-Sale Unstable PTGER4 0 56 O=C(O)/C=C\c1ccccc1CN1CCc2ccccc21 ZINC000217962844 CG For-Sale Unstable PTGER3 18 56 CCc1ncnc(NCc2ccc(C(F)(F)F)cc2)c1F ZINC000217962871 CH On-Demand Unstable PETD 0 43 CCc1ncnc(NCc2ccc(C(F)(F)F)cc2)c1F ZINC000217962871 CH On-Demand Unstable USP10 0 40 CCc1ncnc(NCc2ccc(C(F)(F)F)cc2)c1F ZINC000217962871 CH On-Demand Unstable USP13 0 40 COc1ccc(/C=C2/CC(=O)NC2=O)cc1C ZINC000217962872 BD For-Sale Unstable ESRRA 51 45 COc1ccc(/C=C2/CC(=O)NC2=O)cc1C ZINC000217962872 BD For-Sale Unstable HPGD 45 38 COc1ncccc1N[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217962893 CH For-Sale Unstable TRPM8 15 40 COC(=O)C[C@@H](c1oc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c1O)C(C)C ZINC000217962903 IE In-Stock Unstable CHRNA4 36 47 CCC[C@@H](O)CNC(=O)CNC(=O)CN ZINC000217962933 BA For-Sale Unstable UREB 0 45 COc1cccc(/C=C/NC(=O)NCCCc2ccccc2)c1 ZINC000217962934 DH For-Sale Unstable DRD4 41 32 COc1cccc(/C=C/NC(=O)NCCCc2ccccc2)c1 ZINC000217962934 DH For-Sale Unstable HRH2 34 42 COc1cccc(/C=C/NC(=O)NCCCc2ccccc2)c1 ZINC000217962934 DH For-Sale Unstable GRIN2B 0 42 COc1cccc(/C=C/NC(=O)NCCCc2ccccc2)c1 ZINC000217962934 DH For-Sale Unstable PTAFR 19 42 COc1cccc(/C=C/NC(=O)NCCCc2ccccc2)c1 ZINC000217962934 DH For-Sale Unstable G6PC 24 42 COc1cccc(/C=C/NC(=O)NCCCc2ccccc2)c1 ZINC000217962934 DH For-Sale Unstable SCN2A 17 46 COc1cccc(/C=C/NC(=O)NCCCc2ccccc2)c1 ZINC000217962934 DH For-Sale Unstable MTNR1A 120 60 COc1cccc(/C=C/NC(=O)NCCCc2ccccc2)c1 ZINC000217962934 DH For-Sale Unstable MTNR1B 115 60 COc1cccc(/C=C/NC(=O)NCCCc2ccccc2)c1 ZINC000217962934 DH For-Sale Unstable FAAH 21 45 COc1cccc(/C=C/NC(=O)NCCCc2ccccc2)c1 ZINC000217962934 DH For-Sale Unstable AMP1_PLAFQ 29 45 COc1cccc(/C=C/NC(=O)NCCCc2ccccc2)c1 ZINC000217962934 DH For-Sale Unstable AKR1C3 23 42 COc1cccc(/C=C/NC(=O)NCCCc2ccccc2)c1 ZINC000217962934 DH For-Sale Unstable CRTM 66 45 COc1cccc(/C=C/NC(=O)NCCCc2ccccc2)c1 ZINC000217962934 DH For-Sale Unstable PDS 48 40 COc1ncccc1N[C@H]1C[C@H](C)CC[C@@H]1C(C)C ZINC000217962972 CH For-Sale Unstable TRPM8 15 40 COC(=O)C[C@H](c1oc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c1O)C(C)C ZINC000217962983 IE In-Stock Unstable CHRNA4 28 46 COc1cc(CF)cc(Br)c1OC ZINC000217963007 BF For-Sale Unstable DRTS_TOXGO 40 33 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cc(-c2cc(OC)c(OC)c(OC)c2)n[nH]1 ZINC000217963013 JG For-Sale Unstable TACR3 21 45 CCC[C@H](O)CNC(=O)CNC(=O)CN ZINC000217963016 BA For-Sale Unstable UREB 0 45 COc1cccc(/C=C/NC(=O)NCCCCc2ccccc2)c1 ZINC000217963029 DH For-Sale Unstable DRD4 40 31 COc1cccc(/C=C/NC(=O)NCCCCc2ccccc2)c1 ZINC000217963029 DH For-Sale Unstable HRH2 30 41 COc1cccc(/C=C/NC(=O)NCCCCc2ccccc2)c1 ZINC000217963029 DH For-Sale Unstable DRD3 15 42 COc1cccc(/C=C/NC(=O)NCCCCc2ccccc2)c1 ZINC000217963029 DH For-Sale Unstable PTAFR 21 45 COc1cccc(/C=C/NC(=O)NCCCCc2ccccc2)c1 ZINC000217963029 DH For-Sale Unstable G6PC 23 41 COc1cccc(/C=C/NC(=O)NCCCCc2ccccc2)c1 ZINC000217963029 DH For-Sale Unstable SCN2A 15 50 COc1cccc(/C=C/NC(=O)NCCCCc2ccccc2)c1 ZINC000217963029 DH For-Sale Unstable MTNR1A 112 56 COc1cccc(/C=C/NC(=O)NCCCCc2ccccc2)c1 ZINC000217963029 DH For-Sale Unstable MTNR1B 107 56 COc1cccc(/C=C/NC(=O)NCCCCc2ccccc2)c1 ZINC000217963029 DH For-Sale Unstable FAAH 26 49 COc1cccc(/C=C/NC(=O)NCCCCc2ccccc2)c1 ZINC000217963029 DH For-Sale Unstable AMP1_PLAFQ 28 46 COc1cccc(/C=C/NC(=O)NCCCCc2ccccc2)c1 ZINC000217963029 DH For-Sale Unstable AKR1C3 23 41 COc1cccc(/C=C/NC(=O)NCCCCc2ccccc2)c1 ZINC000217963029 DH For-Sale Unstable CRTM 63 42 COc1cccc(/C=C/NC(=O)NCCCCc2ccccc2)c1 ZINC000217963029 DH For-Sale Unstable PDS 48 37 Cc1noc2nc(C(C)C)cc(C(=O)Nc3cccc(S(=O)(=O)NC(C)(C)C)c3)c12 ZINC000217963061 IH On-Demand Unstable KCNK3 40 35 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cc(-c2cc(OC)c(OC)c(OC)c2)n[nH]1 ZINC000217963083 JG For-Sale Unstable TACR3 21 45 C[C@@H](Oc1ccc2c(c1)OCO2)C(=O)N1CCN(c2cnccn2)CC1 ZINC000217963094 FD In-Stock Unstable SSTR3 109 40 COC(=O)C[C@@H](C1=C(O)C(=O)C([C@H](CC(=O)OC)c2ccncc2)=C(O)C1=O)c1ccncc1 ZINC000217963098 JE In-Stock Unstable KCNA5 32 40 CCC[C@@H]1CC[C@@H](C#N)[C@@H](S(=O)(=O)c2ccccc2)C1 ZINC000217963112 CH For-Sale Unstable CHRM3 47 37 CCOC(CNC(=O)N/C=C/c1cccc(OC)c1)OCC ZINC000217963140 DE For-Sale Unstable MTNR1A 54 43 CCOC(CNC(=O)N/C=C/c1cccc(OC)c1)OCC ZINC000217963140 DE For-Sale Unstable MTNR1B 53 43 C[C@]12C[C@@H]3C[C@](C)(C1)C[C@@](NCc1ccc(C(=O)O)cc1)(C3)C2 ZINC000217963144 DI In-Stock Unstable RARA 43 33 C[C@]12C[C@@H]3C[C@](C)(C1)C[C@@](NCc1ccc(C(=O)O)cc1)(C3)C2 ZINC000217963144 DI In-Stock Unstable RARG 47 34 C[C@]12C[C@@H]3C[C@](C)(C1)C[C@@](NCc1ccc(C(=O)O)cc1)(C3)C2 ZINC000217963144 DI In-Stock Unstable RXRG 52 37 C[C@]12C[C@@H]3C[C@](C)(C1)C[C@@](NCc1ccc(C(=O)O)cc1)(C3)C2 ZINC000217963144 DI In-Stock Unstable RARB 46 34 C[C@]12C[C@@H]3C[C@](C)(C1)C[C@@](NCc1ccc(C(=O)O)cc1)(C3)C2 ZINC000217963144 DI In-Stock Unstable RXRB 53 34 C[C@H](Oc1ccc2c(c1)OCO2)C(=O)N1CCN(c2cnccn2)CC1 ZINC000217963166 FD In-Stock Unstable SSTR3 109 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cc(-c2cc(OC)c(OC)c(OC)c2)n[nH]1 ZINC000217963170 JG For-Sale Unstable TACR3 21 45 COC(=O)C[C@H](C1=C(O)C(=O)C([C@H](CC(=O)OC)c2ccncc2)=C(O)C1=O)c1ccncc1 ZINC000217963185 JE In-Stock Unstable KCNA5 32 40 COc1cccc(/C=C/NC(=O)NCCC#N)c1 ZINC000217963234 BD For-Sale Unstable DRD4 43 33 COc1cccc(/C=C/NC(=O)NCCC#N)c1 ZINC000217963234 BD For-Sale Unstable MTNR1A 53 43 COc1cccc(/C=C/NC(=O)NCCC#N)c1 ZINC000217963234 BD For-Sale Unstable MTNR1B 47 41 Nc1ccc(S(=O)(=O)N2CCC[C@@H]3CCCC[C@H]32)cc1 ZINC000217963235 CF On-Demand Unstable CASP3 44 34 Nc1ccc(S(=O)(=O)N2CCC[C@@H]3CCCC[C@H]32)cc1 ZINC000217963235 CF On-Demand Unstable CASP7 51 34 Nc1ccc(S(=O)(=O)N2CCC[C@@H]3CCCC[C@H]32)cc1 ZINC000217963235 CF On-Demand Unstable AKR1C3 36 43 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cc(-c2cc(OC)c(OC)c(OC)c2)n[nH]1 ZINC000217963257 JG For-Sale Unstable TACR3 21 45 COC(=O)C[C@H](C1=C(O)C(=O)C([C@@H](CC(=O)OC)c2ccncc2)=C(O)C1=O)c1ccncc1 ZINC000217963283 JE In-Stock Unstable KCNA5 32 40 CCC[C@@H]1CC[C@H](C#N)[C@@H](S(=O)(=O)c2ccccc2)C1 ZINC000217963303 CH For-Sale Unstable CHRM3 47 37 CCC[C@@H](O)CNC(=O)CC1(CN)CCC1 ZINC000217963309 BC For-Sale Unstable CACNA2D1 23 40 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217963319 EK In-Stock Unstable PYGL 26 49 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217963319 EK In-Stock Unstable HDAC1 15 41 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217963319 EK In-Stock Unstable HDAC2 0 41 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217963319 EK In-Stock Unstable HDAC4 19 41 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217963319 EK In-Stock Unstable HDAC9 35 41 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217963319 EK In-Stock Unstable HDAC7 43 41 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217963319 EK In-Stock Unstable MMP1 0 41 CC(C)c1ccc(CCCNC(=O)/C=C/c2ccc(Cl)cc2)cc1 ZINC000217963319 EK In-Stock Unstable TRPM2 0 40 CC(C)(C)OC(=O)N1CCN(c2cc(Cl)nc(C3CC3)n2)CC1 ZINC000217963337 EG On-Demand Unstable GPR119 47 48 CCN1CCN(c2ccccc2NC(=O)c2cc(C(C)C)nc3onc(C)c23)CC1 ZINC000217963378 HI On-Demand Unstable KCNQ2 71 36 CCN1CCN(c2ccccc2NC(=O)c2cc(C(C)C)nc3onc(C)c23)CC1 ZINC000217963378 HI On-Demand Unstable NPY2R 47 38 CCOC(=O)c1ccc([C@@H]2CCN(C(=O)OC(C)(C)C)C2)cc1 ZINC000217963391 DH For-Sale Unstable GPR119 50 48 O=C(Cn1ncc2ccccc21)NCCc1noc(C2CCCC2)n1 ZINC000217963392 EE In-Stock Unstable SMO 48 36 CCC[C@H](O)CNC(=O)CC1(CN)CCC1 ZINC000217963405 BC For-Sale Unstable CACNA2D1 23 40 CN(CCCNC(=O)/C=C/c1ccc(Cl)cc1)c1ccccc1 ZINC000217963426 EH In-Stock Unstable DRD3 15 49 CN(CCCNC(=O)/C=C/c1ccc(Cl)cc1)c1ccccc1 ZINC000217963426 EH In-Stock Unstable PYGL 27 49 CN(CCCNC(=O)/C=C/c1ccc(Cl)cc1)c1ccccc1 ZINC000217963426 EH In-Stock Unstable HDAC8 0 42 CN(CCCNC(=O)/C=C/c1ccc(Cl)cc1)c1ccccc1 ZINC000217963426 EH In-Stock Unstable MMP2 17 48 CN(CCCNC(=O)/C=C/c1ccc(Cl)cc1)c1ccccc1 ZINC000217963426 EH In-Stock Unstable HDAC1 23 42 CN(CCCNC(=O)/C=C/c1ccc(Cl)cc1)c1ccccc1 ZINC000217963426 EH In-Stock Unstable HDAC2 21 42 CN(CCCNC(=O)/C=C/c1ccc(Cl)cc1)c1ccccc1 ZINC000217963426 EH In-Stock Unstable HDAC3 16 42 CN(CCCNC(=O)/C=C/c1ccc(Cl)cc1)c1ccccc1 ZINC000217963426 EH In-Stock Unstable HDAC4 24 42 CN(CCCNC(=O)/C=C/c1ccc(Cl)cc1)c1ccccc1 ZINC000217963426 EH In-Stock Unstable HDAC6 23 40 CN(CCCNC(=O)/C=C/c1ccc(Cl)cc1)c1ccccc1 ZINC000217963426 EH In-Stock Unstable HDAC9 42 42 CN(CCCNC(=O)/C=C/c1ccc(Cl)cc1)c1ccccc1 ZINC000217963426 EH In-Stock Unstable HDAC7 54 42 CN(CCCNC(=O)/C=C/c1ccc(Cl)cc1)c1ccccc1 ZINC000217963426 EH In-Stock Unstable MMP1 0 48 COc1cccc(/C=C/NC(=O)N2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000217963447 HE For-Sale Unstable MMP13 30 40 COc1cccc(/C=C/NC(=O)N2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000217963447 HE For-Sale Unstable MMP3 35 40 COc1cccc(/C=C/NC(=O)N2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000217963447 HE For-Sale Unstable MMP9 28 40 COc1cccc(/C=C/NC(=O)N2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000217963447 HE For-Sale Unstable PKM 18 44 COc1cccc(/C=C/NC(=O)N2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000217963447 HE For-Sale Unstable TGM2 64 39 COc1cccc(/C=C/NC(=O)N2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000217963447 HE For-Sale Unstable MMP7 40 38 COc1cccc(/C=C/NC(=O)N2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000217963447 HE For-Sale Unstable MMP1 31 40 COc1cccc(/C=C/NC(=O)N2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000217963447 HE For-Sale Unstable F13A1 85 39 COc1cccc(/C=C/NC(=O)N2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000217963447 HE For-Sale Unstable AKR1C3 47 41 CCOC(=O)c1ccc([C@H]2CCN(C(=O)OC(C)(C)C)C2)cc1 ZINC000217963473 DH For-Sale Unstable GPR119 50 48 CCOc1ccccc1C(=O)Nc1sc2c(c1-c1nc(C)no1)CCOC2 ZINC000217963490 GH In-Stock Unstable HCN1 49 35 CCOc1ccccc1C(=O)Nc1sc2c(c1-c1nc(C)no1)CCOC2 ZINC000217963490 GH In-Stock Unstable HCN4 40 31 O=C1C/C(=C/c2ccc(C(F)(F)F)cc2)C(=O)N1 ZINC000217963520 CE For-Sale Unstable PRKCA 22 40 COc1cccc(/C=C/NC(=O)N2CCN(S(=O)(=O)c3ccc(C)cc3)CC2)c1 ZINC000217963530 HF For-Sale Unstable MMP13 30 41 COc1cccc(/C=C/NC(=O)N2CCN(S(=O)(=O)c3ccc(C)cc3)CC2)c1 ZINC000217963530 HF For-Sale Unstable MMP3 35 41 COc1cccc(/C=C/NC(=O)N2CCN(S(=O)(=O)c3ccc(C)cc3)CC2)c1 ZINC000217963530 HF For-Sale Unstable MMP9 24 41 COc1cccc(/C=C/NC(=O)N2CCN(S(=O)(=O)c3ccc(C)cc3)CC2)c1 ZINC000217963530 HF For-Sale Unstable PKM 18 41 COc1cccc(/C=C/NC(=O)N2CCN(S(=O)(=O)c3ccc(C)cc3)CC2)c1 ZINC000217963530 HF For-Sale Unstable TGM2 64 38 COc1cccc(/C=C/NC(=O)N2CCN(S(=O)(=O)c3ccc(C)cc3)CC2)c1 ZINC000217963530 HF For-Sale Unstable MMP1 28 41 COc1cccc(/C=C/NC(=O)N2CCN(S(=O)(=O)c3ccc(C)cc3)CC2)c1 ZINC000217963530 HF For-Sale Unstable F13A1 79 39 O=C(/C=C/c1ccc(Cl)cc1)NCCCN1CCCc2ccccc21 ZINC000217963547 FI In-Stock Unstable DRD3 26 55 O=C(/C=C/c1ccc(Cl)cc1)NCCCN1CCCc2ccccc21 ZINC000217963547 FI In-Stock Unstable PYGL 27 42 C[C@@H](C(=O)NN)c1ccc(CN2CCC[C@@H](N)C2)cc1 ZINC000217963591 CC For-Sale Unstable BIRC2 44 35 CC[C@@H]1CCCN(Cc2ccccc2/C=C\C(=O)O)C1 ZINC000217963630 CG For-Sale Unstable SLC6A1 142 42 CC[C@@H]1CCCN(Cc2ccccc2/C=C\C(=O)O)C1 ZINC000217963630 CG For-Sale Unstable PTGER2 32 42 CC[C@@H]1CCCN(Cc2ccccc2/C=C\C(=O)O)C1 ZINC000217963630 CG For-Sale Unstable PTGER4 0 42 CC[C@@H]1CCCN(Cc2ccccc2/C=C\C(=O)O)C1 ZINC000217963630 CG For-Sale Unstable SIGMAR1 15 41 COC(=O)N1CCN(C(=O)N/C=C/c2cccc(OC)c2)CC1 ZINC000217963632 DD For-Sale Unstable DRD4 41 31 COC(=O)N1CCN(C(=O)N/C=C/c2cccc(OC)c2)CC1 ZINC000217963632 DD For-Sale Unstable MTNR1A 33 41 COC(=O)N1CCN(C(=O)N/C=C/c2cccc(OC)c2)CC1 ZINC000217963632 DD For-Sale Unstable MTNR1B 41 41 COC(=O)N1CCN(C(=O)N/C=C/c2cccc(OC)c2)CC1 ZINC000217963632 DD For-Sale Unstable AKR1C2 44 34 COc1ccccc1/C=C/C(=O)Nc1ccc(CSc2ccccc2)cc1 ZINC000217963655 GK In-Stock Unstable PTGER2 33 40 COc1ccccc1/C=C/C(=O)Nc1ccc(CSc2ccccc2)cc1 ZINC000217963655 GK In-Stock Unstable PTGER4 23 40 COc1ccccc1/C=C/C(=O)Nc1ccc(CSc2ccccc2)cc1 ZINC000217963655 GK In-Stock Unstable PTGER3 17 40 COc1ccccc1/C=C/C(=O)Nc1ccc(CSc2ccccc2)cc1 ZINC000217963655 GK In-Stock Unstable MMP2 15 47 COc1ccccc1/C=C/C(=O)Nc1ccc(CSc2ccccc2)cc1 ZINC000217963655 GK In-Stock Unstable METAP2 0 42 C[C@@H](CNC(=O)c1cc(N)n[nH]1)N(C)C1CC1 ZINC000217963657 BC For-Sale Unstable ALPL 45 40 C[C@H](C(=O)NN)c1ccc(CN2CCC[C@@H](N)C2)cc1 ZINC000217963669 CC For-Sale Unstable BIRC2 44 35 O=C(CCCN1Cc2ccccc2C1=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217963672 GE In-Stock Unstable CHRNA4 31 57 CCOc1cc(/C=C2/CC(=O)NC2=O)ccc1OC(F)F ZINC000217963676 CE For-Sale Unstable ESRRA 40 41 CCOc1cc(/C=C2/CC(=O)NC2=O)ccc1OC(F)F ZINC000217963676 CE For-Sale Unstable HPGD 48 35 C1=C(c2ccccc2)CCN(C[C@@H]2[C@H]3CNC[C@H]32)C1 ZINC000217963704 CE In-Stock Unstable PARP1 0 44 CC[C@H]1CCCN(Cc2ccccc2/C=C\C(=O)O)C1 ZINC000217963720 CG For-Sale Unstable SLC6A1 142 42 CC[C@H]1CCCN(Cc2ccccc2/C=C\C(=O)O)C1 ZINC000217963720 CG For-Sale Unstable PTGER2 32 42 CC[C@H]1CCCN(Cc2ccccc2/C=C\C(=O)O)C1 ZINC000217963720 CG For-Sale Unstable PTGER4 0 42 CC[C@H]1CCCN(Cc2ccccc2/C=C\C(=O)O)C1 ZINC000217963720 CG For-Sale Unstable SIGMAR1 15 41 C[C@H](CNC(=O)c1cc(N)n[nH]1)N(C)C1CC1 ZINC000217963731 BC For-Sale Unstable ALPL 45 40 CCOC(=O)N(CCN)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217963735 DD For-Sale Unstable MTNR1A 26 43 CCOC(=O)N(CCN)C(=O)N/C=C/c1cccc(OC)c1 ZINC000217963735 DD For-Sale Unstable MTNR1B 31 43 CC[C@@H]1CC[C@@H](C#N)[C@@H](S(=O)(=O)c2ccccc2)C1 ZINC000217963757 CG For-Sale Unstable CHRM3 45 33 COc1ccccc1/C=C/C(=O)NCCSCc1cccc(C)c1 ZINC000217963765 EI In-Stock Unstable DRD3 15 48 O=C1C/C(=C/c2cccc3ccccc23)C(=O)N1 ZINC000217963766 BE For-Sale Unstable CHAT 59 33 CC[C@@H]1CCCN(Cc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217963826 CG For-Sale Unstable SLC6A1 57 33 CC[C@@H]1CCCN(Cc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217963826 CG For-Sale Unstable SIGMAR1 27 45 COc1ccc(NC(=O)c2cc(-c3ccc(C)cc3)nc3onc(C)c23)c([N+](=O)[O-])c1 ZINC000217963834 HJ On-Demand Unstable AKR1C2 18 42 O=C(/C=C\c1ccc2c(c1)OCCO2)CCl ZINC000217963843 BE For-Sale Unstable ITGAL 17 43 O=C(/C=C\c1ccc2c(c1)OCCO2)CCl ZINC000217963843 BE For-Sale Unstable PLK1 19 47 O=C(/C=C\c1ccc2c(c1)OCCO2)CCl ZINC000217963843 BE For-Sale Unstable DYRK2 40 34 CCOC(=O)NCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217963848 DD For-Sale Unstable DRD4 41 32 CCOC(=O)NCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217963848 DD For-Sale Unstable MTNR1A 72 48 CCOC(=O)NCCNC(=O)N/C=C/c1cccc(OC)c1 ZINC000217963848 DD For-Sale Unstable MTNR1B 67 48 COc1ccccc1/C=C/C(=O)NCCSCc1ccc(Cl)cc1Cl ZINC000217963866 GK In-Stock Unstable DRD3 15 45 COc1ccccc1/C=C/C(=O)NCCSCc1ccc(Cl)cc1Cl ZINC000217963866 GK In-Stock Unstable CYSP_PLAFA 41 42 C[C@@H](C(=O)NN)c1ccc(CN2CCC[C@@H](O)C2)cc1 ZINC000217963893 CC For-Sale Unstable MLNR 28 41 C[C@@H](C(=O)NN)c1ccc(CN2CCC[C@@H](O)C2)cc1 ZINC000217963893 CC For-Sale Unstable BIRC2 44 35 CC[C@@H]1CC[C@H](C#N)[C@@H](S(=O)(=O)c2ccccc2)C1 ZINC000217963898 CG For-Sale Unstable CHRM3 45 33 CCCOc1ccc(/C=C\C(=O)CCl)cc1OCCC ZINC000217963913 CI For-Sale Unstable APP 18 41 CCCOc1ccc(/C=C\C(=O)CCl)cc1OCCC ZINC000217963913 CI For-Sale Unstable AKR1C3 28 46 CC[C@H](C(=O)Nc1sc2c(c1-c1nc(C)no1)CCOC2)c1ccccc1 ZINC000217963915 GI In-Stock Unstable KCNQ2 41 35 CC[C@H]1CCCN(Cc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217963916 CG For-Sale Unstable SLC6A1 57 33 CC[C@H]1CCCN(Cc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217963916 CG For-Sale Unstable SIGMAR1 27 45 COc1ccccc1/C=C/C(=O)NCCSCc1ccc(Cl)c(Cl)c1 ZINC000217963971 GK In-Stock Unstable DRD3 16 46 COc1ccccc1/C=C/C(=O)NCCSCc1ccc(Cl)c(Cl)c1 ZINC000217963971 GK In-Stock Unstable PYGL 22 52 COc1ccccc1/C=C/C(=O)NCCSCc1ccc(Cl)c(Cl)c1 ZINC000217963971 GK In-Stock Unstable CYSP_PLAFA 42 36 COc1ccc2c(ccn2CCNC(=O)Cn2c(C)nc3cc(OC)c(OC)cc3c2=O)c1 ZINC000217963973 JF In-Stock Unstable AVPR1B 43 40 COc1ccc2c(ccn2CCNC(=O)Cn2c(C)nc3cc(OC)c(OC)cc3c2=O)c1 ZINC000217963973 JF In-Stock Unstable MTNR1A 32 41 COc1ccc2c(ccn2CCNC(=O)Cn2c(C)nc3cc(OC)c(OC)cc3c2=O)c1 ZINC000217963973 JF In-Stock Unstable MTNR1B 26 41 COc1ccc2c(ccn2CCNC(=O)Cn2c(C)nc3cc(OC)c(OC)cc3c2=O)c1 ZINC000217963973 JF In-Stock Unstable POLR1A 50 30 C[C@H](C(=O)NN)c1ccc(CN2CCC[C@@H](O)C2)cc1 ZINC000217963982 CC For-Sale Unstable MLNR 28 41 C[C@H](C(=O)NN)c1ccc(CN2CCC[C@@H](O)C2)cc1 ZINC000217963982 CC For-Sale Unstable BIRC2 44 35 CC[C@@H](C(=O)Nc1sc2c(c1-c1nc(C)no1)CCOC2)c1ccccc1 ZINC000217963996 GI In-Stock Unstable KCNQ2 41 35 CC[C@@H]1CCCN(Cc2ccc(/C=C\C(=O)O)cc2F)C1 ZINC000217964027 CH For-Sale Unstable SLC6A1 61 36 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cc(-c2ccc3c(c2)OCO3)n[nH]1 ZINC000217964056 JF For-Sale Unstable TACR3 20 43 COc1cccc(/C=C/NC(=O)NCCNC(=O)OC(C)(C)C)c1 ZINC000217964060 EE For-Sale Unstable DRD4 42 32 COc1cccc(/C=C/NC(=O)NCCNC(=O)OC(C)(C)C)c1 ZINC000217964060 EE For-Sale Unstable NQO2 24 40 COc1cccc(/C=C/NC(=O)NCCNC(=O)OC(C)(C)C)c1 ZINC000217964060 EE For-Sale Unstable MTNR1A 71 43 COc1cccc(/C=C/NC(=O)NCCNC(=O)OC(C)(C)C)c1 ZINC000217964060 EE For-Sale Unstable MTNR1B 68 43 COc1ccccc1/C=C/C(=O)NCCSCc1ccco1 ZINC000217964077 DG In-Stock Unstable DRD3 15 47 COc1ccc(Br)cc1/C=C\C(=O)CCl ZINC000217964078 CG For-Sale Unstable TNFRSF1A 26 60 COc1ccc(Br)cc1/C=C\C(=O)CCl ZINC000217964078 CG For-Sale Unstable CYSP_PLAFA 52 42 Nc1ccc(OCCN2CCC[C@@H]3CCCC[C@H]32)cc1 ZINC000217964100 CG For-Sale Unstable LTA4H 51 42 Nc1ccc(OCCN2CCC[C@@H]3CCCC[C@H]32)cc1 ZINC000217964100 CG For-Sale Unstable HRH3 47 42 Nc1ccc(OCCN2CCC[C@@H]3CCCC[C@H]32)cc1 ZINC000217964100 CG For-Sale Unstable PSMB2 46 37 Nc1ccc(OCCN2CCC[C@@H]3CCCC[C@H]32)cc1 ZINC000217964100 CG For-Sale Unstable PSMB1 41 37 CCOC(=O)c1ccc([C@@H]2CCCN(C(=O)OC(C)(C)C)C2)cc1 ZINC000217964101 EH For-Sale Unstable GPR119 44 45 CC[C@H]1CCCN(Cc2ccc(/C=C\C(=O)O)cc2F)C1 ZINC000217964108 CH For-Sale Unstable SLC6A1 61 36 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cc(-c2ccc3c(c2)OCO3)n[nH]1 ZINC000217964138 JF For-Sale Unstable TACR3 20 43 Nc1ccc(OCCN2CCC[C@H]3CCCC[C@H]32)cc1 ZINC000217964184 CG For-Sale Unstable LTA4H 51 42 Nc1ccc(OCCN2CCC[C@H]3CCCC[C@H]32)cc1 ZINC000217964184 CG For-Sale Unstable HRH3 47 42 Nc1ccc(OCCN2CCC[C@H]3CCCC[C@H]32)cc1 ZINC000217964184 CG For-Sale Unstable PSMB2 46 37 Nc1ccc(OCCN2CCC[C@H]3CCCC[C@H]32)cc1 ZINC000217964184 CG For-Sale Unstable PSMB1 41 37 COc1cccc(/C=C/NC(=O)N2CCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000217964186 FF For-Sale Unstable DRD4 40 31 CCOC(=O)c1ccc([C@H]2CCCN(C(=O)OC(C)(C)C)C2)cc1 ZINC000217964197 EH For-Sale Unstable GPR119 44 45 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cc(-c2ccc3c(c2)OCO3)n[nH]1 ZINC000217964214 JF For-Sale Unstable TACR3 20 43 COc1ccccc1/C=C/C(=O)Nc1cc([N+](=O)[O-])ccc1Cl ZINC000217964215 EH In-Stock Unstable EPHX1 0 45 COc1ccccc1/C=C/C(=O)Nc1cc([N+](=O)[O-])ccc1Cl ZINC000217964215 EH In-Stock Unstable KCNMA1 22 47 COc1ccccc1/C=C/C(=O)Nc1cc([N+](=O)[O-])ccc1Cl ZINC000217964215 EH In-Stock Unstable TRPM8 0 60 COc1ccccc1/C=C/C(=O)Nc1cc([N+](=O)[O-])ccc1Cl ZINC000217964215 EH In-Stock Unstable CYSP_PLAFA 43 35 COc1ccc(/C=C\C(=O)CCl)c2ccccc12 ZINC000217964249 CH For-Sale Unstable CYSP_PLAFA 59 44 CCc1ncnc(NCC[C@@H]2CCCO2)c1F ZINC000217964269 BE On-Demand Unstable TNK2 46 35 Nc1ccccc1OCCCC(=O)OCc1ccccc1 ZINC000217964281 CG For-Sale Unstable PTGER2 22 40 Nc1ccccc1OCCCC(=O)OCc1ccccc1 ZINC000217964281 CG For-Sale Unstable PPIA 42 34 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cc(-c2ccc3c(c2)OCO3)n[nH]1 ZINC000217964282 JF For-Sale Unstable TACR3 20 43 COc1cccc(/C=C/NC(=O)NC2CCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000217964308 GG For-Sale Unstable MTNR1A 18 40 COc1cccc(/C=C/NC(=O)NC2CCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000217964308 GG For-Sale Unstable MTNR1B 22 40 COc1cccc(/C=C/NC(=O)NC2CCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000217964308 GG For-Sale Unstable EPHX2 36 42 COc1cccc(/C=C/NC(=O)NC2CCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000217964308 GG For-Sale Unstable GPR119 37 42 COc1ccccc1/C=C/C(=O)NCc1cccc(OC(C)C)c1 ZINC000217964323 EH In-Stock Unstable ANPEP 19 42 COc1ccccc1/C=C/C(=O)NCc1cccc(OC(C)C)c1 ZINC000217964323 EH In-Stock Unstable PDS 45 33 COc1ccc(Cl)cc1CC(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217964348 CE On-Demand Unstable QRFPR 40 39 CCc1ncnc(NCC[C@H]2CCCO2)c1F ZINC000217964352 BE On-Demand Unstable TNK2 46 35 CN(Cc1ccccc1/C=C\C(=O)O)C1CCCCCC1 ZINC000217964374 CH For-Sale Unstable PTGER2 49 50 CN(Cc1ccccc1/C=C\C(=O)O)C1CCCCCC1 ZINC000217964374 CH For-Sale Unstable PTGER4 23 50 CN(Cc1ccccc1/C=C\C(=O)O)C1CCCCCC1 ZINC000217964374 CH For-Sale Unstable PTGER3 18 50 CN(Cc1ccccc1/C=C\C(=O)O)C1CCCCCC1 ZINC000217964374 CH For-Sale Unstable AMY2 44 31 CN(Cc1ccccc1/C=C\C(=O)O)C1CCCCCC1 ZINC000217964374 CH For-Sale Unstable PTGDR 0 48 NCCCCOc1ccccc1N ZINC000217964389 AD For-Sale Unstable TAAR1 15 42 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cc(-c2ccccc2OC)n[nH]1 ZINC000217964400 IG For-Sale Unstable TACR3 18 43 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cc(-c2ccccc2OC)n[nH]1 ZINC000217964400 IG For-Sale Unstable ALPL 44 34 COc1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1OC ZINC000217964406 DH For-Sale Unstable HTR2A 15 43 COc1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1OC ZINC000217964406 DH For-Sale Unstable PDGFRA 34 43 COc1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1OC ZINC000217964406 DH For-Sale Unstable IMPDH2 0 40 COc1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1OC ZINC000217964406 DH For-Sale Unstable ENPP1 69 33 COc1ccc(Cl)cc1CC(=O)N[C@H]1CCC[C@@H]1CO ZINC000217964425 CE For-Sale Unstable CPT1A 40 38 COc1ccc(Cl)cc1CC(=O)N[C@H]1CCC[C@@H]1CO ZINC000217964425 CE For-Sale Unstable QRFPR 40 39 CCOc1ccc(CNC(=O)/C=C/c2ccccc2OC)cc1OCC ZINC000217964428 FH In-Stock Unstable PTGER4 24 45 CCOc1ccc(CNC(=O)/C=C/c2ccccc2OC)cc1OCC ZINC000217964428 FH In-Stock Unstable PTGER3 16 40 CN(Cc1ccc(/C=C\C(=O)O)cc1)C1CCCCCC1 ZINC000217964459 CH For-Sale Unstable NR1H4 32 44 CCc1ncnc(NCC2CC2)c1F ZINC000217964478 AE On-Demand Unstable KHK 69 39 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cc(-c2ccccc2OC)n[nH]1 ZINC000217964488 IG For-Sale Unstable TACR3 18 43 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cc(-c2ccccc2OC)n[nH]1 ZINC000217964488 IG For-Sale Unstable ALPL 44 34 COc1ccc(Cl)cc1CC(=O)N[C@@H]1CCC[C@H]1CO ZINC000217964495 CE For-Sale Unstable CPT1A 40 38 COc1ccc(Cl)cc1CC(=O)N[C@@H]1CCC[C@H]1CO ZINC000217964495 CE For-Sale Unstable QRFPR 40 39 Cc1cc(C(=O)NCCc2cn[nH]c2)ccc1N1CCOCC1 ZINC000217964503 DD In-Stock Unstable DRD4 42 32 COC(=O)C[C@H](c1ccc(OC)cc1)c1cc2c(cc1O)OCO2 ZINC000217964513 EF In-Stock Unstable EDNRB 65 39 COC(=O)C[C@H](c1ccc(OC)cc1)c1cc2c(cc1O)OCO2 ZINC000217964513 EF In-Stock Unstable EDNRA 61 39 COC(=O)C[C@H](c1ccc(OC)cc1)c1cc2c(cc1O)OCO2 ZINC000217964513 EF In-Stock Unstable BMP1 53 44 COC(=O)C[C@H](c1ccc(OC)cc1)c1cc2c(cc1O)OCO2 ZINC000217964513 EF In-Stock Unstable RORC 55 41 COc1ccccc1/C=C/C(=O)NCc1ccc(OC(C)C)c(OC)c1 ZINC000217964556 FH In-Stock Unstable PTGER2 23 42 COc1ccccc1/C=C/C(=O)NCc1ccc(OC(C)C)c(OC)c1 ZINC000217964556 FH In-Stock Unstable PTGER4 18 42 Cn1c(=O)n(C)c2cc(/C=C\C(=O)CCl)ccc21 ZINC000217964563 CD For-Sale Unstable BRPF1 0 44 CCOC1CCN(Cc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217964566 CF For-Sale Unstable HRH1 19 40 CCOC1CCN(Cc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217964566 CF For-Sale Unstable SIGMAR1 41 50 CCOC1CCN(Cc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217964566 CF For-Sale Unstable SSTR5 51 38 CCOC1CCN(Cc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217964566 CF For-Sale Unstable CCR3 16 40 CCOC1CCN(Cc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217964566 CF For-Sale Unstable TIMP3 61 32 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cc(-c2ccccc2OC)n[nH]1 ZINC000217964569 IG For-Sale Unstable TACR3 18 43 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cc(-c2ccccc2OC)n[nH]1 ZINC000217964569 IG For-Sale Unstable ALPL 44 34 COc1ccc(Cl)cc1CC(=O)N[C@H]1CCC[C@H]1CO ZINC000217964583 CE For-Sale Unstable CPT1A 40 38 COc1ccc(Cl)cc1CC(=O)N[C@H]1CCC[C@H]1CO ZINC000217964583 CE For-Sale Unstable QRFPR 40 39 O=C(O)[C@@H]1C[C@@H]2CCCC[C@@H]2N1C(=O)NCC1CC1 ZINC000217964601 CD On-Demand Unstable ACE 16 60 COC(=O)C[C@@H](c1ccc(OC)cc1)c1cc2c(cc1O)OCO2 ZINC000217964605 EF In-Stock Unstable EDNRB 65 39 COC(=O)C[C@@H](c1ccc(OC)cc1)c1cc2c(cc1O)OCO2 ZINC000217964605 EF In-Stock Unstable EDNRA 61 39 COC(=O)C[C@@H](c1ccc(OC)cc1)c1cc2c(cc1O)OCO2 ZINC000217964605 EF In-Stock Unstable BMP1 53 44 COC(=O)C[C@@H](c1ccc(OC)cc1)c1cc2c(cc1O)OCO2 ZINC000217964605 EF In-Stock Unstable RORC 55 41 C[C@H](C(=O)NN)c1ccc(CN2CCN(C)[C@@H](C)C2)cc1 ZINC000217964648 CC For-Sale Unstable MLNR 27 41 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cc(-c2ccccc2OC)n[nH]1 ZINC000217964655 IG For-Sale Unstable TACR3 18 43 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cc(-c2ccccc2OC)n[nH]1 ZINC000217964655 IG For-Sale Unstable ALPL 44 34 COc1ccccc1/C=C/C(=O)NCCCc1ccccc1Cl ZINC000217964662 EI In-Stock Unstable DRD3 26 56 COc1ccccc1/C=C/C(=O)NCCCc1ccccc1Cl ZINC000217964662 EI In-Stock Unstable PTGER2 31 43 COc1ccccc1/C=C/C(=O)NCCCc1ccccc1Cl ZINC000217964662 EI In-Stock Unstable PYGL 0 41 CN1CCN(C)[C@@H](CC(=O)NCCc2cccc(Oc3ccccc3)c2)C1 ZINC000217964668 FF In-Stock Unstable FDFT1 23 52 CN1CCN(C)[C@@H](CC(=O)NCCc2cccc(Oc3ccccc3)c2)C1 ZINC000217964668 FF In-Stock Unstable AMP1_PLAFQ 36 40 CN1CCN(C)[C@@H](CC(=O)NCCc2cccc(Oc3ccccc3)c2)C1 ZINC000217964668 FF In-Stock Unstable CRTM 36 41 O=C(O)[C@@H]1C[C@H]2CCCC[C@@H]2N1C(=O)NCC1CC1 ZINC000217964677 CD On-Demand Unstable ACE 16 60 CCOC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217964686 CF For-Sale Unstable CHRM2 15 40 CCOC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217964686 CF For-Sale Unstable DRD2 21 40 CCOC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217964686 CF For-Sale Unstable DRD4 44 41 CCOC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217964686 CF For-Sale Unstable ACHE 38 42 CCOC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217964686 CF For-Sale Unstable HRH1 21 42 CCOC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217964686 CF For-Sale Unstable CHRM3 24 40 CCOC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217964686 CF For-Sale Unstable SIGMAR1 48 50 CCOC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217964686 CF For-Sale Unstable SSTR5 64 36 CCOC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217964686 CF For-Sale Unstable CCR3 25 42 CCOC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217964686 CF For-Sale Unstable TIMP3 64 33 CCOC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217964686 CF For-Sale Unstable AKR1C3 39 44 CCc1ncnc(NCc2ccc(O)cc2)c1F ZINC000217964698 BE On-Demand Unstable HTT 0 40 CCc1ncnc(NCc2ccc(O)cc2)c1F ZINC000217964698 BE On-Demand Unstable USP10 0 42 CCc1ncnc(NCc2ccc(O)cc2)c1F ZINC000217964698 BE On-Demand Unstable USP13 0 42 O=C(N/C=C/c1cccc(F)c1)Nc1cccc(C(=O)O)c1 ZINC000217964754 DG For-Sale Anodyne CCR3 15 41 O=C(N/C=C/c1cccc(F)c1)Nc1cccc(C(=O)O)c1 ZINC000217964754 DG For-Sale Anodyne AKR1C3 34 49 O=C(N/C=C/c1cccc(F)c1)Nc1cccc(C(=O)O)c1 ZINC000217964754 DG For-Sale Anodyne KCNK3 59 46 O=C(N/C=C/c1cccc(F)c1)Nc1cccc(C(=O)O)c1 ZINC000217964754 DG For-Sale Anodyne KCNK9 23 40 COc1ccccc1/C=C/C(=O)NCCCc1ccc(Cl)cc1 ZINC000217964762 EI In-Stock Unstable DRD3 27 55 COc1ccccc1/C=C/C(=O)NCCCc1ccc(Cl)cc1 ZINC000217964762 EI In-Stock Unstable PTGER2 21 41 COc1ccccc1/C=C/C(=O)NCCCc1ccc(Cl)cc1 ZINC000217964762 EI In-Stock Unstable HDAC7 30 41 COc1ccccc1/C=C/C(=O)NCCCc1ccc(Cl)cc1 ZINC000217964762 EI In-Stock Unstable AKR1B10 33 42 COc1ccccc1/C=C/C(=O)NCCCc1ccc(Cl)cc1 ZINC000217964762 EI In-Stock Unstable CYSP_PLAFA 40 40 C[C@H](C(=O)NN)c1ccc(CN2CCC[C@@H](C)CC2)cc1 ZINC000217964794 CE For-Sale Unstable HRH3 19 50 C[C@H](C(=O)NN)c1ccc(CN2CCC[C@@H](C)CC2)cc1 ZINC000217964794 CE For-Sale Unstable SIGMAR1 27 40 C[C@H](C(=O)NN)c1ccc(CN2CCC[C@@H](C)CC2)cc1 ZINC000217964794 CE For-Sale Unstable BIRC2 46 35 C[C@@H]1CCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217964801 CF For-Sale Unstable ESR1 25 45 C[C@@H]1CCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217964801 CF For-Sale Unstable HRH2 32 40 C[C@@H]1CCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217964801 CF For-Sale Unstable SLC6A1 63 34 C[C@@H]1CCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217964801 CF For-Sale Unstable ESR2 18 45 C[C@@H]1CCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217964801 CF For-Sale Unstable LTA4H 27 43 C[C@@H]1CCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217964801 CF For-Sale Unstable HRH3 20 45 C[C@@H]1CCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217964801 CF For-Sale Unstable SIGMAR1 18 41 C[C@@H]1CCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217964801 CF For-Sale Unstable EBP 24 41 Nc1nc(/C=C\c2ccc(F)cc2)cs1 ZINC000217964804 BG For-Sale Unstable AHR 15 41 Nc1ccc(OCCCN2CCC[C@@H]3CCCC[C@H]32)cc1 ZINC000217964843 CH For-Sale Unstable HTR3A 24 44 Nc1ccc(OCCCN2CCC[C@@H]3CCCC[C@H]32)cc1 ZINC000217964843 CH For-Sale Unstable HRH3 78 49 Nc1ccc(OCCCN2CCC[C@@H]3CCCC[C@H]32)cc1 ZINC000217964843 CH For-Sale Unstable MEN1 40 34 COc1ccccc1/C=C/C(=O)NCCCc1ccc(F)cc1 ZINC000217964875 DH In-Stock Unstable DRD2 18 56 COc1ccccc1/C=C/C(=O)NCCCc1ccc(F)cc1 ZINC000217964875 DH In-Stock Unstable DRD3 30 56 COc1ccccc1/C=C/C(=O)NCCCc1ccc(F)cc1 ZINC000217964875 DH In-Stock Unstable PTGER2 24 41 COc1ccccc1/C=C/C(=O)NCCCc1ccc(F)cc1 ZINC000217964875 DH In-Stock Unstable PTGER4 0 41 COc1ccccc1/C=C/C(=O)NCCCc1ccc(F)cc1 ZINC000217964875 DH In-Stock Unstable PTGER3 15 41 COc1ccccc1/C=C/C(=O)NCCCc1ccc(F)cc1 ZINC000217964875 DH In-Stock Unstable MTNR1B 20 42 COc1ccccc1/C=C/C(=O)NCCCc1ccc(F)cc1 ZINC000217964875 DH In-Stock Unstable AKR1B10 34 43 C[C@H]1CCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217964894 CF For-Sale Unstable ESR1 25 45 C[C@H]1CCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217964894 CF For-Sale Unstable HRH2 32 40 C[C@H]1CCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217964894 CF For-Sale Unstable SLC6A1 63 34 C[C@H]1CCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217964894 CF For-Sale Unstable ESR2 18 45 C[C@H]1CCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217964894 CF For-Sale Unstable LTA4H 27 43 C[C@H]1CCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217964894 CF For-Sale Unstable HRH3 20 45 C[C@H]1CCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217964894 CF For-Sale Unstable SIGMAR1 18 41 C[C@H]1CCN(CCOc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217964894 CF For-Sale Unstable EBP 24 41 O=C(N[C@H]1CCC[C@H]1CO)[C@@H]1CC(=O)N(C2CCCC2)C1 ZINC000217964930 CD On-Demand Unstable INHA 47 48 Nc1ccc(OCCCN2CCC[C@H]3CCCC[C@H]32)cc1 ZINC000217964932 CH For-Sale Unstable HTR3A 24 44 Nc1ccc(OCCCN2CCC[C@H]3CCCC[C@H]32)cc1 ZINC000217964932 CH For-Sale Unstable HRH3 78 49 Nc1ccc(OCCCN2CCC[C@H]3CCCC[C@H]32)cc1 ZINC000217964932 CH For-Sale Unstable MEN1 40 34 O=C(N/C=C/c1cccc(F)c1)Nc1cccc(O)c1 ZINC000217964973 CG For-Sale Anodyne MMP1 0 61 COc1ccccc1/C=C/C(=O)NCCCc1ccccc1OC ZINC000217964981 EG In-Stock Unstable DRD2 18 59 COc1ccccc1/C=C/C(=O)NCCCc1ccccc1OC ZINC000217964981 EG In-Stock Unstable DRD3 31 59 COc1ccccc1/C=C/C(=O)NCCCc1ccccc1OC ZINC000217964981 EG In-Stock Unstable PTGER2 33 46 COc1ccccc1/C=C/C(=O)NCCCc1ccccc1OC ZINC000217964981 EG In-Stock Unstable PTGER4 0 46 COc1ccccc1/C=C/C(=O)NCCCc1ccccc1OC ZINC000217964981 EG In-Stock Unstable MTNR1B 40 44 COc1ccccc1/C=C/C(=O)NCCCc1ccccc1OC ZINC000217964981 EG In-Stock Unstable AKR1B10 28 41 Nc1cccc(CS(=O)(=O)N2CCC[C@@H]3CCCC[C@H]32)c1 ZINC000217965014 DF For-Sale Unstable FKBP1A 15 40 CN[C@@H](Cc1cc(Br)ccc1OC)[C@@H]1CCC[C@@H](C)C1 ZINC000217965041 EI For-Sale Unstable QRFPR 41 34 C[C@@H](OCc1ccccc1)C(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217965052 CD On-Demand Unstable CAPNS1 43 30 C[C@@H](OCc1ccccc1)C(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217965052 CD On-Demand Unstable CAPN2 55 34 C[C@@H](OCc1ccccc1)C(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217965052 CD On-Demand Unstable POL 0 43 C[C@@H](OCc1ccccc1)C(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217965052 CD On-Demand Unstable NPR 45 31 C[C@@H](OCc1ccccc1)C(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217965052 CD On-Demand Unstable Q9NBD4_PLAFA 0 40 C[C@@H](OCc1ccccc1)C(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217965052 CD On-Demand Unstable Q9NAW4_PLAFA 23 40 C[C@@H](N[C@H]1CCCC[C@@H]1c1ccccc1)[C@@H]1CCCO1 ZINC000217965058 CH For-Sale Unstable GRIA4 18 47 Cc1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217965083 CH For-Sale Unstable KIT 27 40 Cc1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217965083 CH For-Sale Unstable KDR 18 40 Cc1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217965083 CH For-Sale Unstable IMPDH2 0 41 Cc1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217965083 CH For-Sale Unstable TEK 22 40 Cc1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217965083 CH For-Sale Unstable IDO1 15 42 COc1cccc(CCCNC(=O)/C=C/c2ccccc2OC)c1 ZINC000217965099 EG In-Stock Unstable DRD2 15 53 COc1cccc(CCCNC(=O)/C=C/c2ccccc2OC)c1 ZINC000217965099 EG In-Stock Unstable DRD4 41 32 COc1cccc(CCCNC(=O)/C=C/c2ccccc2OC)c1 ZINC000217965099 EG In-Stock Unstable DRD3 30 53 COc1cccc(CCCNC(=O)/C=C/c2ccccc2OC)c1 ZINC000217965099 EG In-Stock Unstable PTGER2 32 44 COc1cccc(CCCNC(=O)/C=C/c2ccccc2OC)c1 ZINC000217965099 EG In-Stock Unstable PTAFR 25 48 COc1cccc(CCCNC(=O)/C=C/c2ccccc2OC)c1 ZINC000217965099 EG In-Stock Unstable CYP1B1 36 43 COc1cccc(CCCNC(=O)/C=C/c2ccccc2OC)c1 ZINC000217965099 EG In-Stock Unstable MTNR1A 63 60 COc1cccc(CCCNC(=O)/C=C/c2ccccc2OC)c1 ZINC000217965099 EG In-Stock Unstable MTNR1B 57 60 COc1cccc(CCCNC(=O)/C=C/c2ccccc2OC)c1 ZINC000217965099 EG In-Stock Unstable ABCB1 0 40 COc1cccc(CCCNC(=O)/C=C/c2ccccc2OC)c1 ZINC000217965099 EG In-Stock Unstable CYP1A2 16 43 COc1cccc(CCCNC(=O)/C=C/c2ccccc2OC)c1 ZINC000217965099 EG In-Stock Unstable AMP1_PLAFQ 19 41 COc1cccc(CCCNC(=O)/C=C/c2ccccc2OC)c1 ZINC000217965099 EG In-Stock Unstable ABCG2 25 42 COc1cccc(CCCNC(=O)/C=C/c2ccccc2OC)c1 ZINC000217965099 EG In-Stock Unstable CRTM 67 50 COc1cccc(CCCNC(=O)/C=C/c2ccccc2OC)c1 ZINC000217965099 EG In-Stock Unstable AKR1B10 33 43 COc1cccc(CCCNC(=O)/C=C/c2ccccc2OC)c1 ZINC000217965099 EG In-Stock Unstable CYSP_PLAFA 39 40 Nc1cccc(CS(=O)(=O)N2CCC[C@H]3CCCC[C@H]32)c1 ZINC000217965101 DF For-Sale Unstable FKBP1A 15 40 CN[C@@H](Cc1cc(Br)ccc1OC)[C@H]1CCC[C@@H](C)C1 ZINC000217965108 EI For-Sale Unstable QRFPR 41 34 CCS(=O)(=O)Nc1ccc([N+](=O)[O-])cc1O ZINC000217965125 BD For-Sale Unstable KCNMA1 19 40 C[C@H](OCc1ccccc1)C(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217965135 CD On-Demand Unstable CASP3 15 42 C[C@H](OCc1ccccc1)C(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217965135 CD On-Demand Unstable CAPNS1 43 30 C[C@H](OCc1ccccc1)C(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217965135 CD On-Demand Unstable CAPN2 55 34 C[C@H](OCc1ccccc1)C(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217965135 CD On-Demand Unstable POL 0 43 C[C@H](OCc1ccccc1)C(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217965135 CD On-Demand Unstable NPR 45 31 C[C@H](OCc1ccccc1)C(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217965135 CD On-Demand Unstable Q9NBD4_PLAFA 0 40 C[C@H](OCc1ccccc1)C(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217965135 CD On-Demand Unstable Q9NAW4_PLAFA 23 40 C[C@H](N[C@H]1CCCC[C@@H]1c1ccccc1)[C@@H]1CCCO1 ZINC000217965146 CH For-Sale Unstable GRIA4 18 47 CCOC(=O)c1ccc(OCc2cnn(-c3ccccc3)c2)cc1 ZINC000217965148 DH On-Demand Unstable SRD5A2 0 40 CCOC(=O)c1ccc(OCc2cnn(-c3ccccc3)c2)cc1 ZINC000217965148 DH On-Demand Unstable GRM4 26 43 CCOC(=O)c1ccc(OCc2cnn(-c3ccccc3)c2)cc1 ZINC000217965148 DH On-Demand Unstable F2RL3 20 43 N[C@H](CN1CCN2C(=O)NC[C@@H]2C1)C(=O)O ZINC000217965201 BA For-Sale Unstable GRIK5 49 33 Nc1cccc(OCCCN2CCC[C@@H]3CCCC[C@H]32)c1 ZINC000217965205 CH For-Sale Unstable HTR3A 15 42 Nc1cccc(OCCCN2CCC[C@@H]3CCCC[C@H]32)c1 ZINC000217965205 CH For-Sale Unstable HRH3 57 42 Nc1cccc(OCCCN2CCC[C@@H]3CCCC[C@H]32)c1 ZINC000217965205 CH For-Sale Unstable CHRNA10 77 38 COc1ccc(CCCNC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217965215 EG In-Stock Unstable DRD2 18 56 COc1ccc(CCCNC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217965215 EG In-Stock Unstable DRD3 31 56 COc1ccc(CCCNC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217965215 EG In-Stock Unstable PTGER2 28 46 COc1ccc(CCCNC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217965215 EG In-Stock Unstable PTAFR 21 47 COc1ccc(CCCNC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217965215 EG In-Stock Unstable PTGER4 19 43 COc1ccc(CCCNC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217965215 EG In-Stock Unstable CYP1B1 31 43 COc1ccc(CCCNC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217965215 EG In-Stock Unstable PTGER3 20 46 COc1ccc(CCCNC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217965215 EG In-Stock Unstable SCN2A 15 43 COc1ccc(CCCNC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217965215 EG In-Stock Unstable MTNR1A 48 36 COc1ccc(CCCNC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217965215 EG In-Stock Unstable MTNR1B 45 43 COc1ccc(CCCNC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217965215 EG In-Stock Unstable ABCG2 23 42 COc1ccc(CCCNC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217965215 EG In-Stock Unstable CRTM 40 38 COc1ccc(CCCNC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217965215 EG In-Stock Unstable AKR1B10 37 43 Nc1cccc(OCCCN2CCC[C@H]3CCCC[C@H]32)c1 ZINC000217965277 CH For-Sale Unstable HTR3A 15 42 Nc1cccc(OCCCN2CCC[C@H]3CCCC[C@H]32)c1 ZINC000217965277 CH For-Sale Unstable HRH3 57 42 Nc1cccc(OCCCN2CCC[C@H]3CCCC[C@H]32)c1 ZINC000217965277 CH For-Sale Unstable CHRNA10 77 38 Cc1c(OC(C)C)ncc(OCc2ccccc2)c1C(=O)O ZINC000217965327 DG For-Sale Unstable PPIA 43 33 Cc1c(OC(C)C)ncc(OCc2ccccc2)c1C(=O)O ZINC000217965327 DG For-Sale Unstable PTGER1 45 43 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217965330 EG In-Stock Unstable PTGER2 0 41 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217965330 EG In-Stock Unstable PTAFR 15 42 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217965330 EG In-Stock Unstable PTGER4 0 41 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217965330 EG In-Stock Unstable SDH1 0 40 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217965330 EG In-Stock Unstable CYP1B1 30 43 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217965330 EG In-Stock Unstable KCNQ2 48 34 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217965330 EG In-Stock Unstable UL26 23 40 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217965330 EG In-Stock Unstable U53 0 40 COc1ccc(OC[C@@H](C)NC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217965330 EG In-Stock Unstable SCAF_EBVB9 15 40 O=C1CCC/C1=C/c1ccc(OCc2ccccc2)cc1 ZINC000217965370 CI For-Sale Unstable MAOA 17 54 O=C1CCC/C1=C/c1ccc(OCc2ccccc2)cc1 ZINC000217965370 CI For-Sale Unstable MAOB 41 54 O=C1CCC/C1=C/c1ccc(OCc2ccccc2)cc1 ZINC000217965370 CI For-Sale Unstable LTA4H 17 43 O=C1CCC/C1=C/c1ccc(OCc2ccccc2)cc1 ZINC000217965370 CI For-Sale Unstable TRY1_BOVIN 44 38 O=C1CCC/C1=C/c1ccc(OCc2ccccc2)cc1 ZINC000217965370 CI For-Sale Unstable FFAR1 18 41 O=C1CCC/C1=C/c1ccc(OCc2ccccc2)cc1 ZINC000217965370 CI For-Sale Unstable HPGD 53 49 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217965412 EG In-Stock Unstable PTGER2 0 41 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217965412 EG In-Stock Unstable PTAFR 15 42 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217965412 EG In-Stock Unstable PTGER4 0 41 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217965412 EG In-Stock Unstable SDH1 0 40 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217965412 EG In-Stock Unstable CYP1B1 30 43 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217965412 EG In-Stock Unstable KCNQ2 48 34 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217965412 EG In-Stock Unstable UL26 23 40 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217965412 EG In-Stock Unstable U53 0 40 COc1ccc(OC[C@H](C)NC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217965412 EG In-Stock Unstable SCAF_EBVB9 15 40 CCCCN(Cc1ccccc1/C=C\C(=O)O)C1CC1 ZINC000217965415 CH For-Sale Unstable PTGER2 41 46 CCCCN(Cc1ccccc1/C=C\C(=O)O)C1CC1 ZINC000217965415 CH For-Sale Unstable PTGER4 0 46 CCCCN(Cc1ccccc1/C=C\C(=O)O)C1CC1 ZINC000217965415 CH For-Sale Unstable PTGER3 16 46 CCCCN(Cc1ccccc1/C=C\C(=O)O)C1CC1 ZINC000217965415 CH For-Sale Unstable PTGDR 0 42 Cc1ccc(F)c(C(=O)N[C@@H]2CCC[C@@H]2CO)c1 ZINC000217965423 CE On-Demand Unstable SSTR3 24 42 COC(=O)c1c(OCc2ccccc2)cnc(OC(C)C)c1C ZINC000217965450 DH For-Sale Unstable PPIA 45 36 COC(=O)c1c(OCc2ccccc2)cnc(OC(C)C)c1C ZINC000217965450 DH For-Sale Unstable PTGER1 40 39 CC(=O)Nc1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217965508 DH For-Sale Unstable IMPDH2 0 42 CC(=O)Nc1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217965508 DH For-Sale Unstable IDO1 30 49 Cc1ccc(F)c(C(=O)N[C@H]2CCC[C@@H]2CO)c1 ZINC000217965510 CE For-Sale Unstable SSTR3 25 42 COCCN(Cc1ccccc1/C=C\C(=O)O)C1CC1 ZINC000217965522 CE For-Sale Unstable PTGER2 47 46 COCCN(Cc1ccccc1/C=C\C(=O)O)C1CC1 ZINC000217965522 CE For-Sale Unstable PTGER4 23 46 COCCN(Cc1ccccc1/C=C\C(=O)O)C1CC1 ZINC000217965522 CE For-Sale Unstable PTGER3 18 46 COCCN(Cc1ccccc1/C=C\C(=O)O)C1CC1 ZINC000217965522 CE For-Sale Unstable PTGDR 16 41 COc1ccccc1/C=C/C(=O)Nc1ccccc1C(=O)c1ccccc1 ZINC000217965524 FJ In-Stock Unstable LTB4R 0 46 COc1ccccc1/C=C/C(=O)Nc1ccccc1C(=O)c1ccccc1 ZINC000217965524 FJ In-Stock Unstable MMP2 19 59 COc1ccccc1/C=C/C(=O)Nc1ccccc1C(=O)c1ccccc1 ZINC000217965524 FJ In-Stock Unstable MMP9 17 59 COc1ccccc1/C=C/C(=O)Nc1ccccc1C(=O)c1ccccc1 ZINC000217965524 FJ In-Stock Unstable HDA106 0 47 COc1ccccc1/C=C/C(=O)Nc1ccccc1C(=O)c1ccccc1 ZINC000217965524 FJ In-Stock Unstable TRPM2 0 41 COc1ccccc1/C=C/C(=O)Nc1ccccc1C(=O)c1ccccc1 ZINC000217965524 FJ In-Stock Unstable CYSP_PLAFA 42 35 CCCCCOc1ccc(/C=C2/CC(=O)NC2=O)cc1 ZINC000217965565 CF For-Sale Unstable PLA2G4B 87 37 CCCCCOc1ccc(/C=C2/CC(=O)NC2=O)cc1 ZINC000217965565 CF For-Sale Unstable HPGD 80 43 Cc1ccc(F)c(C(=O)N[C@@H]2CCC[C@H]2CO)c1 ZINC000217965596 CE For-Sale Unstable SSTR3 25 42 COc1ccccc1/C=C/C(=O)NCCCc1cccc(OC(C)C)c1 ZINC000217965619 FI In-Stock Unstable DRD3 20 50 COc1ccccc1/C=C/C(=O)NCCCc1cccc(OC(C)C)c1 ZINC000217965619 FI In-Stock Unstable PTGER2 23 41 COc1ccccc1/C=C/C(=O)NCCCc1cccc(OC(C)C)c1 ZINC000217965619 FI In-Stock Unstable PTAFR 24 46 COc1ccccc1/C=C/C(=O)NCCCc1cccc(OC(C)C)c1 ZINC000217965619 FI In-Stock Unstable PTGER4 0 41 COc1ccccc1/C=C/C(=O)NCCCc1cccc(OC(C)C)c1 ZINC000217965619 FI In-Stock Unstable MTNR1A 24 50 COc1ccccc1/C=C/C(=O)NCCCc1cccc(OC(C)C)c1 ZINC000217965619 FI In-Stock Unstable MTNR1B 25 42 COc1ccccc1/C=C/C(=O)NCCCc1cccc(OC(C)C)c1 ZINC000217965619 FI In-Stock Unstable AMP1_PLAFQ 19 40 COc1ccccc1/C=C/C(=O)NCCCc1cccc(OC(C)C)c1 ZINC000217965619 FI In-Stock Unstable CRTM 59 49 COc1ccccc1/C=C/C(=O)NCCCc1cccc(OC(C)C)c1 ZINC000217965619 FI In-Stock Unstable AKR1B10 28 40 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217965635 EF For-Sale Anodyne IDO1 25 47 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(S(=O)(=O)O)cc1 ZINC000217965635 EF For-Sale Anodyne P96878_MYCTU 45 41 COc1ccccc1-c1ccc(S(=O)(=O)N[C@H](C(=O)O)C(C)C)cc1 ZINC000217965659 FF On-Demand Unstable MMP13 89 69 COc1ccccc1-c1ccc(S(=O)(=O)N[C@H](C(=O)O)C(C)C)cc1 ZINC000217965659 FF On-Demand Unstable CA14 17 40 COc1ccccc1-c1ccc(S(=O)(=O)N[C@H](C(=O)O)C(C)C)cc1 ZINC000217965659 FF On-Demand Unstable MMP2 78 69 COc1ccccc1-c1ccc(S(=O)(=O)N[C@H](C(=O)O)C(C)C)cc1 ZINC000217965659 FF On-Demand Unstable MMP3 42 69 COc1ccccc1-c1ccc(S(=O)(=O)N[C@H](C(=O)O)C(C)C)cc1 ZINC000217965659 FF On-Demand Unstable MMP8 44 67 COc1ccccc1-c1ccc(S(=O)(=O)N[C@H](C(=O)O)C(C)C)cc1 ZINC000217965659 FF On-Demand Unstable MMP14 38 59 COc1ccccc1-c1ccc(S(=O)(=O)N[C@H](C(=O)O)C(C)C)cc1 ZINC000217965659 FF On-Demand Unstable CAPN1 22 42 COc1ccccc1-c1ccc(S(=O)(=O)N[C@H](C(=O)O)C(C)C)cc1 ZINC000217965659 FF On-Demand Unstable MMP9 46 67 COc1ccccc1-c1ccc(S(=O)(=O)N[C@H](C(=O)O)C(C)C)cc1 ZINC000217965659 FF On-Demand Unstable MMP12 116 48 COc1ccccc1-c1ccc(S(=O)(=O)N[C@H](C(=O)O)C(C)C)cc1 ZINC000217965659 FF On-Demand Unstable MMP7 32 50 COc1ccccc1-c1ccc(S(=O)(=O)N[C@H](C(=O)O)C(C)C)cc1 ZINC000217965659 FF On-Demand Unstable ADAMTS4 98 54 COc1ccccc1-c1ccc(S(=O)(=O)N[C@H](C(=O)O)C(C)C)cc1 ZINC000217965659 FF On-Demand Unstable MMP1 25 50 COc1ccccc1-c1ccc(S(=O)(=O)N[C@H](C(=O)O)C(C)C)cc1 ZINC000217965659 FF On-Demand Unstable LEF 31 50 C[C@H]1CN(Cc2ccc([C@H](C)C(=O)NN)cc2)C[C@@H](C)S1 ZINC000217965675 DE For-Sale Unstable MLNR 15 41 Cc1ccc(F)c(C(=O)N[C@H]2CCC[C@H]2CO)c1 ZINC000217965683 CE For-Sale Unstable SSTR3 25 42 COc1ccccc1-c1ccc(S(=O)(=O)N[C@@H](C(=O)O)C(C)C)cc1 ZINC000217965730 FF On-Demand Unstable MMP13 89 69 COc1ccccc1-c1ccc(S(=O)(=O)N[C@@H](C(=O)O)C(C)C)cc1 ZINC000217965730 FF On-Demand Unstable CA14 17 40 COc1ccccc1-c1ccc(S(=O)(=O)N[C@@H](C(=O)O)C(C)C)cc1 ZINC000217965730 FF On-Demand Unstable MMP2 78 69 COc1ccccc1-c1ccc(S(=O)(=O)N[C@@H](C(=O)O)C(C)C)cc1 ZINC000217965730 FF On-Demand Unstable MMP3 42 69 COc1ccccc1-c1ccc(S(=O)(=O)N[C@@H](C(=O)O)C(C)C)cc1 ZINC000217965730 FF On-Demand Unstable MMP8 44 67 COc1ccccc1-c1ccc(S(=O)(=O)N[C@@H](C(=O)O)C(C)C)cc1 ZINC000217965730 FF On-Demand Unstable MMP14 38 59 COc1ccccc1-c1ccc(S(=O)(=O)N[C@@H](C(=O)O)C(C)C)cc1 ZINC000217965730 FF On-Demand Unstable CAPN1 22 42 COc1ccccc1-c1ccc(S(=O)(=O)N[C@@H](C(=O)O)C(C)C)cc1 ZINC000217965730 FF On-Demand Unstable MMP9 46 67 COc1ccccc1-c1ccc(S(=O)(=O)N[C@@H](C(=O)O)C(C)C)cc1 ZINC000217965730 FF On-Demand Unstable MMP12 116 48 COc1ccccc1-c1ccc(S(=O)(=O)N[C@@H](C(=O)O)C(C)C)cc1 ZINC000217965730 FF On-Demand Unstable MMP7 32 50 COc1ccccc1-c1ccc(S(=O)(=O)N[C@@H](C(=O)O)C(C)C)cc1 ZINC000217965730 FF On-Demand Unstable ADAMTS4 98 54 COc1ccccc1-c1ccc(S(=O)(=O)N[C@@H](C(=O)O)C(C)C)cc1 ZINC000217965730 FF On-Demand Unstable MMP1 25 50 COc1ccccc1-c1ccc(S(=O)(=O)N[C@@H](C(=O)O)C(C)C)cc1 ZINC000217965730 FF On-Demand Unstable LEF 31 50 COc1ccccc1/C=C/C(=O)NCCCc1ccc(OC(C)C)cc1 ZINC000217965739 FI In-Stock Unstable DRD3 19 52 COc1ccccc1/C=C/C(=O)NCCCc1ccc(OC(C)C)cc1 ZINC000217965739 FI In-Stock Unstable PTAFR 19 43 CCOc1ccc(-c2nc(CN[C@@H](c3ccc(OC)cc3)C3CC3)cs2)cc1 ZINC000217965744 GK On-Demand Unstable AVPR1B 24 42 O=C(c1ccccc1N1CCOCC1)N1CCN(Cc2nnc[nH]2)CC1 ZINC000217965749 FC In-Stock Unstable AKR1C3 28 40 Cc1cc(OCC(=O)N[C@@H]2CCC[C@@H]2CO)no1 ZINC000217965802 CC For-Sale Unstable S1PR3 0 42 CCOc1ccc(-c2nc(CN[C@H](c3ccc(OC)cc3)C3CC3)cs2)cc1 ZINC000217965821 GK On-Demand Unstable AVPR1B 24 42 O=C1C/C(=C/c2ccc(-c3ccc(Br)cc3)s2)C(=O)N1 ZINC000217965822 EH For-Sale Unstable PRF1 45 38 COc1ccc(/C=C\C(=O)O)cc1CN1CCC[C@H](O)C1 ZINC000217965837 CD For-Sale Unstable SLC6A1 42 36 COc1ccc(/C=C\C(=O)O)cc1CN1CCC[C@H](O)C1 ZINC000217965837 CD For-Sale Unstable ACKR3 44 33 Cc1cc(N)ccc1S(=O)(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217965852 DF For-Sale Unstable EPHX2 15 40 COc1cccc2cc(C(=O)N3CCCN(S(=O)(=O)c4cnn(C)c4)CC3)oc12 ZINC000217965859 HD In-Stock Unstable SSTR1 41 34 C[C@H](C(=O)NN)c1ccc(CN2CCCCC[C@@H]2C)cc1 ZINC000217965889 CF For-Sale Unstable HRH3 41 49 Cc1cc(OCC(=O)N[C@H]2CCC[C@@H]2CO)no1 ZINC000217965895 CC For-Sale Unstable S1PR3 0 42 COc1cc([C@@H]2CC(=O)Oc3cc(C)oc(=O)c32)ccc1O ZINC000217965927 DE In-Stock Unstable CAN2 0 41 Cc1cc(N)ccc1S(=O)(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217965938 DF For-Sale Unstable EPHX2 15 40 CC(=O)NC[C@]1(O)CCN(Cc2ccccc2)C1 ZINC000217965950 BC On-Demand Unstable CHRM2 17 41 CC(=O)NC[C@]1(O)CCN(Cc2ccccc2)C1 ZINC000217965950 BC On-Demand Unstable DRD3 15 41 CC(=O)NC[C@]1(O)CCN(Cc2ccccc2)C1 ZINC000217965950 BC On-Demand Unstable OPRK1 17 49 CC(=O)NC[C@]1(O)CCN(Cc2ccccc2)C1 ZINC000217965950 BC On-Demand Unstable OPRL1 27 43 CC(=O)NC[C@]1(O)CCN(Cc2ccccc2)C1 ZINC000217965950 BC On-Demand Unstable SIGMAR1 69 40 CC(=O)NC[C@]1(O)CCN(Cc2ccccc2)C1 ZINC000217965950 BC On-Demand Unstable NPFFR2 53 49 CC(=O)NC[C@]1(O)CCN(Cc2ccccc2)C1 ZINC000217965950 BC On-Demand Unstable MCHR2 41 36 CC(=O)NC[C@]1(O)CCN(Cc2ccccc2)C1 ZINC000217965950 BC On-Demand Unstable NPFFR1 78 49 COc1ccc(CN2CCC[C@H](O)C2)cc1/C=C\C(=O)O ZINC000217965952 CD For-Sale Unstable DRD4 28 41 COc1ccc(CN2CCC[C@H](O)C2)cc1/C=C\C(=O)O ZINC000217965952 CD For-Sale Unstable ACHE 17 43 COc1ccc(CN2CCC[C@H](O)C2)cc1/C=C\C(=O)O ZINC000217965952 CD For-Sale Unstable SLC6A1 66 39 COc1ccc(CN2CCC[C@H](O)C2)cc1/C=C\C(=O)O ZINC000217965952 CD For-Sale Unstable DRD3 20 41 COc1ccc(CN2CCC[C@H](O)C2)cc1/C=C\C(=O)O ZINC000217965952 CD For-Sale Unstable MCHR1 18 43 CCc1ncnc(NCc2cccc(C)c2)c1F ZINC000217965964 BG On-Demand Unstable ADORA3 24 41 CCc1ncnc(NCc2cccc(C)c2)c1F ZINC000217965964 BG On-Demand Unstable CLK4 22 47 Cc1cc(OCC(=O)N[C@@H]2CCC[C@H]2CO)no1 ZINC000217965971 CC For-Sale Unstable S1PR3 0 42 COc1cc([C@H]2CC(=O)Oc3cc(C)oc(=O)c32)ccc1O ZINC000217966007 DE In-Stock Unstable CAN2 0 41 COC[C@@H]1CCN(Cc2ccc([C@@H](C)C(=O)NN)cc2)C1 ZINC000217966025 CD For-Sale Unstable SLC6A3 16 43 COC[C@@H]1CCN(Cc2ccc([C@@H](C)C(=O)NN)cc2)C1 ZINC000217966025 CD For-Sale Unstable HTR4 32 41 COC[C@@H]1CCN(Cc2ccc([C@@H](C)C(=O)NN)cc2)C1 ZINC000217966025 CD For-Sale Unstable SIGMAR1 30 43 COc1cccc(-c2ccc(S(=O)(=O)N[C@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966031 FF On-Demand Unstable BMP1 50 38 COc1cccc(-c2ccc(S(=O)(=O)N[C@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966031 FF On-Demand Unstable MMP13 110 77 COc1cccc(-c2ccc(S(=O)(=O)N[C@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966031 FF On-Demand Unstable ADAM17 30 40 COc1cccc(-c2ccc(S(=O)(=O)N[C@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966031 FF On-Demand Unstable CYP11B2 16 41 COc1cccc(-c2ccc(S(=O)(=O)N[C@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966031 FF On-Demand Unstable MMP2 86 77 COc1cccc(-c2ccc(S(=O)(=O)N[C@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966031 FF On-Demand Unstable MMP3 56 77 COc1cccc(-c2ccc(S(=O)(=O)N[C@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966031 FF On-Demand Unstable MMP8 52 77 COc1cccc(-c2ccc(S(=O)(=O)N[C@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966031 FF On-Demand Unstable MMP14 44 61 COc1cccc(-c2ccc(S(=O)(=O)N[C@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966031 FF On-Demand Unstable MMP9 61 77 COc1cccc(-c2ccc(S(=O)(=O)N[C@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966031 FF On-Demand Unstable MMP12 124 49 COc1cccc(-c2ccc(S(=O)(=O)N[C@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966031 FF On-Demand Unstable PLAU 17 45 COc1cccc(-c2ccc(S(=O)(=O)N[C@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966031 FF On-Demand Unstable ITGAV 21 44 COc1cccc(-c2ccc(S(=O)(=O)N[C@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966031 FF On-Demand Unstable MMP7 40 52 COc1cccc(-c2ccc(S(=O)(=O)N[C@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966031 FF On-Demand Unstable ADAMTS4 108 63 COc1cccc(-c2ccc(S(=O)(=O)N[C@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966031 FF On-Demand Unstable MMP1 40 55 COc1cccc(-c2ccc(S(=O)(=O)N[C@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966031 FF On-Demand Unstable HSD17B2 23 43 COc1cccc(-c2ccc(S(=O)(=O)N[C@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966031 FF On-Demand Unstable LEF 32 55 CC(=O)NC[C@@]1(O)CCN(Cc2ccccc2)C1 ZINC000217966034 BC On-Demand Unstable CHRM2 17 41 CC(=O)NC[C@@]1(O)CCN(Cc2ccccc2)C1 ZINC000217966034 BC On-Demand Unstable DRD3 15 41 CC(=O)NC[C@@]1(O)CCN(Cc2ccccc2)C1 ZINC000217966034 BC On-Demand Unstable OPRK1 17 49 CC(=O)NC[C@@]1(O)CCN(Cc2ccccc2)C1 ZINC000217966034 BC On-Demand Unstable OPRL1 27 43 CC(=O)NC[C@@]1(O)CCN(Cc2ccccc2)C1 ZINC000217966034 BC On-Demand Unstable SIGMAR1 69 40 CC(=O)NC[C@@]1(O)CCN(Cc2ccccc2)C1 ZINC000217966034 BC On-Demand Unstable NPFFR2 53 49 CC(=O)NC[C@@]1(O)CCN(Cc2ccccc2)C1 ZINC000217966034 BC On-Demand Unstable MCHR2 41 36 CC(=O)NC[C@@]1(O)CCN(Cc2ccccc2)C1 ZINC000217966034 BC On-Demand Unstable NPFFR1 78 49 Cc1cc(OCC(=O)N[C@H]2CCC[C@H]2CO)no1 ZINC000217966052 CC For-Sale Unstable S1PR3 0 42 O=C(O)/C=C\c1ccc(CN2CCC[C@H](O)C2)c(F)c1 ZINC000217966075 CD For-Sale Unstable SLC6A1 72 35 C=C(C)COc1c(OC)cccc1[C@@H]1CC(=O)Oc2ccc3c(c21)OC1(CCCCC1)CC3=O ZINC000217966105 JK In-Stock Unstable MT-ND4 40 31 COc1cccc(-c2ccc(S(=O)(=O)N[C@@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966125 FF On-Demand Unstable BMP1 50 38 COc1cccc(-c2ccc(S(=O)(=O)N[C@@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966125 FF On-Demand Unstable MMP13 110 77 COc1cccc(-c2ccc(S(=O)(=O)N[C@@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966125 FF On-Demand Unstable ADAM17 30 40 COc1cccc(-c2ccc(S(=O)(=O)N[C@@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966125 FF On-Demand Unstable CYP11B2 16 41 COc1cccc(-c2ccc(S(=O)(=O)N[C@@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966125 FF On-Demand Unstable MMP2 86 77 COc1cccc(-c2ccc(S(=O)(=O)N[C@@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966125 FF On-Demand Unstable MMP3 56 77 COc1cccc(-c2ccc(S(=O)(=O)N[C@@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966125 FF On-Demand Unstable MMP8 52 77 COc1cccc(-c2ccc(S(=O)(=O)N[C@@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966125 FF On-Demand Unstable MMP14 44 61 COc1cccc(-c2ccc(S(=O)(=O)N[C@@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966125 FF On-Demand Unstable MMP9 61 77 COc1cccc(-c2ccc(S(=O)(=O)N[C@@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966125 FF On-Demand Unstable MMP12 124 49 COc1cccc(-c2ccc(S(=O)(=O)N[C@@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966125 FF On-Demand Unstable PLAU 17 45 COc1cccc(-c2ccc(S(=O)(=O)N[C@@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966125 FF On-Demand Unstable ITGAV 21 44 COc1cccc(-c2ccc(S(=O)(=O)N[C@@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966125 FF On-Demand Unstable MMP7 40 52 COc1cccc(-c2ccc(S(=O)(=O)N[C@@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966125 FF On-Demand Unstable ADAMTS4 108 63 COc1cccc(-c2ccc(S(=O)(=O)N[C@@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966125 FF On-Demand Unstable MMP1 40 55 COc1cccc(-c2ccc(S(=O)(=O)N[C@@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966125 FF On-Demand Unstable HSD17B2 23 43 COc1cccc(-c2ccc(S(=O)(=O)N[C@@H](C(=O)O)C(C)C)cc2)c1 ZINC000217966125 FF On-Demand Unstable LEF 32 55 CCOc1ccc(CCCNC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217966147 EH In-Stock Unstable DRD3 25 52 CCOc1ccc(CCCNC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217966147 EH In-Stock Unstable PTGER2 28 41 CCOc1ccc(CCCNC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217966147 EH In-Stock Unstable PTAFR 16 43 CCOc1ccc(CCCNC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217966147 EH In-Stock Unstable PTGER4 0 41 CCOc1ccc(CCCNC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217966147 EH In-Stock Unstable SCN2A 16 44 CCOc1ccc(CCCNC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217966147 EH In-Stock Unstable MTNR1A 18 41 CCOc1ccc(CCCNC(=O)/C=C/c2ccccc2OC)cc1 ZINC000217966147 EH In-Stock Unstable AKR1B10 28 40 O=C1C/C(=C/c2ccc(OC(F)F)cc2)C(=O)N1 ZINC000217966166 CD For-Sale Unstable HPGD 52 33 CN(Cc1ccc(/C=C\C(=O)O)cc1)CC1CCCCC1 ZINC000217966176 CH For-Sale Unstable NR1H4 25 40 C=C(C)COc1c(OC)cccc1[C@H]1CC(=O)Oc2ccc3c(c21)OC1(CCCCC1)CC3=O ZINC000217966189 JK In-Stock Unstable MT-ND4 40 31 Nc1cccc(NC(=O)CN2CCC[C@@H]3CCCC[C@H]32)c1 ZINC000217966211 CF For-Sale Unstable CCKBR 17 41 Cn1c(=O)n(CCC(=O)N2CCC(C(=O)Nc3ccccc3O)CC2)c2ccccc21 ZINC000217966233 HE On-Demand Unstable CCR8 41 41 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CNC(=O)OCc1ccccc1 ZINC000217966252 IE For-Sale Unstable PREP 18 46 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CNC(=O)OCc1ccccc1 ZINC000217966252 IE For-Sale Unstable NPR 48 31 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccccc1OC ZINC000217966256 FI In-Stock Unstable DRD3 22 52 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccccc1OC ZINC000217966256 FI In-Stock Unstable PTGER2 31 43 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccccc1OC ZINC000217966256 FI In-Stock Unstable MTNR1A 28 49 CCCOc1ccccc1CCCNC(=O)/C=C/c1ccccc1OC ZINC000217966256 FI In-Stock Unstable MTNR1B 38 42 CN(Cc1cccc(/C=C\C(=O)O)c1)CC1CCCCC1 ZINC000217966259 CH For-Sale Unstable NR1H4 39 42 Nc1cccc(NC(=O)CN2CCC[C@H]3CCCC[C@H]32)c1 ZINC000217966287 CF For-Sale Unstable CCKBR 17 41 Cn1cc(S(=O)(=O)N2CCCN(C(=O)c3ccc(C(C)(C)C)cc3)CC2)cn1 ZINC000217966297 HE In-Stock Unstable MLYCD 18 41 Cn1cc(S(=O)(=O)N2CCCN(C(=O)c3ccc(C(C)(C)C)cc3)CC2)cn1 ZINC000217966297 HE In-Stock Unstable L3MBTL1 0 41 Cn1cc(S(=O)(=O)N2CCCN(C(=O)c3ccc(C(C)(C)C)cc3)CC2)cn1 ZINC000217966297 HE In-Stock Unstable L3MBTL3 34 41 Cn1cc(S(=O)(=O)N2CCCN(C(=O)c3ccc(C(C)(C)C)cc3)CC2)cn1 ZINC000217966297 HE In-Stock Unstable MBTD1 0 41 BrCc1ccc(-n2nnc(-c3ccccc3)n2)nc1 ZINC000217966299 DF For-Sale Unstable GRM5 0 42 O=C([C@@H]1CC[C@@H](Cn2cnnn2)CC1)N1CCC(O)(c2ccc(Cl)cc2)CC1 ZINC000217966320 HF In-Stock Unstable CCR1 69 40 COc1ccccc1/C=C/C(=O)N[C@H](C)COc1ccccc1C ZINC000217966328 EH In-Stock Unstable KCNQ2 48 34 COc1ccccc1/C=C/C(=O)N[C@H](C)COc1ccccc1C ZINC000217966328 EH In-Stock Unstable UL26 25 42 COc1ccccc1/C=C/C(=O)N[C@H](C)COc1ccccc1C ZINC000217966328 EH In-Stock Unstable U53 0 42 COc1ccccc1/C=C/C(=O)N[C@H](C)COc1ccccc1C ZINC000217966328 EH In-Stock Unstable SCAF_EBVB9 20 42 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CNC(=O)OCc1ccccc1 ZINC000217966331 IE For-Sale Unstable PREP 18 46 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)CNC(=O)OCc1ccccc1 ZINC000217966331 IE For-Sale Unstable NPR 48 31 Cc1occc1CN(C)Cc1ccccc1/C=C\C(=O)O ZINC000217966378 CG For-Sale Unstable PTGER2 45 46 Cc1occc1CN(C)Cc1ccccc1/C=C\C(=O)O ZINC000217966378 CG For-Sale Unstable PTGER4 0 46 Cc1occc1CN(C)Cc1ccccc1/C=C\C(=O)O ZINC000217966378 CG For-Sale Unstable PTGER3 17 47 C[C@H](C(=O)NN)c1ccc(CN2C[C@@H](C)[C@@H](C)C2)cc1 ZINC000217966379 CD For-Sale Unstable MLNR 31 43 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(Cl)c(Cl)c1 ZINC000217966394 EJ For-Sale Anodyne IMPDH2 0 42 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(Cl)c(Cl)c1 ZINC000217966394 EJ For-Sale Anodyne IMDH_CRYPV 33 41 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(Cl)c(Cl)c1 ZINC000217966394 EJ For-Sale Anodyne BLM 0 41 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(Cl)c(Cl)c1 ZINC000217966394 EJ For-Sale Anodyne P95276_MYCTO 0 47 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(Cl)c(Cl)c1 ZINC000217966394 EJ For-Sale Anodyne PPX1 0 40 Cn1cc(S(=O)(=O)N2CCCN(C(=O)c3ccc4c(c3)OCO4)CC2)cn1 ZINC000217966396 GC In-Stock Unstable PKM 32 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CNC(=O)OCc1ccccc1 ZINC000217966397 IE For-Sale Unstable PREP 18 46 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CNC(=O)OCc1ccccc1 ZINC000217966397 IE For-Sale Unstable NPR 48 31 C[C@@H]1C[C@@H]1[C@@H](Cl)Cc1ccc2ccccc2c1 ZINC000217966410 BJ For-Sale Unstable CYP2A5 0 44 COc1ccccc1/C=C/C(=O)N[C@@H](C)COc1ccc(C)cc1 ZINC000217966434 EH In-Stock Unstable KCNQ2 47 34 COc1cc2c(cc1Cl)CCCNC2=O ZINC000217966448 BE For-Sale Unstable CSNK1G2 56 31 C[C@H](C(=O)NN)c1ccc(CN2C[C@H](C)[C@@H](C)C2)cc1 ZINC000217966465 CD For-Sale Unstable MLNR 31 43 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CNC(=O)OCc1ccccc1 ZINC000217966475 IE For-Sale Unstable PREP 18 46 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)CNC(=O)OCc1ccccc1 ZINC000217966475 IE For-Sale Unstable NPR 48 31 Cc1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1Cl ZINC000217966486 DJ For-Sale Unstable IMPDH2 0 40 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)Nc3ccc4c(ccn4C)c3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217966492 KI In-Stock Unstable TUBA1A 17 62 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)Nc3ccc4c(ccn4C)c3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217966492 KI In-Stock Unstable TPPP 0 59 COc1ccc(/C=C\C(=O)O)cc1CN(C)CCC#N ZINC000217966496 CE For-Sale Unstable PTGER2 0 42 COc1ccc(/C=C\C(=O)O)cc1CN(C)CCC#N ZINC000217966496 CE For-Sale Unstable AKR1C3 22 40 C[C@H]1C[C@@H]1[C@@H](Cl)Cc1ccc2ccccc2c1 ZINC000217966500 BJ For-Sale Unstable CYP2A5 0 44 COc1ccccc1/C=C/C(=O)N[C@H](C)COc1ccc(C)cc1 ZINC000217966524 EH In-Stock Unstable KCNQ2 47 34 C[C@@H]1C[C@H]1[C@@H](Cl)Cc1ccc2ccccc2c1 ZINC000217966574 BJ For-Sale Unstable CYP2A5 0 44 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cc2ccc(OC)cc2[nH]1 ZINC000217966577 HG For-Sale Unstable TUBB2B 32 42 Nc1ccccc1NC(=O)CN1CCC[C@@H]2CCCC[C@H]21 ZINC000217966587 CF For-Sale Unstable KCNQ2 44 38 Nc1ccccc1NC(=O)CN1CCC[C@@H]2CCCC[C@H]21 ZINC000217966587 CF For-Sale Unstable HDAC1 34 40 COc1ccc(CN(C)CCC#N)cc1/C=C\C(=O)O ZINC000217966611 CE For-Sale Unstable PTGER2 27 41 COc1ccc(CN(C)CCC#N)cc1/C=C\C(=O)O ZINC000217966611 CE For-Sale Unstable PTGER4 0 41 COc1ccccc1/C=C/C(=O)N[C@@H](C)c1ccc(N2CCC(C)CC2)cc1 ZINC000217966626 GJ In-Stock Unstable KCNQ2 56 42 O=C1C/C(=C/c2ccc(Cl)c(Cl)c2)C(=O)N1 ZINC000217966631 CE For-Sale Unstable HPGD 50 38 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1ccc(CC#N)cc1 ZINC000217966638 CJ For-Sale Unstable TRPM8 16 41 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cc2ccc(OC)cc2[nH]1 ZINC000217966655 HG For-Sale Unstable TUBB2B 32 42 C[C@H]1C[C@H]1[C@@H](Cl)Cc1ccc2ccccc2c1 ZINC000217966661 BJ For-Sale Unstable CYP2A5 0 44 Nc1ccccc1NC(=O)CN1CCC[C@H]2CCCC[C@H]21 ZINC000217966675 CF For-Sale Unstable KCNQ2 44 38 Nc1ccccc1NC(=O)CN1CCC[C@H]2CCCC[C@H]21 ZINC000217966675 CF For-Sale Unstable HDAC1 34 40 COc1ccccc1/C=C/C(=O)N[C@H](C)c1ccc(N2CCC(C)CC2)cc1 ZINC000217966709 GJ In-Stock Unstable KCNQ2 56 42 C[C@@H]1CCCN(Cc2ccc(F)c(/C=C\C(=O)O)c2)C1 ZINC000217966711 CG For-Sale Unstable SLC6A1 96 36 C[C@@H]1CCCN(Cc2ccc(F)c(/C=C\C(=O)O)c2)C1 ZINC000217966711 CG For-Sale Unstable CCR1 25 42 C[C@@H]1CCCN(Cc2ccc(F)c(/C=C\C(=O)O)c2)C1 ZINC000217966711 CG For-Sale Unstable MLNR 52 35 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1ccc(CC#N)cc1 ZINC000217966721 CJ For-Sale Unstable TRPM8 16 41 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)c1cc2ccc(OC)cc2[nH]1 ZINC000217966727 HG For-Sale Unstable TUBB2B 32 42 Cc1cc(C(=O)N2Cc3ccccc3C[C@@H]2C(=O)O)cc(=O)[nH]1 ZINC000217966771 DD In-Stock Unstable ACE 19 47 Cc1cc(C(=O)N2Cc3ccccc3C[C@@H]2C(=O)O)cc(=O)[nH]1 ZINC000217966771 DD In-Stock Unstable OPRD1 68 45 Cc1cc(C(=O)N2Cc3ccccc3C[C@@H]2C(=O)O)cc(=O)[nH]1 ZINC000217966771 DD In-Stock Unstable AGTR2 15 40 Cc1cc(C(=O)N2Cc3ccccc3C[C@@H]2C(=O)O)cc(=O)[nH]1 ZINC000217966771 DD In-Stock Unstable CFTR 59 41 CC[C@@H]1CCCCN1C(=O)[C@@H](C)N[C@@H](c1ccccc1)C1CC1 ZINC000217966779 DH On-Demand Unstable ACE 50 42 CC[C@@H]1CCCCN1C(=O)[C@@H](C)N[C@@H](c1ccccc1)C1CC1 ZINC000217966779 DH On-Demand Unstable KCNQ2 45 35 CC[C@@H]1CCCCN1C(=O)[C@@H](C)N[C@@H](c1ccccc1)C1CC1 ZINC000217966779 DH On-Demand Unstable ACE2 19 42 CC(=O)N1CC(Nc2ccc(C(=O)O)cc2)=CC1=O ZINC000217966786 CD In-Stock Unstable AKR1C3 28 45 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1ccc(CC#N)cc1 ZINC000217966795 CJ For-Sale Unstable TRPM8 16 41 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)c1cc2ccc(OC)cc2[nH]1 ZINC000217966797 HG For-Sale Unstable TUBB2B 32 42 C[C@H]1CCCN(Cc2ccc(F)c(/C=C\C(=O)O)c2)C1 ZINC000217966802 CG For-Sale Unstable SLC6A1 96 36 C[C@H]1CCCN(Cc2ccc(F)c(/C=C\C(=O)O)c2)C1 ZINC000217966802 CG For-Sale Unstable CCR1 25 42 C[C@H]1CCCN(Cc2ccc(F)c(/C=C\C(=O)O)c2)C1 ZINC000217966802 CG For-Sale Unstable MLNR 52 35 COc1ccccc1/C=C/C(=O)N[C@@H](C)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217966815 GJ In-Stock Unstable KCNQ2 55 42 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(C(=O)O)cc1 ZINC000217966816 DG For-Sale Anodyne UL80 17 40 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(C(=O)O)cc1 ZINC000217966816 DG For-Sale Anodyne AKR1C3 27 40 Cc1cc(C(=O)N2Cc3ccccc3C[C@H]2C(=O)O)cc(=O)[nH]1 ZINC000217966863 DD In-Stock Unstable ACE 19 47 Cc1cc(C(=O)N2Cc3ccccc3C[C@H]2C(=O)O)cc(=O)[nH]1 ZINC000217966863 DD In-Stock Unstable OPRD1 68 45 Cc1cc(C(=O)N2Cc3ccccc3C[C@H]2C(=O)O)cc(=O)[nH]1 ZINC000217966863 DD In-Stock Unstable AGTR2 15 40 Cc1cc(C(=O)N2Cc3ccccc3C[C@H]2C(=O)O)cc(=O)[nH]1 ZINC000217966863 DD In-Stock Unstable CFTR 59 41 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1ccc(CC#N)cc1 ZINC000217966869 CJ For-Sale Unstable TRPM8 16 41 COc1ccccc1CCC(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217966871 CD On-Demand Unstable MBTPS1 48 41 COc1ccccc1CCC(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217966871 CD On-Demand Unstable SLC5A4 44 34 Cn1cc(S(=O)(=O)N2CCCN(C(=O)CSCc3ccccc3)CC2)cn1 ZINC000217966883 HD In-Stock Unstable TGM2 27 40 Cn1cc(S(=O)(=O)N2CCCN(C(=O)CSCc3ccccc3)CC2)cn1 ZINC000217966883 HD In-Stock Unstable F13A1 34 40 CCCCN(C)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217966891 CF On-Demand Unstable THRA 59 42 CCCCN(C)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217966891 CF On-Demand Unstable FDPS 29 42 CCCCN(C)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217966891 CF On-Demand Unstable LTA4H 22 46 CCCCN(C)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217966891 CF On-Demand Unstable THRB 29 42 CCCCN(C)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217966891 CF On-Demand Unstable SHC 21 40 CCCCN(C)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217966891 CF On-Demand Unstable PLA2G4B 89 38 CCCCN(C)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217966891 CF On-Demand Unstable LSS 49 40 CCCCN(C)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217966891 CF On-Demand Unstable ESRRG 42 32 CCCCN(C)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217966891 CF On-Demand Unstable FAAH 22 40 CCCCN(C)CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217966891 CF On-Demand Unstable AKR1C3 0 43 COc1ccccc1/C=C/C(=O)N[C@H](C)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217966899 GJ In-Stock Unstable KCNQ2 55 42 CC[C@@H]1CCCCN1C(=O)[C@H](C)N[C@@H](c1ccccc1)C1CC1 ZINC000217966937 DH On-Demand Unstable ACE 50 42 CC[C@@H]1CCCCN1C(=O)[C@H](C)N[C@@H](c1ccccc1)C1CC1 ZINC000217966937 DH On-Demand Unstable KCNQ2 45 35 CC[C@@H]1CCCCN1C(=O)[C@H](C)N[C@@H](c1ccccc1)C1CC1 ZINC000217966937 DH On-Demand Unstable ACE2 19 42 Nc1c(Cl)ncnc1N[C@H]1CCc2ccccc21 ZINC000217966951 CF For-Sale Unstable KCNN3 22 45 Cn1nccc1CCNC(=O)c1cc2ccccc2n1C ZINC000217966965 CD In-Stock Unstable PYK 40 42 O=C(O)/C=C\c1ccc(CN2CCc3ccccc32)cc1 ZINC000217966977 CG For-Sale Unstable DRD4 22 44 O=C(O)/C=C\c1ccc(CN2CCc3ccccc32)cc1 ZINC000217966977 CG For-Sale Unstable PTGER2 0 41 C[C@H](O)[C@@H](NC(=O)N1c2ccccc2CC[C@@H]1C)C(=O)O ZINC000217966995 CD For-Sale Unstable ACE 34 45 O=C(NCc1ccccc1F)[C@@H]1CC[C@@H](Cn2cnnn2)CC1 ZINC000217967000 DD In-Stock Unstable CACNA1G 26 41 Nc1c(Cl)ncnc1N[C@@H]1CCc2ccccc21 ZINC000217967024 CF For-Sale Unstable KCNN3 22 45 CCc1ncnc(N[C@@H](C)c2cccc(Br)c2)c1F ZINC000217967039 DI On-Demand Unstable EGFR 37 41 CCOC(=O)c1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217967040 EH For-Sale Unstable ACR 62 36 CCOC(=O)c1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217967040 EH For-Sale Unstable SENP1 0 43 O=C(/C=C\c1ccc2c(c1)OCCCO2)CCl ZINC000217967063 CF For-Sale Unstable PLK1 17 43 C[C@H](O)[C@H](NC(=O)N1c2ccccc2CC[C@@H]1C)C(=O)O ZINC000217967066 CD For-Sale Unstable ACE 34 45 O=C(O)/C=C\c1cccc(CN2CCc3ccccc32)c1 ZINC000217967070 CG For-Sale Unstable PTGER2 25 43 O=C(O)/C=C\c1cccc(CN2CCc3ccccc32)c1 ZINC000217967070 CG For-Sale Unstable HDAC8 44 37 O=C(O)/C=C\c1cccc(CN2CCc3ccccc32)c1 ZINC000217967070 CG For-Sale Unstable HDAC1 21 43 COC(=O)c1cccc(COc2ccc3c(c2)O/C(=C\c2ccco2)C3=O)c1 ZINC000217967090 GI In-Stock Unstable MAOB 38 41 CCc1ncnc(N[C@H](C)c2cccc(Br)c2)c1F ZINC000217967112 DI On-Demand Unstable EGFR 37 41 CCOc1ccc(/C=C\C(=O)CCl)cc1OCC ZINC000217967137 CG For-Sale Unstable TUBB1 27 44 CCOc1ccc(/C=C\C(=O)CCl)cc1OCC ZINC000217967137 CG For-Sale Unstable AKR1C3 29 50 CCOc1ccc(/C=C\C(=O)CCl)cc1OCC ZINC000217967137 CG For-Sale Unstable NFE2L2 0 40 C[C@H]1C[C@@H](C)CN(Cc2ccccc2/C=C\C(=O)O)C1 ZINC000217967168 CG For-Sale Unstable PTGER2 44 47 C[C@H]1C[C@@H](C)CN(Cc2ccccc2/C=C\C(=O)O)C1 ZINC000217967168 CG For-Sale Unstable PTGER4 0 47 C[C@H]1C[C@@H](C)CN(Cc2ccccc2/C=C\C(=O)O)C1 ZINC000217967168 CG For-Sale Unstable PTGER3 17 47 Cn1cc(S(=O)(=O)N2CCCN(C(=O)c3ccco3)CC2)cn1 ZINC000217967199 EC In-Stock Unstable F13A1 42 38 O=C(/C=C\c1ccc(Oc2ccccc2)cc1)CCl ZINC000217967220 CI For-Sale Unstable AKR1B1 21 44 O=C(/C=C\c1ccc(Oc2ccccc2)cc1)CCl ZINC000217967220 CI For-Sale Unstable F3 24 43 O=C(/C=C\c1ccc(Oc2ccccc2)cc1)CCl ZINC000217967220 CI For-Sale Unstable MMP2 20 40 O=C(/C=C\c1ccc(Oc2ccccc2)cc1)CCl ZINC000217967220 CI For-Sale Unstable 17HSDCL 0 40 CSc1ccc(C(=O)N[C@@H]2CCC[C@@H]2CO)cc1[N+](=O)[O-] ZINC000217967223 DE On-Demand Unstable GSTM2 44 32 O=C(Nc1cc(Cl)ccc1[N+](=O)[O-])NC1CCCCC1 ZINC000217967270 CH For-Sale Unstable EPHX2 25 54 O=C(/C=C\c1ccc(F)cc1)CCl ZINC000217967306 AF For-Sale Unstable SSSIM 16 50 N[C@@H]1C(=O)NC[C@@H]1CP(=O)(O)O ZINC000217967310 AA For-Sale Unstable AROB 47 30 COc1ccc2c(c1)[C@@H](NC(=O)/C=C/c1ccccc1OC)CC(C)(C)O2 ZINC000217967349 FI In-Stock Unstable CYP1B1 24 40 C[C@H](N[C@H](c1ccccc1)C1CC1)C(=O)N[C@@H]1CCCC[C@@H]1C ZINC000217967350 DH On-Demand Unstable BIRC8 45 37 CC[C@@H]1CCCN(Cc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217967363 CG For-Sale Unstable DRD2 17 45 CC[C@@H]1CCCN(Cc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217967363 CG For-Sale Unstable SLC6A1 74 35 CC[C@@H]1CCCN(Cc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217967363 CG For-Sale Unstable SIGMAR1 36 45 CC[C@@H]1CCCN(Cc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217967363 CG For-Sale Unstable CCR3 30 41 CC[C@@H]1CCCN(Cc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217967363 CG For-Sale Unstable HDAC8 38 42 CC[C@@H]1CCCN(Cc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217967363 CG For-Sale Unstable HDAC1 18 42 CC[C@@H]1CCCN(Cc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217967363 CG For-Sale Unstable HDAC6 27 42 N[C@@H]1C(=O)NC[C@H]1CP(=O)(O)O ZINC000217967397 AA For-Sale Unstable AROB 47 30 Cn1cc(S(=O)(=O)N2CCCN(C(=O)c3cc(=O)c4ccccc4o3)CC2)cn1 ZINC000217967405 HD In-Stock Unstable TNKS 29 43 CC[C@H]1CCCN(Cc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217967429 CG For-Sale Unstable DRD2 17 45 CC[C@H]1CCCN(Cc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217967429 CG For-Sale Unstable SLC6A1 74 35 CC[C@H]1CCCN(Cc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217967429 CG For-Sale Unstable SIGMAR1 36 45 CC[C@H]1CCCN(Cc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217967429 CG For-Sale Unstable CCR3 30 41 CC[C@H]1CCCN(Cc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217967429 CG For-Sale Unstable HDAC8 38 42 CC[C@H]1CCCN(Cc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217967429 CG For-Sale Unstable HDAC1 18 42 CC[C@H]1CCCN(Cc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217967429 CG For-Sale Unstable HDAC6 27 42 COc1ccc2c(c1)[C@H](NC(=O)/C=C/c1ccccc1OC)CC(C)(C)O2 ZINC000217967433 FI In-Stock Unstable CYP1B1 24 40 O=C(CCSc1nc2ccccc2o1)NCc1ccccc1 ZINC000217967435 DH For-Sale Unstable MTNR1A 17 40 O=C(CCSc1nc2ccccc2o1)NCc1ccccc1 ZINC000217967435 DH For-Sale Unstable MTNR1B 19 40 O=C(CCSc1nc2ccccc2o1)NCc1ccccc1 ZINC000217967435 DH For-Sale Unstable TNKS 66 38 Cc1cc2nc(CNC(=O)CN3CCC[C@@H](O)C3)[nH]c2cc1C ZINC000217967439 DD In-Stock Unstable F9 39 43 O=C(/C=C\c1c(-c2ccccc2)[nH]c2ccccc12)CCl ZINC000217967449 CJ For-Sale Unstable PTGS2 52 38 O=C(/C=C\c1c(-c2ccccc2)[nH]c2ccccc12)CCl ZINC000217967449 CJ For-Sale Unstable TSPO 24 53 N[C@H]1C(=O)NC[C@@H]1CP(=O)(O)O ZINC000217967475 AA For-Sale Unstable AROB 47 30 Cc1cc2nc(CNC(=O)CN3CCC[C@H](O)C3)[nH]c2cc1C ZINC000217967514 DD In-Stock Unstable F9 39 43 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)/C=C/c1ccccc1OC ZINC000217967528 FI In-Stock Unstable CYP1B1 32 41 CC[C@@H]1CCCN(Cc2ccc(F)cc2/C=C\C(=O)O)C1 ZINC000217967534 CH For-Sale Unstable SLC6A1 105 42 CC[C@@H]1CCCN(Cc2ccc(F)cc2/C=C\C(=O)O)C1 ZINC000217967534 CH For-Sale Unstable CCR3 59 36 COc1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1Cl ZINC000217967539 DI For-Sale Unstable EGFR 22 42 COc1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1Cl ZINC000217967539 DI For-Sale Unstable HTR2A 20 41 COc1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1Cl ZINC000217967539 DI For-Sale Unstable PYGL 0 40 COc1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1Cl ZINC000217967539 DI For-Sale Unstable GRM4 15 46 COc1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1Cl ZINC000217967539 DI For-Sale Unstable PDGFRA 25 42 COc1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1Cl ZINC000217967539 DI For-Sale Unstable IMPDH2 0 47 O=C(c1n[nH]c2c1CCC2)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217967550 DD In-Stock Unstable CHRNA4 29 47 N[C@H]1C(=O)NC[C@H]1CP(=O)(O)O ZINC000217967575 AA For-Sale Unstable AROB 47 30 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)/C=C/c1ccccc1OC ZINC000217967609 FI In-Stock Unstable CYP1B1 32 41 CC[C@H]1CCCN(Cc2ccc(F)cc2/C=C\C(=O)O)C1 ZINC000217967619 CH For-Sale Unstable SLC6A1 105 42 CC[C@H]1CCCN(Cc2ccc(F)cc2/C=C\C(=O)O)C1 ZINC000217967619 CH For-Sale Unstable CCR3 59 36 Cn1cc(S(=O)(=O)N2CCCN(C(=O)Cc3ccccc3Cl)CC2)cn1 ZINC000217967627 GD In-Stock Unstable TGM2 31 40 Cn1cc(S(=O)(=O)N2CCCN(C(=O)Cc3ccccc3Cl)CC2)cn1 ZINC000217967627 GD In-Stock Unstable F13A1 41 40 COC(=O)COc1ccc([C@@H](CC(=O)OC)C2=C(O)C(=O)C([C@H](CC(=O)OC)c3ccc(OCC(=O)OC)c(OC)c3)=C(O)C2=O)cc1OC ZINC000217967662 KF In-Stock Unstable TNF 22 41 O=C(N/C=C/c1cccc(F)c1)Nc1cccc(C(F)(F)F)c1 ZINC000217967666 DJ For-Sale Anodyne KIT 17 41 O=C(N/C=C/c1cccc(F)c1)Nc1cccc(C(F)(F)F)c1 ZINC000217967666 DJ For-Sale Anodyne UL80 18 41 O=C(N/C=C/c1cccc(F)c1)Nc1cccc(C(F)(F)F)c1 ZINC000217967666 DJ For-Sale Anodyne KDR 15 41 O=C(N/C=C/c1cccc(F)c1)Nc1cccc(C(F)(F)F)c1 ZINC000217967666 DJ For-Sale Anodyne RIPK1 57 40 O=C(N/C=C/c1cccc(F)c1)Nc1cccc(C(F)(F)F)c1 ZINC000217967666 DJ For-Sale Anodyne TRPM4 0 42 O=C(N/C=C/c1cccc(F)c1)Nc1cccc(C(F)(F)F)c1 ZINC000217967666 DJ For-Sale Anodyne KCNK3 18 42 O=C([C@@H]1C[C@@H](O)CN1)N1CCN2C(=O)NC[C@@H]2C1 ZINC000217967714 CA For-Sale Unstable DPP4 23 42 O=C([C@@H]1C[C@@H](O)CN1)N1CCN2C(=O)NC[C@@H]2C1 ZINC000217967714 CA For-Sale Unstable DPP8 0 42 O=C([C@@H]1C[C@@H](O)CN1)N1CCN2C(=O)NC[C@@H]2C1 ZINC000217967714 CA For-Sale Unstable DPP9 0 42 CC[C@@H](NC(=O)/C=C/c1ccccc1OC)c1ccc(C)c(C)c1 ZINC000217967724 DJ In-Stock Unstable KCNQ2 50 37 CC[C@@H]1CCCN(Cc2ccc(F)c(/C=C\C(=O)O)c2)C1 ZINC000217967726 CH For-Sale Unstable SLC6A1 78 35 CC[C@@H]1CCCN(Cc2ccc(F)c(/C=C\C(=O)O)c2)C1 ZINC000217967726 CH For-Sale Unstable CCR3 64 37 COC(=O)COc1ccc([C@H](CC(=O)OC)C2=C(O)C(=O)C([C@H](CC(=O)OC)c3ccc(OCC(=O)OC)c(OC)c3)=C(O)C2=O)cc1OC ZINC000217967753 KF In-Stock Unstable TNF 22 41 FC(F)(F)c1cc(-n2cccn2)ccc1CBr ZINC000217967802 DH For-Sale Unstable AMP1_PLAFQ 46 37 CC[C@H]1CCCN(Cc2ccc(F)c(/C=C\C(=O)O)c2)C1 ZINC000217967813 CH For-Sale Unstable SLC6A1 78 35 CC[C@H]1CCCN(Cc2ccc(F)c(/C=C\C(=O)O)c2)C1 ZINC000217967813 CH For-Sale Unstable CCR3 64 37 CC[C@H](NC(=O)/C=C/c1ccccc1OC)c1ccc(C)c(C)c1 ZINC000217967815 DJ In-Stock Unstable KCNQ2 50 37 COC(=O)COc1ccc([C@H](CC(=O)OC)C2=C(O)C(=O)C([C@@H](CC(=O)OC)c3ccc(OCC(=O)OC)c(OC)c3)=C(O)C2=O)cc1OC ZINC000217967836 KF In-Stock Unstable TNF 22 41 CN(Cc1cccc(/C=C\C(=O)O)c1)C1CCCCCC1 ZINC000217967907 CH For-Sale Unstable ACE 41 36 CN(Cc1cccc(/C=C\C(=O)O)c1)C1CCCCCC1 ZINC000217967907 CH For-Sale Unstable PTGER2 24 42 CN(Cc1cccc(/C=C\C(=O)O)c1)C1CCCCCC1 ZINC000217967907 CH For-Sale Unstable NR1H4 47 42 CC[C@@H](NC(=O)/C=C/c1ccccc1OC)c1ccc(C)cc1C ZINC000217967917 DJ In-Stock Unstable UL26 15 42 CC[C@@H](NC(=O)/C=C/c1ccccc1OC)c1ccc(C)cc1C ZINC000217967917 DJ In-Stock Unstable U53 0 42 CC[C@@H](NC(=O)/C=C/c1ccccc1OC)c1ccc(C)cc1C ZINC000217967917 DJ In-Stock Unstable SCAF_EBVB9 15 42 COC(=O)C[C@@H](C1=C(O)C(=O)C([C@H](CC(=O)OC)c2ccc(OC(C)C)c(OC)c2)=C(O)C1=O)c1ccc(OC(C)C)c(OC)c1 ZINC000217967939 KK In-Stock Unstable TNF 22 41 CC[C@H](NC(=O)/C=C/c1ccccc1OC)c1ccc(C)cc1C ZINC000217967984 DJ In-Stock Unstable UL26 15 42 CC[C@H](NC(=O)/C=C/c1ccccc1OC)c1ccc(C)cc1C ZINC000217967984 DJ In-Stock Unstable U53 0 42 CC[C@H](NC(=O)/C=C/c1ccccc1OC)c1ccc(C)cc1C ZINC000217967984 DJ In-Stock Unstable SCAF_EBVB9 15 42 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(O)cc1 ZINC000217967988 CG For-Sale Anodyne MMP2 0 50 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(O)cc1 ZINC000217967988 CG For-Sale Anodyne MMP9 0 50 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(O)cc1 ZINC000217967988 CG For-Sale Anodyne MMP1 0 50 COC(=O)C[C@H](C1=C(O)C(=O)C([C@H](CC(=O)OC)c2ccc(OC(C)C)c(OC)c2)=C(O)C1=O)c1ccc(OC(C)C)c(OC)c1 ZINC000217968029 KK In-Stock Unstable TNF 22 41 CN(Cc1ccccc1/C=C\C(=O)O)[C@@H]1CCS(=O)(=O)C1 ZINC000217968032 DD For-Sale Unstable PTGER2 36 45 CN(Cc1ccccc1/C=C\C(=O)O)[C@@H]1CCS(=O)(=O)C1 ZINC000217968032 DD For-Sale Unstable PTGER4 0 45 CN(Cc1ccccc1/C=C\C(=O)O)[C@@H]1CCS(=O)(=O)C1 ZINC000217968032 DD For-Sale Unstable PTGER3 15 45 CN(Cc1ccccc1/C=C\C(=O)O)[C@@H]1CCS(=O)(=O)C1 ZINC000217968032 DD For-Sale Unstable PTGDR 0 41 CN[C@@H](Cc1cc(Cl)ccc1OC)[C@@H]1CCC[C@@H](C)C1 ZINC000217968041 CI For-Sale Unstable QRFPR 46 40 N#CCNC(=O)[C@@H]1C[C@@H]2CC[C@@H]1C2 ZINC000217968091 AD For-Sale Unstable CTSK 16 53 CC[C@@H](NC(=O)/C=C/c1ccccc1OC)c1ccc(OC)c(OC)c1 ZINC000217968099 FH In-Stock Unstable KCNQ2 52 38 CC[C@@H](NC(=O)/C=C/c1ccccc1OC)c1ccc(OC)c(OC)c1 ZINC000217968099 FH In-Stock Unstable CYP1A1 17 45 CC[C@@H](NC(=O)/C=C/c1ccccc1OC)c1ccc(OC)c(OC)c1 ZINC000217968099 FH In-Stock Unstable CYSP_PLAFA 47 34 COc1ccc(Cl)cc1NC(=O)N/C=C/c1cccc(F)c1 ZINC000217968101 DI For-Sale Unstable PYGL 0 43 COc1ccc(Cl)cc1NC(=O)N/C=C/c1cccc(F)c1 ZINC000217968101 DI For-Sale Unstable RBP4 24 41 COC(=O)C[C@H](C1=C(O)C(=O)C([C@@H](CC(=O)OC)c2ccc(OC(C)C)c(OC)c2)=C(O)C1=O)c1ccc(OC(C)C)c(OC)c1 ZINC000217968114 KK In-Stock Unstable TNF 22 41 CN[C@@H](Cc1cc(Cl)ccc1OC)[C@H]1CCC[C@@H](C)C1 ZINC000217968126 CI For-Sale Unstable QRFPR 46 40 N#CCNC(=O)[C@@H]1C[C@H]2CC[C@@H]1C2 ZINC000217968172 AD For-Sale Unstable CTSK 16 53 CC[C@H](NC(=O)/C=C/c1ccccc1OC)c1ccc(OC)c(OC)c1 ZINC000217968179 FH In-Stock Unstable KCNQ2 52 38 CC[C@H](NC(=O)/C=C/c1ccccc1OC)c1ccc(OC)c(OC)c1 ZINC000217968179 FH In-Stock Unstable CYP1A1 17 45 CC[C@H](NC(=O)/C=C/c1ccccc1OC)c1ccc(OC)c(OC)c1 ZINC000217968179 FH In-Stock Unstable CYSP_PLAFA 47 34 CCCCc1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217968223 DJ For-Sale Unstable P96878_MYCTU 15 46 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217968242 II For-Sale Unstable ENV 42 33 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217968242 II For-Sale Unstable SCD1 18 43 C[C@@H]1CCN(CCOc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217968268 CF On-Demand Unstable ESR1 45 47 C[C@@H]1CCN(CCOc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217968268 CF On-Demand Unstable SLC6A1 52 34 C[C@@H]1CCN(CCOc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217968268 CF On-Demand Unstable ESR2 30 47 C[C@@H]1CCN(CCOc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217968268 CF On-Demand Unstable LTA4H 48 46 C[C@@H]1CCN(CCOc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217968268 CF On-Demand Unstable HRH3 40 46 C[C@@H]1CCN(CCOc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217968268 CF On-Demand Unstable SIGMAR1 16 50 C[C@@H]1CCN(CCOc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217968268 CF On-Demand Unstable EBP 27 50 C[C@@H]1CCN(CCOc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217968268 CF On-Demand Unstable PSMB1 43 37 CC[C@@H](NC(=O)/C=C/c1ccccc1OC)c1ccc(S(C)(=O)=O)cc1 ZINC000217968286 FG In-Stock Unstable KCNQ2 46 34 CC[C@@H](NC(=O)/C=C/c1ccccc1OC)c1ccc(S(C)(=O)=O)cc1 ZINC000217968286 FG In-Stock Unstable CTSF 44 32 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217968316 II For-Sale Unstable ENV 42 33 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217968316 II For-Sale Unstable SCD1 18 43 Clc1cc(NCCN2CCCCCC2)nc(C2CC2)n1 ZINC000217968320 CG On-Demand Unstable HNMT 49 35 COc1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217968337 CH For-Sale Unstable AHR 24 40 COc1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217968337 CH For-Sale Unstable MTNR1A 29 44 COc1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217968337 CH For-Sale Unstable MTNR1B 27 44 COc1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217968337 CH For-Sale Unstable TUBB2B 15 40 COc1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217968337 CH For-Sale Unstable CA12 16 41 COc1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217968337 CH For-Sale Unstable PDGFRA 38 42 COc1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217968337 CH For-Sale Unstable CA9 16 41 COc1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217968337 CH For-Sale Unstable Q8MMZ8_EIMTE 0 42 COc1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217968337 CH For-Sale Unstable AKR1C3 15 40 COc1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217968337 CH For-Sale Unstable AKR1C2 41 33 COc1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217968337 CH For-Sale Unstable IMDH_CRYPV 15 42 C[C@H]1CCN(CCOc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217968355 CF On-Demand Unstable ESR1 45 47 C[C@H]1CCN(CCOc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217968355 CF On-Demand Unstable SLC6A1 52 34 C[C@H]1CCN(CCOc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217968355 CF On-Demand Unstable ESR2 30 47 C[C@H]1CCN(CCOc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217968355 CF On-Demand Unstable LTA4H 48 46 C[C@H]1CCN(CCOc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217968355 CF On-Demand Unstable HRH3 40 46 C[C@H]1CCN(CCOc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217968355 CF On-Demand Unstable SIGMAR1 16 50 C[C@H]1CCN(CCOc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217968355 CF On-Demand Unstable EBP 27 50 C[C@H]1CCN(CCOc2ccc(/C=C\C(=O)O)cc2)C1 ZINC000217968355 CF On-Demand Unstable PSMB1 43 37 Nc1nc(/C=C\c2c[nH]c3ccc(F)cc23)cs1 ZINC000217968357 CH For-Sale Unstable MPO 78 40 CC[C@H](NC(=O)/C=C/c1ccccc1OC)c1ccc(S(C)(=O)=O)cc1 ZINC000217968380 FG In-Stock Unstable KCNQ2 46 34 CC[C@H](NC(=O)/C=C/c1ccccc1OC)c1ccc(S(C)(=O)=O)cc1 ZINC000217968380 FG In-Stock Unstable CTSF 44 32 Nc1ccc(CCN2CCC[C@@H]3CCCC[C@H]32)cc1 ZINC000217968384 CG For-Sale Unstable HRH3 54 44 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217968405 II For-Sale Unstable ENV 42 33 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217968405 II For-Sale Unstable SCD1 18 43 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)Nc3cc(C)n(C)n3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217968406 KF In-Stock Unstable TUBA1A 20 66 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)Nc3cc(C)n(C)n3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217968406 KF In-Stock Unstable TPPP 0 63 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(Cl)cc1Cl ZINC000217968438 EJ For-Sale Anodyne PYGL 22 40 Nc1nc(/C=C\c2c[nH]c3ccc(Cl)cc23)cs1 ZINC000217968443 CI For-Sale Unstable TDO2 0 50 Nc1nc(/C=C\c2c[nH]c3ccc(Cl)cc23)cs1 ZINC000217968443 CI For-Sale Unstable MAP3K14 28 42 O=[N+]([O-])[C@@H]1[C@H](c2ccc(F)cc2)[C@H]2CC[C@H]1N2Cc1ccccc1 ZINC000217968453 EH For-Sale Unstable SLC6A3 15 47 Nc1ccc(CCN2CCC[C@H]3CCCC[C@H]32)cc1 ZINC000217968472 CG For-Sale Unstable HRH3 58 51 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217968476 II For-Sale Unstable ENV 42 33 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000217968476 II For-Sale Unstable SCD1 18 43 CCNC(=O)Nc1ccc([N+](=O)[O-])cc1Br ZINC000217968489 CE For-Sale Unstable TBXA2R 27 41 C=CCNC(=O)CNc1ccc2c(cc1=O)[C@@H](NC(C)=O)CCc1cc(OC)c(OC)c(OC)c1-2 ZINC000217968519 JF In-Stock Unstable TUBA1A 19 70 C=CCNC(=O)CNc1ccc2c(cc1=O)[C@@H](NC(C)=O)CCc1cc(OC)c(OC)c(OC)c1-2 ZINC000217968519 JF In-Stock Unstable TPPP 0 69 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)Nc1ccccc1 ZINC000217968572 FG For-Sale Unstable AGTR2 21 41 CC1(C)CC(=O)c2c(O)cc(OCC(=O)N3CCCC[C@H]3c3cccnc3)cc2O1 ZINC000217968621 HH In-Stock Unstable COLA 148 47 CC1(C)CC(=O)c2c(O)cc(OCC(=O)N3CCCC[C@H]3c3cccnc3)cc2O1 ZINC000217968621 HH In-Stock Unstable CPT1A 138 47 CC1(C)CC(=O)c2c(O)cc(OCC(=O)N3CCCC[C@H]3c3cccnc3)cc2O1 ZINC000217968621 HH In-Stock Unstable CPT2 48 40 CC1(C)CC(=O)c2c(O)cc(OCC(=O)N3CCCC[C@H]3c3cccnc3)cc2O1 ZINC000217968621 HH In-Stock Unstable GPBAR1 0 40 CC(C)(C)[C@@H]1CC[C@@H](O)[C@@H](N2CCN(S(C)(=O)=O)CC2)C1 ZINC000217968633 DD For-Sale Unstable SLC18A3 15 56 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)Nc1ccccc1 ZINC000217968637 FG For-Sale Unstable AGTR2 21 41 CC(C)NC(=O)N/C=C/c1cccc(F)c1 ZINC000217968654 BF For-Sale Unstable NR1H4 16 46 CCCCN(Cc1cccc(/C=C\C(=O)O)c1)C1CC1 ZINC000217968696 CH For-Sale Unstable AKR1C3 27 43 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)Nc1ccccc1 ZINC000217968719 FG For-Sale Unstable AGTR2 21 41 CCC[C@@H](O)CNC(=O)CCCNC(C)C ZINC000217968740 BD For-Sale Unstable NOD1 42 33 CC(C)N(Cc1ccccc1)C(=O)N/C=C/c1cccc(F)c1 ZINC000217968752 DI For-Sale Unstable NR1H4 29 44 Cc1ccc(NC(=O)OCCCCCl)cc1Cl ZINC000217968763 CI For-Sale Unstable POLC 66 42 Cc1ccc(NC(=O)OCCCCCl)cc1Cl ZINC000217968763 CI For-Sale Unstable AGPAT2 41 36 CC(C)(C)[C@@H]1CC[C@H](O)[C@@H](N2CCN(S(C)(=O)=O)CC2)C1 ZINC000217968802 DD For-Sale Unstable SLC18A3 15 56 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)Nc1ccccc1 ZINC000217968805 FG For-Sale Unstable AGTR2 21 41 CCC[C@H](O)CNC(=O)CCCNC(C)C ZINC000217968820 BD For-Sale Unstable NOD1 42 33 COCCN(Cc1cccc(/C=C\C(=O)O)c1)C1CC1 ZINC000217968829 CE For-Sale Unstable NR1H4 47 37 O=C(CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)Nc1cc(Cl)ccc1O ZINC000217968840 FF In-Stock Unstable PLCD1 0 42 O=C(CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)Nc1cc(Cl)ccc1O ZINC000217968840 FF In-Stock Unstable AGAL_COFAR 0 47 O=C(CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)Nc1cc(Cl)ccc1O ZINC000217968840 FF In-Stock Unstable HSPA8 0 41 O=C(CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)Nc1cc(Cl)ccc1O ZINC000217968840 FF In-Stock Unstable CYTH3 0 42 O=C(CCCC[C@@H]1SC[C@@H]2NC(=O)N[C@H]12)Nc1cc(Cl)ccc1O ZINC000217968840 FF In-Stock Unstable HLCS 0 48 CN(C(=O)N/C=C/c1cccc(F)c1)C1CCCCC1 ZINC000217968860 CH For-Sale Unstable NR1H4 20 42 CCNC(=O)Nc1ccc(F)cc1[N+](=O)[O-] ZINC000217968871 BD For-Sale Unstable COLA 19 42 NNC(=O)Cc1ccc(CN2C[C@H]3[C@H](O)CC[C@H]3C2)cc1 ZINC000217968886 CC For-Sale Unstable SIGMAR1 16 40 NNC(=O)Cc1ccc(CN2C[C@H]3[C@H](O)CC[C@H]3C2)cc1 ZINC000217968886 CC For-Sale Unstable AOC2 0 43 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccccc3OC)n2)c(OC)c1 ZINC000217968929 GG In-Stock Unstable CYP1B1 31 42 COc1ccc(-c2noc(CNC(=O)/C=C/c3ccccc3OC)n2)c(OC)c1 ZINC000217968929 GG In-Stock Unstable IMPDH2 0 44 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)Nc3cccc(-c4nnn(C)n4)c3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217968949 KG In-Stock Unstable TUBA1A 16 59 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)Nc3cccc(-c4nnn(C)n4)c3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217968949 KG In-Stock Unstable TPPP 0 56 O=C(NCc1ccc(Cl)cc1)[C@@H]1CC[C@@H](Cn2cnnn2)CC1 ZINC000217968997 EE In-Stock Unstable SLC6A1 0 46 CN[C@@H](CCCc1ccccc1)[C@@H]1CCC[C@@H](C)C1 ZINC000217969015 CI For-Sale Unstable SLC18A2 40 43 CN[C@@H](CCCc1ccccc1)[C@@H]1CCC[C@@H](C)C1 ZINC000217969015 CI For-Sale Unstable MMP3 17 42 CN[C@@H](CCCc1ccccc1)[C@@H]1CCC[C@@H](C)C1 ZINC000217969015 CI For-Sale Unstable BIRC2 34 44 COC(=O)C[C@H](c1ccc(OC(=O)c2ccc(OC)cc2)cc1)c1oc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c1O ZINC000217969053 KI In-Stock Unstable CHRNA4 25 41 CN[C@@H](CCCc1ccccc1)[C@H]1CCC[C@@H](C)C1 ZINC000217969097 CI For-Sale Unstable SLC18A2 40 43 CN[C@@H](CCCc1ccccc1)[C@H]1CCC[C@@H](C)C1 ZINC000217969097 CI For-Sale Unstable MMP3 17 42 CN[C@@H](CCCc1ccccc1)[C@H]1CCC[C@@H](C)C1 ZINC000217969097 CI For-Sale Unstable BIRC2 34 44 CCCOc1cccc(/C=C2/CC(=O)NC2=O)c1 ZINC000217969105 BD For-Sale Unstable HPGD 42 33 COC(=O)C[C@@H](c1ccc(OC(=O)c2ccc(OC)cc2)cc1)c1oc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c1O ZINC000217969126 KI In-Stock Unstable CHRNA4 25 41 O=C(O)/C=C\c1cc(F)ccc1CN1CCC[C@H](O)C1 ZINC000217969171 CD For-Sale Unstable SLC6A1 109 44 O=C(O)/C=C\c1cc(F)ccc1CN1CCC[C@H](O)C1 ZINC000217969171 CD For-Sale Unstable CCR3 26 40 O=C(O)/C=C\c1cc(CN2CCC[C@H](O)C2)ccc1F ZINC000217969271 CD For-Sale Unstable SLC6A1 91 37 O=C(O)/C=C\c1cc(CN2CCC[C@H](O)C2)ccc1F ZINC000217969271 CD For-Sale Unstable CCR3 25 40 CCC[C@@H](O)CNC(=O)[C@@H](C)CCN ZINC000217969278 BC For-Sale Unstable DPP7 23 40 CCc1ncnc(NCc2cccc(F)c2)c1F ZINC000217969306 BF On-Demand Unstable EGFR 23 49 CCc1ncnc(NCc2cccc(F)c2)c1F ZINC000217969306 BF On-Demand Unstable CLK4 24 49 CCc1ncnc(NCc2cccc(F)c2)c1F ZINC000217969306 BF On-Demand Unstable USP10 0 43 CCc1ncnc(NCc2cccc(F)c2)c1F ZINC000217969306 BF On-Demand Unstable USP13 0 43 Cc1nc2n(c1C(=O)O)CCC[C@H]2OCc1ccccc1 ZINC000217969326 CF For-Sale Unstable PREP 58 38 Cc1nc2n(c1C(=O)O)CCC[C@H]2OCc1ccccc1 ZINC000217969326 CF For-Sale Unstable SLC12A5 49 34 O=C(N/C=C/c1cccc(F)c1)NC1CCCCC1 ZINC000217969340 CG For-Sale Unstable FAAH 0 47 O=C(N/C=C/c1cccc(F)c1)NC1CCCCC1 ZINC000217969340 CG For-Sale Unstable EPHX2 27 43 C[C@H](C(=O)NN)c1ccc(CN2CC[C@@H](C)[C@@H](C)C2)cc1 ZINC000217969344 CE For-Sale Unstable MLNR 43 42 CCC[C@H](O)CNC(=O)[C@@H](C)CCN ZINC000217969364 BC For-Sale Unstable DPP7 23 40 COc1ccccc1/C=C/C(=O)N(C)Cc1nc(-c2ccc(C)cc2)no1 ZINC000217969367 FH In-Stock Unstable LUCI_PHOPE 28 40 Cc1nc2n(c1C(=O)O)CCC[C@@H]2OCc1ccccc1 ZINC000217969409 CF For-Sale Unstable PREP 58 38 Cc1nc2n(c1C(=O)O)CCC[C@@H]2OCc1ccccc1 ZINC000217969409 CF For-Sale Unstable SLC12A5 49 34 CCC[C@@H](O)CNC(=O)[C@H](C)CCN ZINC000217969442 BC For-Sale Unstable DPP7 23 40 Cc1occc1CN(C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217969498 CG For-Sale Unstable PTGER2 22 42 CCC[C@H](O)CNC(=O)[C@H](C)CCN ZINC000217969514 BC For-Sale Unstable DPP7 23 40 CN(C)c1ccc(CCC(=O)N2CCC[C@@H](N(C)C)CC2)cc1 ZINC000217969536 DF In-Stock Unstable L3MBTL1 0 40 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1ccc(C#N)cc1Br ZINC000217969573 EK For-Sale Unstable TRPM8 0 40 CCCNC(=O)N1C[C@H](Oc2ccccc2F)C[C@@H]1C(=O)OC ZINC000217969576 DD For-Sale Unstable ASAH1 58 34 COc1ccc(-c2noc(CN(C)C(=O)/C=C/c3ccccc3OC)n2)cc1 ZINC000217969578 GG In-Stock Unstable LUCI_PHOPE 29 40 CCC1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217969620 CG For-Sale Unstable ACHE 33 45 CCC1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217969620 CG For-Sale Unstable PTGER2 43 45 CCC1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217969620 CG For-Sale Unstable PTGER4 0 45 CCC1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217969620 CG For-Sale Unstable SIGMAR1 42 40 CCC1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217969620 CG For-Sale Unstable PTGER3 16 45 CCC1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217969620 CG For-Sale Unstable CCR3 34 42 CN(C)c1ccc(CCC(=O)N2CCC[C@H](N(C)C)CC2)cc1 ZINC000217969630 DF In-Stock Unstable L3MBTL1 0 40 CCCNC(=O)N1C[C@@H](Oc2ccccc2F)C[C@@H]1C(=O)OC ZINC000217969648 DD For-Sale Unstable ASAH1 58 34 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1ccc(C#N)cc1Br ZINC000217969649 EK For-Sale Unstable TRPM8 0 40 Nc1ccc(N2CCC[C@@H]3CCCC[C@H]32)cn1 ZINC000217969663 BF For-Sale Unstable GCKR 69 37 O=C([C@@H]1CC[C@@H](Cn2cnnn2)CC1)N1CCN(c2ccccc2)CC1 ZINC000217969670 FD In-Stock Unstable ERBB2 0 43 O=C([C@@H]1CC[C@@H](Cn2cnnn2)CC1)N1CCN(c2ccccc2)CC1 ZINC000217969670 FD In-Stock Unstable MMP2 0 43 O=C([C@@H]1CC[C@@H](Cn2cnnn2)CC1)N1CCN(c2ccccc2)CC1 ZINC000217969670 FD In-Stock Unstable ADAM10 34 43 O=C(N/C=C/c1cccc(F)c1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217969675 HJ For-Sale Unstable NMUR2 0 45 O=C(N/C=C/c1cccc(F)c1)N1CCN(C(c2ccccc2)c2ccccc2)CC1 ZINC000217969675 HJ For-Sale Unstable NMUR1 0 45 COc1ccc(-c2noc(CN(C)C(=O)/C=C/c3ccccc3OC)n2)c(OC)c1 ZINC000217969680 HG In-Stock Unstable CYP1B1 30 41 NC(=O)COc1ccc(/C=C2/CC(=O)NC2=O)cc1 ZINC000217969685 CB For-Sale Unstable TRY1_BOVIN 40 35 NC(=O)COc1ccc(/C=C2/CC(=O)NC2=O)cc1 ZINC000217969685 CB For-Sale Unstable HPGD 62 39 O=C(Cn1nnc(-c2ccc(Cl)cc2)n1)NCc1ccccc1CN1CCCC1 ZINC000217969705 HF On-Demand Unstable SCN2A 19 42 O=C(Cn1nnc(-c2ccc(Cl)cc2)n1)NCc1ccccc1CN1CCCC1 ZINC000217969705 HF On-Demand Unstable SCN10A 37 42 O=C(Cn1nnc(-c2ccc(Cl)cc2)n1)NCc1ccccc1CN1CCCC1 ZINC000217969705 HF On-Demand Unstable SCARB1 46 44 COc1ccc(S(=O)(=O)[C@H]2C[C@@H](C)CC[C@@H]2C#N)cc1 ZINC000217969707 CF For-Sale Unstable CHRM2 16 42 COc1ccc(S(=O)(=O)[C@H]2C[C@@H](C)CC[C@@H]2C#N)cc1 ZINC000217969707 CF For-Sale Unstable MMP13 24 47 COc1ccc(S(=O)(=O)[C@H]2C[C@@H](C)CC[C@@H]2C#N)cc1 ZINC000217969707 CF For-Sale Unstable MMP8 15 45 COc1ccc(S(=O)(=O)[C@H]2C[C@@H](C)CC[C@@H]2C#N)cc1 ZINC000217969707 CF For-Sale Unstable MMP1 25 45 CCCNC(=O)N1C[C@H](Oc2ccccc2F)C[C@H]1C(=O)OC ZINC000217969724 DD For-Sale Unstable ASAH1 58 34 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1ccc(C#N)cc1Br ZINC000217969728 EK For-Sale Unstable TRPM8 0 40 CCCCN(C)Cc1cc(/C=C\C(=O)O)ccc1OC ZINC000217969732 CG For-Sale Unstable AKR1C3 29 44 Nc1ccc(N2CCC[C@H]3CCCC[C@H]32)cn1 ZINC000217969735 BF For-Sale Unstable GCKR 69 37 CCCNC(=O)N1C[C@@H](Oc2ccccc2F)C[C@H]1C(=O)OC ZINC000217969796 DD For-Sale Unstable ASAH1 58 34 COc1ccc(S(=O)(=O)[C@H]2C[C@H](C)CC[C@@H]2C#N)cc1 ZINC000217969799 CF For-Sale Unstable CHRM2 16 42 COc1ccc(S(=O)(=O)[C@H]2C[C@H](C)CC[C@@H]2C#N)cc1 ZINC000217969799 CF For-Sale Unstable MMP13 24 47 COc1ccc(S(=O)(=O)[C@H]2C[C@H](C)CC[C@@H]2C#N)cc1 ZINC000217969799 CF For-Sale Unstable MMP8 15 45 COc1ccc(S(=O)(=O)[C@H]2C[C@H](C)CC[C@@H]2C#N)cc1 ZINC000217969799 CF For-Sale Unstable MMP1 25 45 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1ccc(C#N)cc1Br ZINC000217969806 EK For-Sale Unstable TRPM8 0 40 C[C@@H]1C[C@@H](C)[C@@H](C)N(Cc2ccc(CC(=O)NN)cc2)C1 ZINC000217969817 CE For-Sale Unstable AOC2 0 40 Cn1cc(S(=O)(=O)N2CCCN(C(=O)NCc3cccc4ccccc34)CC2)cn1 ZINC000217969821 IE In-Stock Unstable TGM2 30 41 Cn1cc(S(=O)(=O)N2CCCN(C(=O)NCc3cccc4ccccc34)CC2)cn1 ZINC000217969821 IE In-Stock Unstable F13A1 37 41 Cn1cc(S(=O)(=O)N2CCCN(C(=O)NCc3cccc4ccccc34)CC2)cn1 ZINC000217969821 IE In-Stock Unstable NAMPT 53 42 COCc1n[nH]c(-c2cccc(NC(=O)CCCNc3ccc4c(cc3=O)[C@@H](NC(C)=O)CCc3cc(OC)c(OC)c(OC)c3-4)c2)n1 ZINC000217969823 KJ In-Stock Unstable TUBA1A 15 54 CCCCN(C)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217969843 CG For-Sale Unstable PTGER2 32 43 CCCCN(C)Cc1ccc(OC)c(/C=C\C(=O)O)c1 ZINC000217969843 CG For-Sale Unstable PTGER4 0 43 CC[C@@H]1CC[C@@H](C#N)[C@@H](S(=O)(=O)c2ccc(OC)cc2)C1 ZINC000217969884 DG For-Sale Unstable MMP13 25 44 CC[C@@H]1CC[C@@H](C#N)[C@@H](S(=O)(=O)c2ccc(OC)cc2)C1 ZINC000217969884 DG For-Sale Unstable MMP8 20 42 CC[C@@H]1CC[C@@H](C#N)[C@@H](S(=O)(=O)c2ccc(OC)cc2)C1 ZINC000217969884 DG For-Sale Unstable MMP1 25 42 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)Nc1ccc(F)cc1 ZINC000217969896 GG For-Sale Unstable AGTR2 15 44 O=C(C1CCN(c2nc3ccccc3o2)CC1)N1CCN(c2cccc(O)c2)CC1 ZINC000217969921 HG On-Demand Unstable SSTR2 50 35 O=C(C1CCN(c2nc3ccccc3o2)CC1)N1CCN(c2cccc(O)c2)CC1 ZINC000217969921 HG On-Demand Unstable HTR7 18 45 O=C(C1CCN(c2nc3ccccc3o2)CC1)N1CCN(c2cccc(O)c2)CC1 ZINC000217969921 HG On-Demand Unstable CCKAR 23 40 O=C(C1CCN(c2nc3ccccc3o2)CC1)N1CCN(c2cccc(O)c2)CC1 ZINC000217969921 HG On-Demand Unstable SSTR1 58 37 O=C(C1CCN(c2nc3ccccc3o2)CC1)N1CCN(c2cccc(O)c2)CC1 ZINC000217969921 HG On-Demand Unstable NPBWR1 40 40 CCCOc1ccc([C@@H](NC)[C@@H]2CCC[C@@H](C)C2)cc1 ZINC000217969949 CJ For-Sale Unstable ACACA 33 41 CCCOc1ccc([C@@H](NC)[C@@H]2CCC[C@@H](C)C2)cc1 ZINC000217969949 CJ For-Sale Unstable ACACB 16 41 C[C@H]1C[C@@H](C)CN(Cc2ccc(CC(=O)NN)cc2)[C@@H]1C ZINC000217969968 CE For-Sale Unstable AOC2 0 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)Nc1ccc(F)cc1 ZINC000217969979 GG For-Sale Unstable AGTR2 15 44 CCCCNC(=O)N/C=C/c1cccc(F)c1 ZINC000217969991 BF For-Sale Unstable ACAT 0 45 O=C(COc1ccc(Oc2ccccc2)cc1)N1CCN(c2cccc(O)c2)CC1 ZINC000217970017 HH On-Demand Unstable HTR1A 21 51 O=C(COc1ccc(Oc2ccccc2)cc1)N1CCN(c2cccc(O)c2)CC1 ZINC000217970017 HH On-Demand Unstable HTR1D 19 51 O=C(COc1ccc(Oc2ccccc2)cc1)N1CCN(c2cccc(O)c2)CC1 ZINC000217970017 HH On-Demand Unstable HTR1B 21 48 O=C(COc1ccc(Oc2ccccc2)cc1)N1CCN(c2cccc(O)c2)CC1 ZINC000217970017 HH On-Demand Unstable HTR7 20 41 O=C(COc1ccc(Oc2ccccc2)cc1)N1CCN(c2cccc(O)c2)CC1 ZINC000217970017 HH On-Demand Unstable COLA 128 53 O=C(COc1ccc(Oc2ccccc2)cc1)N1CCN(c2cccc(O)c2)CC1 ZINC000217970017 HH On-Demand Unstable CPT1A 118 53 O=C(COc1ccc(Oc2ccccc2)cc1)N1CCN(c2cccc(O)c2)CC1 ZINC000217970017 HH On-Demand Unstable CPT2 52 53 O=C(COc1ccc(Oc2ccccc2)cc1)N1CCN(c2cccc(O)c2)CC1 ZINC000217970017 HH On-Demand Unstable GRM5 18 54 O=C(COc1ccc(Oc2ccccc2)cc1)N1CCN(c2cccc(O)c2)CC1 ZINC000217970017 HH On-Demand Unstable FAAH 20 40 CCCOc1ccc([C@H](NC)[C@@H]2CCC[C@@H](C)C2)cc1 ZINC000217970021 CJ For-Sale Unstable ACACA 33 41 CCCOc1ccc([C@H](NC)[C@@H]2CCC[C@@H](C)C2)cc1 ZINC000217970021 CJ For-Sale Unstable ACACB 16 41 Cc1ccc(S(=O)(=O)N2CCCN(S(=O)(=O)c3cnn(C)c3)CC2)cc1 ZINC000217970038 GC In-Stock Unstable PKM 37 43 Cc1ccc(S(=O)(=O)N2CCCN(S(=O)(=O)c3cnn(C)c3)CC2)cc1 ZINC000217970038 GC In-Stock Unstable AKR1C3 0 40 CC[C@@H]1CC[C@H](C#N)[C@@H](S(=O)(=O)c2ccc(OC)cc2)C1 ZINC000217970040 DG For-Sale Unstable MMP13 25 44 CC[C@@H]1CC[C@H](C#N)[C@@H](S(=O)(=O)c2ccc(OC)cc2)C1 ZINC000217970040 DG For-Sale Unstable MMP8 20 42 CC[C@@H]1CC[C@H](C#N)[C@@H](S(=O)(=O)c2ccc(OC)cc2)C1 ZINC000217970040 DG For-Sale Unstable MMP1 25 42 [N-]=[N+]=NCCCNCc1ccccc1 ZINC000217970046 AE For-Sale Unstable GPM3 0 58 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)Nc1ccc(F)cc1 ZINC000217970055 GG For-Sale Unstable AGTR2 15 44 O=C(O)[C@@H]1CCCN(C2CCN(C(=O)c3ccc(Cl)cc3O)CC2)C1 ZINC000217970075 FE In-Stock Unstable SLC6A1 138 39 O=C(O)[C@@H]1CCCN(C2CCN(C(=O)c3ccc(Cl)cc3O)CC2)C1 ZINC000217970075 FE In-Stock Unstable L3MBTL1 0 50 O=C(O)[C@@H]1CCCN(C2CCN(C(=O)c3ccc(Cl)cc3O)CC2)C1 ZINC000217970075 FE In-Stock Unstable L3MBTL3 116 50 O=C(O)[C@@H]1CCCN(C2CCN(C(=O)c3ccc(Cl)cc3O)CC2)C1 ZINC000217970075 FE In-Stock Unstable L3MBTL4 0 43 O=C(O)[C@@H]1CCCN(C2CCN(C(=O)c3ccc(Cl)cc3O)CC2)C1 ZINC000217970075 FE In-Stock Unstable MBTD1 0 49 O=C(O)[C@@H]1CCCN(C2CCN(C(=O)c3ccc(Cl)cc3O)CC2)C1 ZINC000217970075 FE In-Stock Unstable TP53BP1 0 50 CCCOc1ccc([C@@H](NC)[C@H]2CCC[C@@H](C)C2)cc1 ZINC000217970103 CJ For-Sale Unstable ACACA 33 41 CCCOc1ccc([C@@H](NC)[C@H]2CCC[C@@H](C)C2)cc1 ZINC000217970103 CJ For-Sale Unstable ACACB 16 41 CC(=O)N1CC(Nc2ccc3oc(-c4ccc(C(C)C)cc4)cc(=O)c3c2)=CC1=O ZINC000217970106 HI In-Stock Unstable TNKS 28 49 COc1ccccc1/C=C/C(=O)NCCCc1ccc(C(C)C)cc1 ZINC000217970113 EJ In-Stock Unstable DRD2 16 56 COc1ccccc1/C=C/C(=O)NCCCc1ccc(C(C)C)cc1 ZINC000217970113 EJ In-Stock Unstable DRD3 29 56 COc1ccccc1/C=C/C(=O)NCCCc1ccc(C(C)C)cc1 ZINC000217970113 EJ In-Stock Unstable AKR1B10 32 41 CCC[C@@H](NC(=O)NCc1ccc(F)cc1)C(=O)N1CCN(c2cccc(O)c2)CC1 ZINC000217970123 IF On-Demand Unstable P2RY12 113 38 CCC[C@@H](NC(=O)NCc1ccc(F)cc1)C(=O)N1CCN(c2cccc(O)c2)CC1 ZINC000217970123 IF On-Demand Unstable MC4R 46 38 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)Nc1ccc(F)cc1 ZINC000217970130 GG For-Sale Unstable AGTR2 15 44 O=C(O)[C@H]1CCCN(C2CCN(C(=O)c3ccc(Cl)cc3O)CC2)C1 ZINC000217970140 FE In-Stock Unstable SLC6A1 138 39 O=C(O)[C@H]1CCCN(C2CCN(C(=O)c3ccc(Cl)cc3O)CC2)C1 ZINC000217970140 FE In-Stock Unstable L3MBTL1 0 50 O=C(O)[C@H]1CCCN(C2CCN(C(=O)c3ccc(Cl)cc3O)CC2)C1 ZINC000217970140 FE In-Stock Unstable L3MBTL3 116 50 O=C(O)[C@H]1CCCN(C2CCN(C(=O)c3ccc(Cl)cc3O)CC2)C1 ZINC000217970140 FE In-Stock Unstable L3MBTL4 0 43 O=C(O)[C@H]1CCCN(C2CCN(C(=O)c3ccc(Cl)cc3O)CC2)C1 ZINC000217970140 FE In-Stock Unstable MBTD1 0 49 O=C(O)[C@H]1CCCN(C2CCN(C(=O)c3ccc(Cl)cc3O)CC2)C1 ZINC000217970140 FE In-Stock Unstable TP53BP1 0 50 Cn1cc(S(=O)(=O)N2CCCN(S(=O)(=O)c3ccc(Cl)cc3)CC2)cn1 ZINC000217970168 HD In-Stock Unstable PKM 43 49 CCC[C@H](NC(=O)NCc1ccc(F)cc1)C(=O)N1CCN(c2cccc(O)c2)CC1 ZINC000217970185 IF On-Demand Unstable P2RY12 113 38 CCC[C@H](NC(=O)NCc1ccc(F)cc1)C(=O)N1CCN(c2cccc(O)c2)CC1 ZINC000217970185 IF On-Demand Unstable MC4R 46 38 CCCOc1ccc([C@H](NC)[C@H]2CCC[C@@H](C)C2)cc1 ZINC000217970192 CJ For-Sale Unstable ACACA 33 41 CCCOc1ccc([C@H](NC)[C@H]2CCC[C@@H](C)C2)cc1 ZINC000217970192 CJ For-Sale Unstable ACACB 16 41 COC(=O)C[C@@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(OCCc2ccc(OC)cc2)c(OC)c1 ZINC000217970211 KJ In-Stock Unstable TNF 21 42 COC(=O)C[C@@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(OCCc2ccc(OC)cc2)c(OC)c1 ZINC000217970211 KJ In-Stock Unstable MTNR1B 19 42 COc1ccccc1/C=C/C(=O)NCCCN(C)c1ccccc1 ZINC000217970223 DG In-Stock Unstable DRD3 25 56 C[C@H](C(=O)NN)c1ccc(CN2CC[C@@H](O)[C@@H](C)C2)cc1 ZINC000217970243 CC For-Sale Unstable MLNR 40 41 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217970260 II For-Sale Unstable TRPM8 62 44 CC(=O)Nc1ccc(S(=O)(=O)N2CCCN(S(=O)(=O)c3cnn(C)c3)CC2)cc1 ZINC000217970268 IC In-Stock Unstable LPL 44 34 CC(=O)Nc1ccc(S(=O)(=O)N2CCCN(S(=O)(=O)c3cnn(C)c3)CC2)cc1 ZINC000217970268 IC In-Stock Unstable TGM2 82 45 CC(=O)Nc1ccc(S(=O)(=O)N2CCCN(S(=O)(=O)c3cnn(C)c3)CC2)cc1 ZINC000217970268 IC In-Stock Unstable F13A1 104 50 CC(=O)Nc1ccc(S(=O)(=O)N2CCCN(S(=O)(=O)c3cnn(C)c3)CC2)cc1 ZINC000217970268 IC In-Stock Unstable RAC1 0 42 CC(=O)Nc1ccc(S(=O)(=O)N2CCCN(S(=O)(=O)c3cnn(C)c3)CC2)cc1 ZINC000217970268 IC In-Stock Unstable NAMPT 58 47 CC(=O)Nc1ccc(S(=O)(=O)N2CCCN(S(=O)(=O)c3cnn(C)c3)CC2)cc1 ZINC000217970268 IC In-Stock Unstable DDIT3 0 42 COC(=O)C[C@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(OCCc2ccc(OC)cc2)c(OC)c1 ZINC000217970293 KJ In-Stock Unstable TNF 21 42 COC(=O)C[C@H](C1=C(O)C(=O)c2ccccc2C1=O)c1ccc(OCCc2ccc(OC)cc2)c(OC)c1 ZINC000217970293 KJ In-Stock Unstable MTNR1B 19 42 O=C1C/C(=C\c2ccc3c(c2)OCCO3)C(=O)N1 ZINC000217970299 BC For-Sale Unstable DYRK1A 23 44 O=C1C/C(=C\c2ccc3c(c2)OCCO3)C(=O)N1 ZINC000217970299 BC For-Sale Unstable CLK1 37 44 O=C1C/C(=C\c2ccc3c(c2)OCCO3)C(=O)N1 ZINC000217970299 BC For-Sale Unstable DYRK2 75 44 COc1ccccc1/C=C/C(=O)NCCCN1CCCc2ccccc21 ZINC000217970330 FH In-Stock Unstable HTR1A 37 40 COc1ccccc1/C=C/C(=O)NCCCN1CCCc2ccccc21 ZINC000217970330 FH In-Stock Unstable DRD2 36 63 COc1ccccc1/C=C/C(=O)NCCCN1CCCc2ccccc21 ZINC000217970330 FH In-Stock Unstable DRD1 0 49 COc1ccccc1/C=C/C(=O)NCCCN1CCCc2ccccc21 ZINC000217970330 FH In-Stock Unstable HTR2A 22 49 COc1ccccc1/C=C/C(=O)NCCCN1CCCc2ccccc21 ZINC000217970330 FH In-Stock Unstable ADRA1A 19 44 COc1ccccc1/C=C/C(=O)NCCCN1CCCc2ccccc21 ZINC000217970330 FH In-Stock Unstable DRD3 55 63 C[C@H]1C[C@@H](C)CN(Cc2cccc(/C=C\C(=O)O)c2)C1 ZINC000217970334 CG For-Sale Unstable SIGMAR1 20 44 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217970338 II For-Sale Unstable TRPM8 62 44 COc1ccc(S(=O)(=O)N2CCCN(S(=O)(=O)c3cnn(C)c3)CC2)cc1OC ZINC000217970384 IC In-Stock Unstable HTR6 16 40 COc1ccc(S(=O)(=O)N2CCCN(S(=O)(=O)c3cnn(C)c3)CC2)cc1OC ZINC000217970384 IC In-Stock Unstable PKM 42 43 O=C(c1n[nH]c2c1CCCC2)N1CCCC[C@H]1c1cccnc1 ZINC000217970394 DG In-Stock Unstable CHRNA2 41 43 O=C(c1n[nH]c2c1CCCC2)N1CCCC[C@H]1c1cccnc1 ZINC000217970394 DG In-Stock Unstable COLA 64 39 O=C(c1n[nH]c2c1CCCC2)N1CCCC[C@H]1c1cccnc1 ZINC000217970394 DG In-Stock Unstable CPT1A 62 36 O=C(c1n[nH]c2c1CCCC2)N1CCCC[C@H]1c1cccnc1 ZINC000217970394 DG In-Stock Unstable GPBAR1 0 45 O=C(N/C=C/c1cccc(F)c1)N1CCCc2ccccc21 ZINC000217970401 CH For-Sale Unstable AVPR2 46 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217970417 II For-Sale Unstable TRPM8 62 44 COc1cc(CNC(=O)CSc2ccccc2)ccc1OC(C)C ZINC000217970444 EH In-Stock Unstable HCRTR1 18 40 COc1cc(CNC(=O)CSc2ccccc2)ccc1OC(C)C ZINC000217970444 EH In-Stock Unstable TRPV1 24 41 COc1cc(CNC(=O)CSc2ccccc2)ccc1OC(C)C ZINC000217970444 EH In-Stock Unstable PDE10A 15 45 COc1cc(CNC(=O)CSc2ccccc2)ccc1OC(C)C ZINC000217970444 EH In-Stock Unstable ENPP1 58 34 COc1cc(CNC(=O)CSc2ccccc2)ccc1OC(C)C ZINC000217970444 EH In-Stock Unstable FAS 58 40 O=C(/C=C\c1ccc(F)cc1F)CCl ZINC000217970463 BF For-Sale Unstable BOTA 15 44 Cn1cc(S(=O)(=O)N2CCCN(S(=O)(=O)c3cccs3)CC2)cn1 ZINC000217970490 GC In-Stock Unstable GCK 0 44 Cn1cc(S(=O)(=O)N2CCCN(S(=O)(=O)c3cccs3)CC2)cn1 ZINC000217970490 GC In-Stock Unstable GCKR 38 44 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000217970497 II For-Sale Unstable TRPM8 62 44 COc1cc2c(cc1OC)CN(C(=O)c1c(C)cc(C)n(C[C@@H]3CCCO3)c1=O)CC2 ZINC000217970499 IF In-Stock Unstable ABCB1B 51 32 COc1cc2c(cc1OC)CN(C(=O)c1c(C)cc(C)n(C[C@@H]3CCCO3)c1=O)CC2 ZINC000217970499 IF In-Stock Unstable ABCB1 0 41 CCS(=O)(=O)[C@@H]1C[C@@]1(N)C(=O)O ZINC000217970520 AA In-Stock Unstable GRM2 0 44 CCS(=O)(=O)[C@@H]1C[C@@]1(N)C(=O)O ZINC000217970520 AA In-Stock Unstable GRM1 0 44 CC(C)N1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217970528 CE For-Sale Unstable PTGER2 44 46 CC(C)N1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217970528 CE For-Sale Unstable PTGER4 21 46 CC(C)N1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217970528 CE For-Sale Unstable PTGER3 18 46 CC(C)N1CCN(Cc2ccccc2/C=C\C(=O)O)CC1 ZINC000217970528 CE For-Sale Unstable PTGDR 17 44 O=C(/C=C\c1ccc(-c2ccccc2)cc1)CCl ZINC000217970548 CI For-Sale Unstable NA 0 41 O=C(/C=C\c1ccc(-c2ccccc2)cc1)CCl ZINC000217970548 CI For-Sale Unstable LTB4R 0 48 O=C(/C=C\c1ccc(-c2ccccc2)cc1)CCl ZINC000217970548 CI For-Sale Unstable F3 26 47 O=C(/C=C\c1ccc(-c2ccccc2)cc1)CCl ZINC000217970548 CI For-Sale Unstable MMP2 15 41 O=C(/C=C\c1ccc(-c2ccccc2)cc1)CCl ZINC000217970548 CI For-Sale Unstable HDAC1 20 43 O=C(/C=C\c1ccc(-c2ccccc2)cc1)CCl ZINC000217970548 CI For-Sale Unstable HDAC2 15 59 O=C(/C=C\c1ccc(-c2ccccc2)cc1)CCl ZINC000217970548 CI For-Sale Unstable HDAC6 26 43 O=C(/C=C\c1ccc(-c2ccccc2)cc1)CCl ZINC000217970548 CI For-Sale Unstable 17HSDCL 0 41 O=C(/C=C\c1ccc(-c2ccccc2)cc1)CCl ZINC000217970548 CI For-Sale Unstable SSSIM 15 47 COc1cc2c(cc1OC)CN(C(=O)c1c(C)cc(C)n(C[C@H]3CCCO3)c1=O)CC2 ZINC000217970577 IF In-Stock Unstable ABCB1B 51 32 COc1cc2c(cc1OC)CN(C(=O)c1c(C)cc(C)n(C[C@H]3CCCO3)c1=O)CC2 ZINC000217970577 IF In-Stock Unstable ABCB1 0 41 CCS(=O)(=O)[C@H]1C[C@@]1(N)C(=O)O ZINC000217970592 AA In-Stock Unstable GRM2 0 44 CCS(=O)(=O)[C@H]1C[C@@]1(N)C(=O)O ZINC000217970592 AA In-Stock Unstable GRM1 0 44 O=C(N/C=C/c1cccc(F)c1)NC1CCCC1 ZINC000217970605 BG For-Sale Unstable CCR3 19 41 O=C(N/C=C/c1cccc(F)c1)NC1CCCC1 ZINC000217970605 BG For-Sale Unstable EPHX2 22 42 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)Nc1cccc(OC)c1 ZINC000217970613 GG For-Sale Unstable CCR3 22 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)Nc1cccc(OC)c1 ZINC000217970613 GG For-Sale Unstable TAAR1 31 44 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)Nc1cccc(OC)c1 ZINC000217970613 GG For-Sale Unstable LIMK2 23 42 CC(C)(C)c1ccc(/C=C\C(=O)CCl)cc1 ZINC000217970623 BH For-Sale Unstable SSSIM 15 47 CC(C)N1CCN(Cc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217970632 CE For-Sale Unstable HRH3 15 51 CC(C)N1CCN(Cc2ccc(/C=C\C(=O)O)cc2)CC1 ZINC000217970632 CE For-Sale Unstable SIGMAR1 21 46 O=C(CSc1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217970656 DI In-Stock Unstable SCN5A 0 45 O=C(CSc1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217970656 DI In-Stock Unstable SLC6A5 20 41 O=C(CSc1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217970656 DI In-Stock Unstable NCE103 23 41 O=C(CSc1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217970656 DI In-Stock Unstable CRTM 46 47 O=C(CSc1ccccc1)NCCCc1ccc(Cl)cc1 ZINC000217970656 DI In-Stock Unstable CAN2 0 41 CCS(=O)(=O)[C@@H]1C[C@]1(N)C(=O)O ZINC000217970665 AA In-Stock Unstable GRM2 0 44 CCS(=O)(=O)[C@@H]1C[C@]1(N)C(=O)O ZINC000217970665 AA In-Stock Unstable GRM1 0 44 COc1ccc(CC(=O)N[C@@H]2CCC[C@@H]2CO)cc1F ZINC000217970679 CD On-Demand Unstable PDE4D 20 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)Nc1cccc(OC)c1 ZINC000217970684 GG For-Sale Unstable CCR3 22 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)Nc1cccc(OC)c1 ZINC000217970684 GG For-Sale Unstable TAAR1 31 44 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)Nc1cccc(OC)c1 ZINC000217970684 GG For-Sale Unstable LIMK2 23 42 COc1ccc(F)cc1S(=O)(=O)N1CCCN(S(=O)(=O)c2cnn(C)c2)CC1 ZINC000217970699 IC In-Stock Unstable PKM 31 41 Cc1nnc(CNC(=O)c2ccc(CN3CCc4ccccc4C3)cc2)o1 ZINC000217970701 FF In-Stock Unstable HDAC6 28 41 Cc1nnc(CNC(=O)c2ccc(CN3CCc4ccccc4C3)cc2)o1 ZINC000217970701 FF In-Stock Unstable NOD1 42 53 Cc1nnc(CNC(=O)c2ccc(CN3CCc4ccccc4C3)cc2)o1 ZINC000217970701 FF In-Stock Unstable NOD2 63 53 O=C(N/C=C/c1cccc(F)c1)NCc1ccccc1Cl ZINC000217970704 DH For-Sale Unstable P2RX7 64 39 CCS(=O)(=O)[C@H]1C[C@]1(N)C(=O)O ZINC000217970727 AA In-Stock Unstable GRM2 0 44 CCS(=O)(=O)[C@H]1C[C@]1(N)C(=O)O ZINC000217970727 AA In-Stock Unstable GRM1 0 44 CC(C)N1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217970734 CE For-Sale Unstable DRD2 18 42 CC(C)N1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217970734 CE For-Sale Unstable SIGMAR1 30 46 CC(C)N1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217970734 CE For-Sale Unstable HDAC8 44 37 CC(C)N1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217970734 CE For-Sale Unstable HDAC1 20 43 CC(C)N1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217970734 CE For-Sale Unstable CACNA1G 22 40 CC(C)N1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217970734 CE For-Sale Unstable AKR1C3 33 43 O=C(CSc1ccccc1)NCCCc1ccc(F)cc1 ZINC000217970752 DH In-Stock Unstable CCR3 19 43 O=C(CSc1ccccc1)NCCCc1ccc(F)cc1 ZINC000217970752 DH In-Stock Unstable CRTM 43 47 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)Nc1cccc(OC)c1 ZINC000217970769 GG For-Sale Unstable CCR3 22 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)Nc1cccc(OC)c1 ZINC000217970769 GG For-Sale Unstable TAAR1 31 44 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)Nc1cccc(OC)c1 ZINC000217970769 GG For-Sale Unstable LIMK2 23 42 Cc1c(OCC(=O)N2CCCC[C@H]2c2cccnc2)ccc2c3c(c(=O)oc12)CCC3 ZINC000217970770 HI In-Stock Unstable COLA 132 43 Cc1c(OCC(=O)N2CCCC[C@H]2c2cccnc2)ccc2c3c(c(=O)oc12)CCC3 ZINC000217970770 HI In-Stock Unstable CPT1A 124 43 COc1ccc(CCNC(=O)N/C=C/c2cccc(F)c2)cc1OC ZINC000217970801 EG For-Sale Unstable MTNR1A 24 41 COc1ccc(CCNC(=O)N/C=C/c2cccc(F)c2)cc1OC ZINC000217970801 EG For-Sale Unstable MTNR1B 26 44 COc1ccc(CCNC(=O)N/C=C/c2cccc(F)c2)cc1OC ZINC000217970801 EG For-Sale Unstable ACKR3 50 42 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)Nc1cccc(OC)c1 ZINC000217970836 GG For-Sale Unstable CCR3 22 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)Nc1cccc(OC)c1 ZINC000217970836 GG For-Sale Unstable TAAR1 31 44 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)Nc1cccc(OC)c1 ZINC000217970836 GG For-Sale Unstable LIMK2 23 42 COc1ccccc1CCCNC(=O)CSc1ccccc1 ZINC000217970851 DH In-Stock Unstable DRD2 22 42 COc1ccccc1CCCNC(=O)CSc1ccccc1 ZINC000217970851 DH In-Stock Unstable MTNR1A 62 40 COc1ccccc1CCCNC(=O)CSc1ccccc1 ZINC000217970851 DH In-Stock Unstable MTNR1B 54 44 COc1ccccc1CCCNC(=O)CSc1ccccc1 ZINC000217970851 DH In-Stock Unstable MBTPS1 40 31 COc1ccccc1CCCNC(=O)CSc1ccccc1 ZINC000217970851 DH In-Stock Unstable FAS 72 44 Cn1cc(/C=C\C(=O)CCl)c2ccccc21 ZINC000217970871 BF For-Sale Unstable PRKCG 45 37 Cn1cc(S(=O)(=O)N2CCCN(S(=O)(=O)c3ccc(F)c(Cl)c3)CC2)cn1 ZINC000217970921 ID In-Stock Unstable PKM 54 45 Cn1cc(S(=O)(=O)N2CCCN(S(=O)(=O)c3ccc(F)c(Cl)c3)CC2)cn1 ZINC000217970921 ID In-Stock Unstable GCK 57 39 CN(CCOc1cccc(/C=C\C(=O)O)c1)CC(F)(F)F ZINC000217970928 DF For-Sale Unstable FDPS 20 40 COc1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217970971 DH In-Stock Unstable SCNN1A 46 41 COc1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217970971 DH In-Stock Unstable BMP1 32 43 COc1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217970971 DH In-Stock Unstable NQO2 25 40 COc1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217970971 DH In-Stock Unstable SIGMAR1 18 47 COc1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217970971 DH In-Stock Unstable MMP13 26 40 COc1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217970971 DH In-Stock Unstable LTB4R 24 45 COc1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217970971 DH In-Stock Unstable SCN2A 23 48 COc1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217970971 DH In-Stock Unstable MTNR1A 112 49 COc1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217970971 DH In-Stock Unstable MTNR1B 102 49 COc1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217970971 DH In-Stock Unstable MMP2 19 42 COc1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217970971 DH In-Stock Unstable MMP3 34 42 COc1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217970971 DH In-Stock Unstable MMP8 15 40 COc1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217970971 DH In-Stock Unstable MMP9 28 40 COc1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217970971 DH In-Stock Unstable CA9 18 44 COc1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217970971 DH In-Stock Unstable MMP1 30 40 COc1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217970971 DH In-Stock Unstable AMP1_PLAFQ 23 40 COc1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217970971 DH In-Stock Unstable CRTM 47 44 COc1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217970971 DH In-Stock Unstable FAS 79 44 CN(CCOc1ccc(/C=C\C(=O)O)cc1)CC(F)(F)F ZINC000217971011 DF On-Demand Unstable FDPS 24 41 CCCCOCCCNC(=O)N/C=C/c1cccc(F)c1 ZINC000217971017 CG For-Sale Unstable ACAT 0 40 CC(=O)c1cccc(S(=O)(=O)N2CCCN(S(=O)(=O)c3cnn(C)c3)CC2)c1 ZINC000217971031 IC In-Stock Unstable PKM 41 41 CC(=O)c1cccc(S(=O)(=O)N2CCCN(S(=O)(=O)c3cnn(C)c3)CC2)c1 ZINC000217971031 IC In-Stock Unstable AKR1C3 69 43 CC(=O)c1cccc(S(=O)(=O)N2CCCN(S(=O)(=O)c3cnn(C)c3)CC2)c1 ZINC000217971031 IC In-Stock Unstable AKR1C1 21 40 O=C(N[C@@H]1CCC[C@@H]1CO)c1c[nH]c2ccccc12 ZINC000217971035 CE For-Sale Unstable GABRA1 15 46 O=C(N[C@@H]1CCC[C@@H]1CO)c1c[nH]c2ccccc12 ZINC000217971035 CE For-Sale Unstable SSTR3 29 52 COc1ccc(OC[C@@H](C)NC(=O)CSc2ccccc2)cc1 ZINC000217971091 EG In-Stock Unstable SDH1 0 44 COc1ccc(OC[C@@H](C)NC(=O)CSc2ccccc2)cc1 ZINC000217971091 EG In-Stock Unstable CYP2D6 0 40 COc1ccc(OC[C@@H](C)NC(=O)CSc2ccccc2)cc1 ZINC000217971091 EG In-Stock Unstable FAS 73 44 COc1ccc(OC[C@@H](C)NC(=O)CSc2ccccc2)cc1 ZINC000217971091 EG In-Stock Unstable GPR88 0 45 O=C(/C=C\c1c[nH]c2ccc(Br)cc12)CCl ZINC000217971115 CH For-Sale Unstable GUSB 0 40 O=C(/C=C\c1c[nH]c2ccc(Br)cc12)CCl ZINC000217971115 CH For-Sale Unstable TDO2 0 41 O=C(N[C@H]1CCC[C@@H]1CO)c1c[nH]c2ccccc12 ZINC000217971121 CE For-Sale Unstable GABRA1 15 46 O=C(N[C@H]1CCC[C@@H]1CO)c1c[nH]c2ccccc12 ZINC000217971121 CE For-Sale Unstable SSTR3 29 52 COc1ccc(/C=C\C(=O)O)cc1CN1CC[C@@H](C)C1 ZINC000217971123 CF For-Sale Unstable RORC 42 35 O=C(N/C=C/c1cccc(F)c1)NCc1cccnc1 ZINC000217971139 CF For-Sale Unstable PTAFR 17 41 O=C(N/C=C/c1cccc(F)c1)NCc1cccnc1 ZINC000217971139 CF For-Sale Unstable SCD 15 40 O=C(N/C=C/c1cccc(F)c1)NCc1cccnc1 ZINC000217971139 CF For-Sale Unstable NAMPT 73 45 COc1ccc(OC[C@H](C)NC(=O)CSc2ccccc2)cc1 ZINC000217971160 EG In-Stock Unstable SDH1 0 44 COc1ccc(OC[C@H](C)NC(=O)CSc2ccccc2)cc1 ZINC000217971160 EG In-Stock Unstable CYP2D6 0 40 COc1ccc(OC[C@H](C)NC(=O)CSc2ccccc2)cc1 ZINC000217971160 EG In-Stock Unstable FAS 73 44 COc1ccc(OC[C@H](C)NC(=O)CSc2ccccc2)cc1 ZINC000217971160 EG In-Stock Unstable GPR88 0 45 O=C1c2ccccc2N2C(=O)c3ccccc3[C@@H]2N1CCCO ZINC000217971162 DE In-Stock Unstable TOP1 0 43 O=C(N[C@@H]1CCC[C@H]1CO)c1c[nH]c2ccccc12 ZINC000217971206 CE For-Sale Unstable GABRA1 15 46 O=C(N[C@@H]1CCC[C@H]1CO)c1c[nH]c2ccccc12 ZINC000217971206 CE For-Sale Unstable SSTR3 29 52 COc1ccc(/C=C\C(=O)O)cc1CN1CC[C@H](C)C1 ZINC000217971208 CF For-Sale Unstable RORC 42 35 O=C1c2ccccc2N2C(=O)c3ccccc3[C@H]2N1CCCO ZINC000217971244 DE In-Stock Unstable TOP1 0 43 Cn1cc(S(=O)(=O)N2CCCN(S(=O)(=O)c3c(F)cccc3F)CC2)cn1 ZINC000217971255 HC In-Stock Unstable PKM 56 59 O=C(CSc1ccccc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217971269 EJ In-Stock Unstable PAGA 0 40 O=C(CSc1ccccc1)Nc1ccccc1C(=O)c1ccccc1 ZINC000217971269 EJ In-Stock Unstable FAS 83 68 O=C(N[C@H]1CCC[C@H]1CO)c1c[nH]c2ccccc12 ZINC000217971292 CE For-Sale Unstable GABRA1 15 46 O=C(N[C@H]1CCC[C@H]1CO)c1c[nH]c2ccccc12 ZINC000217971292 CE For-Sale Unstable SSTR3 29 52 COc1ccc(CN2CC[C@@H](C)C2)cc1/C=C\C(=O)O ZINC000217971321 CF For-Sale Unstable DRD4 34 40 COc1ccc(CN2CC[C@@H](C)C2)cc1/C=C\C(=O)O ZINC000217971321 CF For-Sale Unstable DRD3 0 40 COc1ccc(CN2CC[C@@H](C)C2)cc1/C=C\C(=O)O ZINC000217971321 CF For-Sale Unstable PTGER2 23 40 COc1ccc(CN2CC[C@@H](C)C2)cc1/C=C\C(=O)O ZINC000217971321 CF For-Sale Unstable PTGER4 0 40 COc1ccc(CN2CC[C@@H](C)C2)cc1/C=C\C(=O)O ZINC000217971321 CF For-Sale Unstable SSTR5 47 36 COc1ccc(CN2CC[C@@H](C)C2)cc1/C=C\C(=O)O ZINC000217971321 CF For-Sale Unstable CCR1 0 41 COc1ccc(CN2CC[C@@H](C)C2)cc1/C=C\C(=O)O ZINC000217971321 CF For-Sale Unstable MCHR1 18 42 O=C(N/C=C/c1cccc(F)c1)N1CCC(Cc2ccccc2)CC1 ZINC000217971365 EI For-Sale Unstable GRIN2B 83 47 O=C(N/C=C/c1cccc(F)c1)N1CCC(Cc2ccccc2)CC1 ZINC000217971365 EI For-Sale Unstable SIGMAR1 28 43 O=C(N/C=C/c1cccc(F)c1)N1CCC(Cc2ccccc2)CC1 ZINC000217971365 EI For-Sale Unstable CCR3 98 42 CC(C)Oc1cccc(CCCNC(=O)CSc2ccccc2)c1 ZINC000217971387 EI In-Stock Unstable FDFT1 23 51 CC(C)Oc1cccc(CCCNC(=O)CSc2ccccc2)c1 ZINC000217971387 EI In-Stock Unstable MTNR1A 46 43 CC(C)Oc1cccc(CCCNC(=O)CSc2ccccc2)c1 ZINC000217971387 EI In-Stock Unstable MTNR1B 23 44 CC(C)Oc1cccc(CCCNC(=O)CSc2ccccc2)c1 ZINC000217971387 EI In-Stock Unstable AMP1_PLAFQ 42 46 CC(C)Oc1cccc(CCCNC(=O)CSc2ccccc2)c1 ZINC000217971387 EI In-Stock Unstable CRTM 80 51 CC(C)Oc1cccc(CCCNC(=O)CSc2ccccc2)c1 ZINC000217971387 EI In-Stock Unstable CRTH2 0 44 CC(C)Oc1cccc(CCCNC(=O)CSc2ccccc2)c1 ZINC000217971387 EI In-Stock Unstable PDS 55 41 CC(C)Oc1cccc(CCCNC(=O)CSc2ccccc2)c1 ZINC000217971387 EI In-Stock Unstable FAS 46 39 COc1ccc(CN2CC[C@H](C)C2)cc1/C=C\C(=O)O ZINC000217971402 CF For-Sale Unstable DRD4 34 40 COc1ccc(CN2CC[C@H](C)C2)cc1/C=C\C(=O)O ZINC000217971402 CF For-Sale Unstable DRD3 19 40 COc1ccc(CN2CC[C@H](C)C2)cc1/C=C\C(=O)O ZINC000217971402 CF For-Sale Unstable PTGER2 23 40 COc1ccc(CN2CC[C@H](C)C2)cc1/C=C\C(=O)O ZINC000217971402 CF For-Sale Unstable PTGER4 15 40 COc1ccc(CN2CC[C@H](C)C2)cc1/C=C\C(=O)O ZINC000217971402 CF For-Sale Unstable SSTR5 47 36 COc1ccc(CN2CC[C@H](C)C2)cc1/C=C\C(=O)O ZINC000217971402 CF For-Sale Unstable CCR1 20 41 COc1ccc(CN2CC[C@H](C)C2)cc1/C=C\C(=O)O ZINC000217971402 CF For-Sale Unstable MCHR1 21 42 NC(=O)Cc1c(Cl)cncc1Cl ZINC000217971447 BD For-Sale Unstable PDE4D 16 48 CN1CCC(N(C)C(=O)N/C=C/c2cccc(F)c2)CC1 ZINC000217971469 CF For-Sale Unstable NPY2R 0 42 CC(C)Oc1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217971492 EI In-Stock Unstable AMP1_PLAFQ 24 41 CC(C)Oc1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217971492 EI In-Stock Unstable CRTM 45 42 CC(C)Oc1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217971492 EI In-Stock Unstable FAS 43 39 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)NCCc3ccncc3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217971539 KG In-Stock Unstable TUBA1A 18 66 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)NCCc3ccncc3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217971539 KG In-Stock Unstable TPPP 0 63 COc1cc(F)c(/C=C\C(=O)CCl)cc1OC ZINC000217971549 CF For-Sale Unstable NFE2L2 0 47 COc1cc(F)c(/C=C\C(=O)CCl)cc1OC ZINC000217971549 CF For-Sale Unstable CYSP_PLAFA 49 35 COc1ccc(CCNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217971564 DG For-Sale Unstable MTNR1A 108 43 COc1ccc(CCNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217971564 DG For-Sale Unstable MTNR1B 88 43 COC(=O)c1ccc(S(=O)(=O)N2CCCN(S(=O)(=O)c3cnn(C)c3)CC2)cc1 ZINC000217971592 IC In-Stock Unstable PKM 23 43 COC(=O)c1ccc(S(=O)(=O)N2CCCN(S(=O)(=O)c3cnn(C)c3)CC2)cc1 ZINC000217971592 IC In-Stock Unstable TGM2 61 35 COC(=O)c1ccc(S(=O)(=O)N2CCCN(S(=O)(=O)c3cnn(C)c3)CC2)cc1 ZINC000217971592 IC In-Stock Unstable F13A1 62 38 CC1(C)C[C@@H](NC(=O)CSc2ccccc2)c2ccccc2O1 ZINC000217971600 EI In-Stock Unstable FAS 57 40 CC1(C)C[C@H](NC(=O)CSc2ccccc2)c2ccccc2O1 ZINC000217971682 EI In-Stock Unstable FAS 57 40 CCc1ncnc(NCc2ccc(S(C)(=O)=O)cc2)c1F ZINC000217971704 DE On-Demand Unstable PTGS2 24 46 CCCN1CCC[C@H]([C@@H](C)N[C@H](c2cccs2)C(C)C)C1 ZINC000217971738 DJ For-Sale Unstable BIRC2 40 33 C[C@@H]1CCC[C@H](N(C)Cc2ccccc2/C=C\C(=O)O)C1 ZINC000217971756 CH For-Sale Unstable PTGER2 39 46 C[C@@H]1CCC[C@H](N(C)Cc2ccccc2/C=C\C(=O)O)C1 ZINC000217971756 CH For-Sale Unstable PTGER4 0 46 C[C@@H]1CCC[C@H](N(C)Cc2ccccc2/C=C\C(=O)O)C1 ZINC000217971756 CH For-Sale Unstable PTGER3 15 46 C[C@@H]1CCC[C@H](N(C)Cc2ccccc2/C=C\C(=O)O)C1 ZINC000217971756 CH For-Sale Unstable PTGDR 0 44 COc1cccc2c(O)c(C(=O)NCCCc3nc4ccccc4n3C)cnc12 ZINC000217971769 GG In-Stock Unstable DRD2 16 41 COc1cccc2c(O)c(C(=O)NCCCc3nc4ccccc4n3C)cnc12 ZINC000217971769 GG In-Stock Unstable DRD3 26 41 CCOc1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217971794 EH In-Stock Unstable SCN2A 27 50 CCOc1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217971794 EH In-Stock Unstable PLA2G4A 28 40 CCOc1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217971794 EH In-Stock Unstable PLA2G2A 0 41 CCOc1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217971794 EH In-Stock Unstable MTNR1A 52 39 CCOc1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217971794 EH In-Stock Unstable MTNR1B 42 40 CCOc1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217971794 EH In-Stock Unstable CRTM 46 43 CCOc1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217971794 EH In-Stock Unstable PDS 47 40 CCOc1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217971794 EH In-Stock Unstable FAS 56 40 CCCN1CCC[C@@H]([C@@H](C)N[C@H](c2cccs2)C(C)C)C1 ZINC000217971816 DJ For-Sale Unstable BIRC2 40 33 CC[C@H](C(N)=S)N1C[C@@H](C)Cc2ccccc21 ZINC000217971830 BF For-Sale Unstable TPP2 54 34 Cn1cc(S(=O)(=O)N2CCCN(S(=O)(=O)Cc3cc(F)ccc3F)CC2)cn1 ZINC000217971841 IC In-Stock Unstable PKM 36 40 O=C(COC[C@@H]1CCCCO1)N1CCN(c2nc3ccccc3o2)CC1 ZINC000217971861 FE In-Stock Unstable COLA 53 35 C[C@H]1CCC[C@H](N(C)Cc2ccccc2/C=C\C(=O)O)C1 ZINC000217971863 CH For-Sale Unstable PTGER2 39 46 C[C@H]1CCC[C@H](N(C)Cc2ccccc2/C=C\C(=O)O)C1 ZINC000217971863 CH For-Sale Unstable PTGER4 0 46 C[C@H]1CCC[C@H](N(C)Cc2ccccc2/C=C\C(=O)O)C1 ZINC000217971863 CH For-Sale Unstable PTGER3 15 46 C[C@H]1CCC[C@H](N(C)Cc2ccccc2/C=C\C(=O)O)C1 ZINC000217971863 CH For-Sale Unstable PTGDR 0 44 Clc1cc(CBr)ccc1-n1ccnc1 ZINC000217971870 CG For-Sale Unstable CYP17A1 0 46 CCCOc1ccccc1CCCNC(=O)CSc1ccccc1 ZINC000217971914 EI In-Stock Unstable MTNR1A 44 41 CCCOc1ccccc1CCCNC(=O)CSc1ccccc1 ZINC000217971914 EI In-Stock Unstable MTNR1B 54 42 CCCOc1ccccc1CCCNC(=O)CSc1ccccc1 ZINC000217971914 EI In-Stock Unstable FAS 42 39 CC[C@@H](C(N)=S)N1C[C@@H](C)Cc2ccccc21 ZINC000217971923 BF For-Sale Unstable TPP2 54 34 O=C(COC[C@H]1CCCCO1)N1CCN(c2nc3ccccc3o2)CC1 ZINC000217971945 FE In-Stock Unstable COLA 53 35 Clc1ccc(CBr)c(-n2ccnc2)c1 ZINC000217971969 CG For-Sale Unstable TBXAS1 0 44 CCOc1ccc(S(=O)(=O)N2CCCN(S(=O)(=O)c3cnn(C)c3)CC2)cc1F ZINC000217971971 ID In-Stock Unstable PDE5A 38 42 CCOc1ccc(S(=O)(=O)N2CCCN(S(=O)(=O)c3cnn(C)c3)CC2)cc1F ZINC000217971971 ID In-Stock Unstable PKM 45 40 CCOc1ccc(S(=O)(=O)N2CCCN(S(=O)(=O)c3cnn(C)c3)CC2)cc1F ZINC000217971971 ID In-Stock Unstable GCK 56 38 CCOc1ccc(S(=O)(=O)N2CCCN(S(=O)(=O)c3cnn(C)c3)CC2)cc1F ZINC000217971971 ID In-Stock Unstable GCKR 42 29 CCN(CC(=O)N(C)C)Cc1ccccc1/C=C\C(=O)O ZINC000217971974 CD For-Sale Unstable PTGER2 43 47 CCN(CC(=O)N(C)C)Cc1ccccc1/C=C\C(=O)O ZINC000217971974 CD For-Sale Unstable PTGER4 0 47 CCN(CC(=O)N(C)C)Cc1ccccc1/C=C\C(=O)O ZINC000217971974 CD For-Sale Unstable PTGER3 16 47 Cc1ccccc1OC[C@H](C)NC(=O)CSc1ccccc1 ZINC000217971991 DH In-Stock Unstable FAS 49 42 Cc1noc2nc(C(C)C)cc(C(=O)Nc3cc(C(F)(F)F)ccc3N3CCCC3)c12 ZINC000217971995 IK On-Demand Unstable TEK 23 45 C[C@@H](NC(=O)N/C=C/c1cccc(F)c1)c1ccccc1 ZINC000217971999 CH For-Sale Unstable KCNQ2 50 38 C[C@@H](NC(=O)N/C=C/c1cccc(F)c1)c1ccccc1 ZINC000217971999 CH For-Sale Unstable ACACA 0 40 COc1cc(OC)nc(-n2c(C)ccc2C)n1 ZINC000217972038 BD For-Sale Unstable ALS 76 37 C[C@H](NC(=O)N/C=C/c1cccc(F)c1)c1ccccc1 ZINC000217972074 CH For-Sale Unstable KCNQ2 50 38 C[C@H](NC(=O)N/C=C/c1cccc(F)c1)c1ccccc1 ZINC000217972074 CH For-Sale Unstable ACACA 0 40 Cc1cc(-n2ccnc2)ccc1CBr ZINC000217972077 CG For-Sale Unstable CYP2C19 17 43 Cn1cc(S(=O)(=O)N2CCCN(S(=O)(=O)c3ccc4c(c3)CCO4)CC2)cn1 ZINC000217972078 IC In-Stock Unstable PKM 53 52 C[C@H]1Cc2ccccc2N(C[C@H](C)C(N)=S)C1 ZINC000217972087 BF For-Sale Unstable ACE 15 40 C[C@H]1Cc2ccccc2N(C[C@H](C)C(N)=S)C1 ZINC000217972087 BF For-Sale Unstable TPP2 52 32 Cc1ccc(OC[C@@H](C)NC(=O)CSc2ccccc2)cc1 ZINC000217972104 DH In-Stock Unstable SDH1 0 44 Cc1ccc(OC[C@@H](C)NC(=O)CSc2ccccc2)cc1 ZINC000217972104 DH In-Stock Unstable ACACA 42 35 Cc1ccc(OC[C@@H](C)NC(=O)CSc2ccccc2)cc1 ZINC000217972104 DH In-Stock Unstable PDS 45 36 Cc1ccc(OC[C@@H](C)NC(=O)CSc2ccccc2)cc1 ZINC000217972104 DH In-Stock Unstable FAS 50 42 Cc1ccc(OC[C@@H](C)NC(=O)CSc2ccccc2)cc1 ZINC000217972104 DH In-Stock Unstable GPR88 0 43 COc1ccc(C(=O)N[C@@H]2CCC[C@@H]2CO)cc1F ZINC000217972139 CD On-Demand Unstable SSTR3 26 43 COc1ccc(C(=O)N[C@@H]2CCC[C@@H]2CO)cc1F ZINC000217972139 CD On-Demand Unstable ACKR3 41 34 CC[C@@H](CC(N)=S)N1C[C@@H](C)Cc2ccccc21 ZINC000217972177 CG For-Sale Unstable TPP2 53 33 Cc1ccc(OC[C@H](C)NC(=O)CSc2ccccc2)cc1 ZINC000217972184 DH In-Stock Unstable SDH1 0 44 Cc1ccc(OC[C@H](C)NC(=O)CSc2ccccc2)cc1 ZINC000217972184 DH In-Stock Unstable ACACA 42 35 Cc1ccc(OC[C@H](C)NC(=O)CSc2ccccc2)cc1 ZINC000217972184 DH In-Stock Unstable PDS 41 34 Cc1ccc(OC[C@H](C)NC(=O)CSc2ccccc2)cc1 ZINC000217972184 DH In-Stock Unstable FAS 50 42 Cc1ccc(OC[C@H](C)NC(=O)CSc2ccccc2)cc1 ZINC000217972184 DH In-Stock Unstable GPR88 0 43 Cc1nc2ccccc2n1CCC(=O)NCCc1noc(C2CCC2)n1 ZINC000217972196 FF In-Stock Unstable SMO 57 45 Cc1nc2ccccc2n1CCC(=O)NCCc1noc(C2CCC2)n1 ZINC000217972196 FF In-Stock Unstable ETHR 42 34 CCN(CC(=O)N(C)C)Cc1cccc(/C=C\C(=O)O)c1 ZINC000217972215 CD For-Sale Unstable AKR1C3 30 42 CC[C@H](CC(N)=S)N1C[C@@H](C)Cc2ccccc21 ZINC000217972244 CG For-Sale Unstable TPP2 53 33 COc1ccc(CNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217972269 DG For-Sale Unstable MTNR1A 52 45 COc1ccc(CNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217972269 DG For-Sale Unstable MTNR1B 47 45 COc1ccc(CNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217972269 DG For-Sale Unstable NR1H4 25 40 CC1CCN(c2ccc([C@@H](C)NC(=O)CSc3ccccc3)cc2)CC1 ZINC000217972289 FJ In-Stock Unstable PRCP 15 43 Clc1ccc(-n2ccnc2)c(CBr)c1 ZINC000217972305 CG For-Sale Unstable TBXAS1 0 44 CN(Cc1cnn(C)c1)Cc1ccccc1/C=C\C(=O)O ZINC000217972344 CE For-Sale Unstable PTGER2 36 42 CN(Cc1cnn(C)c1)Cc1ccccc1/C=C\C(=O)O ZINC000217972344 CE For-Sale Unstable PTGER4 16 43 CN(Cc1cnn(C)c1)Cc1ccccc1/C=C\C(=O)O ZINC000217972344 CE For-Sale Unstable PTGER3 19 43 CN(Cc1cnn(C)c1)Cc1ccccc1/C=C\C(=O)O ZINC000217972344 CE For-Sale Unstable PTGDR 16 43 C[C@H]1Cc2ccccc2N([C@H](C)CC(N)=S)C1 ZINC000217972368 BF For-Sale Unstable TPP2 43 30 CCCCOc1ccc(NC(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217972373 II For-Sale Unstable TSHR 48 35 CCCCOc1ccc(NC(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217972373 II For-Sale Unstable PLA2G4B 42 31 CCCCOc1ccc(NC(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217972373 II For-Sale Unstable FAAH 23 53 CCCCOc1ccc(NC(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217972373 II For-Sale Unstable CFTR 42 32 CC1CCN(c2ccc([C@H](C)NC(=O)CSc3ccccc3)cc2)CC1 ZINC000217972374 FJ In-Stock Unstable PRCP 15 43 O=C(COc1ccc(Cl)c(Cl)c1)N[C@@H]1C[C@@H]2OCC[C@@H]21 ZINC000217972444 DF In-Stock Unstable TRAR 32 42 CCCCOc1ccc(NC(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217972449 II For-Sale Unstable TSHR 48 35 CCCCOc1ccc(NC(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217972449 II For-Sale Unstable PLA2G4B 42 31 CCCCOc1ccc(NC(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217972449 II For-Sale Unstable FAAH 23 53 CCCCOc1ccc(NC(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217972449 II For-Sale Unstable CFTR 42 32 CN(Cc1ccc(/C=C\C(=O)O)cc1)Cc1cnn(C)c1 ZINC000217972466 CE For-Sale Unstable PLA2G7 44 38 O=C(N/C=C/c1cccc(F)c1)NCc1ccc2c(c1)OCO2 ZINC000217972490 DG For-Sale Unstable NOS2 79 34 O=C(N/C=C/c1cccc(F)c1)NCc1ccc2c(c1)OCO2 ZINC000217972490 DG For-Sale Unstable MCHR1 15 44 CCCCOc1ccc(NC(=O)N2C[C@H](Oc3ccccc3F)C[C@H]2C(=O)OC)cc1 ZINC000217972528 II For-Sale Unstable TSHR 48 35 CCCCOc1ccc(NC(=O)N2C[C@H](Oc3ccccc3F)C[C@H]2C(=O)OC)cc1 ZINC000217972528 II For-Sale Unstable PLA2G4B 42 31 CCCCOc1ccc(NC(=O)N2C[C@H](Oc3ccccc3F)C[C@H]2C(=O)OC)cc1 ZINC000217972528 II For-Sale Unstable FAAH 23 53 CCCCOc1ccc(NC(=O)N2C[C@H](Oc3ccccc3F)C[C@H]2C(=O)OC)cc1 ZINC000217972528 II For-Sale Unstable CFTR 42 32 CN(Cc1cccc(/C=C\C(=O)O)c1)Cc1cnn(C)c1 ZINC000217972576 CE For-Sale Unstable HDAC8 53 42 CN(Cc1cccc(/C=C\C(=O)O)c1)Cc1cnn(C)c1 ZINC000217972576 CE For-Sale Unstable HDAC1 31 42 CN(Cc1cccc(/C=C\C(=O)O)c1)Cc1cnn(C)c1 ZINC000217972576 CE For-Sale Unstable HDAC6 42 42 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217972602 EE For-Sale Unstable CA2 91 56 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217972602 EE For-Sale Unstable CA1 85 50 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217972602 EE For-Sale Unstable CA7 43 40 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217972602 EE For-Sale Unstable CA5B 45 40 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217972602 EE For-Sale Unstable CA4 76 50 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217972602 EE For-Sale Unstable CA5A 52 40 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217972602 EE For-Sale Unstable CA14 34 40 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217972602 EE For-Sale Unstable CA12 71 56 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217972602 EE For-Sale Unstable CA9 75 49 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217972602 EE For-Sale Unstable IDO1 28 46 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217972602 EE For-Sale Unstable NCE103 39 42 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217972602 EE For-Sale Unstable MTCA1 60 56 NS(=O)(=O)c1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217972602 EE For-Sale Unstable P96878_MYCTU 72 56 CCCCOc1ccc(NC(=O)N2C[C@@H](Oc3ccccc3F)C[C@H]2C(=O)OC)cc1 ZINC000217972607 II For-Sale Unstable TSHR 48 35 CCCCOc1ccc(NC(=O)N2C[C@@H](Oc3ccccc3F)C[C@H]2C(=O)OC)cc1 ZINC000217972607 II For-Sale Unstable PLA2G4B 42 31 CCCCOc1ccc(NC(=O)N2C[C@@H](Oc3ccccc3F)C[C@H]2C(=O)OC)cc1 ZINC000217972607 II For-Sale Unstable FAAH 23 53 CCCCOc1ccc(NC(=O)N2C[C@@H](Oc3ccccc3F)C[C@H]2C(=O)OC)cc1 ZINC000217972607 II For-Sale Unstable CFTR 42 32 O=C1C/C(=C/c2ccc(-c3ccc(Cl)cc3)s2)C(=O)N1 ZINC000217972616 DG For-Sale Unstable PRF1 45 38 BrCc1ccc(-n2ccnc2)nc1 ZINC000217972619 BE For-Sale Unstable CYP11B1 33 43 Cc1ccc2c(c1)[C@@H](NC(=O)CSc1ccccc1)CC(C)(C)O2 ZINC000217972670 EJ In-Stock Unstable FAS 41 36 CCC1CCN(Cc2ccc(/C=C\C(=O)O)cc2F)CC1 ZINC000217972683 CH For-Sale Unstable CCR2 53 45 O=C(N/C=C/c1cccc(F)c1)NCc1ccccc1 ZINC000217972722 CG For-Sale Unstable AMP1_PLAFQ 31 42 O=C(N/C=C/c1cccc(F)c1)NCc1ccccc1 ZINC000217972722 CG For-Sale Unstable PDS 54 42 CN(C)CCOc1ccc(/C=C2/CC(=O)NC2=O)cc1 ZINC000217972727 CD For-Sale Unstable ESRRG 45 33 CN(C)CCOc1ccc(/C=C2/CC(=O)NC2=O)cc1 ZINC000217972727 CD For-Sale Unstable HPGD 71 42 BrCc1cnc(-n2ccnc2)nc1 ZINC000217972749 BD For-Sale Unstable CYP11B1 26 40 BrCc1cnc(-n2ccnc2)nc1 ZINC000217972749 BD For-Sale Unstable CYP11B2 21 40 Cc1ccc2c(c1)[C@H](NC(=O)CSc1ccccc1)CC(C)(C)O2 ZINC000217972751 EJ In-Stock Unstable FAS 41 36 CC(C)Oc1cccc(/C=C2/CC(=O)NC2=O)c1 ZINC000217972805 BD For-Sale Unstable AKR1B1 21 42 CCC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217972806 CG For-Sale Unstable CHRM2 15 42 CCC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217972806 CG For-Sale Unstable DRD2 26 47 CCC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217972806 CG For-Sale Unstable DRD4 56 47 CCC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217972806 CG For-Sale Unstable ACHE 55 49 CCC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217972806 CG For-Sale Unstable HRH1 23 40 CCC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217972806 CG For-Sale Unstable DRD3 23 42 CCC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217972806 CG For-Sale Unstable CHRM3 22 42 CCC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217972806 CG For-Sale Unstable GRIN2B 27 40 CCC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217972806 CG For-Sale Unstable VACHT_TETCF 0 41 CCC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217972806 CG For-Sale Unstable SIGMAR1 63 53 CCC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217972806 CG For-Sale Unstable CCR3 48 42 CCC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217972806 CG For-Sale Unstable HDAC1 17 42 CCC1CCN(Cc2cccc(/C=C\C(=O)O)c2)CC1 ZINC000217972806 CG For-Sale Unstable AKR1C3 29 42 Cc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)CSc1ccccc1 ZINC000217972843 EJ In-Stock Unstable FAS 45 37 COc1ccc(C(=O)NCC2(C)COC2)c(F)c1F ZINC000217972867 CD In-Stock Unstable KCNA3 37 40 COc1ccc(C(=O)NCC2(C)COC2)c(F)c1F ZINC000217972867 CD In-Stock Unstable HCN1 50 34 COc1ccc(C(=O)NCC2(C)COC2)c(F)c1F ZINC000217972867 CD In-Stock Unstable HCN4 48 34 CN(C)CCCNS(=O)(=O)c1ccc(N2CCC[C@@H]2c2ccccc2)c([N+](=O)[O-])c1 ZINC000217972904 IG On-Demand Unstable BDKRB1 33 43 CN(C)CCCNS(=O)(=O)c1ccc(N2CCC[C@@H]2c2ccccc2)c([N+](=O)[O-])c1 ZINC000217972904 IG On-Demand Unstable BCL2L1 69 34 CN(C)CCCNS(=O)(=O)c1ccc(N2CCC[C@@H]2c2ccccc2)c([N+](=O)[O-])c1 ZINC000217972904 IG On-Demand Unstable BCL2 52 32 Cc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)CSc1ccccc1 ZINC000217972924 EJ In-Stock Unstable FAS 45 37 O=C(O)/C=C\c1ccccc1CN1CCC(CO)CC1 ZINC000217972925 CD For-Sale Unstable ACHE 29 43 O=C(O)/C=C\c1ccccc1CN1CCC(CO)CC1 ZINC000217972925 CD For-Sale Unstable PTGER2 38 46 O=C(O)/C=C\c1ccccc1CN1CCC(CO)CC1 ZINC000217972925 CD For-Sale Unstable PTGER4 0 46 O=C(O)/C=C\c1ccccc1CN1CCC(CO)CC1 ZINC000217972925 CD For-Sale Unstable SIGMAR1 39 40 O=C(O)/C=C\c1ccccc1CN1CCC(CO)CC1 ZINC000217972925 CD For-Sale Unstable PTGER3 18 46 O=C(O)/C=C\c1ccccc1CN1CCC(CO)CC1 ZINC000217972925 CD For-Sale Unstable CCR3 31 43 CN(C)CCCNS(=O)(=O)c1ccc(N2CCC[C@H]2c2ccccc2)c([N+](=O)[O-])c1 ZINC000217972981 IG On-Demand Unstable BDKRB1 33 43 CN(C)CCCNS(=O)(=O)c1ccc(N2CCC[C@H]2c2ccccc2)c([N+](=O)[O-])c1 ZINC000217972981 IG On-Demand Unstable BCL2L1 69 34 CN(C)CCCNS(=O)(=O)c1ccc(N2CCC[C@H]2c2ccccc2)c([N+](=O)[O-])c1 ZINC000217972981 IG On-Demand Unstable BCL2 52 32 COc1ccc2c(c1)[C@@H](NC(=O)CSc1ccccc1)CC(C)(C)O2 ZINC000217973021 FI In-Stock Unstable FAS 62 41 O=C(O)/C=C\c1ccc(CN2CCC(CO)CC2)cc1 ZINC000217973024 CD For-Sale Unstable DRD2 0 51 O=C(O)/C=C\c1ccc(CN2CCC(CO)CC2)cc1 ZINC000217973024 CD For-Sale Unstable ACHE 42 44 O=C(O)/C=C\c1ccc(CN2CCC(CO)CC2)cc1 ZINC000217973024 CD For-Sale Unstable SIGMAR1 53 51 O=C(O)/C=C\c1ccc(CN2CCC(CO)CC2)cc1 ZINC000217973024 CD For-Sale Unstable CCR3 17 40 COc1ccc2c(c1)[C@H](NC(=O)CSc1ccccc1)CC(C)(C)O2 ZINC000217973108 FI In-Stock Unstable FAS 62 41 Cc1cc(O)ccc1NC(=O)N/C=C/c1cccc(F)c1 ZINC000217973125 CH For-Sale Unstable MMP1 0 44 O=C(O)/C=C\c1ccc(CN2CCC(CO)CC2)c(F)c1 ZINC000217973140 CE For-Sale Unstable SIGMAR1 18 40 O=C(O)/C=C\c1ccc(CN2CCC(CO)CC2)c(F)c1 ZINC000217973140 CE For-Sale Unstable CCR2 33 45 c1cnn(CCNCCCN2CCCCC2)c1 ZINC000217973153 BD For-Sale Unstable HNMT 70 40 COc1ccccc1CCN1Cc2ccccc2C1=N ZINC000217973215 CG For-Sale Unstable HTR1A 15 45 COc1ccccc1CCN1Cc2ccccc2C1=N ZINC000217973215 CG For-Sale Unstable HTR7 16 44 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)CSc1ccccc1 ZINC000217973225 FI In-Stock Unstable MTNR1A 41 35 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)CSc1ccccc1 ZINC000217973225 FI In-Stock Unstable FAS 66 42 C[C@@H]1CCCCN1CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217973264 CG For-Sale Unstable HRH3 60 41 C[C@@H]1CCCCN1CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217973264 CG For-Sale Unstable COLA 68 35 C[C@@H]1CCCCN1CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217973264 CG For-Sale Unstable CPT1A 65 35 C[C@@H]1CCCCN1CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217973264 CG For-Sale Unstable ACKR3 42 44 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)CSc1ccccc1 ZINC000217973305 FI In-Stock Unstable MTNR1A 41 35 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)CSc1ccccc1 ZINC000217973305 FI In-Stock Unstable FAS 66 42 C[C@H]1CCCCN1CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217973350 CG For-Sale Unstable HRH3 60 41 C[C@H]1CCCCN1CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217973350 CG For-Sale Unstable COLA 68 35 C[C@H]1CCCCN1CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217973350 CG For-Sale Unstable CPT1A 65 35 C[C@H]1CCCCN1CCOc1cccc(/C=C\C(=O)O)c1 ZINC000217973350 CG For-Sale Unstable ACKR3 42 44 CC[C@@H](NC(=O)CSc1ccccc1)c1ccc(C)c(C)c1 ZINC000217973434 DJ In-Stock Unstable TACR3 44 34 CC[C@@H](NC(=O)CSc1ccccc1)c1ccc(C)c(C)c1 ZINC000217973434 DJ In-Stock Unstable PDS 43 33 CC[C@@H](NC(=O)CSc1ccccc1)c1ccc(C)c(C)c1 ZINC000217973434 DJ In-Stock Unstable FAS 36 40 C[C@@H]1CCCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217973458 CG On-Demand Unstable ESR1 25 41 C[C@@H]1CCCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217973458 CG On-Demand Unstable HTR3A 16 43 C[C@@H]1CCCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217973458 CG On-Demand Unstable ESR2 18 41 C[C@@H]1CCCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217973458 CG On-Demand Unstable LTA4H 43 44 C[C@@H]1CCCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217973458 CG On-Demand Unstable HRH3 84 47 C[C@@H]1CCCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217973458 CG On-Demand Unstable PSMB2 48 37 C[C@@H]1CCCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217973458 CG On-Demand Unstable PSMB1 42 37 CCCn1cccc(C(N)=O)c1=O ZINC000217973486 AC For-Sale Unstable PARP1 24 40 CC[C@H](NC(=O)CSc1ccccc1)c1ccc(C)c(C)c1 ZINC000217973509 DJ In-Stock Unstable TACR3 44 34 CC[C@H](NC(=O)CSc1ccccc1)c1ccc(C)c(C)c1 ZINC000217973509 DJ In-Stock Unstable PDS 50 33 CC[C@H](NC(=O)CSc1ccccc1)c1ccc(C)c(C)c1 ZINC000217973509 DJ In-Stock Unstable FAS 36 40 C[C@H]1CCCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217973548 CG On-Demand Unstable ESR1 25 41 C[C@H]1CCCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217973548 CG On-Demand Unstable HTR3A 16 43 C[C@H]1CCCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217973548 CG On-Demand Unstable ESR2 18 41 C[C@H]1CCCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217973548 CG On-Demand Unstable LTA4H 43 44 C[C@H]1CCCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217973548 CG On-Demand Unstable HRH3 84 47 C[C@H]1CCCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217973548 CG On-Demand Unstable PSMB2 48 37 C[C@H]1CCCCN1CCOc1ccc(/C=C\C(=O)O)cc1 ZINC000217973548 CG On-Demand Unstable PSMB1 42 37 CCOC(=O)N1CCN(c2nc3ccccc3nc2NS(=O)(=O)c2cnn(C)c2)CC1 ZINC000217973557 ID In-Stock Unstable P2RY12 118 40 CC[C@@H](NC(=O)CSc1ccccc1)c1ccc(C)cc1C ZINC000217973628 DJ In-Stock Unstable CTSA 40 34 COc1ccc(CN2CCCCCC2)cc1/C=C\C(=O)O ZINC000217973640 CG For-Sale Unstable ACHE 25 56 COc1ccc(CN2CCCCCC2)cc1/C=C\C(=O)O ZINC000217973640 CG For-Sale Unstable HRH2 26 41 COc1ccc(CN2CCCCCC2)cc1/C=C\C(=O)O ZINC000217973640 CG For-Sale Unstable PTGER2 39 43 COc1ccc(CN2CCCCCC2)cc1/C=C\C(=O)O ZINC000217973640 CG For-Sale Unstable PTGER4 22 43 COc1ccc(CN2CCCCCC2)cc1/C=C\C(=O)O ZINC000217973640 CG For-Sale Unstable HRH3 21 41 COc1ccc(CN2CCCCCC2)cc1/C=C\C(=O)O ZINC000217973640 CG For-Sale Unstable SIGMAR1 17 40 COc1ccc(CN2CCCCCC2)cc1/C=C\C(=O)O ZINC000217973640 CG For-Sale Unstable PTGER3 18 43 COc1ccc(CN2CCCCCC2)cc1/C=C\C(=O)O ZINC000217973640 CG For-Sale Unstable SSTR5 40 35 COc1ccc(CN2CCCCCC2)cc1/C=C\C(=O)O ZINC000217973640 CG For-Sale Unstable MCHR1 17 40 COc1cc(OC)c([C@@H]2CC(=O)Oc3ccc4c(c32)OC2(CCCCC2)CC4=O)cc1OC ZINC000217973641 JJ In-Stock Unstable MT-ND4 51 32 O=C(NC[C@@H]1CC[C@@H](C(=O)Oc2ccc3c(=O)c(-c4ccc([N+](=O)[O-])cc4)coc3c2)CC1)OCc1ccccc1 ZINC000217973649 KK In-Stock Unstable ALDH2 101 40 Cc1n[nH]c(C)c1CCN(C)C(=O)COc1ccc(F)cc1F ZINC000217973655 DE In-Stock Unstable HAO2 45 38 COc1cc(Br)c(Br)c(Br)c1Oc1ccc(Br)cc1Br ZINC000217973686 KK For-Sale Unstable AKR1B1 0 45 COc1cc(Br)c(Br)c(Br)c1Oc1ccc(Br)cc1Br ZINC000217973686 KK For-Sale Unstable ALOX12 19 57 COc1cc(Br)c(Br)c(Br)c1Oc1ccc(Br)cc1Br ZINC000217973686 KK For-Sale Unstable ALOX15 0 64 O=C(O)/C=C\c1ccc(CN2CCCCCC2)c(F)c1 ZINC000217973726 CG For-Sale Unstable GPR183 0 42 COc1cc(OC)c([C@H]2CC(=O)Oc3ccc4c(c32)OC2(CCCCC2)CC4=O)cc1OC ZINC000217973727 JJ In-Stock Unstable MT-ND4 51 32 O=C(O)CCCCCNC(=O)N/C=C/c1cccc(F)c1 ZINC000217973735 CF For-Sale Unstable HDAC9 34 40 O=C(O)CCCCCNC(=O)N/C=C/c1cccc(F)c1 ZINC000217973735 CF For-Sale Unstable HDAC7 32 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)NC1CCCCC1 ZINC000217973780 FF For-Sale Unstable EPHX2 17 40 CC[C@@H](NC(=O)CSc1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217973826 EI In-Stock Unstable ENPP1 63 38 CC[C@@H](NC(=O)CSc1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217973826 EI In-Stock Unstable PDS 48 34 CC[C@@H](NC(=O)CSc1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217973826 EI In-Stock Unstable FAS 63 43 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)NC1CCCCC1 ZINC000217973846 FF For-Sale Unstable EPHX2 17 40 CCc1ncnc(NCCN2CCCCC2)c1F ZINC000217973902 CE On-Demand Unstable HNMT 49 38 CC[C@H](NC(=O)CSc1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217973909 EI In-Stock Unstable TACR3 41 37 CC[C@H](NC(=O)CSc1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217973909 EI In-Stock Unstable ENPP1 63 38 CC[C@H](NC(=O)CSc1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217973909 EI In-Stock Unstable PDS 48 34 CC[C@H](NC(=O)CSc1ccccc1)c1ccc(OC)c(OC)c1 ZINC000217973909 EI In-Stock Unstable FAS 63 43 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)NC1CCCCC1 ZINC000217973931 FF For-Sale Unstable EPHX2 17 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)NC1CCCCC1 ZINC000217974005 FF For-Sale Unstable EPHX2 17 40 CC[C@@H](NC(=O)CSc1ccccc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217974028 FG In-Stock Unstable PTGS2 26 40 CC[C@@H](NC(=O)CSc1ccccc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217974028 FG In-Stock Unstable CTSF 49 37 CC[C@@H](NC(=O)CSc1ccccc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217974028 FG In-Stock Unstable TACR3 47 38 C[C@H]1C[C@@H](C)CN(Cc2ccc(F)c(/C=C\C(=O)O)c2)C1 ZINC000217974048 CG For-Sale Unstable CCR1 25 40 CC[C@H](NC(=O)CSc1ccccc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217974101 FG In-Stock Unstable PTGS2 26 40 CC[C@H](NC(=O)CSc1ccccc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217974101 FG In-Stock Unstable CTSF 49 37 CC[C@H](NC(=O)CSc1ccccc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217974101 FG In-Stock Unstable TACR3 47 38 CCOc1ccc(NC(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217974105 HG For-Sale Unstable TSHR 49 36 CCCCc1ccc(/C=C\C(=O)CCl)cc1 ZINC000217974110 BH For-Sale Unstable S1PR2 43 38 CCCCc1ccc(/C=C\C(=O)CCl)cc1 ZINC000217974110 BH For-Sale Unstable TRPM2 0 47 CC(C)C[C@@H](NC(=O)N/C=C/c1cccc(F)c1)C(=O)O ZINC000217974152 CF For-Sale Unstable FOLH1 57 39 CC(C)C[C@@H](NC(=O)N/C=C/c1cccc(F)c1)C(=O)O ZINC000217974152 CF For-Sale Unstable MME 17 44 CC(C)C[C@@H](NC(=O)N/C=C/c1cccc(F)c1)C(=O)O ZINC000217974152 CF For-Sale Unstable ANPEP 32 48 CC(C)C[C@@H](NC(=O)N/C=C/c1cccc(F)c1)C(=O)O ZINC000217974152 CF For-Sale Unstable NAALAD2 28 40 CC(C)C[C@@H](NC(=O)N/C=C/c1cccc(F)c1)C(=O)O ZINC000217974152 CF For-Sale Unstable FPR1 69 40 CCOc1ccc(NC(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217974195 HG For-Sale Unstable TSHR 49 36 CCN(Cc1ccccc1/C=C\C(=O)O)c1ccccc1 ZINC000217974216 CH For-Sale Unstable PTGER2 47 50 CCN(Cc1ccccc1/C=C\C(=O)O)c1ccccc1 ZINC000217974216 CH For-Sale Unstable PTGER4 23 50 CCN(Cc1ccccc1/C=C\C(=O)O)c1ccccc1 ZINC000217974216 CH For-Sale Unstable PTGER3 18 50 CCN(Cc1ccccc1/C=C\C(=O)O)c1ccccc1 ZINC000217974216 CH For-Sale Unstable PTGDR 0 48 CC(C)C[C@H](NC(=O)N/C=C/c1cccc(F)c1)C(=O)O ZINC000217974221 CF For-Sale Unstable FOLH1 57 39 CC(C)C[C@H](NC(=O)N/C=C/c1cccc(F)c1)C(=O)O ZINC000217974221 CF For-Sale Unstable MME 17 44 CC(C)C[C@H](NC(=O)N/C=C/c1cccc(F)c1)C(=O)O ZINC000217974221 CF For-Sale Unstable ANPEP 32 48 CC(C)C[C@H](NC(=O)N/C=C/c1cccc(F)c1)C(=O)O ZINC000217974221 CF For-Sale Unstable NAALAD2 28 40 CC(C)C[C@H](NC(=O)N/C=C/c1cccc(F)c1)C(=O)O ZINC000217974221 CF For-Sale Unstable FPR1 69 40 COc1ccc(-c2noc(CNC(=O)CSc3ccccc3)n2)c(OC)c1 ZINC000217974231 GG In-Stock Unstable MTNR1A 64 37 COc1ccc(-c2noc(CNC(=O)CSc3ccccc3)n2)c(OC)c1 ZINC000217974231 GG In-Stock Unstable MTNR1B 57 37 COc1ccc(-c2noc(CNC(=O)CSc3ccccc3)n2)c(OC)c1 ZINC000217974231 GG In-Stock Unstable NR4A2 0 40 COc1ccc(-c2noc(CNC(=O)CSc3ccccc3)n2)c(OC)c1 ZINC000217974231 GG In-Stock Unstable FAS 43 36 CCOc1ccc(NC(=O)N2C[C@H](Oc3ccccc3F)C[C@H]2C(=O)OC)cc1 ZINC000217974283 HG For-Sale Unstable TSHR 49 36 CSCC[C@@H](NC(=O)N/C=C/c1cccc(F)c1)C(=O)O ZINC000217974341 DE For-Sale Unstable NAALAD2 42 34 CSCC[C@@H](NC(=O)N/C=C/c1cccc(F)c1)C(=O)O ZINC000217974341 DE For-Sale Unstable PAM 0 41 Cn1cc(S(=O)(=O)Nc2nc3ccccc3nc2NCCc2c[nH]c3ccccc23)cn1 ZINC000217974342 IG In-Stock Unstable ALOX15 27 46 C[C@@H]1CN(CC(=O)N2CCc3ccc(Nc4ccccc4)cc32)CCN1 ZINC000217974343 FF Annotated Unstable MLNR 61 37 COc1ccc2[nH]cc(/C=C\C(=O)CCl)c2c1 ZINC000217974359 BF For-Sale Unstable HTR1D 17 48 COc1ccc2[nH]cc(/C=C\C(=O)CCl)c2c1 ZINC000217974359 BF For-Sale Unstable NQO2 22 49 COc1ccc2[nH]cc(/C=C\C(=O)CCl)c2c1 ZINC000217974359 BF For-Sale Unstable HTR1E 15 43 COc1ccc2[nH]cc(/C=C\C(=O)CCl)c2c1 ZINC000217974359 BF For-Sale Unstable MTNR1A 60 50 COc1ccc2[nH]cc(/C=C\C(=O)CCl)c2c1 ZINC000217974359 BF For-Sale Unstable MTNR1B 45 49 COc1ccc2[nH]cc(/C=C\C(=O)CCl)c2c1 ZINC000217974359 BF For-Sale Unstable TDO2 0 43 COc1ccc2[nH]cc(/C=C\C(=O)CCl)c2c1 ZINC000217974359 BF For-Sale Unstable TUBB2B 41 39 CCOc1ccc(NC(=O)N2C[C@@H](Oc3ccccc3F)C[C@H]2C(=O)OC)cc1 ZINC000217974362 HG For-Sale Unstable TSHR 49 36 CSCC[C@H](NC(=O)N/C=C/c1cccc(F)c1)C(=O)O ZINC000217974430 DE For-Sale Unstable NAALAD2 42 34 CSCC[C@H](NC(=O)N/C=C/c1cccc(F)c1)C(=O)O ZINC000217974430 DE For-Sale Unstable PAM 0 41 CC[C@@H](C)c1ccc(NC(=O)CN2CCC[C@@H](C(=O)N3CCOCC3)C2)cc1 ZINC000217974431 GF On-Demand Unstable MTOR 40 33 O=C(/C=C\c1c[nH]c2ccc([N+](=O)[O-])cc12)CCl ZINC000217974436 CF For-Sale Unstable GABRA1 15 48 O=C(/C=C\c1c[nH]c2ccc([N+](=O)[O-])cc12)CCl ZINC000217974436 CF For-Sale Unstable TDO2 0 41 COc1cccc(-c2noc(CN(C)C(=O)CSc3ccccc3)n2)c1 ZINC000217974476 FG In-Stock Unstable HSD17B2 20 40 CC[C@H](C)c1ccc(NC(=O)CN2CCC[C@@H](C(=O)N3CCOCC3)C2)cc1 ZINC000217974516 GF On-Demand Unstable MTOR 40 33 COc1ccc(-c2noc(CN(C)C(=O)CSc3ccccc3)n2)c(OC)c1 ZINC000217974584 GH In-Stock Unstable NR4A2 0 40 CC(C)c1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217974713 EJ In-Stock Unstable ANPEP 15 44 CC(C)c1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217974713 EJ In-Stock Unstable SDH1 0 42 CC(C)c1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217974713 EJ In-Stock Unstable MTNR1A 24 40 CC(C)c1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217974713 EJ In-Stock Unstable MTNR1B 34 40 CC(C)c1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217974713 EJ In-Stock Unstable AMP1_PLAFQ 28 44 CC(C)c1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217974713 EJ In-Stock Unstable CRTM 43 45 CC(C)c1ccc(CCCNC(=O)CSc2ccccc2)cc1 ZINC000217974713 EJ In-Stock Unstable FAS 43 40 Cc1ccc(COc2ccc(/C=C\C(=O)O)cc2)cc1C ZINC000217974719 CH For-Sale Unstable PTGER2 45 47 Cc1ccc(COc2ccc(/C=C\C(=O)O)cc2)cc1C ZINC000217974719 CH For-Sale Unstable PTGER4 26 40 Cc1ccc(COc2ccc(/C=C\C(=O)O)cc2)cc1C ZINC000217974719 CH For-Sale Unstable FFAR1 65 43 Cc1ccc(COc2ccc(/C=C\C(=O)O)cc2)cc1C ZINC000217974719 CH For-Sale Unstable AKR1C3 33 43 COc1ccc([C@@H](C)NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217974735 DH For-Sale Unstable ACACA 23 41 COc1ccc([C@@H](C)NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217974735 DH For-Sale Unstable ACACB 26 47 COc1ccc([C@@H](C)NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217974735 DH For-Sale Unstable MTNR1A 21 41 COc1ccc([C@@H](C)NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217974735 DH For-Sale Unstable MTNR1B 20 41 Cc1ccc(COc2ccccc2/C=C\C(=O)O)cc1C ZINC000217974798 CH For-Sale Unstable PTGER2 31 56 Cc1ccc(COc2ccccc2/C=C\C(=O)O)cc1C ZINC000217974798 CH For-Sale Unstable PTGER4 57 56 Cc1ccc(COc2ccccc2/C=C\C(=O)O)cc1C ZINC000217974798 CH For-Sale Unstable PTGER3 50 56 Cc1ccc(COc2ccccc2/C=C\C(=O)O)cc1C ZINC000217974798 CH For-Sale Unstable PTGDR 0 47 Cc1ccc(COc2ccccc2/C=C\C(=O)O)cc1C ZINC000217974798 CH For-Sale Unstable AKR1C3 33 44 Cc1ccc(COc2ccccc2/C=C\C(=O)O)cc1C ZINC000217974798 CH For-Sale Unstable AKR1B10 38 42 COc1ccc([C@H](C)NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217974815 DH For-Sale Unstable ACACA 23 41 COc1ccc([C@H](C)NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217974815 DH For-Sale Unstable ACACB 26 47 COc1ccc([C@H](C)NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217974815 DH For-Sale Unstable MTNR1A 21 41 COc1ccc([C@H](C)NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217974815 DH For-Sale Unstable MTNR1B 20 41 Cc1ccc(COc2cccc(/C=C\C(=O)O)c2)cc1C ZINC000217974872 CH For-Sale Unstable MAOB 38 46 Cc1ccc(COc2cccc(/C=C\C(=O)O)c2)cc1C ZINC000217974872 CH For-Sale Unstable PTGER2 24 51 Cc1ccc(COc2cccc(/C=C\C(=O)O)c2)cc1C ZINC000217974872 CH For-Sale Unstable PTGER4 35 48 Cc1ccc(COc2cccc(/C=C\C(=O)O)c2)cc1C ZINC000217974872 CH For-Sale Unstable PTGER3 48 38 Cc1ccc(COc2cccc(/C=C\C(=O)O)c2)cc1C ZINC000217974872 CH For-Sale Unstable LTB4R 17 41 Cc1ccc(COc2cccc(/C=C\C(=O)O)c2)cc1C ZINC000217974872 CH For-Sale Unstable NR1H4 54 35 Cc1ccc(COc2cccc(/C=C\C(=O)O)c2)cc1C ZINC000217974872 CH For-Sale Unstable PTGDR 0 44 Cc1ccc(COc2cccc(/C=C\C(=O)O)c2)cc1C ZINC000217974872 CH For-Sale Unstable FFAR1 76 42 Cc1ccc(COc2cccc(/C=C\C(=O)O)c2)cc1C ZINC000217974872 CH For-Sale Unstable AKR1C3 34 46 C[C@@H](CNC(=O)c1cc(N)ccc1Cl)N(C)C1CC1 ZINC000217974894 CE On-Demand Unstable P2RX7 18 48 Cc1cc2ncn(-c3ccccc3CBr)c2cc1C ZINC000217974901 DJ For-Sale Unstable PDGFRB 23 47 COc1ccc(CNC(=O)CSc2ccc(C)cc2)c(OC)c1OC ZINC000217974954 FG In-Stock Unstable SLC9A1 59 37 COc1ccc(CNC(=O)CSc2ccc(C)cc2)c(OC)c1OC ZINC000217974954 FG In-Stock Unstable ENPP1 49 30 COc1ccc(CNC(=O)CSc2ccc(C)cc2)c(OC)c1OC ZINC000217974954 FG In-Stock Unstable FAS 46 36 C[C@H](CNC(=O)c1cc(N)ccc1Cl)N(C)C1CC1 ZINC000217974972 CE On-Demand Unstable P2RX7 18 48 COc1cc(CNC(=O)CSc2ccc(C)cc2)ccc1OC(C)C ZINC000217975072 FI In-Stock Unstable TRPV1 0 41 COc1cc(CNC(=O)CSc2ccc(C)cc2)ccc1OC(C)C ZINC000217975072 FI In-Stock Unstable ENPP1 57 33 CN[C@@H](c1ccc(Cl)c(Cl)c1)[C@@H]1CCC[C@@H](C)C1 ZINC000217975076 CK For-Sale Unstable AKT1 0 40 COC(=O)c1ccc(Nc2nc3ccccc3nc2NS(=O)(=O)c2cnn(C)c2)cc1 ZINC000217975104 IF In-Stock Unstable PYGM 40 37 O=C(CCCC[C@H]1CCSS1)N1CCCC[C@H]1c1cccnc1 ZINC000217975137 FJ In-Stock Unstable CHRNA2 39 40 O=C(CCCC[C@H]1CCSS1)N1CCCC[C@H]1c1cccnc1 ZINC000217975137 FJ In-Stock Unstable COLA 102 44 O=C(CCCC[C@H]1CCSS1)N1CCCC[C@H]1c1cccnc1 ZINC000217975137 FJ In-Stock Unstable CPT1A 97 44 O=C(CCCC[C@H]1CCSS1)N1CCCC[C@H]1c1cccnc1 ZINC000217975137 FJ In-Stock Unstable GPBAR1 0 41 O=C(CCCC[C@H]1CCSS1)N1CCCC[C@H]1c1cccnc1 ZINC000217975137 FJ In-Stock Unstable CRTY 0 40 O=C(COc1cccc(F)c1)N[C@H]1CCC[C@H]1CO ZINC000217975150 CD On-Demand Unstable CHRNA10 29 40 CN[C@@H](c1ccc(Cl)c(Cl)c1)[C@H]1CCC[C@@H](C)C1 ZINC000217975158 CK For-Sale Unstable AKT1 0 40 C[C@@H](C(=O)Nc1ccc(Cl)cn1)N1CCC[C@@H](C(=O)N2CCOCC2)C1 ZINC000217975164 GD On-Demand Unstable F10 18 45 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)NC12CC3CC(CC(C3)C1)C2 ZINC000217975183 HG For-Sale Unstable EPHX2 57 41 Cc1ccc(SCC(=O)NCCCc2ccccc2Cl)cc1 ZINC000217975192 EI In-Stock Unstable FAS 43 33 Nc1nc(/C=C\c2c[nH]c3cc(Cl)ccc23)cs1 ZINC000217975206 CI For-Sale Unstable TDO2 0 50 O=C(CCCC[C@@H]1CCSS1)N1CCCC[C@H]1c1cccnc1 ZINC000217975219 FJ In-Stock Unstable CHRNA2 39 40 O=C(CCCC[C@@H]1CCSS1)N1CCCC[C@H]1c1cccnc1 ZINC000217975219 FJ In-Stock Unstable COLA 102 44 O=C(CCCC[C@@H]1CCSS1)N1CCCC[C@H]1c1cccnc1 ZINC000217975219 FJ In-Stock Unstable CPT1A 97 44 O=C(CCCC[C@@H]1CCSS1)N1CCCC[C@H]1c1cccnc1 ZINC000217975219 FJ In-Stock Unstable GPBAR1 0 41 O=C(CCCC[C@@H]1CCSS1)N1CCCC[C@H]1c1cccnc1 ZINC000217975219 FJ In-Stock Unstable CRTY 0 40 C[C@H](C(=O)Nc1ccc(Cl)cn1)N1CCC[C@@H](C(=O)N2CCOCC2)C1 ZINC000217975237 GD On-Demand Unstable F10 18 45 CN[C@@H](Cc1ccc(Cl)cc1)[C@@H]1CCC[C@@H](C)C1 ZINC000217975239 CI For-Sale Unstable AVPR1A 31 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)NC12CC3CC(CC(C3)C1)C2 ZINC000217975250 HG For-Sale Unstable EPHX2 57 41 CC(C)Oc1ccc(C(=O)N[C@@H]2CCC[C@@H]2CO)cc1 ZINC000217975251 CE On-Demand Unstable SSTR3 26 43 CCc1ccc([C@@H](C)NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217975276 DI For-Sale Unstable KCNQ2 45 34 CCc1ccc([C@@H](C)NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217975276 DI For-Sale Unstable NR1H4 15 40 Cc1ccc(SCC(=O)NCCCc2ccc(Cl)cc2)cc1 ZINC000217975281 EI In-Stock Unstable CRTM 29 40 CN[C@@H](Cc1ccc(Cl)cc1)[C@H]1CCC[C@@H](C)C1 ZINC000217975312 CI For-Sale Unstable AVPR1A 31 40 Cn1cc(S(=O)(=O)Nc2nc3ccccc3nc2Nc2ccc(F)c(Cl)c2)cn1 ZINC000217975319 IH In-Stock Unstable EGFR 42 41 Cn1cc(S(=O)(=O)Nc2nc3ccccc3nc2Nc2ccc(F)c(Cl)c2)cn1 ZINC000217975319 IH In-Stock Unstable ERBB2 20 41 Cn1cc(S(=O)(=O)Nc2nc3ccccc3nc2Nc2ccc(F)c(Cl)c2)cn1 ZINC000217975319 IH In-Stock Unstable ERBB4 46 35 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)NC12CC3CC(CC(C3)C1)C2 ZINC000217975327 HG For-Sale Unstable EPHX2 57 41 CC(C)Oc1ccc(C(=O)N[C@H]2CCC[C@@H]2CO)cc1 ZINC000217975337 CE For-Sale Unstable SSTR3 27 43 CC(C)Oc1ccc(C(=O)N[C@H]2CCC[C@@H]2CO)cc1 ZINC000217975337 CE For-Sale Unstable PLAU 24 43 CCc1ccc([C@H](C)NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217975358 DI For-Sale Unstable KCNQ2 45 34 CCc1ccc([C@H](C)NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217975358 DI For-Sale Unstable NR1H4 15 40 Cc1ccc(SCC(=O)NCCCc2ccc(F)cc2)cc1 ZINC000217975392 DH In-Stock Unstable CRTM 17 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)NC12CC3CC(CC(C3)C1)C2 ZINC000217975409 HG For-Sale Unstable EPHX2 57 41 COc1ccc(Nc2nc3ccccc3nc2NS(=O)(=O)c2cnn(C)c2)c(OC)c1 ZINC000217975423 IF In-Stock Unstable MAPK7 47 33 CC(C)Oc1ccc(C(=O)N[C@@H]2CCC[C@H]2CO)cc1 ZINC000217975424 CE For-Sale Unstable SSTR3 27 43 CC(C)Oc1ccc(C(=O)N[C@@H]2CCC[C@H]2CO)cc1 ZINC000217975424 CE For-Sale Unstable PLAU 24 43 C[C@@H](NC(=O)N/C=C/c1cccc(F)c1)c1ccc2c(c1)CCCC2 ZINC000217975465 EJ For-Sale Unstable KCNQ2 46 34 COc1ccccc1CCCNC(=O)CSc1ccc(C)cc1 ZINC000217975490 EH In-Stock Unstable DRD2 22 41 COc1ccccc1CCCNC(=O)CSc1ccc(C)cc1 ZINC000217975490 EH In-Stock Unstable HTR7 15 41 COc1ccccc1CCCNC(=O)CSc1ccc(C)cc1 ZINC000217975490 EH In-Stock Unstable MTNR1B 43 42 COc1ccccc1CCCNC(=O)CSc1ccc(C)cc1 ZINC000217975490 EH In-Stock Unstable FAS 62 37 CC(C)Oc1ccc(C(=O)N[C@H]2CCC[C@H]2CO)cc1 ZINC000217975506 CE For-Sale Unstable SSTR3 27 43 CC(C)Oc1ccc(C(=O)N[C@H]2CCC[C@H]2CO)cc1 ZINC000217975506 CE For-Sale Unstable PLAU 24 43 C[C@H](NC(=O)N/C=C/c1cccc(F)c1)c1ccc2c(c1)CCCC2 ZINC000217975547 EJ For-Sale Unstable KCNQ2 46 34 C[C@@H](C(=O)Nc1sc2c(c1C#N)CCCCC2)N1CCC[C@@H](C(=O)N2CCOCC2)C1 ZINC000217975558 IF On-Demand Unstable MAPK10 0 43 Cc1cc2ncn(-c3ccc(CBr)cc3)c2cc1C ZINC000217975559 DJ For-Sale Unstable PDGFRB 27 52 COc1cccc(CCCNC(=O)CSc2ccc(C)cc2)c1 ZINC000217975598 EH In-Stock Unstable DRD4 45 39 COc1cccc(CCCNC(=O)CSc2ccc(C)cc2)c1 ZINC000217975598 EH In-Stock Unstable HRH2 26 41 COc1cccc(CCCNC(=O)CSc2ccc(C)cc2)c1 ZINC000217975598 EH In-Stock Unstable MTNR1A 78 48 COc1cccc(CCCNC(=O)CSc2ccc(C)cc2)c1 ZINC000217975598 EH In-Stock Unstable MTNR1B 65 61 COc1cccc(CCCNC(=O)CSc2ccc(C)cc2)c1 ZINC000217975598 EH In-Stock Unstable ROCK2 41 33 COc1cccc(CCCNC(=O)CSc2ccc(C)cc2)c1 ZINC000217975598 EH In-Stock Unstable FPR2 20 41 COc1cccc(CCCNC(=O)CSc2ccc(C)cc2)c1 ZINC000217975598 EH In-Stock Unstable CRTM 73 46 COc1cccc(CCCNC(=O)CSc2ccc(C)cc2)c1 ZINC000217975598 EH In-Stock Unstable CRTH2 0 41 COc1cccc(CCCNC(=O)CSc2ccc(C)cc2)c1 ZINC000217975598 EH In-Stock Unstable FAS 54 41 C[C@H](C(=O)Nc1sc2c(c1C#N)CCCCC2)N1CCC[C@@H](C(=O)N2CCOCC2)C1 ZINC000217975643 IF On-Demand Unstable MAPK10 0 43 COc1ccc(CCCNC(=O)CSc2ccc(C)cc2)cc1 ZINC000217975674 EH In-Stock Unstable MTNR1A 56 38 COc1ccc(CCCNC(=O)CSc2ccc(C)cc2)cc1 ZINC000217975674 EH In-Stock Unstable MTNR1B 47 42 COc1ccc(CCCNC(=O)CSc2ccc(C)cc2)cc1 ZINC000217975674 EH In-Stock Unstable CA9 15 44 COc1ccc(CCCNC(=O)CSc2ccc(C)cc2)cc1 ZINC000217975674 EH In-Stock Unstable CRTM 40 38 COc1ccc(CCCNC(=O)CSc2ccc(C)cc2)cc1 ZINC000217975674 EH In-Stock Unstable FAS 53 45 COc1ccc2c(ccn2CCNC(=O)CCCCCNc2ccc3c(cc2=O)[C@@H](NC(C)=O)CCc2cc(OC)c(OC)c(OC)c2-3)c1 ZINC000217975741 KK In-Stock Unstable TUBA1A 15 57 COc1ccc(OC[C@@H](C)NC(=O)CSc2ccc(C)cc2)cc1 ZINC000217975771 EH In-Stock Unstable FAS 43 45 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217975780 EK For-Sale Anodyne CA1 36 45 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217975780 EK For-Sale Anodyne RAF1 28 41 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217975780 EK For-Sale Anodyne NPY5R 21 40 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000217975780 EK For-Sale Anodyne Q8MMZ8_EIMTE 46 41 COC(=O)C[C@H](c1ccc(O)c(OC)c1)c1oc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c1O ZINC000217975853 KF In-Stock Unstable CHRNA4 26 43 COc1ccc(OC[C@H](C)NC(=O)CSc2ccc(C)cc2)cc1 ZINC000217975857 EH In-Stock Unstable FAS 43 45 Cc1ccc(Cl)cc1NC(=O)N/C=C/c1cccc(F)c1 ZINC000217975884 DJ For-Sale Unstable CMA1 23 40 COC(=O)C[C@@H](c1ccc(O)c(OC)c1)c1oc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c1O ZINC000217975934 KF In-Stock Unstable CHRNA4 26 43 CCc1ncnc(NCc2cccc(COC)c2)c1F ZINC000217975940 CF On-Demand Unstable CLK4 22 41 Cc1ccc(SCC(=O)NCCCc2cccc(OC(C)C)c2)cc1 ZINC000217975974 FJ In-Stock Unstable HRH2 22 40 Cc1ccc(SCC(=O)NCCCc2cccc(OC(C)C)c2)cc1 ZINC000217975974 FJ In-Stock Unstable AMP1_PLAFQ 15 40 Cc1ccc(SCC(=O)NCCCc2cccc(OC(C)C)c2)cc1 ZINC000217975974 FJ In-Stock Unstable CRTM 66 44 Cc1ccc(SCC(=O)NCCCc2cccc(OC(C)C)c2)cc1 ZINC000217975974 FJ In-Stock Unstable CRTH2 0 41 COc1ccc(OC)c(NC(=O)N/C=C/c2cccc(F)c2)c1 ZINC000217975990 DH For-Sale Unstable CYP1B1 46 35 COc1ccc(OC)c(NC(=O)N/C=C/c2cccc(F)c2)c1 ZINC000217975990 DH For-Sale Unstable MTNR1A 29 44 COc1ccc(OC)c(NC(=O)N/C=C/c2cccc(F)c2)c1 ZINC000217975990 DH For-Sale Unstable MTNR1B 31 44 COc1ccc(OC)c(NC(=O)N/C=C/c2cccc(F)c2)c1 ZINC000217975990 DH For-Sale Unstable AKR1C2 45 34 Cc1noc(C)c1CCC(=O)N1CCCC[C@H]1c1cccnc1 ZINC000217976047 DG In-Stock Unstable CHRNA2 41 42 Cc1noc(C)c1CCC(=O)N1CCCC[C@H]1c1cccnc1 ZINC000217976047 DG In-Stock Unstable COLA 116 42 Cc1noc(C)c1CCC(=O)N1CCCC[C@H]1c1cccnc1 ZINC000217976047 DG In-Stock Unstable CPT1A 101 41 Cc1noc(C)c1CCC(=O)N1CCCC[C@H]1c1cccnc1 ZINC000217976047 DG In-Stock Unstable C3AR1 42 36 Cc1noc(C)c1CCC(=O)N1CCCC[C@H]1c1cccnc1 ZINC000217976047 DG In-Stock Unstable GPBAR1 0 46 COc1cccc(CCNc2cc(Cl)nc(C3CC3)n2)c1 ZINC000217976059 DH On-Demand Unstable PTGDR 29 40 CCC[C@@H](O)CNC(=O)[C@@H](N)COC ZINC000217976114 BB On-Demand Unstable DPP7 0 40 CCC[C@H](O)CNC(=O)[C@@H](N)COC ZINC000217976187 BB On-Demand Unstable DPP7 0 40 Cc1ccc(SCC(=O)NCCN(C)c2ccccc2)cc1 ZINC000217976201 DG In-Stock Unstable FAS 52 37 Cc1cc(C)c(NC(=O)N/C=C/c2cccc(F)c2)c(C)c1 ZINC000217976210 CJ For-Sale Unstable PYGL 42 39 CCC[C@@H](O)CNC(=O)[C@H](N)COC ZINC000217976280 BB On-Demand Unstable DPP7 0 40 Cc1ccc(SCC(=O)Nc2ccc(OC3CCCC3)cc2)cc1 ZINC000217976310 EK In-Stock Unstable FAS 53 39 Cn1ccc2ccc(C(=O)NCC(=O)NCC(=O)O)cc21 ZINC000217976341 CC In-Stock Unstable CA2 23 47 Cn1ccc2ccc(C(=O)NCC(=O)NCC(=O)O)cc21 ZINC000217976341 CC In-Stock Unstable EGLN1 0 40 CCC[C@H](O)CNC(=O)[C@H](N)COC ZINC000217976366 BB On-Demand Unstable DPP7 0 40 Cc1ccc(SCC(=O)N[C@@H]2CC(C)(C)Oc3ccccc32)cc1 ZINC000217976403 EJ In-Stock Unstable FAS 48 34 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(F)cc1 ZINC000217976406 CH For-Sale Anodyne IMPDH2 0 43 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(F)cc1 ZINC000217976406 CH For-Sale Anodyne MMP1 0 52 N[C@H](C(=O)O)c1nonc1OCc1ccccc1 ZINC000217976408 BC For-Sale Unstable CACNA2D1 20 40 Cn1cc(S(=O)(=O)Nc2nc3ccccc3nc2Nc2cccc(OC(F)F)c2)cn1 ZINC000217976423 IH In-Stock Unstable GALR2 22 40 CCOc1cccc(CNc2cc(Cl)nc(C3CC3)n2)c1 ZINC000217976443 DI On-Demand Unstable PDS 44 37 CC(C)c1ccc(N2C(=O)N[C@@H](CC(=O)NCCc3c[nH]c4ccccc34)C2=O)cc1 ZINC000217976446 HG In-Stock Unstable EDNRA 32 40 CC(C)c1ccc(N2C(=O)N[C@@H](CC(=O)NCCc3c[nH]c4ccccc34)C2=O)cc1 ZINC000217976446 HG In-Stock Unstable TACR1 32 42 CC(C)c1ccc(N2C(=O)N[C@@H](CC(=O)NCCc3c[nH]c4ccccc34)C2=O)cc1 ZINC000217976446 HG In-Stock Unstable MC4R 36 41 CC(C)c1ccc(N2C(=O)N[C@@H](CC(=O)NCCc3c[nH]c4ccccc34)C2=O)cc1 ZINC000217976446 HG In-Stock Unstable TACR2 41 36 CC(C)c1ccc(N2C(=O)N[C@@H](CC(=O)NCCc3c[nH]c4ccccc34)C2=O)cc1 ZINC000217976446 HG In-Stock Unstable CCKAR 41 39 CC(C)c1ccc(N2C(=O)N[C@@H](CC(=O)NCCc3c[nH]c4ccccc34)C2=O)cc1 ZINC000217976446 HG In-Stock Unstable BRS3 27 42 CC(C)c1ccc(N2C(=O)N[C@@H](CC(=O)NCCc3c[nH]c4ccccc34)C2=O)cc1 ZINC000217976446 HG In-Stock Unstable NMBR 42 41 CC(C)c1ccc(N2C(=O)N[C@@H](CC(=O)NCCc3c[nH]c4ccccc34)C2=O)cc1 ZINC000217976446 HG In-Stock Unstable CFTR 17 41 CC(C)c1ccc(N2C(=O)N[C@@H](CC(=O)NCCc3c[nH]c4ccccc34)C2=O)cc1 ZINC000217976446 HG In-Stock Unstable ALOX15 18 46 CC(C)c1ccc(N2C(=O)N[C@@H](CC(=O)NCCc3c[nH]c4ccccc34)C2=O)cc1 ZINC000217976446 HG In-Stock Unstable MMP9 15 44 Cc1ccc(SCC(=O)N[C@H]2CC(C)(C)Oc3ccccc32)cc1 ZINC000217976477 EJ In-Stock Unstable FAS 48 34 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(Cl)c([N+](=O)[O-])c1 ZINC000217976493 EI For-Sale Bother IMDH_CRYPV 33 46 N[C@@H](C(=O)O)c1nonc1OCc1ccccc1 ZINC000217976497 BC For-Sale Unstable CACNA2D1 20 40 CCOc1ccc(/C=C2/CC(=O)NC2=O)cc1OC ZINC000217976503 CD For-Sale Unstable ESRRA 53 41 CCOc1ccc(/C=C2/CC(=O)NC2=O)cc1OC ZINC000217976503 CD For-Sale Unstable HPGD 49 47 CCOc1cccc(CNc2ncnc(CC)c2F)c1 ZINC000217976540 CG On-Demand Unstable CLK4 25 44 CCOc1cccc(CNc2ncnc(CC)c2F)c1 ZINC000217976540 CG On-Demand Unstable PDS 52 35 COC(=O)C[C@@H](C1=C(O)C(=O)C([C@@H](CC(=O)OC)c2cc3ccccc3[nH]c2=O)=C(O)C1=O)c1cc2ccccc2[nH]c1=O ZINC000217976547 KG In-Stock Unstable DDO 0 42 CCOc1ccc(CCCNC(=O)CSc2ccc(C)cc2)cc1 ZINC000217976574 EI In-Stock Unstable SCN2A 21 42 COc1cc([N+](=O)[O-])ccc1NC(=O)N/C=C/c1cccc(F)c1 ZINC000217976594 EH For-Sale Unstable CACNA1D 46 36 COc1cc([N+](=O)[O-])ccc1NC(=O)N/C=C/c1cccc(F)c1 ZINC000217976594 EH For-Sale Unstable KCNMA1 23 50 COC(=O)C[C@@H](C1=C(O)C(=O)C([C@H](CC(=O)OC)c2cc3ccccc3[nH]c2=O)=C(O)C1=O)c1cc2ccccc2[nH]c1=O ZINC000217976632 KG In-Stock Unstable DDO 0 42 COc1cc(/C=C2/CC(=O)NC2=O)ccc1OC(C)C ZINC000217976647 CD For-Sale Unstable ESRRA 51 41 COc1cc(/C=C2/CC(=O)NC2=O)ccc1OC(C)C ZINC000217976647 CD For-Sale Unstable HPGD 26 40 CC(C)(C)OC(=O)N1C[C@@H]2CN(C(=O)c3ccc(S(N)(=O)=O)cc3)C[C@@H]2C1 ZINC000217976651 GD On-Demand Unstable CA2 50 42 CC(C)(C)OC(=O)N1C[C@@H]2CN(C(=O)c3ccc(S(N)(=O)=O)cc3)C[C@@H]2C1 ZINC000217976651 GD On-Demand Unstable CA1 31 42 CC(C)(C)OC(=O)N1C[C@@H]2CN(C(=O)c3ccc(S(N)(=O)=O)cc3)C[C@@H]2C1 ZINC000217976651 GD On-Demand Unstable CA7 36 42 CC(C)(C)OC(=O)N1C[C@@H]2CN(C(=O)c3ccc(S(N)(=O)=O)cc3)C[C@@H]2C1 ZINC000217976651 GD On-Demand Unstable CA4 24 42 CC(C)(C)OC(=O)N1C[C@@H]2CN(C(=O)c3ccc(S(N)(=O)=O)cc3)C[C@@H]2C1 ZINC000217976651 GD On-Demand Unstable CA14 33 40 CC(C)(C)OC(=O)N1C[C@@H]2CN(C(=O)c3ccc(S(N)(=O)=O)cc3)C[C@@H]2C1 ZINC000217976651 GD On-Demand Unstable CA12 26 42 CC(C)(C)OC(=O)N1C[C@@H]2CN(C(=O)c3ccc(S(N)(=O)=O)cc3)C[C@@H]2C1 ZINC000217976651 GD On-Demand Unstable CA9 26 42 CC(C)(C)OC(=O)N1C[C@@H]2CN(C(=O)c3ccc(S(N)(=O)=O)cc3)C[C@@H]2C1 ZINC000217976651 GD On-Demand Unstable GPR119 42 45 CCCOc1ccccc1CCCNC(=O)CSc1ccc(C)cc1 ZINC000217976678 FJ In-Stock Unstable MTNR1B 41 38 O=C(N/C=C/c1cccc(F)c1)Nc1ccc([N+](=O)[O-])cc1 ZINC000217976699 DH For-Sale Bother TRPM8 15 43 COC(=O)C[C@H](C1=C(O)C(=O)C([C@@H](CC(=O)OC)c2cc3ccccc3[nH]c2=O)=C(O)C1=O)c1cc2ccccc2[nH]c1=O ZINC000217976712 KG In-Stock Unstable DDO 0 42 NCc1cccc(CN2CCC[C@@H]3CCCC[C@H]32)c1 ZINC000217976722 CG For-Sale Unstable SLC18A3 20 43 Cc1ccc(SCC(=O)N[C@@H](C)COc2ccccc2C)cc1 ZINC000217976745 EH In-Stock Unstable FAS 46 35 Fc1cccc(CN[C@@H]2C[C@@H]3CC=C[C@H]32)c1 ZINC000217976776 BF For-Sale Unstable HRH2 0 50 NCc1cccc(CN2CCC[C@H]3CCCC[C@H]32)c1 ZINC000217976802 CG For-Sale Unstable SLC18A3 20 43 O=C(N/C=C/c1cccc(F)c1)Nc1cccc([N+](=O)[O-])c1 ZINC000217976804 DH For-Sale Bother TRPM8 17 53 O=C(Cn1ccc2c(Cl)cccc21)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217976822 GG In-Stock Unstable CHRNA4 30 48 Cc1ccc(OC[C@@H](C)NC(=O)CSc2ccc(C)cc2)cc1 ZINC000217976858 EH In-Stock Unstable ACACA 43 36 Cc1ccc(OC[C@@H](C)NC(=O)CSc2ccc(C)cc2)cc1 ZINC000217976858 EH In-Stock Unstable FAS 41 38 Fc1cccc(CN[C@H]2C[C@@H]3CC=C[C@H]32)c1 ZINC000217976871 BF For-Sale Unstable HRH2 0 50 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)Nc1ccc(OC)cc1 ZINC000217976898 GG For-Sale Unstable TSHR 41 34 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)Nc1ccc(OC)cc1 ZINC000217976898 GG For-Sale Unstable AGTR2 21 43 O=C(N/C=C/c1cccc(F)c1)Nc1cc([N+](=O)[O-])ccc1Cl ZINC000217976909 EI For-Sale Bother TRPM8 0 49 Cc1ccc(OC[C@H](C)NC(=O)CSc2ccc(C)cc2)cc1 ZINC000217976923 EH In-Stock Unstable ACACA 43 36 Cc1ccc(OC[C@H](C)NC(=O)CSc2ccc(C)cc2)cc1 ZINC000217976923 EH In-Stock Unstable FAS 41 38 CC(C)CCn1cnc2ccc(NC(=O)CCCn3cnc4ccccc4c3=O)cc2c1=O ZINC000217976928 IH In-Stock Unstable HTR7 24 42 CC(C)CCn1cnc2ccc(NC(=O)CCCn3cnc4ccccc4c3=O)cc2c1=O ZINC000217976928 IH In-Stock Unstable SCD1 0 48 CC(C)CCn1cnc2ccc(NC(=O)CCCn3cnc4ccccc4c3=O)cc2c1=O ZINC000217976928 IH In-Stock Unstable SCD 0 43 CC(C)CCn1cnc2ccc(NC(=O)CCCn3cnc4ccccc4c3=O)cc2c1=O ZINC000217976928 IH In-Stock Unstable IMDH_CRYPV 40 39 Fc1cccc(CN[C@@H]2C[C@H]3CC=C[C@H]32)c1 ZINC000217976944 BF For-Sale Unstable HRH2 0 50 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)Nc1ccc(OC)cc1 ZINC000217976973 GG For-Sale Unstable TSHR 41 34 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)Nc1ccc(OC)cc1 ZINC000217976973 GG For-Sale Unstable AGTR2 21 43 Fc1cccc(CN[C@H]2C[C@H]3CC=C[C@@H]23)c1 ZINC000217977016 BF For-Sale Unstable HRH2 0 50 CC(C)Oc1ccc(C(=O)N2CCN(C(=O)c3cnn4c3CCCC4)CC2)cc1 ZINC000217977064 GF In-Stock Unstable L3MBTL3 54 33 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)Nc1ccc(OC)cc1 ZINC000217977069 GG For-Sale Unstable TSHR 41 34 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)Nc1ccc(OC)cc1 ZINC000217977069 GG For-Sale Unstable AGTR2 21 43 CS(=O)(=O)c1ccc(C2(C(=O)O)CC2)c(F)c1 ZINC000217977138 CD For-Sale Unstable PTGS2 29 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)Nc1ccc(OC)cc1 ZINC000217977162 GG For-Sale Unstable TSHR 41 34 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)Nc1ccc(OC)cc1 ZINC000217977162 GG For-Sale Unstable AGTR2 21 43 CCCCCOc1ccc(/C=C/C=C\C(=O)O)cc1 ZINC000217977172 CH For-Sale Unstable PPARG 16 44 CCCCCOc1ccc(/C=C/C=C\C(=O)O)cc1 ZINC000217977172 CH For-Sale Unstable PLA2G4A 30 48 CCCCCOc1ccc(/C=C/C=C\C(=O)O)cc1 ZINC000217977172 CH For-Sale Unstable PLA2G4B 113 48 CCCCCOc1ccc(/C=C/C=C\C(=O)O)cc1 ZINC000217977172 CH For-Sale Unstable FAAH 26 44 O=C(c1cccc(C(F)(F)F)c1)N1CCN(C(=O)c2cnn3c2CCCC3)CC1 ZINC000217977180 HF In-Stock Unstable CACNA1B 46 38 O=C(c1cccc(C(F)(F)F)c1)N1CCN(C(=O)c2cnn3c2CCCC3)CC1 ZINC000217977180 HF In-Stock Unstable HPGD 25 44 O=C(c1cccc(C(F)(F)F)c1)N1CCN(C(=O)c2cnn3c2CCCC3)CC1 ZINC000217977180 HF In-Stock Unstable SLC6A7 0 42 C[C@@H](NC(=O)N1CCCC[C@H]1C(=O)O)[C@@H]1C[C@@H]2CC[C@@H]1C2 ZINC000217977217 CE For-Sale Unstable ACE 42 43 C[C@@H](NC(=O)N1CCCC[C@H]1C(=O)O)[C@@H]1C[C@@H]2CC[C@@H]1C2 ZINC000217977217 CE For-Sale Unstable REN 15 41 O=C(N/C=C/c1cccc(F)c1)N1CCN(c2ccc(F)cc2)CC1 ZINC000217977236 EG For-Sale Unstable AKR1C3 0 44 CCCc1ccc(/C=C\C(=O)CCl)cc1 ZINC000217977240 BG For-Sale Unstable NA 0 40 CCCc1ccc(/C=C\C(=O)CCl)cc1 ZINC000217977240 BG For-Sale Unstable SSSIM 15 44 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)NCc1ccc(OC)cc1 ZINC000217977269 HF For-Sale Unstable MMP13 29 43 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)NCc1ccc(OC)cc1 ZINC000217977269 HF For-Sale Unstable MMP3 27 43 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)NCc1ccc(OC)cc1 ZINC000217977269 HF For-Sale Unstable MMP9 18 43 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)NCc1ccc(OC)cc1 ZINC000217977269 HF For-Sale Unstable MMP7 22 43 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)NCc1ccc(OC)cc1 ZINC000217977269 HF For-Sale Unstable MMP1 23 43 C[C@H](NC(=O)N1CCCC[C@H]1C(=O)O)[C@@H]1C[C@@H]2CC[C@@H]1C2 ZINC000217977304 CE For-Sale Unstable ACE 42 43 C[C@H](NC(=O)N1CCCC[C@H]1C(=O)O)[C@@H]1C[C@@H]2CC[C@@H]1C2 ZINC000217977304 CE For-Sale Unstable REN 15 41 CCCCCOc1ccc(/C=C/C=C/C(=O)O)cc1 ZINC000217977305 CH For-Sale Unstable ALOX5 15 56 CCCCCOc1ccc(/C=C/C=C/C(=O)O)cc1 ZINC000217977305 CH For-Sale Unstable THRA 53 42 CCCCCOc1ccc(/C=C/C=C/C(=O)O)cc1 ZINC000217977305 CH For-Sale Unstable PPARG 16 44 CCCCCOc1ccc(/C=C/C=C/C(=O)O)cc1 ZINC000217977305 CH For-Sale Unstable RARB 16 50 CCCCCOc1ccc(/C=C/C=C/C(=O)O)cc1 ZINC000217977305 CH For-Sale Unstable THRB 34 42 CCCCCOc1ccc(/C=C/C=C/C(=O)O)cc1 ZINC000217977305 CH For-Sale Unstable PLA2G4A 30 48 CCCCCOc1ccc(/C=C/C=C/C(=O)O)cc1 ZINC000217977305 CH For-Sale Unstable PLA2G4B 113 48 CCCCCOc1ccc(/C=C/C=C/C(=O)O)cc1 ZINC000217977305 CH For-Sale Unstable FAAH 26 44 CCOCCOc1ccccc1C(=O)N(C)Cc1nc(C)c[nH]1 ZINC000217977329 DE In-Stock Unstable HCN1 40 32 CCOCCOc1ccccc1C(=O)N(C)Cc1nc(C)c[nH]1 ZINC000217977329 DE In-Stock Unstable HCN4 40 32 O=C(N/C=C/c1cccc(F)c1)Nc1ccccc1O ZINC000217977350 CG For-Sale Anodyne MMP1 0 49 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)NCc1ccc(OC)cc1 ZINC000217977356 HF For-Sale Unstable MMP13 29 43 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)NCc1ccc(OC)cc1 ZINC000217977356 HF For-Sale Unstable MMP3 27 43 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)NCc1ccc(OC)cc1 ZINC000217977356 HF For-Sale Unstable MMP9 18 43 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)NCc1ccc(OC)cc1 ZINC000217977356 HF For-Sale Unstable MMP7 22 43 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)NCc1ccc(OC)cc1 ZINC000217977356 HF For-Sale Unstable MMP1 23 43 C=C(CCCC)C(=O)[C@H](NC(=O)OC(C)(C)C)C(C)C ZINC000217977381 CH For-Sale Unstable CTSK 22 46 C=C(CCCC)C(=O)[C@H](NC(=O)OC(C)(C)C)C(C)C ZINC000217977381 CH For-Sale Unstable PGA5 29 51 C=C(CCCC)C(=O)[C@H](NC(=O)OC(C)(C)C)C(C)C ZINC000217977381 CH For-Sale Unstable POLG_HCV1 22 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)NCc1ccc(OC)cc1 ZINC000217977435 HF For-Sale Unstable MMP13 29 43 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)NCc1ccc(OC)cc1 ZINC000217977435 HF For-Sale Unstable MMP3 27 43 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)NCc1ccc(OC)cc1 ZINC000217977435 HF For-Sale Unstable MMP9 18 43 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)NCc1ccc(OC)cc1 ZINC000217977435 HF For-Sale Unstable MMP7 22 43 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)NCc1ccc(OC)cc1 ZINC000217977435 HF For-Sale Unstable MMP1 23 43 NCc1cccc(OCCN2CCC[C@@H]3CCCC[C@H]32)c1 ZINC000217977475 CG For-Sale Unstable HRH3 24 44 NCc1cccc(OCCN2CCC[C@@H]3CCCC[C@H]32)c1 ZINC000217977475 CG For-Sale Unstable CHRNA10 54 36 CC[C@@H](CCO)NC(=O)[C@H](C#N)CC ZINC000217977509 AC On-Demand Unstable CTSC 16 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)NCc1ccc(OC)cc1 ZINC000217977518 HF For-Sale Unstable MMP13 29 43 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)NCc1ccc(OC)cc1 ZINC000217977518 HF For-Sale Unstable MMP3 27 43 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)NCc1ccc(OC)cc1 ZINC000217977518 HF For-Sale Unstable MMP9 18 43 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)NCc1ccc(OC)cc1 ZINC000217977518 HF For-Sale Unstable MMP7 22 43 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)NCc1ccc(OC)cc1 ZINC000217977518 HF For-Sale Unstable MMP1 23 43 CC[C@H](C(=O)N1CCN(C(=O)c2cnn3c2CCCC3)CC1)c1ccccc1 ZINC000217977521 GF In-Stock Unstable KCNQ2 44 39 O=[N+]([O-])c1ccccc1CNc1cc(Cl)nc(C2CC2)n1 ZINC000217977540 DH In-Stock Unstable PRKCQ 26 44 NCc1cccc(OCCN2CCC[C@H]3CCCC[C@H]32)c1 ZINC000217977554 CG For-Sale Unstable HRH3 24 44 NCc1cccc(OCCN2CCC[C@H]3CCCC[C@H]32)c1 ZINC000217977554 CG For-Sale Unstable CHRNA10 54 36 COC(=O)[C@@H](C)N[C@@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217977573 BF For-Sale Unstable TRPM8 18 47 CC[C@@H](CCO)NC(=O)[C@@H](C#N)CC ZINC000217977594 AC On-Demand Unstable CTSC 16 40 CC[C@@H](C(=O)N1CCN(C(=O)c2cnn3c2CCCC3)CC1)c1ccccc1 ZINC000217977599 GF In-Stock Unstable KCNQ2 44 39 COc1ccc(N2C(=O)N[C@@H](CC(=O)NCCc3c[nH]c4ccccc34)C2=O)cc1 ZINC000217977602 HE In-Stock Unstable TACR1 19 40 COc1ccc(N2C(=O)N[C@@H](CC(=O)NCCc3c[nH]c4ccccc34)C2=O)cc1 ZINC000217977602 HE In-Stock Unstable NQO2 26 46 COc1ccc(N2C(=O)N[C@@H](CC(=O)NCCc3c[nH]c4ccccc34)C2=O)cc1 ZINC000217977602 HE In-Stock Unstable CCKAR 51 45 COc1ccc(N2C(=O)N[C@@H](CC(=O)NCCc3c[nH]c4ccccc34)C2=O)cc1 ZINC000217977602 HE In-Stock Unstable BRS3 25 41 COc1ccc(N2C(=O)N[C@@H](CC(=O)NCCc3c[nH]c4ccccc34)C2=O)cc1 ZINC000217977602 HE In-Stock Unstable NMBR 26 41 COc1ccc(N2C(=O)N[C@@H](CC(=O)NCCc3c[nH]c4ccccc34)C2=O)cc1 ZINC000217977602 HE In-Stock Unstable MC5R 32 40 COc1ccc(N2C(=O)N[C@@H](CC(=O)NCCc3c[nH]c4ccccc34)C2=O)cc1 ZINC000217977602 HE In-Stock Unstable MTNR1A 71 49 COc1ccc(N2C(=O)N[C@@H](CC(=O)NCCc3c[nH]c4ccccc34)C2=O)cc1 ZINC000217977602 HE In-Stock Unstable MTNR1B 54 46 COc1ccc(N2C(=O)N[C@@H](CC(=O)NCCc3c[nH]c4ccccc34)C2=O)cc1 ZINC000217977602 HE In-Stock Unstable CCKBR 45 41 COc1ccc(N2C(=O)N[C@@H](CC(=O)NCCc3c[nH]c4ccccc34)C2=O)cc1 ZINC000217977602 HE In-Stock Unstable GHSR 47 40 Cc1ccc(SCC(=O)N[C@@H]2CC(C)(C)Oc3cc(C)ccc32)cc1 ZINC000217977609 FJ In-Stock Unstable FAS 40 32 CCc1ncnc(NCc2ccccc2[N+](=O)[O-])c1F ZINC000217977653 CF On-Demand Unstable COLA 51 35 CCc1ncnc(NCc2ccccc2[N+](=O)[O-])c1F ZINC000217977653 CF On-Demand Unstable PRKCQ 27 44 COC(=O)[C@@H](C)N[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217977659 BF For-Sale Unstable TRPM8 18 47 NCc1ccc(OCCN2CCC[C@@H]3CCCC[C@H]32)cc1 ZINC000217977664 CG For-Sale Unstable LTA4H 51 46 NCc1ccc(OCCN2CCC[C@@H]3CCCC[C@H]32)cc1 ZINC000217977664 CG For-Sale Unstable HRH3 56 41 NCc1ccc(OCCN2CCC[C@@H]3CCCC[C@H]32)cc1 ZINC000217977664 CG For-Sale Unstable PSMB2 40 41 NCc1ccc(OCCN2CCC[C@@H]3CCCC[C@H]32)cc1 ZINC000217977664 CG For-Sale Unstable PSMB1 40 41 CC[C@@H](C#N)C(=O)N[C@H](CC)CCO ZINC000217977667 AC On-Demand Unstable CTSC 16 40 Cc1ccc(SCC(=O)N[C@H]2CC(C)(C)Oc3cc(C)ccc32)cc1 ZINC000217977675 FJ In-Stock Unstable FAS 40 32 CC(=O)c1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217977694 CH For-Sale Unstable IMPDH2 0 40 NCc1ccc(OCCN2CCC[C@H]3CCCC[C@H]32)cc1 ZINC000217977729 CG For-Sale Unstable LTA4H 51 46 NCc1ccc(OCCN2CCC[C@H]3CCCC[C@H]32)cc1 ZINC000217977729 CG For-Sale Unstable HRH3 56 41 NCc1ccc(OCCN2CCC[C@H]3CCCC[C@H]32)cc1 ZINC000217977729 CG For-Sale Unstable PSMB2 40 41 NCc1ccc(OCCN2CCC[C@H]3CCCC[C@H]32)cc1 ZINC000217977729 CG For-Sale Unstable PSMB1 40 41 O=C(/C=C\c1c[nH]c2ccc(F)cc12)CCl ZINC000217977736 BG For-Sale Unstable MPO 94 45 O=C(/C=C\c1c[nH]c2ccc(F)cc12)CCl ZINC000217977736 BG For-Sale Unstable CAPN1 23 53 COC(=O)[C@H](C)N[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217977743 BF For-Sale Unstable TRPM8 18 47 COc1ccc2c(c1)[C@@H](NC(=O)CSc1ccc(C)cc1)CC(C)(C)O2 ZINC000217977784 FJ In-Stock Unstable FAS 45 39 CC(=O)c1cccc(NC(=O)N/C=C/c2cccc(F)c2)c1 ZINC000217977796 CH For-Sale Unstable CCR3 22 46 CC(=O)c1cccc(NC(=O)N/C=C/c2cccc(F)c2)c1 ZINC000217977796 CH For-Sale Unstable IMPDH2 0 40 CC(=O)c1cccc(NC(=O)N/C=C/c2cccc(F)c2)c1 ZINC000217977796 CH For-Sale Unstable AKR1C3 24 47 CC(=O)c1cccc(NC(=O)N/C=C/c2cccc(F)c2)c1 ZINC000217977796 CH For-Sale Unstable KCNK3 78 44 CC(=O)c1cccc(NC(=O)N/C=C/c2cccc(F)c2)c1 ZINC000217977796 CH For-Sale Unstable KCNK9 37 44 O=C(/C=C\c1c[nH]c2ccc(Cl)cc12)CCl ZINC000217977813 CH For-Sale Unstable TDO2 0 48 COc1ccc2c(c1)[C@H](NC(=O)CSc1ccc(C)cc1)CC(C)(C)O2 ZINC000217977856 FJ In-Stock Unstable FAS 45 39 NC[C@H](c1cc(Br)cs1)N1CCC[C@@H]1c1cccnc1 ZINC000217977876 FH For-Sale Unstable CHRNA2 44 45 NC[C@H](c1cc(Br)cs1)N1CCC[C@@H]1c1cccnc1 ZINC000217977876 FH For-Sale Unstable CRTY 0 45 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)CSc1ccc(C)cc1 ZINC000217977958 FJ In-Stock Unstable FAS 56 39 COc1ccc([C@@H]2CCCCCN2C(=O)c2cc(C(C)C)nc3onc(C)c23)cc1 ZINC000217977978 HK On-Demand Unstable COLA 45 37 COc1ccc([C@@H]2CCCCCN2C(=O)c2cc(C(C)C)nc3onc(C)c23)cc1 ZINC000217977978 HK On-Demand Unstable CPT1A 44 37 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)NCCCc1ccccc1 ZINC000217977993 HG For-Sale Unstable FKBP1A 46 37 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1C(=O)NCCCc1ccccc1 ZINC000217977993 HG For-Sale Unstable ASAH1 42 34 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)CSc1ccc(C)cc1 ZINC000217978039 FJ In-Stock Unstable FAS 56 39 COc1ccc([C@@H]2CC(=O)Oc3ccc4c(c32)O/C(=C\c2cccc(OC)c2OC)C4=O)cc1 ZINC000217978046 JJ In-Stock Unstable MT-ND4 49 30 COc1ccc([C@H]2CCCCCN2C(=O)c2cc(C(C)C)nc3onc(C)c23)cc1 ZINC000217978050 HK On-Demand Unstable COLA 45 37 COc1ccc([C@H]2CCCCCN2C(=O)c2cc(C(C)C)nc3onc(C)c23)cc1 ZINC000217978050 HK On-Demand Unstable CPT1A 44 37 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)NCCCc1ccccc1 ZINC000217978059 HG For-Sale Unstable FKBP1A 46 37 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1C(=O)NCCCc1ccccc1 ZINC000217978059 HG For-Sale Unstable ASAH1 42 34 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)NCCCc1ccccc1 ZINC000217978133 HG For-Sale Unstable FKBP1A 46 37 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)NCCCc1ccccc1 ZINC000217978133 HG For-Sale Unstable ASAH1 42 34 COc1ccc([C@H]2CC(=O)Oc3ccc4c(c32)O/C(=C\c2cccc(OC)c2OC)C4=O)cc1 ZINC000217978137 JJ In-Stock Unstable MT-ND4 49 30 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)NCCCc1ccccc1 ZINC000217978222 HG For-Sale Unstable FKBP1A 46 37 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1C(=O)NCCCc1ccccc1 ZINC000217978222 HG For-Sale Unstable ASAH1 42 34 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)NCCN3CCOCC3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217978235 KD In-Stock Unstable TUBA1A 17 64 Cc1cccc(NC(=O)N/C=C/c2cccc(F)c2)c1 ZINC000217978313 CH For-Sale Unstable CCKAR 17 43 Cc1cccc(NC(=O)N/C=C/c2cccc(F)c2)c1 ZINC000217978313 CH For-Sale Unstable CCKBR 25 41 Cc1cccc(NC(=O)N/C=C/c2cccc(F)c2)c1 ZINC000217978313 CH For-Sale Unstable IMPDH2 0 42 Cc1cccc(NC(=O)N/C=C/c2cccc(F)c2)c1 ZINC000217978313 CH For-Sale Unstable MMP1 0 51 Cc1cccc(NC(=O)N/C=C/c2cccc(F)c2)c1 ZINC000217978313 CH For-Sale Unstable KCNK3 64 50 Cc1cccc(NC(=O)N/C=C/c2cccc(F)c2)c1 ZINC000217978313 CH For-Sale Unstable KCNK9 47 50 CC[C@H](CCO)NC(=O)[C@@H](C#N)CC ZINC000217978361 AC On-Demand Unstable CTSC 16 40 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217978412 FK For-Sale Anodyne GUAB 0 48 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217978412 FK For-Sale Anodyne RAF1 29 45 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217978412 FK For-Sale Anodyne Q8MMZ8_EIMTE 48 45 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217978412 FK For-Sale Anodyne BRAF 16 41 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217978412 FK For-Sale Anodyne RIPK1 15 44 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217978412 FK For-Sale Anodyne IMDH_CRYPV 37 50 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000217978412 FK For-Sale Anodyne BLM 0 45 COC(=O)c1ccc(S(=O)(=O)N2CCN(C(=O)c3cnn4c3CCCC4)CC2)cc1 ZINC000217978434 ID In-Stock Unstable TGM2 59 36 COC(=O)c1ccc(S(=O)(=O)N2CCN(C(=O)c3cnn4c3CCCC4)CC2)cc1 ZINC000217978434 ID In-Stock Unstable F13A1 57 37 CC[C@@H](NC(=O)CSc1ccc(C)cc1)c1ccc(OC)c(OC)c1 ZINC000217978512 FI In-Stock Unstable ENPP1 62 37 CC[C@@H](NC(=O)CSc1ccc(C)cc1)c1ccc(OC)c(OC)c1 ZINC000217978512 FI In-Stock Unstable FAS 42 36 O=C(c1cnn2c1CCCC2)N1CCN(S(=O)(=O)c2ccc3c(c2)CCO3)CC1 ZINC000217978545 HD In-Stock Unstable PKM 36 41 CC[C@H](NC(=O)CSc1ccc(C)cc1)c1ccc(OC)c(OC)c1 ZINC000217978596 FI In-Stock Unstable ENPP1 62 37 CC[C@H](NC(=O)CSc1ccc(C)cc1)c1ccc(OC)c(OC)c1 ZINC000217978596 FI In-Stock Unstable FAS 42 36 COC(=O)Nc1ccc(S(=O)(=O)N2CCN(C(=O)c3cnn4c3CCCC4)CC2)cc1 ZINC000217978654 ID In-Stock Unstable TGM2 76 43 COC(=O)Nc1ccc(S(=O)(=O)N2CCN(C(=O)c3cnn4c3CCCC4)CC2)cc1 ZINC000217978654 ID In-Stock Unstable F13A1 101 45 CC[C@@H](NC(=O)CSc1ccc(C)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217978693 GH In-Stock Unstable CTSF 45 32 O=C(N[C@@H](c1cccnc1)C1CCOCC1)c1ccccc1 ZINC000217978756 CF In-Stock Unstable KCNA5 53 38 O=C(N[C@@H](c1cccnc1)C1CCOCC1)c1ccccc1 ZINC000217978756 CF In-Stock Unstable AKT1 26 51 CC[C@H](NC(=O)CSc1ccc(C)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217978760 GH In-Stock Unstable CTSF 45 32 C[C@H](O)[C@@H](NC(=O)N1c2ccccc2C[C@@H]1C)C(=O)O ZINC000217978797 CC For-Sale Unstable ACE 30 46 C[C@H](O)[C@@H](NC(=O)N1c2ccccc2C[C@@H]1C)C(=O)O ZINC000217978797 CC For-Sale Unstable DRD4 26 41 C[C@H](O)[C@@H](NC(=O)N1c2ccccc2C[C@@H]1C)C(=O)O ZINC000217978797 CC For-Sale Unstable TPP2 59 37 O=C(N[C@H](c1cccnc1)C1CCOCC1)c1ccccc1 ZINC000217978821 CF In-Stock Unstable KCNA5 53 38 O=C(N[C@H](c1cccnc1)C1CCOCC1)c1ccccc1 ZINC000217978821 CF In-Stock Unstable AKT1 26 51 O=C(N/C=C/c1cccc(F)c1)Nc1cccc(Cl)c1 ZINC000217978836 CI For-Sale Anodyne PPIA 16 40 COc1cccc(-c2noc(CNC(=O)CSc3ccc(C)cc3)n2)c1 ZINC000217978865 FG In-Stock Unstable MTNR1A 44 37 COc1cccc(-c2noc(CNC(=O)CSc3ccc(C)cc3)n2)c1 ZINC000217978865 FG In-Stock Unstable WNT3A 19 40 COc1cccc(-c2noc(CNC(=O)CSc3ccc(C)cc3)n2)c1 ZINC000217978865 FG In-Stock Unstable TNKS2 15 43 COc1cccc(-c2noc(CNC(=O)CSc3ccc(C)cc3)n2)c1 ZINC000217978865 FG In-Stock Unstable AXIN2 0 40 C[C@H](O)[C@H](NC(=O)N1c2ccccc2C[C@@H]1C)C(=O)O ZINC000217978885 CC For-Sale Unstable ACE 30 46 C[C@H](O)[C@H](NC(=O)N1c2ccccc2C[C@@H]1C)C(=O)O ZINC000217978885 CC For-Sale Unstable DRD4 26 41 C[C@H](O)[C@H](NC(=O)N1c2ccccc2C[C@@H]1C)C(=O)O ZINC000217978885 CC For-Sale Unstable TPP2 59 37 O=C(N[C@H](CN1C(=O)COC1=O)c1ccccc1)C1CC1 ZINC000217978934 CD In-Stock Unstable CCR5 21 43 O=C(N[C@H](CN1C(=O)COC1=O)c1ccccc1)C1CC1 ZINC000217978934 CD In-Stock Unstable F11 48 41 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(Cl)cc1 ZINC000217978945 CI For-Sale Anodyne GUAB 0 41 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(Cl)cc1 ZINC000217978945 CI For-Sale Anodyne MMP1 0 49 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(Cl)cc1 ZINC000217978945 CI For-Sale Anodyne P95276_MYCTO 0 42 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(Cl)cc1 ZINC000217978945 CI For-Sale Anodyne SENP1 0 41 Cc1noc2nc(C(C)C)cc(C(=O)Nc3ccccc3OC(F)(F)F)c12 ZINC000217978948 GJ On-Demand Unstable KCNK3 40 44 Cc1noc2nc(C(C)C)cc(C(=O)Nc3ccccc3OC(F)(F)F)c12 ZINC000217978948 GJ On-Demand Unstable KCNK9 43 48 Cc1cc(N)n(CC(=O)NCC2(c3ccccc3)CCCC2)n1 ZINC000217978952 DE In-Stock Unstable ACAT 0 49 Cc1cc(N)n(CC(=O)NCC2(c3ccccc3)CCCC2)n1 ZINC000217978952 DE In-Stock Unstable NPFFR1 31 41 O=C(N[C@@H](CN1C(=O)COC1=O)c1ccccc1)C1CC1 ZINC000217978996 CD In-Stock Unstable CCR5 21 43 O=C(N[C@@H](CN1C(=O)COC1=O)c1ccccc1)C1CC1 ZINC000217978996 CD In-Stock Unstable F11 48 41 O=C(N[C@H](CN1C(=O)COC1=O)c1ccccc1)c1ccco1 ZINC000217979082 DD In-Stock Unstable SOAT1 24 40 COC(=O)C[C@@H](C1=C(O)C(=O)C([C@H](CC(=O)OC)c2ccccc2)=C(O)C1=O)c1ccccc1 ZINC000217979094 JG In-Stock Unstable KCNA5 42 48 O=C(N/C=C/c1cccc(F)c1)N1CCN(Cc2ccccc2)CC1 ZINC000217979134 EG For-Sale Unstable DRD2 22 45 O=C(N/C=C/c1cccc(F)c1)N1CCN(Cc2ccccc2)CC1 ZINC000217979134 EG For-Sale Unstable DRD4 42 45 O=C(N/C=C/c1cccc(F)c1)N1CCN(Cc2ccccc2)CC1 ZINC000217979134 EG For-Sale Unstable ACHE 23 44 O=C(N/C=C/c1cccc(F)c1)N1CCN(Cc2ccccc2)CC1 ZINC000217979134 EG For-Sale Unstable SIGMAR1 51 49 O=C(N/C=C/c1cccc(F)c1)N1CCN(Cc2ccccc2)CC1 ZINC000217979134 EG For-Sale Unstable CCR3 37 50 O=C(N/C=C/c1cccc(F)c1)N1CCN(Cc2ccccc2)CC1 ZINC000217979134 EG For-Sale Unstable MLNR 40 39 O=C(N/C=C/c1cccc(F)c1)N1CCN(Cc2ccccc2)CC1 ZINC000217979134 EG For-Sale Unstable FAAH 32 52 O=C(N/C=C/c1cccc(F)c1)N1CCN(Cc2ccccc2)CC1 ZINC000217979134 EG For-Sale Unstable MGLL 0 40 N#Cc1cnc2ccc(N)cc2c1Nc1cccnc1 ZINC000217979154 CF For-Sale Unstable EGFR 30 55 N#Cc1cnc2ccc(N)cc2c1Nc1cccnc1 ZINC000217979154 CF For-Sale Unstable ERBB2 17 41 N#Cc1cnc2ccc(N)cc2c1Nc1cccnc1 ZINC000217979154 CF For-Sale Unstable SRC 64 44 N#Cc1cnc2ccc(N)cc2c1Nc1cccnc1 ZINC000217979154 CF For-Sale Unstable MAP2K1 54 50 N#Cc1cnc2ccc(N)cc2c1Nc1cccnc1 ZINC000217979154 CF For-Sale Unstable MAP3K8 57 48 O=C(N[C@@H](CN1C(=O)COC1=O)c1ccccc1)c1ccco1 ZINC000217979161 DD In-Stock Unstable SOAT1 24 40 COC(=O)C[C@H](C1=C(O)C(=O)C([C@H](CC(=O)OC)c2ccccc2)=C(O)C1=O)c1ccccc1 ZINC000217979171 JG In-Stock Unstable KCNA5 42 48 COC(=O)[C@H]1C[C@H](NC(=O)c2ccc(Cl)cc2)CN1 ZINC000217979177 CC On-Demand Unstable SLC6A1 15 40 NC[C@H](c1cccc(Cl)c1)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217979192 CH For-Sale Unstable OPRL1 0 43 Cc1ccc(SCC(=O)N(C)Cc2nc(-c3cccc(C)c3)no2)cc1 ZINC000217979201 FI In-Stock Unstable GRM5 15 41 COC(=O)C[C@H](C1=C(O)C(=O)C([C@@H](CC(=O)OC)c2ccccc2)=C(O)C1=O)c1ccccc1 ZINC000217979246 JG In-Stock Unstable KCNA5 42 48 O=C(N[C@H](CN1C(=O)COC1=O)c1ccccc1)c1ccccn1 ZINC000217979275 ED In-Stock Unstable TACR3 41 33 O=C(N[C@H](CN1C(=O)COC1=O)c1ccccc1)c1ccccn1 ZINC000217979275 ED In-Stock Unstable GRM4 40 37 NC[C@@H](c1cccc(Cl)c1)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217979281 CH For-Sale Unstable OPRL1 0 43 Clc1ccc(Br)c(OCCBr)c1 ZINC000217979282 DH For-Sale Unstable S1PR4 29 43 COc1cccc(-c2noc(CN(C)C(=O)CSc3ccc(C)cc3)n2)c1 ZINC000217979311 GH In-Stock Unstable HSD17B2 21 41 O=C(N[C@@H](CN1C(=O)COC1=O)c1ccccc1)c1ccccn1 ZINC000217979355 ED In-Stock Unstable TACR3 41 33 O=C(N[C@@H](CN1C(=O)COC1=O)c1ccccc1)c1ccccn1 ZINC000217979355 ED In-Stock Unstable GRM4 40 37 COc1cccc([C@@H](CN)N2CCC[C@@H]3CCCC[C@H]32)c1 ZINC000217979385 CG For-Sale Unstable CHRNA10 31 41 CCCOc1cc(/C=C2/CC(=O)NC2=O)ccc1OC ZINC000217979399 CD For-Sale Unstable ESRRA 49 38 CCCOc1cc(/C=C2/CC(=O)NC2=O)ccc1OC ZINC000217979399 CD For-Sale Unstable HPGD 54 45 O=C(N/C=C/c1cccc(F)c1)NC1CCCCCCCCCCC1 ZINC000217979436 EK For-Sale Unstable FAAH 0 47 O=C(N/C=C/c1cccc(F)c1)NC1CCCCCCCCCCC1 ZINC000217979436 EK For-Sale Unstable EPHX2 27 43 COc1cccc([C@H](CN)N2CCC[C@@H]3CCCC[C@H]32)c1 ZINC000217979460 CG For-Sale Unstable CHRNA10 31 41 Cc1ccc(SCC(=O)N(C)Cc2nc(-c3ccccc3Cl)no2)cc1 ZINC000217979516 GI In-Stock Unstable GPBAR1 24 42 O=C(N/C=C/c1cccc(F)c1)NCCN1CCOCC1 ZINC000217979544 CD For-Sale Unstable DRD4 40 31 O=C(N/C=C/c1cccc(F)c1)NCCN1CCOCC1 ZINC000217979544 CD For-Sale Unstable CASR 41 36 O=C(N/C=C/c1cccc(F)c1)NCCN1CCOCC1 ZINC000217979544 CD For-Sale Unstable EPHX2 26 47 O=C(N/C=C/c1cccc(F)c1)NCCN1CCOCC1 ZINC000217979544 CD For-Sale Unstable PLD2 58 36 COc1cc([C@@H]2CC(=O)Oc3cc(OC)c(OC)c(OC)c32)ccc1O ZINC000217979623 FF In-Stock Unstable CAN2 0 43 COc1cc([C@@H]2CC(=O)Oc3cc(OC)c(OC)c(OC)c32)ccc1O ZINC000217979623 FF In-Stock Unstable TAS2R31 0 43 O=C(N[C@H](CN1C(=O)COC1=O)c1ccccc1)c1ccccc1F ZINC000217979625 EE In-Stock Unstable CTSA 38 40 COc1cc([C@H]2CC(=O)Oc3cc(OC)c(OC)c(OC)c32)ccc1O ZINC000217979697 FF In-Stock Unstable CAN2 0 43 COc1cc([C@H]2CC(=O)Oc3cc(OC)c(OC)c(OC)c32)ccc1O ZINC000217979697 FF In-Stock Unstable TAS2R31 0 43 O=C(N[C@@H](CN1C(=O)COC1=O)c1ccccc1)c1ccccc1F ZINC000217979717 EE In-Stock Unstable CTSA 38 40 COC(=O)c1ccc(CSc2ccc(N)cc2Cl)cc1F ZINC000217979727 EI On-Demand Unstable PTPRG 0 42 O=C(N/C=C/c1cccc(F)c1)NCCN1CCNCC1 ZINC000217979832 CD For-Sale Unstable PLD2 63 36 Clc1cccc(-n2cnc3ccccc32)c1CBr ZINC000217979923 DJ For-Sale Unstable PDGFRB 0 45 COc1cc(CNC(=O)CSc2ccc(Cl)cc2)ccc1OC(C)C ZINC000217979955 GJ In-Stock Unstable TRPV1 23 40 COc1cc(CNC(=O)CSc2ccc(Cl)cc2)ccc1OC(C)C ZINC000217979955 GJ In-Stock Unstable U38 0 41 COc1cc(CNC(=O)CSc2ccc(Cl)cc2)ccc1OC(C)C ZINC000217979955 GJ In-Stock Unstable ENPP1 70 37 Cc1cc(CBr)cnc1-n1cnc2ccccc21 ZINC000217980034 DH For-Sale Unstable PDGFRB 0 43 O=C(CSc1ccc(Cl)cc1)NCCCc1ccccc1Cl ZINC000217980071 FJ In-Stock Unstable SCN10A 23 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccccc1 ZINC000217980095 GE For-Sale Unstable MMP13 55 43 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccccc1 ZINC000217980095 GE For-Sale Unstable MMP2 28 67 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccccc1 ZINC000217980095 GE For-Sale Unstable MMP3 68 43 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccccc1 ZINC000217980095 GE For-Sale Unstable MMP9 32 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccccc1 ZINC000217980095 GE For-Sale Unstable MMP7 63 39 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccccc1 ZINC000217980095 GE For-Sale Unstable MMP1 58 43 C[C@@H](N[C@H]1CCOc2ccccc21)[C@@H]1CCCN(C)C1 ZINC000217980154 CF For-Sale Unstable XIAP 19 42 C[C@@H](N[C@H]1CCOc2ccccc21)[C@@H]1CCCN(C)C1 ZINC000217980154 CF For-Sale Unstable BIRC3 36 42 C[C@@H](N[C@H]1CCOc2ccccc21)[C@@H]1CCCN(C)C1 ZINC000217980154 CF For-Sale Unstable BIRC2 21 42 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccccc1 ZINC000217980165 GE For-Sale Unstable MMP13 55 43 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccccc1 ZINC000217980165 GE For-Sale Unstable MMP2 28 67 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccccc1 ZINC000217980165 GE For-Sale Unstable MMP3 68 43 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccccc1 ZINC000217980165 GE For-Sale Unstable MMP9 32 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccccc1 ZINC000217980165 GE For-Sale Unstable MMP7 63 39 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccccc1 ZINC000217980165 GE For-Sale Unstable MMP1 58 43 O=C(N/C=C/c1cccc(F)c1)NCCCN1CCOCC1 ZINC000217980166 DD For-Sale Unstable HTR2A 19 41 O=C(N/C=C/c1cccc(F)c1)NCCCN1CCOCC1 ZINC000217980166 DD For-Sale Unstable CASR 40 35 O=C(N/C=C/c1cccc(F)c1)NCCCN1CCOCC1 ZINC000217980166 DD For-Sale Unstable TACR2 27 45 O=C(N/C=C/c1cccc(F)c1)NCCCN1CCOCC1 ZINC000217980166 DD For-Sale Unstable CCR3 35 41 O=C(N/C=C/c1cccc(F)c1)NCCCN1CCOCC1 ZINC000217980166 DD For-Sale Unstable EPHX2 25 45 O=C(N/C=C/c1cccc(F)c1)NCCCN1CCOCC1 ZINC000217980166 DD For-Sale Unstable ACKR3 18 41 COC(=O)C[C@H](c1cnn(C)c1)c1c(O)c2ccccc2oc1=O ZINC000217980177 ED In-Stock Unstable NQO1 45 48 O=C(CSc1ccc(Cl)cc1)NCCCc1ccc(Cl)cc1 ZINC000217980184 FJ In-Stock Unstable CRTM 31 41 CC(C)Cc1ccc(/C=C\C(=O)CCl)cc1 ZINC000217980221 BH For-Sale Unstable SLC22A20 0 44 C[C@H](N[C@H]1CCOc2ccccc21)[C@@H]1CCCN(C)C1 ZINC000217980227 CF For-Sale Unstable XIAP 19 42 C[C@H](N[C@H]1CCOc2ccccc21)[C@@H]1CCCN(C)C1 ZINC000217980227 CF For-Sale Unstable BIRC3 36 42 C[C@H](N[C@H]1CCOc2ccccc21)[C@@H]1CCCN(C)C1 ZINC000217980227 CF For-Sale Unstable BIRC2 21 42 N[C@]1(C(=O)O)C[C@@H]1S(=O)(=O)c1ccccc1 ZINC000217980230 BC In-Stock Unstable GRM3 43 36 COC(=O)C[C@@H](c1cnn(C)c1)c1c(O)c2ccccc2oc1=O ZINC000217980247 ED In-Stock Unstable NQO1 45 48 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccccc1 ZINC000217980249 GE For-Sale Unstable MMP13 55 43 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccccc1 ZINC000217980249 GE For-Sale Unstable MMP2 28 67 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccccc1 ZINC000217980249 GE For-Sale Unstable MMP3 68 43 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccccc1 ZINC000217980249 GE For-Sale Unstable MMP9 32 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccccc1 ZINC000217980249 GE For-Sale Unstable MMP7 63 39 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccccc1 ZINC000217980249 GE For-Sale Unstable MMP1 58 43 O=[N+]([O-])c1cc(Cl)ccc1OCc1cnn(-c2ccccc2)c1 ZINC000217980256 EI On-Demand Unstable PTGER1 54 39 CCN(C(=O)N/C=C/c1cccc(F)c1)c1ccccc1 ZINC000217980264 CI For-Sale Unstable NR1H4 26 42 N[C@@]1(C(=O)O)C[C@@H]1S(=O)(=O)c1ccccc1 ZINC000217980293 BC In-Stock Unstable GRM3 43 36 O=C(N[C@H](CN1C(=O)COC1=O)c1ccccc1)c1ccc(Cl)s1 ZINC000217980321 FF In-Stock Unstable F10 24 41 COc1ccc2c(c1OC)C(=O)N1[C@@H](C(=O)Nc3ccc(NC(C)=O)cc3)CS[C@H]21 ZINC000217980344 IF In-Stock Unstable TSHR 61 33 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccccc1 ZINC000217980346 GE For-Sale Unstable MMP13 55 43 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccccc1 ZINC000217980346 GE For-Sale Unstable MMP2 28 67 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccccc1 ZINC000217980346 GE For-Sale Unstable MMP3 68 43 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccccc1 ZINC000217980346 GE For-Sale Unstable MMP9 32 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccccc1 ZINC000217980346 GE For-Sale Unstable MMP7 63 39 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccccc1 ZINC000217980346 GE For-Sale Unstable MMP1 58 43 CN(Cc1ccccc1)C(=O)N/C=C/c1cccc(F)c1 ZINC000217980367 CH For-Sale Unstable NR1H4 26 42 CN(Cc1ccccc1)C(=O)N/C=C/c1cccc(F)c1 ZINC000217980367 CH For-Sale Unstable LIMK2 30 47 N[C@]1(C(=O)O)C[C@H]1S(=O)(=O)c1ccccc1 ZINC000217980369 BC In-Stock Unstable GRM3 43 36 O=C(/C=C\c1ccc(I)cc1)CCl ZINC000217980385 DG For-Sale Unstable SSSIM 16 50 COc1ccccc1CCCNC(=O)CSc1ccc(Cl)cc1 ZINC000217980393 EI In-Stock Unstable DRD2 23 44 COc1ccccc1CCCNC(=O)CSc1ccc(Cl)cc1 ZINC000217980393 EI In-Stock Unstable DRD3 32 44 COc1ccccc1CCCNC(=O)CSc1ccc(Cl)cc1 ZINC000217980393 EI In-Stock Unstable FAS 68 38 O=C(N[C@@H](CN1C(=O)COC1=O)c1ccccc1)c1ccc(Cl)s1 ZINC000217980405 FF In-Stock Unstable F10 24 41 COc1ccc2c(c1OC)C(=O)N1[C@@H](C(=O)Nc3ccc(NC(C)=O)cc3)CS[C@@H]21 ZINC000217980418 IF In-Stock Unstable TSHR 61 33 N[C@@]1(C(=O)O)C[C@H]1S(=O)(=O)c1ccccc1 ZINC000217980437 BC In-Stock Unstable GRM3 43 36 Clc1cc(CBr)ccc1-n1cnc2ccccc21 ZINC000217980455 DJ For-Sale Unstable PDGFRB 0 44 Clc1cc(CBr)ccc1-n1cnc2ccccc21 ZINC000217980455 DJ For-Sale Unstable PLK1 19 41 O=C(N[C@@H]1CCC[C@@H]1CO)c1ccc(F)c(Br)c1 ZINC000217980476 DE For-Sale Unstable SSTR3 28 45 O=C(/C=C\c1ccc(F)c(F)c1)CCl ZINC000217980488 BF For-Sale Unstable NFE2L2 0 41 COc1cccc(CCCNC(=O)CSc2ccc(Cl)cc2)c1 ZINC000217980496 EI In-Stock Unstable DRD4 48 40 COc1cccc(CCCNC(=O)CSc2ccc(Cl)cc2)c1 ZINC000217980496 EI In-Stock Unstable PTGS1 0 41 COc1cccc(CCCNC(=O)CSc2ccc(Cl)cc2)c1 ZINC000217980496 EI In-Stock Unstable HRH2 24 41 COc1cccc(CCCNC(=O)CSc2ccc(Cl)cc2)c1 ZINC000217980496 EI In-Stock Unstable PTGS2 32 43 COc1cccc(CCCNC(=O)CSc2ccc(Cl)cc2)c1 ZINC000217980496 EI In-Stock Unstable MTNR1B 60 60 COc1cccc(CCCNC(=O)CSc2ccc(Cl)cc2)c1 ZINC000217980496 EI In-Stock Unstable CRTM 75 54 COc1cccc(CCCNC(=O)CSc2ccc(Cl)cc2)c1 ZINC000217980496 EI In-Stock Unstable CAN2 0 51 COc1cccc(CCCNC(=O)CSc2ccc(Cl)cc2)c1 ZINC000217980496 EI In-Stock Unstable PDS 41 36 COc1cccc(CCCNC(=O)CSc2ccc(Cl)cc2)c1 ZINC000217980496 EI In-Stock Unstable FAS 60 41 COc1ccc2c(c1OC)C(=O)N1[C@H](C(=O)Nc3ccc(NC(C)=O)cc3)CS[C@H]21 ZINC000217980504 IF In-Stock Unstable TSHR 61 33 O=C(N[C@H]1CCC[C@@H]1CO)c1ccc(F)c(Br)c1 ZINC000217980533 DE For-Sale Unstable SSTR3 28 45 Clc1ccc(CBr)c(-n2cnc3ccccc32)c1 ZINC000217980557 DJ For-Sale Unstable PDGFRB 0 48 Clc1ccc(CBr)c(-n2cnc3ccccc32)c1 ZINC000217980557 DJ For-Sale Unstable PLK1 19 41 COc1ccc(CCCNC(=O)CSc2ccc(Cl)cc2)cc1 ZINC000217980562 EI In-Stock Unstable PTGS1 0 41 COc1ccc(CCCNC(=O)CSc2ccc(Cl)cc2)cc1 ZINC000217980562 EI In-Stock Unstable PTGS2 34 41 COc1ccc(CCCNC(=O)CSc2ccc(Cl)cc2)cc1 ZINC000217980562 EI In-Stock Unstable SCNN1A 50 42 COc1ccc(CCCNC(=O)CSc2ccc(Cl)cc2)cc1 ZINC000217980562 EI In-Stock Unstable MTNR1B 41 41 COc1ccc(CCCNC(=O)CSc2ccc(Cl)cc2)cc1 ZINC000217980562 EI In-Stock Unstable U38 0 42 COc1ccc(CCCNC(=O)CSc2ccc(Cl)cc2)cc1 ZINC000217980562 EI In-Stock Unstable CRTM 36 43 COc1ccc(CCCNC(=O)CSc2ccc(Cl)cc2)cc1 ZINC000217980562 EI In-Stock Unstable PROKR1 41 33 COc1ccc(CCCNC(=O)CSc2ccc(Cl)cc2)cc1 ZINC000217980562 EI In-Stock Unstable FAS 53 44 COc1cc(Cl)c(/C=C\C(=O)CCl)cc1OC ZINC000217980569 CG For-Sale Unstable CYSP_PLAFA 53 40 COc1ccc2c(c1OC)C(=O)N1[C@H]2SC[C@H]1C(=O)Nc1ccc(NC(C)=O)cc1 ZINC000217980584 IF In-Stock Unstable TSHR 61 33 Cc1csc(NC(=O)N/C=C/c2cccc(F)c2)n1 ZINC000217980587 CG For-Sale Unstable GCK 16 50 CCn1nc2c(C(=O)O)cccn2c1=O ZINC000217980590 BC For-Sale Unstable POLR1A 55 33 O=C(N[C@@H]1CCC[C@H]1CO)c1ccc(F)c(Br)c1 ZINC000217980622 DE For-Sale Unstable SSTR3 28 45 Cn1nc2c(C(=O)O)cccn2c1=O ZINC000217980679 AB For-Sale Unstable POLR1A 63 33 COc1ccc(OC[C@@H](C)NC(=O)CSc2ccc(Cl)cc2)cc1 ZINC000217980680 FI In-Stock Unstable PTGS1 0 48 COc1ccc(OC[C@@H](C)NC(=O)CSc2ccc(Cl)cc2)cc1 ZINC000217980680 FI In-Stock Unstable PTGS2 33 48 COc1ccc(OC[C@@H](C)NC(=O)CSc2ccc(Cl)cc2)cc1 ZINC000217980680 FI In-Stock Unstable FAS 43 44 Cc1cc(-n2cnc3ccccc32)ccc1CBr ZINC000217980683 DI For-Sale Unstable PDGFRB 28 51 Cc1cc(-n2cnc3ccccc32)ccc1CBr ZINC000217980683 DI For-Sale Unstable PLK1 19 41 COc1ccc2c(c1)C[C@@H]2CC(=O)O ZINC000217980695 AD For-Sale Unstable PPARG 36 51 COc1ccc2c(c1)C[C@@H]2CC(=O)O ZINC000217980695 AD For-Sale Unstable PPARA 26 49 COc1ccc2c(c1)C[C@@H]2CC(=O)O ZINC000217980695 AD For-Sale Unstable NQO2 41 43 COc1ccc2c(c1)C[C@@H]2CC(=O)O ZINC000217980695 AD For-Sale Unstable MTR1B_CHICK 0 51 COc1ccc2c(c1)C[C@@H]2CC(=O)O ZINC000217980695 AD For-Sale Unstable PPARD 66 61 COc1ccc2c(c1)C[C@@H]2CC(=O)O ZINC000217980695 AD For-Sale Unstable MTNR1A 61 45 COc1ccc2c(c1)C[C@@H]2CC(=O)O ZINC000217980695 AD For-Sale Unstable MTNR1B 58 43 COc1ccc2c(c1)C[C@@H]2CC(=O)O ZINC000217980695 AD For-Sale Unstable EBP 17 41 COc1ccc2c(c1)C[C@@H]2CC(=O)O ZINC000217980695 AD For-Sale Unstable AADAT 47 40 COc1ccc2c(c1)C[C@@H]2CC(=O)O ZINC000217980695 AD For-Sale Unstable FFAR1 58 56 COc1ccc2c(c1)C[C@@H]2CC(=O)O ZINC000217980695 AD For-Sale Unstable AKR1C2 41 33 COc1ccc2c(c1)C[C@@H]2CC(=O)O ZINC000217980695 AD For-Sale Unstable CYP27A1 0 40 COc1ccc2c(c1)C[C@@H]2CC(=O)O ZINC000217980695 AD For-Sale Unstable CCBL2 0 40 O=C(N[C@H](CN1C(=O)COC1=O)c1ccccc1)c1ccc(F)cc1Cl ZINC000217980703 GF In-Stock Unstable CTSA 41 35 O=C(N[C@H]1CCC[C@H]1CO)c1ccc(F)c(Br)c1 ZINC000217980712 DE On-Demand Unstable SSTR3 26 43 COc1ccc(OC[C@H](C)NC(=O)CSc2ccc(Cl)cc2)cc1 ZINC000217980768 FI In-Stock Unstable PTGS1 0 48 COc1ccc(OC[C@H](C)NC(=O)CSc2ccc(Cl)cc2)cc1 ZINC000217980768 FI In-Stock Unstable PTGS2 33 48 COc1ccc(OC[C@H](C)NC(=O)CSc2ccc(Cl)cc2)cc1 ZINC000217980768 FI In-Stock Unstable FAS 43 44 COc1ccc2c(c1)C[C@H]2CC(=O)O ZINC000217980786 AD For-Sale Unstable PPARG 36 51 COc1ccc2c(c1)C[C@H]2CC(=O)O ZINC000217980786 AD For-Sale Unstable PPARA 26 49 COc1ccc2c(c1)C[C@H]2CC(=O)O ZINC000217980786 AD For-Sale Unstable NQO2 41 43 COc1ccc2c(c1)C[C@H]2CC(=O)O ZINC000217980786 AD For-Sale Unstable MTR1B_CHICK 0 51 COc1ccc2c(c1)C[C@H]2CC(=O)O ZINC000217980786 AD For-Sale Unstable PPARD 66 61 COc1ccc2c(c1)C[C@H]2CC(=O)O ZINC000217980786 AD For-Sale Unstable MTNR1A 61 45 COc1ccc2c(c1)C[C@H]2CC(=O)O ZINC000217980786 AD For-Sale Unstable MTNR1B 58 43 COc1ccc2c(c1)C[C@H]2CC(=O)O ZINC000217980786 AD For-Sale Unstable EBP 17 41 COc1ccc2c(c1)C[C@H]2CC(=O)O ZINC000217980786 AD For-Sale Unstable AADAT 47 40 COc1ccc2c(c1)C[C@H]2CC(=O)O ZINC000217980786 AD For-Sale Unstable FFAR1 58 56 COc1ccc2c(c1)C[C@H]2CC(=O)O ZINC000217980786 AD For-Sale Unstable AKR1C2 41 33 COc1ccc2c(c1)C[C@H]2CC(=O)O ZINC000217980786 AD For-Sale Unstable CYP27A1 0 40 COc1ccc2c(c1)C[C@H]2CC(=O)O ZINC000217980786 AD For-Sale Unstable CCBL2 0 40 O=C(N[C@@H](CN1C(=O)COC1=O)c1ccccc1)c1ccc(F)cc1Cl ZINC000217980791 GF In-Stock Unstable CTSA 41 35 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1cccc(C)c1 ZINC000217980796 GF For-Sale Unstable ADAM17 16 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1cccc(C)c1 ZINC000217980796 GF For-Sale Unstable MMP2 15 56 COc1cccc(NC(=O)N/C=C/c2cccc(F)c2)c1 ZINC000217980801 CH For-Sale Unstable CCR3 22 41 COc1cccc(NC(=O)N/C=C/c2cccc(F)c2)c1 ZINC000217980801 CH For-Sale Unstable MTNR1A 26 49 COc1cccc(NC(=O)N/C=C/c2cccc(F)c2)c1 ZINC000217980801 CH For-Sale Unstable MTNR1B 31 49 COc1cccc(NC(=O)N/C=C/c2cccc(F)c2)c1 ZINC000217980801 CH For-Sale Unstable TAAR1 35 47 COc1cccc(NC(=O)N/C=C/c2cccc(F)c2)c1 ZINC000217980801 CH For-Sale Unstable KCNK3 41 36 CC(C)Oc1cccc(CCCNC(=O)CSc2ccc(Cl)cc2)c1 ZINC000217980873 GJ In-Stock Unstable MTNR1A 27 50 CC(C)Oc1cccc(CCCNC(=O)CSc2ccc(Cl)cc2)c1 ZINC000217980873 GJ In-Stock Unstable MTNR1B 26 50 CC(C)Oc1cccc(CCCNC(=O)CSc2ccc(Cl)cc2)c1 ZINC000217980873 GJ In-Stock Unstable CRTM 73 52 CC(C)Oc1cccc(CCCNC(=O)CSc2ccc(Cl)cc2)c1 ZINC000217980873 GJ In-Stock Unstable CAN2 0 40 CC(C)Oc1cccc(CCCNC(=O)CSc2ccc(Cl)cc2)c1 ZINC000217980873 GJ In-Stock Unstable PDS 57 37 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1cccc(C)c1 ZINC000217980883 GF For-Sale Unstable ADAM17 16 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1cccc(C)c1 ZINC000217980883 GF For-Sale Unstable MMP2 15 56 O=C(N[C@H](CN1C(=O)COC1=O)c1ccccc1)c1ccc(C(F)(F)F)cc1 ZINC000217980901 GG In-Stock Unstable MTTP 70 42 O=C(N/C=C/c1cccc(F)c1)Nc1cc(Cl)ccc1O ZINC000217980908 DH For-Sale Anodyne KCNMA1 20 44 O=C(N/C=C/c1cccc(F)c1)Nc1cc(Cl)ccc1O ZINC000217980908 DH For-Sale Anodyne MMP1 15 41 Clc1ccc(-n2cnc3ccccc32)c(CBr)c1 ZINC000217980909 DJ For-Sale Unstable PDGFRB 0 48 Clc1ccc(-n2cnc3ccccc32)c(CBr)c1 ZINC000217980909 DJ For-Sale Unstable PLK1 19 41 O=C(N[C@@H](CN1C(=O)COC1=O)c1ccccc1)c1ccc(C(F)(F)F)cc1 ZINC000217980969 GG In-Stock Unstable MTTP 66 42 CC(C)Oc1ccc(CCCNC(=O)CSc2ccc(Cl)cc2)cc1 ZINC000217980994 GJ In-Stock Unstable CRTM 35 41 ClCc1c(Cl)ncnc1-n1cnc2ccccc21 ZINC000217981017 CG For-Sale Unstable PDGFRB 0 45 Cc1noc(NC(=O)c2cn(-c3ccccc3)nc2-c2cccs2)c1C ZINC000217981020 FI On-Demand Unstable EDNRA 22 44 Cc1noc(NC(=O)c2cn(-c3ccccc3)nc2-c2cccs2)c1C ZINC000217981020 FI On-Demand Unstable CDK2 17 45 Cc1noc(NC(=O)c2cn(-c3ccccc3)nc2-c2cccs2)c1C ZINC000217981020 FI On-Demand Unstable GPR142 48 31 O=C(CSc1ccc(Cl)cc1)Nc1ccc(OC2CCCC2)cc1 ZINC000217981106 FK In-Stock Unstable EPHX2 22 48 O=C(CSc1ccc(Cl)cc1)Nc1ccc(OC2CCCC2)cc1 ZINC000217981106 FK In-Stock Unstable FAS 48 39 O=C(N/C=C/c1cccc(F)c1)Nc1nccs1 ZINC000217981151 CG For-Sale Anodyne MAP 0 47 O=C(N/C=C/c1cccc(F)c1)Nc1nccs1 ZINC000217981151 CG For-Sale Anodyne MAP1 106 41 CC1(C)C[C@@H](NC(=O)CSc2ccc(Cl)cc2)c2ccccc2O1 ZINC000217981205 FJ In-Stock Unstable FAS 51 37 BrCc1ccc(-n2cnc3ccccc32)nc1 ZINC000217981222 CG For-Sale Unstable PDGFRB 0 47 CC(C)(C)OC(=O)N1CCc2cc(CC#N)ccc21 ZINC000217981224 CG For-Sale Unstable GPR119 22 47 CC1(C)C[C@H](NC(=O)CSc2ccc(Cl)cc2)c2ccccc2O1 ZINC000217981275 FJ In-Stock Unstable FAS 51 37 BrCc1cnc(-n2cnc3ccccc32)nc1 ZINC000217981328 CF For-Sale Unstable PDGFRB 0 50 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)cc1 ZINC000217981343 GE For-Sale Unstable MMP13 61 42 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)cc1 ZINC000217981343 GE For-Sale Unstable ADAM17 38 41 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)cc1 ZINC000217981343 GE For-Sale Unstable MMP2 31 59 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)cc1 ZINC000217981343 GE For-Sale Unstable MMP3 73 42 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)cc1 ZINC000217981343 GE For-Sale Unstable MMP8 34 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)cc1 ZINC000217981343 GE For-Sale Unstable MMP9 34 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)cc1 ZINC000217981343 GE For-Sale Unstable MMP7 69 42 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)cc1 ZINC000217981343 GE For-Sale Unstable MMP1 64 45 O=C(N/C=C/c1cccc(F)c1)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000217981360 IG For-Sale Unstable PKM 33 42 CCOc1ccc(CCCNC(=O)CSc2ccc(Cl)cc2)cc1 ZINC000217981391 FJ In-Stock Unstable SCN2A 17 41 CCOc1ccc(CCCNC(=O)CSc2ccc(Cl)cc2)cc1 ZINC000217981391 FJ In-Stock Unstable CRTM 35 41 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)cc1 ZINC000217981414 GE For-Sale Unstable MMP13 61 42 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)cc1 ZINC000217981414 GE For-Sale Unstable ADAM17 38 41 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)cc1 ZINC000217981414 GE For-Sale Unstable MMP2 31 59 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)cc1 ZINC000217981414 GE For-Sale Unstable MMP3 73 42 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)cc1 ZINC000217981414 GE For-Sale Unstable MMP8 34 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)cc1 ZINC000217981414 GE For-Sale Unstable MMP9 34 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)cc1 ZINC000217981414 GE For-Sale Unstable MMP7 69 42 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)cc1 ZINC000217981414 GE For-Sale Unstable MMP1 64 45 BrCc1ccc(Br)cc1-n1cnc2ccccc21 ZINC000217981449 FJ For-Sale Unstable PDGFRB 0 45 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217981470 ED For-Sale Unstable CA2 100 52 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217981470 ED For-Sale Unstable CA1 83 52 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217981470 ED For-Sale Unstable CA7 47 46 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217981470 ED For-Sale Unstable CA5B 55 46 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217981470 ED For-Sale Unstable CA4 76 52 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217981470 ED For-Sale Unstable CA5A 58 46 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217981470 ED For-Sale Unstable CA14 37 47 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217981470 ED For-Sale Unstable CA12 63 51 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217981470 ED For-Sale Unstable ALPL 15 50 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217981470 ED For-Sale Unstable CA9 71 51 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217981470 ED For-Sale Unstable CYNT 23 41 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217981470 ED For-Sale Unstable MTCA1 45 47 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217981470 ED For-Sale Unstable P96878_MYCTU 56 47 NS(=O)(=O)c1ccc(CNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217981470 ED For-Sale Unstable NAMPT 35 40 CCCOc1ccccc1CCCNC(=O)CSc1ccc(Cl)cc1 ZINC000217981478 GJ In-Stock Unstable MTNR1A 38 44 CCCOc1ccccc1CCCNC(=O)CSc1ccc(Cl)cc1 ZINC000217981478 GJ In-Stock Unstable MTNR1B 37 44 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)cc1 ZINC000217981499 GE For-Sale Unstable MMP13 61 42 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)cc1 ZINC000217981499 GE For-Sale Unstable ADAM17 38 41 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)cc1 ZINC000217981499 GE For-Sale Unstable MMP2 31 59 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)cc1 ZINC000217981499 GE For-Sale Unstable MMP3 73 42 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)cc1 ZINC000217981499 GE For-Sale Unstable MMP8 34 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)cc1 ZINC000217981499 GE For-Sale Unstable MMP9 34 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)cc1 ZINC000217981499 GE For-Sale Unstable MMP7 69 42 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)cc1 ZINC000217981499 GE For-Sale Unstable MMP1 64 45 O=C1N[C@H]2CCC[C@@H]1CN(C(=O)c1cc(Cl)ccc1F)C2 ZINC000217981546 DE In-Stock Unstable PARP1 46 35 BrCc1ccccc1-n1cnc2ccccc21 ZINC000217981569 CH For-Sale Unstable PDGFRB 21 51 BrCc1ccccc1-n1cnc2ccccc21 ZINC000217981569 CH For-Sale Unstable PLK1 20 40 O=C(N/C=C/c1cccc(F)c1)Nc1cccnc1Cl ZINC000217981574 CH For-Sale Anodyne G2YM83_BOTF4 59 33 Cc1ccccc1OC[C@@H](C)NC(=O)CSc1ccc(Cl)cc1 ZINC000217981577 EI In-Stock Unstable SDH1 0 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)cc1 ZINC000217981586 GE For-Sale Unstable MMP13 61 42 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)cc1 ZINC000217981586 GE For-Sale Unstable ADAM17 38 41 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)cc1 ZINC000217981586 GE For-Sale Unstable MMP2 31 59 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)cc1 ZINC000217981586 GE For-Sale Unstable MMP3 73 42 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)cc1 ZINC000217981586 GE For-Sale Unstable MMP8 34 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)cc1 ZINC000217981586 GE For-Sale Unstable MMP9 34 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)cc1 ZINC000217981586 GE For-Sale Unstable MMP7 69 42 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)cc1 ZINC000217981586 GE For-Sale Unstable MMP1 64 45 CC(C)c1ccc(N2C(=O)N[C@@H](CC(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)C2=O)cc1 ZINC000217981632 IE In-Stock Unstable CHRNA4 27 43 Cc1ccccc1OC[C@H](C)NC(=O)CSc1ccc(Cl)cc1 ZINC000217981645 EI In-Stock Unstable SDH1 0 40 Cc1ccc(S(=O)(=O)N[C@@H](CN2C(=O)COC2=O)c2ccccc2)cc1C ZINC000217981659 GE In-Stock Unstable LEF 39 40 CCc1ncnc(NCc2ccc([N+](=O)[O-])cc2)c1F ZINC000217981672 CF On-Demand Unstable SLC29A1 33 41 CN(CC(=O)Nc1cc(Cl)ccc1F)S(=O)(=O)c1cccc([N+](=O)[O-])c1 ZINC000217981736 HF On-Demand Unstable CA1 18 40 CN(CC(=O)Nc1cc(Cl)ccc1F)S(=O)(=O)c1cccc([N+](=O)[O-])c1 ZINC000217981736 HF On-Demand Unstable COLA 31 40 CN(CC(=O)Nc1cc(Cl)ccc1F)S(=O)(=O)c1cccc([N+](=O)[O-])c1 ZINC000217981736 HF On-Demand Unstable CA4 22 42 CN(CC(=O)Nc1cc(Cl)ccc1F)S(=O)(=O)c1cccc([N+](=O)[O-])c1 ZINC000217981736 HF On-Demand Unstable MMP2 16 45 CN(CC(=O)Nc1cc(Cl)ccc1F)S(=O)(=O)c1cccc([N+](=O)[O-])c1 ZINC000217981736 HF On-Demand Unstable MMP8 33 45 CN(CC(=O)Nc1cc(Cl)ccc1F)S(=O)(=O)c1cccc([N+](=O)[O-])c1 ZINC000217981736 HF On-Demand Unstable MMP9 17 45 CN(CC(=O)Nc1cc(Cl)ccc1F)S(=O)(=O)c1cccc([N+](=O)[O-])c1 ZINC000217981736 HF On-Demand Unstable MMP1 27 45 Cc1ccc(S(=O)(=O)N[C@H](CN2C(=O)COC2=O)c2ccccc2)cc1C ZINC000217981743 GE In-Stock Unstable LEF 39 40 Cc1cc(CBr)ccc1-n1cnc2ccccc21 ZINC000217981773 DI For-Sale Unstable PDGFRB 22 44 Cc1cc(CBr)ccc1-n1cnc2ccccc21 ZINC000217981773 DI For-Sale Unstable PLK1 19 41 CN(CC(=O)NCCc1cccc(Cl)c1)S(=O)(=O)c1cccc([N+](=O)[O-])c1 ZINC000217981844 HE On-Demand Unstable MMP2 15 46 CN(CC(=O)NCCc1cccc(Cl)c1)S(=O)(=O)c1cccc([N+](=O)[O-])c1 ZINC000217981844 HE On-Demand Unstable MMP8 32 46 CN(CC(=O)NCCc1cccc(Cl)c1)S(=O)(=O)c1cccc([N+](=O)[O-])c1 ZINC000217981844 HE On-Demand Unstable MMP9 17 46 CN(CC(=O)NCCc1cccc(Cl)c1)S(=O)(=O)c1cccc([N+](=O)[O-])c1 ZINC000217981844 HE On-Demand Unstable MMP1 26 46 Fc1cc(CBr)ccc1-n1cnc2ccccc21 ZINC000217981873 DI For-Sale Unstable PDGFRB 0 44 C/C(=C1/CC(=O)NC1=O)c1ccc(S(C)(=O)=O)cc1 ZINC000217981882 CC For-Sale Unstable PTGS2 24 40 C/C(=C1/CC(=O)NC1=O)c1ccc(S(C)(=O)=O)cc1 ZINC000217981882 CC For-Sale Unstable LOX1.1 42 35 C/C(=C1/CC(=O)NC1=O)c1ccc(S(C)(=O)=O)cc1 ZINC000217981882 CC For-Sale Unstable O49150_SOLTU 49 33 CC1CCN(c2ccc([C@@H](C)NC(=O)CSc3ccc(Cl)cc3)cc2)CC1 ZINC000217981919 HK In-Stock Unstable SDH1 0 43 CC1CCN(c2ccc([C@@H](C)NC(=O)CSc3ccc(Cl)cc3)cc2)CC1 ZINC000217981919 HK In-Stock Unstable PRCP 22 46 Fc1ccc(-n2cnc3ccccc32)c(CBr)c1 ZINC000217981959 DI For-Sale Unstable PDGFRB 0 44 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1ccc(CC(N)=O)cc1 ZINC000217981998 CH For-Sale Unstable TRPM8 18 50 CC1CCN(c2ccc([C@H](C)NC(=O)CSc3ccc(Cl)cc3)cc2)CC1 ZINC000217982000 HK In-Stock Unstable SDH1 0 43 CC1CCN(c2ccc([C@H](C)NC(=O)CSc3ccc(Cl)cc3)cc2)CC1 ZINC000217982000 HK In-Stock Unstable PRCP 22 46 Cc1nn(C)c(-n2cnc3ccccc32)c1CBr ZINC000217982065 DF For-Sale Unstable PDGFRB 0 44 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1ccc(CC(N)=O)cc1 ZINC000217982071 CH For-Sale Unstable TRPM8 18 50 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)CSc3ccc(Cl)cc3)cc2)C1 ZINC000217982095 HK In-Stock Unstable SLC6A1 0 40 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)CSc3ccc(Cl)cc3)cc2)C1 ZINC000217982095 HK In-Stock Unstable SDH1 0 41 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)CSc3ccc(Cl)cc3)cc2)C1 ZINC000217982095 HK In-Stock Unstable PRCP 18 44 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)CSc3ccc(Cl)cc3)cc2)C1 ZINC000217982095 HK In-Stock Unstable ADAM17 0 40 COC(=O)c1cc(OC)c(Cl)cc1Br ZINC000217982133 CF For-Sale Unstable HTR4 48 38 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1ccc(CC(N)=O)cc1 ZINC000217982158 CH For-Sale Unstable TRPM8 18 50 C[C@H](NC(=O)CSc1ccc(Cl)cc1)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217982171 HK In-Stock Unstable SLC6A1 0 40 C[C@H](NC(=O)CSc1ccc(Cl)cc1)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217982171 HK In-Stock Unstable SDH1 0 41 C[C@H](NC(=O)CSc1ccc(Cl)cc1)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217982171 HK In-Stock Unstable PRCP 18 44 C[C@H](NC(=O)CSc1ccc(Cl)cc1)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217982171 HK In-Stock Unstable ADAM17 0 40 COc1cc(Br)ccc1C(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217982206 EE For-Sale Unstable DRD2 34 41 COc1cc(Br)ccc1C(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217982206 EE For-Sale Unstable DRD3 22 40 CCc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217982240 HF For-Sale Unstable FKBP1A 22 44 CCc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217982240 HF For-Sale Unstable MMP13 65 43 CCc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217982240 HF For-Sale Unstable ADAM17 47 42 CCc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217982240 HF For-Sale Unstable MMP2 33 43 CCc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217982240 HF For-Sale Unstable MMP3 78 43 CCc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217982240 HF For-Sale Unstable MMP9 36 41 CCc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217982240 HF For-Sale Unstable MMP7 75 40 CCc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217982240 HF For-Sale Unstable MMP1 71 43 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1ccc(CC(N)=O)cc1 ZINC000217982247 CH For-Sale Unstable TRPM8 18 50 Fc1cc(CBr)cc(F)c1-n1cnc2ccccc21 ZINC000217982278 DI For-Sale Unstable PDGFRB 23 46 Fc1cc(CBr)cc(F)c1-n1cnc2ccccc21 ZINC000217982278 DI For-Sale Unstable PLK1 19 40 COc1cc(Br)ccc1C(=O)N[C@H]1CCC[C@@H]1CO ZINC000217982282 EE For-Sale Unstable DRD2 34 41 COc1cc(Br)ccc1C(=O)N[C@H]1CCC[C@@H]1CO ZINC000217982282 EE For-Sale Unstable DRD3 22 40 COc1ccc(CCNC(=O)COc2c(C)occc2=O)cc1 ZINC000217982304 DD In-Stock Unstable NQO2 21 40 COc1ccc(CCNC(=O)COc2c(C)occc2=O)cc1 ZINC000217982304 DD In-Stock Unstable MTNR1A 61 41 COc1ccc(CCNC(=O)COc2c(C)occc2=O)cc1 ZINC000217982304 DD In-Stock Unstable MTNR1B 48 39 COc1ccc(CCNC(=O)COc2c(C)occc2=O)cc1 ZINC000217982304 DD In-Stock Unstable CA9 18 47 COc1ccc(CCNC(=O)COc2c(C)occc2=O)cc1 ZINC000217982304 DD In-Stock Unstable PROKR1 51 31 CCc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217982306 HF For-Sale Unstable FKBP1A 22 44 CCc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217982306 HF For-Sale Unstable MMP13 65 43 CCc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217982306 HF For-Sale Unstable ADAM17 47 42 CCc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217982306 HF For-Sale Unstable MMP2 33 43 CCc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217982306 HF For-Sale Unstable MMP3 78 43 CCc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217982306 HF For-Sale Unstable MMP9 36 41 CCc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217982306 HF For-Sale Unstable MMP7 75 40 CCc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217982306 HF For-Sale Unstable MMP1 71 43 NC[C@H](c1ccccc1Cl)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217982310 CH For-Sale Unstable OPRL1 29 42 CCN(C)C(=O)CNc1cc(OC)ccc1C#N ZINC000217982319 BD For-Sale Unstable AKR1C2 45 34 O=C(O)[C@@H]1C[C@@H]2CCCC[C@@H]2N1C(=O)NCC(F)(F)F ZINC000217982343 CD On-Demand Unstable ACE 15 60 COc1cc(Br)ccc1C(=O)N[C@@H]1CCC[C@H]1CO ZINC000217982370 EE For-Sale Unstable DRD2 34 41 COc1cc(Br)ccc1C(=O)N[C@@H]1CCC[C@H]1CO ZINC000217982370 EE For-Sale Unstable DRD3 22 40 BrCc1ccc(-n2cnc3ccccc32)cc1 ZINC000217982372 CH For-Sale Unstable PDGFRB 31 66 NC[C@@H](c1ccccc1Cl)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217982386 CH For-Sale Unstable OPRL1 29 42 O=C(O)c1cc(Br)c(Cl)cn1 ZINC000217982416 BE For-Sale Anodyne KMO 0 44 O=C(O)[C@@H]1C[C@H]2CCCC[C@@H]2N1C(=O)NCC(F)(F)F ZINC000217982423 CD On-Demand Unstable ACE 15 60 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)Nc3ccncc3)[C@H]21 ZINC000217982424 IF In-Stock Unstable TSHR 48 32 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C)c(C)c1 ZINC000217982435 HF For-Sale Unstable MMP2 17 52 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C)c(C)c1 ZINC000217982435 HF For-Sale Unstable MMP3 48 39 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C)c(C)c1 ZINC000217982435 HF For-Sale Unstable MMP7 45 35 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C)c(C)c1 ZINC000217982435 HF For-Sale Unstable MMP1 41 39 COc1cc(Br)ccc1C(=O)N[C@H]1CCC[C@H]1CO ZINC000217982444 EE For-Sale Unstable DRD2 34 41 COc1cc(Br)ccc1C(=O)N[C@H]1CCC[C@H]1CO ZINC000217982444 EE For-Sale Unstable DRD3 22 40 COc1ccc2c(c1OC)C(=O)N1c3ccccc3C(=O)N(CC(=O)Nc3ccncc3)[C@@H]21 ZINC000217982506 IF In-Stock Unstable TSHR 48 32 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C)c(C)c1 ZINC000217982510 HF For-Sale Unstable MMP2 17 52 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C)c(C)c1 ZINC000217982510 HF For-Sale Unstable MMP3 48 39 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C)c(C)c1 ZINC000217982510 HF For-Sale Unstable MMP7 45 35 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C)c(C)c1 ZINC000217982510 HF For-Sale Unstable MMP1 41 39 C[C@@](O)(CNC(=O)C1CC1)c1cc2ccccc2o1 ZINC000217982595 CE In-Stock Unstable VCP 42 36 COc1cccc2c1ccn2CCNC(=O)[C@@H](NC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)C(C)C ZINC000217982600 KF In-Stock Unstable CHRNA4 25 41 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C)cc1C ZINC000217982605 HF For-Sale Unstable EPHX2 15 45 CC(C)(C)OC(=O)N1CC[C@]2(CC(=O)c3cc(Cl)ccc3O2)C1 ZINC000217982619 EH For-Sale Unstable ACACA 46 36 CC(C)(C)OC(=O)N1CC[C@]2(CC(=O)c3cc(Cl)ccc3O2)C1 ZINC000217982619 EH For-Sale Unstable ACACB 39 48 COc1ccc2c(c1)[C@@H](NC(=O)CSc1ccc(Cl)cc1)CC(C)(C)O2 ZINC000217982629 GJ In-Stock Unstable FAS 51 39 Cc1ccc(S(=O)(=O)Nc2ccc(NC(=O)CCn3c(=O)n(C)c4ccccc43)cc2)cc1 ZINC000217982668 JG On-Demand Unstable CA2 20 46 Cc1ccc(S(=O)(=O)Nc2ccc(NC(=O)CCn3c(=O)n(C)c4ccccc43)cc2)cc1 ZINC000217982668 JG On-Demand Unstable CA1 21 46 Cc1ccc(S(=O)(=O)Nc2ccc(NC(=O)CCn3c(=O)n(C)c4ccccc43)cc2)cc1 ZINC000217982668 JG On-Demand Unstable CA4 19 45 Cc1ccc(S(=O)(=O)Nc2ccc(NC(=O)CCn3c(=O)n(C)c4ccccc43)cc2)cc1 ZINC000217982668 JG On-Demand Unstable CA9 15 46 Cc1ccc(S(=O)(=O)Nc2ccc(NC(=O)CCn3c(=O)n(C)c4ccccc43)cc2)cc1 ZINC000217982668 JG On-Demand Unstable CALCRL 28 43 Cc1ccc(S(=O)(=O)Nc2ccc(NC(=O)CCn3c(=O)n(C)c4ccccc43)cc2)cc1 ZINC000217982668 JG On-Demand Unstable LIMK2 44 34 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C)cc1C ZINC000217982676 HF For-Sale Unstable EPHX2 15 45 C[C@](O)(CNC(=O)C1CC1)c1cc2ccccc2o1 ZINC000217982682 CE In-Stock Unstable VCP 42 36 CC(C)(C)OC(=O)N1CC[C@@]2(CC(=O)c3cc(Cl)ccc3O2)C1 ZINC000217982705 EH For-Sale Unstable ACACA 46 36 CC(C)(C)OC(=O)N1CC[C@@]2(CC(=O)c3cc(Cl)ccc3O2)C1 ZINC000217982705 EH For-Sale Unstable ACACB 39 48 COc1ccc2c(c1)[C@H](NC(=O)CSc1ccc(Cl)cc1)CC(C)(C)O2 ZINC000217982708 GJ In-Stock Unstable FAS 51 39 CCc1ncnc(N2C[C@@H]3CNC[C@@H]3C2)c1F ZINC000217982710 BC On-Demand Unstable CHRNA4 29 40 CCc1ncnc(N2C[C@H]3CNC[C@@H]3C2)c1F ZINC000217982776 BC On-Demand Unstable CHRNA4 29 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)CCc1ccccc1 ZINC000217982779 HE For-Sale Unstable MMP13 18 42 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)CCc1ccccc1 ZINC000217982779 HE For-Sale Unstable MMP3 22 45 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)CCc1ccccc1 ZINC000217982779 HE For-Sale Unstable MMP1 17 40 COCC(=O)NC[C@@](C)(O)c1cc2ccccc2o1 ZINC000217982794 CD In-Stock Unstable KCNJ11 16 40 CCCCCNC(=O)N/C=C/c1cccc(F)c1 ZINC000217982802 CG For-Sale Unstable ASAH1 80 33 CCCCCNC(=O)N/C=C/c1cccc(F)c1 ZINC000217982802 CG For-Sale Unstable ACAT 0 50 COc1ccc2c(c1)OC(C)(C)C[C@@H]2NC(=O)CSc1ccc(Cl)cc1 ZINC000217982815 GJ In-Stock Unstable FAS 62 39 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)CCc1ccccc1 ZINC000217982842 HE For-Sale Unstable MMP13 18 42 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)CCc1ccccc1 ZINC000217982842 HE For-Sale Unstable MMP3 22 45 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)CCc1ccccc1 ZINC000217982842 HE For-Sale Unstable MMP1 17 40 CCc1ncnc(N2C[C@@H]3CNC[C@H]3C2)c1F ZINC000217982859 BC On-Demand Unstable CHRNA4 29 40 COCC(=O)NC[C@](C)(O)c1cc2ccccc2o1 ZINC000217982863 CD In-Stock Unstable KCNJ11 16 40 COc1ccc2c(c1)OC(C)(C)C[C@H]2NC(=O)CSc1ccc(Cl)cc1 ZINC000217982902 GJ In-Stock Unstable FAS 62 39 O=C(N/C=C/c1cccc(F)c1)Nc1ccccc1 ZINC000217982912 CH For-Sale Anodyne MMP1 0 55 O=C(N/C=C/c1cccc(F)c1)Nc1ccccc1 ZINC000217982912 CH For-Sale Anodyne KCNK3 39 44 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)CCc1ccccc1 ZINC000217982915 HE For-Sale Unstable MMP13 18 42 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)CCc1ccccc1 ZINC000217982915 HE For-Sale Unstable MMP3 22 45 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)CCc1ccccc1 ZINC000217982915 HE For-Sale Unstable MMP1 17 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)CCc1ccccc1 ZINC000217982990 HE For-Sale Unstable MMP13 18 42 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)CCc1ccccc1 ZINC000217982990 HE For-Sale Unstable MMP3 22 45 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)CCc1ccccc1 ZINC000217982990 HE For-Sale Unstable MMP1 17 40 CC[C@@H](NC(=O)CSc1ccc(Cl)cc1)c1ccc(C)c(C)c1 ZINC000217983013 EK In-Stock Unstable UTS2 42 33 CCOC(=O)[C@@H]1CCCN(C(=O)N/C=C/c2cccc(F)c2)C1 ZINC000217983015 DF For-Sale Unstable SLC6A1 51 38 CCOC(=O)[C@@H]1CCCN(C(=O)N/C=C/c2cccc(F)c2)C1 ZINC000217983015 DF For-Sale Unstable FDFT1 28 41 CCOC(=O)[C@@H]1CCCN(C(=O)N/C=C/c2cccc(F)c2)C1 ZINC000217983015 DF For-Sale Unstable NR1H4 19 40 Cc1noc2nc(C(C)C)cc(C(=O)Nc3ccc(Sc4nccn4C)cc3)c12 ZINC000217983054 HJ On-Demand Unstable GCK 16 42 CCOC(=O)[C@H]1CCCN(C(=O)N/C=C/c2cccc(F)c2)C1 ZINC000217983096 DF For-Sale Unstable SLC6A1 51 38 CCOC(=O)[C@H]1CCCN(C(=O)N/C=C/c2cccc(F)c2)C1 ZINC000217983096 DF For-Sale Unstable FDFT1 28 41 CCOC(=O)[C@H]1CCCN(C(=O)N/C=C/c2cccc(F)c2)C1 ZINC000217983096 DF For-Sale Unstable NR1H4 19 40 CC[C@H](NC(=O)CSc1ccc(Cl)cc1)c1ccc(C)c(C)c1 ZINC000217983107 EK In-Stock Unstable UTS2 42 33 COC(=O)c1cc(C=O)cn1Cc1ccccc1 ZINC000217983114 BE For-Sale Unstable PLA2G2A 56 35 COC(=O)c1cc(C=O)cn1Cc1ccccc1 ZINC000217983114 BE For-Sale Unstable HDAC6 17 41 COC(=O)c1cc(C=O)cn1Cc1ccccc1 ZINC000217983114 BE For-Sale Unstable FAS 44 36 O=C(O)Cc1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217983198 DG For-Sale Unstable HPSE 41 38 NC(=O)c1ccc(/C=C2/CC(=O)NC2=O)cc1 ZINC000217983224 BC For-Sale Unstable TRY1_BOVIN 50 50 C[C@@](O)(CNC(=O)c1ccccc1)c1cc2ccccc2o1 ZINC000217983318 CG In-Stock Unstable KCNJ11 54 39 O=C(N/C=C/c1cccc(F)c1)NCc1ccc(C(=O)O)cc1 ZINC000217983320 DF For-Sale Unstable UL80 20 41 CC(F)(F)CCS(=O)(=O)c1ccc(N)cc1 ZINC000217983354 BE For-Sale Unstable DYR_PNECA 18 43 CC(F)(F)CCS(=O)(=O)c1ccc(N)cc1 ZINC000217983354 BE For-Sale Unstable CAH_METTE 18 42 CC(F)(F)CCS(=O)(=O)c1ccc(N)cc1 ZINC000217983354 BE For-Sale Unstable CYNT 19 43 O=C1C/C(=C\c2ccc3c(c2)OCCCO3)C(=O)N1 ZINC000217983374 CD For-Sale Unstable DYRK1A 22 40 O=C1C/C(=C\c2ccc3c(c2)OCCCO3)C(=O)N1 ZINC000217983374 CD For-Sale Unstable CLK1 34 40 O=C1C/C(=C\c2ccc3c(c2)OCCCO3)C(=O)N1 ZINC000217983374 CD For-Sale Unstable DYRK2 72 40 C[C@](O)(CNC(=O)c1ccccc1)c1cc2ccccc2o1 ZINC000217983381 CG In-Stock Unstable KCNJ11 54 39 CC[C@@H](NC(=O)CSc1ccc(Cl)cc1)c1ccc(OC)c(OC)c1 ZINC000217983389 GJ In-Stock Unstable ENPP1 63 39 CC[C@@H](NC(=O)CSc1ccc(Cl)cc1)c1ccc(OC)c(OC)c1 ZINC000217983389 GJ In-Stock Unstable UTS2 42 33 CC[C@@H](NC(=O)CSc1ccc(Cl)cc1)c1ccc(OC)c(OC)c1 ZINC000217983389 GJ In-Stock Unstable FAS 39 41 Cn1nc(CC(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)c2ccccc2c1=O ZINC000217983438 GD In-Stock Unstable CHRNA4 30 48 Cn1nc(CC(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)c2ccccc2c1=O ZINC000217983438 GD In-Stock Unstable IMDH_CRYPV 26 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1cccc(OC)c1 ZINC000217983449 HE For-Sale Unstable MMP13 47 42 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1cccc(OC)c1 ZINC000217983449 HE For-Sale Unstable ADAM17 19 42 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1cccc(OC)c1 ZINC000217983449 HE For-Sale Unstable MMP2 22 56 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1cccc(OC)c1 ZINC000217983449 HE For-Sale Unstable MMP3 58 42 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1cccc(OC)c1 ZINC000217983449 HE For-Sale Unstable MMP9 34 42 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1cccc(OC)c1 ZINC000217983449 HE For-Sale Unstable PKM 19 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1cccc(OC)c1 ZINC000217983449 HE For-Sale Unstable MMP7 55 38 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1cccc(OC)c1 ZINC000217983449 HE For-Sale Unstable MMP1 50 42 CC[C@H](NC(=O)CSc1ccc(Cl)cc1)c1ccc(OC)c(OC)c1 ZINC000217983459 GJ In-Stock Unstable ENPP1 76 39 CC[C@H](NC(=O)CSc1ccc(Cl)cc1)c1ccc(OC)c(OC)c1 ZINC000217983459 GJ In-Stock Unstable UTS2 44 33 CC[C@H](NC(=O)CSc1ccc(Cl)cc1)c1ccc(OC)c(OC)c1 ZINC000217983459 GJ In-Stock Unstable FAS 39 41 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1cccc(OC)c1 ZINC000217983527 HE For-Sale Unstable MMP13 47 42 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1cccc(OC)c1 ZINC000217983527 HE For-Sale Unstable ADAM17 19 42 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1cccc(OC)c1 ZINC000217983527 HE For-Sale Unstable MMP2 22 56 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1cccc(OC)c1 ZINC000217983527 HE For-Sale Unstable MMP3 58 42 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1cccc(OC)c1 ZINC000217983527 HE For-Sale Unstable MMP9 34 42 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1cccc(OC)c1 ZINC000217983527 HE For-Sale Unstable PKM 19 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1cccc(OC)c1 ZINC000217983527 HE For-Sale Unstable MMP7 55 38 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1cccc(OC)c1 ZINC000217983527 HE For-Sale Unstable MMP1 50 42 CCN[C@@H](Cc1cc(F)ccc1F)[C@@H]1CCC[C@@H](C)C1 ZINC000217983529 CI For-Sale Unstable DPP4 20 42 COc1ccc([C@@H]2CC(=O)Oc3ccc4c(c32)O/C(=C\c2cccc(OC)c2OC)C4=O)c(OC)c1 ZINC000217983544 JJ In-Stock Unstable MT-ND4 52 34 CC[C@@H](NC(=O)CSc1ccc(Cl)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217983562 GI In-Stock Unstable PTGS2 18 43 CC[C@@H](NC(=O)CSc1ccc(Cl)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217983562 GI In-Stock Unstable UTS2 42 33 CCN[C@H](Cc1cc(F)ccc1F)[C@@H]1CCC[C@@H](C)C1 ZINC000217983612 CI For-Sale Unstable DPP4 20 42 COc1ccc([C@H]2CC(=O)Oc3ccc4c(c32)O/C(=C\c2cccc(OC)c2OC)C4=O)c(OC)c1 ZINC000217983621 JJ In-Stock Unstable MT-ND4 52 34 CC[C@H](NC(=O)CSc1ccc(Cl)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217983637 GI In-Stock Unstable PTGS2 16 43 CC[C@H](NC(=O)CSc1ccc(Cl)cc1)c1ccc(S(C)(=O)=O)cc1 ZINC000217983637 GI In-Stock Unstable UTS2 42 33 CCN[C@@H](Cc1cc(F)ccc1F)[C@H]1CCC[C@@H](C)C1 ZINC000217983695 CI For-Sale Unstable DPP4 20 42 O=C(Nc1ccc(Br)cc1)[C@@H]1CC[C@@H](Cn2cnnn2)CC1 ZINC000217983699 FF In-Stock Unstable DHODH 19 40 Cc1cccc(-c2noc(CNC(=O)CSc3ccc(Cl)cc3)n2)c1 ZINC000217983749 FI In-Stock Unstable GRM5 23 45 CCN[C@H](Cc1cc(F)ccc1F)[C@H]1CCC[C@@H](C)C1 ZINC000217983770 CI For-Sale Unstable DPP4 20 42 NCCc1ccc(S(=O)(=O)CC(F)F)cc1 ZINC000217983775 BD For-Sale Unstable CA2 21 42 NCCc1ccc(S(=O)(=O)CC(F)F)cc1 ZINC000217983775 BD For-Sale Unstable CA1 20 56 NCCc1ccc(S(=O)(=O)CC(F)F)cc1 ZINC000217983775 BD For-Sale Unstable CA9 15 42 NCCc1ccc(S(=O)(=O)CC(F)F)cc1 ZINC000217983775 BD For-Sale Unstable CAH_METTE 21 56 NCCc1ccc(S(=O)(=O)CC(F)F)cc1 ZINC000217983775 BD For-Sale Unstable TAAR1 20 44 NCCc1ccc(S(=O)(=O)CC(F)F)cc1 ZINC000217983775 BD For-Sale Unstable NCE103 16 56 NCCc1ccc(S(=O)(=O)CC(F)F)cc1 ZINC000217983775 BD For-Sale Unstable CA15 15 56 Cc1ccc(-c2noc(CNC(=O)CSc3ccc(Cl)cc3)n2)cc1 ZINC000217983815 FI In-Stock Unstable TSPO 15 48 Cc1ccc(-c2noc(CNC(=O)CSc3ccc(Cl)cc3)n2)cc1 ZINC000217983815 FI In-Stock Unstable TNKS2 15 43 CCc1ncnc(NCCc2ccc(O)cc2)c1F ZINC000217983842 CF On-Demand Unstable HTT 0 55 CC1(C)CC(NC(=O)N/C=C/c2cccc(F)c2)CC(C)(C)N1 ZINC000217983864 DG For-Sale Unstable ENV 23 41 CC1(C)CC(NC(=O)N/C=C/c2cccc(F)c2)CC(C)(C)N1 ZINC000217983864 DG For-Sale Unstable EZH2 52 40 NCc1ccc(S(=O)(=O)CCC(F)F)cc1 ZINC000217983886 BD For-Sale Unstable CAH_METTE 15 50 COCc1cccc(N[C@H]2C[C@@H](C)CC[C@@H]2C(C)C)c1 ZINC000217983909 CJ For-Sale Unstable TRPM8 17 45 COc1cccc(-c2noc(CNC(=O)CSc3ccc(Cl)cc3)n2)c1 ZINC000217983930 GH In-Stock Unstable MTNR1A 47 37 COc1cccc(-c2noc(CNC(=O)CSc3ccc(Cl)cc3)n2)c1 ZINC000217983930 GH In-Stock Unstable MTNR1B 43 37 COc1cccc(-c2noc(CNC(=O)CSc3ccc(Cl)cc3)n2)c1 ZINC000217983930 GH In-Stock Unstable GRM5 19 44 COCc1cccc(N[C@H]2C[C@H](C)CC[C@@H]2C(C)C)c1 ZINC000217983995 CJ For-Sale Unstable TRPM8 17 45 COc1ccc(-c2noc(CNC(=O)CSc3ccc(Cl)cc3)n2)cc1 ZINC000217984035 GH In-Stock Unstable TSPO 15 44 COc1ccc(-c2noc(CNC(=O)CSc3ccc(Cl)cc3)n2)cc1 ZINC000217984035 GH In-Stock Unstable WNT3A 20 40 COc1ccc(-c2noc(CNC(=O)CSc3ccc(Cl)cc3)n2)cc1 ZINC000217984035 GH In-Stock Unstable TNKS2 16 41 COc1ccc(-c2noc(CNC(=O)CSc3ccc(Cl)cc3)n2)cc1 ZINC000217984035 GH In-Stock Unstable AXIN2 0 44 NCCc1cccc(S(=O)(=O)CC(F)F)c1 ZINC000217984108 BD For-Sale Unstable TAAR1 18 46 C[C@@](O)(CNC(=O)/C=C/c1ccccc1)c1cc2ccccc2o1 ZINC000217984235 DG In-Stock Unstable HDAC8 52 47 C[C@@](O)(CNC(=O)/C=C/c1ccccc1)c1cc2ccccc2o1 ZINC000217984235 DG In-Stock Unstable MMP2 16 45 C[C@@](O)(CNC(=O)/C=C/c1ccccc1)c1cc2ccccc2o1 ZINC000217984235 DG In-Stock Unstable HDAC1 24 46 C[C@@](O)(CNC(=O)/C=C/c1ccccc1)c1cc2ccccc2o1 ZINC000217984235 DG In-Stock Unstable HDAC6 39 41 CC(C)[C@@H]1CC[C@@H](C(=O)N[C@@H](Cc2ccccc2)C(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)CC1 ZINC000217984278 JH In-Stock Unstable ACE 42 37 CC(C)[C@@H]1CC[C@@H](C(=O)N[C@@H](Cc2ccccc2)C(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)CC1 ZINC000217984278 JH In-Stock Unstable MC4R 44 40 CC(C)[C@@H]1CC[C@@H](C(=O)N[C@@H](Cc2ccccc2)C(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)CC1 ZINC000217984278 JH In-Stock Unstable CHRNA4 27 48 CC(C)[C@@H]1CC[C@@H](C(=O)N[C@@H](Cc2ccccc2)C(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)CC1 ZINC000217984278 JH In-Stock Unstable NPFFR2 57 32 CC(C)[C@@H]1CC[C@@H](C(=O)N[C@@H](Cc2ccccc2)C(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)CC1 ZINC000217984278 JH In-Stock Unstable MC5R 40 32 CC(C)[C@@H]1CC[C@@H](C(=O)N[C@@H](Cc2ccccc2)C(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)CC1 ZINC000217984278 JH In-Stock Unstable F11 44 36 CC(C)[C@@H]1CC[C@@H](C(=O)N[C@@H](Cc2ccccc2)C(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)CC1 ZINC000217984278 JH In-Stock Unstable NPFFR1 40 30 C[C@](O)(CNC(=O)/C=C/c1ccccc1)c1cc2ccccc2o1 ZINC000217984316 DG In-Stock Unstable HDAC8 52 47 C[C@](O)(CNC(=O)/C=C/c1ccccc1)c1cc2ccccc2o1 ZINC000217984316 DG In-Stock Unstable MMP2 16 45 C[C@](O)(CNC(=O)/C=C/c1ccccc1)c1cc2ccccc2o1 ZINC000217984316 DG In-Stock Unstable HDAC1 24 46 C[C@](O)(CNC(=O)/C=C/c1ccccc1)c1cc2ccccc2o1 ZINC000217984316 DG In-Stock Unstable HDAC6 39 41 CCn1cc(C=O)cc1C(=O)OCc1ccccc1 ZINC000217984326 CF For-Sale Unstable CHRM5 17 43 CCn1cc(C=O)cc1C(=O)OCc1ccccc1 ZINC000217984326 CF For-Sale Unstable KLK3 41 31 CCn1cc(C=O)cc1C(=O)OCc1ccccc1 ZINC000217984326 CF For-Sale Unstable CAPN1 42 37 CCn1cc(C=O)cc1C(=O)OCc1ccccc1 ZINC000217984326 CF For-Sale Unstable CAPN2 59 33 CCn1cc(C=O)cc1C(=O)OCc1ccccc1 ZINC000217984326 CF For-Sale Unstable SLC12A5 66 34 O=C(CSc1ccc(Cl)cc1)NCc1nc(-c2cccs2)no1 ZINC000217984336 FH In-Stock Unstable ETHR 29 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(C)c1 ZINC000217984369 HF For-Sale Unstable MMP2 17 52 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(C)c1 ZINC000217984369 HF For-Sale Unstable MMP3 46 37 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(C)c1 ZINC000217984369 HF For-Sale Unstable MMP7 45 35 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(C)c1 ZINC000217984369 HF For-Sale Unstable MMP1 40 37 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(C)c1 ZINC000217984369 HF For-Sale Unstable LEF 57 35 Nc1nc(Cl)c2ccc(Br)cc2n1 ZINC000217984413 CF For-Sale Unstable PTGES 0 41 Cc1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1C ZINC000217984431 CI For-Sale Unstable IMPDH2 0 42 CN(Cc1nc(-c2ccccc2)no1)C(=O)CSc1ccc(Cl)cc1 ZINC000217984438 FI In-Stock Unstable TSPO 30 47 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(C)c1 ZINC000217984440 HF For-Sale Unstable MMP2 17 52 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(C)c1 ZINC000217984440 HF For-Sale Unstable MMP3 46 37 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(C)c1 ZINC000217984440 HF For-Sale Unstable MMP7 45 35 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(C)c1 ZINC000217984440 HF For-Sale Unstable MMP1 40 37 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(C)c1 ZINC000217984440 HF For-Sale Unstable LEF 57 35 CC(=O)c1oc2ccc(Cl)cc2c1C=O ZINC000217984445 BG For-Sale Unstable AHR 18 41 Cc1ccc(-c2noc(CN(C)C(=O)CSc3ccc(Cl)cc3)n2)cc1 ZINC000217984522 GI In-Stock Unstable TSPO 24 53 Cc1ccc(-c2noc(CN(C)C(=O)CSc3ccc(Cl)cc3)n2)cc1 ZINC000217984522 GI In-Stock Unstable TNKS2 15 42 CCN(Cc1ccccc1)C(=O)N/C=C/c1cccc(F)c1 ZINC000217984544 CI For-Sale Unstable TSPO 24 44 CCN(Cc1ccccc1)C(=O)N/C=C/c1cccc(F)c1 ZINC000217984544 CI For-Sale Unstable NR1H4 22 41 CCN(Cc1ccccc1)C(=O)N/C=C/c1cccc(F)c1 ZINC000217984544 CI For-Sale Unstable LIMK2 24 42 CC(C)(C)OC(=O)N1CC(c2cccc(O)c2)C1 ZINC000217984629 BF For-Sale Unstable GPR119 36 43 COc1ccc(-c2noc(CN(C)C(=O)CSc3ccc(Cl)cc3)n2)cc1 ZINC000217984634 HI In-Stock Unstable TSPO 21 48 COc1ccc(-c2noc(CN(C)C(=O)CSc3ccc(Cl)cc3)n2)cc1 ZINC000217984634 HI In-Stock Unstable TNKS2 16 40 COc1ccc(-c2noc(CN(C)C(=O)CSc3ccc(Cl)cc3)n2)cc1 ZINC000217984634 HI In-Stock Unstable AXIN2 0 43 COc1ccc(C(=O)NC[C@@](C)(O)c2cc3ccccc3o2)cc1 ZINC000217984650 EG In-Stock Unstable MAOB 15 46 COc1ccc(C(=O)NC[C@@](C)(O)c2cc3ccccc3o2)cc1 ZINC000217984650 EG In-Stock Unstable KCNJ11 38 46 COc1ccc(C(=O)NC[C@@](C)(O)c2cc3ccccc3o2)cc1 ZINC000217984650 EG In-Stock Unstable NQO2 19 42 COc1ccc(C(=O)NC[C@@](C)(O)c2cc3ccccc3o2)cc1 ZINC000217984650 EG In-Stock Unstable ECR 24 41 CN1[C@@H]2CC[C@@H]1CC(N[C@H](c1ccccc1)C1CC1)C2 ZINC000217984654 CG For-Sale Unstable CHRM1 22 60 CN1[C@@H]2CC[C@@H]1CC(N[C@H](c1ccccc1)C1CC1)C2 ZINC000217984654 CG For-Sale Unstable SLC6A1 23 60 CN1[C@@H]2CC[C@@H]1CC(N[C@H](c1ccccc1)C1CC1)C2 ZINC000217984654 CG For-Sale Unstable SLC6A3 31 60 CN1[C@@H]2CC[C@@H]1CC(N[C@H](c1ccccc1)C1CC1)C2 ZINC000217984654 CG For-Sale Unstable CHRM4 18 49 CN1[C@@H]2CC[C@@H]1CC(N[C@H](c1ccccc1)C1CC1)C2 ZINC000217984654 CG For-Sale Unstable CHRM5 20 40 CN1[C@@H]2CC[C@@H]1CC(N[C@H](c1ccccc1)C1CC1)C2 ZINC000217984654 CG For-Sale Unstable GLRA1 43 32 COc1ccc(C(=O)NC[C@](C)(O)c2cc3ccccc3o2)cc1 ZINC000217984728 EG In-Stock Unstable MAOB 15 46 COc1ccc(C(=O)NC[C@](C)(O)c2cc3ccccc3o2)cc1 ZINC000217984728 EG In-Stock Unstable KCNJ11 38 46 COc1ccc(C(=O)NC[C@](C)(O)c2cc3ccccc3o2)cc1 ZINC000217984728 EG In-Stock Unstable NQO2 19 42 COc1ccc(C(=O)NC[C@](C)(O)c2cc3ccccc3o2)cc1 ZINC000217984728 EG In-Stock Unstable ECR 24 41 CN1[C@H]2CC[C@@H]1CC(N[C@H](c1ccccc1)C1CC1)C2 ZINC000217984735 CG For-Sale Unstable CHRM1 22 60 CN1[C@H]2CC[C@@H]1CC(N[C@H](c1ccccc1)C1CC1)C2 ZINC000217984735 CG For-Sale Unstable SLC6A1 23 60 CN1[C@H]2CC[C@@H]1CC(N[C@H](c1ccccc1)C1CC1)C2 ZINC000217984735 CG For-Sale Unstable SLC6A3 31 60 CN1[C@H]2CC[C@@H]1CC(N[C@H](c1ccccc1)C1CC1)C2 ZINC000217984735 CG For-Sale Unstable CHRM4 18 49 CN1[C@H]2CC[C@@H]1CC(N[C@H](c1ccccc1)C1CC1)C2 ZINC000217984735 CG For-Sale Unstable CHRM5 20 40 CN1[C@H]2CC[C@@H]1CC(N[C@H](c1ccccc1)C1CC1)C2 ZINC000217984735 CG For-Sale Unstable GLRA1 43 32 CC(C)(C)OC(=O)N1CC[C@@H]1c1cccc(O)c1 ZINC000217984739 BG For-Sale Unstable KIF11 30 42 CC(C)(C)OC(=O)N1CC[C@@H]1c1cccc(O)c1 ZINC000217984739 BG For-Sale Unstable GPR119 28 42 Cn1c(C(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc2ccccc21 ZINC000217984767 EF In-Stock Unstable CHRNA4 31 52 CN1[C@H]2CC[C@H]1CC(N[C@H](c1ccccc1)C1CC1)C2 ZINC000217984806 CG On-Demand Unstable CHRM1 22 60 CN1[C@H]2CC[C@H]1CC(N[C@H](c1ccccc1)C1CC1)C2 ZINC000217984806 CG On-Demand Unstable SLC6A1 23 60 CN1[C@H]2CC[C@H]1CC(N[C@H](c1ccccc1)C1CC1)C2 ZINC000217984806 CG On-Demand Unstable SLC6A3 31 60 CN1[C@H]2CC[C@H]1CC(N[C@H](c1ccccc1)C1CC1)C2 ZINC000217984806 CG On-Demand Unstable CHRM4 18 49 CN1[C@H]2CC[C@H]1CC(N[C@H](c1ccccc1)C1CC1)C2 ZINC000217984806 CG On-Demand Unstable CHRM5 20 40 CN1[C@H]2CC[C@H]1CC(N[C@H](c1ccccc1)C1CC1)C2 ZINC000217984806 CG On-Demand Unstable GLRA1 43 32 CC(C)(C)OC(=O)N1CC[C@H]1c1cccc(O)c1 ZINC000217984810 BG For-Sale Unstable KIF11 30 42 CC(C)(C)OC(=O)N1CC[C@H]1c1cccc(O)c1 ZINC000217984810 BG For-Sale Unstable GPR119 28 42 Cn1cccc(C(=O)NC[C@@](C)(O)c2cc3ccccc3o2)c1=O ZINC000217984837 ED In-Stock Unstable POLR1A 70 33 CN(Cc1nc(-c2ccccc2Cl)no1)C(=O)CSc1ccc(Cl)cc1 ZINC000217984845 HJ In-Stock Unstable GPBAR1 28 40 CC[C@@H]1CCCCN1C(=O)N/C=C/c1cccc(F)c1 ZINC000217984877 CH For-Sale Unstable ACKR3 61 38 Cn1cccc(C(=O)NC[C@](C)(O)c2cc3ccccc3o2)c1=O ZINC000217984926 ED In-Stock Unstable POLR1A 70 33 CC(C)(C)OC(=O)N1CC(c2ccccc2O)C1 ZINC000217984929 BF For-Sale Unstable GPR119 38 42 O=c1c2c(-c3ccc(F)cc3)csc2ncn1Cc1cnn(-c2ccccc2)c1 ZINC000217984930 HI On-Demand Unstable TGM2 18 46 CN(Cc1nc(-c2ccc(Cl)cc2)no1)C(=O)CSc1ccc(Cl)cc1 ZINC000217984955 HJ In-Stock Unstable TSPO 21 53 CN(Cc1nc(-c2ccc(Cl)cc2)no1)C(=O)CSc1ccc(Cl)cc1 ZINC000217984955 HJ In-Stock Unstable LIPE 23 41 CN(Cc1nc(-c2ccc(Cl)cc2)no1)C(=O)CSc1ccc(Cl)cc1 ZINC000217984955 HJ In-Stock Unstable UTS2 40 30 CC[C@H]1CCCCN1C(=O)N/C=C/c1cccc(F)c1 ZINC000217984970 CH For-Sale Unstable ACKR3 61 38 CC(C)(C)OC(=O)N1CC[C@@H]1c1ccccc1O ZINC000217985028 BG For-Sale Unstable GPR119 31 42 O=C(N/C=C/c1cccc(F)c1)N(Cc1ccccc1)Cc1ccccc1 ZINC000217985080 FK For-Sale Unstable NR1H4 23 42 O=C(N/C=C/c1cccc(F)c1)N(Cc1ccccc1)Cc1ccccc1 ZINC000217985080 FK For-Sale Unstable PTGES 25 40 O=C(N/C=C/c1cccc(F)c1)N(Cc1ccccc1)Cc1ccccc1 ZINC000217985080 FK For-Sale Unstable LIMK2 24 42 CC(C)(C)OC(=O)N1CC[C@H]1c1ccccc1O ZINC000217985104 BG For-Sale Unstable GPR119 31 42 CSc1ccccc1C(=O)Nc1ccc(NC(=O)c2ccco2)cc1C(F)(F)F ZINC000217985123 HK On-Demand Unstable GRM4 20 55 CSc1ccccc1C(=O)Nc1ccc(NC(=O)c2ccco2)cc1C(F)(F)F ZINC000217985123 HK On-Demand Unstable MTTP 42 35 CSc1ccccc1C(=O)Nc1ccc(NC(=O)c2ccco2)cc1C(F)(F)F ZINC000217985123 HK On-Demand Unstable KCNK3 50 43 CC[C@@H](CCO)Nc1ccc(C(=O)O)cn1 ZINC000217985153 BD On-Demand Unstable RXRA 41 34 CC[C@@H](CCO)Nc1ccc(C(=O)O)cn1 ZINC000217985153 BD On-Demand Unstable P4HTM 0 44 CC(C)CCCNC(=O)N1[C@H](C(=O)O)C[C@@H]2CCCC[C@@H]21 ZINC000217985219 CF On-Demand Unstable ACE 28 57 CC(C)(C)OC(=O)N1CC(c2ccc(O)cc2)C1 ZINC000217985221 BF For-Sale Unstable GPR119 42 44 CC[C@H](CCO)Nc1ccc(C(=O)O)cn1 ZINC000217985242 BD On-Demand Unstable RXRA 41 34 CC[C@H](CCO)Nc1ccc(C(=O)O)cn1 ZINC000217985242 BD On-Demand Unstable P4HTM 0 44 COc1ccc(NC(=O)N/C=C/c2cccc(F)c2)c(OC)c1 ZINC000217985305 DH For-Sale Unstable CYP1B1 48 45 COc1ccc(NC(=O)N/C=C/c2cccc(F)c2)c(OC)c1 ZINC000217985305 DH For-Sale Unstable MTNR1A 30 42 COc1ccc(NC(=O)N/C=C/c2cccc(F)c2)c(OC)c1 ZINC000217985305 DH For-Sale Unstable MTNR1B 29 42 CC(C)CCCNC(=O)N1[C@H](C(=O)O)C[C@H]2CCCC[C@@H]21 ZINC000217985310 CF On-Demand Unstable ACE 28 57 CCCCCCCCOc1ccc([C@@H]2CC(=O)Oc3c(C(C)=O)c(O)c4c(C)cc(=O)oc4c32)cc1 ZINC000217985312 JK In-Stock Unstable PLA2G4B 64 31 CCCCCCCCOc1ccc([C@@H]2CC(=O)Oc3c(C(C)=O)c(O)c4c(C)cc(=O)oc4c32)cc1 ZINC000217985312 JK In-Stock Unstable NTBBF1.1 0 41 Cc1ccc(C(=O)N[C@@H]2CCC[C@@H]2CO)c(F)c1 ZINC000217985313 CE On-Demand Unstable SSTR3 24 42 CC(C)(C)OC(=O)N1CC[C@@H]1c1ccc(O)cc1 ZINC000217985344 BG For-Sale Unstable GPR119 37 42 CCCCCCCCOc1ccc([C@H]2CC(=O)Oc3c(C(C)=O)c(O)c4c(C)cc(=O)oc4c32)cc1 ZINC000217985391 JK In-Stock Unstable PLA2G4B 64 31 CCCCCCCCOc1ccc([C@H]2CC(=O)Oc3c(C(C)=O)c(O)c4c(C)cc(=O)oc4c32)cc1 ZINC000217985391 JK In-Stock Unstable NTBBF1.1 0 41 Cc1ccc(C(=O)N[C@H]2CCC[C@@H]2CO)c(F)c1 ZINC000217985398 CE For-Sale Unstable SSTR3 25 42 CC(C)(C)OC(=O)N1CC[C@H]1c1ccc(O)cc1 ZINC000217985410 BG For-Sale Unstable GPR119 37 42 Cc1ccc(C(=O)N[C@@H]2CCC[C@H]2CO)c(F)c1 ZINC000217985470 CE For-Sale Unstable SSTR3 25 42 Cc1cc(Cl)ccc1NC(=O)N/C=C/c1cccc(F)c1 ZINC000217985487 DJ For-Sale Unstable CMA1 23 40 Cc1cc(Cl)ccc1NC(=O)N/C=C/c1cccc(F)c1 ZINC000217985487 DJ For-Sale Unstable H9CNL0_SPOEX 0 40 CN(C)[C@@H]1CCN(C[C@@H](C(=O)O)c2ccccc2)C1 ZINC000217985528 CD For-Sale Unstable CHRM1 18 41 CN(C)[C@@H]1CCN(C[C@@H](C(=O)O)c2ccccc2)C1 ZINC000217985528 CD For-Sale Unstable OPRM1 15 46 CN(C)[C@@H]1CCN(C[C@@H](C(=O)O)c2ccccc2)C1 ZINC000217985528 CD For-Sale Unstable OPRD1 17 46 CN(C)[C@@H]1CCN(C[C@@H](C(=O)O)c2ccccc2)C1 ZINC000217985528 CD For-Sale Unstable OPRK1 34 49 CN(C)[C@@H]1CCN(C[C@@H](C(=O)O)c2ccccc2)C1 ZINC000217985528 CD For-Sale Unstable SIGMAR1 20 44 CN(C)[C@@H]1CCN(C[C@@H](C(=O)O)c2ccccc2)C1 ZINC000217985528 CD For-Sale Unstable CCR5 91 51 O=C1[C@H]2[C@@H](c3ccc([N+](=O)[O-])cc3)N(c3ccccc3)O[C@H]2C(=O)N1c1ccc([N+](=O)[O-])cc1 ZINC000217985540 JH In-Stock Bother ACHE 20 86 O=C(Nc1ccc(NC(=O)c2ccco2)cc1C(F)(F)F)c1csc(-c2cccc(Cl)c2)n1 ZINC000217985544 JK On-Demand Anodyne GRM4 26 42 O=C(Nc1ccc(NC(=O)c2ccco2)cc1C(F)(F)F)c1csc(-c2cccc(Cl)c2)n1 ZINC000217985544 JK On-Demand Anodyne KISS1R 55 33 Cc1ccc(C(=O)N[C@H]2CCC[C@H]2CO)c(F)c1 ZINC000217985552 CE For-Sale Unstable SSTR3 25 42 CN(C)[C@H]1CCN(C[C@@H](C(=O)O)c2ccccc2)C1 ZINC000217985604 CD For-Sale Unstable CHRM1 18 41 CN(C)[C@H]1CCN(C[C@@H](C(=O)O)c2ccccc2)C1 ZINC000217985604 CD For-Sale Unstable OPRM1 15 46 CN(C)[C@H]1CCN(C[C@@H](C(=O)O)c2ccccc2)C1 ZINC000217985604 CD For-Sale Unstable OPRD1 17 46 CN(C)[C@H]1CCN(C[C@@H](C(=O)O)c2ccccc2)C1 ZINC000217985604 CD For-Sale Unstable OPRK1 34 49 CN(C)[C@H]1CCN(C[C@@H](C(=O)O)c2ccccc2)C1 ZINC000217985604 CD For-Sale Unstable SIGMAR1 20 44 CN(C)[C@H]1CCN(C[C@@H](C(=O)O)c2ccccc2)C1 ZINC000217985604 CD For-Sale Unstable CCR5 91 51 [C-]#[N+]C1(c2cccc(OCc3ccccc3)c2)CC1 ZINC000217985616 BI For-Sale Unstable ALOX5 16 44 O=C1[C@H]2ON(c3ccccc3)[C@H](c3ccc([N+](=O)[O-])cc3)[C@@H]2C(=O)N1c1ccc([N+](=O)[O-])cc1 ZINC000217985622 JH In-Stock Bother ACHE 20 86 C[C@@](O)(CNC(=O)c1c(F)cccc1F)c1cc2ccccc2o1 ZINC000217985640 EG In-Stock Unstable KCNJ11 55 35 O=C(N[C@@H]1CCC[C@@H]1CO)c1ccc(I)c(Cl)c1 ZINC000217985650 GF For-Sale Unstable SSTR3 33 42 CCOc1ccc(CNC(=O)[C@@H](C)Sc2ccc(Cl)cc2)cc1OCC ZINC000217985692 GJ In-Stock Unstable PDS 46 37 [C-]#[N+]C1(c2ccc(OCc3ccccc3)cc2)CC1 ZINC000217985713 BI For-Sale Unstable MAOB 26 40 [C-]#[N+]C1(c2ccc(OCc3ccccc3)cc2)CC1 ZINC000217985713 BI For-Sale Unstable LTA4H 23 44 [C-]#[N+]C1(c2ccc(OCc3ccccc3)cc2)CC1 ZINC000217985713 BI For-Sale Unstable TAAR1 19 44 [C-]#[N+]C1(c2ccc(OCc3ccccc3)cc2)CC1 ZINC000217985713 BI For-Sale Unstable FFAR1 19 43 O=C(Cc1csc(-c2ccccc2)n1)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217985715 GG In-Stock Unstable CHRNA4 30 50 C[C@](O)(CNC(=O)c1c(F)cccc1F)c1cc2ccccc2o1 ZINC000217985723 EG In-Stock Unstable KCNJ11 55 35 O=C(N[C@H]1CCC[C@@H]1CO)c1ccc(I)c(Cl)c1 ZINC000217985724 GF For-Sale Unstable SSTR3 33 42 CCOc1ccc(CNC(=O)[C@H](C)Sc2ccc(Cl)cc2)cc1OCC ZINC000217985781 GJ In-Stock Unstable PDS 46 37 O=C(N[C@@H]1CCC[C@H]1CO)c1ccc(I)c(Cl)c1 ZINC000217985800 GF For-Sale Unstable SSTR3 33 42 Cc1nc(-c2ccccc2)sc1C(=O)N1CCCC[C@H]1c1cccnc1 ZINC000217985825 FJ In-Stock Unstable CHRNA2 42 43 Cc1nc(-c2ccccc2)sc1C(=O)N1CCCC[C@H]1c1cccnc1 ZINC000217985825 FJ In-Stock Unstable CPT1A 95 46 Cc1nc(-c2ccccc2)sc1C(=O)N1CCCC[C@H]1c1cccnc1 ZINC000217985825 FJ In-Stock Unstable CRTY 0 43 C[C@@](O)(CNC(=O)c1ccc(F)c(F)c1)c1cc2ccccc2o1 ZINC000217985832 EG In-Stock Unstable KCNJ11 49 34 COc1cc(CNC(=O)[C@@H](C)Sc2ccc(Cl)cc2)ccc1OC(C)C ZINC000217985870 GJ In-Stock Unstable TRPV1 0 40 COc1cc(CNC(=O)[C@@H](C)Sc2ccc(Cl)cc2)ccc1OC(C)C ZINC000217985870 GJ In-Stock Unstable U38 0 41 CCN(CC)[C@@H]1CCN(C[C@@H](C(=O)O)c2ccccc2)C1 ZINC000217985886 CE For-Sale Unstable CHRM1 15 42 CCN(CC)[C@@H]1CCN(C[C@@H](C(=O)O)c2ccccc2)C1 ZINC000217985886 CE For-Sale Unstable OPRM1 15 47 CCN(CC)[C@@H]1CCN(C[C@@H](C(=O)O)c2ccccc2)C1 ZINC000217985886 CE For-Sale Unstable OPRD1 21 47 CCN(CC)[C@@H]1CCN(C[C@@H](C(=O)O)c2ccccc2)C1 ZINC000217985886 CE For-Sale Unstable OPRK1 29 45 CCN(CC)[C@@H]1CCN(C[C@@H](C(=O)O)c2ccccc2)C1 ZINC000217985886 CE For-Sale Unstable CCR5 96 47 O=C(N[C@H]1CCC[C@H]1CO)c1ccc(I)c(Cl)c1 ZINC000217985887 GF On-Demand Unstable SSTR3 33 42 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(F)c1 ZINC000217985888 HE For-Sale Unstable MMP13 46 39 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(F)c1 ZINC000217985888 HE For-Sale Unstable MMP2 22 54 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(F)c1 ZINC000217985888 HE For-Sale Unstable MMP3 56 39 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(F)c1 ZINC000217985888 HE For-Sale Unstable MMP7 50 36 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(F)c1 ZINC000217985888 HE For-Sale Unstable MMP1 48 39 C[C@](O)(CNC(=O)c1ccc(F)c(F)c1)c1cc2ccccc2o1 ZINC000217985910 EG In-Stock Unstable KCNJ11 49 34 Cc1cc(C)n(C[C@@H]2CCCO2)c(=O)c1C(=O)NCCc1c[nH]c2ccccc12 ZINC000217985915 GG In-Stock Unstable MC4R 40 41 COc1cc(CNC(=O)[C@H](C)Sc2ccc(Cl)cc2)ccc1OC(C)C ZINC000217985945 GJ In-Stock Unstable TRPV1 0 40 COc1cc(CNC(=O)[C@H](C)Sc2ccc(Cl)cc2)ccc1OC(C)C ZINC000217985945 GJ In-Stock Unstable U38 0 41 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(F)c1 ZINC000217985949 HE For-Sale Unstable MMP13 46 39 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(F)c1 ZINC000217985949 HE For-Sale Unstable MMP2 22 54 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(F)c1 ZINC000217985949 HE For-Sale Unstable MMP3 56 39 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(F)c1 ZINC000217985949 HE For-Sale Unstable MMP7 50 36 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(F)c1 ZINC000217985949 HE For-Sale Unstable MMP1 48 39 CCN(CC)[C@H]1CCN(C[C@@H](C(=O)O)c2ccccc2)C1 ZINC000217985967 CE For-Sale Unstable CHRM1 15 42 CCN(CC)[C@H]1CCN(C[C@@H](C(=O)O)c2ccccc2)C1 ZINC000217985967 CE For-Sale Unstable OPRM1 15 47 CCN(CC)[C@H]1CCN(C[C@@H](C(=O)O)c2ccccc2)C1 ZINC000217985967 CE For-Sale Unstable OPRD1 21 47 CCN(CC)[C@H]1CCN(C[C@@H](C(=O)O)c2ccccc2)C1 ZINC000217985967 CE For-Sale Unstable OPRK1 29 45 CCN(CC)[C@H]1CCN(C[C@@H](C(=O)O)c2ccccc2)C1 ZINC000217985967 CE For-Sale Unstable CCR5 96 47 CN(C(=O)CCC(=O)NCc1ccc2[nH]c(=O)[nH]c2c1)C1CCCCC1 ZINC000217985985 FE In-Stock Unstable P2RY12 22 52 CN(C(=O)CCC(=O)NCc1ccc2[nH]c(=O)[nH]c2c1)C1CCCCC1 ZINC000217985985 FE In-Stock Unstable PYGL 27 43 Cc1cc(C)n(C[C@H]2CCCO2)c(=O)c1C(=O)NCCc1c[nH]c2ccccc12 ZINC000217986014 GG In-Stock Unstable MC4R 40 41 Cc1cc(C)n(C[C@H]2CCCO2)c(=O)c1C(=O)NCCc1c[nH]c2ccccc12 ZINC000217986014 GG In-Stock Unstable NMBR 42 39 C[C@@](O)(CNC(=O)c1ccc(Cl)s1)c1cc2ccccc2o1 ZINC000217986024 EH In-Stock Unstable F10 22 45 C[C@@](O)(CNC(=O)c1ccc(Cl)s1)c1cc2ccccc2o1 ZINC000217986024 EH In-Stock Unstable KCNJ11 58 33 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(F)c1 ZINC000217986035 HE For-Sale Unstable MMP13 46 39 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(F)c1 ZINC000217986035 HE For-Sale Unstable MMP2 22 54 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(F)c1 ZINC000217986035 HE For-Sale Unstable MMP3 56 39 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(F)c1 ZINC000217986035 HE For-Sale Unstable MMP7 50 36 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(F)c1 ZINC000217986035 HE For-Sale Unstable MMP1 48 39 C[C@@H](Sc1ccc(Cl)cc1)C(=O)NCCCc1ccccc1Cl ZINC000217986068 FK In-Stock Unstable SCN10A 22 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(F)c1 ZINC000217986108 HE For-Sale Unstable MMP13 46 39 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(F)c1 ZINC000217986108 HE For-Sale Unstable MMP2 22 54 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(F)c1 ZINC000217986108 HE For-Sale Unstable MMP3 56 39 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(F)c1 ZINC000217986108 HE For-Sale Unstable MMP7 50 36 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(F)c1 ZINC000217986108 HE For-Sale Unstable MMP1 48 39 C[C@](O)(CNC(=O)c1ccc(Cl)s1)c1cc2ccccc2o1 ZINC000217986116 EH In-Stock Unstable F10 22 45 C[C@](O)(CNC(=O)c1ccc(Cl)s1)c1cc2ccccc2o1 ZINC000217986116 EH In-Stock Unstable KCNJ11 58 33 N#Cc1cncc2c1CN(Cc1ccccc1)CC2 ZINC000217986141 BF For-Sale Unstable SIGMAR1 28 40 N#Cc1cncc2c1CN(Cc1ccccc1)CC2 ZINC000217986141 BF For-Sale Unstable NOD2 40 33 C[C@H](Sc1ccc(Cl)cc1)C(=O)NCCCc1ccccc1Cl ZINC000217986170 FK In-Stock Unstable SCN10A 22 40 O=C(COc1ccc(F)c(Cl)c1)N1CCC(n2cnnc2)CC1 ZINC000217986196 EE In-Stock Unstable HTR1B 17 40 O=C(COc1ccc(F)c(Cl)c1)N1CCC(n2cnnc2)CC1 ZINC000217986196 EE In-Stock Unstable HRH1 17 40 O=C(COc1ccc(F)c(Cl)c1)N1CCC(n2cnnc2)CC1 ZINC000217986196 EE In-Stock Unstable CCR3 21 40 O=C(COc1ccc(F)c(Cl)c1)N1CCC(n2cnnc2)CC1 ZINC000217986196 EE In-Stock Unstable GPR183 0 43 N#Cc1cncc2c1CCN(Cc1ccccc1)C2 ZINC000217986256 BF For-Sale Unstable SIGMAR1 28 41 C[C@@H](Sc1ccc(Cl)cc1)C(=O)NCCCc1ccc(Cl)cc1 ZINC000217986275 FK In-Stock Unstable SLC6A5 16 42 C[C@@H](Sc1ccc(Cl)cc1)C(=O)NCCCc1ccc(Cl)cc1 ZINC000217986275 FK In-Stock Unstable AMP1_PLAFQ 35 41 O=C(Cn1ncc2ccccc21)N[C@@H](CCn1cncn1)c1ccccc1 ZINC000217986287 FF In-Stock Unstable HIS3 50 37 O=C(Cn1ncc2ccccc21)N[C@@H](CCn1cncn1)c1ccccc1 ZINC000217986287 FF In-Stock Unstable CYP51 0 43 CC[C@@H](CCO)Nc1ccc(C(=O)O)nc1 ZINC000217986342 BD For-Sale Unstable P4HTM 0 44 CC[C@@H](CCO)Nc1ccc(C(=O)O)nc1 ZINC000217986342 BD For-Sale Unstable P4HA1 0 41 C[C@H](Sc1ccc(Cl)cc1)C(=O)NCCCc1ccc(Cl)cc1 ZINC000217986351 FK In-Stock Unstable SLC6A5 16 42 C[C@H](Sc1ccc(Cl)cc1)C(=O)NCCCc1ccc(Cl)cc1 ZINC000217986351 FK In-Stock Unstable AMP1_PLAFQ 35 41 O=C(Cn1ncc2ccccc21)N[C@H](CCn1cncn1)c1ccccc1 ZINC000217986373 FF In-Stock Unstable HIS3 50 37 O=C(Cn1ncc2ccccc21)N[C@H](CCn1cncn1)c1ccccc1 ZINC000217986373 FF In-Stock Unstable CYP51 0 43 CCOc1ccccc1C(=O)NC[C@](C)(O)c1cc2ccccc2o1 ZINC000217986388 EG In-Stock Unstable HCN1 52 39 CCOc1ccccc1C(=O)NC[C@](C)(O)c1cc2ccccc2o1 ZINC000217986388 EG In-Stock Unstable HCN4 49 38 CCOc1ccccc1C(=O)NC[C@](C)(O)c1cc2ccccc2o1 ZINC000217986388 EG In-Stock Unstable KCNK3 46 44 CCOc1ccccc1C(=O)NC[C@](C)(O)c1cc2ccccc2o1 ZINC000217986388 EG In-Stock Unstable KCNK9 44 44 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1ccccc1S(C)(=O)=O ZINC000217986411 DH For-Sale Unstable TRPM8 18 45 CC[C@H](CCO)Nc1ccc(C(=O)O)nc1 ZINC000217986423 BD For-Sale Unstable P4HTM 0 44 CC[C@H](CCO)Nc1ccc(C(=O)O)nc1 ZINC000217986423 BD For-Sale Unstable P4HA1 0 41 O=C(O)C[C@@H](N1CC[C@H](N2CCCC2)C1)C(F)(F)F ZINC000217986427 CD For-Sale Unstable L3MBTL3 40 35 C[C@@H](Sc1ccc(Cl)cc1)C(=O)NCCCc1ccc(F)cc1 ZINC000217986448 FJ In-Stock Unstable LEF 61 37 CCOc1ccccc1C(=O)NC[C@@](C)(O)c1cc2ccccc2o1 ZINC000217986469 EG In-Stock Unstable HCN1 52 39 CCOc1ccccc1C(=O)NC[C@@](C)(O)c1cc2ccccc2o1 ZINC000217986469 EG In-Stock Unstable HCN4 49 38 CCOc1ccccc1C(=O)NC[C@@](C)(O)c1cc2ccccc2o1 ZINC000217986469 EG In-Stock Unstable KCNK3 46 44 CCOc1ccccc1C(=O)NC[C@@](C)(O)c1cc2ccccc2o1 ZINC000217986469 EG In-Stock Unstable KCNK9 44 44 Cc1ccc(OCCOc2cc(Cl)cc(Cl)c2)cn1 ZINC000217986493 CI On-Demand Unstable S1PR4 18 44 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1ccccc1S(C)(=O)=O ZINC000217986495 DH For-Sale Unstable TRPM8 18 45 O=C(O)[C@@H]1CCC[C@@H]1N1CC[C@H](N2CCCC2)C1 ZINC000217986513 CD For-Sale Unstable L3MBTL1 0 45 O=C(O)[C@@H]1CCC[C@@H]1N1CC[C@H](N2CCCC2)C1 ZINC000217986513 CD For-Sale Unstable L3MBTL3 97 45 O=C(O)[C@@H]1CCC[C@@H]1N1CC[C@H](N2CCCC2)C1 ZINC000217986513 CD For-Sale Unstable L3MBTL4 0 40 O=C(O)[C@@H]1CCC[C@@H]1N1CC[C@H](N2CCCC2)C1 ZINC000217986513 CD For-Sale Unstable MBTD1 0 41 O=C(O)[C@@H]1CCC[C@@H]1N1CC[C@H](N2CCCC2)C1 ZINC000217986513 CD For-Sale Unstable TP53BP1 0 40 C[C@H](Sc1ccc(Cl)cc1)C(=O)NCCCc1ccc(F)cc1 ZINC000217986535 FJ In-Stock Unstable LEF 61 37 CC[C@@H](CCO)Nc1ccnc(C(=O)O)c1 ZINC000217986539 BD On-Demand Unstable FTO 0 41 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1c(F)cccc1F ZINC000217986541 HE For-Sale Unstable PKM 19 41 COc1cccc(CC(=O)NC[C@@](C)(O)c2cc3ccccc3o2)c1 ZINC000217986565 EG In-Stock Unstable MTNR1A 45 42 COc1cccc(CC(=O)NC[C@@](C)(O)c2cc3ccccc3o2)c1 ZINC000217986565 EG In-Stock Unstable MTNR1B 45 41 COc1cccc(CC(=O)NC[C@@](C)(O)c2cc3ccccc3o2)c1 ZINC000217986565 EG In-Stock Unstable CRTM 45 37 COc1cccc(CC(=O)NC[C@@](C)(O)c2cc3ccccc3o2)c1 ZINC000217986565 EG In-Stock Unstable CAN2 0 44 C=C(C)COc1ccccc1C(=O)N[C@@H]1C[C@@H](c2nnc(CO)n2C)C1 ZINC000217986586 FD In-Stock Unstable HCN1 40 32 C=C(C)COc1ccccc1C(=O)N[C@@H]1C[C@@H](c2nnc(CO)n2C)C1 ZINC000217986586 FD In-Stock Unstable HCN4 40 32 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1ccccc1S(C)(=O)=O ZINC000217986588 DH For-Sale Unstable TRPM8 18 45 O=C(O)[C@H]1CCC[C@@H]1N1CC[C@H](N2CCCC2)C1 ZINC000217986594 CD For-Sale Unstable L3MBTL3 97 45 CC[C@H](CCO)Nc1ccnc(C(=O)O)c1 ZINC000217986623 BD On-Demand Unstable FTO 0 41 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1c(F)cccc1F ZINC000217986630 HE For-Sale Unstable PKM 19 41 COc1ccccc1CCCNC(=O)[C@@H](C)Sc1ccc(Cl)cc1 ZINC000217986635 FJ In-Stock Unstable DRD2 16 42 COc1ccccc1CCCNC(=O)[C@@H](C)Sc1ccc(Cl)cc1 ZINC000217986635 FJ In-Stock Unstable DRD3 26 42 COc1ccccc1CCCNC(=O)[C@@H](C)Sc1ccc(Cl)cc1 ZINC000217986635 FJ In-Stock Unstable MTNR1B 36 41 COc1cccc(CC(=O)NC[C@](C)(O)c2cc3ccccc3o2)c1 ZINC000217986651 EG In-Stock Unstable MTNR1A 45 42 COc1cccc(CC(=O)NC[C@](C)(O)c2cc3ccccc3o2)c1 ZINC000217986651 EG In-Stock Unstable MTNR1B 45 41 COc1cccc(CC(=O)NC[C@](C)(O)c2cc3ccccc3o2)c1 ZINC000217986651 EG In-Stock Unstable CRTM 45 37 COc1cccc(CC(=O)NC[C@](C)(O)c2cc3ccccc3o2)c1 ZINC000217986651 EG In-Stock Unstable CAN2 0 44 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1ccccc1S(C)(=O)=O ZINC000217986665 DH For-Sale Unstable TRPM8 18 45 O=C(O)[C@@H]1CCC[C@H]1N1CC[C@H](N2CCCC2)C1 ZINC000217986667 CD For-Sale Unstable L3MBTL1 0 45 O=C(O)[C@@H]1CCC[C@H]1N1CC[C@H](N2CCCC2)C1 ZINC000217986667 CD For-Sale Unstable L3MBTL3 97 45 O=C(O)[C@@H]1CCC[C@H]1N1CC[C@H](N2CCCC2)C1 ZINC000217986667 CD For-Sale Unstable L3MBTL4 0 40 O=C(O)[C@@H]1CCC[C@H]1N1CC[C@H](N2CCCC2)C1 ZINC000217986667 CD For-Sale Unstable MBTD1 0 41 O=C(O)[C@@H]1CCC[C@H]1N1CC[C@H](N2CCCC2)C1 ZINC000217986667 CD For-Sale Unstable TP53BP1 0 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1c(F)cccc1F ZINC000217986723 HE For-Sale Unstable PKM 19 41 COc1ccccc1CCCNC(=O)[C@H](C)Sc1ccc(Cl)cc1 ZINC000217986724 FJ In-Stock Unstable DRD2 16 42 COc1ccccc1CCCNC(=O)[C@H](C)Sc1ccc(Cl)cc1 ZINC000217986724 FJ In-Stock Unstable DRD3 26 42 COc1ccccc1CCCNC(=O)[C@H](C)Sc1ccc(Cl)cc1 ZINC000217986724 FJ In-Stock Unstable MTNR1B 36 41 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1c(F)cccc1F ZINC000217986807 HE For-Sale Unstable PKM 19 41 COc1cccc(CCCNC(=O)[C@@H](C)Sc2ccc(Cl)cc2)c1 ZINC000217986820 FJ In-Stock Unstable DRD4 45 38 COc1cccc(CCCNC(=O)[C@@H](C)Sc2ccc(Cl)cc2)c1 ZINC000217986820 FJ In-Stock Unstable NQO2 19 40 COc1cccc(CCCNC(=O)[C@@H](C)Sc2ccc(Cl)cc2)c1 ZINC000217986820 FJ In-Stock Unstable MTNR1A 47 59 COc1cccc(CCCNC(=O)[C@@H](C)Sc2ccc(Cl)cc2)c1 ZINC000217986820 FJ In-Stock Unstable MTNR1B 43 57 COc1cccc(CCCNC(=O)[C@@H](C)Sc2ccc(Cl)cc2)c1 ZINC000217986820 FJ In-Stock Unstable AMP1_PLAFQ 38 42 COc1cccc(CCCNC(=O)[C@@H](C)Sc2ccc(Cl)cc2)c1 ZINC000217986820 FJ In-Stock Unstable AKR1C3 16 41 COc1cccc(CCCNC(=O)[C@@H](C)Sc2ccc(Cl)cc2)c1 ZINC000217986820 FJ In-Stock Unstable CRTM 65 48 COc1cccc(CCCNC(=O)[C@@H](C)Sc2ccc(Cl)cc2)c1 ZINC000217986820 FJ In-Stock Unstable PDS 60 38 CNC(=O)[C@@H]1CCCN1[C@@H](C)c1ccc(C(=O)O)o1 ZINC000217986856 CD For-Sale Unstable XPNPEP1 0 42 CNC(=O)[C@@H]1CCCN1[C@@H](C)c1ccc(C(=O)O)o1 ZINC000217986856 CD For-Sale Unstable XPNPEP2 0 42 N[C@H](/C=C/F)C(=O)O ZINC000217986891 AB For-Sale Unstable ACS5 0 43 COc1cccc(CCCNC(=O)[C@H](C)Sc2ccc(Cl)cc2)c1 ZINC000217986893 FJ In-Stock Unstable DRD4 45 38 COc1cccc(CCCNC(=O)[C@H](C)Sc2ccc(Cl)cc2)c1 ZINC000217986893 FJ In-Stock Unstable NQO2 19 40 COc1cccc(CCCNC(=O)[C@H](C)Sc2ccc(Cl)cc2)c1 ZINC000217986893 FJ In-Stock Unstable MTNR1A 47 59 COc1cccc(CCCNC(=O)[C@H](C)Sc2ccc(Cl)cc2)c1 ZINC000217986893 FJ In-Stock Unstable MTNR1B 43 57 COc1cccc(CCCNC(=O)[C@H](C)Sc2ccc(Cl)cc2)c1 ZINC000217986893 FJ In-Stock Unstable AMP1_PLAFQ 38 42 COc1cccc(CCCNC(=O)[C@H](C)Sc2ccc(Cl)cc2)c1 ZINC000217986893 FJ In-Stock Unstable AKR1C3 16 41 COc1cccc(CCCNC(=O)[C@H](C)Sc2ccc(Cl)cc2)c1 ZINC000217986893 FJ In-Stock Unstable CRTM 65 48 COc1cccc(CCCNC(=O)[C@H](C)Sc2ccc(Cl)cc2)c1 ZINC000217986893 FJ In-Stock Unstable PDS 60 38 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(Cl)s1 ZINC000217986913 HF For-Sale Unstable CCR4 49 33 Cc1noc2nc(C(C)C)cc(C(=O)Nc3ccccc3OCC(F)(F)F)c12 ZINC000217986940 GJ On-Demand Unstable KCNK3 42 36 Cc1noc2nc(C(C)C)cc(C(=O)Nc3ccccc3OCC(F)(F)F)c12 ZINC000217986940 GJ On-Demand Unstable KCNK9 42 38 O=C(O)[C@@H]1CCC[C@@H]1N1CC[C@H](N2CCCCC2)C1 ZINC000217986947 CD For-Sale Unstable L3MBTL1 0 44 O=C(O)[C@@H]1CCC[C@@H]1N1CC[C@H](N2CCCCC2)C1 ZINC000217986947 CD For-Sale Unstable L3MBTL3 99 44 O=C(O)[C@@H]1CCC[C@@H]1N1CC[C@H](N2CCCCC2)C1 ZINC000217986947 CD For-Sale Unstable MBTD1 0 44 COc1ccc(CCCNC(=O)[C@@H](C)Sc2ccc(Cl)cc2)cc1 ZINC000217986976 FJ In-Stock Unstable SCNN1A 46 41 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(Cl)s1 ZINC000217986990 HF For-Sale Unstable CCR4 49 33 O=C(O)[C@H]1CCC[C@@H]1N1CC[C@H](N2CCCCC2)C1 ZINC000217987035 CD For-Sale Unstable L3MBTL1 0 44 O=C(O)[C@H]1CCC[C@@H]1N1CC[C@H](N2CCCCC2)C1 ZINC000217987035 CD For-Sale Unstable L3MBTL3 99 44 O=C(O)[C@H]1CCC[C@@H]1N1CC[C@H](N2CCCCC2)C1 ZINC000217987035 CD For-Sale Unstable MBTD1 0 44 COc1ccc(CCCNC(=O)[C@H](C)Sc2ccc(Cl)cc2)cc1 ZINC000217987044 FJ In-Stock Unstable SCNN1A 46 41 COc1ccc2nc(NC(=O)[C@@H]3CC[C@@H](Cn4cnnn4)CC3)sc2c1 ZINC000217987048 FF In-Stock Unstable LCK 17 44 COc1ccc2nc(NC(=O)[C@@H]3CC[C@@H](Cn4cnnn4)CC3)sc2c1 ZINC000217987048 FF In-Stock Unstable CSNK1D 47 51 COc1ccc2nc(NC(=O)[C@@H]3CC[C@@H](Cn4cnnn4)CC3)sc2c1 ZINC000217987048 FF In-Stock Unstable NMT1 39 42 COc1ccc2nc(NC(=O)[C@@H]3CC[C@@H](Cn4cnnn4)CC3)sc2c1 ZINC000217987048 FF In-Stock Unstable FABK 0 44 COc1ccc2nc(NC(=O)[C@@H]3CC[C@@H](Cn4cnnn4)CC3)sc2c1 ZINC000217987048 FF In-Stock Unstable PORCN 0 43 COc1ccc2nc(NC(=O)[C@@H]3CC[C@@H](Cn4cnnn4)CC3)sc2c1 ZINC000217987048 FF In-Stock Unstable ISPD 0 45 Cc1ccccc1OCC(=O)NC[C@](C)(O)c1cc2ccccc2o1 ZINC000217987077 EG In-Stock Unstable CETP 22 43 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(Cl)s1 ZINC000217987083 HF For-Sale Unstable CCR4 49 33 O=C(O)[C@@H]1CCC[C@H]1N1CC[C@H](N2CCCCC2)C1 ZINC000217987105 CD For-Sale Unstable L3MBTL1 0 44 O=C(O)[C@@H]1CCC[C@H]1N1CC[C@H](N2CCCCC2)C1 ZINC000217987105 CD For-Sale Unstable L3MBTL3 99 44 O=C(O)[C@@H]1CCC[C@H]1N1CC[C@H](N2CCCCC2)C1 ZINC000217987105 CD For-Sale Unstable MBTD1 0 44 COc1ccc(OC[C@@H](C)NC(=O)[C@@H](C)Sc2ccc(Cl)cc2)cc1 ZINC000217987141 GI In-Stock Unstable PTGS2 0 41 COc1ccc(OC[C@@H](C)NC(=O)[C@@H](C)Sc2ccc(Cl)cc2)cc1 ZINC000217987141 GI In-Stock Unstable SDH1 0 41 Cc1ccccc1OCC(=O)NC[C@@](C)(O)c1cc2ccccc2o1 ZINC000217987154 EG In-Stock Unstable CETP 22 43 CC[C@@H](CCO)NC(=N)Nc1ccccc1 ZINC000217987160 BD For-Sale Unstable SCN2A 35 41 CC[C@@H](C(=O)N[C@@H](CC(=O)OC(C)C)c1ccccc1[N+](=O)[O-])c1ccccc1 ZINC000217987167 GI On-Demand Unstable COLA 91 34 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(Cl)s1 ZINC000217987169 HF For-Sale Unstable CCR4 49 33 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217987187 EK For-Sale Anodyne MMP1 0 50 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217987187 EK For-Sale Anodyne AKR1C3 21 40 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(Nc2ccccc2)cc1 ZINC000217987187 EK For-Sale Anodyne P95276_MYCTO 0 40 O=C(O)[C@@H]1CCCC[C@@H]1N1CC[C@H](N2CCCCC2)C1 ZINC000217987217 CE For-Sale Unstable L3MBTL3 97 44 COc1ccc(OC[C@H](C)NC(=O)[C@@H](C)Sc2ccc(Cl)cc2)cc1 ZINC000217987227 GI In-Stock Unstable PTGS2 0 41 COc1ccc(OC[C@H](C)NC(=O)[C@@H](C)Sc2ccc(Cl)cc2)cc1 ZINC000217987227 GI In-Stock Unstable SDH1 0 41 CC[C@H](CCO)NC(=N)Nc1ccccc1 ZINC000217987229 BD For-Sale Unstable SCN2A 35 41 CC[C@H](C(=O)N[C@@H](CC(=O)OC(C)C)c1ccccc1[N+](=O)[O-])c1ccccc1 ZINC000217987242 GI On-Demand Unstable COLA 91 34 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(C)=O)cc1 ZINC000217987279 HE For-Sale Unstable MMP13 55 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(C)=O)cc1 ZINC000217987279 HE For-Sale Unstable MMP2 28 55 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(C)=O)cc1 ZINC000217987279 HE For-Sale Unstable MMP3 64 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(C)=O)cc1 ZINC000217987279 HE For-Sale Unstable MMP7 63 38 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(C)=O)cc1 ZINC000217987279 HE For-Sale Unstable MMP1 58 40 O=C(O)[C@H]1CCCC[C@@H]1N1CC[C@H](N2CCCCC2)C1 ZINC000217987302 CE For-Sale Unstable L3MBTL3 97 44 COc1ccc(OC[C@@H](C)NC(=O)[C@H](C)Sc2ccc(Cl)cc2)cc1 ZINC000217987303 GI In-Stock Unstable PTGS2 0 41 COc1ccc(OC[C@@H](C)NC(=O)[C@H](C)Sc2ccc(Cl)cc2)cc1 ZINC000217987303 GI In-Stock Unstable SDH1 0 41 O=C(N/C=C/c1cccc(F)c1)N1CCc2ccccc2C1 ZINC000217987305 CH For-Sale Unstable HDAC6 36 40 CC[C@@H](C(=O)N[C@H](CC(=O)OC(C)C)c1ccccc1[N+](=O)[O-])c1ccccc1 ZINC000217987327 GI On-Demand Unstable COLA 91 34 COC(=O)C[C@H](c1ccc(OCCc2ccc(OC)cc2)c(OC)c1)c1c(O)c2ccccc2oc1=O ZINC000217987359 KJ In-Stock Unstable NQO1 41 52 COC(=O)C[C@H](c1ccc(OCCc2ccc(OC)cc2)c(OC)c1)c1c(O)c2ccccc2oc1=O ZINC000217987359 KJ In-Stock Unstable ABCG2 25 41 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(C)=O)cc1 ZINC000217987364 HE For-Sale Unstable MMP13 55 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(C)=O)cc1 ZINC000217987364 HE For-Sale Unstable MMP2 28 55 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(C)=O)cc1 ZINC000217987364 HE For-Sale Unstable MMP3 64 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(C)=O)cc1 ZINC000217987364 HE For-Sale Unstable MMP7 63 38 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(C)=O)cc1 ZINC000217987364 HE For-Sale Unstable MMP1 58 40 O=C(O)[C@@H]1CCCC[C@H]1N1CC[C@H](N2CCCCC2)C1 ZINC000217987382 CE For-Sale Unstable L3MBTL3 97 44 COc1ccc(OC[C@H](C)NC(=O)[C@H](C)Sc2ccc(Cl)cc2)cc1 ZINC000217987383 GI In-Stock Unstable PTGS2 0 41 COc1ccc(OC[C@H](C)NC(=O)[C@H](C)Sc2ccc(Cl)cc2)cc1 ZINC000217987383 GI In-Stock Unstable SDH1 0 41 Cc1cccc(NC(=O)N/C=C/c2cccc(F)c2)n1 ZINC000217987415 CG For-Sale Unstable GRM5 22 49 Cc1cccc(NC(=O)N/C=C/c2cccc(F)c2)n1 ZINC000217987415 CG For-Sale Unstable SORT1 16 40 CC[C@H](C(=O)N[C@H](CC(=O)OC(C)C)c1ccccc1[N+](=O)[O-])c1ccccc1 ZINC000217987416 GI On-Demand Unstable COLA 91 34 COC(=O)C[C@@H](c1ccc(OCCc2ccc(OC)cc2)c(OC)c1)c1c(O)c2ccccc2oc1=O ZINC000217987443 KJ In-Stock Unstable NQO1 41 52 COC(=O)C[C@@H](c1ccc(OCCc2ccc(OC)cc2)c(OC)c1)c1c(O)c2ccccc2oc1=O ZINC000217987443 KJ In-Stock Unstable ABCG2 25 41 Cc1ccc(OCCNC(=O)[C@@H](C)Sc2ccc(Cl)cc2)cc1 ZINC000217987482 EI In-Stock Unstable PTGES 0 45 Cc1c(CN)c(=O)[nH]c2ccccc12 ZINC000217987511 AD In-Stock Unstable PTGS2 51 34 Cn1ccnc1CCNC(=O)c1ccc(N2CCCCC2)cc1 ZINC000217987534 DE In-Stock Unstable HTR1A 15 43 Cn1ccnc1CCNC(=O)c1ccc(N2CCCCC2)cc1 ZINC000217987534 DE In-Stock Unstable DRD2 20 43 Cn1ccnc1CCNC(=O)c1ccc(N2CCCCC2)cc1 ZINC000217987534 DE In-Stock Unstable DRD4 46 38 Cn1ccnc1CCNC(=O)c1ccc(N2CCCCC2)cc1 ZINC000217987534 DE In-Stock Unstable HTR2A 16 41 Cn1ccnc1CCNC(=O)c1ccc(N2CCCCC2)cc1 ZINC000217987534 DE In-Stock Unstable DRD3 29 41 Cn1ccnc1CCNC(=O)c1ccc(N2CCCCC2)cc1 ZINC000217987534 DE In-Stock Unstable CTSK 15 42 Cn1ccnc1CCNC(=O)c1ccc(N2CCCCC2)cc1 ZINC000217987534 DE In-Stock Unstable PRNP 51 38 COc1ccc(-c2cc(C(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)[nH]n2)cc1OC ZINC000217987555 HF In-Stock Unstable CHRNA4 27 43 COc1ccc(-c2cc(C(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)[nH]n2)cc1OC ZINC000217987555 HF In-Stock Unstable TACR3 21 42 Cc1ccc(OCCNC(=O)[C@H](C)Sc2ccc(Cl)cc2)cc1 ZINC000217987559 EI In-Stock Unstable PTGES 0 45 COCCn1c(C)cc(C)c(C(=O)N2CCCC[C@H]2c2cccnc2)c1=O ZINC000217987652 FF In-Stock Unstable CHRNA2 41 43 COCCn1c(C)cc(C)c(C(=O)N2CCCC[C@H]2c2cccnc2)c1=O ZINC000217987652 FF In-Stock Unstable CPT1A 65 34 COCCn1c(C)cc(C)c(C(=O)N2CCCC[C@H]2c2cccnc2)c1=O ZINC000217987652 FF In-Stock Unstable CRTY 0 43 CCCc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217987657 HG For-Sale Unstable FKBP1A 24 41 CCCc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217987657 HG For-Sale Unstable MMP13 65 46 CCCc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217987657 HG For-Sale Unstable ADAM17 42 41 CCCc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217987657 HG For-Sale Unstable MMP2 33 46 CCCc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217987657 HG For-Sale Unstable MMP3 75 46 CCCc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217987657 HG For-Sale Unstable MMP9 34 41 CCCc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217987657 HG For-Sale Unstable MMP7 75 41 CCCc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217987657 HG For-Sale Unstable MMP1 67 46 C[C@H]1Cc2ccccc2N([C@@H]2C[C@H](C)CC[C@@H]2C(=O)O)C1 ZINC000217987714 CH For-Sale Unstable TPP2 43 31 CCCc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217987731 HG For-Sale Unstable FKBP1A 24 41 CCCc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217987731 HG For-Sale Unstable MMP13 65 46 CCCc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217987731 HG For-Sale Unstable ADAM17 42 41 CCCc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217987731 HG For-Sale Unstable MMP2 33 46 CCCc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217987731 HG For-Sale Unstable MMP3 75 46 CCCc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217987731 HG For-Sale Unstable MMP9 34 41 CCCc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217987731 HG For-Sale Unstable MMP7 75 41 CCCc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217987731 HG For-Sale Unstable MMP1 67 46 O=C(N[C@@H](c1ccc(F)cc1)[C@@H]1C[C@H](O)C1)c1ccc2[nH]ccc2c1 ZINC000217987746 EH In-Stock Unstable AKT1 22 40 O=C(N[C@@H](c1ccc(F)cc1)[C@@H]1C[C@H](O)C1)c1ccc2[nH]ccc2c1 ZINC000217987746 EH In-Stock Unstable TTK 30 41 COc1ccc2cnn(CC(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)c(=O)c2c1OC ZINC000217987768 ID In-Stock Unstable CHRNA4 26 42 C[C@H]1CC[C@H](C(=O)O)[C@H](N2C[C@@H](C)Cc3ccccc32)C1 ZINC000217987790 CH For-Sale Unstable TPP2 43 31 CC(C)Oc1cccc(CCCNC(=O)[C@@H](C)Sc2ccc(Cl)cc2)c1 ZINC000217987825 GK In-Stock Unstable FDFT1 0 48 CC(C)Oc1cccc(CCCNC(=O)[C@@H](C)Sc2ccc(Cl)cc2)c1 ZINC000217987825 GK In-Stock Unstable MTNR1A 26 47 CC(C)Oc1cccc(CCCNC(=O)[C@@H](C)Sc2ccc(Cl)cc2)c1 ZINC000217987825 GK In-Stock Unstable MTNR1B 27 47 CC(C)Oc1cccc(CCCNC(=O)[C@@H](C)Sc2ccc(Cl)cc2)c1 ZINC000217987825 GK In-Stock Unstable AMP1_PLAFQ 38 42 CC(C)Oc1cccc(CCCNC(=O)[C@@H](C)Sc2ccc(Cl)cc2)c1 ZINC000217987825 GK In-Stock Unstable CRTM 66 48 CC(C)Oc1cccc(CCCNC(=O)[C@@H](C)Sc2ccc(Cl)cc2)c1 ZINC000217987825 GK In-Stock Unstable PDS 68 38 O=C(N[C@H](c1ccc(F)cc1)[C@@H]1C[C@H](O)C1)c1ccc2[nH]ccc2c1 ZINC000217987832 EH In-Stock Unstable AKT1 22 40 O=C(N[C@H](c1ccc(F)cc1)[C@@H]1C[C@H](O)C1)c1ccc2[nH]ccc2c1 ZINC000217987832 EH In-Stock Unstable TTK 30 41 C[C@H]1Cc2ccccc2N([C@@H]2C[C@H](C)CC[C@H]2C(=O)O)C1 ZINC000217987868 CH For-Sale Unstable TPP2 43 31 CC(C)Oc1cccc(CCCNC(=O)[C@H](C)Sc2ccc(Cl)cc2)c1 ZINC000217987906 GK In-Stock Unstable FDFT1 0 48 CC(C)Oc1cccc(CCCNC(=O)[C@H](C)Sc2ccc(Cl)cc2)c1 ZINC000217987906 GK In-Stock Unstable MTNR1A 26 47 CC(C)Oc1cccc(CCCNC(=O)[C@H](C)Sc2ccc(Cl)cc2)c1 ZINC000217987906 GK In-Stock Unstable MTNR1B 27 47 CC(C)Oc1cccc(CCCNC(=O)[C@H](C)Sc2ccc(Cl)cc2)c1 ZINC000217987906 GK In-Stock Unstable AMP1_PLAFQ 38 42 CC(C)Oc1cccc(CCCNC(=O)[C@H](C)Sc2ccc(Cl)cc2)c1 ZINC000217987906 GK In-Stock Unstable CRTM 66 48 CC(C)Oc1cccc(CCCNC(=O)[C@H](C)Sc2ccc(Cl)cc2)c1 ZINC000217987906 GK In-Stock Unstable PDS 68 38 O=C(O)c1cccc(N[C@@H]2C[C@@H]3CC=C[C@H]32)c1 ZINC000217987913 BF For-Sale Unstable AKR1C3 47 44 O=C(COc1ccccc1Cl)NC1CCN(C(=O)N2CCCC2)CC1 ZINC000217987933 FF In-Stock Unstable EPHX2 32 45 O=C(COc1ccccc1Cl)NC1CCN(C(=O)N2CCCC2)CC1 ZINC000217987933 FF In-Stock Unstable LUXN 0 42 O=C(COc1ccccc1Cl)NC1CCN(C(=O)N2CCCC2)CC1 ZINC000217987933 FF In-Stock Unstable ADIPOR1 0 45 O=C(COc1ccccc1Cl)NC1CCN(C(=O)N2CCCC2)CC1 ZINC000217987933 FF In-Stock Unstable ADIPOR2 0 45 C[C@H]1CC[C@@H](C(=O)O)[C@H](N2C[C@@H](C)Cc3ccccc32)C1 ZINC000217987939 CH For-Sale Unstable TPP2 43 31 O=C(O)c1cccc(N[C@H]2C[C@@H]3CC=C[C@H]32)c1 ZINC000217987986 BF For-Sale Unstable AKR1C3 47 44 CC[C@H](C(=O)O)N1C[C@@H](C)Cc2ccccc21 ZINC000217988023 BF For-Sale Unstable ACE 32 43 CC[C@H](C(=O)O)N1C[C@@H](C)Cc2ccccc21 ZINC000217988023 BF For-Sale Unstable KCNQ2 45 33 CC[C@H](C(=O)O)N1C[C@@H](C)Cc2ccccc21 ZINC000217988023 BF For-Sale Unstable TPP2 61 39 Cc1ccc(S(=O)(=O)N2CCC(NC(=O)c3cc(N4CCCC4)ccn3)CC2)cc1 ZINC000217988042 IF On-Demand Unstable CNR1 15 42 Cc1ccc(S(=O)(=O)N2CCC(NC(=O)c3cc(N4CCCC4)ccn3)CC2)cc1 ZINC000217988042 IF On-Demand Unstable EPHX2 41 58 Cc1ccc(S(=O)(=O)N2CCC(NC(=O)c3cc(N4CCCC4)ccn3)CC2)cc1 ZINC000217988042 IF On-Demand Unstable TGM2 54 41 Cc1ccc(S(=O)(=O)N2CCC(NC(=O)c3cc(N4CCCC4)ccn3)CC2)cc1 ZINC000217988042 IF On-Demand Unstable FPR1 15 40 Cc1ccc(S(=O)(=O)N2CCC(NC(=O)c3cc(N4CCCC4)ccn3)CC2)cc1 ZINC000217988042 IF On-Demand Unstable F13A1 43 36 CC(=O)NCC1CCN(c2cc(Cl)nc(C3CC3)n2)CC1 ZINC000217988055 DE On-Demand Unstable CACNA1I 46 34 C=C(C)COc1cc([C@@H](CC(=O)OC)c2c(O)c3ccccc3oc2=O)ccc1OC ZINC000217988066 HI In-Stock Unstable NQO1 46 46 O=C(O)c1cccc(N[C@@H]2C[C@H]3CC=C[C@H]32)c1 ZINC000217988075 BF For-Sale Unstable AKR1C3 47 44 CC[C@@H](C(=O)O)N1C[C@@H](C)Cc2ccccc21 ZINC000217988121 BF For-Sale Unstable ACE 32 43 CC[C@@H](C(=O)O)N1C[C@@H](C)Cc2ccccc21 ZINC000217988121 BF For-Sale Unstable KCNQ2 45 33 CC[C@@H](C(=O)O)N1C[C@@H](C)Cc2ccccc21 ZINC000217988121 BF For-Sale Unstable TPP2 61 39 C=C(C)COc1cc([C@H](CC(=O)OC)c2c(O)c3ccccc3oc2=O)ccc1OC ZINC000217988139 HI In-Stock Unstable NQO1 46 46 O=C(O)c1cccc(N[C@H]2C[C@H]3CC=C[C@@H]23)c1 ZINC000217988152 BF For-Sale Unstable AKR1C3 47 44 COc1ccc(/C=C2/C[C@@H](C)Cc3c2nc2ccccc2c3C(=O)N(CC(N)=O)C(C)C)cc1 ZINC000217988165 JJ On-Demand Unstable TACR3 40 34 CCO[C@@H](CN1C[C@@H](C)Cc2ccccc21)C(=O)O ZINC000217988213 CE For-Sale Unstable TPP2 61 36 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(C)C)cc1 ZINC000217988227 HG For-Sale Unstable MMP13 52 39 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(C)C)cc1 ZINC000217988227 HG For-Sale Unstable MMP2 26 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(C)C)cc1 ZINC000217988227 HG For-Sale Unstable MMP3 64 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(C)C)cc1 ZINC000217988227 HG For-Sale Unstable MMP7 55 37 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(C)C)cc1 ZINC000217988227 HG For-Sale Unstable MMP1 53 40 C[C@@H](Sc1ccc(Cl)cc1)C(=O)Nc1ccc(OC2CCCC2)cc1 ZINC000217988238 GK In-Stock Unstable EPHX2 22 47 COC(=O)C[C@H](c1ccccc1)c1oc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c1O ZINC000217988243 JF In-Stock Unstable CHRNA4 29 49 COc1ccc(/C=C2/C[C@H](C)Cc3c2nc2ccccc2c3C(=O)N(CC(N)=O)C(C)C)cc1 ZINC000217988255 JJ On-Demand Unstable TACR3 40 34 CCO[C@H](CN1C[C@@H](C)Cc2ccccc21)C(=O)O ZINC000217988292 CE For-Sale Unstable TPP2 61 36 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(C)C)cc1 ZINC000217988317 HG For-Sale Unstable MMP13 52 39 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(C)C)cc1 ZINC000217988317 HG For-Sale Unstable MMP2 26 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(C)C)cc1 ZINC000217988317 HG For-Sale Unstable MMP3 64 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(C)C)cc1 ZINC000217988317 HG For-Sale Unstable MMP7 55 37 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(C)C)cc1 ZINC000217988317 HG For-Sale Unstable MMP1 53 40 C[C@H](Sc1ccc(Cl)cc1)C(=O)Nc1ccc(OC2CCCC2)cc1 ZINC000217988323 GK In-Stock Unstable EPHX2 22 47 COC(=O)C[C@@H](c1ccccc1)c1oc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c1O ZINC000217988327 JF In-Stock Unstable CHRNA4 29 49 CCO[C@@H](CCN1C[C@@H](C)Cc2ccccc21)C(=O)O ZINC000217988369 CF For-Sale Unstable TPP2 60 35 C[C@H]1c2ccsc2CCN1[C@H](C)c1ccc(C(=O)O)o1 ZINC000217988438 CH For-Sale Unstable TRPM8 17 40 COC(=O)C[C@H](c1cc(OC)c(OC(C)=O)c(OC)c1)c1oc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c1O ZINC000217988455 KF In-Stock Unstable CHRNA4 25 41 CCO[C@H](CCN1C[C@@H](C)Cc2ccccc21)C(=O)O ZINC000217988456 CF For-Sale Unstable TPP2 60 35 COC(=O)c1ccc([C@@H](C)N2CCc3sccc3[C@@H]2C)o1 ZINC000217988524 DH For-Sale Unstable TRPM8 17 42 COC(=O)C[C@@H](c1cc(OC)c(OC(C)=O)c(OC)c1)c1oc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c1O ZINC000217988544 KF In-Stock Unstable CHRNA4 25 41 C[C@H]1Cc2ccccc2N([C@H](C)C(=O)O)C1 ZINC000217988569 BE For-Sale Unstable ACE 29 45 C[C@H]1Cc2ccccc2N([C@H](C)C(=O)O)C1 ZINC000217988569 BE For-Sale Unstable TPP2 53 32 CC(=O)Nc1cccc(NC(=O)N/C=C/c2cccc(F)c2)c1 ZINC000217988601 DH For-Sale Unstable IMPDH2 0 41 CC(=O)Nc1cccc(NC(=O)N/C=C/c2cccc(F)c2)c1 ZINC000217988601 DH For-Sale Unstable IDO1 16 45 CC(=O)Nc1cccc(NC(=O)N/C=C/c2cccc(F)c2)c1 ZINC000217988601 DH For-Sale Unstable KCNK3 67 43 CC(=O)Nc1cccc(NC(=O)N/C=C/c2cccc(F)c2)c1 ZINC000217988601 DH For-Sale Unstable KCNK9 45 43 C[C@@](O)(CNC(=O)c1nc2ccccc2s1)c1cc2ccccc2o1 ZINC000217988603 FH In-Stock Unstable TMPRSS6 47 32 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1ccc(SC(F)F)cc1 ZINC000217988626 DK For-Sale Unstable TRPM8 15 42 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(C)c1 ZINC000217988628 HF For-Sale Unstable MMP13 48 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(C)c1 ZINC000217988628 HF For-Sale Unstable ADAM17 26 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(C)c1 ZINC000217988628 HF For-Sale Unstable MMP2 23 52 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(C)c1 ZINC000217988628 HF For-Sale Unstable MMP3 60 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(C)c1 ZINC000217988628 HF For-Sale Unstable MMP9 31 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(C)c1 ZINC000217988628 HF For-Sale Unstable MMP7 53 38 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(C)c1 ZINC000217988628 HF For-Sale Unstable MMP1 51 40 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)N3CCN(Cc4nc5ccccc5c(=O)[nH]4)CC3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217988661 KF In-Stock Unstable TUBA1A 15 55 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)N3CCN(Cc4nc5ccccc5c(=O)[nH]4)CC3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217988661 KF In-Stock Unstable TPPP 0 52 CC[C@@H](CC(=O)O)N1C[C@@H](C)Cc2ccccc21 ZINC000217988663 BF For-Sale Unstable ACE 29 46 CC[C@@H](CC(=O)O)N1C[C@@H](C)Cc2ccccc21 ZINC000217988663 BF For-Sale Unstable TPP2 60 38 C[C@](O)(CNC(=O)c1nc2ccccc2s1)c1cc2ccccc2o1 ZINC000217988681 FH In-Stock Unstable TMPRSS6 47 32 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1ccc(SC(F)F)cc1 ZINC000217988707 DK For-Sale Unstable TRPM8 15 42 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(C)c1 ZINC000217988716 HF For-Sale Unstable MMP13 48 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(C)c1 ZINC000217988716 HF For-Sale Unstable ADAM17 26 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(C)c1 ZINC000217988716 HF For-Sale Unstable MMP2 23 52 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(C)c1 ZINC000217988716 HF For-Sale Unstable MMP3 60 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(C)c1 ZINC000217988716 HF For-Sale Unstable MMP9 31 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(C)c1 ZINC000217988716 HF For-Sale Unstable MMP7 53 38 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(C)c1 ZINC000217988716 HF For-Sale Unstable MMP1 51 40 CC[C@H](CC(=O)O)N1C[C@@H](C)Cc2ccccc21 ZINC000217988745 BF For-Sale Unstable ACE 29 46 CC[C@H](CC(=O)O)N1C[C@@H](C)Cc2ccccc21 ZINC000217988745 BF For-Sale Unstable TPP2 60 38 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1ccc(SC(F)F)cc1 ZINC000217988771 DK For-Sale Unstable TRPM8 15 42 CCOc1ccc(CCCNC(=O)[C@@H](C)Sc2ccc(Cl)cc2)cc1 ZINC000217988792 GJ In-Stock Unstable SCN2A 18 41 CCOc1ccc(CCCNC(=O)[C@@H](C)Sc2ccc(Cl)cc2)cc1 ZINC000217988792 GJ In-Stock Unstable PDS 43 37 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1cc(C)ccc1OC ZINC000217988814 HF For-Sale Unstable CPT1A 40 38 C[C@H]1Cc2ccccc2N([C@H](C)CC(=O)O)C1 ZINC000217988831 BF For-Sale Unstable ACE 33 46 C[C@H]1Cc2ccccc2N([C@H](C)CC(=O)O)C1 ZINC000217988831 BF For-Sale Unstable TPP2 57 34 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1ccc(SC(F)F)cc1 ZINC000217988847 DK For-Sale Unstable TRPM8 15 42 CCOc1ccc(CCCNC(=O)[C@H](C)Sc2ccc(Cl)cc2)cc1 ZINC000217988865 GJ In-Stock Unstable SCN2A 18 41 CCOc1ccc(CCCNC(=O)[C@H](C)Sc2ccc(Cl)cc2)cc1 ZINC000217988865 GJ In-Stock Unstable PDS 43 37 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1cc(C)ccc1OC ZINC000217988892 HF For-Sale Unstable CPT1A 40 38 C[C@H]1Cc2ccccc2N(C[C@H](C)C(=O)O)C1 ZINC000217988932 BE For-Sale Unstable ACE 56 49 C[C@H]1Cc2ccccc2N(C[C@H](C)C(=O)O)C1 ZINC000217988932 BE For-Sale Unstable TPP2 60 35 CCCOc1ccccc1CCCNC(=O)[C@@H](C)Sc1ccc(Cl)cc1 ZINC000217988966 GK In-Stock Unstable MTNR1A 27 44 CCCOc1ccccc1CCCNC(=O)[C@@H](C)Sc1ccc(Cl)cc1 ZINC000217988966 GK In-Stock Unstable MTNR1B 28 44 O=C(c1cc(-c2ccc3c(c2)CCO3)n[nH]1)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000217988976 HE In-Stock Unstable CHRNA4 25 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)cc1C ZINC000217989000 HF For-Sale Unstable MMP2 17 47 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)cc1C ZINC000217989000 HF For-Sale Unstable MMP3 42 38 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)cc1C ZINC000217989000 HF For-Sale Unstable MMP7 46 35 CCCOc1ccccc1CCCNC(=O)[C@H](C)Sc1ccc(Cl)cc1 ZINC000217989052 GK In-Stock Unstable MTNR1A 27 44 CCCOc1ccccc1CCCNC(=O)[C@H](C)Sc1ccc(Cl)cc1 ZINC000217989052 GK In-Stock Unstable MTNR1B 28 44 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)cc1C ZINC000217989072 HF For-Sale Unstable MMP2 17 47 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)cc1C ZINC000217989072 HF For-Sale Unstable MMP3 42 38 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)cc1C ZINC000217989072 HF For-Sale Unstable MMP7 46 35 CC(=O)c1ccc(S(=O)(=O)NCCC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217989084 HF On-Demand Unstable TBXA2R 50 39 CC(=O)c1ccc(S(=O)(=O)NCCC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217989084 HF On-Demand Unstable MMP13 23 41 CC(=O)c1ccc(S(=O)(=O)NCCC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217989084 HF On-Demand Unstable MMP2 23 41 CC(=O)c1ccc(S(=O)(=O)NCCC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217989084 HF On-Demand Unstable ADAMTS4 49 41 CC(=O)c1ccc(S(=O)(=O)NCCC(=O)N(Cc2ccccc2)C(C)C)cc1 ZINC000217989084 HF On-Demand Unstable LIMK2 51 45 COc1ccc(CCCNC(=O)[C@@H](C)Sc2ccc(Cl)cc2)cc1OC ZINC000217989159 GJ In-Stock Unstable TRPV1 0 48 COc1ccc(CCCNC(=O)[C@@H](C)Sc2ccc(Cl)cc2)cc1OC ZINC000217989159 GJ In-Stock Unstable MTNR1B 15 47 COc1ccc(CCCNC(=O)[C@@H](C)Sc2ccc(Cl)cc2)cc1OC ZINC000217989159 GJ In-Stock Unstable CAN2 0 47 Cc1c([C@@H](C)C(=O)O)ccc(O)c1Br ZINC000217989161 CF For-Sale Unstable PTGS1 21 45 Cc1c([C@@H](C)C(=O)O)ccc(O)c1Br ZINC000217989161 CF For-Sale Unstable PTGS2 16 45 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(F)c1 ZINC000217989179 IE For-Sale Unstable MMP13 41 39 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(F)c1 ZINC000217989179 IE For-Sale Unstable MMP2 20 54 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(F)c1 ZINC000217989179 IE For-Sale Unstable MMP3 53 39 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(F)c1 ZINC000217989179 IE For-Sale Unstable MMP7 49 37 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(F)c1 ZINC000217989179 IE For-Sale Unstable MMP1 45 39 Cc1c([C@H](C)C(=O)O)ccc(O)c1Br ZINC000217989221 CF For-Sale Unstable PTGS1 21 45 Cc1c([C@H](C)C(=O)O)ccc(O)c1Br ZINC000217989221 CF For-Sale Unstable PTGS2 16 45 COc1ccc(CCCNC(=O)[C@H](C)Sc2ccc(Cl)cc2)cc1OC ZINC000217989235 GJ In-Stock Unstable TRPV1 0 48 COc1ccc(CCCNC(=O)[C@H](C)Sc2ccc(Cl)cc2)cc1OC ZINC000217989235 GJ In-Stock Unstable MTNR1B 15 47 COc1ccc(CCCNC(=O)[C@H](C)Sc2ccc(Cl)cc2)cc1OC ZINC000217989235 GJ In-Stock Unstable CAN2 0 47 C=C(CCCC)[C@H](O)CC ZINC000217989243 AF For-Sale Unstable CQSS 70 50 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(F)c1 ZINC000217989270 IE For-Sale Unstable MMP13 41 39 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(F)c1 ZINC000217989270 IE For-Sale Unstable MMP2 20 54 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(F)c1 ZINC000217989270 IE For-Sale Unstable MMP3 53 39 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(F)c1 ZINC000217989270 IE For-Sale Unstable MMP7 49 37 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(F)c1 ZINC000217989270 IE For-Sale Unstable MMP1 45 39 O=C(COc1cccc(Cl)c1)N[C@H]1CCC[C@H]1CO ZINC000217989332 CD On-Demand Unstable ADIPOR1 0 40 O=C(COc1cccc(Cl)c1)N[C@H]1CCC[C@H]1CO ZINC000217989332 CD On-Demand Unstable ADIPOR2 0 40 Clc1cc2c(cc1Br)OCOC2 ZINC000217989335 BF For-Sale Unstable AHR 15 47 Cc1c(O)cc([C@@H](C)C(=O)O)cc1Br ZINC000217989336 CF For-Sale Unstable PTGS1 19 48 Cc1ccccc1OC[C@@H](C)NC(=O)[C@@H](C)Sc1ccc(Cl)cc1 ZINC000217989363 FJ In-Stock Unstable SDH1 0 43 O=C(Nc1nc2ccccc2[nH]1)[C@@H]1CC[C@@H](Cn2cnnn2)CC1 ZINC000217989385 ED In-Stock Unstable KCNN3 41 38 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1cc(F)ccc1OC ZINC000217989389 IE For-Sale Unstable CPT1A 42 39 Cc1c(O)cc([C@H](C)C(=O)O)cc1Br ZINC000217989425 CF For-Sale Unstable PTGS1 19 48 Cc1nnnn1Cc1ccc(C(=O)N[C@@H]2COCC[C@@H]2OCC(N)=O)cc1 ZINC000217989435 FB In-Stock Unstable ADAM17 17 40 COc1ccc2[nH]c3c(c2c1)CCC[C@@H]3NC(=O)c1cn(C)c(=O)c2ccccc12 ZINC000217989439 HH In-Stock Unstable MAPKAPK2 22 49 Cc1ccc(C(=O)N[C@@H]2CCC[C@@H]2CO)cc1 ZINC000217989440 BD On-Demand Unstable PRKCD 0 40 Cc1ccc(C(=O)N[C@@H]2CCC[C@@H]2CO)cc1 ZINC000217989440 BD On-Demand Unstable SSTR3 0 54 Cc1ccc(C(=O)N[C@@H]2CCC[C@@H]2CO)cc1 ZINC000217989440 BD On-Demand Unstable MMP7 0 43 Cc1ccc(C(=O)N[C@@H]2CCC[C@@H]2CO)cc1 ZINC000217989440 BD On-Demand Unstable HSPB1 0 40 Cc1ccccc1OC[C@H](C)NC(=O)[C@@H](C)Sc1ccc(Cl)cc1 ZINC000217989441 FJ In-Stock Unstable SDH1 0 43 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1cc(F)ccc1OC ZINC000217989464 IE For-Sale Unstable CPT1A 42 39 COC(=O)C[C@@H](NC1C[C@@H]2CC[C@@H](C1)N2C)c1cccs1 ZINC000217989469 DF For-Sale Unstable SLC6A1 73 40 COC(=O)C[C@@H](NC1C[C@@H]2CC[C@@H](C1)N2C)c1cccs1 ZINC000217989469 DF For-Sale Unstable SLC6A4 18 40 COC(=O)C[C@@H](NC1C[C@@H]2CC[C@@H](C1)N2C)c1cccs1 ZINC000217989469 DF For-Sale Unstable SLC6A3 42 41 COC(=O)C[C@@H](NC1C[C@@H]2CC[C@@H](C1)N2C)c1cccs1 ZINC000217989469 DF For-Sale Unstable GLRA1 54 46 Cc1ccccc1OC[C@@H](C)NC(=O)[C@H](C)Sc1ccc(Cl)cc1 ZINC000217989508 FJ In-Stock Unstable SDH1 0 43 Cc1ccc(C(=O)N[C@H]2CCC[C@@H]2CO)cc1 ZINC000217989513 BD For-Sale Unstable PRKCD 0 40 Cc1ccc(C(=O)N[C@H]2CCC[C@@H]2CO)cc1 ZINC000217989513 BD For-Sale Unstable SSTR3 28 54 Cc1ccc(C(=O)N[C@H]2CCC[C@@H]2CO)cc1 ZINC000217989513 BD For-Sale Unstable MMP7 0 43 Cc1ccc(C(=O)N[C@H]2CCC[C@@H]2CO)cc1 ZINC000217989513 BD For-Sale Unstable HSPB1 0 40 C[C@@](O)(CNC(=O)COc1ccc(Cl)cc1)c1cc2ccccc2o1 ZINC000217989516 FG In-Stock Unstable CETP 0 40 COc1ccc2[nH]c3c(c2c1)CCC[C@H]3NC(=O)c1cn(C)c(=O)c2ccccc12 ZINC000217989519 HH In-Stock Unstable MAPKAPK2 22 49 COC(=O)C[C@@H](NC1C[C@@H]2CC[C@H](C1)N2C)c1cccs1 ZINC000217989542 DF For-Sale Unstable SLC6A1 73 40 COC(=O)C[C@@H](NC1C[C@@H]2CC[C@H](C1)N2C)c1cccs1 ZINC000217989542 DF For-Sale Unstable SLC6A4 18 40 COC(=O)C[C@@H](NC1C[C@@H]2CC[C@H](C1)N2C)c1cccs1 ZINC000217989542 DF For-Sale Unstable SLC6A3 42 41 COC(=O)C[C@@H](NC1C[C@@H]2CC[C@H](C1)N2C)c1cccs1 ZINC000217989542 DF For-Sale Unstable GLRA1 54 46 C[C@@]12CC3CC(C(=O)NCCc4ccc(-n5cccn5)cc4)(C1)C[C@](C)(C3)C2 ZINC000217989563 GJ On-Demand Unstable AMP1_PLAFQ 52 36 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C)c(Cl)c1 ZINC000217989571 IG For-Sale Unstable MMP13 40 38 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C)c(Cl)c1 ZINC000217989571 IG For-Sale Unstable MMP2 18 50 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C)c(Cl)c1 ZINC000217989571 IG For-Sale Unstable MMP3 43 38 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C)c(Cl)c1 ZINC000217989571 IG For-Sale Unstable MMP7 46 36 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C)c(Cl)c1 ZINC000217989571 IG For-Sale Unstable MMP1 42 38 Cc1ccc(C(=O)N[C@@H]2CCC[C@H]2CO)cc1 ZINC000217989592 BD For-Sale Unstable PRKCD 0 40 Cc1ccc(C(=O)N[C@@H]2CCC[C@H]2CO)cc1 ZINC000217989592 BD For-Sale Unstable SSTR3 28 54 Cc1ccc(C(=O)N[C@@H]2CCC[C@H]2CO)cc1 ZINC000217989592 BD For-Sale Unstable MMP7 0 43 Cc1ccc(C(=O)N[C@@H]2CCC[C@H]2CO)cc1 ZINC000217989592 BD For-Sale Unstable HSPB1 0 40 Cc1ccccc1OC[C@H](C)NC(=O)[C@H](C)Sc1ccc(Cl)cc1 ZINC000217989602 FJ In-Stock Unstable SDH1 0 43 C[C@](O)(CNC(=O)COc1ccc(Cl)cc1)c1cc2ccccc2o1 ZINC000217989618 FG In-Stock Unstable CETP 0 40 COC(=O)COc1cc([C@@H](CC(=O)OC)C2=C(O)C(=O)C([C@H](CC(=O)OC)c3ccc(OC)c(OCC(=O)OC)c3)=C(O)C2=O)ccc1OC ZINC000217989628 KF In-Stock Unstable TNF 22 41 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C)c(Cl)c1 ZINC000217989656 IG For-Sale Unstable MMP13 40 38 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C)c(Cl)c1 ZINC000217989656 IG For-Sale Unstable MMP2 18 50 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C)c(Cl)c1 ZINC000217989656 IG For-Sale Unstable MMP3 43 38 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C)c(Cl)c1 ZINC000217989656 IG For-Sale Unstable MMP7 46 36 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C)c(Cl)c1 ZINC000217989656 IG For-Sale Unstable MMP1 42 38 Cc1ccc(C(=O)N[C@H]2CCC[C@H]2CO)cc1 ZINC000217989684 BD For-Sale Unstable PRKCD 0 40 Cc1ccc(C(=O)N[C@H]2CCC[C@H]2CO)cc1 ZINC000217989684 BD For-Sale Unstable SSTR3 28 54 Cc1ccc(C(=O)N[C@H]2CCC[C@H]2CO)cc1 ZINC000217989684 BD For-Sale Unstable MMP7 0 43 Cc1ccc(C(=O)N[C@H]2CCC[C@H]2CO)cc1 ZINC000217989684 BD For-Sale Unstable HSPB1 0 40 Cc1ccc(OC[C@@H](C)NC(=O)[C@@H](C)Sc2ccc(Cl)cc2)cc1 ZINC000217989699 FJ In-Stock Unstable SDH1 0 41 COC(=O)COc1cc([C@H](CC(=O)OC)C2=C(O)C(=O)C([C@H](CC(=O)OC)c3ccc(OC)c(OCC(=O)OC)c3)=C(O)C2=O)ccc1OC ZINC000217989709 KF In-Stock Unstable TNF 22 41 C[C@@](O)(CNC(=O)c1ccccc1C(F)(F)F)c1cc2ccccc2o1 ZINC000217989720 FI In-Stock Unstable KCNJ11 59 32 Cc1cc([C@@H](C)C(=O)O)cc(O)c1Br ZINC000217989730 CF For-Sale Unstable PTGS1 19 40 Cc1ccc(OC[C@H](C)NC(=O)[C@@H](C)Sc2ccc(Cl)cc2)cc1 ZINC000217989783 FJ In-Stock Unstable SDH1 0 41 C[C@](O)(CNC(=O)c1ccccc1C(F)(F)F)c1cc2ccccc2o1 ZINC000217989786 FI In-Stock Unstable KCNJ11 59 32 COC(=O)COc1cc([C@H](CC(=O)OC)C2=C(O)C(=O)C([C@@H](CC(=O)OC)c3ccc(OC)c(OCC(=O)OC)c3)=C(O)C2=O)ccc1OC ZINC000217989796 KF In-Stock Unstable TNF 22 41 Cc1cc([C@H](C)C(=O)O)cc(O)c1Br ZINC000217989805 CF For-Sale Unstable PTGS1 19 40 O=C(N/C=C/c1cccc(F)c1)Nc1ccccc1N1CCOCC1 ZINC000217989826 EG For-Sale Unstable KCNQ2 84 47 O=C(N/C=C/c1cccc(F)c1)Nc1ccccc1N1CCOCC1 ZINC000217989826 EG For-Sale Unstable CSF1R 0 44 Cc1ccc(OC[C@@H](C)NC(=O)[C@H](C)Sc2ccc(Cl)cc2)cc1 ZINC000217989873 FJ In-Stock Unstable SDH1 0 41 C[C@@](O)(CNC(=O)c1cc(=O)c2ccccc2o1)c1cc2ccccc2o1 ZINC000217989886 FG In-Stock Unstable KCNJ11 61 32 C[C@@](O)(CNC(=O)c1cc(=O)c2ccccc2o1)c1cc2ccccc2o1 ZINC000217989886 FG In-Stock Unstable BCHE 28 43 O=C(NCCc1ccc(Br)s1)c1ccnc2ccccc12 ZINC000217989896 FI On-Demand Unstable PREP 22 43 O=C(NCCc1ccc(Br)s1)c1ccnc2ccccc12 ZINC000217989896 FI On-Demand Unstable FAP 0 48 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@H](C)C(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217989907 KG In-Stock Unstable TUBA1A 17 60 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@H](C)C(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217989907 KG In-Stock Unstable TPPP 0 57 COC(=O)c1ccc(COc2ccccc2OC)c(Br)c1 ZINC000217989922 FH On-Demand Unstable ACR 31 40 COC(=O)c1ccc(COc2ccccc2OC)c(Br)c1 ZINC000217989922 FH On-Demand Unstable MT-CYB 47 34 COc1ccccc1CCC(=O)N[C@@H]1C[C@H](c2nnc(CO)n2C)C1 ZINC000217989923 ED In-Stock Unstable MBTPS1 40 31 CN1CCN(c2ccc(NC(=O)N/C=C/c3cccc(F)c3)cc2)CC1 ZINC000217989933 FG For-Sale Unstable HTR1B 16 42 CN1CCN(c2ccc(NC(=O)N/C=C/c3cccc(F)c3)cc2)CC1 ZINC000217989933 FG For-Sale Unstable PRNP 37 44 Cc1ccc(OC[C@H](C)NC(=O)[C@H](C)Sc2ccc(Cl)cc2)cc1 ZINC000217989956 FJ In-Stock Unstable SDH1 0 41 C[C@](O)(CNC(=O)c1cc(=O)c2ccccc2o1)c1cc2ccccc2o1 ZINC000217989965 FG In-Stock Unstable KCNJ11 61 32 C[C@](O)(CNC(=O)c1cc(=O)c2ccccc2o1)c1cc2ccccc2o1 ZINC000217989965 FG In-Stock Unstable BCHE 28 43 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(N2CCCCC2)cc1 ZINC000217990059 EJ For-Sale Unstable IMPDH2 0 41 CC1CCN(c2ccc([C@@H](C)NC(=O)[C@@H](C)Sc3ccc(Cl)cc3)cc2)CC1 ZINC000217990079 HK In-Stock Unstable SDH1 0 40 CC1CCN(c2ccc([C@@H](C)NC(=O)[C@@H](C)Sc3ccc(Cl)cc3)cc2)CC1 ZINC000217990079 HK In-Stock Unstable ADAM17 0 41 CCCCc1ccc(NC(=O)[C@@H]2CC[C@@H](Cn3cnnn3)CC2)cc1 ZINC000217990121 EG In-Stock Unstable CFTR 42 37 C=C(C)/C=C\CC[C@H](NC(=O)OC(C)(C)C)C(=O)OC ZINC000217990149 CF For-Sale Unstable PAPA1_CARPA 35 41 C=C(C)/C=C\CC[C@H](NC(=O)OC(C)(C)C)C(=O)OC ZINC000217990149 CF For-Sale Unstable CTSK 17 46 CC1CCN(c2ccc([C@H](C)NC(=O)[C@@H](C)Sc3ccc(Cl)cc3)cc2)CC1 ZINC000217990173 HK In-Stock Unstable SDH1 0 40 CC1CCN(c2ccc([C@H](C)NC(=O)[C@@H](C)Sc3ccc(Cl)cc3)cc2)CC1 ZINC000217990173 HK In-Stock Unstable ADAM17 0 41 C=C(C)/C=C\CC[C@@H](NC(=O)OC(C)(C)C)C(=O)OC ZINC000217990231 CF For-Sale Unstable PAPA1_CARPA 35 41 C=C(C)/C=C\CC[C@@H](NC(=O)OC(C)(C)C)C(=O)OC ZINC000217990231 CF For-Sale Unstable CTSK 17 46 CC1CCN(c2ccc([C@@H](C)NC(=O)[C@H](C)Sc3ccc(Cl)cc3)cc2)CC1 ZINC000217990249 HK In-Stock Unstable SDH1 0 40 CC1CCN(c2ccc([C@@H](C)NC(=O)[C@H](C)Sc3ccc(Cl)cc3)cc2)CC1 ZINC000217990249 HK In-Stock Unstable ADAM17 0 41 O=C(c1cc(N2CCOCC2)ccn1)N1CCN(Cc2nc(-c3cccs3)no2)CC1 ZINC000217990252 ID On-Demand Unstable ETHR 30 40 C[C@@H](c1ccc(C(=O)O)o1)N1CC[C@@H](c2ccccc2)C1 ZINC000217990294 CH On-Demand Unstable CCR5 61 35 C=C(C)/C=C/CC[C@@H](NC(=O)OC(C)(C)C)C(=O)OC ZINC000217990304 CF For-Sale Unstable PAPA1_CARPA 35 41 C=C(C)/C=C/CC[C@@H](NC(=O)OC(C)(C)C)C(=O)OC ZINC000217990304 CF For-Sale Unstable CTSK 17 46 CCc1ncnc(NCc2ccc(F)c(F)c2)c1F ZINC000217990315 CG On-Demand Unstable USP10 0 41 CCc1ncnc(NCc2ccc(F)c(F)c2)c1F ZINC000217990315 CG On-Demand Unstable USP13 0 41 COc1cc2c(c(OC)c1OC)-c1ccc(NCCCCCC(=O)NCCCCCC(=O)O)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217990327 KJ In-Stock Unstable TUBA1A 18 68 CC1CCN(c2ccc([C@H](C)NC(=O)[C@H](C)Sc3ccc(Cl)cc3)cc2)CC1 ZINC000217990334 HK In-Stock Unstable SDH1 0 40 CC1CCN(c2ccc([C@H](C)NC(=O)[C@H](C)Sc3ccc(Cl)cc3)cc2)CC1 ZINC000217990334 HK In-Stock Unstable ADAM17 0 41 C[C@H](c1ccc(C(=O)O)o1)N1CC[C@@H](c2ccccc2)C1 ZINC000217990373 CH On-Demand Unstable CCR5 61 35 O=C(c1cc(N2CCCC2)ccn1)N1CCN(Cc2nc(-c3cccs3)no2)CC1 ZINC000217990379 HF On-Demand Unstable ETHR 41 41 C[C@@H]1CCCN(c2ccc([C@@H](C)NC(=O)[C@@H](C)Sc3ccc(Cl)cc3)cc2)C1 ZINC000217990425 HK In-Stock Unstable ADAM17 0 43 O=C(NCC(=O)N1CCN(Cc2nc(-c3cccs3)no2)CC1)c1ccc(Br)cc1 ZINC000217990490 JF On-Demand Unstable ETHR 49 46 O=C(N/C=C/c1cccc(F)c1)Nc1cccc2ccccc12 ZINC000217990495 DJ For-Sale Anodyne TRPV1 27 47 CC(C)c1ccc(C(=O)N[C@@H]2CCC[C@@H]2CO)cc1 ZINC000217990501 CF On-Demand Unstable SSTR3 28 41 C[C@H](NC(=O)[C@@H](C)Sc1ccc(Cl)cc1)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217990510 HK In-Stock Unstable ADAM17 0 43 c1ccc(-c2nnc3ccccc3n2)nc1 ZINC000217990511 BE For-Sale Anodyne METAP1 34 44 c1ccc(-c2nnc3ccccc3n2)nc1 ZINC000217990511 BE For-Sale Anodyne LUCI_PHOPE 23 41 CC(C)c1ccc(C(=O)N[C@H]2CCC[C@@H]2CO)cc1 ZINC000217990572 CF For-Sale Unstable SSTR3 29 41 C[C@H](Sc1ccc(Cl)cc1)C(=O)N[C@H](C)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217990583 HK In-Stock Unstable ADAM17 0 43 Cc1nn(C)c(C)c1C(=O)C(=O)N1CCN(Cc2nc(-c3cccs3)no2)CC1 ZINC000217990604 HD On-Demand Unstable ETHR 31 42 COC(=O)c1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217990630 DG For-Sale Unstable ACR 39 40 CCc1ncnc(NC[C@@H]2CCCCO2)c1F ZINC000217990638 BE On-Demand Unstable TNK2 64 43 CCCNCCCCS(=O)(=O)NCc1ccc(C)cc1 ZINC000217990648 CE For-Sale Unstable RELA 19 43 CC(C)c1ccc(C(=O)N[C@@H]2CCC[C@H]2CO)cc1 ZINC000217990649 CF For-Sale Unstable SSTR3 29 41 COc1ccc(O)c(CC(C)=O)c1Br ZINC000217990653 CE For-Sale Unstable TUBB1 42 37 C[C@H](Sc1ccc(Cl)cc1)C(=O)N[C@@H](C)c1ccc(N2CCC[C@@H](C)C2)cc1 ZINC000217990663 HK In-Stock Unstable ADAM17 0 43 O=C(c1nn(-c2ccccc2)cc1O)N1CCN(Cc2nc(-c3cccs3)no2)CC1 ZINC000217990705 IF On-Demand Unstable ETHR 35 41 CCc1ncnc(NC[C@H]2CCCCO2)c1F ZINC000217990727 BE On-Demand Unstable TNK2 64 43 CC(C)c1ccc(C(=O)N[C@H]2CCC[C@H]2CO)cc1 ZINC000217990728 CF For-Sale Unstable SSTR3 29 41 O=C(N/C=C/c1cccc(F)c1)N(Cc1ccccc1)c1ccccc1 ZINC000217990734 EK For-Sale Unstable NR1H4 48 50 COc1cccc(N2CCC(N[C@@H]3CCOC[C@H]3OC)CC2)c1 ZINC000217990739 DE In-Stock Unstable CCR2 36 49 O=C(N/C=C/c1cccc(F)c1)Nc1ccc2ccccc2c1 ZINC000217990830 DJ For-Sale Anodyne IMPDH2 0 42 O=C(N/C=C/c1cccc(F)c1)Nc1ccc2ccccc2c1 ZINC000217990830 DJ For-Sale Anodyne IMDH_CRYPV 28 41 CN1CCC[C@@H]1CNc1cc(Cl)nc(C2CC2)n1 ZINC000217990832 CF On-Demand Unstable CHRNA10 46 42 C[C@@](O)(CNC(=O)C1CCN(S(C)(=O)=O)CC1)c1cc2ccccc2o1 ZINC000217990848 GD In-Stock Unstable EPHX2 42 41 C[C@@](O)(CNC(=O)C1CCN(S(C)(=O)=O)CC1)c1cc2ccccc2o1 ZINC000217990848 GD In-Stock Unstable CACNA1G 33 40 CCOCCOc1cccc(C(=O)N2CCC(c3noc(C)n3)CC2)c1 ZINC000217990853 FF In-Stock Unstable ETHR 46 34 C[C@](O)(CNC(=O)C1CCN(S(C)(=O)=O)CC1)c1cc2ccccc2o1 ZINC000217990929 GD In-Stock Unstable EPHX2 42 41 C[C@](O)(CNC(=O)C1CCN(S(C)(=O)=O)CC1)c1cc2ccccc2o1 ZINC000217990929 GD In-Stock Unstable CACNA1G 33 40 CN1CCC[C@H]1CNc1cc(Cl)nc(C2CC2)n1 ZINC000217990935 CF On-Demand Unstable CHRNA10 46 42 COc1ccc(-c2n[nH]cc2C(=O)N2CCN(c3ccccc3C)CC2)cc1 ZINC000217990936 GG On-Demand Unstable HTR1A 17 43 COc1ccc(-c2n[nH]cc2C(=O)N2CCN(c3ccccc3C)CC2)cc1 ZINC000217990936 GG On-Demand Unstable HTR7 15 40 COc1ccc(-c2n[nH]cc2C(=O)N2CCN(c3ccccc3C)CC2)cc1 ZINC000217990936 GG On-Demand Unstable CCKAR 41 49 COc1ccc(-c2n[nH]cc2C(=O)N2CCN(c3ccccc3C)CC2)cc1 ZINC000217990936 GG On-Demand Unstable TACR3 27 49 COc1ccc(-c2n[nH]cc2C(=O)N2CCN(c3ccccc3C)CC2)cc1 ZINC000217990936 GG On-Demand Unstable ABCB1 30 40 COc1ccc(-c2n[nH]cc2C(=O)N2CCN(c3ccccc3C)CC2)cc1 ZINC000217990936 GG On-Demand Unstable SMO 15 48 Cn1ncc(C(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)c1-n1cccc1 ZINC000217991008 FD In-Stock Unstable CHRNA4 29 47 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(Cl)c1 ZINC000217991014 IG For-Sale Unstable MMP2 17 51 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(Cl)c1 ZINC000217991014 IG For-Sale Unstable MMP3 41 37 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(Cl)c1 ZINC000217991014 IG For-Sale Unstable MMP7 43 36 CN1CCC[C@@H]1CNc1ccc(C(F)(F)F)nn1 ZINC000217991055 CE On-Demand Unstable CHRNA10 49 36 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(Cl)c1 ZINC000217991096 IG For-Sale Unstable MMP2 17 51 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(Cl)c1 ZINC000217991096 IG For-Sale Unstable MMP3 41 37 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(Cl)c1 ZINC000217991096 IG For-Sale Unstable MMP7 43 36 Cc1nnnn1-c1ccccc1C(=O)N1CCCC[C@H]1c1cccnc1 ZINC000217991121 EF In-Stock Unstable CHRNA2 41 42 Cc1nnnn1-c1ccccc1C(=O)N1CCCC[C@H]1c1cccnc1 ZINC000217991121 EF In-Stock Unstable CRTY 0 42 CN1CCC[C@H]1CNc1ccc(C(F)(F)F)nn1 ZINC000217991138 CE On-Demand Unstable CHRNA10 49 36 Cc1nc2ccccc2cc1C(=O)N[C@@H](C)c1ccc2c(c1)OCO2 ZINC000217991155 EH On-Demand Unstable EDNRA 25 42 Cc1nc2ccccc2cc1C(=O)N[C@@H](C)c1ccc2c(c1)OCO2 ZINC000217991155 EH On-Demand Unstable KCNQ2 23 49 CCc1cccc(OCC(=O)N[C@@H]2CCC[C@@H]2CO)c1 ZINC000217991170 CD On-Demand Unstable FAAH 17 40 Cc1c(CCC(=O)O)ccc(O)c1Br ZINC000217991181 CE For-Sale Unstable FFAR1 29 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(Cl)c1 ZINC000217991185 IG For-Sale Unstable MMP2 17 51 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(Cl)c1 ZINC000217991185 IG For-Sale Unstable MMP3 41 37 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(Cl)c1 ZINC000217991185 IG For-Sale Unstable MMP7 43 36 Cc1nc2ccccc2cc1C(=O)N[C@H](C)c1ccc2c(c1)OCO2 ZINC000217991245 EH On-Demand Unstable EDNRA 25 42 Cc1nc2ccccc2cc1C(=O)N[C@H](C)c1ccc2c(c1)OCO2 ZINC000217991245 EH On-Demand Unstable KCNQ2 23 49 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(Cl)c1 ZINC000217991259 IG For-Sale Unstable MMP2 17 51 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(Cl)c1 ZINC000217991259 IG For-Sale Unstable MMP3 41 37 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(F)c(Cl)c1 ZINC000217991259 IG For-Sale Unstable MMP7 43 36 CCc1ncnc(NC[C@@H]2CCCN2C)c1F ZINC000217991263 BD On-Demand Unstable CHRNA10 52 39 Cc1cc(Br)c(O)cc1CCC(=O)O ZINC000217991280 CE For-Sale Unstable THRA 32 41 Cc1cc(Br)c(O)cc1CCC(=O)O ZINC000217991280 CE For-Sale Unstable THRB 28 45 CCc1ncnc(NC[C@H]2CCCN2C)c1F ZINC000217991342 BD On-Demand Unstable CHRNA10 52 39 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc2c(c1)CCCC2 ZINC000217991360 IG For-Sale Unstable MMP2 15 49 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc2c(c1)CCCC2 ZINC000217991360 IG For-Sale Unstable MMP3 41 36 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc2c(c1)CCCC2 ZINC000217991360 IG For-Sale Unstable MMP7 43 34 Cc1cc(CCC(=O)O)cc(O)c1Br ZINC000217991386 CE For-Sale Unstable THRA 27 49 Cc1cc(CCC(=O)O)cc(O)c1Br ZINC000217991386 CE For-Sale Unstable THRB 21 45 Cc1cc(CCC(=O)O)cc(O)c1Br ZINC000217991386 CE For-Sale Unstable FFAR1 61 43 CCCCCCCCOc1ccc([C@@H]2CC(=O)Oc3cc(C)oc(=O)c32)cc1 ZINC000217991387 GK In-Stock Unstable THRA 40 39 CCCCCCCCOc1ccc([C@@H]2CC(=O)Oc3cc(C)oc(=O)c32)cc1 ZINC000217991387 GK In-Stock Unstable PLA2G4B 68 33 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc2c(c1)CCCC2 ZINC000217991450 IG For-Sale Unstable MMP2 15 49 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc2c(c1)CCCC2 ZINC000217991450 IG For-Sale Unstable MMP3 41 36 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc2c(c1)CCCC2 ZINC000217991450 IG For-Sale Unstable MMP7 43 34 COC(=O)[C@@H]1CCCN1C(=O)c1cc(C)ccc1N=[N+]=[N-] ZINC000217991463 CF For-Sale Unstable PREP 22 46 CCCCCCCCOc1ccc([C@H]2CC(=O)Oc3cc(C)oc(=O)c32)cc1 ZINC000217991468 GK In-Stock Unstable THRA 40 39 CCCCCCCCOc1ccc([C@H]2CC(=O)Oc3cc(C)oc(=O)c32)cc1 ZINC000217991468 GK In-Stock Unstable PLA2G4B 78 33 COc1ccc(-c2noc(CN3CCN(C(=O)c4cc(N5CCCC5)ccn4)CC3)n2)cc1 ZINC000217991474 IF On-Demand Unstable CCKAR 39 41 Cc1cc(O)c(CCC(=O)O)c(Br)c1 ZINC000217991496 CE For-Sale Unstable THRB 18 41 Cc1cc(O)c(CCC(=O)O)c(Br)c1 ZINC000217991496 CE For-Sale Unstable FFAR1 16 43 Cc1cc(O)c(CCC(=O)O)c(Br)c1 ZINC000217991496 CE For-Sale Unstable GPR17 27 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc2c(c1)CCCC2 ZINC000217991522 IG For-Sale Unstable MMP2 15 49 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc2c(c1)CCCC2 ZINC000217991522 IG For-Sale Unstable MMP3 41 36 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc2c(c1)CCCC2 ZINC000217991522 IG For-Sale Unstable MMP7 43 34 CCO[C@@H]1COCC[C@H]1NC(=O)CCc1ccccc1 ZINC000217991571 CD In-Stock Unstable NAAA 40 47 CCO[C@@H]1COCC[C@H]1NC(=O)CCc1ccccc1 ZINC000217991571 CD In-Stock Unstable LUXR 40 37 COc1ccc(-c2cc(C(=O)N3CCCC[C@H]3c3cccnc3)[nH]n2)cc1OC ZINC000217991579 GH In-Stock Unstable COLA 80 39 COc1ccc(-c2cc(C(=O)N3CCCC[C@H]3c3cccnc3)[nH]n2)cc1OC ZINC000217991579 GH In-Stock Unstable CPT1A 71 39 COc1ccc(-c2cc(C(=O)N3CCCC[C@H]3c3cccnc3)[nH]n2)cc1OC ZINC000217991579 GH In-Stock Unstable TACR3 22 43 Cc1ccc(O)c(CCC(=O)O)c1Br ZINC000217991606 CE For-Sale Unstable THRA 28 43 Cc1ccc(O)c(CCC(=O)O)c1Br ZINC000217991606 CE For-Sale Unstable THRB 18 43 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc2c(c1)CCCC2 ZINC000217991608 IG For-Sale Unstable MMP2 15 49 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc2c(c1)CCCC2 ZINC000217991608 IG For-Sale Unstable MMP3 41 36 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc2c(c1)CCCC2 ZINC000217991608 IG For-Sale Unstable MMP7 43 34 C[C@@H](c1ccc(Cl)cc1)N(C)[C@H](C)c1ccc(C(=O)O)o1 ZINC000217991612 DI For-Sale Unstable UTS2 51 38 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)N[C@@H](C)c3nnc4ccccn34)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217991693 KG In-Stock Unstable TUBA1A 17 59 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)N[C@@H](C)c3nnc4ccccn34)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217991693 KG In-Stock Unstable TPPP 0 56 C[C@@H](c1ccccc1Cl)N(C)[C@H](C)c1ccc(C(=O)O)o1 ZINC000217991718 DI For-Sale Unstable MAP 0 46 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(C)(C)C)cc1 ZINC000217991730 IH For-Sale Unstable HSD11B1 21 43 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(C)(C)C)cc1 ZINC000217991730 IH For-Sale Unstable MMP13 52 41 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(C)(C)C)cc1 ZINC000217991730 IH For-Sale Unstable MMP2 28 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(C)(C)C)cc1 ZINC000217991730 IH For-Sale Unstable MMP3 64 41 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(C)(C)C)cc1 ZINC000217991730 IH For-Sale Unstable MMP7 61 37 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(C)(C)C)cc1 ZINC000217991730 IH For-Sale Unstable MMP1 54 41 CC1(C)C[C@H]2C[C@@](C)(CN2C(=O)N/C=C/c2cccc(F)c2)C1 ZINC000217991757 DI For-Sale Unstable AVPR2 17 43 CC1(C)C[C@H]2C[C@@](C)(CN2C(=O)N/C=C/c2cccc(F)c2)C1 ZINC000217991757 DI For-Sale Unstable AVPR1A 36 43 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(C)(C)C)cc1 ZINC000217991813 IH For-Sale Unstable HSD11B1 21 43 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(C)(C)C)cc1 ZINC000217991813 IH For-Sale Unstable MMP13 52 41 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(C)(C)C)cc1 ZINC000217991813 IH For-Sale Unstable MMP2 28 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(C)(C)C)cc1 ZINC000217991813 IH For-Sale Unstable MMP3 64 41 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(C)(C)C)cc1 ZINC000217991813 IH For-Sale Unstable MMP7 61 37 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(C)(C)C)cc1 ZINC000217991813 IH For-Sale Unstable MMP1 54 41 C[C@@H](c1cccc(Cl)c1)N(C)[C@H](C)c1ccc(C(=O)O)o1 ZINC000217991832 DI For-Sale Unstable ADRB1 30 48 C[C@@H](c1cccc(Cl)c1)N(C)[C@H](C)c1ccc(C(=O)O)o1 ZINC000217991832 DI For-Sale Unstable ADRB3 48 48 Cc1ccccc1OCCC(=O)N[C@@H]1CCC[C@@H]1CO ZINC000217991861 CE For-Sale Unstable SLC5A4 40 33 Cc1ccccc1OCCC(=O)N[C@H]1CCC[C@@H]1CO ZINC000217991934 CE For-Sale Unstable SLC5A4 40 33 Cc1ccccc1OCCC(=O)N[C@@H]1CCC[C@H]1CO ZINC000217992006 CE For-Sale Unstable SLC5A4 40 33 Cc1cc(C(=O)Nc2cccnc2Cl)c(C)nn1 ZINC000217992015 CE For-Sale Unstable GRM4 40 40 Cc1cc(C(=O)Nc2cccnc2Cl)c(C)nn1 ZINC000217992015 CE For-Sale Unstable G2YM83_BOTF4 90 46 CN1CCc2nc(NC(=O)N/C=C/c3cccc(F)c3)sc2C1 ZINC000217992077 EG For-Sale Unstable F10 26 42 Cc1ccccc1OCCC(=O)N[C@H]1CCC[C@H]1CO ZINC000217992088 CE For-Sale Unstable SLC5A4 40 33 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000217992104 IE For-Sale Unstable MMP13 50 39 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000217992104 IE For-Sale Unstable MMP2 25 54 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000217992104 IE For-Sale Unstable MMP3 62 39 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000217992104 IE For-Sale Unstable TGM2 43 33 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000217992104 IE For-Sale Unstable MMP7 55 37 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000217992104 IE For-Sale Unstable MMP1 52 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000217992104 IE For-Sale Unstable F13A1 76 33 Cc1cccnc1CN1CCN(Cc2nnc([C@@H]3C[C@H](N)C3)n2C)CC1 ZINC000217992178 FD In-Stock Unstable EGLN1 0 41 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000217992186 IE For-Sale Unstable MMP13 50 39 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000217992186 IE For-Sale Unstable MMP2 25 54 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000217992186 IE For-Sale Unstable MMP3 62 39 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000217992186 IE For-Sale Unstable TGM2 43 33 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000217992186 IE For-Sale Unstable MMP7 55 37 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000217992186 IE For-Sale Unstable MMP1 52 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000217992186 IE For-Sale Unstable F13A1 76 33 CCOc1ccc(OCC(=O)N[C@@H]2CCC[C@@H]2CO)cc1 ZINC000217992195 CD On-Demand Unstable LUXN 0 44 CCOc1ccc(OCC(=O)N[C@@H]2CCC[C@@H]2CO)cc1 ZINC000217992195 CD On-Demand Unstable ADIPOR1 0 42 CCOc1ccc(OCC(=O)N[C@@H]2CCC[C@@H]2CO)cc1 ZINC000217992195 CD On-Demand Unstable ADIPOR2 0 42 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc2c(c1)OCCO2 ZINC000217992292 ID For-Sale Unstable PKM 49 48 CCCN(CC)CCNC(=O)c1c(N)cccc1Cl ZINC000217992328 CE For-Sale Unstable ECR 43 34 Cn1cccc1/C=C1/Oc2cc(OCc3ccccc3)ccc2C1=O ZINC000217992346 EI In-Stock Unstable MAOA 24 41 Cn1cccc1/C=C1/Oc2cc(OCc3ccccc3)ccc2C1=O ZINC000217992346 EI In-Stock Unstable ACHE 17 44 Cn1cccc1/C=C1/Oc2cc(OCc3ccccc3)ccc2C1=O ZINC000217992346 EI In-Stock Unstable MAOB 54 38 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc2c(c1)OCCO2 ZINC000217992380 ID For-Sale Unstable PKM 49 48 N[C@@H](Cc1cc(C(F)F)ccc1Cl)C(=O)O ZINC000217992408 BE For-Sale Unstable CACNA2D1 43 44 N[C@@H](Cc1cc(C(F)F)ccc1Cl)C(=O)O ZINC000217992408 BE For-Sale Unstable TPH1 40 34 C[C@@](O)(CNC(=O)c1cc(C2CC2)on1)c1cc2ccccc2o1 ZINC000217992411 EF In-Stock Unstable S1PR3 0 41 CC(C)Cc1cc(C(=O)N2CCCC[C@H]2c2cccnc2)[nH]n1 ZINC000217992448 DG In-Stock Unstable CHRNA2 40 41 CC(C)Cc1cc(C(=O)N2CCCC[C@H]2c2cccnc2)[nH]n1 ZINC000217992448 DG In-Stock Unstable COLA 72 36 CC(C)Cc1cc(C(=O)N2CCCC[C@H]2c2cccnc2)[nH]n1 ZINC000217992448 DG In-Stock Unstable CPT1A 71 35 CC(C)Cc1cc(C(=O)N2CCCC[C@H]2c2cccnc2)[nH]n1 ZINC000217992448 DG In-Stock Unstable GPBAR1 0 45 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc2c(c1)OCCO2 ZINC000217992463 ID For-Sale Unstable PKM 49 48 N[C@H](Cc1cc(C(F)F)ccc1Cl)C(=O)O ZINC000217992485 BE For-Sale Unstable CACNA2D1 43 44 N[C@H](Cc1cc(C(F)F)ccc1Cl)C(=O)O ZINC000217992485 BE For-Sale Unstable TPH1 40 34 C[C@](O)(CNC(=O)c1cc(C2CC2)on1)c1cc2ccccc2o1 ZINC000217992489 EF In-Stock Unstable S1PR3 0 41 C[C@@H](c1ccc(C(=O)O)o1)N1CC[C@@H](N2CCCC2)C1 ZINC000217992500 CE On-Demand Unstable L3MBTL3 108 47 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc2c(c1)OCCO2 ZINC000217992529 ID For-Sale Unstable PKM 49 48 C[C@@H]1CCCN(S(=O)(=O)N[C@H](C)c2ccc(Br)cc2)C1 ZINC000217992546 FG For-Sale Unstable SDH1 0 44 O=[N+]([O-])c1cccc(CNc2cc(Cl)nc(C3CC3)n2)c1 ZINC000217992553 DH In-Stock Unstable CACNA1D 61 35 O=[N+]([O-])c1cccc(CNc2cc(Cl)nc(C3CC3)n2)c1 ZINC000217992553 DH In-Stock Unstable LUXR 16 43 COc1cc(CC(=O)O)cc(C)c1Br ZINC000217992564 CE For-Sale Unstable THRA 29 40 COc1cc(CC(=O)O)cc(C)c1Br ZINC000217992564 CE For-Sale Unstable THRB 23 40 C[C@H](c1ccc(C(=O)O)o1)N1CC[C@@H](N2CCCC2)C1 ZINC000217992577 CE On-Demand Unstable L3MBTL3 108 47 C[C@H]1CCCCN1S(=O)(=O)N[C@H](C)c1ccc(Br)cc1 ZINC000217992630 FG For-Sale Unstable SDH1 0 45 COc1ccc(CNC(=O)c2ccccc2NC(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc1 ZINC000217992638 JG In-Stock Unstable CHRNA4 27 42 CCc1ncnc(NCc2cccc([N+](=O)[O-])c2)c1F ZINC000217992660 CF On-Demand Unstable ADORA3 25 45 CCc1ncnc(NCc2cccc([N+](=O)[O-])c2)c1F ZINC000217992660 CF On-Demand Unstable CLK4 22 42 C[C@@H](c1ccc(C(=O)O)o1)N1CC[C@@H](N2CCCCC2)C1 ZINC000217992690 CF On-Demand Unstable L3MBTL3 104 46 O=C(CCc1nnc(-c2ccccc2)o1)N1CCN(Cc2nc(-c3ccc(Cl)cc3)no2)CC1 ZINC000217992731 JH On-Demand Unstable S1PR4 15 41 O=C(CCc1nnc(-c2ccccc2)o1)N1CCN(Cc2nc(-c3ccc(Cl)cc3)no2)CC1 ZINC000217992731 JH On-Demand Unstable S1PR1 17 41 C[C@@H]1CCCN(S(=O)(=O)N[C@H](C)c2cccc(Br)c2)C1 ZINC000217992732 FG For-Sale Unstable MBTD1 0 40 C[C@H](c1ccc(C(=O)O)o1)N1CC[C@@H](N2CCCCC2)C1 ZINC000217992770 CF On-Demand Unstable L3MBTL3 104 46 O=C(/C=C/c1cccc(Br)c1)N[C@H]1CCC[C@H]1CO ZINC000217992776 DF On-Demand Unstable HDAC8 47 37 NC[C@@H](C(=O)O)c1cc(C(F)F)ccc1Cl ZINC000217992780 BE For-Sale Unstable CACNA2D1 20 42 CCN[C@@H](CCCc1ccccc1)[C@@H]1CCC[C@@H](C)C1 ZINC000217992816 CJ For-Sale Unstable SLC18A2 37 41 NC[C@H](C(=O)O)c1cc(C(F)F)ccc1Cl ZINC000217992855 BE For-Sale Unstable CACNA2D1 20 42 COc1ccc(O)c(C(=O)N2CCN(Cc3nc(-c4ccc(Cl)cc4)no3)CC2)c1 ZINC000217992863 IG On-Demand Unstable PDK1 60 39 CCN[C@H](CCCc1ccccc1)[C@@H]1CCC[C@@H](C)C1 ZINC000217992905 CJ For-Sale Unstable SLC18A2 37 41 CC(C)(C)c1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217992940 DJ For-Sale Unstable TRPV1 20 41 CC(C)(C)c1ccc(NC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217992940 DJ For-Sale Unstable IMDH_CRYPV 54 35 N[C@@H](Cc1cc(Cl)ccc1C(F)F)C(=O)O ZINC000217992958 BE For-Sale Unstable CACNA2D1 42 47 CCN[C@@H](CCCc1ccccc1)[C@H]1CCC[C@@H](C)C1 ZINC000217992988 CJ For-Sale Unstable SLC18A2 37 41 CCOc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1C ZINC000217993013 IF For-Sale Unstable MMP2 16 47 CCOc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1C ZINC000217993013 IF For-Sale Unstable MMP3 43 36 CCOc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1C ZINC000217993013 IF For-Sale Unstable MMP7 46 35 N[C@H](Cc1cc(Cl)ccc1C(F)F)C(=O)O ZINC000217993037 BE For-Sale Unstable CACNA2D1 42 47 CCN[C@H](CCCc1ccccc1)[C@H]1CCC[C@@H](C)C1 ZINC000217993049 CJ For-Sale Unstable SLC18A2 37 41 CCOc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1C ZINC000217993102 IF For-Sale Unstable MMP2 16 47 CCOc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1C ZINC000217993102 IF For-Sale Unstable MMP3 43 36 CCOc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1C ZINC000217993102 IF For-Sale Unstable MMP7 46 35 O=C(Nc1ccc(Br)c(Cl)c1)[C@H]1[C@H]2C=C[C@H](C2)[C@H]1C(=O)O ZINC000217993108 FH In-Stock Unstable F13A1 16 50 COc1ccc(-c2n[nH]cc2C(=O)Nc2nc(-c3ccccc3)cs2)cc1 ZINC000217993137 GI On-Demand Unstable MAOA 19 42 COc1ccc(-c2n[nH]cc2C(=O)Nc2nc(-c3ccccc3)cs2)cc1 ZINC000217993137 GI On-Demand Unstable MAOB 27 42 COc1ccc(-c2n[nH]cc2C(=O)Nc2nc(-c3ccccc3)cs2)cc1 ZINC000217993137 GI On-Demand Unstable ADORA1 15 69 COc1ccc(-c2n[nH]cc2C(=O)Nc2nc(-c3ccccc3)cs2)cc1 ZINC000217993137 GI On-Demand Unstable ROCK1 31 45 COc1ccc(-c2n[nH]cc2C(=O)Nc2nc(-c3ccccc3)cs2)cc1 ZINC000217993137 GI On-Demand Unstable ROCK2 25 45 COc1ccc(-c2n[nH]cc2C(=O)Nc2nc(-c3ccccc3)cs2)cc1 ZINC000217993137 GI On-Demand Unstable HDAC9 15 43 COc1ccc(-c2n[nH]cc2C(=O)Nc2nc(-c3ccccc3)cs2)cc1 ZINC000217993137 GI On-Demand Unstable GCK 18 43 COc1ccc(-c2n[nH]cc2C(=O)Nc2nc(-c3ccccc3)cs2)cc1 ZINC000217993137 GI On-Demand Unstable LUCI_LUCLA 22 40 O=C(N[C@@H](c1ccccn1)[C@@H]1C[C@H](O)C1)c1ccn2nnnc2c1 ZINC000217993194 DC In-Stock Unstable TTK 39 49 O=C(Nc1ccc(Br)c(Cl)c1)[C@H]1[C@H]2C=C[C@@H](C2)[C@H]1C(=O)O ZINC000217993203 FH In-Stock Unstable F13A1 16 50 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1cc(C)c(OC)c(C)c1 ZINC000217993215 IF For-Sale Unstable MMP2 15 56 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1cc(C)c(OC)c(C)c1 ZINC000217993215 IF For-Sale Unstable MMP7 42 34 O=C(N[C@@H]1CCC[C@@H]1CO)c1ccc(=O)[nH]c1 ZINC000217993226 BC For-Sale Unstable SSTR3 27 40 C[C@@](O)(CNC(=O)Cc1c(F)cccc1Cl)c1cc2ccccc2o1 ZINC000217993261 FH In-Stock Unstable P2RX7 21 43 O=C(N[C@H](c1ccccn1)[C@@H]1C[C@H](O)C1)c1ccn2nnnc2c1 ZINC000217993265 DC In-Stock Unstable TTK 39 49 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1cc(C)c(OC)c(C)c1 ZINC000217993297 IF For-Sale Unstable MMP2 15 56 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1cc(C)c(OC)c(C)c1 ZINC000217993297 IF For-Sale Unstable MMP7 42 34 O=C(N[C@H]1CCC[C@@H]1CO)c1ccc(=O)[nH]c1 ZINC000217993317 BC For-Sale Unstable SSTR3 27 40 C[C@](O)(CNC(=O)Cc1c(F)cccc1Cl)c1cc2ccccc2o1 ZINC000217993327 FH In-Stock Unstable P2RX7 21 43 O=C(N/C=C/c1cccc(F)c1)Nc1ccc2cn[nH]c2c1 ZINC000217993362 CG For-Sale Anodyne PLK4 19 40 O=C(N[C@@H]1CCC[C@H]1CO)c1ccc(=O)[nH]c1 ZINC000217993392 BC For-Sale Unstable SSTR3 27 40 CCc1ccc(OC)c(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)c1 ZINC000217993409 IF For-Sale Unstable CPT1B 44 34 O=C(N[C@H]1CCC[C@H]1CO)c1ccc(=O)[nH]c1 ZINC000217993468 BC On-Demand Unstable SSTR3 25 40 CC(C)(C)c1ccccc1NC(=O)N/C=C/c1cccc(F)c1 ZINC000217993469 DJ For-Sale Unstable P2RY1 21 41 CCc1ccc(OC)c(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)c1 ZINC000217993483 IF For-Sale Unstable CPT1B 44 34 C[C@H](C(=O)O)c1ccc(Br)cc1CO ZINC000217993491 CE For-Sale Unstable PTGS1 27 42 C[C@H](C(=O)O)c1ccc(Br)cc1CO ZINC000217993491 CE For-Sale Unstable PTGS2 20 41 N[C@@H](Cc1ccc(C(F)F)cc1Cl)C(=O)O ZINC000217993519 BE For-Sale Unstable CACNA2D1 41 45 N[C@@H](Cc1ccc(C(F)F)cc1Cl)C(=O)O ZINC000217993519 BE For-Sale Unstable TPH1 41 36 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217993562 FD For-Sale Unstable CA2 97 58 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217993562 FD For-Sale Unstable CA6 17 40 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217993562 FD For-Sale Unstable CA1 82 58 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217993562 FD For-Sale Unstable CA7 48 48 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217993562 FD For-Sale Unstable CA13 19 40 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217993562 FD For-Sale Unstable CA5B 53 48 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217993562 FD For-Sale Unstable CA4 70 54 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217993562 FD For-Sale Unstable CA5A 54 48 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217993562 FD For-Sale Unstable CA14 40 48 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217993562 FD For-Sale Unstable CA12 62 58 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217993562 FD For-Sale Unstable CA9 73 58 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217993562 FD For-Sale Unstable CYNT 25 43 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217993562 FD For-Sale Unstable NCE103 31 49 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217993562 FD For-Sale Unstable LIG1 0 43 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217993562 FD For-Sale Unstable MTCA1 40 38 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217993562 FD For-Sale Unstable P96878_MYCTU 50 44 NS(=O)(=O)c1ccc(CCNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217993562 FD For-Sale Unstable A6YCJ1_9METZ 24 48 C[C@@H](C(=O)O)c1ccc(Br)cc1CO ZINC000217993572 CE For-Sale Unstable PTGS1 27 42 C[C@@H](C(=O)O)c1ccc(Br)cc1CO ZINC000217993572 CE For-Sale Unstable PTGS2 20 41 N[C@H](Cc1ccc(C(F)F)cc1Cl)C(=O)O ZINC000217993591 BE For-Sale Unstable CACNA2D1 41 45 N[C@H](Cc1ccc(C(F)F)cc1Cl)C(=O)O ZINC000217993591 BE For-Sale Unstable TPH1 41 36 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)CCc1ccc(OC)cc1 ZINC000217993593 IE For-Sale Unstable FKBP1A 21 44 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)CCc1ccc(OC)cc1 ZINC000217993593 IE For-Sale Unstable MMP13 45 50 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)CCc1ccc(OC)cc1 ZINC000217993593 IE For-Sale Unstable MMP2 25 45 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)CCc1ccc(OC)cc1 ZINC000217993593 IE For-Sale Unstable MMP3 59 44 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)CCc1ccc(OC)cc1 ZINC000217993593 IE For-Sale Unstable MMP8 19 50 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)CCc1ccc(OC)cc1 ZINC000217993593 IE For-Sale Unstable MMP12 21 50 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)CCc1ccc(OC)cc1 ZINC000217993593 IE For-Sale Unstable MMP7 47 39 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)CCc1ccc(OC)cc1 ZINC000217993593 IE For-Sale Unstable MMP1 50 44 O=C(N/C=C/c1cccc(F)c1)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000217993667 GK For-Sale Mild PTPA 0 42 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)CCc1ccc(OC)cc1 ZINC000217993681 IE For-Sale Unstable FKBP1A 21 44 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)CCc1ccc(OC)cc1 ZINC000217993681 IE For-Sale Unstable MMP13 45 50 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)CCc1ccc(OC)cc1 ZINC000217993681 IE For-Sale Unstable MMP2 25 45 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)CCc1ccc(OC)cc1 ZINC000217993681 IE For-Sale Unstable MMP3 59 44 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)CCc1ccc(OC)cc1 ZINC000217993681 IE For-Sale Unstable MMP8 19 50 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)CCc1ccc(OC)cc1 ZINC000217993681 IE For-Sale Unstable MMP12 21 50 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)CCc1ccc(OC)cc1 ZINC000217993681 IE For-Sale Unstable MMP7 47 39 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)CCc1ccc(OC)cc1 ZINC000217993681 IE For-Sale Unstable MMP1 50 44 O=C(O)CCc1ccc(Br)cc1CO ZINC000217993698 CD For-Sale Unstable FFAR1 26 40 O=C(Cn1cc(Br)c(=O)[nH]c1=O)Nc1ccc(CN2CCOCC2)cc1 ZINC000217993741 HC On-Demand Unstable EPHX2 16 42 CN1C[C@@H](NC(=O)c2ccccc2Oc2ccccc2)C[C@H]1C(=O)O ZINC000217993763 EE In-Stock Unstable FABH 0 42 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1cc(OC)ccc1OC ZINC000217993797 IE For-Sale Unstable MMP13 43 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1cc(OC)ccc1OC ZINC000217993797 IE For-Sale Unstable MMP2 23 48 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1cc(OC)ccc1OC ZINC000217993797 IE For-Sale Unstable MMP3 54 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1cc(OC)ccc1OC ZINC000217993797 IE For-Sale Unstable MMP7 51 38 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1cc(OC)ccc1OC ZINC000217993797 IE For-Sale Unstable MMP1 47 40 C[C@H](C(=O)O)c1ccc(CO)cc1Br ZINC000217993825 CE For-Sale Unstable PTGS1 33 60 C[C@H](C(=O)O)c1ccc(CO)cc1Br ZINC000217993825 CE For-Sale Unstable PTGS2 25 60 C[C@H](C(=O)O)c1ccc(CO)cc1Br ZINC000217993825 CE For-Sale Unstable CXCL8 17 41 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1cc(OC)ccc1OC ZINC000217993875 IE For-Sale Unstable MMP13 43 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1cc(OC)ccc1OC ZINC000217993875 IE For-Sale Unstable MMP2 23 48 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1cc(OC)ccc1OC ZINC000217993875 IE For-Sale Unstable MMP3 54 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1cc(OC)ccc1OC ZINC000217993875 IE For-Sale Unstable MMP7 51 38 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1cc(OC)ccc1OC ZINC000217993875 IE For-Sale Unstable MMP1 47 40 C[C@H]1CCC[C@H](C)N1C(=O)N[C@@H](C(=O)O)[C@@H](C)O ZINC000217993886 CC For-Sale Unstable EDNRB 48 38 Cc1cccc(-c2noc(CNC(=O)[C@@H](C)Sc3ccc(Cl)cc3)n2)c1 ZINC000217993892 GI In-Stock Unstable GRM5 21 44 C[C@@H](C(=O)O)c1ccc(CO)cc1Br ZINC000217993909 CE For-Sale Unstable PTGS1 33 60 C[C@@H](C(=O)O)c1ccc(CO)cc1Br ZINC000217993909 CE For-Sale Unstable PTGS2 25 60 C[C@@H](C(=O)O)c1ccc(CO)cc1Br ZINC000217993909 CE For-Sale Unstable CXCL8 17 41 Cc1cc(-c2cc(C(=O)Nc3ccc(CN4CCOCC4)cc3)c3cnn(C(C)C)c3n2)c(C)o1 ZINC000217993928 JJ On-Demand Unstable EZH2 17 40 COC(=O)C(C)(C)N[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000217993933 CF For-Sale Unstable TRPM8 17 50 C[C@H](O)[C@@H](NC(=O)N1[C@@H](C)CCC[C@@H]1C)C(=O)O ZINC000217993959 CC On-Demand Unstable EDNRB 48 38 Cc1cccc(-c2noc(CNC(=O)[C@H](C)Sc3ccc(Cl)cc3)n2)c1 ZINC000217993963 GI In-Stock Unstable GRM5 21 44 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(OC)c1 ZINC000217993991 IE For-Sale Unstable MMP13 41 39 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(OC)c1 ZINC000217993991 IE For-Sale Unstable MMP2 21 54 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(OC)c1 ZINC000217993991 IE For-Sale Unstable MMP3 53 39 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(OC)c1 ZINC000217993991 IE For-Sale Unstable MMP7 49 37 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(OC)c1 ZINC000217993991 IE For-Sale Unstable MMP1 44 39 COC(=O)C(C)(C)N[C@H]1C[C@H](C)CC[C@@H]1C(C)C ZINC000217994008 CF For-Sale Unstable TRPM8 17 50 O=C(O)CCc1ccc(CO)cc1Br ZINC000217994010 CD For-Sale Unstable THRA 34 44 O=C(O)CCc1ccc(CO)cc1Br ZINC000217994010 CD For-Sale Unstable THRB 29 44 O=C(O)CCc1ccc(CO)cc1Br ZINC000217994010 CD For-Sale Unstable FFAR1 71 47 O=C(O)CCc1ccc(CO)cc1Br ZINC000217994010 CD For-Sale Unstable FFAR4 59 38 C[C@H](O)[C@H](NC(=O)N1[C@@H](C)CCC[C@@H]1C)C(=O)O ZINC000217994044 CC On-Demand Unstable EDNRB 48 38 Cc1ccc(-c2noc(CNC(=O)[C@@H](C)Sc3ccc(Cl)cc3)n2)cc1 ZINC000217994073 GI In-Stock Unstable SCN10A 40 36 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(F)c(Cl)c1 ZINC000217994079 DI For-Sale Anodyne IMPDH2 0 41 O=C(N/C=C/c1cccc(F)c1)Nc1ccc(F)c(Cl)c1 ZINC000217994079 DI For-Sale Anodyne P95276_MYCTO 0 43 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(OC)c1 ZINC000217994083 IE For-Sale Unstable MMP13 41 39 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(OC)c1 ZINC000217994083 IE For-Sale Unstable MMP2 21 54 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(OC)c1 ZINC000217994083 IE For-Sale Unstable MMP3 53 39 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(OC)c1 ZINC000217994083 IE For-Sale Unstable MMP7 49 37 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(OC)c1 ZINC000217994083 IE For-Sale Unstable MMP1 44 39 CC(F)(F)c1ccc([C@H](N)C(=O)O)c(Cl)c1 ZINC000217994089 BF For-Sale Unstable CACNA2D1 26 44 Cc1ccc(-c2noc(CNC(=O)[C@H](C)Sc3ccc(Cl)cc3)n2)cc1 ZINC000217994141 GI In-Stock Unstable SCN10A 40 36 Cc1ccccc1-c1cc(C(=O)Nc2ccc(CN3CCOCC3)cc2)c2cnn(C(C)C)c2n1 ZINC000217994146 JK On-Demand Unstable PIK3CA 21 41 Cc1ccccc1-c1cc(C(=O)Nc2ccc(CN3CCOCC3)cc2)c2cnn(C(C)C)c2n1 ZINC000217994146 JK On-Demand Unstable MTOR 38 40 Cc1ccccc1-c1cc(C(=O)Nc2ccc(CN3CCOCC3)cc2)c2cnn(C(C)C)c2n1 ZINC000217994146 JK On-Demand Unstable EZH2 23 42 CC(F)(F)c1ccc([C@@H](N)C(=O)O)c(Cl)c1 ZINC000217994167 BF For-Sale Unstable CACNA2D1 26 44 COC(=O)C[C@H](c1ccc(OC)c(OC)c1)c1oc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c1O ZINC000217994189 KF In-Stock Unstable CHRNA4 26 43 CCOc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1F ZINC000217994205 IF For-Sale Unstable MMP13 44 37 CCOc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1F ZINC000217994205 IF For-Sale Unstable MMP2 20 48 CCOc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1F ZINC000217994205 IF For-Sale Unstable MMP3 49 37 CCOc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1F ZINC000217994205 IF For-Sale Unstable MMP7 52 34 CCOc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1F ZINC000217994205 IF For-Sale Unstable MMP1 44 37 CC[C@@H](C)[C@@H](NC(=O)N1[C@@H](C)CCC[C@@H]1C)C(=O)O ZINC000217994209 CE On-Demand Unstable EDNRB 37 45 COc1cccc(-c2noc(CNC(=O)[C@@H](C)Sc3ccc(Cl)cc3)n2)c1 ZINC000217994248 HI In-Stock Unstable GRM5 16 43 O=C(Nc1ccc(CN2CCOCC2)cc1)c1cc(-c2ccc(Cl)cc2)n[nH]1 ZINC000217994271 GH On-Demand Unstable DRD4 35 42 O=C(Nc1ccc(CN2CCOCC2)cc1)c1cc(-c2ccc(Cl)cc2)n[nH]1 ZINC000217994271 GH On-Demand Unstable F10 23 49 O=C(Nc1ccc(CN2CCOCC2)cc1)c1cc(-c2ccc(Cl)cc2)n[nH]1 ZINC000217994271 GH On-Demand Unstable PTGER1 19 48 O=C(Nc1ccc(CN2CCOCC2)cc1)c1cc(-c2ccc(Cl)cc2)n[nH]1 ZINC000217994271 GH On-Demand Unstable PIK3CA 29 44 O=C(Nc1ccc(CN2CCOCC2)cc1)c1cc(-c2ccc(Cl)cc2)n[nH]1 ZINC000217994271 GH On-Demand Unstable CHRNA7 21 44 O=C(Nc1ccc(CN2CCOCC2)cc1)c1cc(-c2ccc(Cl)cc2)n[nH]1 ZINC000217994271 GH On-Demand Unstable AURKB 17 42 O=C(Nc1ccc(CN2CCOCC2)cc1)c1cc(-c2ccc(Cl)cc2)n[nH]1 ZINC000217994271 GH On-Demand Unstable JAK3 20 45 O=C(Nc1ccc(CN2CCOCC2)cc1)c1cc(-c2ccc(Cl)cc2)n[nH]1 ZINC000217994271 GH On-Demand Unstable PRNP 52 37 O=C(Nc1ccc(CN2CCOCC2)cc1)c1cc(-c2ccc(Cl)cc2)n[nH]1 ZINC000217994271 GH On-Demand Unstable JAK2 16 41 O=C(Nc1ccc(CN2CCOCC2)cc1)c1cc(-c2ccc(Cl)cc2)n[nH]1 ZINC000217994271 GH On-Demand Unstable FLT1 22 41 O=C(Nc1ccc(CN2CCOCC2)cc1)c1cc(-c2ccc(Cl)cc2)n[nH]1 ZINC000217994271 GH On-Demand Unstable KDR 21 55 O=C(Nc1ccc(CN2CCOCC2)cc1)c1cc(-c2ccc(Cl)cc2)n[nH]1 ZINC000217994271 GH On-Demand Unstable TACR3 15 46 O=C(Nc1ccc(CN2CCOCC2)cc1)c1cc(-c2ccc(Cl)cc2)n[nH]1 ZINC000217994271 GH On-Demand Unstable FAAH 20 41 O=C(Nc1ccc(CN2CCOCC2)cc1)c1cc(-c2ccc(Cl)cc2)n[nH]1 ZINC000217994271 GH On-Demand Unstable MTOR 48 44 O=C(Nc1ccc(CN2CCOCC2)cc1)c1cc(-c2ccc(Cl)cc2)n[nH]1 ZINC000217994271 GH On-Demand Unstable EPHX2 25 48 O=C(Nc1ccc(CN2CCOCC2)cc1)c1cc(-c2ccc(Cl)cc2)n[nH]1 ZINC000217994271 GH On-Demand Unstable PIK3CG 23 44 O=C(Nc1ccc(CN2CCOCC2)cc1)c1cc(-c2ccc(Cl)cc2)n[nH]1 ZINC000217994271 GH On-Demand Unstable FLT3 37 55 O=C(Nc1ccc(CN2CCOCC2)cc1)c1cc(-c2ccc(Cl)cc2)n[nH]1 ZINC000217994271 GH On-Demand Unstable ALPL 64 37 O=C(Nc1ccc(CN2CCOCC2)cc1)c1cc(-c2ccc(Cl)cc2)n[nH]1 ZINC000217994271 GH On-Demand Unstable MCHR1 29 52 O=C(Nc1ccc(CN2CCOCC2)cc1)c1cc(-c2ccc(Cl)cc2)n[nH]1 ZINC000217994271 GH On-Demand Unstable AURKA 29 49 O=C(Nc1ccc(CN2CCOCC2)cc1)c1cc(-c2ccc(Cl)cc2)n[nH]1 ZINC000217994271 GH On-Demand Unstable DPOL_VZVD 24 42 O=C(Nc1ccc(CN2CCOCC2)cc1)c1cc(-c2ccc(Cl)cc2)n[nH]1 ZINC000217994271 GH On-Demand Unstable DGAT1 21 42 O=C(Nc1ccc(CN2CCOCC2)cc1)c1cc(-c2ccc(Cl)cc2)n[nH]1 ZINC000217994271 GH On-Demand Unstable NOD1 29 45 O=C(Nc1ccc(CN2CCOCC2)cc1)c1cc(-c2ccc(Cl)cc2)n[nH]1 ZINC000217994271 GH On-Demand Unstable NOD2 41 34 COC(=O)C[C@@H](c1ccc(OC)c(OC)c1)c1oc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c1O ZINC000217994278 KF In-Stock Unstable CHRNA4 26 43 CCOc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1F ZINC000217994279 IF For-Sale Unstable MMP13 44 37 CCOc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1F ZINC000217994279 IF For-Sale Unstable MMP2 20 48 CCOc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1F ZINC000217994279 IF For-Sale Unstable MMP3 49 37 CCOc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1F ZINC000217994279 IF For-Sale Unstable MMP7 52 34 CCOc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1F ZINC000217994279 IF For-Sale Unstable MMP1 44 37 CC(F)(F)c1c(Cl)cccc1[C@H](N)C(=O)O ZINC000217994280 BF For-Sale Unstable CACNA2D1 25 51 O=C([C@H](Cl)c1ccccc1)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217994285 CI For-Sale Unstable PREP 45 37 O=C(N/C=C/c1cccc(F)c1)NCc1ccc(F)cc1 ZINC000217994311 CG For-Sale Unstable Q76353_9HIV1 0 41 COc1cccc(-c2noc(CNC(=O)[C@H](C)Sc3ccc(Cl)cc3)n2)c1 ZINC000217994334 HI In-Stock Unstable GRM5 16 43 CC(F)(F)c1c(Cl)cccc1[C@@H](N)C(=O)O ZINC000217994356 BF For-Sale Unstable CACNA2D1 25 51 O=C([C@@H](Cl)c1ccccc1)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217994365 CI For-Sale Unstable PREP 45 37 Cc1ccc(-c2cc(C(=O)Nc3ccc(CN4CCOCC4)cc3)[nH]n2)cc1 ZINC000217994373 GG On-Demand Unstable KIT 24 45 Cc1ccc(-c2cc(C(=O)Nc3ccc(CN4CCOCC4)cc3)[nH]n2)cc1 ZINC000217994373 GG On-Demand Unstable PTGER1 17 46 Cc1ccc(-c2cc(C(=O)Nc3ccc(CN4CCOCC4)cc3)[nH]n2)cc1 ZINC000217994373 GG On-Demand Unstable PIK3CA 34 42 Cc1ccc(-c2cc(C(=O)Nc3ccc(CN4CCOCC4)cc3)[nH]n2)cc1 ZINC000217994373 GG On-Demand Unstable CHRNA7 23 46 Cc1ccc(-c2cc(C(=O)Nc3ccc(CN4CCOCC4)cc3)[nH]n2)cc1 ZINC000217994373 GG On-Demand Unstable AURKB 25 41 Cc1ccc(-c2cc(C(=O)Nc3ccc(CN4CCOCC4)cc3)[nH]n2)cc1 ZINC000217994373 GG On-Demand Unstable JAK3 24 47 Cc1ccc(-c2cc(C(=O)Nc3ccc(CN4CCOCC4)cc3)[nH]n2)cc1 ZINC000217994373 GG On-Demand Unstable PRNP 54 39 Cc1ccc(-c2cc(C(=O)Nc3ccc(CN4CCOCC4)cc3)[nH]n2)cc1 ZINC000217994373 GG On-Demand Unstable JAK2 18 43 Cc1ccc(-c2cc(C(=O)Nc3ccc(CN4CCOCC4)cc3)[nH]n2)cc1 ZINC000217994373 GG On-Demand Unstable FLT1 25 42 Cc1ccc(-c2cc(C(=O)Nc3ccc(CN4CCOCC4)cc3)[nH]n2)cc1 ZINC000217994373 GG On-Demand Unstable KDR 27 49 Cc1ccc(-c2cc(C(=O)Nc3ccc(CN4CCOCC4)cc3)[nH]n2)cc1 ZINC000217994373 GG On-Demand Unstable NR1H4 21 40 Cc1ccc(-c2cc(C(=O)Nc3ccc(CN4CCOCC4)cc3)[nH]n2)cc1 ZINC000217994373 GG On-Demand Unstable MTOR 60 42 Cc1ccc(-c2cc(C(=O)Nc3ccc(CN4CCOCC4)cc3)[nH]n2)cc1 ZINC000217994373 GG On-Demand Unstable EPHX2 23 41 Cc1ccc(-c2cc(C(=O)Nc3ccc(CN4CCOCC4)cc3)[nH]n2)cc1 ZINC000217994373 GG On-Demand Unstable SCN10A 41 32 Cc1ccc(-c2cc(C(=O)Nc3ccc(CN4CCOCC4)cc3)[nH]n2)cc1 ZINC000217994373 GG On-Demand Unstable FLT3 45 49 Cc1ccc(-c2cc(C(=O)Nc3ccc(CN4CCOCC4)cc3)[nH]n2)cc1 ZINC000217994373 GG On-Demand Unstable MCHR1 29 44 Cc1ccc(-c2cc(C(=O)Nc3ccc(CN4CCOCC4)cc3)[nH]n2)cc1 ZINC000217994373 GG On-Demand Unstable AURKA 37 49 Cc1ccc(-c2cc(C(=O)Nc3ccc(CN4CCOCC4)cc3)[nH]n2)cc1 ZINC000217994373 GG On-Demand Unstable NOD2 43 37 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(Cl)c1 ZINC000217994381 IF For-Sale Unstable MMP2 18 52 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(Cl)c1 ZINC000217994381 IF For-Sale Unstable MMP3 42 38 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(Cl)c1 ZINC000217994381 IF For-Sale Unstable MMP7 44 35 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(Cl)c1 ZINC000217994381 IF For-Sale Unstable MMP1 40 38 COc1ccccc1N1CCN(C(=O)N/C=C/c2cccc(F)c2)CC1 ZINC000217994422 FG For-Sale Unstable HTR1A 89 50 COc1ccccc1N1CCN(C(=O)N/C=C/c2cccc(F)c2)CC1 ZINC000217994422 FG For-Sale Unstable DRD2 68 46 COc1ccccc1N1CCN(C(=O)N/C=C/c2cccc(F)c2)CC1 ZINC000217994422 FG For-Sale Unstable DRD4 36 43 COc1ccccc1N1CCN(C(=O)N/C=C/c2cccc(F)c2)CC1 ZINC000217994422 FG For-Sale Unstable ADRA1D 72 39 COc1ccccc1N1CCN(C(=O)N/C=C/c2cccc(F)c2)CC1 ZINC000217994422 FG For-Sale Unstable HTR1D 25 47 COc1ccccc1N1CCN(C(=O)N/C=C/c2cccc(F)c2)CC1 ZINC000217994422 FG For-Sale Unstable HTR1B 21 50 COc1ccccc1N1CCN(C(=O)N/C=C/c2cccc(F)c2)CC1 ZINC000217994422 FG For-Sale Unstable HTR2A 33 46 COc1ccccc1N1CCN(C(=O)N/C=C/c2cccc(F)c2)CC1 ZINC000217994422 FG For-Sale Unstable ADRA1A 67 40 COc1ccccc1N1CCN(C(=O)N/C=C/c2cccc(F)c2)CC1 ZINC000217994422 FG For-Sale Unstable ADRA1B 58 39 COc1ccccc1N1CCN(C(=O)N/C=C/c2cccc(F)c2)CC1 ZINC000217994422 FG For-Sale Unstable DRD3 70 46 COc1ccccc1N1CCN(C(=O)N/C=C/c2cccc(F)c2)CC1 ZINC000217994422 FG For-Sale Unstable HTR7 58 48 COc1ccccc1N1CCN(C(=O)N/C=C/c2cccc(F)c2)CC1 ZINC000217994422 FG For-Sale Unstable TACR3 22 52 COc1ccccc1N1CCN(C(=O)N/C=C/c2cccc(F)c2)CC1 ZINC000217994422 FG For-Sale Unstable RBP4 22 43 COc1ccccc1N1CCN(C(=O)N/C=C/c2cccc(F)c2)CC1 ZINC000217994422 FG For-Sale Unstable ACKR3 53 37 O=C([C@H](Cl)c1ccccc1)N1CCC[C@H]2CCCC[C@H]21 ZINC000217994430 CI For-Sale Unstable PREP 45 37 N[C@@H](Cc1cccc(Cl)c1C(F)F)C(=O)O ZINC000217994459 BE For-Sale Unstable CACNA2D1 57 47 N[C@@H](Cc1cccc(Cl)c1C(F)F)C(=O)O ZINC000217994459 BE For-Sale Unstable GRIK1 19 41 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(Cl)c1 ZINC000217994461 IF For-Sale Unstable MMP2 18 52 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(Cl)c1 ZINC000217994461 IF For-Sale Unstable MMP3 42 38 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(Cl)c1 ZINC000217994461 IF For-Sale Unstable MMP7 44 35 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC)c(Cl)c1 ZINC000217994461 IF For-Sale Unstable MMP1 40 38 O=C(CC1CCCC1)N[C@@H]1CCOC[C@H]1OCc1ccccc1 ZINC000217994479 DG In-Stock Unstable KLK5 46 42 O=C(CCc1ncc(-c2ccc(Cl)cc2Cl)o1)Nc1ccc(CN2CCOCC2)cc1 ZINC000217994485 JK On-Demand Unstable HTR2A 15 42 O=C(CCc1ncc(-c2ccc(Cl)cc2Cl)o1)Nc1ccc(CN2CCOCC2)cc1 ZINC000217994485 JK On-Demand Unstable EPHX2 16 45 O=C([C@@H](Cl)c1ccccc1)N1CCC[C@H]2CCCC[C@H]21 ZINC000217994504 CI For-Sale Unstable PREP 45 37 N[C@H](Cc1cccc(Cl)c1C(F)F)C(=O)O ZINC000217994541 BE For-Sale Unstable CACNA2D1 57 47 N[C@H](Cc1cccc(Cl)c1C(F)F)C(=O)O ZINC000217994541 BE For-Sale Unstable GRIK1 19 41 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000217994574 IG For-Sale Unstable MMP13 54 39 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000217994574 IG For-Sale Unstable CACNA1B 16 41 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000217994574 IG For-Sale Unstable ADAM17 25 41 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000217994574 IG For-Sale Unstable MMP2 28 54 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000217994574 IG For-Sale Unstable MMP3 63 39 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000217994574 IG For-Sale Unstable MMP8 33 41 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000217994574 IG For-Sale Unstable MMP7 57 39 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000217994574 IG For-Sale Unstable MMP1 53 39 CC(C)[C@@H](Br)C(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217994611 DH For-Sale Unstable DPP4 21 42 CC(C)[C@@H](Br)C(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217994611 DH For-Sale Unstable DPP7 18 42 CC(C)[C@@H](Br)C(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217994611 DH For-Sale Unstable DPP9 16 42 CC[C@H](C)[C@@H](NC(=O)CS[C@@H](C(=O)O)C(C)C)C(=O)OC ZINC000217994612 DD For-Sale Unstable ENPEP 51 32 CC[C@H](C)[C@@H](NC(=O)CS[C@@H](C(=O)O)C(C)C)C(=O)OC ZINC000217994612 DD For-Sale Unstable LASB 0 40 CC(C)CN(CC(C)C)C(=O)N/C=C/c1cccc(F)c1 ZINC000217994649 CI For-Sale Unstable NR1H4 17 42 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000217994653 IG For-Sale Unstable MMP13 54 39 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000217994653 IG For-Sale Unstable CACNA1B 16 41 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000217994653 IG For-Sale Unstable ADAM17 25 41 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000217994653 IG For-Sale Unstable MMP2 28 54 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000217994653 IG For-Sale Unstable MMP3 63 39 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000217994653 IG For-Sale Unstable MMP8 33 41 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000217994653 IG For-Sale Unstable MMP7 57 39 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000217994653 IG For-Sale Unstable MMP1 53 39 N[C@H](CC(=O)O)c1cccc(Cl)c1C(F)F ZINC000217994663 BF For-Sale Unstable CXCL8 50 31 CC(C)[C@H](Br)C(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217994674 DH For-Sale Unstable DPP4 21 42 CC(C)[C@H](Br)C(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217994674 DH For-Sale Unstable DPP7 18 42 CC(C)[C@H](Br)C(=O)N1CCC[C@@H]2CCCC[C@H]21 ZINC000217994674 DH For-Sale Unstable DPP9 16 42 N[C@@H](CC(=O)O)c1cccc(Cl)c1C(F)F ZINC000217994737 BF For-Sale Unstable CXCL8 50 31 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000217994738 IG For-Sale Unstable MMP13 54 39 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000217994738 IG For-Sale Unstable CACNA1B 16 41 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000217994738 IG For-Sale Unstable ADAM17 25 41 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000217994738 IG For-Sale Unstable MMP2 28 54 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000217994738 IG For-Sale Unstable MMP3 63 39 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000217994738 IG For-Sale Unstable MMP8 33 41 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000217994738 IG For-Sale Unstable MMP7 57 39 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000217994738 IG For-Sale Unstable MMP1 53 39 CC(C)[C@@H](Br)C(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217994757 DH For-Sale Unstable DPP4 21 42 CC(C)[C@@H](Br)C(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217994757 DH For-Sale Unstable DPP7 18 42 CC(C)[C@@H](Br)C(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217994757 DH For-Sale Unstable DPP9 16 42 CC[C@H](C)[C@H](NC(=O)CS[C@@H](C(=O)O)C(C)C)C(=O)OC ZINC000217994781 DD For-Sale Unstable ENPEP 51 32 CC[C@H](C)[C@H](NC(=O)CS[C@@H](C(=O)O)C(C)C)C(=O)OC ZINC000217994781 DD For-Sale Unstable LASB 0 40 C[C@H]1CCC[C@H](C)N1C(=O)N[C@H](C)CC(=O)O ZINC000217994782 BD On-Demand Unstable EDNRB 48 39 Cc1ccc2[nH]c(CCNC(=O)C[C@@H]3C=CS(=O)(=O)C3)nc2c1 ZINC000217994792 ED In-Stock Unstable F9 27 52 Cc1ccc2[nH]c(CCNC(=O)C[C@@H]3C=CS(=O)(=O)C3)nc2c1 ZINC000217994792 ED In-Stock Unstable CYSP_TRYCR 0 51 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000217994814 IG For-Sale Unstable MMP13 54 39 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000217994814 IG For-Sale Unstable CACNA1B 16 41 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000217994814 IG For-Sale Unstable ADAM17 25 41 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000217994814 IG For-Sale Unstable MMP2 28 54 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000217994814 IG For-Sale Unstable MMP3 63 39 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000217994814 IG For-Sale Unstable MMP8 33 41 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000217994814 IG For-Sale Unstable MMP7 57 39 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000217994814 IG For-Sale Unstable MMP1 53 39 CCC[C@@H](NC(=O)NCc1ccc(F)cc1)C(=O)Nc1ccc(CN2CCOCC2)cc1 ZINC000217994818 IG On-Demand Unstable TACR2 27 46 CCC[C@@H](NC(=O)NCc1ccc(F)cc1)C(=O)Nc1ccc(CN2CCOCC2)cc1 ZINC000217994818 IG On-Demand Unstable CCR3 45 37 CCC[C@@H](NC(=O)NCc1ccc(F)cc1)C(=O)Nc1ccc(CN2CCOCC2)cc1 ZINC000217994818 IG On-Demand Unstable F2R 57 39 CCC[C@@H](NC(=O)NCc1ccc(F)cc1)C(=O)Nc1ccc(CN2CCOCC2)cc1 ZINC000217994818 IG On-Demand Unstable MLNR 42 36 CCC[C@@H](NC(=O)NCc1ccc(F)cc1)C(=O)Nc1ccc(CN2CCOCC2)cc1 ZINC000217994818 IG On-Demand Unstable EPHX2 22 43 C[C@@H](Sc1ccc(Cl)cc1)C(=O)NCc1nc(-c2ccccc2Cl)no1 ZINC000217994828 HJ In-Stock Unstable GPBAR1 26 40 O=C(N/C=C/c1cccc(F)c1)NC1CCCCCC1 ZINC000217994833 CH For-Sale Unstable FAAH 0 47 O=C(N/C=C/c1cccc(F)c1)NC1CCCCCC1 ZINC000217994833 CH For-Sale Unstable EPHX2 27 43 NC[C@@H](C(=O)O)c1cccc(Cl)c1C(F)F ZINC000217994834 BE For-Sale Unstable CXCL8 33 40 CCOC(=O)[C@H](Cc1cccc(C)c1)NC(=O)OC(C)(C)C ZINC000217994837 DF For-Sale Unstable TACR1 23 51 CCOC(=O)[C@H](Cc1cccc(C)c1)NC(=O)OC(C)(C)C ZINC000217994837 DF For-Sale Unstable PGC 57 38 CCOC(=O)[C@H](Cc1cccc(C)c1)NC(=O)OC(C)(C)C ZINC000217994837 DF For-Sale Unstable CMA1 43 36 CCOC(=O)[C@H](Cc1cccc(C)c1)NC(=O)OC(C)(C)C ZINC000217994837 DF For-Sale Unstable CTRA_BOVIN 23 44 CCOC(=O)[C@H](Cc1cccc(C)c1)NC(=O)OC(C)(C)C ZINC000217994837 DF For-Sale Unstable CTSB 47 42 CCOC(=O)[C@H](Cc1cccc(C)c1)NC(=O)OC(C)(C)C ZINC000217994837 DF For-Sale Unstable PAPA1_CARPA 72 53 CCOC(=O)[C@H](Cc1cccc(C)c1)NC(=O)OC(C)(C)C ZINC000217994837 DF For-Sale Unstable CYSP_TRYCR 54 37 CCOC(=O)[C@H](Cc1cccc(C)c1)NC(=O)OC(C)(C)C ZINC000217994837 DF For-Sale Unstable CCKAR 48 41 CCOC(=O)[C@H](Cc1cccc(C)c1)NC(=O)OC(C)(C)C ZINC000217994837 DF For-Sale Unstable CTSK 46 47 CCOC(=O)[C@H](Cc1cccc(C)c1)NC(=O)OC(C)(C)C ZINC000217994837 DF For-Sale Unstable CTSL 44 54 CCOC(=O)[C@H](Cc1cccc(C)c1)NC(=O)OC(C)(C)C ZINC000217994837 DF For-Sale Unstable CCR3 19 51 CCOC(=O)[C@H](Cc1cccc(C)c1)NC(=O)OC(C)(C)C ZINC000217994837 DF For-Sale Unstable SCN9A 31 40 CCOC(=O)[C@H](Cc1cccc(C)c1)NC(=O)OC(C)(C)C ZINC000217994837 DF For-Sale Unstable TACR3 17 43 CCOC(=O)[C@H](Cc1cccc(C)c1)NC(=O)OC(C)(C)C ZINC000217994837 DF For-Sale Unstable CAPNS1 49 35 CCOC(=O)[C@H](Cc1cccc(C)c1)NC(=O)OC(C)(C)C ZINC000217994837 DF For-Sale Unstable HLA-DRB1 57 38 CCOC(=O)[C@H](Cc1cccc(C)c1)NC(=O)OC(C)(C)C ZINC000217994837 DF For-Sale Unstable REN 59 47 CCOC(=O)[C@H](Cc1cccc(C)c1)NC(=O)OC(C)(C)C ZINC000217994837 DF For-Sale Unstable CTSS 45 54 CCOC(=O)[C@H](Cc1cccc(C)c1)NC(=O)OC(C)(C)C ZINC000217994837 DF For-Sale Unstable CAPN2 61 36 CCOC(=O)[C@H](Cc1cccc(C)c1)NC(=O)OC(C)(C)C ZINC000217994837 DF For-Sale Unstable EPHX2 17 48 CCOC(=O)[C@H](Cc1cccc(C)c1)NC(=O)OC(C)(C)C ZINC000217994837 DF For-Sale Unstable CTSV 35 40 CCOC(=O)[C@H](Cc1cccc(C)c1)NC(=O)OC(C)(C)C ZINC000217994837 DF For-Sale Unstable FPR1 58 44 CCOC(=O)[C@H](Cc1cccc(C)c1)NC(=O)OC(C)(C)C ZINC000217994837 DF For-Sale Unstable CTRB_BOVIN 60 59 COc1ccc([C@@H]2CC(=O)Oc3ccc4c(c32)O/C(=C\c2cccnc2)C4=O)cc1 ZINC000217994840 GI In-Stock Unstable DAPK3 20 41 COc1ccc([C@@H]2CC(=O)Oc3ccc4c(c32)O/C(=C\c2cccnc2)C4=O)cc1 ZINC000217994840 GI In-Stock Unstable CYP11B2 15 43 CC(C)[C@H](Br)C(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217994849 DH For-Sale Unstable DPP4 21 42 CC(C)[C@H](Br)C(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217994849 DH For-Sale Unstable DPP7 18 42 CC(C)[C@H](Br)C(=O)N1CCC[C@H]2CCCC[C@H]21 ZINC000217994849 DH For-Sale Unstable DPP9 16 42 Cc1ccc2[nH]c(CCNC(=O)C[C@H]3C=CS(=O)(=O)C3)nc2c1 ZINC000217994881 ED In-Stock Unstable F9 27 52 Cc1ccc2[nH]c(CCNC(=O)C[C@H]3C=CS(=O)(=O)C3)nc2c1 ZINC000217994881 ED In-Stock Unstable CYSP_TRYCR 0 51 CCC[C@H](NC(=O)NCc1ccc(F)cc1)C(=O)Nc1ccc(CN2CCOCC2)cc1 ZINC000217994898 IG On-Demand Unstable TACR2 27 46 CCC[C@H](NC(=O)NCc1ccc(F)cc1)C(=O)Nc1ccc(CN2CCOCC2)cc1 ZINC000217994898 IG On-Demand Unstable CCR3 45 37 CCC[C@H](NC(=O)NCc1ccc(F)cc1)C(=O)Nc1ccc(CN2CCOCC2)cc1 ZINC000217994898 IG On-Demand Unstable F2R 57 39 CCC[C@H](NC(=O)NCc1ccc(F)cc1)C(=O)Nc1ccc(CN2CCOCC2)cc1 ZINC000217994898 IG On-Demand Unstable MLNR 42 36 CCC[C@H](NC(=O)NCc1ccc(F)cc1)C(=O)Nc1ccc(CN2CCOCC2)cc1 ZINC000217994898 IG On-Demand Unstable EPHX2 22 43 C[C@H](Sc1ccc(Cl)cc1)C(=O)NCc1nc(-c2ccccc2Cl)no1 ZINC000217994904 HJ In-Stock Unstable GPBAR1 26 40 CCc1ncnc(NCc2ccccc2C(F)(F)F)c1F ZINC000217994907 CH On-Demand Unstable PTK2 42 34 NC[C@H](C(=O)O)c1cccc(Cl)c1C(F)F ZINC000217994911 BE For-Sale Unstable CXCL8 33 40 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1cccc(C(F)(F)F)c1 ZINC000217994920 IG For-Sale Unstable CACNA1B 57 39 COc1ccc([C@H]2CC(=O)Oc3ccc4c(c32)O/C(=C\c2cccnc2)C4=O)cc1 ZINC000217994929 GI In-Stock Unstable DAPK3 20 41 COc1ccc([C@H]2CC(=O)Oc3ccc4c(c32)O/C(=C\c2cccnc2)C4=O)cc1 ZINC000217994929 GI In-Stock Unstable CYP11B2 15 43 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1cccc(C(F)(F)F)c1 ZINC000217994989 IG For-Sale Unstable CACNA1B 57 39 O=C(Nc1ccc(CN2CCOCC2)cc1)c1cc(-c2ccccc2)nc2c1cnn2Cc1ccco1 ZINC000217995010 JJ On-Demand Unstable PIK3CA 21 42 O=C(Nc1ccc(CN2CCOCC2)cc1)c1cc(-c2ccccc2)nc2c1cnn2Cc1ccco1 ZINC000217995010 JJ On-Demand Unstable MTOR 35 41 CCc1ncnc(NCc2cccc(Br)c2)c1F ZINC000217995025 DH On-Demand Unstable ABL1 0 42 CCc1ncnc(NCc2cccc(Br)c2)c1F ZINC000217995025 DH On-Demand Unstable ADORA3 24 42 CCc1ncnc(NCc2cccc(Br)c2)c1F ZINC000217995025 DH On-Demand Unstable HTT 0 46 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](C)C(=O)NCc3ccccn3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217995040 KG In-Stock Unstable TUBA1A 18 62 COc1cc2c(c(OC)c1OC)-c1ccc(N[C@@H](C)C(=O)NCc3ccccn3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217995040 KG In-Stock Unstable TPPP 0 59 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1cccc(C(F)(F)F)c1 ZINC000217995072 IG For-Sale Unstable CACNA1B 57 39 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1cccc(C(F)(F)F)c1 ZINC000217995145 IG For-Sale Unstable CACNA1B 57 39 CCOc1ccccc1NC(=O)N/C=C/c1cccc(F)c1 ZINC000217995155 DI For-Sale Unstable P2RY1 20 41 COc1cccc(C(=O)NCC(=O)Nc2nc(CN3CCC(C)CC3)cs2)c1 ZINC000217995161 HF On-Demand Unstable DRD4 53 41 COc1cccc(C(=O)NCC(=O)Nc2nc(CN3CCC(C)CC3)cs2)c1 ZINC000217995161 HF On-Demand Unstable CCR3 17 45 COc1cccc(C(=O)NCC(=O)Nc2nc(CN3CCC(C)CC3)cs2)c1 ZINC000217995161 HF On-Demand Unstable CCR2 37 44 COc1cccc(C(=O)NCC(=O)Nc2nc(CN3CCC(C)CC3)cs2)c1 ZINC000217995161 HF On-Demand Unstable MCHR1 24 41 COc1cccc(C(=O)NCC(=O)Nc2nc(CN3CCC(C)CC3)cs2)c1 ZINC000217995161 HF On-Demand Unstable TRPC6 47 39 O=C(O)Cc1cc(I)c(Cc2cc(I)c(O)c(I)c2)c(I)c1 ZINC000217995231 KK For-Sale Unstable THRA 27 44 O=C(O)Cc1cc(I)c(Cc2cc(I)c(O)c(I)c2)c(I)c1 ZINC000217995231 KK For-Sale Unstable THRB 21 40 COc1ccccc1C(=O)NCC(=O)Nc1nc(CN2CCC(C)CC2)cs1 ZINC000217995272 HF On-Demand Unstable DRD2 21 41 COc1ccccc1C(=O)NCC(=O)Nc1nc(CN2CCC(C)CC2)cs1 ZINC000217995272 HF On-Demand Unstable DRD4 31 41 COc1ccccc1C(=O)NCC(=O)Nc1nc(CN2CCC(C)CC2)cs1 ZINC000217995272 HF On-Demand Unstable KCNA3 42 38 COc1ccccc1C(=O)NCC(=O)Nc1nc(CN2CCC(C)CC2)cs1 ZINC000217995272 HF On-Demand Unstable HCN1 62 36 COc1ccccc1C(=O)NCC(=O)Nc1nc(CN2CCC(C)CC2)cs1 ZINC000217995272 HF On-Demand Unstable HCN4 51 35 COc1ccccc1C(=O)NCC(=O)Nc1nc(CN2CCC(C)CC2)cs1 ZINC000217995272 HF On-Demand Unstable TRPC6 46 36 Nc1nc(C2CC(N)C2)cc(N2CCCN(Cc3cccc(F)c3)CC2)n1 ZINC000217995355 FE In-Stock Unstable HRH4 25 43 COc1ccc(OCCNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217995358 EG For-Sale Unstable HRH2 23 41 COc1ccc(OCCNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217995358 EG For-Sale Unstable MTNR1A 75 48 COc1ccc(OCCNC(=O)N/C=C/c2cccc(F)c2)cc1 ZINC000217995358 EG For-Sale Unstable MTNR1B 62 48 CCCOc1ccc([C@@H](NCC)[C@@H]2CCC[C@@H](C)C2)cc1 ZINC000217995375 CJ For-Sale Unstable ACACA 30 41 CCCOc1ccc([C@H](NCC)[C@@H]2CCC[C@@H](C)C2)cc1 ZINC000217995450 CJ For-Sale Unstable ACACA 30 41 CCc1nccn1CCNC(=O)c1ccc2[nH]c(=O)c(=O)[nH]c2c1 ZINC000217995459 EC In-Stock Unstable DRD4 41 32 CCc1nccn1CCNC(=O)c1ccc2[nH]c(=O)c(=O)[nH]c2c1 ZINC000217995459 EC In-Stock Unstable PLD2 63 36 CCCOc1ccc([C@@H](NCC)[C@H]2CCC[C@@H](C)C2)cc1 ZINC000217995531 CJ For-Sale Unstable ACACA 30 41 COc1ccc2[nH]c3c(c2c1)CCC[C@@H]3NC(=O)c1n[nH]c2c1Cc1cc(OC)c(OC)cc1-2 ZINC000217995533 JI In-Stock Unstable MAPKAPK2 0 41 COc1ccc2[nH]c3c(c2c1)CCC[C@@H]3NC(=O)c1n[nH]c2c1Cc1cc(OC)c(OC)cc1-2 ZINC000217995533 JI In-Stock Unstable CHEK1 40 39 CN1CCN(c2ccc(C(=O)N3CC[C@@H]3c3ccc(F)cc3)cc2)CC1 ZINC000217995555 FG In-Stock Unstable SSTR1 18 40 CN1CCN(c2ccc(C(=O)N3CC[C@@H]3c3ccc(F)cc3)cc2)CC1 ZINC000217995555 FG In-Stock Unstable SLC6A7 0 46 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OCC(C)C)cc1 ZINC000217995594 JG For-Sale Unstable MMP13 87 47 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OCC(C)C)cc1 ZINC000217995594 JG For-Sale Unstable ADAM17 68 45 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OCC(C)C)cc1 ZINC000217995594 JG For-Sale Unstable MMP2 44 50 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OCC(C)C)cc1 ZINC000217995594 JG For-Sale Unstable MMP3 87 47 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OCC(C)C)cc1 ZINC000217995594 JG For-Sale Unstable MMP8 36 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OCC(C)C)cc1 ZINC000217995594 JG For-Sale Unstable MMP9 48 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OCC(C)C)cc1 ZINC000217995594 JG For-Sale Unstable MMP7 76 40 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OCC(C)C)cc1 ZINC000217995594 JG For-Sale Unstable MMP1 86 47 CCc1ncnc(NCc2ccc(F)cc2F)c1F ZINC000217995605 CG On-Demand Unstable USP10 0 40 CCc1ncnc(NCc2ccc(F)cc2F)c1F ZINC000217995605 CG On-Demand Unstable USP13 0 40 COc1ccc2[nH]c3c(c2c1)CCC[C@H]3NC(=O)c1n[nH]c2c1Cc1cc(OC)c(OC)cc1-2 ZINC000217995614 JI In-Stock Unstable MAPKAPK2 0 41 COc1ccc2[nH]c3c(c2c1)CCC[C@H]3NC(=O)c1n[nH]c2c1Cc1cc(OC)c(OC)cc1-2 ZINC000217995614 JI In-Stock Unstable CHEK1 40 39 CCCOc1ccc([C@H](NCC)[C@H]2CCC[C@@H](C)C2)cc1 ZINC000217995621 CJ For-Sale Unstable ACACA 30 41 CN1CCN(c2ccc(C(=O)N3CC[C@H]3c3ccc(F)cc3)cc2)CC1 ZINC000217995635 FG In-Stock Unstable SSTR1 18 40 CN1CCN(c2ccc(C(=O)N3CC[C@H]3c3ccc(F)cc3)cc2)CC1 ZINC000217995635 FG In-Stock Unstable SLC6A7 0 46 CCc1c(C)nn(-c2cc(Cl)ccc2CBr)c1C ZINC000217995643 EJ For-Sale Unstable P2RX7 23 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OCC(C)C)cc1 ZINC000217995670 JG For-Sale Unstable MMP13 87 47 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OCC(C)C)cc1 ZINC000217995670 JG For-Sale Unstable ADAM17 68 45 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OCC(C)C)cc1 ZINC000217995670 JG For-Sale Unstable MMP2 44 50 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OCC(C)C)cc1 ZINC000217995670 JG For-Sale Unstable MMP3 87 47 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OCC(C)C)cc1 ZINC000217995670 JG For-Sale Unstable MMP8 36 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OCC(C)C)cc1 ZINC000217995670 JG For-Sale Unstable MMP9 48 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OCC(C)C)cc1 ZINC000217995670 JG For-Sale Unstable MMP7 76 40 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OCC(C)C)cc1 ZINC000217995670 JG For-Sale Unstable MMP1 86 47 C[C@@](O)(CNC(=O)c1noc2c1CCCC2)c1cc2ccccc2o1 ZINC000217995697 EF In-Stock Unstable PANC 57 40 Cc1cc2c(cnn2-c2ccc(F)cc2)cc1C=O ZINC000217995740 CG For-Sale Unstable NR3C1 23 47 Nc1cc(O)nc(CCNC(=O)c2ccc(CN3CCCCCC3)cc2)n1 ZINC000217995747 FE In-Stock Unstable TGFBR1 0 40 C[C@@H](Sc1ccc(Cl)cc1)C(=O)N(C)Cc1nc(-c2ccccc2Cl)no1 ZINC000217995756 HK In-Stock Unstable GPBAR1 24 42 C[C@](O)(CNC(=O)c1noc2c1CCCC2)c1cc2ccccc2o1 ZINC000217995778 EF In-Stock Unstable PANC 57 40 CCCOc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1C ZINC000217995787 JG For-Sale Unstable MMP13 40 38 CCCOc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1C ZINC000217995787 JG For-Sale Unstable MMP3 41 38 CCCOc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1C ZINC000217995787 JG For-Sale Unstable MMP7 50 37 O=C(N/C=C/c1cccc(F)c1)NC12CC3CC(CC(C3)C1)C2 ZINC000217995797 DI For-Sale Unstable EPHX2 99 47 C[C@H](Sc1ccc(Cl)cc1)C(=O)N(C)Cc1nc(-c2ccccc2Cl)no1 ZINC000217995834 HK In-Stock Unstable GPBAR1 24 42 CCCOc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1C ZINC000217995858 JG For-Sale Unstable MMP13 40 38 CCCOc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1C ZINC000217995858 JG For-Sale Unstable MMP3 41 38 CCCOc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1C ZINC000217995858 JG For-Sale Unstable MMP7 50 37 O=C(N/C=C/c1cccc(F)c1)Nc1cccc2cccnc12 ZINC000217995899 DI For-Sale Anodyne PFHDAC1 0 41 CCc1ccc(CNc2ncnc(CC)c2F)cc1 ZINC000217995948 CG On-Demand Unstable USP10 0 48 CCc1ccc(CNc2ncnc(CC)c2F)cc1 ZINC000217995948 CG On-Demand Unstable USP13 0 48 O=C(N[C@@H]1CCOC[C@H]1OCc1ccccc1)c1nccnc1O ZINC000217995982 ED In-Stock Unstable KLK5 41 38 O=C(CSCc1ccc(F)cc1)N[C@@H]1CCC[C@@H]1CO ZINC000217996034 CE For-Sale Unstable SSTR3 20 43 COC(=O)C[C@H](C1=Cc2ccccc2OC1)c1oc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c1O ZINC000217996042 KG In-Stock Unstable CHRNA4 26 42 COc1ccnc(C(=O)N[C@@H](C)c2n[nH]c(C)n2)c1 ZINC000217996099 CD In-Stock Unstable Q8MMZ8_EIMTE 40 35 O=C(CSCc1ccc(F)cc1)N[C@H]1CCC[C@@H]1CO ZINC000217996122 CE For-Sale Unstable SSTR3 20 43 COC(=O)C[C@@H](C1=Cc2ccccc2OC1)c1oc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c1O ZINC000217996131 KG In-Stock Unstable CHRNA4 26 42 C[C@@H]1Cc2ccccc2N1C(=O)N/C=C/c1cccc(F)c1 ZINC000217996137 CH For-Sale Unstable DRD4 27 54 COc1ccnc(C(=O)N[C@H](C)c2n[nH]c(C)n2)c1 ZINC000217996188 CD In-Stock Unstable Q8MMZ8_EIMTE 40 35 O=C(CSCc1ccc(F)cc1)N[C@@H]1CCC[C@H]1CO ZINC000217996212 CE For-Sale Unstable SSTR3 20 43 C[C@H]1Cc2ccccc2N1C(=O)N/C=C/c1cccc(F)c1 ZINC000217996214 CH For-Sale Unstable DRD4 27 54 Cc1noc(C)c1CO[C@H]1CCOC[C@H]1NC(=O)c1ccc(CN)cc1 ZINC000217996283 FD In-Stock Unstable ADAM17 18 40 C[C@@H]1CN(Cc2csc(NC(=O)CNC(=O)c3ccc(C(F)(F)F)cc3)n2)C[C@@H](C)O1 ZINC000217996286 JG On-Demand Unstable CCR2 76 38 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1Nc1ccccc1N(C)C ZINC000217996321 CJ For-Sale Unstable TRPM8 17 46 COc1ccc(CC[C@@H](C)N[C@@H]2CCC[C@@H](C)C2)cc1 ZINC000217996330 CI For-Sale Unstable SLC18A2 31 43 COc1ccc(CC[C@@H](C)N[C@@H]2CCC[C@@H](C)C2)cc1 ZINC000217996330 CI For-Sale Unstable ACACA 0 44 COc1ccc(CC[C@@H](C)N[C@@H]2CCC[C@@H](C)C2)cc1 ZINC000217996330 CI For-Sale Unstable BIRC2 24 41 C[C@H]1CN(Cc2csc(NC(=O)CNC(=O)c3ccc(C(F)(F)F)cc3)n2)C[C@@H](C)O1 ZINC000217996372 JG On-Demand Unstable CCR2 76 38 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1Nc1ccccc1N(C)C ZINC000217996401 CJ For-Sale Unstable TRPM8 17 46 COc1ccc(CC[C@@H](C)N[C@H]2CCC[C@@H](C)C2)cc1 ZINC000217996414 CI For-Sale Unstable SLC18A2 31 43 COc1ccc(CC[C@@H](C)N[C@H]2CCC[C@@H](C)C2)cc1 ZINC000217996414 CI For-Sale Unstable ACACA 0 44 COc1ccc(CC[C@@H](C)N[C@H]2CCC[C@@H](C)C2)cc1 ZINC000217996414 CI For-Sale Unstable BIRC2 24 41 COc1ccccc1CNC(=O)N/C=C/c1cccc(F)c1 ZINC000217996444 DG For-Sale Unstable GRIN2B 0 49 COc1ccccc1CNC(=O)N/C=C/c1cccc(F)c1 ZINC000217996444 DG For-Sale Unstable ACKR3 61 38 COC(=O)C[C@@H]1c2cccnc2Oc2cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc3c21 ZINC000217996455 II In-Stock Unstable AKR1B1 0 45 COC(=O)Cn1cc(NC(=O)c2ccn(C)n2)cn1 ZINC000217996456 CC On-Demand Unstable PANC 52 34 C[C@H]1CN(Cc2csc(NC(=O)CNC(=O)c3ccc(C(F)(F)F)cc3)n2)C[C@H](C)O1 ZINC000217996461 JG On-Demand Unstable CCR2 76 38 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1Nc1ccccc1N(C)C ZINC000217996478 CJ For-Sale Unstable TRPM8 17 46 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217996525 JG For-Sale Unstable MMP13 70 46 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217996525 JG For-Sale Unstable ADAM17 41 41 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217996525 JG For-Sale Unstable MMP2 41 52 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217996525 JG For-Sale Unstable MMP3 79 42 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217996525 JG For-Sale Unstable MMP9 44 46 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217996525 JG For-Sale Unstable MMP7 76 39 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217996525 JG For-Sale Unstable MMP1 71 46 COC(=O)C[C@H]1c2cccnc2Oc2cc(O)c3c(=O)cc(-c4ccc(O)cc4)oc3c21 ZINC000217996539 II In-Stock Unstable AKR1B1 0 45 O=C(N/C=C/c1cccc(F)c1)N1CCN(c2ncccn2)CC1 ZINC000217996544 EE For-Sale Unstable FAAH 28 43 O=C(N/C=C/c1cccc(F)c1)N1CCN(c2ncccn2)CC1 ZINC000217996544 EE For-Sale Unstable SLC6A7 0 45 CC(C)[C@H]1CC[C@H](C)C[C@@H]1Nc1ccccc1N(C)C ZINC000217996565 CJ For-Sale Unstable TRPM8 17 46 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217996616 JG For-Sale Unstable MMP13 70 46 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217996616 JG For-Sale Unstable ADAM17 41 41 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217996616 JG For-Sale Unstable MMP2 41 52 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217996616 JG For-Sale Unstable MMP3 79 42 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217996616 JG For-Sale Unstable MMP9 44 46 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217996616 JG For-Sale Unstable MMP7 76 39 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217996616 JG For-Sale Unstable MMP1 71 46 N#C[C@@]1(C(=O)O)C[C@@H]1S(=O)(=O)c1ccc(Cl)cc1 ZINC000217996701 CD In-Stock Unstable ADAMTS5 24 41 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217996705 JG For-Sale Unstable MMP13 70 46 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217996705 JG For-Sale Unstable ADAM17 41 41 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217996705 JG For-Sale Unstable MMP2 41 52 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217996705 JG For-Sale Unstable MMP3 79 42 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217996705 JG For-Sale Unstable MMP9 44 46 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217996705 JG For-Sale Unstable MMP7 76 39 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217996705 JG For-Sale Unstable MMP1 71 46 C[C@@H](Sc1ccc(Cl)cc1)C(=O)NCCCN1CCCc2ccccc21 ZINC000217996711 GJ In-Stock Unstable DRD2 15 40 C[C@@H](Sc1ccc(Cl)cc1)C(=O)NCCCN1CCCc2ccccc21 ZINC000217996711 GJ In-Stock Unstable MC4R 32 41 CCOC(=O)N1CCC(NC(=O)N/C=C/c2cccc(F)c2)CC1 ZINC000217996772 EF For-Sale Unstable GRIN2B 16 40 CC[C@@H](CCO)Nc1ccnc(C)c1 ZINC000217996777 AD On-Demand Unstable ISPA 0 51 N#C[C@]1(C(=O)O)C[C@@H]1S(=O)(=O)c1ccc(Cl)cc1 ZINC000217996784 CD In-Stock Unstable ADAMTS5 24 41 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217996790 JG For-Sale Unstable MMP13 70 46 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217996790 JG For-Sale Unstable ADAM17 41 41 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217996790 JG For-Sale Unstable MMP2 41 52 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217996790 JG For-Sale Unstable MMP3 79 42 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217996790 JG For-Sale Unstable MMP9 44 46 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217996790 JG For-Sale Unstable MMP7 76 39 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000217996790 JG For-Sale Unstable MMP1 71 46 C[C@H](Sc1ccc(Cl)cc1)C(=O)NCCCN1CCCc2ccccc21 ZINC000217996802 GJ In-Stock Unstable DRD2 15 40 C[C@H](Sc1ccc(Cl)cc1)C(=O)NCCCN1CCCc2ccccc21 ZINC000217996802 GJ In-Stock Unstable MC4R 32 41 COc1ccc([C@@H](NC(=O)CCc2nc3ccccc3[nH]2)[C@@H]2C[C@H](O)C2)cn1 ZINC000217996822 GF In-Stock Unstable CYSP_TRYCR 0 40 COc1ccc([C@@H](NC(=O)CCc2nc3ccccc3[nH]2)[C@@H]2C[C@H](O)C2)cn1 ZINC000217996822 GF In-Stock Unstable PARP3 22 40 CC[C@H](CCO)Nc1ccnc(C)c1 ZINC000217996846 AD On-Demand Unstable ISPA 0 51 N#C[C@@]1(C(=O)O)C[C@H]1S(=O)(=O)c1ccc(Cl)cc1 ZINC000217996863 CD In-Stock Unstable ADAMTS5 24 41 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)NC[C@@H]3CCCO3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217996878 KF In-Stock Unstable TUBA1A 18 65 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)NC[C@@H]3CCCO3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217996878 KF In-Stock Unstable TPPP 0 62 COc1ccc([C@H](NC(=O)CCc2nc3ccccc3[nH]2)[C@@H]2C[C@H](O)C2)cn1 ZINC000217996904 GF In-Stock Unstable CYSP_TRYCR 0 40 COc1ccc([C@H](NC(=O)CCc2nc3ccccc3[nH]2)[C@@H]2C[C@H](O)C2)cn1 ZINC000217996904 GF In-Stock Unstable PARP3 22 40 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1cccc(Br)c1 ZINC000217996914 EJ For-Sale Unstable TRPM8 23 75 O=C(Nc1cc([N+](=O)[O-])ccc1Cl)c1ccc(CSc2ccccc2)cc1 ZINC000217996920 GK In-Stock Unstable HDAC1 22 40 N#C[C@]1(C(=O)O)C[C@H]1S(=O)(=O)c1ccc(Cl)cc1 ZINC000217996957 CD In-Stock Unstable ADAMTS5 24 41 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)NC[C@H]3CCCO3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217996966 KF In-Stock Unstable TUBA1A 18 65 COc1cc2c(c(OC)c1OC)-c1ccc(NCC(=O)NC[C@H]3CCCO3)c(=O)cc1[C@@H](NC(C)=O)CC2 ZINC000217996966 KF In-Stock Unstable TPPP 0 62 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1cccc(Br)c1 ZINC000217996992 EJ For-Sale Unstable TRPM8 23 75 Cc1ccc2nc(-c3ccc(NC(=O)N/C=C/c4cccc(F)c4)cc3)sc2c1 ZINC000217996997 HK For-Sale Unstable APP 24 49 CC(C)Oc1cccc(CNC(=O)c2ccc(CSc3ccccc3)cc2)c1 ZINC000217997030 GK In-Stock Unstable PRSS1 18 43 CC(C)Oc1cccc(CNC(=O)c2ccc(CSc3ccccc3)cc2)c1 ZINC000217997030 GK In-Stock Unstable PPARA 16 46 CC(C)Oc1cccc(CNC(=O)c2ccc(CSc3ccccc3)cc2)c1 ZINC000217997030 GK In-Stock Unstable ANPEP 17 41 CC(C)Oc1cccc(CNC(=O)c2ccc(CSc3ccccc3)cc2)c1 ZINC000217997030 GK In-Stock Unstable PDS 65 38 CCc1c(C)nn(-c2ccc(F)cc2CBr)c1C ZINC000217997059 DI For-Sale Unstable P2RX7 26 41 COC(=O)C[C@H](c1ccsc1)c1oc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c1O ZINC000217997064 JF In-Stock Unstable CHRNA4 27 44 CCCC[C@@H](NC(=O)N1C[C@H](C)C[C@@H](C)C1)C(=O)O ZINC000217997069 CE For-Sale Unstable NOD1 90 45 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)c1cccc(Br)c1 ZINC000217997074 EJ For-Sale Unstable TRPM8 23 75 O=C(N/C=C/c1cccc(F)c1)Nc1ccc2c(c1)OCO2 ZINC000217997098 DG For-Sale Unstable CCR2 0 42 O=C(N/C=C/c1cccc(F)c1)Nc1ccc2c(c1)OCO2 ZINC000217997098 DG For-Sale Unstable IMPDH2 0 47 COc1ccc(CNC(=O)c2ccc(CSc3ccccc3)cc2)c(OC)c1OC ZINC000217997133 HJ In-Stock Unstable PPARG 17 48 COc1ccc(CNC(=O)c2ccc(CSc3ccccc3)cc2)c(OC)c1OC ZINC000217997133 HJ In-Stock Unstable PPARA 21 48 COc1ccc(CNC(=O)c2ccc(CSc3ccccc3)cc2)c(OC)c1OC ZINC000217997133 HJ In-Stock Unstable PPARD 28 48 COc1ccc(CNC(=O)c2ccc(CSc3ccccc3)cc2)c(OC)c1OC ZINC000217997133 HJ In-Stock Unstable SLC9A1 57 33 COc1ccc(CNC(=O)c2ccc(CSc3ccccc3)cc2)c(OC)c1OC ZINC000217997133 HJ In-Stock Unstable MT-ND1 23 40 CCCC[C@H](NC(=O)N1C[C@H](C)C[C@@H](C)C1)C(=O)O ZINC000217997140 CE For-Sale Unstable NOD1 90 45 CO/C(=C/c1ccccc1)CO ZINC000217997147 AD For-Sale Unstable LSDA 41 33 CO/C(=C/c1ccccc1)CO ZINC000217997147 AD For-Sale Unstable TLR4 29 52 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)c1cccc(Br)c1 ZINC000217997154 EJ For-Sale Unstable TRPM8 23 75 COC(=O)C[C@@H](c1ccsc1)c1oc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c1O ZINC000217997156 JF In-Stock Unstable CHRNA4 27 44 CC(C)(C)OC(=O)NCCNc1cnn(CC(=O)NC2CC2)c1 ZINC000217997177 DD For-Sale Unstable PANC 52 34 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1ccccc1Br ZINC000217997237 EJ For-Sale Unstable TRPM8 22 60 CCOc1ccc(CNC(=O)c2ccc(CSc3ccccc3)cc2)cc1OCC ZINC000217997247 HK In-Stock Unstable PPARG 15 41 CCOc1ccc(CNC(=O)c2ccc(CSc3ccccc3)cc2)cc1OCC ZINC000217997247 HK In-Stock Unstable PPARA 20 43 CCOc1ccc(CNC(=O)c2ccc(CSc3ccccc3)cc2)cc1OCC ZINC000217997247 HK In-Stock Unstable PPARD 26 40 CCOc1ccc(CNC(=O)c2ccc(CSc3ccccc3)cc2)cc1OCC ZINC000217997247 HK In-Stock Unstable MT-ND1 17 43 CCOc1ccc(CNC(=O)c2ccc(CSc3ccccc3)cc2)cc1OCC ZINC000217997247 HK In-Stock Unstable PDS 42 34 COC(=O)C[C@@H](c1cc(OC)c(OC)cc1OC)c1oc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c1O ZINC000217997269 KF In-Stock Unstable CHRNA4 26 44 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1ccccc1Br ZINC000217997323 EJ For-Sale Unstable TRPM8 22 60 O=C(N/C=C/c1cccc(F)c1)Nc1cccc(F)c1 ZINC000217997326 CH For-Sale Anodyne IMPDH2 0 44 O=C(N/C=C/c1cccc(F)c1)Nc1cccc(F)c1 ZINC000217997326 CH For-Sale Anodyne MMP1 0 56 O=C(N/C=C/c1cccc(F)c1)Nc1cccc(F)c1 ZINC000217997326 CH For-Sale Anodyne KCNK3 15 42 COC(=O)C[C@H](c1cc(OC)c(OC)cc1OC)c1oc(CN2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)cc(=O)c1O ZINC000217997343 KF In-Stock Unstable CHRNA4 26 44 COc1cc(CNC(=O)c2ccc(CSc3ccccc3)cc2)ccc1OC(C)C ZINC000217997358 HK In-Stock Unstable PPARA 20 45 COc1cc(CNC(=O)c2ccc(CSc3ccccc3)cc2)ccc1OC(C)C ZINC000217997358 HK In-Stock Unstable PPARD 26 45 COc1cc(CNC(=O)c2ccc(CSc3ccccc3)cc2)ccc1OC(C)C ZINC000217997358 HK In-Stock Unstable MT-ND1 28 50 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)c1ccccc1Br ZINC000217997404 EJ For-Sale Unstable TRPM8 23 62 CCC[C@@H](NC(=O)N1C[C@H](C)C[C@@H](C)C1)C(=O)O ZINC000217997411 CD For-Sale Unstable NOD1 60 38 COC(=O)c1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217997461 ID For-Sale Unstable MMP13 55 40 COC(=O)c1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217997461 ID For-Sale Unstable MMP2 27 55 COC(=O)c1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217997461 ID For-Sale Unstable MMP3 64 40 COC(=O)c1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217997461 ID For-Sale Unstable MMP7 61 38 COC(=O)c1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217997461 ID For-Sale Unstable MMP1 57 40 C[C@@](O)(CNS(=O)(=O)c1cccc(Cl)c1)c1cc2ccccc2o1 ZINC000217997473 FG In-Stock Unstable FBP1 34 40 Cc1ccc(C)c([C@@H](C)NC(=O)c2ccc(CSc3ccccc3)cc2)c1 ZINC000217997476 GK In-Stock Unstable UTS2 40 37 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)c1ccccc1Br ZINC000217997486 EJ For-Sale Unstable TRPM8 23 62 CCC[C@H](NC(=O)N1C[C@H](C)C[C@@H](C)C1)C(=O)O ZINC000217997497 CD For-Sale Unstable NOD1 60 38 COC(=O)c1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217997547 ID For-Sale Unstable MMP13 55 40 COC(=O)c1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217997547 ID For-Sale Unstable MMP2 27 55 COC(=O)c1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217997547 ID For-Sale Unstable MMP3 64 40 COC(=O)c1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217997547 ID For-Sale Unstable MMP7 61 38 COC(=O)c1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217997547 ID For-Sale Unstable MMP1 57 40 CC(C)(C)OC(=O)NCCNc1cnn(Cc2ccccc2)c1 ZINC000217997548 DF For-Sale Unstable PAPA1_CARPA 29 43 CC(C)(C)OC(=O)NCCNc1cnn(Cc2ccccc2)c1 ZINC000217997548 DF For-Sale Unstable ITK 33 46 CC(C)(C)OC(=O)NCCNc1cnn(Cc2ccccc2)c1 ZINC000217997548 DF For-Sale Unstable FPR1 41 34 CC(C)(C)OC(=O)NCCNc1cnn(Cc2ccccc2)c1 ZINC000217997548 DF For-Sale Unstable PANC 64 47 Cc1ccc(C)c([C@H](C)NC(=O)c2ccc(CSc3ccccc3)cc2)c1 ZINC000217997556 GK In-Stock Unstable UTS2 40 37 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1ccc(Br)cc1 ZINC000217997558 EJ For-Sale Unstable TRPM8 23 76 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1ccc(Br)cc1 ZINC000217997558 EJ For-Sale Unstable PHZR 0 43 COc1ccc(C(=O)C2CCN(C(=O)c3nn(-c4ccccc4)cc3O)CC2)cc1 ZINC000217997560 HG On-Demand Unstable SLC18A3 45 52 COc1ccc(C(=O)C2CCN(C(=O)c3nn(-c4ccccc4)cc3O)CC2)cc1 ZINC000217997560 HG On-Demand Unstable L3MBTL3 42 34 C[C@](O)(CNS(=O)(=O)c1cccc(Cl)c1)c1cc2ccccc2o1 ZINC000217997562 FG In-Stock Unstable FBP1 34 40 COc1coc(C(=O)NC[C@@H]2CCCO2)cc1=O ZINC000217997648 CC On-Demand Unstable OXTR 0 40 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1ccc(Br)cc1 ZINC000217997654 EJ For-Sale Unstable TRPM8 23 76 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1ccc(Br)cc1 ZINC000217997654 EJ For-Sale Unstable PHZR 0 43 O=C(NCCCc1ccccc1Cl)c1ccc(CSc2ccccc2)cc1 ZINC000217997679 GK In-Stock Unstable DRD3 27 45 COc1coc(C(=O)NC[C@H]2CCCO2)cc1=O ZINC000217997733 CC On-Demand Unstable OXTR 0 40 O=C(N/C=C/c1cccc(F)c1)NCCc1c[nH]c2ccccc12 ZINC000217997736 DH For-Sale Unstable NQO2 16 40 O=C(N/C=C/c1cccc(F)c1)NCCc1c[nH]c2ccccc12 ZINC000217997736 DH For-Sale Unstable CCKAR 21 40 O=C(N/C=C/c1cccc(F)c1)NCCc1c[nH]c2ccccc12 ZINC000217997736 DH For-Sale Unstable MPO 93 41 O=C(N/C=C/c1cccc(F)c1)NCCc1c[nH]c2ccccc12 ZINC000217997736 DH For-Sale Unstable NMBR 28 42 O=C(N/C=C/c1cccc(F)c1)NCCc1c[nH]c2ccccc12 ZINC000217997736 DH For-Sale Unstable MTNR1A 21 43 O=C(N/C=C/c1cccc(F)c1)NCCc1c[nH]c2ccccc12 ZINC000217997736 DH For-Sale Unstable MTNR1B 16 41 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)c1ccc(Br)cc1 ZINC000217997744 EJ For-Sale Unstable TRPM8 23 76 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)c1ccc(Br)cc1 ZINC000217997744 EJ For-Sale Unstable PHZR 0 43 COc1ccc(-c2n[nH]cc2C(=O)N2CCN(Cc3cc(F)ccc3OC)CC2)cc1 ZINC000217997770 HG On-Demand Unstable CCKAR 23 40 COc1ccc(-c2n[nH]cc2C(=O)N2CCN(Cc3cc(F)ccc3OC)CC2)cc1 ZINC000217997770 HG On-Demand Unstable TACR3 22 49 O=C(NCCCc1ccc(Cl)cc1)c1ccc(CSc2ccccc2)cc1 ZINC000217997787 GK In-Stock Unstable DRD3 18 41 O=C(NCCCc1ccc(Cl)cc1)c1ccc(CSc2ccccc2)cc1 ZINC000217997787 GK In-Stock Unstable SCN5A 0 47 O=C(NCCCc1ccc(Cl)cc1)c1ccc(CSc2ccccc2)cc1 ZINC000217997787 GK In-Stock Unstable SLC6A5 21 43 O=C(NCCCc1ccc(Cl)cc1)c1ccc(CSc2ccccc2)cc1 ZINC000217997787 GK In-Stock Unstable HAO1 22 41 O=C(NCCCc1ccc(Cl)cc1)c1ccc(CSc2ccccc2)cc1 ZINC000217997787 GK In-Stock Unstable CRTM 41 41 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)c1ccc(Br)cc1 ZINC000217997824 EJ For-Sale Unstable TRPM8 23 76 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)c1ccc(Br)cc1 ZINC000217997824 EJ For-Sale Unstable PHZR 0 43 COc1ccc(N2C[C@H](C(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)CC2=O)c(OC)c1 ZINC000217997855 ID In-Stock Unstable CHRNA4 25 41 CC(=O)Nc1ccc(S(=O)(=O)NC[C@](C)(O)c2cc3ccccc3o2)cc1 ZINC000217997881 GF In-Stock Unstable ALOX15 18 41 CC(=O)Nc1ccc(S(=O)(=O)NC[C@](C)(O)c2cc3ccccc3o2)cc1 ZINC000217997881 GF In-Stock Unstable IDO1 33 42 COc1ccc(F)cc1CN1CCN(C(=O)C[C@@H](NC(N)=O)c2cccs2)CC1 ZINC000217997887 HE On-Demand Unstable SLC9A1 40 36 O=C(NCCCc1ccc(F)cc1)c1ccc(CSc2ccccc2)cc1 ZINC000217997896 GK In-Stock Unstable DRD3 19 40 O=C(NCCCc1ccc(F)cc1)c1ccc(CSc2ccccc2)cc1 ZINC000217997896 GK In-Stock Unstable BCHE 22 43 O=C(NCCCc1ccc(F)cc1)c1ccc(CSc2ccccc2)cc1 ZINC000217997896 GK In-Stock Unstable KCNA3 0 42 O=C(NCCCc1ccc(F)cc1)c1ccc(CSc2ccccc2)cc1 ZINC000217997896 GK In-Stock Unstable EPHX2 0 46 O=C(NCCCc1ccc(F)cc1)c1ccc(CSc2ccccc2)cc1 ZINC000217997896 GK In-Stock Unstable HAO1 22 41 O=C(NCCCc1ccc(F)cc1)c1ccc(CSc2ccccc2)cc1 ZINC000217997896 GK In-Stock Unstable CRTM 29 41 C#CC[C@H](O)CCCC=O ZINC000217997903 AC For-Sale Unstable CYP4A4 50 34 CCC(CC)(CN[C@@H](C)c1ccccc1)NC(=O)OC(C)(C)C ZINC000217997910 DI For-Sale Unstable PAPA1_CARPA 40 36 CCC(CC)(CN[C@@H](C)c1ccccc1)NC(=O)OC(C)(C)C ZINC000217997910 DI For-Sale Unstable CTSK 22 45 CCC(CC)(CN[C@@H](C)c1ccccc1)NC(=O)OC(C)(C)C ZINC000217997910 DI For-Sale Unstable FPR1 43 35 CCC(CC)(CN[C@@H](C)c1ccccc1)NC(=O)OC(C)(C)C ZINC000217997910 DI For-Sale Unstable POL 0 43 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1ccc(F)cc1Br ZINC000217997917 FJ For-Sale Unstable TRPM8 20 56 COc1ccc(N2C[C@@H](C(=O)N3C[C@@H]4C[C@H](C3)c3cccc(=O)n3C4)CC2=O)c(OC)c1 ZINC000217997945 ID In-Stock Unstable CHRNA4 25 41 CC(=O)Nc1ccc(S(=O)(=O)NC[C@@](C)(O)c2cc3ccccc3o2)cc1 ZINC000217997963 GF In-Stock Unstable ALOX15 18 41 CC(=O)Nc1ccc(S(=O)(=O)NC[C@@](C)(O)c2cc3ccccc3o2)cc1 ZINC000217997963 GF In-Stock Unstable IDO1 33 42 COc1ccc(F)cc1CN1CCN(C(=O)C[C@H](NC(N)=O)c2cccs2)CC1 ZINC000217997972 HE On-Demand Unstable SLC9A1 40 36 C#CC[C@@H](O)CCCC=O ZINC000217997981 AC For-Sale Unstable CYP4A4 50 34 COc1ccccc1CCCNC(=O)c1ccc(CSc2ccccc2)cc1 ZINC000217997994 GK In-Stock Unstable HTR1A 18 48 COc1ccccc1CCCNC(=O)c1ccc(CSc2ccccc2)cc1 ZINC000217997994 GK In-Stock Unstable DRD2 25 48 COc1ccccc1CCCNC(=O)c1ccc(CSc2ccccc2)cc1 ZINC000217997994 GK In-Stock Unstable DRD1 0 43 COc1ccccc1CCCNC(=O)c1ccc(CSc2ccccc2)cc1 ZINC000217997994 GK In-Stock Unstable DRD4 17 48 COc1ccccc1CCCNC(=O)c1ccc(CSc2ccccc2)cc1 ZINC000217997994 GK In-Stock Unstable DRD3 46 48 COc1ccccc1CCCNC(=O)c1ccc(CSc2ccccc2)cc1 ZINC000217997994 GK In-Stock Unstable PPARD 19 40 COc1ccccc1CCCNC(=O)c1ccc(CSc2ccccc2)cc1 ZINC000217997994 GK In-Stock Unstable MTNR1B 43 40 COc1ccccc1CCCNC(=O)c1ccc(CSc2ccccc2)cc1 ZINC000217997994 GK In-Stock Unstable MBTPS1 52 35 CCC(CC)(CN[C@H](C)c1ccccc1)NC(=O)OC(C)(C)C ZINC000217997996 DI For-Sale Unstable PAPA1_CARPA 40 36 CCC(CC)(CN[C@H](C)c1ccccc1)NC(=O)OC(C)(C)C ZINC000217997996 DI For-Sale Unstable CTSK 22 45 CCC(CC)(CN[C@H](C)c1ccccc1)NC(=O)OC(C)(C)C ZINC000217997996 DI For-Sale Unstable FPR1 43 35 CCC(CC)(CN[C@H](C)c1ccccc1)NC(=O)OC(C)(C)C ZINC000217997996 DI For-Sale Unstable POL 0 43 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1ccc(F)cc1Br ZINC000217998006 FJ For-Sale Unstable TRPM8 20 56 CC[C@@H](C)[C@H](NC(=O)N1C[C@H](C)C[C@@H](C)C1)C(=O)O ZINC000217998016 CE For-Sale Unstable ENPEP 65 38 CC(C)CCCCCCNC(=N)Nc1ccccc1 ZINC000217998033 CI On-Demand Unstable CXCR4 16 64 CC(C)CCCCCCNC(=N)Nc1ccccc1 ZINC000217998033 CI On-Demand Unstable MMP2 15 43 CC(C)CCCCCCNC(=N)Nc1ccccc1 ZINC000217998033 CI On-Demand Unstable MMP3 33 43 CC(C)CCCCCCNC(=N)Nc1ccccc1 ZINC000217998033 CI On-Demand Unstable HDAC2 19 40 CC(C)CCCCCCNC(=N)Nc1ccccc1 ZINC000217998033 CI On-Demand Unstable PAO 48 44 Cc1ccc(-c2noc(CN3CCN(C(=O)c4cc(N5CCOCC5)ccn4)CC3)n2)cc1 ZINC000217998079 IE On-Demand Unstable PIK3CA 42 37 Cc1ccc(-c2noc(CN3CCN(C(=O)c4cc(N5CCOCC5)ccn4)CC3)n2)cc1 ZINC000217998079 IE On-Demand Unstable MTOR 58 37 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)c1ccc(F)cc1Br ZINC000217998096 FJ For-Sale Unstable TRPM8 20 56 COc1cccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)c1 ZINC000217998107 GK In-Stock Unstable DRD2 15 42 COc1cccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)c1 ZINC000217998107 GK In-Stock Unstable DRD4 49 39 COc1cccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)c1 ZINC000217998107 GK In-Stock Unstable DRD3 31 42 COc1cccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)c1 ZINC000217998107 GK In-Stock Unstable PTAFR 27 52 COc1cccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)c1 ZINC000217998107 GK In-Stock Unstable CASR 18 40 COc1cccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)c1 ZINC000217998107 GK In-Stock Unstable NQO2 18 48 COc1cccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)c1 ZINC000217998107 GK In-Stock Unstable FDFT1 15 46 COc1cccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)c1 ZINC000217998107 GK In-Stock Unstable SCN2A 15 42 COc1cccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)c1 ZINC000217998107 GK In-Stock Unstable NPFFR2 17 41 COc1cccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)c1 ZINC000217998107 GK In-Stock Unstable MTNR1A 70 58 COc1cccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)c1 ZINC000217998107 GK In-Stock Unstable MTNR1B 68 58 COc1cccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)c1 ZINC000217998107 GK In-Stock Unstable AMP1_PLAFQ 26 42 COc1cccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)c1 ZINC000217998107 GK In-Stock Unstable TAAR1 21 41 COc1cccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)c1 ZINC000217998107 GK In-Stock Unstable CRTM 75 46 COc1cccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)c1 ZINC000217998107 GK In-Stock Unstable NPFFR1 19 41 CCOC(=O)/C=C(/Cl)C=O ZINC000217998153 AC For-Sale Unstable HCAR2 15 43 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)c1ccc(F)cc1Br ZINC000217998173 FJ For-Sale Unstable TRPM8 20 56 COc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998204 GK In-Stock Unstable DRD2 18 43 COc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998204 GK In-Stock Unstable DRD4 41 33 COc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998204 GK In-Stock Unstable DRD3 36 43 COc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998204 GK In-Stock Unstable CYSLTR1 18 41 COc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998204 GK In-Stock Unstable PTAFR 21 44 COc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998204 GK In-Stock Unstable BMP1 35 41 COc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998204 GK In-Stock Unstable NQO2 16 49 COc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998204 GK In-Stock Unstable LTB4R 22 46 COc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998204 GK In-Stock Unstable SCN2A 17 50 COc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998204 GK In-Stock Unstable HDAC8 15 42 COc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998204 GK In-Stock Unstable MTNR1A 61 42 COc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998204 GK In-Stock Unstable MTNR1B 55 44 COc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998204 GK In-Stock Unstable HDAC2 16 43 COc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998204 GK In-Stock Unstable HDAC6 17 43 COc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998204 GK In-Stock Unstable SLC6A5 25 46 COc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998204 GK In-Stock Unstable MMP1 16 42 COc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998204 GK In-Stock Unstable CRTM 42 39 Cc1ccc(-c2noc(CN3CCN(C(=O)c4cc(N5CCCC5)ccn4)CC3)n2)cc1 ZINC000217998206 IF On-Demand Unstable CCKAR 40 37 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1cc(F)ccc1Br ZINC000217998249 FJ For-Sale Unstable TRPM8 20 56 CCCC[C@@H](CC)CNC(=N)Nc1ccccc1 ZINC000217998276 BH On-Demand Unstable SCN2A 36 40 COc1ccc(OC[C@@H](C)NC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998306 HK In-Stock Unstable LTA4H 15 40 COc1ccc(OC[C@@H](C)NC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998306 HK In-Stock Unstable PPARD 17 42 COc1ccc(OC[C@@H](C)NC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998306 HK In-Stock Unstable CYP2D6 22 43 COc1ccc(OC[C@@H](C)NC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998306 HK In-Stock Unstable UTS2 40 41 COc1ccc(OC[C@@H](C)NC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998306 HK In-Stock Unstable PDS 40 35 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1cc(F)ccc1Br ZINC000217998336 FJ For-Sale Unstable TRPM8 20 56 CCCC[C@H](CC)CNC(=N)Nc1ccccc1 ZINC000217998368 BH On-Demand Unstable SCN2A 36 40 COc1ccc(OC[C@H](C)NC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998371 HK In-Stock Unstable LTA4H 15 40 COc1ccc(OC[C@H](C)NC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998371 HK In-Stock Unstable PPARD 17 42 COc1ccc(OC[C@H](C)NC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998371 HK In-Stock Unstable CYP2D6 22 43 COc1ccc(OC[C@H](C)NC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998371 HK In-Stock Unstable UTS2 40 41 COc1ccc(OC[C@H](C)NC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998371 HK In-Stock Unstable PDS 40 35 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)c1cc(F)ccc1Br ZINC000217998430 FJ For-Sale Unstable TRPM8 20 56 CC[C@@H](CCO)Nc1nccs1 ZINC000217998432 AD On-Demand Unstable MAP 74 38 CC[C@@H](CCO)Nc1nccs1 ZINC000217998432 AD On-Demand Unstable MAP1 81 37 COc1cc(NC(=O)N/C=C/c2cccc(F)c2)c(OC)cc1Cl ZINC000217998440 FI For-Sale Unstable PYGL 15 41 COc1ccc(CCS(=O)(=O)NC[C@@](C)(O)c2cc3ccccc3o2)cc1 ZINC000217998467 GF In-Stock Unstable MMP12 17 47 Cc1ccc(OCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998488 GK In-Stock Unstable DRD4 16 52 Cc1ccc(OCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998488 GK In-Stock Unstable DRD3 15 52 Cc1ccc(OCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998488 GK In-Stock Unstable PPARG 22 43 Cc1ccc(OCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998488 GK In-Stock Unstable PPARA 22 43 Cc1ccc(OCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998488 GK In-Stock Unstable GRIN2B 17 40 Cc1ccc(OCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998488 GK In-Stock Unstable LTA4H 31 40 Cc1ccc(OCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998488 GK In-Stock Unstable PLA2G4B 40 37 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)c1cc(F)ccc1Br ZINC000217998498 FJ For-Sale Unstable TRPM8 20 56 CCc1ccc(CNC(=N)Nc2ccccc2)s1 ZINC000217998502 CG On-Demand Unstable SCN2A 32 40 CC[C@H](CCO)Nc1nccs1 ZINC000217998518 AD On-Demand Unstable MAP 74 38 CC[C@H](CCO)Nc1nccs1 ZINC000217998518 AD On-Demand Unstable MAP1 81 37 CCOc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217998531 HF For-Sale Unstable MMP13 90 45 CCOc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217998531 HF For-Sale Unstable ADAM17 72 47 CCOc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217998531 HF For-Sale Unstable MMP2 42 52 CCOc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217998531 HF For-Sale Unstable MMP3 87 45 CCOc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217998531 HF For-Sale Unstable MMP8 34 42 CCOc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217998531 HF For-Sale Unstable MMP9 50 45 CCOc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217998531 HF For-Sale Unstable MMP7 82 42 CCOc1ccc(S(=O)(=O)N2C[C@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217998531 HF For-Sale Unstable MMP1 93 45 COc1ccc(CCS(=O)(=O)NC[C@](C)(O)c2cc3ccccc3o2)cc1 ZINC000217998546 GF In-Stock Unstable MMP12 18 47 O=C(Cc1ccsc1)N1CCN(Cc2nc(-c3cccc(C(F)(F)F)c3)no2)CC1 ZINC000217998572 IH On-Demand Unstable KCNJ1 44 33 O=C(Cc1ccsc1)N1CCN(Cc2nc(-c3cccc(C(F)(F)F)c3)no2)CC1 ZINC000217998572 IH On-Demand Unstable ETHR 50 40 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1cc(Br)ccc1F ZINC000217998579 FJ For-Sale Unstable TRPM8 20 62 Cc1cc(Cl)c(F)c(C[C@H](N)C(=O)O)c1F ZINC000217998602 BD For-Sale Unstable GRIA3 55 40 Cc1cc(Cl)c(F)c(C[C@H](N)C(=O)O)c1F ZINC000217998602 BD For-Sale Unstable GRIA1 39 40 Cc1cc(Cl)c(F)c(C[C@H](N)C(=O)O)c1F ZINC000217998602 BD For-Sale Unstable GRIA2 53 40 Cc1cc(Cl)c(F)c(C[C@H](N)C(=O)O)c1F ZINC000217998602 BD For-Sale Unstable GRIA4 45 40 Cc1cc(Cl)c(F)c(C[C@H](N)C(=O)O)c1F ZINC000217998602 BD For-Sale Unstable GRIK1 37 40 Cc1cc(Cl)c(F)c(C[C@H](N)C(=O)O)c1F ZINC000217998602 BD For-Sale Unstable SLC1A2 41 38 O=C(Nc1ccccc1C(=O)c1ccccc1)c1ccc(CSc2ccccc2)cc1 ZINC000217998610 HK In-Stock Unstable HDAC8 0 44 O=C(Nc1ccccc1C(=O)c1ccccc1)c1ccc(CSc2ccccc2)cc1 ZINC000217998610 HK In-Stock Unstable NR1H4 24 47 O=C(Nc1ccccc1C(=O)c1ccccc1)c1ccc(CSc2ccccc2)cc1 ZINC000217998610 HK In-Stock Unstable HDAC1 39 45 O=C(Nc1ccccc1C(=O)c1ccccc1)c1ccc(CSc2ccccc2)cc1 ZINC000217998610 HK In-Stock Unstable HDAC2 33 44 O=C(Nc1ccccc1C(=O)c1ccccc1)c1ccc(CSc2ccccc2)cc1 ZINC000217998610 HK In-Stock Unstable HDAC3 0 42 O=C(Nc1ccccc1C(=O)c1ccccc1)c1ccc(CSc2ccccc2)cc1 ZINC000217998610 HK In-Stock Unstable HAO1 16 42 O=C(Nc1ccccc1C(=O)c1ccccc1)c1ccc(CSc2ccccc2)cc1 ZINC000217998610 HK In-Stock Unstable KCNK3 43 35 O=C(Nc1ccccc1C(=O)c1ccccc1)c1ccc(CSc2ccccc2)cc1 ZINC000217998610 HK In-Stock Unstable FAS 16 42 CCOc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217998621 HF For-Sale Unstable MMP13 90 45 CCOc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217998621 HF For-Sale Unstable ADAM17 72 47 CCOc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217998621 HF For-Sale Unstable MMP2 42 52 CCOc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217998621 HF For-Sale Unstable MMP3 87 45 CCOc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217998621 HF For-Sale Unstable MMP8 34 42 CCOc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217998621 HF For-Sale Unstable MMP9 50 45 CCOc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217998621 HF For-Sale Unstable MMP7 82 42 CCOc1ccc(S(=O)(=O)N2C[C@@H](Oc3ccccc3F)C[C@@H]2C(=O)OC)cc1 ZINC000217998621 HF For-Sale Unstable MMP1 93 45 N=C(NCCc1ccc(Cl)s1)Nc1ccccc1 ZINC000217998629 CH On-Demand Unstable CXCR4 15 49 CCO[C@@H]1COCC[C@H]1NC(=O)c1ccc(C)nc1 ZINC000217998650 CD In-Stock Unstable ADAM17 23 42 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1cc(Br)ccc1F ZINC000217998653 FJ For-Sale Unstable TRPM8 20 62 COc1ccc(CCNC(=O)C[C@H](CC(C)C)c2c(O)cc(O)c3c(=O)cc(-c4ccccc4)oc23)cc1 ZINC000217998662 KK In-Stock Unstable CAPN2 15 40 Cc1cc(Cl)c(F)c(C[C@@H](N)C(=O)O)c1F ZINC000217998689 BD For-Sale Unstable GRIA3 55 40 Cc1cc(Cl)c(F)c(C[C@@H](N)C(=O)O)c1F ZINC000217998689 BD For-Sale Unstable GRIA1 39 40 Cc1cc(Cl)c(F)c(C[C@@H](N)C(=O)O)c1F ZINC000217998689 BD For-Sale Unstable GRIA2 53 40 Cc1cc(Cl)c(F)c(C[C@@H](N)C(=O)O)c1F ZINC000217998689 BD For-Sale Unstable GRIA4 45 40 Cc1cc(Cl)c(F)c(C[C@@H](N)C(=O)O)c1F ZINC000217998689 BD For-Sale Unstable GRIK1 37 40 Cc1cc(Cl)c(F)c(C[C@@H](N)C(=O)O)c1F ZINC000217998689 BD For-Sale Unstable SLC1A2 41 38 CC(C)Oc1cccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)c1 ZINC000217998719 HK In-Stock Unstable PTAFR 20 43 CC(C)Oc1cccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)c1 ZINC000217998719 HK In-Stock Unstable FDFT1 16 45 CC(C)Oc1cccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)c1 ZINC000217998719 HK In-Stock Unstable AMP1_PLAFQ 34 42 CC(C)Oc1cccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)c1 ZINC000217998719 HK In-Stock Unstable CRTM 68 45 CC(C)Oc1cccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)c1 ZINC000217998719 HK In-Stock Unstable PDS 41 38 Cc1cccc(C(=O)N2CCN(Cc3nc(-c4cccc(C(F)(F)F)c4)no3)CC2)c1O ZINC000217998723 IH On-Demand Unstable CCR2 15 40 CCN1CCC[C@@H]1CNC(=O)N1C[C@@H](O)C[C@@H]1C(=O)O ZINC000217998733 CB For-Sale Unstable DRD2 32 40 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)c1cc(Br)ccc1F ZINC000217998747 FJ For-Sale Unstable TRPM8 20 62 COc1ccc(CCNC(=O)C[C@@H](CC(C)C)c2c(O)cc(O)c3c(=O)cc(-c4ccccc4)oc23)cc1 ZINC000217998751 KK In-Stock Unstable CAPN2 15 40 O=C(N[C@@H]1CCC[C@@H]1CO)c1cc2cc(F)ccc2s1 ZINC000217998764 CF For-Sale Unstable SSTR3 27 40 O=C(N[C@@H]1CCC[C@@H]1CO)c1cc2cc(F)ccc2s1 ZINC000217998764 CF For-Sale Unstable PIN1 21 40 O=C(N/C=C/c1cccc(F)c1)N1CCN(c2ccccc2)CC1 ZINC000217998793 EG For-Sale Unstable FAAH 0 44 O=C(N/C=C/c1cccc(F)c1)N1CCN(c2ccccc2)CC1 ZINC000217998793 EG For-Sale Unstable AKR1C3 0 40 CCN1CCC[C@H]1CNC(=O)N1C[C@@H](O)C[C@@H]1C(=O)O ZINC000217998818 CB For-Sale Unstable DRD2 32 40 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)c1cc(Br)ccc1F ZINC000217998824 FJ For-Sale Unstable TRPM8 20 62 CC(C)Oc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217998843 HK In-Stock Unstable CRTM 40 37 O=C(N[C@H]1CCC[C@@H]1CO)c1cc2cc(F)ccc2s1 ZINC000217998846 CF For-Sale Unstable SSTR3 27 40 O=C(N[C@H]1CCC[C@@H]1CO)c1cc2cc(F)ccc2s1 ZINC000217998846 CF For-Sale Unstable PIN1 21 40 COc1ccc(SCC(=O)N2CCN(Cc3nc(-c4cccc(C(F)(F)F)c4)no3)CC2)cc1 ZINC000217998862 JI On-Demand Unstable HRH3 18 40 COc1ccc(Cl)cc1S(=O)(=O)NC[C@@](C)(O)c1cc2ccccc2o1 ZINC000217998864 GG In-Stock Unstable COLA 74 39 COc1ccc(Cl)cc1S(=O)(=O)NC[C@@](C)(O)c1cc2ccccc2o1 ZINC000217998864 GG In-Stock Unstable CPT1A 70 39 COc1ccc(Cl)cc1S(=O)(=O)NC[C@@](C)(O)c1cc2ccccc2o1 ZINC000217998864 GG In-Stock Unstable CPT1B 71 35 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1ccc(Br)cc1F ZINC000217998903 FJ For-Sale Unstable TRPM8 20 59 CC(C)C/C=C\[C@H](O)[C@H](NC(=O)OC(C)(C)C)C(C)C ZINC000217998910 CG For-Sale Unstable CTSK 17 47 O=C(N[C@@H]1CCC[C@H]1CO)c1cc2cc(F)ccc2s1 ZINC000217998937 CF For-Sale Unstable SSTR3 27 40 O=C(N[C@@H]1CCC[C@H]1CO)c1cc2cc(F)ccc2s1 ZINC000217998937 CF For-Sale Unstable PIN1 21 40 CN(CCNC(=O)c1ccc(CSc2ccccc2)cc1)c1ccccc1 ZINC000217998946 GJ In-Stock Unstable HAO1 15 41 COc1ccc(Cl)cc1S(=O)(=O)NC[C@](C)(O)c1cc2ccccc2o1 ZINC000217998957 GG In-Stock Unstable COLA 74 39 COc1ccc(Cl)cc1S(=O)(=O)NC[C@](C)(O)c1cc2ccccc2o1 ZINC000217998957 GG In-Stock Unstable CPT1A 70 39 COc1ccc(Cl)cc1S(=O)(=O)NC[C@](C)(O)c1cc2ccccc2o1 ZINC000217998957 GG In-Stock Unstable CPT1B 71 35 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1ccc(Br)cc1F ZINC000217998979 FJ For-Sale Unstable TRPM8 20 59 CC(C)C/C=C/[C@H](O)[C@H](NC(=O)OC(C)(C)C)C(C)C ZINC000217998988 CG For-Sale Unstable CTSK 17 47 O=C(N[C@H]1CCC[C@H]1CO)c1cc2cc(F)ccc2s1 ZINC000217999009 CF On-Demand Unstable SSTR3 18 40 O=C(N[C@H]1CCC[C@H]1CO)c1cc2cc(F)ccc2s1 ZINC000217999009 CF On-Demand Unstable PIN1 21 40 Cc1cccc(C)c1NC(=O)N/C=C/c1cccc(F)c1 ZINC000217999028 CI For-Sale Unstable S1PR4 0 40 O=C(Nc1ccc(OC2CCCC2)cc1)c1ccc(CSc2ccccc2)cc1 ZINC000217999057 HK In-Stock Unstable PRSS1 24 50 O=C(Nc1ccc(OC2CCCC2)cc1)c1ccc(CSc2ccccc2)cc1 ZINC000217999057 HK In-Stock Unstable PRNP 42 36 O=C(Nc1ccc(OC2CCCC2)cc1)c1ccc(CSc2ccccc2)cc1 ZINC000217999057 HK In-Stock Unstable PLAT 15 45 O=C(Nc1ccc(OC2CCCC2)cc1)c1ccc(CSc2ccccc2)cc1 ZINC000217999057 HK In-Stock Unstable PLAU 27 50 O=C(Nc1ccc(OC2CCCC2)cc1)c1ccc(CSc2ccccc2)cc1 ZINC000217999057 HK In-Stock Unstable NOD2 46 39 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)c1ccc(Br)cc1F ZINC000217999067 FJ For-Sale Unstable TRPM8 20 59 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)Cc1ccccc1 ZINC000217999128 GE In-Stock Unstable FKBP1A 23 43 N=C(NCCc1ccc(Br)s1)Nc1ccccc1 ZINC000217999132 DH On-Demand Unstable CXCR4 15 49 COc1ccc([N+](=O)[O-])cc1NC(=O)N/C=C/c1cccc(F)c1 ZINC000217999139 EH For-Sale Unstable PYGL 31 40 COc1ccc([N+](=O)[O-])cc1NC(=O)N/C=C/c1cccc(F)c1 ZINC000217999139 EH For-Sale Unstable KCNMA1 21 50 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)c1ccc(Br)cc1F ZINC000217999144 FJ For-Sale Unstable TRPM8 20 59 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)Cc1ccccc1 ZINC000217999215 GE In-Stock Unstable FKBP1A 23 43 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1cc(Br)cn1C ZINC000217999243 EH For-Sale Unstable TRPM8 19 54 COc1cc(Cl)c(C)cc1NC(=O)N/C=C/c1cccc(F)c1 ZINC000217999250 EJ For-Sale Unstable PYGL 15 40 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)Cc1ccccc1 ZINC000217999298 GE In-Stock Unstable FKBP1A 23 43 COC(=O)c1cc2cccc(F)c2o1 ZINC000217999313 AE In-Stock Unstable RPS6KA2 40 33 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1cc(Br)cn1C ZINC000217999340 EH For-Sale Unstable TRPM8 19 54 O=C(c1cc(-c2cccs2)on1)N1CCN(Cc2nc(-c3cccc(C(F)(F)F)c3)no2)CC1 ZINC000217999349 JI On-Demand Unstable ETHR 56 38 CC[C@@H](NC(=O)c1ccc(Cl)cc1O)c1ccnn1C ZINC000217999371 CF In-Stock Unstable UTS2 43 33 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)Cc1ccccc1 ZINC000217999375 GE In-Stock Unstable FKBP1A 23 43 CCOc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217999386 HK In-Stock Unstable PPARG 17 41 CCOc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217999386 HK In-Stock Unstable PPARA 15 41 CCOc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217999386 HK In-Stock Unstable CYSLTR1 19 42 CCOc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217999386 HK In-Stock Unstable SCN2A 21 52 CCOc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217999386 HK In-Stock Unstable PLA2G4A 25 42 CCOc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217999386 HK In-Stock Unstable PLA2G2A 0 43 CCOc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217999386 HK In-Stock Unstable PLA2G4B 36 42 CCOc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217999386 HK In-Stock Unstable CRTM 41 37 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)c1cc(Br)cn1C ZINC000217999426 EH For-Sale Unstable TRPM8 19 54 CC[C@H](NC(=O)c1ccc(Cl)cc1O)c1ccnn1C ZINC000217999460 CF In-Stock Unstable UTS2 43 33 Cc1cc(OCC(=O)Nc2ccc(SC[C@@H]3CCCN4CCCC[C@H]34)nc2)ccc1Cl ZINC000217999473 JK In-Stock Unstable MCHR1 18 41 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1cc(F)cc(F)c1 ZINC000217999487 HE For-Sale Unstable MMP2 16 54 COC(=O)[C@@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1cc(F)cc(F)c1 ZINC000217999487 HE For-Sale Unstable MMP7 42 36 CCN(C(=O)N/C=C/c1cccc(F)c1)c1cccc(C)c1 ZINC000217999497 CI For-Sale Unstable NR1H4 42 44 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)c1cc(Br)cn1C ZINC000217999510 EH For-Sale Unstable TRPM8 19 54 CCCOc1ccccc1CCCNC(=O)c1ccc(CSc2ccccc2)cc1 ZINC000217999524 HK In-Stock Unstable PPARG 15 43 CCCOc1ccccc1CCCNC(=O)c1ccc(CSc2ccccc2)cc1 ZINC000217999524 HK In-Stock Unstable MTNR1B 42 40 Cc1noc2nc(C(C)C)cc(C(=O)NC3CCN(C(=O)Nc4ccccc4)CC3)c12 ZINC000217999530 HI On-Demand Unstable SMO 33 41 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1cc(F)cc(F)c1 ZINC000217999572 HE For-Sale Unstable MMP2 16 54 COC(=O)[C@H]1C[C@H](Oc2ccccc2F)CN1S(=O)(=O)c1cc(F)cc(F)c1 ZINC000217999572 HE For-Sale Unstable MMP7 42 36 COc1cccc([C@@H]2CC(=O)Oc3cc(OC)c(OC)c(OC)c32)c1OCCc1ccccc1 ZINC000217999595 JJ In-Stock Unstable ADRA1A 15 41 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1cc(Br)c[nH]1 ZINC000217999598 EH For-Sale Unstable TRPM8 19 55 COc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1OC ZINC000217999631 HK In-Stock Unstable DRD2 20 43 COc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1OC ZINC000217999631 HK In-Stock Unstable DRD1 0 41 COc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1OC ZINC000217999631 HK In-Stock Unstable DRD4 15 41 COc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1OC ZINC000217999631 HK In-Stock Unstable DRD3 31 43 COc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1OC ZINC000217999631 HK In-Stock Unstable PTAFR 18 50 COc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1OC ZINC000217999631 HK In-Stock Unstable TRPV1 0 45 COc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1OC ZINC000217999631 HK In-Stock Unstable MTNR1A 15 46 COc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1OC ZINC000217999631 HK In-Stock Unstable MTNR1B 27 53 COc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1OC ZINC000217999631 HK In-Stock Unstable SCN5A 0 43 COc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1OC ZINC000217999631 HK In-Stock Unstable MT-ND1 27 44 COc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1OC ZINC000217999631 HK In-Stock Unstable ABCG2 18 43 COc1ccc(CCCNC(=O)c2ccc(CSc3ccccc3)cc2)cc1OC ZINC000217999631 HK In-Stock Unstable CRTM 41 36 C1=C(c2c[nH]c3ccccc23)CNC1 ZINC000217999645 AE For-Sale Unstable PRKCB 15 45 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1cc(F)cc(F)c1 ZINC000217999656 HE For-Sale Unstable MMP2 16 54 COC(=O)[C@@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1cc(F)cc(F)c1 ZINC000217999656 HE For-Sale Unstable MMP7 42 36 COc1cccc([C@H]2CC(=O)Oc3cc(OC)c(OC)c(OC)c32)c1OCCc1ccccc1 ZINC000217999682 JJ In-Stock Unstable ADRA1A 15 41 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1cc(Br)c[nH]1 ZINC000217999683 EH For-Sale Unstable TRPM8 19 55 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1cc(F)cc(F)c1 ZINC000217999730 HE For-Sale Unstable MMP2 16 54 COC(=O)[C@H]1C[C@@H](Oc2ccccc2F)CN1S(=O)(=O)c1cc(F)cc(F)c1 ZINC000217999730 HE For-Sale Unstable MMP7 42 36 CCc1ncnc(NCCc2cc(F)cc(F)c2)c1F ZINC000217999736 CG On-Demand Unstable HTT 0 40 CC(C)[C@@H]1CC[C@H](C)C[C@@H]1NC(=O)c1cc(Br)c[nH]1 ZINC000217999761 EH For-Sale Unstable TRPM8 19 55 COc1ccc2[nH]cc(C3=CCNC3)c2c1 ZINC000217999763 BE For-Sale Unstable HTR1A 19 78 COc1ccc2[nH]cc(C3=CCNC3)c2c1 ZINC000217999763 BE For-Sale Unstable HTR1D 17 78 COc1ccc2[nH]cc(C3=CCNC3)c2c1 ZINC000217999763 BE For-Sale Unstable HTR1B 20 78 COc1cccc(C(=O)Nc2nc3c(s2)CCCCC3)c1O ZINC000217999776 DG On-Demand Unstable SLC27A1 39 42 O=C(N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2)C1(n2cnnn2)CCCCC1 ZINC000217999799 FD In-Stock Unstable CHRNA4 28 44 CC(C)[C@H]1CC[C@H](C)C[C@@H]1NC(=O)c1cc(Br)c[nH]1 ZINC000217999852 EH For-Sale Unstable TRPM8 19 55 CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1csc(Br)c1 ZINC000217999928 EJ For-Sale Unstable TRPM8 22 63 COC(=O)c1ccnc(N(C)C2CCCC2)c1 ZINC000217999931 BE For-Sale Unstable KDM4C 0 48 COC(=O)c1ccnc(N(C)C2CCCC2)c1 ZINC000217999931 BE For-Sale Unstable SCARB1 47 35 COC(=O)c1ccnc(N(C)C2CCCC2)c1 ZINC000217999931 BE For-Sale Unstable KDM3A 0 48 COC(=O)c1ccnc(N(C)C2CCCC2)c1 ZINC000217999931 BE For-Sale Unstable KDM5C 0 48 CC1=C(c2ccccc2)[C@@H]1C(=O)NCc1ccc2c(c1)nc(C)n2C ZINC000217999935 EH In-Stock Unstable NAMPT 40 34 Cc1ccc(OC[C@@H](C)NC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217999957 GK In-Stock Unstable PTGER3 44 36 Cc1ccc(OC[C@@H](C)NC(=O)c2ccc(CSc3ccccc3)cc2)cc1 ZINC000217999957 GK In-Stock Unstable PDS 40 33 CC(C)[C@H]1CC[C@@H](C)C[C@@H]1NC(=O)c1csc(Br)c1 ZINC000217999997 EJ For-Sale Unstable TRPM8 22 63